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PDSP
Ki Database
Tracer Database
GPCR Datbase
Rothlab
UNC
Binding/Functional Assay
MDR-1/CaCo2
Publications
USCD-Nature
Instructions:
Select a receptor and a Ki condition. Experiment results for experiments with the selected receptor and ki values will be presented on the following page. The resulting set of test ligands can optionally be graphed against all the receptors in the KiDB using our color coded Ki Graph Tool.
Receptor:
Adrenaline Alpha1
Alpha2B
(+) CIMBI-772
(+)CIMBI-775
(-) CIMBI-772
(-)CIMBI-775
1200015E14Rik
17Beta-HSD Type 3
3-Ethyl-3-{4-[4-(3-hydroxyphenyl)piperazin-1-yl]butyl}-1,3-dihydro-2H-indol-2-one
3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-1,3-dimethyl-1,3-dihydro-2H-indol-2-one
3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-3-(2-fluoroethyl)-1,3-dihydro-2H-indol-2-one
3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-3-methyl-1,3-dihydro-2H-indol-2-one
3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-3-propyl-1,3-dihydro-2H-indol-2-one
5-HT Transporter
5-HT uptake
5-HT-S1
5-HT-S1A
5-HT-S2
5-HT1
5-HT1 like
5-HT1A
5-HT1B
5-HT1C
5-HT1D
5-HT1Dalpha
5-HT1Db
5-HT1DBeta
5-HT1E
5-HT1F
5-HT2
5-HT2A
5-HT2B
5-HT2C
5-HT2c VGI
5-HT2C-INI
5-HT3
5-HT4
5-HT4a
5-HT4b
5-HT4c
5-HT4d
5-HT4hb
5-HT4L
5-HT4S
5-HT5
5-HT5a
5-HT5B
5-HT6
5-HT7
5-HT7A
5-HT7b
5-HT7L
5-HT7S
5-Lipoxygenase
5HT Transporter
A2
a2b2 nicotinic cholinergic
a2b4 nicotinic cholinergic
A3
a3b2 nicotinic cholinergic
a3b4 nicotinic cholinergic
A4
a4b2 nicotinic cholinergic
a4b4 nicotinic cholinergic
Ac-AChBP
Acetylcholinesterase
Acetylcholinesterase, AChE
AChE
Activated p21cdc42Hs kinase
Activator Protein AP-1
ADENOSINE
ADENOSINE A1
ADENOSINE A1 high
ADENOSINE A1 low
ADENOSINE A2
ADENOSINE A2a
ADENOSINE A2B
ADENOSINE A3
Adenosine A4
Adenosine Deaminase ADA
Adenosine Kinase, AK
Adenosine transporter
ADENOSINE UPTAKE
Adenylate cyclase
Adenylate cyclase Forskolin
Adrenaline
Adrenaline Alpha1
Adrenaline Alpha2
Adrenaline Beta
Adrenaline 1
Adrenaline 2
Adrenaline alpha1
Adrenaline alpha2
Adrenaline Beta
Adrenaline beta1
Adrenergic Alpha
adrenergic Alpha1
adrenergic Alpha1A
Adrenergic alpha1A/B
adrenergic Alpha1B
adrenergic Alpha1C
adrenergic Alpha1D
adrenergic Alpha2
adrenergic Alpha2A
adrenergic Alpha2B
adrenergic Alpha2C
adrenergic Alpha2D
adrenergic Beta
adrenergic Beta1
adrenergic Beta1,2
adrenergic Beta2
adrenergic Beta3
Adrenomedullin AM1
Adrenomedullin AM2
Akt
aldose reductase
Aldosterone
all-trans-retinoic acid, atRA
Alpha 1 Adrenergic Receptor
Alpha 1A Adrenergic Receptor
Alpha 1B Adrenergic Receptor
Alpha 2 Adrenergic Receptor
Alpha 2A Adrenergic Receptor
Alpha 2B Adrenergic Receptor
Alpha 2C Adrenergic Receptor
alpha-1
Alpha-1A
Alpha-1B
alpha-2
Alpha-2A
alpha-2C
Alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid
alpha1
alpha1-Adrenocepter
alpha1-GABA-A
alpha1A
alpha1B
alpha1beta3gamma2
Alpha1D
alpha2
alpha2-Adrenocepter
alpha2-GABA-A
Alpha2A
Alpha2B
alpha2beta2
alpha2beta3gamma2
alpha2beta4
Alpha2C
alpha3-GABA-A
alpha3beta2
alpha3beta3gamma2
alpha3beta4
alpha4bet2
alpha4beta2
alpha4beta3gamma2
alpha4beta4
alpha5-GABA-A
alpha5beta3gamma2
alpha6-GABA-A
alpha6beta3gamma2
alpha7
alphabeta3gamma2
AMPA
Anandamid membrane transporter, AMT
Anaphylatoxin C5a
Anaplastic lymphoma kinase (Ki-1)
androgen
Androgen Receptor
ANF
Angiotensin
ANGIOTENSIN AT1
Angiotensin AT2
Angiotensin II AT1
Angiotensin II AT1A
Angiotensin II AT1B
Angiotensin II AT2
Angiotensin II, central
Angiotensin IV
Angiotensin-converting enzyme, ACE
ANP (Atrial natriuretic peptide)
AP2 associated kinase 1
Apelin
Arg-vasopressin V1
ATPase (Na+, K+)
Atrial Natriuretic Factor
atrial natriuretic peptide, ANP
Aurora kinase C
B lymphoid tyrosine kinase
B1
B1 BRADYKININ
B2
B2 BRADYKININ
B3
BChE
Benzodiazepine central
Benzodiazepine peripheral
Beta 1
Beta 2
Beta 3
Beta-1
Beta-2
beta-amyloid
Beta-Amyloid (1-40)
Beta-Amyloid (1-42)
beta1
beta2
beta3
BHE
BHSK
BHSP
Bile Salt Export Pump, BSEP
BMP2 inducible kinase
BMX non-receptor tyrosine kinase
Bombesin
Bombesin 1
Bombesin 2
Bombesin 3
Bombesin 4
Bombesin BB1
Bombesin BB2
Bombesin BB3
Bradykinin
Bradykinin B1
Bradykinin B2
Bruton agammaglobulinemia tyrosine kinase
butyrylcholinesterase, BuChE
BZP
BZP Rat Brain
BZP Rat Brain Site
C-src tyrosine kinase
calcineurin
Calcitonin
Calcitonin Gene-Related Peptide
Calcitonin Gene-related Peptide (CGRP)
Calcitonin Gene-Related Peptide 1
Calcium (type L)
Calcium channel
Calcium channel (DHP)
Calcium channel (Type L)
Calcium channel (Type N)
Calcium channel (Type T,L)
Calcium channel (VER)
Calcium channel diltiazem
Calcium Channel L-Type, Benzothiazepine
Calcium Channel L-Type, Dihydropyridine
Calcium Channel L-Type, Phenylalkylamine
Calcium Channel N-Type
Calcium channel verapamil binding site
Calcium/calmodulin-dependent protein kinase (CaM kinase) II alpha
Calcium/calmodulin-dependent protein kinase (CaM kinase) II beta
Calcium/calmodulin-dependent protein kinase (CaM kinase) II delta
Calcium/calmodulin-dependent protein kinase (CaM kinase) II gamma
Calcium/calmodulin-dependent protein kinase I
Calcium/calmodulin-dependent protein kinase ID
Calcium/calmodulin-dependent protein kinase IG
Calcium/calmodulin-dependent protein kinase kinase 1, alpha
Calcium/calmodulin-dependent protein kinase kinase 2, beta
calmodulin kinase
calpain
calpain-1
CANNABINOID CB1
CANNABINOID CB2
Carbonic Anhydrase Isozymes, CA I
Carbonic Anhydrase Isozymes, CA II
Carbonic Anhydrase Isozymes, CA IX
Carboxypeptidase CPG2
Casein kinase 1 Delta
Casein kinase 1, epsilon
Casein kinase 1, gamma 1
Casein kinase 1, gamma 2
casein kinase-1
casein kinase-2
caspase-2
caspase-3
caspase-6
caspase-7
caspase-8
Cathepsin D
CB1
CB2
CBR
CCK A
CCK B
CCR5
CD-45
CDC-like kinase 1
CDC-like kinase 2
CDC-like kinase 3
CDC-like kinase 4
CDC25
CDK1
CDK2
CDK4
CDK5 activator-binding protein C53
CGRP
CGRP1
Chemoattractant receptor-homologous, CRTH2
Chemokine CCR1
Chemokine CCR2B
Chemokine CCR4
Chemokine CCR5
Chemokine CX3CR1
Chemokine CXCR1
Chemokine CXCR2
Chemokine CXCR3
Chemokine CXCR4
Chemokine CXCR5
Chemokine CXCR7
Chemokine receptor 5
Chemokine US28
Chloride channel, TBOB
Chloride ionophore
Cholecystokinin
Cholecystokinin 1
Cholecystokinin 2
Cholecystokinin A
Cholecystokinin B
Cholecystokinin central
Cholecystokinin peripheral
Choline Acetyltransferase
Choline Transporter
Choline Uptake
Cholinergic, muscarinic
Cholinergic, muscarinic M1
Cholinergic, muscarinic M2
Cholinergic, muscarinic M3
Cholinergic, muscarinic M4
Cholinergic, muscarinic M5
Cholinergic, nicotinic
Cholinergic, nicotinic Alpha1
Cholinergic, Nicotinic Alpha1Beta1DeltaGamma
Cholinergic, Nicotinic Alpha1Beta2
Cholinergic, Nicotinic Alpha2Beta2
Cholinergic, Nicotinic Alpha2Beta4
Cholinergic, Nicotinic Alpha3Beta2
Cholinergic, Nicotinic Alpha3Beta4
Cholinergic, Nicotinic Alpha3Beta4x
Cholinergic, Nicotinic Alpha4Beta2
Cholinergic, Nicotinic Alpha4Beta2**
Cholinergic, Nicotinic Alpha4Beta2X
Cholinergic, Nicotinic Alpha4Beta4
Cholinergic, Nicotinic Alpha6
Cholinergic, Nicotinic Alpha6Beta2
Cholinergic, Nicotinic Alpha6Beta3Beta4Alpha5
Cholinergic, Nicotinic Alpha6Beta4
Cholinergic, Nicotinic Alpha7
Cholinergic, Nicotinic Alpha7/5-HT3
Cholinergic, Nicotinic Muscle
CIMBI-712
CIMBI-717
CIMBI-772
CIMBI-775
Colchicine
Corticotropin-Releasing Factor
COX-1
COX-2
CRF
CRF-R1
CRF-R2 Alpha
CRF-R2 Beta
CRF1
CRF2 Beta
Ct-AChBP
Cyclin G associated kinase
Cyclin-dependent kinase 2
D1
D2
D2L
D2S
D3
D4
D4.4
D5
DAT
Death-associated kinase 3
Death-associated protein kinase 2
Delta
Delta Opiate Receptor
Deoxyuridine triphosphatase
Dihyrofolate Reductase, DHFR
Dipeptidyl peptidase DPP II
Dipeptidyl peptidase DPP IV
DOP
DOPAMINE
DOPAMINE D1
Dopamine D1 high
Dopamine D1 low
Dopamine D1A
Dopamine D1B
DOPAMINE D2
DOPAMINE D2 Long
DOPAMINE D2 Short
DOPAMINE D2/D4
Dopamine D2A
Dopamine D2B
DOPAMINE D3
Dopamine D3A
DOPAMINE D4
DOPAMINE D4.2
DOPAMINE D4.4
DOPAMINE D4.7
DOPAMINE D5
Dopamine Transporter
Dopamine Uptake
Dopamine, cocaine site
Dopamine1-like
Dopamine2-like
DOR
DP1
DRI
Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A
dUTPase
EGF
EGF-R
Eledoisin
ENDOTHELIN
ENDOTHELIN A
ENDOTHELIN B
EP1
EP2
EP3
EP4
EPH receptor A2
EPH receptor A3
EPH receptor A4
EPH receptor A5
EPH receptor A6
EPH receptor A7
EPH receptor A8
EPH receptor B1
EPH receptor B2
EPH receptor B4
Epidermal growth factor receptor
Erythropietin EPOR
estrogen
estrogen alpha
estrogen beta
Estrogen receptor alpha
Estrogen receptor beta
estrogen, ER alpha
estrogen, ER beta
Excitatory Amino Acid EAAT1
Excitatory Amino Acid EAAT2
Excitatory Amino Acid EAAT3
Export Pump, ABCC2
extracellular-regulated protein kinase, ERK
Fatty Acid Amide Hydrolic, FAAH
Fer (fps/fes related) tyrosine kinase (phosphoprotein NCP94)
FGF
FGF-R2
FGFR-1, (cyto)
FGFR-1, (FL)
Fibroblast growth factor receptor 1
Fibroblast growth factor receptor 2
Fibroblast growth factor receptor 3
FKBP12
Fms-related tyrosine kinase 3
Fms-related tyrosine kinase 4
Follicle-Stimulating Hormone, FSH
Formyl peptide Receptor
FP
FYN oncogene related to SRC, FGR, YES
Fyn-related kinase
GABA
GABA A
GABA A alpha1
GABA A Alpha1Beta1Gamma2
GABA A Alpha1Beta2
GABA A Alpha1Beta2Gamma2
GABA A Alpha1Beta3Gamma2
GABA A alpha2
GABA A Alpha2Beta1Gamma2
GABA A Alpha2Beta2Gamma2
GABA A Alpha2Beta3Gamma2
GABA A alpha3
GABA A Alpha3Beta1Gamma2
GABA A Alpha3Beta2Gamma2
GABA A Alpha3Beta3Gamma2
GABA A Alpha4Beta2Gamma2
GABA A Alpha4Beta3Gamma2
GABA A Alpha4Gamma2
GABA A alpha5
GABA A Alpha5Beta1Gamma2
GABA A Alpha5Beta2Gamma2
GABA A Alpha5Beta3Gamma2
GABA A Alpha5m10Beta2Gamma2
GABA A Alpha5m8Beta2Gamma2
GABA A Alpha5m9Beta2Gamma2
GABA A alpha6
GABA A Alpha6Beta1Gamma2
GABA A Alpha6Beta2Gamma2
GABA A Alpha6Beta3Gamma2
GABA A anti-Alpha1
GABA A anti-Alpha3
GABA A Benzodiazepine
GABA A Benzodiazepine brain
GABA A Benzodiazepine liver
GABA A Benzodiazepine omega1
GABA A Benzodiazepine omega2
GABA A Benzodiazepine omega5
GABA A Benzodiazepine Type I
GABA A Benzodiazepine Type II
GABA A Benzodiazepine Type IIL
GABA A Benzodiazepine Type IIM
GABA A Beta2Gamma2
GABA A Flunitrazepam, Central
GABA A Muscimol, Central
GABA A, agonist site
GABA alpha1beta3gamma2
GABA alpha2beta3gamma2
GABA alpha3beta3gamma2
GABA alpha4beta3gamma2
GABA alpha5beta3gamma2
GABA alpha6beta3gamma2
GABA B
GABA B rho 1
GABA B1A
GABA B1B
GABA C
GABA receptor alpha-1 subunit
GABA receptor alpha-2 subunit
GABA receptor alpha-3 subunit
GABA receptor alpha-5 subunit
GABA transporter
GABA uptake
GABA, Chloride, TBOB
GABA-A
GABA-PICROTOXIN
GABAA
GABAa (Cl channel)
GABAA alpha1beta3gamma2
GABAA alpha2beta3gamma2
GABAA alpha3beta3gamma2
GABAA alpha4beta3gamma2
GABAA alpha5beta3gamma2
GABAA alpha6beta3gamma2
GABAa1 receptor
Gabapentin
GALANIN
Galanin R1
Galanin R2
Galanin R3
Gamma hydroxybutyric, GHB
Gardner-Rasheed feline sarcoma viral (v-fgr) oncogene homolog
Gastrin-Releasing peptide
glucagon
Glucocorticoid
Glucocorticoid receptor
GLUK5
GluR1 -40 mV
GluR1 -80 mV
Glutamate AMPA 1
Glutamate AMPA 2
Glutamate AMPA 3
Glutamate AMPA 4
Glutamate AMPA 5
Glutamate AMPA 6
Glutamate Chloride
Glutamate delta 2
Glutamate, GluR1
Glutamate, GluR2
Glutamate, GluR4
Glutamate, GluR6 + KA2
Glutamate, GluR7
Glutamate, Non-selective
Glutamate-AMPA
Glutamate-AMPA, GluR1
Glutamate-AMPA, GluR2 (Q/R)
Glutamate-AMPA, GluR3
Glutamate-AMPA, GluR4c
Glutamate-KA
Glutamate-Kainate
Glutamate-Kainate 2
Glutamate-Kainate 4
Glutamate-Kainate 5
Glutamate-Kainate 7
Glutamate-Kainate EAA1
Glutamate-Kainate, GluR5
Glutamate-Kainate, GluR6
Glutamate-NMDA
Glutamate-NMDA-Channel
Glutamate-NMDA-Glycine
Glutamate-NMDA-MK801
Glutamate-NMDA-Polyamine
Glutamic acid decarboxylase
Glutamine synthetase
Glutaminyl cyclase
Glycine
Glycine, non-strychnine
Glycine, strychnine
Glycine-1-transporter
Glycine-2-transporter
Glycogen synthase kinase 3
Glycogen Synthase Kinase 3
Gonadotropin-Releasing Hormone, GnRH-R
GPR103
GPR109B
GPR7
GPR8
GR Alkaline Fosfatase
Grb2-SH2
Growth Hormone
Growth Hormone Secretagogue Receptor
GSK-3
H1
H2
H3
H4
h5-HT1A
h5-HT2A
h5-HT2B
halpha1B-adrenergic
halpha2C-adrenergic
HCV NS3
hD2L
hD3
Hemopoietic cell kinase
Heptyrosine aminotransferase, HepTAT
HER1
HER2
HERG
hH1
HISTAMINE H1
HISTAMINE H2
Histamine H2-Gs alpha S
HISTAMINE H3
Histamine H3L
HISTAMINE H4
Histaminergic H2
HIV-1 Protease Receptor
hM1
HSST1
HSST2
HSST3
HSST4
HSST5
hY1
hY2
hY5
Hypocretin receptor 1
Hypocretin receptor 2
ICaL
IGF-IR
IK1
IKK
IKr
Iks
IKv 1.1
IKv1.1
IKv1.5
Imidazoline 1
Imidazoline I1
Imidazoline I2
imipramine
INa
Indoleamine 2,3-Dioxygenase, IDO
Inositol Triphosphate
Inositol Triphosphate IP3
Inositol Trisphosphate 1
Inositol Trisphosphate 4
Inositol Trisphosphate 5
Insulin
insulin kinase-beta
Insulin receptor
Interleukin
Interleukin 1-Alpha
Interleukin 1-beta
Interleukin IL-1
Interleukin IL-2
Interleukin IL-6
interleukine-6
IP
IRK1
Itk
Ito
JAK3
Janus kinase 1 (a protein tyrosine kinase)
Janus kinase 2 (a protein tyrosine kinase)
KA
Kainate
Kappa
Kappa Opiate Receptor
KDR
KHEYLRF-NH2 (AF2)
Kinase insert domain receptor (a type III receptor tyrosine kinase)
Kinase insert domain(KDR)
KOP
KOR
L-type calcium channel (nifedipine)
Lck
Leptin
Leukocyte Antigen-Related tyrosine phosphatase
Leukotriene 2
Leukotriene b1
Leukotriene B4
Leukotriene B4 R1
Leukotriene B4 R2
Leukotriene Cysteinyl 1
Leukotriene Cysteinyl 2
Leukotriene D4
Leukotriene D4 Alpha
Leukotriene D4 Beta
Leukotriene LTB4
Leukotriene, Cysteinyl CysLT1
LIM domain kinase 1
Liver X, LXR alpha
Liver X, LXR beta
Luteinizing Hormone-Releasing Hormone LHRH
Lymphocyte-specific protein tyrosine kinase
Lysophosphatidic Acid 1
Lysophosphatidic Acid 2
Lysophosphatidic Acid 3
m-AChR
M1
M2
M3
M4
M5
malonyl-CoA decarboxylase, MCD
MAO A
MAO B
MAP kinase
MAP kinase interacting serine/threonine kinase 2
Map Kinase P38 Alpha
MAP Kinase P38 Beta
MAP Kinase P38 Delta
MAP Kinase P38 Gamma
MAP/microtubule affinity-regulating kinase 2
Matrix Metalloproteinase, MMP-1
Matrix Metalloproteinase, MMP-13
Matrix Metalloproteinase, MMP-2
Matrix Metalloproteinase, MMP-3
Matrix Metalloproteinase, MMP-8
Matrix Metalloproteinase, MMP-9
Matrix Metalloproteinase, MPP-2
Matrix Metalloproteinase, MPP-9
MDR1
MEK
Melanin Concentrating Hormone 1
Melanin Concentrating Hormone 2
Melanocortin MC1
Melanocortin MC3
Melanocortin MC4
Melanocortin MC5
Melatonin
Melatonin 1A
Melatonin 1B
Melatonin 1C
Met
Met proto-oncogene (hepatocyte growth factor receptor)
metabotropic glutamate 1
metabotropic glutamate 1/2
metabotropic glutamate 1/5-D
metabotropic glutamate 1/DA
Metabotropic Glutamate 1a
metabotropic glutamate 1b
metabotropic glutamate 1c
metabotropic glutamate 2
metabotropic glutamate 2/1
metabotropic glutamate 2/3
metabotropic glutamate 3
metabotropic glutamate 3/1a
metabotropic glutamate 3/1c
metabotropic glutamate 4
metabotropic glutamate 4/1-F
metabotropic glutamate 4a
metabotropic glutamate 5
metabotropic glutamate 5/1-C
metabotropic glutamate 5/1-F
metabotropic glutamate 5a
metabotropic glutamate 5b
metabotropic glutamate 6
metabotropic glutamate 7
metabotropic glutamate 8
Methionine Aminopeptidase, ecMetAP
mGluR5
mineralocorticoid
Mineralocorticoid receptor
Mitegen-Activated Protein Kinase Kinase
Mitogen-activated protein kinase 10
Mitogen-activated protein kinase 11
Mitogen-activated protein kinase 12
Mitogen-activated protein kinase 8
Mitogen-activated protein kinase 9
Mitogen-activated protein kinase kinase kinase 4
Mitogen-activated protein kinase kinase kinase 5
Mitogen-activated protein kinase kinase kinase kinase 5
Mixed Lineage Kinase-7, MLK-7K
MK2
Monoamine Oxidase A
Monoamine Oxidase B
Monoamine oxidaxe A
Monoamine oxidaxe B
Monoamine transporter
MOP
MOR
Motilin
MT1
MT1R
MT2
MT2R
Mu
Mu Opiate Receptor
Multidrug Resistance Transporter MDR 1
Muscarine Acetylcholine
Muscarinic
Muscarinic 1
Muscarinic 2
Muscarinic 3
Muscarinic 4
Muscarinic 5
Muscarinic Acetylcholine Receptor
Muscarinic Cholinergic
Muscarinic M1
Muscarinic M2
Muscarinic M3
Muscarinic M4
Muscarinic M5
Myosin light chain kinase 2, skeletal muscle
n-AChR
N-Formyl Peptide Receptor FPR1
N-Formyl Peptide Receptor-Like FPRL1
N-Methyl-D-Aspartate
NET
Neurokinin NK1
Neurokinin NK2
Neurokinin NK3
Neuromedin B
Neuromedin U NMU1
Neuromedin U NMU2
Neuronal acetylcholine receptor protein alpha-3 subunit
Neuronal acetylcholine receptor protein alpha-4 subunit
Neuronal acetylcholine receptor protein alpha-7 subunit
Neuropeptide Y
Neuropeptide Y1
Neuropeptide Y2
Neuropeptide Y5 long
Neuropeptide Y5 short
Neurotensin
Neurotensin 1
Neurotensin 2
Neurotensin receptor subtype 1
Neurotrophic tyrosine kinase, receptor, type 1
Neurotrophic tyrosine kinase, receptor, type 2
NGF
Nicotinic Acetlycholine
Nicotinic Acetylcholine alpha1
Nicotinic Acetylcholine alpha7
Nicotinic Acetylcholine, CNS
nicotinic ACh receptor (muscle)
nicotinic ACh receptor (neuronal)
Nicotinic Alpha-Bungarotoxin
Nicotinic Alpha2Beta2
Nicotinic Alpha2Beta4
Nicotinic Alpha3Beta2
Nicotinic Alpha3Beta4
Nicotinic Alpha4Beta2
Nicotinic Alpha4Beta4
Nicotinic Alpha7
nicotinic central
Nicotinic neuronal, alpha-BGTX-insensitive
NIH 3T3
NIMA (never in mitosis gene a)- related kinase 9
NIMA (never in mitosis gene a)-related kinase 2
NIMA (never in mitosis gene a)-related kinase 6
Nischarin
Nitric-oxide synthase, NOS (constitutive )
Nitric-oxide synthase, NOS (inducible)
Nitrogen oxide synthase - neuronal
NK
NMB
NMDA
NMDA PCP SITE
NMDA, agonism
NMDA, Glycine
NMDA, Phencyclidine
NMDA, Polyamine
Nociceptin receptor
Nociceptin/Orphanin FQ, NOP receptor
Non-receptor tyrosine kinase Tyk2
NOP
Noradrenaline Uptake
noradrenaline-alpha1
noradrenaline-alpha2A
noradrenaline-alpha2C
Norepinephrine transporter
Norepinephrine transporter
Norepinephrine Uptake
NOS
NOS neuronal
NPFF
NPFF2
NPY-Y1
NPY-Y2
NPY-Y4
NPY-Y5
NR2B
NR2B Channel Blocker
NRI
NT
OPIATE Delta
Opiate Delta 1
OPIATE Kappa
Opiate Kappa 1
OPIATE Kappa 3
OPIATE Mu
OPIATE Mu 1
OPIATE Mu 1B1
OPIATE Mu 1B2
OPIATE Mu 1B3
OPIATE Mu 1B4
OPIATE Mu 1B5
OPIATE Mu 2
Opiate non-selective
OPIATE ORL-1
OPIATE Sigma
OPIOID Delta
OPIOID Kappa
OPIOID Kappa 3
OPIOID Mu
OPIOID Mu 2
OPIOID Sigma
Organic Anion Transporter OATP1B3
Orphanin ORL1
ouabain
OX1R
OX2R
Oxytocin
P21 (CDKN1A)-activated kinase 3
P21 (CDKN1A)-activated kinase 6
P21(CDKN1A)-activated kinase 4
P21(CDKN1A)-activated kinase 7
P21/Cdc42/Rac1-activated kinase 1 (STE20 homolog, yeast)
P38 mitogen activated protein kinase
p3TP-Lux
PACAP
PACAP-27
PACAP-38
PAF Platelet activating factor
papain
PAR2
PARATHYROID HT1
PARATHYROID HT2
PBR
PCTAIRE protein kinase 1
PDE1
PDGF
PDGF-Rbeta
PGD2
phencyclidine
Phenylethanolamine-N-methyl transferase, PNMT
Phenylethanolamine-N-methyl transferase, PNMT-3
Phorbol ester
Phosphatidylcholine specific phospholipase C, PC-PLC
Phosphodiesterase 1
Phosphodiesterase 1-4
Phosphodiesterase 3
Phosphodiesterase 3A
Phosphodiesterase 3B
Phosphodiesterase 4
Phosphodiesterase 4A
Phosphodiesterase 4B
Phosphodiesterase 4C
Phosphodiesterase 4D
Phosphodiesterase 5
Phosphodiesterase 7A
Phosphodiesterase 8B
Phosphoinositide specific phospholipase C, PI-PLC
Phosphorylase kinase, gamma 1 (muscle)
Phosphorylase kinase, gamma 2 (testis)
Pim-1 oncogene
Pim-2 oncogene
PKA
PKC alpha
PKC beta
PKC gamma
PKC-alpha
PKC-beta2
Plasmepsin I
Plasmepsin II
Platelet-derived growth factor receptor, alpha polypeptid
Platelet-derived growth factor receptor, beta polypeptide
Polyamine Transporter
Potassium (voltage dependent)
Potassium Channel
Potassium channel (ATP modulatory)
Potassium Channel (Ca2+ dependent)
Potassium Channel HERG
Potassium Channel KA
Potassium Channel KATP
Potassium Channel SKCA
Potassium channel, Apamin
Potassium Channel, Ca2+ Act., VI
Potassium Channel, Ca2+ Act., VS
PPAR-delta
Pregnane X receptor
progesterone
Progesterone PR-B
Progesterone receptor
Prolactin Releasing Peptide Receptor
Prostaglandin D
Prostaglandin D2
Prostaglandin E1
Prostaglandin E2
Prostaglandin E3
Prostaglandin E4
Prostaglandin EP1
Prostaglandin EP2
Prostaglandin EP3
Prostaglandin EP4
Prostaglandin F
Prostaglandin H2
Prostaglandin I
Prostaglandin I2
Prostaglandin Transporter
ProstaglandinF2Alpha
Prostanid EP4
Prostanoid CRTH2
Prostanoid DP
Prostanoid EP2
Prostanoid, Thromboxane A2
Proteasome
Protein Kinase
Protein kinase C
Protein Kinase C- alpha
Protein Kinase C- delta
Protein Kinase D-GST
Protein Kinase G
Protein kinase, AMP-activated, alpha 1 catalytic subunit
Protein kinase, cAMP-dependent, catalytic, alpha
Protein kinase, membrane associated tyrosine/threonine 1
Protein Tyrosine Phosphatase 1B
Protein-tyrosine kinase Tie2
Proteinase-Activated Receptor 2
PrRP
PTK2 protein tyrosine kinase 2
PTK6 protein tyrosine kinase 6
Purinergic, P2X
Purinergic, P2X1
Purinergic, P2X2
Purinergic, P2X3
Purinergic, P2X4
Purinergic, P2X7
Purinergic, P2Y
PurinergicP2X2/3
r5-HT1A
Raf
rD2
Receptor-interacting serine-threonine kinase 2
Ret proto-oncogene
Retinoid X Receptor RXRalpha
Rho Kinase
Ribosomal protein S6 kinase, 90kDa, polypeptide 2
Ribosomal protein S6 kinase, 90kDa, polypeptide 3
Ribosomal protein S6 kinase, 90kDa, polypeptide 5
Rolipram
Ryanodine RyR3
S643b
Serine/threonine kinase 10
Serine/threonine kinase 16
Serine/threonine kinase 17a (apoptosis-inducing)
Serine/threonine kinase 17b (apoptosis-inducing)
Serine/threonine kinase 18
Serine/threonine kinase 3 mouse
Serine/threonine kinase 36 (fused homolog, Drosophila)
Serine/threonine kinase 38 like
Serine/threonine kinase 4
Serine/threonine kinase 6
Serotonin
Serotonin 5-HT1A
Serotonin 5-HT2A
Serotonin 5-HT2B
Serotonin 5-HT2C
Serotonin 5-HT7
Serotonin Reuptake Inhibitor
Serotonin Transporter
Serotonin Transporter (SERT)
Serotonin uptake
SERT
Serum/glucocorticoid regulated kinase
SH2-domain-containing phosphotyrosine phosphatase-2
Sigma
Sigma 1
Sigma 2
Sigma 2 PC12
Sigma 2 receptor
Sigma opioid receptor
Sigma, Non-Selective
Sigma-1
Sigma-2
Signal transducer and activator of transcription 3,Stat3
SLC-1
Small conductance calcium-activated potassium channel protein 3
Smoothened
Sodium (Site 1)
Sodium (Site 2)
Sodium Channel
Sodium Channel, Site 2
SOMATOSTATIN
SOMATOSTATIN SST1
SOMATOSTATIN SST2
SOMATOSTATIN SST3
SOMATOSTATIN SST4
SOMATOSTATIN SST5
sphingosine-1-phosphate 1 S1P1
sphingosine-1-phosphate 3 S1P3
sphingosine-1-phosphate 4 S1P4
sphingosine-1-phosphate 5 S1P5
Spleen tyrosine kinase
Src Kinase
STE20-like kinase (yeast)
Substance K
Substance P
Syk
Synaptic vesicular amine transporter
T Cell PTPase
TA1
TAAR1
tachykinin
Tachykinin NK1
Tachykinin NK2
Tachykinin NK3
TBOB
TBPS
TEK tyrosine kinase, endothelial (venous malformations, multiple cutaneous and mucosal)
Testosterone
TG 1019
Thrombin
Thrombin FIIa
Thrombin FXa
Thrombin trypsin
Thromboxane
Thromboxane A2
Thromboxane Alpha
Thromboxane B2
Thromboxane Beta
Thromboxane prostanoid
Thymidylate Synthase
thyroid alpha
thyroid beta
Thyroid Hormone
Thyrotropin Releasing Hormone
Thyrotropin-releasing Hormone
thyrotropin-releasing hormone R1
thyrotropin-releasing hormone R2
thyrotropin-releasing hormone R3
TMEM97
TNF-alpha
Topoisomerase I
TP
trace amine-associated receptor
TRAF2 and NCK interacting kinase
Transforming Growth Factor Beta RIIK
Transforming Growth Factor Beta RIK
Transforming Growth Factor-beta
TRH
Tripeptidyl Peptidase TPP II
tryptamine
TSPO
TTK protein kinase
Tumor Necrosis Factor alpha
Tumor Necrosis Factor, Non-selective
TXA2/PGH2
Tyrosine kinase receptor ron
Urotensin II
Urotensin-II
V-abl Abelson murine leukemia viral oncogene homolog
V-abl Abelson murine leukemia viral oncogene homolog 1
V-abl Abelson murine leukemia viral oncogene homolog 1 (E255K)
V-abl Abelson murine leukemia viral oncogene homolog 1 (H396P)
V-abl Abelson murine leukemia viral oncogene homolog 1 (M351T)
V-abl Abelson murine leukemia viral oncogene homolog 1 (Q252H)
V-abl Abelson murine leukemia viral oncogene homolog 1 (T3151)
V-abl Abelson murine leukemia viral oncogene homolog 1 (Y253F)
V-abl Abelson murine leukemia viral oncogene homolog 2
V-erb-b2 erythroblastic leukemia viral oncogene homolog 2
V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog (avian)
V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian)
V-yes-1 Yamaguchi sarcoma viral oncogene homolog 1
V-yes-1 Yamaguchi sarcoma viral related oncogene homolog
V1
V2
Vanilloid
Vanilloid receptor
Vanilloid VR1
Vascular Endothelial Growth Factor
Vasoactive Intestinal Peptide
Vasoactive Intestinal Peptide 1
VASOPRESSIN V1
VASOPRESSIN V1A
VASOPRESSIN V1B
VASOPRESSIN V2
Vasopressin V3
VEGF-R2
VIP
VIP 1
VIP 2
Vitamin D, VDR
Vitamin D3
VMAT1
VMAT2
Y1
Y2
Y4
Y5
Zacopride site-R
Zeta-chain (TCR) associated protein kinase 70kDa
Ki value (nM) less than
Ki value (nM) greater than