Configure Receptors:

Adrenaline Alpha1 Alpha2B (+) CIMBI-772 (+)CIMBI-775 (-) CIMBI-772 (-)CIMBI-775 1200015E14Rik 17Beta-HSD Type 3 3-Ethyl-3-{4-[4-(3-hydroxyphenyl)piperazin-1-yl]butyl}-1,3-dihydro-2H-indol-2-one 3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-1,3-dimethyl-1,3-dihydro-2H-indol-2-one 3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-3-(2-fluoroethyl)-1,3-dihydro-2H-indol-2-one 3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-3-methyl-1,3-dihydro-2H-indol-2-one 3-{4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl}-3-propyl-1,3-dihydro-2H-indol-2-one 5-HT Transporter 5-HT uptake 5-HT-S1 5-HT-S1A 5-HT1 5-HT1 like 5-HT1A 5-HT1B 5-HT1C 5-HT1D 5-HT1Dalpha 5-HT1Db 5-HT1DBeta 5-HT1E 5-HT1F 5-HT2 5-HT2A 5-HT2B 5-HT2C 5-HT2c VGI 5-HT3 5-HT4 5-HT5 5-HT5a 5-HT5B 5-HT6 5-HT7 5-HT7A 5-Lipoxygenase 5HT Transporter A2 a2b2 nicotinic cholinergic a2b4 nicotinic cholinergic A3 a3b2 nicotinic cholinergic a3b4 nicotinic cholinergic A4 a4b2 nicotinic cholinergic a4b4 nicotinic cholinergic Ac-AChBP Acetylcholinesterase Acetylcholinesterase, AChE AChE Activated p21cdc42Hs kinase Activator Protein AP-1 ADENOSINE ADENOSINE A1 ADENOSINE A1 high ADENOSINE A1 low ADENOSINE A2 ADENOSINE A2a ADENOSINE A2B ADENOSINE A3 Adenosine A4 Adenosine Deaminase ADA Adenosine Kinase, AK Adenosine transporter ADENOSINE UPTAKE Adenylate cyclase Adenylate cyclase Forskolin Adrenaline Adrenaline Alpha1 Adrenaline Alpha2 Adrenaline Beta Adrenaline 1 Adrenaline 2 Adrenaline alpha1 Adrenaline alpha2 Adrenaline Beta Adrenaline beta1 Adrenergic Alpha adrenergic Alpha1 adrenergic Alpha1A Adrenergic alpha1A/B adrenergic Alpha1B adrenergic Alpha1C adrenergic Alpha1D adrenergic Alpha2 adrenergic Alpha2A adrenergic Alpha2B adrenergic Alpha2C adrenergic Alpha2D adrenergic Beta adrenergic Beta1 adrenergic Beta1,2 adrenergic Beta2 adrenergic Beta3 Adrenomedullin AM1 Adrenomedullin AM2 Akt aldose reductase Aldosterone all-trans-retinoic acid, atRA Alpha 1 Adrenergic Receptor Alpha 1A Adrenergic Receptor Alpha 1B Adrenergic Receptor Alpha 2 Adrenergic Receptor Alpha 2A Adrenergic Receptor Alpha 2B Adrenergic Receptor Alpha 2C Adrenergic Receptor alpha-1 Alpha-1A Alpha-1B alpha-2 Alpha-2A alpha-2C Alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid alpha1 alpha1-Adrenocepter alpha1-GABA-A alpha1A alpha1B alpha1beta3gamma2 Alpha1D alpha2 alpha2-Adrenocepter alpha2-GABA-A Alpha2A Alpha2B alpha2beta2 alpha2beta3gamma2 alpha2beta4 Alpha2C alpha3-GABA-A alpha3beta2 alpha3beta3gamma2 alpha3beta4 alpha4bet2 alpha4beta2 alpha4beta3gamma2 alpha4beta4 alpha5-GABA-A alpha5beta3gamma2 alpha6-GABA-A alpha6beta3gamma2 alpha7 alphabeta3gamma2 AMPA Anandamid membrane transporter, AMT Anaphylatoxin C5a Anaplastic lymphoma kinase (Ki-1) androgen Androgen Receptor ANF Angiotensin ANGIOTENSIN AT1 Angiotensin AT2 Angiotensin II AT1 Angiotensin II AT1A Angiotensin II AT1B Angiotensin II AT2 Angiotensin II, central Angiotensin IV Angiotensin-converting enzyme, ACE ANP (Atrial natriuretic peptide) AP2 associated kinase 1 Apelin Arg-vasopressin V1 ATPase (Na+, K+) Atrial Natriuretic Factor atrial natriuretic peptide, ANP Aurora kinase C B lymphoid tyrosine kinase B1 B1 BRADYKININ B2 B2 BRADYKININ B3 BChE Benzodiazepine central Benzodiazepine peripheral Beta 1 Beta 2 Beta 3 Beta-1 Beta-2 beta-amyloid Beta-Amyloid (1-40) Beta-Amyloid (1-42) beta1 beta2 beta3 BHE BHSK BHSP Bile Salt Export Pump, BSEP BMP2 inducible kinase BMX non-receptor tyrosine kinase Bombesin Bombesin 1 Bombesin 2 Bombesin 3 Bombesin 4 Bombesin BB1 Bombesin BB2 Bombesin BB3 Bradykinin Bradykinin B1 Bradykinin B2 Bruton agammaglobulinemia tyrosine kinase butyrylcholinesterase, BuChE BZP BZP Rat Brain BZP Rat Brain Site C-src tyrosine kinase calcineurin Calcitonin Calcitonin Gene-Related Peptide Calcitonin Gene-related Peptide (CGRP) Calcitonin Gene-Related Peptide 1 Calcium (type L) Calcium channel Calcium channel (DHP) Calcium channel (Type L) Calcium channel (Type N) Calcium channel (Type T,L) Calcium channel (VER) Calcium channel diltiazem Calcium Channel L-Type, Benzothiazepine Calcium Channel L-Type, Dihydropyridine Calcium Channel L-Type, Phenylalkylamine Calcium Channel N-Type Calcium channel verapamil binding site Calcium/calmodulin-dependent protein kinase (CaM kinase) II alpha Calcium/calmodulin-dependent protein kinase (CaM kinase) II beta Calcium/calmodulin-dependent protein kinase (CaM kinase) II delta Calcium/calmodulin-dependent protein kinase (CaM kinase) II gamma Calcium/calmodulin-dependent protein kinase I Calcium/calmodulin-dependent protein kinase ID Calcium/calmodulin-dependent protein kinase IG Calcium/calmodulin-dependent protein kinase kinase 1, alpha Calcium/calmodulin-dependent protein kinase kinase 2, beta calmodulin kinase calpain calpain-1 CANNABINOID CB1 CANNABINOID CB2 Carbonic Anhydrase Isozymes, CA I Carbonic Anhydrase Isozymes, CA II Carbonic Anhydrase Isozymes, CA IX Carboxypeptidase CPG2 Casein kinase 1 Delta Casein kinase 1, epsilon Casein kinase 1, gamma 1 Casein kinase 1, gamma 2 casein kinase-1 casein kinase-2 caspase-2 caspase-3 caspase-6 caspase-7 caspase-8 Cathepsin D CB1 CB2 CBR CCK A CCK B CCR5 CD-45 CDC-like kinase 1 CDC-like kinase 2 CDC-like kinase 3 CDC-like kinase 4 CDC25 CDK1 CDK2 CDK4 CDK5 activator-binding protein C53 CGRP CGRP1 Chemoattractant receptor-homologous, CRTH2 Chemokine CCR1 Chemokine CCR2B Chemokine CCR4 Chemokine CCR5 Chemokine CX3CR1 Chemokine CXCR1 Chemokine CXCR2 Chemokine CXCR3 Chemokine CXCR4 Chemokine CXCR5 Chemokine CXCR7 Chemokine receptor 5 Chemokine US28 Chloride channel, TBOB Chloride ionophore Cholecystokinin Cholecystokinin 1 Cholecystokinin 2 Cholecystokinin A Cholecystokinin B Cholecystokinin central Cholecystokinin peripheral Choline Acetyltransferase Choline Transporter Choline Uptake Cholinergic, muscarinic Cholinergic, muscarinic M1 Cholinergic, muscarinic M2 Cholinergic, muscarinic M3 Cholinergic, muscarinic M4 Cholinergic, muscarinic M5 Cholinergic, nicotinic Cholinergic, nicotinic Alpha1 Cholinergic, Nicotinic Alpha1Beta1DeltaGamma Cholinergic, Nicotinic Alpha1Beta2 Cholinergic, Nicotinic Alpha2Beta2 Cholinergic, Nicotinic Alpha2Beta4 Cholinergic, Nicotinic Alpha3Beta2 Cholinergic, Nicotinic Alpha3Beta4 Cholinergic, Nicotinic Alpha3Beta4x Cholinergic, Nicotinic Alpha4Beta2 Cholinergic, Nicotinic Alpha4Beta2** Cholinergic, Nicotinic Alpha4Beta2X Cholinergic, Nicotinic Alpha4Beta4 Cholinergic, Nicotinic Alpha6 Cholinergic, Nicotinic Alpha6Beta2 Cholinergic, Nicotinic Alpha6Beta3Beta4Alpha5 Cholinergic, Nicotinic Alpha6Beta4 Cholinergic, Nicotinic Alpha7 Cholinergic, Nicotinic Alpha7/5-HT3 Cholinergic, Nicotinic Muscle CIMBI-712 CIMBI-717 CIMBI-772 CIMBI-775 Colchicine Corticotropin-Releasing Factor COX-1 COX-2 CRF CRF-R1 CRF-R2 Alpha CRF-R2 Beta CRF1 CRF2 Beta Ct-AChBP Cyclin G associated kinase Cyclin-dependent kinase 2 D1 D2 D2L D2S D3 D4 D4.4 D5 DAT Death-associated kinase 3 Death-associated protein kinase 2 Delta Delta Opiate Receptor Deoxyuridine triphosphatase Dihyrofolate Reductase, DHFR Dipeptidyl peptidase DPP II Dipeptidyl peptidase DPP IV DOP DOPAMINE DOPAMINE D1 Dopamine D1 high Dopamine D1 low Dopamine D1A Dopamine D1B DOPAMINE D2 DOPAMINE D2 Long DOPAMINE D2 Short DOPAMINE D2/D4 Dopamine D2A Dopamine D2B DOPAMINE D3 Dopamine D3A DOPAMINE D4 DOPAMINE D5 Dopamine Transporter Dopamine Uptake Dopamine, cocaine site Dopamine1-like Dopamine2-like DOR DP1 DRI Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A dUTPase EGF EGF-R Eledoisin ENDOTHELIN ENDOTHELIN A ENDOTHELIN B EP1 EP2 EP3 EP4 EPH receptor A2 EPH receptor A3 EPH receptor A4 EPH receptor A5 EPH receptor A6 EPH receptor A7 EPH receptor A8 EPH receptor B1 EPH receptor B2 EPH receptor B4 Epidermal growth factor receptor Erythropietin EPOR estrogen estrogen alpha estrogen beta Estrogen receptor alpha Estrogen receptor beta estrogen, ER alpha estrogen, ER beta Excitatory Amino Acid EAAT1 Excitatory Amino Acid EAAT2 Excitatory Amino Acid EAAT3 Export Pump, ABCC2 extracellular-regulated protein kinase, ERK Fatty Acid Amide Hydrolic, FAAH Fer (fps/fes related) tyrosine kinase (phosphoprotein NCP94) FGF FGF-R2 FGFR-1, (cyto) FGFR-1, (FL) Fibroblast growth factor receptor 1 Fibroblast growth factor receptor 2 Fibroblast growth factor receptor 3 FKBP12 Fms-related tyrosine kinase 3 Fms-related tyrosine kinase 4 Follicle-Stimulating Hormone, FSH Formyl peptide Receptor FP FYN oncogene related to SRC, FGR, YES Fyn-related kinase GABA GABA A GABA A alpha1 GABA A Alpha1Beta1Gamma2 GABA A Alpha1Beta2 GABA A Alpha1Beta2Gamma2 GABA A Alpha1Beta3Gamma2 GABA A alpha2 GABA A Alpha2Beta1Gamma2 GABA A Alpha2Beta2Gamma2 GABA A Alpha2Beta3Gamma2 GABA A alpha3 GABA A Alpha3Beta1Gamma2 GABA A Alpha3Beta2Gamma2 GABA A Alpha3Beta3Gamma2 GABA A Alpha4Beta2Gamma2 GABA A Alpha4Beta3Gamma2 GABA A Alpha4Gamma2 GABA A alpha5 GABA A Alpha5Beta1Gamma2 GABA A Alpha5Beta2Gamma2 GABA A Alpha5Beta3Gamma2 GABA A Alpha5m10Beta2Gamma2 GABA A Alpha5m8Beta2Gamma2 GABA A Alpha5m9Beta2Gamma2 GABA A alpha6 GABA A Alpha6Beta1Gamma2 GABA A Alpha6Beta2Gamma2 GABA A Alpha6Beta3Gamma2 GABA A anti-Alpha1 GABA A anti-Alpha3 GABA A Benzodiazepine GABA A Benzodiazepine brain GABA A Benzodiazepine liver GABA A Benzodiazepine omega1 GABA A Benzodiazepine omega2 GABA A Benzodiazepine omega5 GABA A Benzodiazepine Type I GABA A Benzodiazepine Type II GABA A Benzodiazepine Type IIL GABA A Benzodiazepine Type IIM GABA A Beta2Gamma2 GABA A Flunitrazepam, Central GABA A Muscimol, Central GABA A, agonist site GABA alpha1beta3gamma2 GABA alpha2beta3gamma2 GABA alpha3beta3gamma2 GABA alpha4beta3gamma2 GABA alpha5beta3gamma2 GABA alpha6beta3gamma2 GABA B GABA B rho 1 GABA B1A GABA B1B GABA C GABA receptor alpha-1 subunit GABA receptor alpha-2 subunit GABA receptor alpha-3 subunit GABA receptor alpha-5 subunit GABA transporter GABA uptake GABA, Chloride, TBOB GABA-A GABA-PICROTOXIN GABAA GABAa (Cl channel) GABAA alpha1beta3gamma2 GABAA alpha2beta3gamma2 GABAA alpha3beta3gamma2 GABAA alpha4beta3gamma2 GABAA alpha5beta3gamma2 GABAA alpha6beta3gamma2 GABAa1 receptor Gabapentin GALANIN Galanin R1 Galanin R2 Galanin R3 Gamma hydroxybutyric, GHB Gardner-Rasheed feline sarcoma viral (v-fgr) oncogene homolog Gastrin-Releasing peptide glucagon Glucocorticoid Glucocorticoid receptor GLUK5 GluR1 -40 mV GluR1 -80 mV Glutamate AMPA 1 Glutamate AMPA 2 Glutamate AMPA 3 Glutamate AMPA 4 Glutamate AMPA 5 Glutamate AMPA 6 Glutamate Chloride Glutamate delta 2 Glutamate, GluR1 Glutamate, GluR2 Glutamate, GluR4 Glutamate, GluR6 + KA2 Glutamate, GluR7 Glutamate, Non-selective Glutamate-AMPA Glutamate-AMPA, GluR1 Glutamate-AMPA, GluR2 (Q/R) Glutamate-AMPA, GluR3 Glutamate-AMPA, GluR4c Glutamate-KA Glutamate-Kainate Glutamate-Kainate 2 Glutamate-Kainate 4 Glutamate-Kainate 5 Glutamate-Kainate 7 Glutamate-Kainate EAA1 Glutamate-Kainate, GluR5 Glutamate-Kainate, GluR6 Glutamate-NMDA Glutamate-NMDA-Channel Glutamate-NMDA-Glycine Glutamate-NMDA-MK801 Glutamate-NMDA-Polyamine Glutamic acid decarboxylase Glutamine synthetase Glutaminyl cyclase Glycine Glycine, non-strychnine Glycine, strychnine Glycine-1-transporter Glycine-2-transporter Glycogen synthase kinase 3 Glycogen Synthase Kinase 3 Gonadotropin-Releasing Hormone, GnRH-R GPR103 GPR109B GPR7 GPR8 GR Alkaline Fosfatase Grb2-SH2 Growth Hormone Growth Hormone Secretagogue Receptor GSK-3 H1 H2 H3 H4 h5-HT1A h5-HT2A h5-HT2B halpha1B-adrenergic halpha2C-adrenergic HCV NS3 hD2L hD3 Hemopoietic cell kinase Heptyrosine aminotransferase, HepTAT HER1 HER2 HERG hH1 HISTAMINE H1 HISTAMINE H2 Histamine H2-Gs alpha S HISTAMINE H3 Histamine H3L HISTAMINE H4 Histaminergic H2 HIV-1 Protease Receptor hM1 HSST1 HSST2 HSST3 HSST4 HSST5 hY1 hY2 hY5 Hypocretin receptor 1 Hypocretin receptor 2 ICaL IGF-IR IK1 IKK IKr Iks IKv 1.1 IKv1.1 IKv1.5 Imidazoline 1 Imidazoline I1 Imidazoline I2 imipramine INa Indoleamine 2,3-Dioxygenase, IDO Inositol Triphosphate Inositol Triphosphate IP3 Inositol Trisphosphate 1 Inositol Trisphosphate 4 Inositol Trisphosphate 5 Insulin insulin kinase-beta Insulin receptor Interleukin Interleukin 1-Alpha Interleukin 1-beta Interleukin IL-1 Interleukin IL-2 Interleukin IL-6 interleukine-6 IP IRK1 Itk Ito JAK3 Janus kinase 1 (a protein tyrosine kinase) Janus kinase 2 (a protein tyrosine kinase) KA Kainate Kappa Kappa Opiate Receptor KDR KHEYLRF-NH2 (AF2) Kinase insert domain receptor (a type III receptor tyrosine kinase) Kinase insert domain(KDR) KOP KOR L-type calcium channel (nifedipine) Lck Leptin Leukocyte Antigen-Related tyrosine phosphatase Leukotriene 2 Leukotriene b1 Leukotriene B4 Leukotriene B4 R1 Leukotriene B4 R2 Leukotriene Cysteinyl 1 Leukotriene Cysteinyl 2 Leukotriene D4 Leukotriene D4 Alpha Leukotriene D4 Beta Leukotriene LTB4 Leukotriene, Cysteinyl CysLT1 LIM domain kinase 1 Liver X, LXR alpha Liver X, LXR beta Luteinizing Hormone-Releasing Hormone LHRH Lymphocyte-specific protein tyrosine kinase Lysophosphatidic Acid 1 Lysophosphatidic Acid 2 Lysophosphatidic Acid 3 m-AChR M1 M2 M3 M4 M5 malonyl-CoA decarboxylase, MCD MAO A MAO B MAP kinase MAP kinase interacting serine/threonine kinase 2 Map Kinase P38 Alpha MAP Kinase P38 Beta MAP Kinase P38 Delta MAP Kinase P38 Gamma MAP/microtubule affinity-regulating kinase 2 Matrix Metalloproteinase, MMP-1 Matrix Metalloproteinase, MMP-13 Matrix Metalloproteinase, MMP-2 Matrix Metalloproteinase, MMP-3 Matrix Metalloproteinase, MMP-8 Matrix Metalloproteinase, MMP-9 Matrix Metalloproteinase, MPP-2 Matrix Metalloproteinase, MPP-9 MDR1 MEK Melanin Concentrating Hormone 1 Melanin Concentrating Hormone 2 Melanocortin MC1 Melanocortin MC3 Melanocortin MC4 Melanocortin MC5 Melatonin Melatonin 1A Melatonin 1B Melatonin 1C Met Met proto-oncogene (hepatocyte growth factor receptor) metabotropic glutamate 1 metabotropic glutamate 1/2 metabotropic glutamate 1/5-D metabotropic glutamate 1/DA Metabotropic Glutamate 1a metabotropic glutamate 1b metabotropic glutamate 1c metabotropic glutamate 2 metabotropic glutamate 2/1 metabotropic glutamate 2/3 metabotropic glutamate 3 metabotropic glutamate 3/1a metabotropic glutamate 3/1c metabotropic glutamate 4 metabotropic glutamate 4/1-F metabotropic glutamate 4a metabotropic glutamate 5 metabotropic glutamate 5/1-C metabotropic glutamate 5/1-F metabotropic glutamate 5a metabotropic glutamate 5b metabotropic glutamate 6 metabotropic glutamate 7 metabotropic glutamate 8 Methionine Aminopeptidase, ecMetAP mGluR5 mineralocorticoid Mineralocorticoid receptor Mitegen-Activated Protein Kinase Kinase Mitogen-activated protein kinase 10 Mitogen-activated protein kinase 11 Mitogen-activated protein kinase 12 Mitogen-activated protein kinase 8 Mitogen-activated protein kinase 9 Mitogen-activated protein kinase kinase kinase 4 Mitogen-activated protein kinase kinase kinase 5 Mitogen-activated protein kinase kinase kinase kinase 5 Mixed Lineage Kinase-7, MLK-7K MK2 Monoamine Oxidase A Monoamine Oxidase B Monoamine oxidaxe A Monoamine oxidaxe B Monoamine transporter MOP MOR Motilin MT1 MT1R MT2 MT2R Mu Mu Opiate Receptor Multidrug Resistance Transporter MDR 1 Muscarine Acetylcholine Muscarinic Muscarinic 1 Muscarinic 2 Muscarinic 3 Muscarinic 4 Muscarinic 5 Muscarinic Acetylcholine Receptor Muscarinic Cholinergic Muscarinic M1 Muscarinic M2 Muscarinic M3 Muscarinic M4 Muscarinic M5 Myosin light chain kinase 2, skeletal muscle n-AChR N-Formyl Peptide Receptor FPR1 N-Formyl Peptide Receptor-Like FPRL1 N-Methyl-D-Aspartate NET Neurokinin NK1 Neurokinin NK2 Neurokinin NK3 Neuromedin B Neuromedin U NMU1 Neuromedin U NMU2 Neuronal acetylcholine receptor protein alpha-3 subunit Neuronal acetylcholine receptor protein alpha-4 subunit Neuronal acetylcholine receptor protein alpha-7 subunit Neuropeptide Y Neuropeptide Y1 Neuropeptide Y2 Neuropeptide Y5 long Neuropeptide Y5 short Neurotensin Neurotensin 1 Neurotensin 2 Neurotensin receptor subtype 1 Neurotrophic tyrosine kinase, receptor, type 1 Neurotrophic tyrosine kinase, receptor, type 2 NGF Nicotinic Acetlycholine Nicotinic Acetylcholine alpha1 Nicotinic Acetylcholine alpha7 Nicotinic Acetylcholine, CNS nicotinic ACh receptor (muscle) nicotinic ACh receptor (neuronal) Nicotinic Alpha-Bungarotoxin Nicotinic Alpha2Beta2 Nicotinic Alpha2Beta4 Nicotinic Alpha3Beta2 Nicotinic Alpha3Beta4 Nicotinic Alpha4Beta2 Nicotinic Alpha4Beta4 Nicotinic Alpha7 nicotinic central Nicotinic neuronal, alpha-BGTX-insensitive NIH 3T3 NIMA (never in mitosis gene a)- related kinase 9 NIMA (never in mitosis gene a)-related kinase 2 NIMA (never in mitosis gene a)-related kinase 6 Nischarin Nitric-oxide synthase, NOS (constitutive ) Nitric-oxide synthase, NOS (inducible) Nitrogen oxide synthase - neuronal NK NMB NMDA NMDA PCP SITE NMDA, agonism NMDA, Glycine NMDA, Phencyclidine NMDA, Polyamine Nociceptin receptor Nociceptin/Orphanin FQ, NOP receptor Non-receptor tyrosine kinase Tyk2 NOP Noradrenaline Uptake noradrenaline-alpha1 noradrenaline-alpha2A noradrenaline-alpha2C Norepinephrine transporter Norepinephrine transporter Norepinephrine Uptake NOS NOS neuronal NPFF NPFF2 NPY-Y1 NPY-Y2 NPY-Y4 NPY-Y5 NR2B NR2B Channel Blocker NRI NT OPIATE Delta Opiate Delta 1 OPIATE Kappa Opiate Kappa 1 OPIATE Kappa 3 OPIATE Mu OPIATE Mu 1 OPIATE Mu 1B1 OPIATE Mu 1B2 OPIATE Mu 1B3 OPIATE Mu 1B4 OPIATE Mu 1B5 OPIATE Mu 2 Opiate non-selective OPIATE ORL-1 OPIATE Sigma OPIOID Delta OPIOID Kappa OPIOID Kappa 3 OPIOID Mu OPIOID Mu 2 OPIOID Sigma Organic Anion Transporter OATP1B3 Orphanin ORL1 ouabain OX1R OX2R Oxytocin P21 (CDKN1A)-activated kinase 3 P21 (CDKN1A)-activated kinase 6 P21(CDKN1A)-activated kinase 4 P21(CDKN1A)-activated kinase 7 P21/Cdc42/Rac1-activated kinase 1 (STE20 homolog, yeast) P38 mitogen activated protein kinase p3TP-Lux PACAP PACAP-27 PACAP-38 PAF Platelet activating factor papain PAR2 PARATHYROID HT1 PARATHYROID HT2 PBR PCTAIRE protein kinase 1 PDE1 PDGF PDGF-Rbeta PGD2 phencyclidine Phenylethanolamine-N-methyl transferase, PNMT Phenylethanolamine-N-methyl transferase, PNMT-3 Phorbol ester Phosphatidylcholine specific phospholipase C, PC-PLC Phosphodiesterase 1 Phosphodiesterase 1-4 Phosphodiesterase 3 Phosphodiesterase 3A Phosphodiesterase 3B Phosphodiesterase 4 Phosphodiesterase 4A Phosphodiesterase 4B Phosphodiesterase 4C Phosphodiesterase 4D Phosphodiesterase 5 Phosphodiesterase 7A Phosphodiesterase 8B Phosphoinositide specific phospholipase C, PI-PLC Phosphorylase kinase, gamma 1 (muscle) Phosphorylase kinase, gamma 2 (testis) Pim-1 oncogene Pim-2 oncogene PKA PKC alpha PKC beta PKC gamma PKC-alpha PKC-beta2 Plasmepsin I Plasmepsin II Platelet-derived growth factor receptor, alpha polypeptid Platelet-derived growth factor receptor, beta polypeptide Polyamine Transporter Potassium (voltage dependent) Potassium Channel Potassium channel (ATP modulatory) Potassium Channel (Ca2+ dependent) Potassium Channel HERG Potassium Channel KA Potassium Channel KATP Potassium Channel SKCA Potassium channel, Apamin Potassium Channel, Ca2+ Act., VI Potassium Channel, Ca2+ Act., VS PPAR-delta Pregnane X receptor progesterone Progesterone PR-B Progesterone receptor Prolactin Releasing Peptide Receptor Prostaglandin D Prostaglandin D2 Prostaglandin E1 Prostaglandin E2 Prostaglandin E3 Prostaglandin E4 Prostaglandin EP1 Prostaglandin EP2 Prostaglandin EP3 Prostaglandin EP4 Prostaglandin F Prostaglandin H2 Prostaglandin I Prostaglandin I2 Prostaglandin Transporter ProstaglandinF2Alpha Prostanid EP4 Prostanoid CRTH2 Prostanoid DP Prostanoid EP2 Prostanoid, Thromboxane A2 Proteasome Protein Kinase Protein kinase C Protein Kinase C- alpha Protein Kinase C- delta Protein Kinase D-GST Protein Kinase G Protein kinase, AMP-activated, alpha 1 catalytic subunit Protein kinase, cAMP-dependent, catalytic, alpha Protein kinase, membrane associated tyrosine/threonine 1 Protein Tyrosine Phosphatase 1B Protein-tyrosine kinase Tie2 Proteinase-Activated Receptor 2 PrRP PTK2 protein tyrosine kinase 2 PTK6 protein tyrosine kinase 6 Purinergic, P2X Purinergic, P2X1 Purinergic, P2X2 Purinergic, P2X3 Purinergic, P2X4 Purinergic, P2X7 Purinergic, P2Y PurinergicP2X2/3 r5-HT1A Raf rD2 Receptor-interacting serine-threonine kinase 2 Ret proto-oncogene Retinoid X Receptor RXRalpha Rho Kinase Ribosomal protein S6 kinase, 90kDa, polypeptide 2 Ribosomal protein S6 kinase, 90kDa, polypeptide 3 Ribosomal protein S6 kinase, 90kDa, polypeptide 5 Rolipram Ryanodine RyR3 S643b Serine/threonine kinase 10 Serine/threonine kinase 16 Serine/threonine kinase 17a (apoptosis-inducing) Serine/threonine kinase 17b (apoptosis-inducing) Serine/threonine kinase 18 Serine/threonine kinase 3 mouse Serine/threonine kinase 36 (fused homolog, Drosophila) Serine/threonine kinase 38 like Serine/threonine kinase 4 Serine/threonine kinase 6 Serotonin Serotonin 5-HT1A Serotonin 5-HT2A Serotonin 5-HT2B Serotonin 5-HT2C Serotonin 5-HT7 Serotonin Reuptake Inhibitor Serotonin Transporter Serotonin Transporter (SERT) Serotonin uptake SERT Serum/glucocorticoid regulated kinase SH2-domain-containing phosphotyrosine phosphatase-2 Sigma Sigma 1 Sigma 2 Sigma 2 PC12 Sigma 2 receptor Sigma opioid receptor Sigma, Non-Selective Sigma-1 Sigma-2 Signal transducer and activator of transcription 3,Stat3 SLC-1 Small conductance calcium-activated potassium channel protein 3 Smoothened Sodium (Site 1) Sodium (Site 2) Sodium Channel Sodium Channel, Site 2 SOMATOSTATIN SOMATOSTATIN SST1 SOMATOSTATIN SST2 SOMATOSTATIN SST3 SOMATOSTATIN SST4 SOMATOSTATIN SST5 sphingosine-1-phosphate 1 S1P1 sphingosine-1-phosphate 3 S1P3 sphingosine-1-phosphate 4 S1P4 sphingosine-1-phosphate 5 S1P5 Spleen tyrosine kinase Src Kinase STE20-like kinase (yeast) Substance K Substance P Syk Synaptic vesicular amine transporter T Cell PTPase TA1 TAAR1 tachykinin Tachykinin NK1 Tachykinin NK2 Tachykinin NK3 TBOB TBPS TEK tyrosine kinase, endothelial (venous malformations, multiple cutaneous and mucosal) Testosterone TG 1019 Thrombin Thrombin FIIa Thrombin FXa Thrombin trypsin Thromboxane Thromboxane A2 Thromboxane Alpha Thromboxane B2 Thromboxane Beta Thromboxane prostanoid Thymidylate Synthase thyroid alpha thyroid beta Thyroid Hormone Thyrotropin Releasing Hormone Thyrotropin-releasing Hormone thyrotropin-releasing hormone R1 thyrotropin-releasing hormone R2 thyrotropin-releasing hormone R3 TMEM97 TNF-alpha Topoisomerase I TP trace amine-associated receptor TRAF2 and NCK interacting kinase Transforming Growth Factor Beta RIIK Transforming Growth Factor Beta RIK Transforming Growth Factor-beta TRH Tripeptidyl Peptidase TPP II tryptamine TSPO TTK protein kinase Tumor Necrosis Factor alpha Tumor Necrosis Factor, Non-selective TXA2/PGH2 Tyrosine kinase receptor ron Urotensin II Urotensin-II V-abl Abelson murine leukemia viral oncogene homolog V-abl Abelson murine leukemia viral oncogene homolog 1 V-abl Abelson murine leukemia viral oncogene homolog 1 (E255K) V-abl Abelson murine leukemia viral oncogene homolog 1 (H396P) V-abl Abelson murine leukemia viral oncogene homolog 1 (M351T) V-abl Abelson murine leukemia viral oncogene homolog 1 (Q252H) V-abl Abelson murine leukemia viral oncogene homolog 1 (T3151) V-abl Abelson murine leukemia viral oncogene homolog 1 (Y253F) V-abl Abelson murine leukemia viral oncogene homolog 2 V-erb-b2 erythroblastic leukemia viral oncogene homolog 2 V-kit Hardy-Zuckerman 4 feline sarcoma viral oncogene homolog (avian) V-src sarcoma (Schmidt-Ruppin A-2) viral oncogene homolog (avian) V-yes-1 Yamaguchi sarcoma viral oncogene homolog 1 V-yes-1 Yamaguchi sarcoma viral related oncogene homolog V1 V2 Vanilloid Vanilloid receptor Vanilloid VR1 Vascular Endothelial Growth Factor Vasoactive Intestinal Peptide Vasoactive Intestinal Peptide 1 VASOPRESSIN V1 VASOPRESSIN V1A VASOPRESSIN V1B VASOPRESSIN V2 Vasopressin V3 VEGF-R2 VIP VIP 1 VIP 2 Vitamin D, VDR Vitamin D3 VMAT1 VMAT2 Y1 Y2 Y4 Y5 Zacopride site-R Zeta-chain (TCR) associated protein kinase 70kDa

Receptor List:

Configure Compounds:

1-( 2,5-Dimet hoxy-4-propionylphenyl)-2-aminopropane HydrochlorideN-n -Propyl-2,5-dimethoxy-4-( 2-aminopropy1)benzamide Hydr... 1-(5-Chloropyridin-2-yl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(Aminomethyl)dibenzo[b,e]bicyclo[2.2.2]octadiene Hydrochloride 1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3-Iodophenyl-[2-methyl-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone 9-Aminomethyl-10,10-dimethyl-9,10-dihydroanthracene Oxalate 9-Aminomethyl-9,10-dihydro-9,10-methanoanthracene Hydrochloride 9-Methyl-9-aminomethyl-9,10-dihydroanthracene Oxalate α-Methylalanyl-L-proline butylamide hydrochloride hemihydrate (()-3-(2-Chloropyrimidin-5-yl)-8-azabicyclo[3/2/1]oct-2-ene Hydrochloride (()-3-(3-Pyridinyl)-8-azabicyclo[3/2/1]-oct-2-ene Maleate ((2R),1R, 2S,4R)-tetrahydrofuran-2-carboxylic acid [1-(3-bromobenzyl)-6-(2,4-dichlorophenyl)-4-(4-fluorophenylsulfanyl)-2-hyd... ((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methanamine ((4R,6S,7R)-7-phenyl-1-azaspiro[5.5]undecan-4-yl)methanol ((±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine ((±)-3,4-Methylenedioxymethamphetamine ((RS)-alpha-M4CPG) ((S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione (+) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin (+) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (+) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (+) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)(R)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+)(R)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+)(S)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2-(piperidin-1-yl)ethanone (+)(S)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2-(pyrrolidin-1-yl)ethanone (+)(S)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2-(thiomorpholin-4-yl)ethanone (+)-(1R,3'R)-Quinuclidin-3'-yl 1-(3-Thienyl)1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monooxalate (+)-(1S,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (+)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (+)-(3'R)-Quinuclidin-3'-yl 1-Benzyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (+)-(R)-4-Methyl-1-[2-(4-chlorophenoxy)-1-methyl-ethyl]piperidine hydrochloride (+)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-2-methyl-propyl]piperidine hydrochloride (+)-(S)-4-Methyl-1-[2-(4-chlorophenoxy)-propyl]piperidine hydrochloride (+)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-1-methyl-propyl]piperidine hydrochloride (+)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-butyl]piperidine hydrochloride (+)-1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (+)-1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (+)-1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine (+)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide (+)-1-[(1R)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride (+)-1-[(1S)-1-(3-Chlorophenyl)-2-(dimethylamino)ethyl]cyclohexanol (+)-1-[(1S)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride (+)-1-[(1S,2R,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (+)-1-[(1S,2S,5R)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (+)-1-{(1R)-2-(4-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride (+)-1-{(1S)-2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride (+)-1-{(1S,2R,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (+)-1-{(1S,2S,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (+)-2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole 2HCl (+)-2-Amino-6-propyltetrahydrobenzothiazole Dihydro 2HCl (+)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid (+)-2-Iodophenyl-[2-methyl-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone (+)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine (+)-3-(4-Chlorophenyl)-N'-[(4-cyanophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (+)-3-(4-Chlorophenyl)-N'-[(4-iodophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (+)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide (+)-5-(1-Methyl-2-pyrrolidinyl)-2-(3-phenylpropyl)pyridine (+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (+)-6-chloro-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (+)-6-fluorodinapsoline hydrobromide (+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazo... (+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazo... (+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole (+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole (+)-7-(2'-methylphenyl)-azepinoindoline (+)-7-Chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3] benzothiazepine (+)-8-hydroxy-2-(di-n-propylamino)tetralin (+)-9-Amino-6-methyl-5,6,6a,7-tetrahydro-4H-benzo [de]-thiazolo[4,5-g]quinoline 2HCl .5H2O (+)-alpha-Methylphenylethylamine (+)-Amphetamine (+)-Bridge-nicotine, (+)-Butaclamol (+)-Cimbi-772 (+)-Cimbi-775 (+)-Mefloquine (+)-Methyl(1S,2R,5R)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (+)-MK-801 (+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine (+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine (+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (+)-Phenmetrazine (+)-Pseudophenmetrazine (+)-SYA 09 (+)-t-ADA (+)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine (+)-trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione (+)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol (+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol (+)Mianserin (+)Niguldipine (+)Org3770 (+)trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (+)trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (+)trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+)trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+-)-MCPG (+-)Mianserin (+-)Org3770 (+/-) 9-Amino-6-methyl-5,6,6a,7-tetrahydro-4H-benzo [de]-thiazolo[4,5-g]quinoline (+/-) BMY-14802 (+/-) trans-4-(4' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid (+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]... (+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol (+/-)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+/-)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (+/-)-11-chlorodinapsoline hydrobromide (+/-)-11-nitrodinapsoline hydrobromide (+/-)-2,3-Dimethyldinapsoline hydrobromide (+/-)-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (+/-)-2-methyldinapsoline hydrobromide (+/-)-2-propyldinapsoline hydrobromide (+/-)-3,4-Dimethylnicotine Dioxalate (+/-)-3-Ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxylic Acid (+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide (+/-)-3-Fluoromethyl-7-(N-2,2,2-trifluoroethylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-3,3,3-trifluoropropylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-3-methoxypropylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-ethylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-propylaminosulfonyl)-THIQ (+/-)-3-Fluoromethyl-7-(N-thiomorpholinoaminosulfonyl)-THIQ (+/-)-3-Methyl-1,2,3,4-tetrahydroisoquinoline (+/-)-3-methyldinapsoline hydrobromide (+/-)-3-n-butyldinapsoline hydrobromide (+/-)-3-perfluorobutyldinapsoline hydrobromide (+/-)-3-trans-(Fluoromethyl)nicotine Oxalate (+/-)-3-trans-(Hydroxymethyl)nicotine (+/-)-3-trans-(Methoxymethyl)nicotine Dioxalate (+/-)-3-trans-Methylnicotine Dioxalate (+/-)-3alpha-Diphenylmethoxy-6beta-methoxymethoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-3alpha-Diphenylmethoxy-8-methyl-8-aza-bicyclo[3.2.1]octan-6beta-ol (+/-)-3alpha-[(4-Chlorophenyl)phenylmethoxy]-6beta-methoxymethoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-3alpha-[(4-Chlorophenyl)phenylmethoxy]-8-methyl-8-aza-bicyclo[3.2.1]octan-6beta-ol (+/-)-3alpha-[Bis(4-fluorophenyl)methoxy]-6alpha-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-3alpha-[Bis(4-fluorophenyl)methoxy]-6alpha-methoxymethoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-3alpha-[Bis(4-fluorophenyl)methoxy]-6beta-methoxymethoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-3alpha-[Bis-(4-fluorophenyl)methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octan-6alpha-ol (+/-)-3alpha-[Bis-(4-fluorophenyl)methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octan-6beta-ol (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(1-cyclopropylethyl)pyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(1-methylcyclopropyl)pyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(cyclopropylmethyl)pyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine (+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-tert-butylpyrimidin-2-amine (+/-)-6alpha-[Bis-(4-fluorophenyl)methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-6beta-[Bis-(4-fluorophenyl)methoxy]-8-methyl-8-aza-bicyclo[3.2.1]octane (+/-)-7,7'-dimethyldinapsoline hydrobromide (+/-)-7-Bromo-9,10-dihydro-9-(4-ethylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Bromo-9,10-dihydro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Bromo-9,10-dihydro-9-[4-(2'-hydroxy)ethylpiperazin-1-yl]pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9,10-dihydro-9-(4-ethylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9,10-dihydro-9-(4-methylhexahydro-1H-1,4-diazepin-1-yl)pyrrolo-[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9,10-dihydro-9-[4-(2'-hydroxy)ethylpiperazin-1-yl]pyrrolo-[2,1-b][1,3]benzothiazepine (+/-)-7-Chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3] benzothiazepine (+/-)-7-chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (+/-)-7-ethyldinapsoline hydrobromide (+/-)-7-methoxycarbonylmethyldinapsoline (+/-)-7-methyldinapsoline hydrobromide (+/-)-8-hydroxy-2-(di-n-propylamino)tetralin (+/-)-9,10-Dihydro-7-fluoro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-9,10-Dihydro-7-fluoro-9-[4-(2'-hydroxy)ethylpiperazin-1-yl]pyrrolo[2,1-b][1,3]benzothiazepine (+/-)-9,10-Dihydro-9-(4-ethylpiperazin-1-yl)-7-fluoropyrrolo[2,1-b][1,3]benzothiazepine (+/-)-9-(4-Methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (+/-)-AP5 (+/-)-BMY-1402 (+/-)-cis-1-Phenyl-3-(trimethylammoniumyl)-1,2,3,4-tetrahydronaphthalene Iodide (+/-)-Methyl 5-[({trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazin-1-yl}carbonyl)amino]pyridine-2-carboxylat... (+/-)-N-(4-(2-(Dimethylamino)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide monohydrochloride (+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride (+/-)-o-chloro-trans-H2-PAT (+/-)-o-methyl-trans-H2-PAT (+/-)-p-chloro-trans-H2-PAT (+/-)-p-fluoro-trans-H2-PAT (+/-)-p-methyl-trans-H2-PAT (+/-)-trans-10,11-dihydroxy-5,6,6a,7,8,12b-hexahydrobenzo[a]phenanthridine (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(1-oxidopyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(2-methylpyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(4-methylpyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(5-methylpyridin-3-yl)piperazine-1-carboxamide hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(6-methylpyridin-3-yl)piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-2-ylpiperazine-1-carboxamide Hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-3-ylpiperazine-1-carboxamide Hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-4-ylpiperazine-1-carboxamide Hydrochloride (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-2-ylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-4-ylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-5-ylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(methylthio)pyridin-3-yl]piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]piperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(2-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(4-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide Hydrochlorid... (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(5-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(6-hydroxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(6-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-ACPD (+/-)-trans-N-(2-Hydroxycyclopropyl)palmitamide (+/-)-trans-N-(6-Acetylpyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-N-(6-Aminopyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-N-(6-Chloropyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)-trans-N-(6-Cyanopyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide (+/-)3-(1-Phenylethoxycarbonyl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide (+/-)trans-4-(4' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (+_)-erythro-2-(1-Methylpiperidin-2-yl)-Chroman (+_)-erythro-5-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)-erythro-6-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)-erythro-7-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)-erythro-7-Hydroxy-2-(1-methylpyrrolidin-2-yl)chroman (+_)-erythro-8-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-2-(1-Methylpiperidin-2-yl)-Chroman (+_)threo-5-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-6-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-7-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (+_)threo-7-Hydroxy-2-(1-methylpyrrolidin-2-yl)chroman (+_)threo-8-Hydroxy-2-(1-methylpiperidin-2-yl)chroman (-) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin (-) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (-) trans-4-(3'-Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (-) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (-) trans-4-(4'-Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)(R)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2(thiomorphin-4-yl)ethanone (-)(R)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2(thiomorpholin-4-yl)ethanone (-)(R)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2-(piperidin-1-yl)ethanone (-)(R)-1-(1-Methyl-1H-pyrrol-2-yl)-2-phenyl-2-(pyrrolidin-1-yl)ethanone (-)(S)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (-)(S)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole (-)-(1S,3'R)-Quinuclidin-3'-yl 1-(3-Thienyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Mono-(-)-tartrate (-)-(2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (-)-(2S,5R)-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]piperazine-1-carboxamide (-)-(3'R)-Quinuclidin-3'-yl 1-Benzyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (-)-(R)-4-Methyl-1-[2-(4-chlorophenoxy)-propyl]piperidine hydrochloride (-)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-1-methyl-propyl]piperidine hydrochloride (-)-(R)-4-Methyl-1-[3-(4-chlorophenoxy)-butyl]piperidine hydrochloride (-)-(S)-4-Methyl-1-[2-(4-chlorophenoxy)-1-methyl-ethyl]piperidine hydrochloride (-)-(S)-4-Methyl-1-[3-(4-chlorophenoxy)-2-methyl-propyl]piperidine hydrochloride (-)-1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (-)-1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine (-)-1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine (-)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide (-)-1-[(1R)-1-(3-Chlorophenyl)-2-(dimethylamino)ethyl]cyclohexanol (-)-1-[(1R)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride (-)-1-[(1R,2R,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (-)-1-[(1R,2S,5S)-6-Benzyl-2-(pyrrolidin-1-yl)-6,8-diazabicyclo-[3.2.2]nonan-8-yl]-2-(3,4-dichlorophenyl)ethanone (-)-1-[(1S)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride (-)-1-{(1R)-2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride (-)-1-{(1R,2R,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (-)-1-{(1R,2S,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonan-8-yl}propan-1-one (-)-1-{(1S)-2-(4-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride (-)-2,6-Diamino-4,5,6,7-tetrahydrobenzothiazole 2HCl (-)-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine (-)-2-Amino-6-propyltetrahydrobenzothiazole Dihydro 2HCl (-)-2-aminoadipic acid (-)-2-Iodophenyl-[2-methyl-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone (-)-3-(3-Hydroxyphenyl)-N-nonylpyrrolidine (-)-3-(4-Chlorophenyl)-N'-[(4-cyanophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (-)-3-(4-Chlorophenyl)-N'-[(4-iodophenyl)sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine (-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide (-)-3-{(Cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)-1-methylpropyl]amino}-8-fluorochromane-5-carboxamide (-)-3-{Cyclobutyl[3-(5,7-difluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide (-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane- (-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-propylpyrimidin-2-amine (-)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide (-)-5-(1-Methyl-2-pyrrolidinyl)-2-(3-phenylpropyl)pyridine (-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (-)-5-OH-DPAT (-)-6-fluorodinapsoline hydrobromide (-)-7,9-difluoro-5-(6-methyl-7-oxa-bicyclo[4.1.0]hept-2-yl)-2,2,4-trimethyl 2,5-dihydro-(1H)-6-oxa-1-aza-chrysen (-)-7-Chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3] benzothiazepine (-)-8-hydroxy-2-(di-n-propylamino)tetralin (-)-9-Amino-6-methyl-5,6,6a,7-tetrahydro-4H-benzo [de]-thiazolo[4,5-g]quinoline 2HCl .5H2O (-)-Amphetamine (-)-Cimbi-772 (-)-Cimbi-775 (-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol (-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)-ferruginine (-)-Indolactam V (-)-Indolactam V (low PS) (-)-Mefloquine (-)-Methyl(1R,2S,5S)-8-[2-(3,4-Dichlorophenyl)acetyl]-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine (-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine (-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (-)-NANM (-)-nicotine (-)-Octylindolactam V (-)-Phenmetrazine (-)-Pseudophenmetrazine (-)-SYA 09 (-)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine (-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone (-)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol (-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol (-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline (-)cis-flupentixol (-)Mianserin (-)Org3770 (-)trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (-)trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine (-)trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (-)trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (1'RS)-(2S)-2-Amino-4-[(1'-aminoethyl)(hydroxy)phosphinyl]butyric Acid (1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-ylcarbamoyl)(phenyl)methyl acetate (1,2,3,4-Tetrahydro-acridin-9-yl)-[8-(1,2,3,4-tetrahydro-acridin-9-ylsulfanyl)-octyl]-amine (1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-carbamic acid benzyl ester (1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-yl)methanol (1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane (1-Benzenesulfonyl-5-fluoro-2-methyl-1H-indol-3-yl)-acetic acid (1-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (1-pentyl-3-(1-naphthoyl)indole) (JWH-018) (14-dimethylaminomethyl-6H,13H-pyrazino[1,2-a;4,5-a']diindol-7-ylmethyl)-dimethyl-amine (14S)-14-Hydroxydihydromorphinone (15R)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide (15R)-8-cyano-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxami... (15S)-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide (15S)-8-cyano-15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxami... (1H-Benzimidazol-2-yl)-thiazol-2-yl-amin (1H-Indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (1H-Indol-2-yl)-(4-phenethyl-piperazin-1-yl)-methanone (1H-Indol-2-yl)-(piperazin-1-yl)-methanone (1R)-2-(2-Chloropyrimidin-5-yl)-8-azabiyclo[3/2/1]oct-2-ene Hydrochloride (1R)-2-(2-Chloropyrimidin-5-yl)-9-azabicyclo[4/2/1]non-2-ene Hydrochloride (1R)-2-(3-Chloropyrazin-2-yl)-8-azabicyclo[3/2/1]oct2-ene (1R)-2-(3-Pyridinyl)-8-azabicyclo[3/2/1]oct-2-ene (1R)-3alpha-(4-Bromophenyl)tropane-2beta-carboxylic Acid Methyl Ester Tosylate (1R)-3alpha-(4-Chlorophenyl)tropane-2alpha-carboxylic Acid Methyl Ester tosylate (1R)-3alpha-(4-Methylphenyl)tropane-2alpha-carboxylic Acid Methyl Ester Tosylate (1R)-3alpha-Diphenylmethoxy-6beta-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (1R)-3alpha-Phenyltropane-2beta-carboxylic Acid Methyl Ester Tosylate (1R)-3alpha-[(4-Chlorophenyl)phenyl-methoxy]-6beta-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (1R)-3alpha-[Bis(4-fluorophenyl)methoxy]-6beta-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (1R)-3beta-(4-Bromophenyl)tropane-2alpha-carboxylic Acid Methyl Ester Fumarate (1R)-8-Azabicyclo[3/2/1]oct-2-ene-2-thiocarboxylic Acid Dimethylamide (1R)-8-Azabicyclo[3/2/1]oct-2-ene-carbocylic Acid Dimethylamide (1R)-8-Methyl-8-azabicyclo[3/2/1]oct-2-ene-2-carboxylic Acid Dimethylamide (1R)-8-Methyl-8-azabicyclo[3/2/1]oct-2-ene-2-thiocarboxylic Acid Dimethylamide (1R)-benzo[b]thiophen-3-yl((4aR)-1-(4-fluorophenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl)methanol (1R,13S,14R)-24-(cyclopropylmethyl)-13,20-dihydroxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa... (1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 (1R,2R,3R,4R,5S,7R,9S,10R)-1-Benzoyloxy-9-cinnamoyloxy-2,3-diacetoxy-dihydro-beta-agarofuran (1R,2R,3R,4R,5S,7R,9S,10R)-1-Benzoyloxy-9-cinnamoyloxy-2,3-dihydroxy-dihydro-beta-agarofuran (1R,2R,3R,4R,5S,7R,9S,10R)-2-Acetoxy-1-benzoyloxy-9-cinnamoyloxy-3-hydroxy-dihydro-beta-agarofuran (1R,2R,3R,4R,5S,7R,9S,10R)-3-Acetoxy-1-benzoyloxy-9-cinnamoyloxy-2-hydroxy-dihydro-beta-agarofuran (1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[... (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1R)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexa... (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1R)-cyclopropylpropyl)amino)- 9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((1S)-cyclopropyl-2- methylpropyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo- [3.1.0]hexa... (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((R)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- h... (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(((S)-cyclobutyl(cyclopropyl)- methyl)amino)-9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]- h... (1R,2R,3S,4R,5S)-4-(2-Chloro-6-((1-cyclopropylpropyl)amino)-9Hpurin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)amino)- 9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)amino)- 9H-purin-9-yl)-1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol(1R... (1R,2R,3S,4R,5S)-4-(2-Chloro-6-(dimethylamino)-9H-purin-9-yl)- 1-(hydroxymethyl)bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-... (1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol (1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol (1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol (1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol (1R,2R,3S,4S,5S,6R,7R,9S,10S)-1-Benzoyloxy-4-hydroxy-2,3,6,9,15-pentaacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1R,2R,4S)-2-(6-chloro-5-(3-methoxyphenyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane (1R,2R,4S)-2-(6-chloro-5-(4-fluorophenyl)pyridin-3-yl)-7-azabicyclo[2.2.1]heptane (1R,2R,4S)-2-(6-chloro-5-phenylpyridin-3-yl)-7-azabicyclo[2.2.1]heptane (1R,2R,5S )-6-benzyl-2-benzyloxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane (1R,2R,5S )-6-benzyl-2-methoxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane (1R,2R,5S )-6-benzyl-8-(2-phenylethyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol (1R,2R,5S )-6-benzyl-8-methyl-6,8-diazabicyclo[3.2.2]nonan-2-ol (1R,2R,5S)-methyl 8-(2-(3,4-dichlorophenyl)acetyl)-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (1R,2S)-(−)-N,N-diethylnorephedrine (1R,2S)-2-(tert-butylamino)-1-phenylpropan-1-ol (1R,2S)-N-Arachidonoylcyclopropanolamide (1R,2S)-N-Oleoylcyclopropanolamide (1R,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1R,2S,4R,5S,6R,7R,8S,9R,10S)-8,9-Dibenzoyloxy-1,2,6,15-tetraacetoxy-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-1,2,6,9,15-pentaacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-1,9-Dibenzoyloxy-2,6,15-triacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-9-Benzoyloxy-1,2,6,15-tetraacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4R,5S,6R,7R,9S,10S)-9-Benzoyloxy-1-hydroxy-2,6,15-triacetoxy-8-oxo-dihydro-beta-agarofuran (1R,2S,4S,5S) Acetic Acid 4-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonooxy-bicyclo[3.1.0]hex-1-ylmethyl Ester (1R,2S,4S,5S) Acetic Acid 4-(2-chloro-6-methylamino-purin-9-yl)-phosphonooxymethyl-bicyclo[3.1.0]hex-2-yl Ester (1R,2S,4S,5S) Phosphoric Acid mono-[4-(2-chloro-6-methylamino-purin-9-yl)-1-hydroxymethyl-bicyclo-[3.1.0] hex-2-yl] Ester (1R,2S,4S,5S) Phosphoric Acid mono-[4-(2-chloro-6-methylamino-purin-9-yl)-2-hydroxy-bicyclo[3.1.0]hex-1-ylmethyl] Ester (1R,2S,4S,5S,6R,7R,8S,9R,10R)-6-Acetoxy-4,8-dihydroxy-1,2,9-tribenzoyloxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,8S,9R,10S)-2,6-Diacetoxy-4-hydroxy,1,8,9-tribenzoyloxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,8S,9R,10S)-8,9-Dibenzoyloxy-4,15-dihydroxy-1,2,6-triacetoxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,8S,9R,10S)-8,9-Dibenzoyloxy-4-hydroxy-1,2,6,15-tetraacetoxy-dihydro-beta-agarofuran (1R,2S,4S,5S,6R,7R,9S,10S)-2,15-Diacetoxy-1,9-dibenzoyloxy-4,6-dihydroxy-8-oxo-dihydro-beta-agarofuran (1R,2S,5S )-6-Benzyl-8-(2-phenylethyl)-6,8-diazabidiazabicyclo (1R,2S,5S )-6-Benzyl-8-methyl-6,8-diazabicyclo-[3.2.2]nonan-2-ol (1R,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (1R,3'S)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (1R,3S)-1-(Aminomethyl)-3,4-dihydro-5,6-dihydroxy-3-phenyl-1H-2-benzopyran Hydrochloride (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid (1R,4R)-2-(2,5-diazabicyclo[2.2.1]hept-2-yl)-thieno[3,2-b]pyridine (1R,4R)-2-(3-methyl-(1,2,4)-thiadiazol-5-yl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(3-pyridinylmethyl)-2,5-diazabicyclo[2.2.1]-heptane (1R,4R)-2-(5,6-dichloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1R,4R)-2-(5-bromo-6-chloropyridine-3-sulfonyl)-2,5-diazabicyclo[2.2.1]heptane (1R,4R)-2-(5-trifluoromethyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-chloro-5-methoxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-chloro-5-methyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-chloropyridine-3-carbonyl)-2,5-diazabicyclo-[2.2.1]heptane (1R,4R)-2-(6-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1R,4R)-3-(2,5-diazabicyclo[2.2.1]hept-2-yl)-thieno[3,2-b]pyridine (1R,5S )-6-benzyl-8-methyl-6,8-diazabicyclo[3.2.2]-nonane-2-one dimethyl acetal (1R,9R,10S)-4-carbamoyl-17-(cyclopropylmethyl)-3,10-dihydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptad... (1R,9R,10S,13R)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-... (1R,9R,10S,13S)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-... (1R,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-15-(prop-2-en-1-yl)-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5... (1R,9R,18S,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^{1,32}.0^{2,7}.... (1RS,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate (1RS,3'R)-Quinuclidin-3'-yl 1-Phenylisoindoline-2-carboxylate (1S)-1-((4aR)-1-(4-fluorophenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl)but-3-en-1-ol (1S)-1-(4-ethoxyphenyl)-2-[4-(2-fluorophenyl)piperazin-1-yl]ethanol (1S)-3alpha-Diphenylmethoxy-6beta-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (1S)-3alpha-[(4-Chlorophenyl)phenylmethoxy]-6beta-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (1S)-3alpha-[Bis(4-fluorophenyl)methoxy]-6beta-methoxy-8-methyl-8-aza-bicyclo[3.2.1]octane (1S,11S,13S,17R,18R,20R,27S,29R,30R,31S,35E)-14,26-bis(cyclohex-2-en-1-yl)-35-(2-hydroxyethylidene)-19-phenyl-21-oxa-8,14,19,... (1S,11S,13S,17R,18R,20R,27S,29R,30R,31S,35E)-14,26-bis[(3,4-dimethoxyphenyl)methyl]-35-(2-hydroxyethylidene)-19-phenyl-21-oxa... (1S,11S,13S,17R,18R,20R,27S,29R,30R,31S,35E)-35-(2-hydroxyethylidene)-14,26-dimethyl-19-phenyl-21-oxa-8,14,19,26-tetraazadeca... (1S,11S,13S,18R,20R,27S,29R,30R,31S,35E)-35-(2-hydroxyethylidene)-14,26-bis[(4-nitrophenyl)methyl]-19-phenyl-21-oxa-8,14,19,2... (1S,2R)-(−)-N,N-diethylnorephedrine (1S,2R)-1-(3-methyl-1H-indol-1-yl)-3-(methylamino)-1-phenylpropan-2-ol (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((2-methoxyphenyl)ethynyl)- 6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((3-methoxyphenyl)ethynyl)- 6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((4-(hydroxymethyl)phenyl)- ethynyl)-6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((4-methoxyphenyl)ethynyl)- 6-(methylamino)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(2-((Z)-2-hydroxy-2-(pyrazin-2- yl)vinyl)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexane-1-carb... (1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-6-(methylamino)-9H-purin-9-yl)-N-methyl bicycle[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-6-(phenethylamino)-9H-purin-9-yl)-N-methyl bicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-4-(6-((Z)-2-hydroxy-2-phenylvinyl)-2-(phenylethynyl)-9H-purin-9-yl)-N-methylbicyclo[3.1.0]hexa... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(2-((1-methyl-1H-pyrazol-4-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)bicyclo[3.1.0]... (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(2-(4-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,3- triazol-1-yl)-6-(methylamino)-9H-purin-9... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(2-(methylamino)- 9H-purin-9-yl)bicycle[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (phenylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamid... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyrazin-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carb... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyridazin-3-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-ca... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyridin-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carb... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyridin-3-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carb... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyridin-4-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carb... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (pyrimidin-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-ca... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiophen-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-car... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiophen-3-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-car... (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2-(4-(pyrazin-2-yl)-1H-1,2,3- triazol-1-yl)-9H-purin-9-yl)bicyclo[... (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2-(4-(pyridin-2-yl)-1H-1,2,3- triazol-1-yl)-9H-purin-9-yl)bicyclo[... (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2-(4-(pyrimidin-2-yl)-1H-1,2,3- triazol-1-yl)-9H-purin-9-yl)bicycl... (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2-(4-phenyl-1H-1,2,3-triazol-1- yl)-9H-purin-9-yl)bicyclo[3.1.0]he... (1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-methyl-2-(pyrazin2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-... (1S,2R,3S,4R,5S)-4-(2-((1H-Pyrazol-3-yl)ethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1... (1S,2R,3S,4R,5S)-4-(2-((2-Chlorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1- ... (1S,2R,3S,4R,5S)-4-(2-((2-Fluorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1- ... (1S,2R,3S,4R,5S)-4-(2-((3,4-Difluorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane... (1S,2R,3S,4R,5S)-4-(2-((3,4-Difluorophenyl)ethynyl)-6-methyl-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carbo... (1S,2R,3S,4R,5S)-4-(2-((3,4-Difluorophenyl)ethynyl)-9H-purin-9- yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-((3-Fluorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1- ... (1S,2R,3S,4R,5S)-4-(2-((4,5-Dimethylfuran-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- ... (1S,2R,3S,4R,5S)-4-(2-((4-Chlorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1- ... (1S,2R,3S,4R,5S)-4-(2-((4-Fluorophenyl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1- ... (1S,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- he... (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((2-hydroxyethyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo... (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-((3,3,3-trifluoropropyl)-amino)-9H-purin-9-yl)-2,3-dihydroxy-N-methy... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-((cyclobutylmethyl)amino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicycl... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-((cyclopropylmethyl)amino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyc... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-((cyclopropylmethyl)amino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyc... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-(cyclobutylamino)-9H-purin-9-yl)- 2,3-dihydroxy-N-methylbicyclo[3.1.... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-(cyclopropylamino)-9H-purin-9-yl)- 2,3-dihydroxy-N-methylbicyclo[3.1... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-(ethylamino)-9H-purin-9-yl)-2,3- dihydroxy-N-methylbicyclo[3.1.0]hex... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-(isopropylamino)-9H-purin-9-yl)- 2,3-dihydroxy-N-methylbicyclo[3.1.0... (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]- h... (1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-2,3- dihydroxy-N-methylbicyclo[3.1.0]he... (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-methoxy-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane1-c... (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-6-methyl9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-ca... (1S,2R,3S,4R,5S)-4-(2-((5-Chlorothiophen-2-yl)ethynyl)-9H-purin9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-((5-Ethylfuran-2-yl)ethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane... (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexa... (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexa... (1S,2R,3S,4R,5S)-4-(2-((Ferrocen-yl)ethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carbo... (1S,2R,3S,4R,5S)-4-(2-(4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9H-purin-9- yl)-2,3-dihydroxy-N-methylbicycl... (1S,2R,3S,4R,5S)-4-(2-(4-(3,4-difluorophenyl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicy... (1S,2R,3S,4R,5S)-4-(2-(4-(5-bromothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbi... (1S,2R,3S,4R,5S)-4-(2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6- ((cyclobutylmethyl)amino)-9H-purin-9-yl)-2,3-dihyd... (1S,2R,3S,4R,5S)-4-(2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6- ((cyclopropylmethyl)amino)-9H-purin-9-yl)-2,3-dihy... (1S,2R,3S,4R,5S)-4-(2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6-(cyclobutylamino) - 9H-purin-9-yl)-2,3-dihydroxy-N-... (1S,2R,3S,4R,5S)-4-(2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6-(ethylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbi... (1S,2R,3S,4R,5S)-4-(2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylb... (1S,2R,3S,4R,5S)-4-(2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-6-(phenethylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-me... (1S,2R,3S,4R,5S)-4-(2-(4-(benzofuran-2-yl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9H-purin- 9-yl)-2,3-dihydroxy-N-methylbicyc... (1S,2R,3S,4R,5S)-4-(2-(4-(ferrocene-2-yl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9H-purin-9- yl)-2,3-dihydroxy-N-methylbicycl... (1S,2R,3S,4R,5S)-4-(2-(4-(furan-2-yl)-1H-1,2,3-triazol-1-yl)-6-(methylamino)-9H-purin-9-yl)- 2,3-dihydroxy-N-methylbicyclo[3.... (1S,2R,3S,4R,5S)-4-(2-(Benzofuran-2-ylethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-c... (1S,2R,3S,4R,5S)-4-(2-(Biphenyl-4-ylethynyl)-6-(methylamino)- 9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-car... (1S,2R,3S,4R,5S)-4-(2-(Cyclohexylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxam... (1S,2R,3S,4R,5S)-4-(2-(Cyclopropylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxa... (1S,2R,3S,4R,5S)-4-(2-(Furan-2-ylethynyl)-6-(methylamino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxam... (1S,2R,3S,4R,5S)-4-(2-azido-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-azido-6-(cyclobutylamino)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-azido-6-(ethylamino)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-azido-6-(methylamino)-9H-purin-9-yl)-2,3-dihydroxy-N-methyl bicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-azido-6-(phenethylamino)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)amino)-9Hpurin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carbox... (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)amino)-9Hpurin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((Z)-2-hydroxy-2-phenylvinyl)-9H-purin-9-yl)-2,3-dihydroxy)-N-methylbicyclo[3.1.0]hexane-1-car... (1S,2R,3S,4R,5S)-4-(2-Chloro-6-(dimethylamino)-9H-purin-9-yl)- 2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(2-Chloro-6-(dimethylamino)-9H-purin-9-yl)- 2,3-dihydroxybicyclo [3.1.0]hexane-1-carboxylic acid (1S,2R,3S,4R,5S)-4-(5-((5-chlorothiophen-2-yl)ethynyl)-7-(cyclopropylamino)-3H-imidazo[4,5- b]pyridin-3-yl)-2,3-dihydroxy-N-m... (1S,2R,3S,4R,5S)-4-(5-((5-chlorothiophen-2-yl)ethynyl)-7-(ethylamino)-3H-imidazo[4,5- b]pyridin-3-yl)-2,3-dihydroxy-N-methylb... (1S,2R,3S,4R,5S)-4-(5-((5-chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5- b]pyridin-3-yl)-2,3-dihydroxy-N-methyl... (1S,2R,3S,4R,5S)-4-(5-((5-chlorothiophen-2-yl)ethynyl)-7-(propylamino)-3H-imidazo[4,5- b]pyridin-3-yl)-2,3-dihydroxy-N-methyl... (1S,2R,3S,4R,5S)-4-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5b]pyridin-3-yl)-2,3-dihydroxy-N-methylbi... (1S,2R,3S,4R,5S)-4-(5-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol-1-yl)-7-(propylamino)-3Himidazo[4,5-b]pyridin-3-yl)-2,3-dih... (1S,2R,3S,4R,5S)-4-(6-((3-chlorobenzyl)amino)-2-(4-(5-chlorothiophen-2-yl)-1H-1,2,3-triazol- 1-yl)-9H-purin-9-yl)-2,3-dihydro... (1S,2R,3S,4R,5S)-4-(6-((3-chlorobenzyl)amino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(6-((Z)-2-(2-Chlorophenyl)-2-hydroxyvinyl)-2- (2-chlorophenyl)ethynyl)-9H-purin-9-yl)-2,3-dihydroxy-Nmethy... (1S,2R,3S,4R,5S)-4-(6-((Z)-2-(4-(tert-Butyl)phenyl)-2-hydroxyvinyl)-2-(4-(tert-butyl) phenyl)ethynyl)-9H-purin-9-yl)-2,3-dihy... (1S,2R,3S,4R,5S)-4-(6-(3-Chlorobenzylamino)-2-((3,4- difluorophenyl)ethynyl)-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.... (1S,2R,3S,4R,5S)-4-(6-(butylamino)-2-((5-chlorothiophen-2-yl)ethynyl)-9H-purin-9-yl)-2,3- dihydroxy-N-methylbicyclo[3.1.0]hex... (1S,2R,3S,4R,5S)-4-(6-(cyclobutylamino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxy-Nmethylbicyclo[3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(6-(ethylamino)-2-iodo-9H-purin-9-yl)-2,3-dihydroxy-N-methylbicyclo [3.1.0]hexane-1-carboxamide (1S,2R,3S,4R,5S)-4-(7-(Ethylamino)-5-((5-fluorothiophen-2-yl)ethynyl)-3H-imidazo[4,5b]pyridin-3-yl)-2,3-dihydroxy-N-methylbic... (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxam... (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-car... (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.... (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1... (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-car... (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane... (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexan... (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbo... (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexan... (1S,2R,3S,4R,5S)-4-[5-[2-(5-chlorothiophen-2-yl)ethynyl]-7-(methylamino)imidazo[4,5-b]pyridin-3-yl]-2,3-dihydroxy-N-methylbic... (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane... (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicycl... (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.... (1S,2R,3S,4R,5S)-N-(2-Acetamidoethyl)-4-(2-chloro-6- ((dicyclopropylmethyl)amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo- [3.1.0... (1S,2R,3S,4R,5S)-N-(2-Aminoethyl)-4-(2-chloro-6- ((dicyclopropylmethyl)amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo- [3.1.0]hex... (1S,2R,3S,4R,5S)-N-(2-aminoethyl)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1... (1S,2R,3S,4R,5S)-N-(3-Acetamidopropyl)-4-(2-chloro-6- ((dicyclopropylmethyl)amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo- [3.1.... (1S,2R,3S,4R,5S)-N-(3-Aminopropyl)-4-(2-chloro-6- ((dicyclopropylmethyl)amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo- [3.1.0]he... (1S,2R,4S)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1S,2R,6S,14R,15S,16R)-3-(cyclopropylmethyl)-16-[(2R)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-3-azahexacyclo[13.2... (1S,2S)-1-[(R)-2-[4-(2,4-Dimethylphenyl)piperazyl]-ethyl]-2-methyl-2-phenylcyclopropane (1S,2S)-1-[(S)-2-[4-(2,4-Dimethylphenyl)piperazyl]-ethyl]-2-methyl-2-phenylcyclopropane (1S,2S)-1-[4-(2,4-Dimethylphenyl)piperazyl]methyl-2-methyl-2-phenylcyclopropane (1S,2S)-N-Arachidonoylcyclopropanolamide (1S,2S)-N-Oleoylcyclopropanolamide (1S,2S,13R,21R)-22-(cyclopropylmethyl)-2-hydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{1... (1S,2S,3R,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- ((3-(trifluoromethyl)phenyl)ethynyl)-9H-purin-9-yl)bicyclo[3.1.... (1S,2S,3R,4R,5S)-2,3-dihydroxy-N-methyl-4-(6-(methylamino)-2- (thiazol-2-ylethynyl)-9H-purin-9-yl)bicyclo[3.1.0]hexane-1-carb... (1S,2S,4R)-1-aminocyclopentane-1,2,4-tricarboxylic acid (1S,2S,5R)-methyl 8-(2-(3,4-dichlorophenyl)acetyl)-2-(pyrrolidin-1-yl)-6,8-diazabicyclo[3.2.2]nonane-6-carboxylate (1S,2S,5R,6S)-2-[(2'S)-(2'-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylicAcid (1S,2S,7S,8R,12S,20R,24R,32R)-9,33-bis(cyclopropylmethyl)-2,7-dihydroxy-19,25-dioxa-9,22,33-triazaundecacyclo[24.9.1.1^{8,14}... (1S,3'S)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate Monohydrochloride (1S,3R)-1-aminocyclopentane-1,3-dicarboxylic (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid (1S,4S)-2-(2-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(2-quinolinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(2-thiazolyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-methylisothiazol-5-yl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(3-nitrophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-pyridazinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(3-quinolinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(4-chloro-1-phthalazinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(4-nitrophenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(4-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-(5-aminocarbonyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(5-aminomethyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(5-cyano-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(5-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(5-pyrimidinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-1,3-pyrimidin-4-yl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-3-pyridinyl)-5,5-dimethyl-2,5-diazabicyclo-[2.2.1]heptanium iodide (1S,4S)-2-(6-chloro-3-pyridinyl)-5-ethyl-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-chloro-3-pyridinyl)-5-methyl-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(6-chloro-5-hydroxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(6-chloro-5-methyl-3-pyridazinyl)-2,5-diazabicyclo-[2.2.1]heptane (1S,4S)-2-(6-chloropyridin-3-yl)-2,5-diazabicyclo[2.2.1]-heptanone (1S,4S)-2-(6-fluoro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-methyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(6-nitro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane (1S,4S)-2-(phenyl)-2,5-diazabicyclo[2.2.1]heptane (1S,4S)-2-[5-hydroxy-3-pyridinyl]-2,5-diazabicyclo[2.2.1]-heptane (1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,... (1S,5R,13R,14S,17S)-4-(cyclobutylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(1... (1S,5R,13R,14S,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,... (1S,5R,13R,17R)-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxa... (1S,5R,13R,17S)-10-carbamoyl-4-(cyclopropylmethyl)-17-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.... (1S,5R,13R,17S)-17-hydroxy-14-oxo-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18... (1S,5R,13S,14S,17R)-14-hydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)... (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-... (1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octad... (1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide (1S,9R,10S)-17-(cyclobutylmethyl)-10-hydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-triene-4-carboxamide (1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxa... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis(cyclohex-2-en-1-yl)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundeca... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis(naphthalen-2-ylmethyl)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaund... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(2E)-but-2-en-1-yl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundeca... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(3,4-dimethoxyphenyl)methyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetra... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(4-bromophenyl)methyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaund... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[(4-nitrophenyl)methyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaund... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-bis[2-(acetyloxy)ethyl]-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundeca... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-dibenzyl-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-dimethyl-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^... (1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-15,31-bis(prop-2-en-1-yl)-10,26-dioxa-8,15,24,31-tetraazaundecacycl... (2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(4,4-difluoropiperidin-1-yl)methanone (2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2,2-diphenyl-[1,3]dioxolo[4,5-c]pyridin-6-yl)-piperidin-1-ylmethanone (2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(1‐phenylpiperidin‐4‐yl)methyl]amine (2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(4‐phenylphenyl)methyl]amine (2-(2,4-dichlorophenyl)-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2-(2,4-dichlorophenyl)-6-fluoro-2-(2-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone (2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2-(2,4-dichlorophenyl)-6-fluoro-2-(4-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (2-(2-chloro-4-fluorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3,4-dichlorophenoxy)-5-(4-(4-fluoropiperidin-1-yl)but-1-ynyl)phenyl)-N-methylmethanamine (2-(3,4-dichlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3,4-dichlorophenoxy)-5-(4-thiomorpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3-chlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(3-fluorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(4-chloro-3-(trifluoromethyl)phenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(4-chlorophenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)-N-methylmethanamine (2-(Methylamino)-4-phenylthiazol-5-yl)(phenyl)methanone (2-Amino-1-(4-chlorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone (2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ2-(4-chlorophenylamino)-4-methylthiazol-5-yl)methanone (2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (p-tolylamino)thiazol-5-yl)methanone (2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone (2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-phenyl-2- (phenylamino)thiazol-5-yl)methanone (2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2- morpholino-4-phenylthiazol-5-yl)methanone (2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2-(4- chlorophenylamino)-4-methylthiazol-5-yl)methanone (2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-methyl2-(phenylamino)thiazol-5-yl)methanone (2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-phenyl2-(phenylamino) thiazol-5-yl)methanone (2-Amino-1-p-tolyl-1H-imidazol-5-yl)IJ2-morpholino-4- phenylthiazol-5-yl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(2,6-difluorophenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(2-methoxyphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(2-methylphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(3,4- methylenedioxyphenyl)thiophen-3-yl)(4-chlorophenyl) methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(3-methoxyphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(3-methylphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4- (trifluoromethoxy)phenyl)thiophen-3-yl)(4-chlorophenyl) methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-(1-(methyl)ethyl) phenyl)thiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-(2-(methoxy) ethoxy)phenyl)thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-fluorophenyl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(3,4-dichloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(3-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(3-trifluoro-methylphenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methoxyphenyl) thiophen-3-yl)(4-methyl-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(4-methylphenyl) thiophen-3-yl)(4-chloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(furan-2-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(furan-3-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(pyrazol-4-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(pyridin-2-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(pyridin-3-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(pyridine-4-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(thiophen-2-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-(thiophen-3-yl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3,4-dichloro-phenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3-chlorophenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (3-trifluoromethylphenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-bromothiophen-3-yl) (4-methylphenyl)methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (2,4-dichlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (2-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3,4-dichlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (3-trifluoromethylphenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (4-chlorophenyl)-methanone (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (4-methylphenyl)-methanone (2-Amino-4-isobutylthiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-(2,3-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-(2,4-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-(2,5-difluorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-(3,4-dichlorophenyl)-4-(2,2- dimethylpropyl)thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-5-(3,5-dimethylisoxazol-4-yl)-4-(2,2- dimethylpropyl)thiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-(4-chlorophenyl)-4-(2,2-dimethylpropyl) thiophen-3-yl)(4-chlorophenyl)-methanone (2-Amino-5-bromo-4-methylthiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-methyl-4-phenylthiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-p-methoxyphenyl-4-methylthiophen-3-yl)(4-chlorophenyl)methanone (2-Amino-5-phenyl-4-methylthiophen-3-yl)(4-chlorophenyl)methanone (2-Aminoethyl)benzene (2-Bromo-5-(4-(((2,4-difluorobenzyl)(2-methyl-3-((methylsulfonyl)amino)phenyl)amino)methyl)phenoxy)phenoxy)acetic Acid (2-Chloro-5-{4-[((2,4-difluorobenzyl){2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic Acid (2-chloroethyl)(2-(methylsulfonyloxyethyl)amino)aminobenzyl-L-glutamic acid (23R, 25R)-DLAM-03I (23R, 25R)-DLAM-2P (23R, 25R)-DLAM-3P (23R, 25R)-DLAM-4P (23R, 25R)-DLAM-MPM (23R, 25S)-DLAM-03I (23R, 25S)-DLAM-2P (23R, 25S)-DLAM-3P (23R, 25S)-DLAM-4P (23R, 25S)-DLAM-MPM (23R,25R)-DLAM-1P (23R,25S)-DLAM-1P (23S, 25R)-DLAM-03I (23S, 25R)-DLAM-2P (23S, 25R)-DLAM-3P (23S, 25R)-DLAM-4P (23S, 25R)-DLAM-MPM (23S, 25S)-DLAM-03I (23S, 25S)-DLAM-1P (23S, 25S)-DLAM-2P (23S, 25S)-DLAM-3P (23S, 25S)-DLAM-4P (23S, 25S)-DLAM-MPM (23S,25R)-DLAM-1P (2E)-3-[6-(Acetylamino)-3-pyridinyl]-N-{2-[2,4-dichloro-3-({[2-methoxy-1-(2-methoxyethyl)-1H-benzimidazol-4-yl]oxy}methyl)met... (2E)-N-{2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(2-pyridinylmethoxy)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl}-3-{6-[(4-py... (2R)-1-(4-pyridin-2-ylpiperazin-1-yl)-3-(thiophen-2-ylmethoxy)propan-2-ol (2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine (2R)-1-indol-1-yl-N-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]propan-2-amine (2R)-1-[(2-amino-6-chloropyrimidin-4-yl)amino]-3-(3,4-dihydro-1H-isoquinolin-2-yl)propan-2-ol (2R)-1-[(2-methylpropan-2-yl)oxy]-3-[4-(thiophen-2-ylmethyl)piperazin-1-yl]propan-2-ol (2R)-1-[4-(2-fluorophenyl)piperazin-1-yl]-3-[[(2S)-oxolan-2-yl]methoxy]propan-2-ol (2R)-1-[4-[(5-chlorothiophen-2-yl)methyl]piperazin-1-yl]-3-[(2-methylpropan-2-yl)oxy]propan-2-ol (2R)-2-(4-fluorophenyl)-2-[[1-(pyridin-2-ylmethyl)piperidin-4-yl]amino]acetamide (2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine (2R)-8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one (2R)-8-{4-[3-(7-Fluoro-1H-indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one (2R)-Amino-3-(4-hydroxyphenyl)-N-{1-[4-(3-hydroxyphenyl)-3R,4R-dimethyl-piperidin-1-ylmethyl]-2-methyl-1-propyl}propanamide (2R,2'R))-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2R,2'R)-2-(1-methyl-2-pyrrolidinyl)-1,4-benzodioxane hydrochloride (2R,2'S)-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2R,3R)-3-chloro-N-[2-(1H-imidazol-4-yl)ethyl]-2,3-dihydro-1-benzothiophene-2-carboxamide (2R,3R)-Hydroxybupropion (2R,3R)-OH-bupropion (2R,4S)-4-Cyanonicotine Dioxalate (2R,6S)-1-Methyl-2,6-bis-(2-naphthalen-1-yl-ethyl)-piperidine (2RS,3'R)-Quinuclidin-3'-yl 1-Phenyl-1,2,3,4-tetrahydroquinoline-2-carboxylate (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-bromo-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-chloro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2RS,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (2RS,3RS)-Hydroxybupropion (2S)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}pyrrolidine-2-carboxamide (2S)-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)amino]-2-benzyl-3-oxopropanoyl}amino)p... (2S)-2-Amino-4-[(1'-aminoethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(2'-Aminoethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(2'-Carboxyethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(aminomethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-Amino-4-[(hydroxymethyl)(hydroxy)phosphinyl]butyric Acid (2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]-3-phenylpropanoic acid bis(tetraflurobor... (2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]-3-phenylpropanoic acid bis(tetrafluorobor... (2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]propanoic acid bis(tetrafluoroborate) (2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]propanoic acid bis(tetrafluoroborate) (2S)-2-{[4-(6-Bromoquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-2-{[4-(6-Chloroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-2-{[4-(6-Fluoroquinolin-2-yl)-1,4-diazepan-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline (2S)-2-{[4-(6-Fluoroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-4-methyl-2-[[(3S)-3-methyl-4-[2-(3-methylphenoxy)ethyl]piperazin-1-yl]methyl]morpholine (2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine (2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl (2S)-6-allyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol (2S)-8-Methyl-2-({4-[6-(trifluoromethoxy)quinolin-2-yl]piperazin-1-yl}methyl)-2,3-dihydro-[1,4]dioxino[2,3-f]quinoline (2S)-8-Methyl-2-[(4-quinolin-2-yl-1,4-diazepan-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]-quinoline (2S)-8-Methyl-2-[(4-quinolin-2-ylpiperazin-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-8-Methyl-2-{[(2R)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline (2S)-8-Methyl-2-{[(2S)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline (2S)-8-Methyl-2-{[4-(6-nitroquinolin-2-yl)piperazin-1-yl]-methyl}-2,3-dihydro[1,4]dioxino[2,3-f]quinoline (2S)-8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one (2S)-8-{4-[3-(5-Fluoro-1H-indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one (2S)-8-{4-[3-(7-Fluoro-1H-indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one (2S)-Amino-3-(4-hydroxyphenyl)-N-{1-[4-(3-hydroxyphenyl)-3R,4R-dimethylpiperidin-1-ylmethyl]-2-methyl-1-propyl}propanamide (2S)-Aminobutyryl-(2S)-azetidine carboxamide trifluoroacetate hydrate (2S)-Aminobutyryl-(2S)-indoline carboxylic acid ethylamide hydrogen oxalate hydrate (2S)-Aminobutyryl-(2S)-indoline carboxylic acid methylamide hydrogen oxalate hydrate (2S)-Aminobutyryl-(2S)-indoline carboxylic acid propylamide hydrogen oxalate hydrate (2S)-Aminobutyryl-(4S)-fluoro-L-proline n-Butylamide Trifluoroacetate (2S)-Aminobutyryl-(R)-pipecolinic acid amide trifluoroacetate (2S)-Aminobutyryl-(S)-nipecotamide hydrogen oxalate (2S)-Aminobutyryl-4-cis-benzyl-L-proline n-butylamide Hydrogen Oxalate (2S)-Aminobutyryl-4-thia-L-prolinamide trifluoroacetate hemihydrate (2S)-Aminobutyryl-L-pipecolinic acid n-butylamide trifluoroacetate (2S)-Aminobutyryl-L-prolinamide trifluoroacetate hemihydrate (2S)-Aminobutyryl-L-proline (R)-sec-butylamide hydrogen oxalate (2S)-Aminobutyryl-L-proline 3-methylthiopropylamide hydrogen oxalate hemihydrate (2S)-Aminobutyryl-L-proline isobutylamide trifluoroacetate (2S)-Aminobutyryl-L-proline n-butylamide hydrogen oxalate (2S)-Aminobutyryl-L-proline n-pentylamide hydrogen oxalate (2S)-Aminobutyryl-L-proline n-propylamide trifluoroacetate (2S)-Aminobutyryl-L-proline-(2S)-methylbutylamide hydrogen oxalate hemihydrate (2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine (2S, 1'S, 2'S)-2-(carboxycyclopropyl)glycine (2S,2'R-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2S,2'S)-2-(1-methyl-2-pyrrolidinyl)-1,4-benzodioxane hydrochloride (2S,2'S-2-(2,3-dihydrobenzo[b][1,4]dioxin-2-yl)pyrrolidine hydrochloride (2S,3S) OH-bupropion (2S,3S)-2-(2-morpholin-2-yl-2-phenylmethoxy) phenol (2S,3S)-Hydroxybupropion (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carbox... (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-ca... (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-car... (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-ca... (2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-car... (2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetr... (2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetra... (2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide (2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate (2S,3S,4R,5S)-5-(6-(cyclopentylamino)-9H-purin-8-yl)-3,4-dihydroxy-N-(1-(4-(N-(1-phenethylpiperidin-4-yl)propionamido)phenyl)... (2S,3S,4S,5R,6S)-6-(5-((R)-2-(5,6-diethyl-2,3-dihydro-1H-inden-2-ylamino)-1-hydroxyethyl)-2-oxo-1,2-dihydroquinolin-8-yloxy)-... (2S,4R)-4-(Acetyloxy)nicotine Dioxalate (2S,4R)-4-(Cyanomethyl)nicotine Dioxalate (2S,4R)-4-(Fluoromethyl)nicotine Dioxalate (2S,4R)-4-(Methoxymethyl)nicotine Dioxalate (2S,4R)-4-Benzylnicotine Dioxalate (2S,4R)-4-Ethylnicotine Dioxalate (2S,4R)-4-Hydroxynicotine Dioxalate (2S,4R)-4-Methylnicotine Dioxalate (2S,4R)-4-[(Methylsulfonyl)oxy]nicotine Dioxalate (2S,4R)-4-[(Methylthio)methyl]nicotine Dioxalate (2S,4R,5R)-2-benzhydryl-5-benzylaminotetrahydropyran-4-ol (2S,4S)-4-(Hydroxynethyl)nicotine (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamid... (2S,5R)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(piperidin-1-ylsulfonyl)piperidine (2S,5R)-5-Butylnicotine Oxalate (2S,5R)-5-Methylnicotine Oxalate (2S,5R)-5-Phenylnicotine Oxalate (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid (2S,5S)-5-Butylnicotine Oxalate (2S,5S)-5-Methylnicotine Oxalate (2S,5S)-5-Phenylnicotine Oxalate (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid (2S,6S,2R)-2-[6-(2-(1-Naphthalene)-sulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-(2-Naphthalene)-sulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-(2-Thiophen)-carboxyl-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-(2-Thiophene)-sulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Acetyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Anisoyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Benzoyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Benzylsulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Butylsulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Butyryloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Isobutyryloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Isopropylsulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Chloro-benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Fluoro-benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Nitro-benzenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-p-Toluenesulfonyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Propionyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2S,6S,2R)-2-[6-(2-Toluyloxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone hydrochloride (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-bromo-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-chloro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin (2SR,3aRS,12bSR)-2-N,N-Dimethylaminomethyl-11-fluoro-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]tiepin (3'R)-Quinuclidin-3'-yl 1-(2-Thienyl)1,2,3,4-tetrahydroisoquinoline-2-carboxylate (3'R)-Quinuclidin-3'-yl 1-Cyclohexyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate (3'R,4RS)-Quinuclidin-3'-yl 4-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone (3,5-dichlorophenyl)-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methanone (3,5-Dinitropyridin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (3-((2-(4,6-dimorpholino-1,3,5-triazin-2-yl)hydrazono)methyl)-1H-indol-1-yl)(p-tolyl)methanone (3-Amino-1(R,S)-ethylpropyl)methylphosphinic acid (3-Amino-1(R,S)-hydroxypropyl)methylphosphinic acid (3-Amino-2(R)-hydroxypropyl)methylphosphinic acid (3-Amino-2(R,S)-hydroxypropyl)(cyclohexylmethyl)phosphinic Acid Hydrochloride (3-Amino-2(R,S)-hydroxypropyl)(diethoxymethyl)phosphinic Acid (3-Amino-2(R,S)-hydroxypropyl)(difluoromethyl)phosphinic acid (3-Amino-2(R,S)-hydroxypropyl)benzylphosphinic Acid Hydrochloride (3-Amino-2(R,S)-hydroxypropyl)n-butylphosphinic Acid Hydrochloride (3-Amino-2(S)-hydroxypropyl)(1,1-diethoxymethyl)phosphinic Acid (3-Amino-2(S)-hydroxypropyl)methylphosphinic acid (3-Aminopropyl)(1(R,S)-hydroxybenzyl)phosphinic acid (3-Aminopropyl)(1,1-difluoro-n-butyl)phosphinic acid hydrochloride (3-Aminopropyl)(2-cyclohexylethyl)phosphinic acid hydrochloride (3-Aminopropyl)(2-phenylethyl)phosphinic acid (3-Aminopropyl)(2-pyridylmethyl)phosphinic acid (3-Aminopropyl)(3-N-phthalimido-2-(R,S)-hydroxypropyl)phosphinic Acid (3-Aminopropyl)(3-oxobutyl)phosphinic Acid (3-Aminopropyl)(cyclohexylmethyl)phosphinic acid (3-Aminopropyl)(hydroxymethyl)phosphinic acid (3-Aminopropyl)benzylphosphinic acid (3-Aminopropyl)isobutylphosphinic acid (3-Aminopropyl)methylphosphinic acid (3-Aminopropyl)phenylphosphinic acid (3-Aminopropyl)tert-butylphosphinic acid (3-Aminopropyl)[(R,S)-tetrahydrofuran-2-yl]phosphinic acid (3-Aminopropyl)[(R,S)-tetrahydropyran-2-yl]phosphinic acid (3-Aminopropyl)[(tetrahydropyran-2(R,S)-yl)ethyl]phosphinic acid (3-Aminopropyl)[[(R,S)-tetrahydropyran-2-yl]methyl]phosphinic acid (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone (3-Ph-Pr6)His7,DAla11,DPro13,Psi13-14,Phe14-Bn(6-14) (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3,5-dimethyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3-ethyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3-trifluoromethyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-ethyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-hydroxyphenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-isopropyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-propyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-trifluoromethyl-phenyl)-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-m-tolyl-methanone (30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-p-tolyl-methanone (30,50-Dichloro-2,6-dimethoxy-biphenyl-4-yl)-p-tolyl-methanone (30,50-Dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-p-tolyl-methanone (3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,4S,7R,7aS)-2-(6-(4-(3-trifluoromethylphenyl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione (3aR,5R,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aR,6aS)-2-(5-fluoro-4-((R)-1-(3-fluorophenyl)ethoxy)pyrimidin-2-yl)octahydropyrrolo[3,4-c]pyrrole (3aR,6aS)-2-(5-fluoro-4-((R)-1-(4-fluorophenyl)ethoxy)pyrimidin-2-yl)octahydropyrrolo[3,4-c]pyrrole (3aR,7aS)-2-[3-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-propyl]-... (3aR,7aS)-2-[4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-butyl]-h... (3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aS,13bR)-12-methoxy-5-methylene-2,3,4,5,6,7,9,13boctahydro-1H-cyclopenta[c]pyrido[1,2-b]isoquinoline (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid (3R)-(-)-3-((Cyclopropylmethyl){[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}amino)-8-fluorochromane-5-carboxamide (3R)-(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide (3R)-(-)-8-Fluoro-3-[{[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}(propyl)amino]chromane-5-carboxamide (3R)-(-)-8-Fluoro-3-{[(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl]amino}chromane-5-carboxamide (3R)-(-)-8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)-amino}-N-methylchromane-5-carboxamide (3R)-(-)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine (3R)-1,1-Dibutyl-3-(4,5-diphenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Dibutyl-3-(4-phenyl-1,3-thiazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline Hydrochloride (3R)-1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-1,2,3,4-tetrahydro[1]benzothieno[2,3-c]pyridine (3R)-1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Diethyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Dihexyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1,1-Dipentyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(2-Nitrophenyl)-3-(4-phenyl-1H-imidazol-2-y1)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(4-Dimethylaminophenyl)-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(4-Methoxyphenyl)-3-(4-phenyl-1H-imidazol-2-y1)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-(n-Pentyl)-3-(4-Phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-Cyclohexyl-1-methyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-1-Cyclohexyl-3-(4-Phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline Fumarate (3R)-2-(N,N-Dimethylglycyl)-7-hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]-methyl}-2-methylpro... (3R)-2-Acetyl-7-hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-te... (3R)-3-((3-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-8-azabicyclo[3.2.1]octan-8-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[... (3R)-3-(4-Phenyl-1H-imidazol-2-yl)-1-(4-pyridinyl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3R)-3-(4-Phenyl-1H-imidazol-2-yl)spiro[Beta-carboline-1,2'-adamantyl] Dihydrochloride (3R)-3-(imidazol-1-ylmethyl)piperidine (3R)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide (3R)-3-{[((1S)-1-{[(3R,4R)-4-(3-Hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)amino]-methyl}-1,2,3,4-tetra... (3R)-7-Hydroxy-N-((1S)-1-{[(3S,4S)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-... (3R)-N-((1S)-1-{[(3R,4R)-4-(3-Hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquino... (3R)-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-3,4-dihydro-2H-chromen- (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dion... (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6a... (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-di... (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6... (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2... (3R,4S)-3-(benzofuran-2-ylmethyl)-4-(4-methoxyphenyl)-1-phenylazetidin-2-one (3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin-3-yl)propyl)azetidin-2-one (3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-N-isobutylpiperidine-3-carboxamide (3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-N-isobutylpiperidine-3-sulfonamide (3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-N-isopentylpiperidine-3-sulfonamide (3R,6S)-1-(4-chlorophenyl)-N-cyclobutyl-6-(2,4-dichlorophenyl)piperidine-3-carboxamide (3R,6S)-1-(4-chlorophenyl)-N-cyclohexyl-6-(2,4-dichlorophenyl)piperidine-3-carboxamide (3R,6S)-1-(4-chlorophenyl)-N-cyclohexyl-6-(2,4-dichlorophenyl)piperidine-3-sulfonamide (3R,6S)-N-(4-chlorobenzyl)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidine-3-carboxamide (3S)-(+)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine (3S)-1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline (3S)-1-(2-methoxyethyl)-N-[(5-methylimidazo[1,2-a]pyridin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide (3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (3S)-3-(((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (3S)-3-((2-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)ethylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (3S)-3-((2-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)ethylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one... (3S)-3-((3-( 6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propylamino)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-o... (3S)-3-({[2-({4-[amino(imino)methyl]benzyl}oxy)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}carbonyl}amino)-3-phenylpro... (3S)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide (3S)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-... (3S)-7-Hydroxy-N-((1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-2-methyl-1,2,3,4-te... (3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-one (3S,4S)-5-(4-Bromobenzyloxy)-3-hydroxy-4-(2-thiophen-2-ylacetylamino)pentanoic Acid [(S)-1-((S)-1-Carbamoyl-3-methylbutylcarb... (3S,4S)-5-(4-Bromobenzyloxy)-4-(3,3-diphenylpropionylamino)-3-hydroxypentanoic Acid [(S)-1-((S)-1-Carbamoyl-3-methylbutylcarb... (3S,4S)-5-(4-Bromobenzyloxy)-4-diphenylacetylamino-3-hydroxypentanoic Acid [(S)-1-((S)-1-Carbamoyl-3-methylbutylcarbamoyl)eth... (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6a... (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine... (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',... (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione (4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxybenzofuran-2-yl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methan... (4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione (4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione (4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol (4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)(1-methyl-1H-pyrrol-2-yl)meth... (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine (4-(4-(5-chloropyridin-2-yl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl) butan-1-one oxime (4-(Benzylamino)piperidin-1-yl)-(naphthalen-2-yl)methadone (4-(furan-2-yl)-2-(2-(thiophen-2-yl)ethylamino)thiazol-5-yl)(phenyl)methanone (4-(Methylsulfonyl)phenyl)(4-phenyl-2-(phenylamino)-thiazol-5-yl)methanone (4-amino)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Asp-NH2 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Thr-NH2 (4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 (4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 (4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 (4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 (4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2 (4-benzhydrylpiperazin-1-yl)(cyclohexyl)methanone (4-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (4-Butyl-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone (4-Butyl-phenyl)-(30,50-dichloro-2,6-dimethoxy-biphenyl-4-yl)-methanone (4-Butyl-phenyl)-(30,50-dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-methanone (4-Chloro-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone (4-Chloro-phenyl)-(30,50-dichloro-2,6-dimethoxy-biphenyl-4-yl)-methanone (4-Chloro-phenyl)-(30,50-dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-methanone (4-Chlorophenyl)(2-(methylamino)-4-phenylthiazol-5-yl)methanone (4-Ethyl-piperazin-1-yl)-(1H-indol-2-yl)-methanone (4-Ethynyl-cyclohex-3-enyl)-dipropyl-amine (4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol (4-Methoxyphenyl)(2-(methylamino)-4-phenylthiazol-5-yl)methanone (4-Methoxyphenyl)(4-phenyl-2-(phenylamino)thiazol-5-yl)methanone (4-Nitrobenzyl)-6-thioguanosine (4-Phenyl-2-(phenylamino)thiazol-5-yl)(p-toluyl)methanone (4-tert-Butyl-2-aminothiophen-3-yl)(4-chlorophenyl)methanone (4-tert-Butyl-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy]phenyl)imidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2,3-dichlorophenyl)piperazin-1-yl]propoxy]phenyl)imidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]butoxy]phenyl)imidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-6-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-7-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-8-methylimidazo[1,2-a]pyridine (4-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]phenyl)-imidazo[1,2-a]pyridine (4-{2-[4-(2,2-Dimethyl-[1,3]dioxan-5-ylmethoxy)phenyl]vinyl}phenyl)dimethylamine (4-{4-[(Benzyl{2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic Acid (4aR,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol (4aR,8S,8aR)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (4aR,8S,8aR)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (4aS,14bR)-13-methoxy-6-methylene-1,2,3,4,5,6,7,8,10,14bdecahydropyrido[2,1-e]phenanthridine (4aS,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,5R)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-D-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,5S)-2-Benzyl-5-[N-[tert-butoxycarbonyl)-L-tryptophyl]amino]-1,3-dioxoperhydropyrido[1,2-c]pyrimidine (4aS,8R,8aS)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (4aS,8R,8aS)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol (4bS,7R,8aR)-4b-benzyl-7-hydroxy-7-(prop-1-ynyl)-N-(pyridin-4-ylmethyl)-4b,5,6,7,8,8a,9,10-octahydrophenanthrene-2-carboxamid... (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzof... (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzo... (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-meth... (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methano... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-me... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanob... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanob... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-met... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methan... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenz... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-metha... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methan... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanob... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-met... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenz... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenz... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-metha... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-met... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-me... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzo... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenz... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofu... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofu... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-me... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzo... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenz... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzo... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofu... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofu... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofu... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofu... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzo... (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzo... (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3... (4R)-3,4-Dihydrosalvinorin C (4R)-3,4-Dihydrosalvinorin E (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid (4R,7S,10S,13R,16S,19R)-13-((1H-indol-3-yl)methyl)-N-((2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl)-10-(3-guanidinopropyl)-16-(4... (5,7- Dichloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5,7-Difluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5,7-Dimethyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol (5-(4-(((2,4-Difluorobenzyl)(2-methyl-3-((methylsulfonyl)amino)phenyl)amino)methyl)phenoxy)-2-fluorophenoxy)acetic Acid (5-(4-(4-cyclopropylpiperazin-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-cyclopropylpiperazin-1-yl)butyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-fluoropiperidin-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-isopropyl-1,4-diazepan-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-isopropylpiperazin-1-yl)but-1-ynyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-(4-(4-isopropylpiperazin-1-yl)butyl)-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-bromo-2-(4-(methylthio)phenoxy)phenyl)-N-methylmethanamine (5-Bromopyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (5-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine (5-Fluoro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Hydroxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Methoxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate (5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate (5aR,6S)-1-(4-Fluorophenyl)-6-((S)-1-methoxy-1-(thiophen-2-yl)-ethyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinol... (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione (5E)-5-((1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one (5E)-5-((4-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one (5E)-5-((5-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one (5E)-5-((6-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one (5E)-5-((7-bromo-1H-indol-3-yl)methylene)-1,3-dimethyl-2-(methylimino)imidazolidin-4-one (5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid (5R,2'R)-5-(1-methyl-2-pyrrolidinyl)oxazolidinone (5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid (5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5R,2'S)-5[1'-methylpyrrolidin-2'-yl]-1,3-oxazolidin-2-one (5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5S,2'S)-5-(1-methyl-2-pyrrolidinyl)oxazolidinone (5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16-triol (6-(4-((phenethylamino)methyl)phenoxy)pyridin-3-yl)(piperidin-1-yl)methanone (6-(methylsulfonyl)-1-pentyl-1H-indol-3-yl)(naphthalen-2-yl)methanone (6-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (6-bromo-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone (6-chloro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone (6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine (6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone (6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (6-fluoro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-ylmethanone (6-fluoro-2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone (6-methyl-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone (6aR,12bS)-6a,7,8,12b-Tetrahydro-6H-chromeno[3,4-c]isoquinoline-2,3-diol (6aS,12bR)-6a,7,8,12b-Tetrahydro-6H-chromeno[3,4-c]isoquinoline-2,3-diol (6bR,10aS)-1-(4-Fluorophenyl)-4-(1,1,3-trimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin... (6bR,10aS)-1-(4-fluorophenyl)-4-(1,3-dimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin-8(... (6bR,10aS)-1-(4-fluorophenyl)-4-(1,3-dimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin-8(... (6bR,10aS)-8-[3-(1,2-Benzisoxazol-3yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quin... (6bR,10aS)-8-[3-(4-Fluoro-phenyl)-4,5-dihydro-isoxazol-5-ylmethyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]p... (6bR,10aS)-8-[3-(4-Fluorophenoxy)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahy-dro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,... (6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,... (6bR,10aS)-8-[3-(6-Fluoro-1H-indazol-3-yl)-propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de... (6bR,11aR)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophen... (6bS, 11aS)-4-(1,2,6b,7,8,10,11,11a-Octahydro-9H-azepino[4,5-b][1,4]oxazino[2,3,4-hi]indol-9-yl)-1-(4-fluorophenyl)-1-butanon... (6bS,11aS)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophen... (6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one (6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride (6R,7S)-1-benzyl-4-methylene-7-phenyl-1,9-diazaspiro[5.5] undecane (6S,10bR)-6-(4-methoxyphenyl)-9-(3-(piperidin-1-yl)propoxy)-1,2,3,5,6,10b-hexahydropyrrolo[2,1-a]isoquinoline (6S,7R)-7-(1H-Indol-3-yl)-4-methylene-1-azaspiro[5.5] undecane (6S,7S)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride (7-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone (7-{4-[4-(3-chloro-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride) (8R,9S,13S,14S,17S)-17-(2-(2-(2-hydroxyphenyl)-1H-indol-3-yl)ethynyl)-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclo... (8R,9S,13S,14S,17S)-17-(2-(2-(2-methoxyphenyl)-1H-indol-3-yl)ethynyl)-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclo... (8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one (8S,9R,10S)-15,16-epoxy-9α-hydroxylabda-5,13(16),14-trien-7-one (9,13-epoxy-15,16-dihydroxylabd-5-en-7-one (9,13-epoxy-6-hydroxylabdan-15,16-olide (9,13-epoxylabd-5-ene-7 b,15,16-triol (9,13:15,16-diepoxylabdane-6b,16b-diol (9-pentyl-9H-carbazol-3-yl)(piperazin-1-yl)methanone (9S,10R,11S,13S,14S,17R)-11,17-dihydroxy-17-(2-hydroxyacetyl)-10,13-dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-1H-c... (anthracen-9-ylmethyl)-3,3-triamine (anthracen-9-ylmethyl)-4,4-triamine (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate (±)-((4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-proline (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-valine (±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine (±)-(3aR,3a1R,6aR,9aS)-1-propyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aR,3a1R,6aS,12bS,12cS)-12b-ethyl-4-propyl-1,2,3,3a,3a1,4,5,6,6a,7,12b,12c-dodecahydroquinolino[4,5-bc]carbazole (±)-(3aR,3a1S,6aS,7R,13bR)-11-chloro-7-ethyl-3-propyl-2,3,3a,3a1,4,5,6,6a,7,13b-decahydro-1H-dibenzo[de,j][3,7]phenanthrol... (±)-(3aR,3a1S,6aS,7R,13bR)-7-ethyl-3-methyl-2,3,3a,3a1,4,5,6,6a,7,13b-decahydro-1H-dibenzo[de,j][3,7]phenanthroline (±)-(3aR,3a1S,6aS,7R,13bR)-7-ethyl-3-propyl-10-(trifluoromethyl)-2,3,3a,3a1,4,5,6,6a,7,13b-decahydro-1H-dibenzo[de,j][3,7]... (±)-(3aR,3a1S,6aS,7R,13bR)-7-ethyl-3-propyl-2,3,3a,3a1,4,5,6,6a,7,13b-decahydro-1H-dibenzo[de,j][3,7]phenanthroline (±)-(3aR,3a1S,6aS,7R,13bR)-7-ethyl-9-methoxy-3-propyl-2,3,3a,3a1,4,5,6,6a,7,13b-decahydro-1H-dibenzo[de,j][3,7]phenanthrol... (±)-(3aS,3a1R,5R,6R,6aS,9aR)-6-ethyl-1-propyldodecahydro-1H-benzo[de]quinolin-5-ol (±)-(3aS,3a1R,6R,6aS,9aR)-1-(cyclohexylmethyl)-6-(4-methoxybenzyl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-1-(cyclohexylmethyl)-6-ethyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-1-isopentyl-6-(4-methoxybenzyl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-(4-methoxybenzyl)-1-methyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-(4-methoxybenzyl)-1-propyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-(2-methoxyethyl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-(cyclohexylmethyl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-(thiazol-2-yl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-(thiophen-2-yl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-isopentyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-methyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-benzyl-1-propyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-(2-methoxyethyl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-(thiazol-2-yl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-(thiophen-2-yl)decahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-heptyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-isopentyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-methyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-propyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-6-ethyl-1-tosyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,3a1R,6R,6aS,9aR)-N-(4-chlorobenzyl)-6-ethyl-5-oxododecahydro-1H-benzo[de]quinoline-1-carboxamide (±)-(3aS,3a1S,6aR,9aR)-1-propyldecahydro-1H-benzo[de]quinolin-5(3a1H)-one (±)-(3aS,4R,7aS)-2-benzyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-benzyl-3-oxo-N-phenyl-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-benzyl-N-(3-chlorophenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-cyclohexyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-cyclohexyl-3-oxo-N-phenyl-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-2-cyclohexyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxami... (±)-(3aS,4R,7aS)-N,2-dicyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-N-(3-chlorophenyl)-2-cyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(3aS,4R,7aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxam... (±)-(3aS,4R,7aS)-N-cyclohexyl-2-benzyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-N-(2,4-dichlorophenyl)-1,2,3,4,4a,7,8,8a-octahydroiso... (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-(3,4-dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-benzyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-butyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclohexyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-2-cyclopropyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-N,2-dibutyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-N,2-dicyclohexyl-1-oxo- 1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-N-(2,4-dichlorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-N-(2,6-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoli... (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinol... (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aR,8S,8aR)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carb... (±)-(4aR,8S,8aR)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aR,8S,8aR)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-(4aS,8R,8aS)-2-benzyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N,2-bis(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N-(cyclopropylmethyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-(4-(trifluoromethyl)benzyl)-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline... (±)-(4aS,8R,8aS)-1-oxo-2-(4-(trifluoromethyl)benzyl)-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline... (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-... (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-N-(thiazol-2-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-2-((3-fluoro-4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline... (±)-(4aS,8R,8aS)-2-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxa... (±)-(4aS,8R,8aS)-2-(2-fluoro-6-methoxybenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoq... (±)-(4aS,8R,8aS)-2-(2-fluorobenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8... (±)-(4aS,8R,8aS)-2-(2-methoxybenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-... (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-(3,4dimethoxybenzyl)-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-c... (±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-... (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxam... (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxam... (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(2,6-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(3-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(4-chlorobenzyl)-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-bemzyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-((3-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoli... (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4a... (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3-(thiophen-2-yl)benzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-benzyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-benzyl-N,N-dicyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-((3-chloro-4-fluoro-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-... (±)-(4aS,8R,8aS)-2-benzyl-N-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxa... (±)-(4aS,8R,8aS)-2-benzyl-N-(2,3,4,5,6-pentafluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(2,3-difluoro-4-methylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(2-carbamoylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(3-bromobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(3-chloro-4-methylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)benzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-3,3-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-methylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluoro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aS,8R,8aS)-2-benzyl-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-([1,1-biphenyl]-2-yl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-benzyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-butyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aS,8R,8aS)-2-butyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-butyl-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)... (±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-cyclohexyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-cyclohexyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aS,8R,8aS)-2-cyclohexyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-2-cyclohexyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid (±)-(4aS,8R,8aS)-2-cyclopropyl-1-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-cyclopropyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-2-cyclopropyl-N-(2,4-dichlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-N-(4-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-cyclopropyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-isopropyl-1-oxo-N-(3-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-isopropyl-1-oxo-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-2-isopropyl-N-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydro-1H-isochromen-1-one (±)-(4aS,8R,8aS)-8-(pyrrolidine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-8-amino-2-benzyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-8-amino-2-cyclohexyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one (±)-(4aS,8R,8aS)-N,2-dibenzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N,2-dibutyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N,2-dicyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N,N-dicyclohexyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N,N-dimethyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-((4-acetamido-[1,1-biphenyl]-3-yl)methyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carb... (±)-(4aS,8R,8aS)-N-((4-acetyl-[1,1-biphenyl]-3-yl)methyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxa... (±)-(4aS,8R,8aS)-N-(2,3-difluoro-4-methylphenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin... (±)-(4aS,8R,8aS)-N-(2,4,6-trimethylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(2,4-dichlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2,4-dichlorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2,4-dichlorophenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aS,8R,8aS)-N-(2,4-dichlorophenyl)-2-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2,6-difluorophenyl)-1-oxo-2-(4-(trifluoromethyl)benzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carb... (±)-(4aS,8R,8aS)-N-(2,6-difluorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2,6-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2,6-difluorophenyl)-2-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(2-chloro-4-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(2-chloro-4-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-N-(2-chloro-4-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aS,8R,8aS)-N-(2-chloro-5-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide ... (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-(4-(trifluoromethyl)benzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carb... (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-2-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-(5-acetylthiophen-2-yl)benzyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and ... (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxa... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoqu... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-fluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline... (±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(4-chloro-2-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(4-chloro-2-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-N-(4-chloro-2-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)benzyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)benzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)benzyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-o... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoq... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoli... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinol... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carb... (±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbox... (±)-(4aS,8R,8aS)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chloro-3-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chloro-3-methylphenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamid (±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-methoxyphenyl)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-3-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-4-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... (±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(4-nitrophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(6-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... (±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-([1,1-biphenyl]-2-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-allyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-allyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-allyl-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-allyl-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-benzyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-benzyl-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclohexylmethyl)-N-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-2-cyclopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-cyclohexyl-N-isopropyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-methoxy-N-methyl-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-methyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-methyl-1-oxo-N,2-diphenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide (±)-(4aS,8R,8aS)-N-methyl-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide (±)-(4aS,8R,8aS)-N-phenyl-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoli... (±)-(4aS,8S,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... (±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine (±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-phenyl-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-2-benzyl-N-(3-chlorophenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-car... (±)-(5aS,9R,9aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-ca... (±)-(5aS,9R,9aS)-2-benzyl-N-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-2-benzyl-N-phenyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-N,2-dicyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-N-(3-chlorlophenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide (±)-(5aS,9R,9aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9... (±)-(5aS,9R,9aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-... (±)-(5S)-8-(4-Methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine (±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine (±)-2,4,5-Trimethoxamphetamine (±)-2,5-Dimethoxy-4-bromoamphetamine (±)-2,5-Dimethoxy-4-ethoxyamphetamine (±)-2,5-Dimethoxy-4-ethylamphetamine (±)-2,5-Dimethoxy-4-iodoamphetamine (±)-2,5-Dimethoxy-4-methylamphetamine (±)-2-((3,5-Dichlorophenyl)sulfonyl)-7-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine (±)-2-((3,5-Dichlorophenyl)sulfonyl)-8-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine (±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine (±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine (±)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-7-yl)morpholine38a (±)-2-Benzyl-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine (±)-2-Benzyl-8-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine (±)-3,4,5-Trimethoxamphetamine (±)-3,4-Methylenedioxyamphetamine (±)-3,4-Methylenedioxymethamphetamine (±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-3-chloro-4-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-3-chloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-4-bromo-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-4-bromo-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-4-chloro-2-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-4-chloro-3-(trifluoromethyl)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-4-chloro-3-methyl-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-4-chloro-N-(((4aS,8R,8aS)-2-benzyl-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)methyl)-3-(trifluoromethyl)aniline (±)-4-Ethylthio-2,5-dimethoxyamphetamine (±)-7-Chloro-1-hydroxymethyl-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (±)-7-Chloro-1-methoxymethyl-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (±)-7-Chloro-9-[4-[2-(imidazolidin-2-on-1-yl)ethyl]piperazin-1-yl]-9,10-dihydro pyrrolo[2,1-b][1,3]benzothiazepine (±)-alpha-Methylbenzeneethanamine (±)-Benzyl(5S)-8-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2- carboxylate (±)-Benzyl-7-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-(3-ethoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate (±)-Benzyl-7-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate (±)-Benzyl-7-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-7-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate (±)-Benzyl-7-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate (±)-Benzyl-8-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate (±)-Benzyl-8-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate (±)-Benzyl-8-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate (±)-Benzyl-8-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate (±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine (±)-cis-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine (±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine (±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine (±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine (±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine (±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine (±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine (±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine (±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine (±)-N-(((4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)methyl)aniline (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3,5-dichlorobenzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3-chloro-4-methylbenzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3-chlorobenzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-bromo-3-(trifluoromethyl)benzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-bromobenzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-2-methylbenzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-(trifluoromethyl)benzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-methylbenzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide (±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide (±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide (±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide (±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide (±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine (±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine (±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine (±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine (±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine (±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine (±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine (±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine (±)-trans-(6-Phenyl-1,4-dioxan-2-yl)methanamine (±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine (±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine (±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine (±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate (C33H41N3O5Cl2·0.7F3CCO2H) C, H, N (C34H40N3O6Cl) C, H, N (C34H42N3O5Cl·2F3CCO2H) C, H, N (C34H46Cl2N6O8•1.5H2O), C, H, N (C34H46Cl2N6O8•3H2O), C, H, N (C34H46Cl2N6O8•H2O), C, H, N (C35H40N3O7Cl) C, H, N (C35H41N4O6Cl·1.3H2O) C, H, N (C35H48Cl2N6O8), C, H, N (C35H48Cl2N6O8•2.5H2O), C, H, N (C35H48Cl2N6O8•H2O), C, H, N (C37H52Cl2N6O8), C, H, N (C37H52Cl2N6O8•1.5H2O), C, H, N (C37H52Cl2N6O8•2.5H2O), C, H, N (C38H36N3O8Cl) C, H, N (C38H54Cl2N6O10•H2O), C, H, N (C40H41N3O8·0.5H2O) C, H, N (C41H49N3O7·0.9F3CCO2H) C, H, N (C42H51N3O7) C, H, N (C42H62Cl2N6O8•0.5H2O), C, H, N (C42H62Cl2N6O8•1.5H2O), C, H, N (C43H49N3O9·0.8H2O) C, H, N (C46H45N3O10) C, H, N (D-Ala(2),MePhe(4),Gly-ol(5))enkephalin (D-Ala2)-MEGY (D-Ala2, Val5)-MEGY (D-T6-D-W8,9)galol (E)-(2-Amino-5-(2-(4-chlorophenyl)ethen-1-yl)-4-(2,2- dimethylpropyl)thiophen-3-yl)(4-chlorophenyl)methanone (E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-propenone (E)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one (E)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one (E)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one (E)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-4(5H)-one (E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide (E)-3-(3-cyanophenyl)-N-methyl-N-[(4-oxo-3H-quinazolin-2-yl)methyl]prop-2-enamide (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide (E)-3-Aminopropen-2-yl)methylphosphinic acid (E)-3-[2-(2-Methyl-4-thiazolyl)vinyl]pyridine (E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide (E)-4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)prop-1-en-1-yl)-2-methoxyphenol (E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide (E)-4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)but-2-en-1-yl)- morpholine (E)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol (E)-5-((1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one (E)-5-((1H-indol-3-yl)methylene)-2-amino-1-methyl-1H-imidazol-4(5H)-one (E)-5-((1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one (E)-5-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one (E)-5-((4-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one (E)-5-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one (E)-5-((5-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one (E)-5-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one (E)-5-((6-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one (E)-5-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-4(5H)-one (E)-5-((7-bromo-1H-indol-3-yl)methylene)-2-imino-1,3-dimethylimidazolidin-4-one (E)-9-(2-(cinnamyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione (E)-CH2OCOC(CH3)3 (E)-N-((3R,3aR,3a1S,9aR)-9-(N-(cyclopropylmethyl)phenylsulfonamido)-5-methoxy-1,2,3,3a,3a1,8,9,9a-octahydrophenanthro[4,5-bcd... (E)-N-((3R,3aR,3a1S,9aS)-9-(N-(cyclopropylmethyl)phenylsulfonamido)-9a-hydroxy-5-methoxy-1,2,3,3a,3a1,8,9,9a-octahydrophenant... (E)-N-((3R,4aR,10R,10aS)-10-(N-(cyclopropylmethyl)phenylsulfonamido)-10a-hydroxy-6-methoxy-1,2,3,4,4a,9,10,10a-octahydrophena... (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide (E)-N-(Adamant-1-yl)-6-[2-(4-methoxyphenyl)vinyl]-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinol... (E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-1... (E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinol... (E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-1... (E/Z)-11-(2-butenyloxy)-N-propylnoraporphine (N-acetyl 2-benzyltryptamine) (R)(+)-BrAPB (R)-(+)-2-(1-Methyl-2-phenylethyl)-4,5-dihydro-1H-imidazole Oxalate (R)-(+)-3-Fluoromethyl-7-(N-2,2,2-trifluoroethylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-3,3,3-trifluoropropylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-3-methoxypropylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-ethylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-propylaminosulfonyl)-THIQ (R)-(+)-3-Fluoromethyl-7-(N-thiomorpholinoaminosulfonyl)-THIQ (R)-(+)-AM2233 (R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride (R)-(-)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid (R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine (R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine (R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine (R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine (R)-(-)-7-chloro-9-(4-methylpiperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine (R)-(-)-9,10-Dihydro-7-fluoro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine (R)-(-)-N-butyl-2-methoxy-11-hydroxynoraporphine (R)-(-)-N-ethyl-2-methoxy-11-hydroxynoraporphine (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine (R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine (R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine (R)-(--)-2-(2-Phenylpropyl)-4,5-dihydro-1H-imidazole Maleate (R)-(1-benzyl-4-(4-methoxybenzyl)piperazin-2-yl)methanol (R)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; iodide (R)-1,3-Dimethyl-8-(2,1,3,4-tetrahydronaphthalen-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione (R)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(tetrahydro-2H-pyran-4-y... (R)-1-(10,11-dihydro-dibenzo[b,f]azepin-5-yl)-3-methylamino-propan-2-ol (R)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol (R)-1-(2-(1-(3,4-Dichloro-benzene sulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine (R)-1-(2-(1-(3-bromo-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl)-4-methyl piperidine (R)-1-(2-(1-(3-methoxy-benzenesulfonyl)-pyrrolidin-2-yl)-ethyl-4-methyl piperidine (R)-1-(2-(2-ethoxyphenyl)-1-phenylethyl)piperazine (R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine (R)-1-(4-Fluorophenyl)-2-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)propan-2... (R)-1-(5-fluoro-4-(1-(3-fluorophenyl)ethoxy)pyrimidin-2-yl)-1,4-diazepane (R)-1-(5-fluoro-4-(1-(4-fluorophenyl)ethoxy)pyrimidin-2-yl)-1,4-diazepane (R)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol (R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine (R)-1-(Indolin-1-yl)-2-(2-(((4-methylpyridin-2-yl)oxy)methyl)morpholino)ethanone (R)-1-(Indolin-1-yl)-2-(2-((pyridin-2-yloxy)methyl)morpholino)ethanone (R)-1-(Indolin-1-yl)-2-(2-((pyridin-3-yloxy)methyl)morpholino)ethanone (R)-1-Cyclohexyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol (R)-1-Cyclopropyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol (R)-10-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-10-Methyl-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-11-(2-methylallyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-11-(3-methylbut-2-enyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-11-(allyloxy)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-11-Amino-2-methoxyaporphine (R)-11-Ethyl-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (R)-2,11-Diaminoaporphine (R)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine (R)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine (R)-2-((1-methylpyrrolidin-2-yl)methyl)-1H-pyrrolo[2,3-b]pyridine (R)-2-((3-Chlorophenoxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-4-methylpentan-2-ol (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-4-phenylbutan-2-ol (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)hexan-2-ol (R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)pent-4-en-2-ol (R)-2-((R)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine (R)-2-((R)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine (R)-2-((R)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine (R)-2-((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)-1-methylpyrrolidine hydrochloride (R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid (R)-2-(2-((3-chlorophenoxy)methyl)morpholino)-1-(indolin-1-yl)ethanone (R)-2-(2-phenyl-2-(piperazin-1-yl)ethyl)phenol (R)-2-(4-hydroxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-2-(4-Hydroxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol (R)-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid (R)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid (R)-2-Me-Tet-AMPA (R)-2-Methoxyaporphin-11-yl pentanoate (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydro... (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroi... (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran... (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-... (R)-3-((1-Methylpyrrolidin-2-yl)methoxy)-5-(phenoxymethyl)isoxazole Hydrochloride (R)-3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate (R)-3-((4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)piperidin-1-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)... (R)-3-((4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)methyl)-7,9-dihydro-2H-[1,4]dioxino[2,3-e]indol-8(3H)-one (R)-3-(1H-indol-4-yl)-N-methyl-3-(thiophen-2-yl)propan-1-amine hydrochloride (R)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride (R)-3-(3,4-dichlorophenyl)-N-methyl-3-(naphthalen-1-yl)propan-1-amine hydrochloride (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole (R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (R)-3-Carboxy-4-hydroxyphenylglycine (R)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (R)-3-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (R)-3-Hydroxyphenylglycine (R)-3alpha-(Methylphenyl)-2alpha-phenyltropane (R)-3beta-(Methylphenyl)-2beta-phenyltropane (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl) (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline (R)-4-(1H-indol-4-yl)-N-methyl-4-(thiophen-2-yl)butan-1-amine hydrochloride (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((4-methylpyridin-2-yl)oxy)methyl)morpholine (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine (R)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine (R)-4-(2-(Indolin-1-yl)ethyl)-2-((pyridin-2-yloxy)methyl)morpholine (R)-4-(2-(Indolin-1-yl)ethyl)-2-((pyridin-3-yloxy)methyl)morpholine (R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide (R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide (R)-4-(3,4-dichlorophenyl)-4-(1H-indol-4-yl)-N-methylbutan-1-amine hydrochloride (R)-4-(3,4-dichlorophenyl)-N-methyl-4-(naphthalen-1-yl)butan-1-amine hydrochloride (R)-4-(3-(2-amino-4-(4-fluorophenyl)thiazol-5-yl)pyrrolidin-1-yl)-1-(4-fluorophenyl)butan-1-one (R)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline (R)-4-(4-Methylpentanoyl)-8-(4-methylpentylidene)-1-thia-4-azaspiro[4.5]decane-3-carboxylic Acid (R)-4-(5-Fluoro-4-(3-fluorophenoxy)pyrimidin-2-yl)-3-methylpiperazin-1-ium·hydrochloride (R)-4-(5-Fluoro-4-(4-fluorophenoxy)pyrimidin-2-yl)-3-methylpiperazin-1-ium·hydrochloride (R)-4-Carboxyphenylglycine (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(10) (R)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) (R)-4-Methyl-1-(2-(1-toluene-3-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine (Oxalate salt) (R)-4-Methylhomoibotenic acid (R)-4-Oxo-1-pentyl-N-(1-phenylethyl)-7-(pyrrolidin-1-yl)-1,4-dihydroquinoline-3-carboxamide (R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide (R)-5,6,6a,7-Tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) (R)-5-(2-Azetidnylmethoxy)-2-Chloropyridine (R)-5-(Phenoxymethyl)-3-(pyrrolidin-2-ylmethoxy)isoxazoleHydrochloride (R)-5-2-Azetidnylmethoxy)-2-Chloropyridine (R)-5-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (R)-5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (R)-5a,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene (R)-6,10-Dimethyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-6-(1-methyl-pyrrolidin-2-yl)-quinoline (R)-6-bromo-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-6-chloro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-6-Chloro-3-(1-phenylethyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide (R)-6-fluoro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole (R)-6-Methyl-2-phenyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol (R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] (R)-7-Ethoxy-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide (R)-7-Fluoro-4-oxo-1-pentyl-N-(1-phenylethyl)-1,4-dihydroquinoline-3-carboxamide (R)-7-Methyl-1,6,6a,7,8,9-hexahydro-1,7-diaza-benzo[cd]pyren-2-one (R)-7-Methyl-6a,7,8,9-tetrahydro-2H,6H-2,7-diaza-benzo[cd]pyren-1-one (R)-7-Methyl-6a,7,8,9-tetrahydro-6H-1-oxa-7-aza-benzo[cd]pyren-2-one (R)-7-Methyl-6a,7,8,9-tetrahydro-6H-2-oxa-7-aza-benzo[cd]pyren-1-one (R)-7-[8-(2-Oxo-1,2,3,4-tetrahydro-quinolin-7-ylmethyl)-3-aza-bicyclo[3.2.1]oct-3-ylmethyl]-7,8-dihydro-3H-1,6,9-trioxa-3-aza... (R)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7, 8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione (R)-8-(3-Methylbutylidene)-4-(5-methylhexanoyl)-1-thia-4-azaspiro[4.5]decane-3-carboxylic Acid (R)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide (R)-8-OH-DPAT (R)-ABT-089 [2-Methyl-3-(2-(S)-pyrrolidinylmethoxy)pyridine] (R)-ACPA (R)-AMPA (R)-AP5 (R)-aspartic acid (R)-ATPA (R)-BrHlbo (R)-Bu-HIBO (R)-Chlopheniramine (R)-chlorpheniramine (R)-CPPene (R)-Demethyl-ACPA (R)-Epinephrine (R)-Hexbutinol (R)-HIBO (R)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-benzo[d]imidazol-2-amine (R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(1H-indol-3-yl)-2-oxoacetamide (R)-N-(2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide (R)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide (R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide (R)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea (R)-N-methyl-3-(naphthalen-1-yl)-3-(thiophen-2-yl)propan-1-amine hydrochloride (R)-N-methyl-4-(naphthalen-1-yl)-4-(thiophen-2-yl)butan-1-amine hydrochloride (R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide (R)-N3-(1-(1-Naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (R)-N3-(1-(2-Naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (R)-N3-(1-Phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide (R)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexa-hydropyrazino[1,2-a]quinolin-3-yl)butyl]amide (R)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (R)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}am... (R)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide (R)-SIB-1508Y (R)-Trihexyphenidyl (R)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone (R,S)-4-Carboxy-3-hydroxyphenylglycine (R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione (R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione (R,S)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione (R,S)-alpha-Methyl-4-carboxyphenylglycine (R/S)-2-(1H-indol-3-yl)-N-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-2-oxoacetamide (R/S)-2-(5-nitro-1H-indol-3-yl)-N-(5-nitro-2,3-dihydro-1H-inden-1-yl)-2-oxoacetamide (R/S)-N-(5-fluoro-2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide (R/S)-N-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide (Rac)-4-(Dimethylamino)-N-(4-(3-(3-hydroxyphenyl)pyrrolidin-1-yl)butyl)-benzamide (RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine (RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine (RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine (RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine (RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine (RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine (RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine (RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine (RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine (RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine (RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate (RS) PPG (RS)-2-Amino-3-(3-hydroxy-4-pentyl-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-(3-hydroxy-4-phenylethyl-5-isoxazolyl)-propionic Acid (RS)-2-amino-3-(3-hydroxy-5-isoxazolyl)propionic acid (RS)-2-Amino-3-(4-heptyl-3-hydroxy-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid (RS)-2-Amino-3-[3-hydroxy-4-(2-phenolyl)-5-isoxazolyl]-propionic Acid (RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate (RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate (RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate (RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate (RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate (RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid (RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate (RS)-2-amino-5-(3-hydoxy-5-methylisoxazol-4-yl)pentanoic acid (RS)-2-amino-5-(3-hydroxy-5-methylisoxazol-4-yl)pentanoic acid (RS)-3-sec-Butyl-2-chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]-pyridin-6(7H)-one (RS)-3-sec-Butyl-2-chloro-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one (RS)-3-sec-Butyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one (RS)-3-sec-Butyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one (RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine (RS)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) (RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride (RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine (RS)-HIBO (RS)-N3-(1-(1,2,3,4-Tetrahydronaphthyl))-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (RS)-N3-(1-(1-Naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (RS)-N3-(1-(2-Naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (RS)-N3-(1-Phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine (S)- (-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tet... (S)- (-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(4-propyl-4H-1,2,4-tri azol-3-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetr... (S)-(+)-2-(2-Phenylpropyl)-4,5-dihydro-1H-imidazole Maleate (S)-(+)-2-Amino-3-(4-hexyl-3-hydroxy-5-isoxazolyl)propionic Acid (S)-(+)-Amphetamine (S)-(+)-Br-HIBO (S)-(+)-Bu-HIBO (S)-(+)-ketamine (S)-(-)-10-{4-[2-(Butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4,5,6-hexa... (S)-(-)-10-{4-[2-(Butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4,5,6-hexahy... (S)-(-)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride (S)-(-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydr... (S)-(-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-1,2,3,4-tetrahydro-... (S)-(-)-8-{4-[2-(Butoxy)ethoxy]phenyl}-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl... (S)-(-)-9-{4-[2-(Butoxy)ethoxy]phenyl}-1-isobutyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-2,3,4,5-tetrahydr... (S)-(-)-9-{4-[2-(Butoxy)ethoxy]phenyl}-1-propyl-N-(4-{[(1-propyl-1H-imidazol-5-yl)methyl]sulfinyl}phenyl)-2,3,4,5-tetrahydro-... (S)-(-)-AM2233 (S)-(--)-2-(1-Methyl-2-phenylethyl)-4,5-dihydro-1H-imidazole Oxalate (S)-(2)-Me-Tet-AMPA (S)-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(2-methoxypyrrolidin-1-yl)methanone (S)-(3-(Pyrrolidin-2-ylmethoxy)isoxazol-5-yl)methyl Phenyl-carbamate Trifluoroacetate (S)-1,1,1-Trifluoro-2-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)propan-2-ol (S)-1,1-Dimethyl-2-quinolin-6-yl-pyrrolidinium; iodide (S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxop... (S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopro-pan... (S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-... (S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)-2-oxoethoxy)-ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-amini... (S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethoxy)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trif... (S)-1-((3-((3,4-Dihydroisoquinolin-2(1H)-yl)methyl)benzyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifl... (S)-1-((5-(3,4-Dihydroisoquinolin-2(1H)-yl)pentyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacet... (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[,5-b]isoquinolin-6-yl)-1-(thiazol-2-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(3-methylthiophen-2-yl)-... (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(5-methylthiophen-2-yl)-... (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-2-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-3-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-4-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-2-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-3-yl)ethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-m-tolylethanol (S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-o-tolylethanol (S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-phenylethanol (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)-2-methylpropan-2-ol (S)-1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol (S)-1-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-N-(5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl)pyrrolidine-2-carboxami... (S)-1-(2-Amino-2-carboxyethyl)-3-(2-carboxy-5-phenylthiophene-3-yl-methylpyrimidine-2,4-dione (S)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine (S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperazin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Tri... (S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperidin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Tri... (S)-1-(4-Chlorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol (S)-1-(4-Fluorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]-isoquinolin-6-yl)ethanol (S)-1-(4-Fluorophenyl)-1-(3-(methyl(4-(4-(prop-2-yn-1-yloxy)benzoyl)benzyl)amino)propyl)-1,3-dihydroisobenzofuran-5-carbonitr... (S)-1-(5-Chlorothiophen-2-yl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-... (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-2-methyl-propan-2-ol (S)-1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol (S)-1-(adamantan-2-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol (S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-amide (S)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine (S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide (S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide (S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-oxopyrrolidine-2-carboxamide (S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide (S)-1-(Indolin-1-yl)-2-(2-((3-methoxyphenoxy)methyl)morpholino)ethanone (S)-1-(Indolin-1-yl)-2-(2-((pyridin-3-yloxy)methyl)morpholino)ethanone (S)-1-(Indolin-1-yl)-2-(2-(phenoxymethyl)morpholino)ethanone (S)-1-acetyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide (S)-1-acetyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)pyrrolidine-2-carboxamide (S)-1-benzoyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide (S)-1-benzoyl-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide (S)-1-benzoyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-5-oxopyrrolidine-2-carboxamide (S)-1-benzoyl-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide (S)-1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-1-thiophen-3-yl-ethanol (S)-1-{2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-isochroman-6-carboxylic acid methylamide (S)-2,3-dichloro-N-(2-cyclopropylethyl)-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-(2H-pyran-4-yl)-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-(pentan-3-yl)-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-(pyrrolidin-3-yl)-N-(2,2,2-trifluoroethyl)benzamide (S)-2,3-dichloro-N-cyclopentyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-ethyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-neopentyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-phenyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-dichloro-N-propyl-N-(pyrrolidin-3-yl)benzamide (S)-2,3-Dihydro-1H-indole-2-carboxylic Acid {(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbam... (S)-2,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine (S)-2-((1-methylpyrrolidin-2-yl)methyl)-1H-pyrrolo[2,3-b]pyridine (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione (S)-2-((3-chlorophenoxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine (S)-2-((4-(1H-Indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)-methyl)-8-methyl-2,3-dihydro-[1,4]dioxino-[2,3-f]quinoline (S)-2-((R)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)-1-methylpyrrolidine hydrochloride (S)-2-((S)-(2,3-dichlorophenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-chloro-4-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-methoxy-4-(trifluoromethyl)phenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-bromo-2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(2-fluorophenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(3-fluorophenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(4-fluorophenyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(m-tolyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(o-tolyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(p-tolyl)methyl)morpholine (S)-2-((S)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-1-yl)propano... (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-2-yl)propano... (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-phenylpropanoic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-4-phenylbutanoic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanedioic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid (S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)succinic acid (S)-2-((S)-2-Aminopropanoylamino)-4-methylpentanoic Acid Amide (S)-2-(2-((3-Chlorophenoxy)methyl)morpholino)-1-(indolin-1-yl)ethanone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(... (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3... (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(... (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S... (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-... (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-d... (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-isobutylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-methylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenethylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenylpropanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-4-phenylbutanoic acid (S)-2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,4-diol (S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionyl}-amino)-3-phenyl-propionic... (S)-2-(methylamino)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-3-phenylpropanamide (S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(N-ethyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid (S)-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (S)-2-amino-3-(1H-indol-3-yl)-N-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-2-amino-3-(1H-indol-3-yl)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-2-amino-3-(1H-indol-3-yl)-N-(3-oxo-3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl)propanamide (S)-2-Amino-3-(3-hydroxy-4-phenyl-5-isoxazolyl)propionic Acid (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid (S)-2-amino-3-(naphthalen-2-yl)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-2-amino-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-3-phenylpropanamide (S)-2-amino-N1,N5-bis(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)pentanediamide (S)-2-Aminoadipic acid (S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine (S)-2-chloro-3-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2-chloro-4-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-2-chloro-5-((1-methylpyrrolidin-2-yl)methoxy)-3-(2-(pyridin-4-yl)vinyl)pyridine (S)-2-chloro-N-isobutyl-N-(pyrrolidin-3-yl)-3-(trifluoromethyl)benzamide (S)-2-Me-Tet-AMPA (S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4- chloroph enyl)-1-({3-[(S)-5-cyano-1-(4-fluorop... (S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophe... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydrois... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydrois... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroiso... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisoben... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4- chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl... (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)... (S)-2-[(S)-2-Amino-3-(tetrahydroisoquinoline-3-carboxamide)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-d... (S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-3-biphenyl-4-yl-propionic ac... (S)-3,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3,5-DHPG (S)-3,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3,5-dihydroxyphenylglycine; (S)-3-((1-Methylpyrrolidin-2-yl)methoxy)-5-(phenoxymethyl)isoxazole Hydrochloride (S)-3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate (S)-3-(1H-indol-3-yl)-2-(methylamino)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)propanamide (S)-3-(1H-indol-4-yl)-N-methyl-3-(thiophen-2-yl)propan-1-amine hydrochloride (S)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride (S)-3-(3,4-dichlorophenyl)-N-methyl-3-(naphthalen-1-yl)propan-1-amine hydrochloride (S)-3-(3-Methanesulfonyl-phenyl)-1-propyl-piperidine (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole (S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole (S)-3-(4-chlorophenyl)-N-(4-chlorophenylsulfonyl)-N'-methyl-4-phenyl-4,5-dihydropyrazole-1-carboxamidine (S)-3-(Pyrrolidin-2-ylmethoxy)-5-((3-(trifluoromethyl)-phenoxy)methyl)isoxazole Trifluoroacetate (S)-3-(Pyrrolidin-2-ylmethoxy)-5-((4-(trifluoromethyl)-phenoxy)methyl)isoxazole Trifluoroacetate (S)-3-(Pyrrolidin-2-ylmethoxy)-5-((m-tolyloxy)methyl)-isoxazole Hydrochloride (S)-3-Azido-5-(azidomethyl)-N-((1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-yl)methyl)benzamide (S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-propionic acid (S)-3-bromo-1,2,9,10-tetramethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (S)-3-bromo-1,9,10-trimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-2-ol (S)-3-Carboxy-4-hydroxyphenylglycine (S)-3-chloro-2-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (S)-3-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (S)-3-chloro-N-isobutyl-2-methyl-N-(pyrrolidin-3-yl)benzamide (S)-3-chloro-N-isobutyl-N-(pyrrolidin-3-yl)benzamide (S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid (S)-3-cyclohexyl-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)propanoic acid (S)-3-fluoro-N-isobutyl-2-methyl-N-(pyrrolidin-3-yl)benzamide (S)-3-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)-2-(trifluoromethyl)benzamide (S)-3-hydroxyphenylglycine (S)-3-Hydroxyphenylglycine (S)-3-iodo-1,2,9,10-tetramethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline (S)-3-iodo-1,9,10-trimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-2-ol (S)-3-methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole (S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline ) (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline (S)-4-(1-(3,4-dimethylphenyl)hexyl)-1H-indene hydrochloride (S)-4-(1H-indol-4-yl)-N-methyl-4-(thiophen-2-yl)butan-1-amine hydrochloride (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((2-methylpyridin-3-yl)oxy)methyl)morpholine (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine (S)-4-(2-(Indolin-1-yl)ethyl)-2-((3-methoxyphenoxy)methyl)morpholine (S)-4-(2-(Indolin-1-yl)ethyl)-2-((pyridin-3-yloxy)methyl)morpholine (S)-4-(2-(Indolin-1-yl)ethyl)-2-(phenoxymethyl)morpholine (S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide (S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide (S)-4-(3,4-dichlorophenyl)-N-methyl-4-(naphthalen-1-yl)butan-1-amine hydrochloride (S)-4-(4-methoxyphenyl)-2-methyl-7-(3-((S)-3-methylmorpholino)propoxy)-1,2,3,4-tetrahydroisoquinoline (S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol (S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol (S)-4-(5-((5-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)pentyl)benzene-1,2-diol (S)-4-carboxy-3-hydroxyphenylglycine (S)-4-carboxy-phenylglycine (S)-4-Carboxyphenylglycine (S)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-piperidin-2-yl)-ethyl)-piperidine(5) (S)-4-Methyl-1-(2-(1-(naphthalene-1-sulfonyl)-pyrrolidin-2-yl)-ethyl)-piperidine(10) (S)-4-Methylhomoibotenic acid (S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide (S)-4C3HPG (S)-4CPG (S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl) (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) (S)-5-((2-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((2-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((3-Bromophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((3-Chlorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride (S)-5-((3-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate (S)-5-((3-Fluorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride (S)-5-((3-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((3-Methoxyphenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((4-Bromophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((4-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((4-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((4-Methoxyphenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride (S)-5-((Naphthalen-2-yloxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate (S)-5-((Phenylthio)methyl)-3-(pyrrolidin-2-ylmethoxy)-isoxazole Trifluoroacetate (S)-5-((R)-1-methylpyrrolidin-2-yl)oxazolidin-2-one (S)-5-(5-methoxypyridin-3-yl)-N-methylpent-4-en-2-amine (S)-5-allyl-10-ethynyl-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-5-allyl-9-(ethynyloxy)-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-5-allyl-9-cyanato-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-5-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanoic acid (S)-5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide (S)-6-(1-methylpyrrolidin-2-yl)-quinoline (S)-6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)5,6,7,8-tetrahydronaphthalen-1-ol (S)-6-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)hexanoic acid (S)-6-chloro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (S)-6-Chloro-3-(1-phenylethyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide (S)-6-fluoro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole (S)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline (S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] (S)-7-ethynyl-1-(3-methyl-1,2,4-oxadiazol-5-yl)-12,13,13a,14-tetrahydro-9H,11H-benzo[f]imidazo[5,1-d]pyrrolo[1,2-a][1,5]diazo... (S)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7, 8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione (S)-8-(5-Methoxy-2,1,3,4-tetrahydronaphth-2-yl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione (S)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide (S)-8-OH-DPAT (S)-9-methoxy-2,2,4-trimethyl-5-phenyl-2,5-dihydro-1H-chromeno[3,4-f]quinoline (S)-ABT-089 [2-Methyl-3-(2-(S)-pyrrolidinylmethoxy)pyridine] (S)-ACPA (S)-alpha-Phenylethylamine (S)-AMPA (S)-AP5 (S)-aspartic acid (S)-ATPA (S)-BrHlbo (S)-Chlopheniramine (S)-Demethyl-ACPA (S)-Glu (S)-Hexbutinol (S)-HIBO (S)-Indolin-1-yl(3-(pyrrolidin-2-ylmethoxy)isoxazol-5-yl)-methanone Hydrochloride (S)-N-((1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-yl)methyl)-4-(4-(prop-2-yn-1-yloxy)benzoyl)... (S)-N-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)benzamide (S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide (S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide (S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide (S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)benzamide (S)-N-(2,3-dichlorobenzyl)-N-(pyrrolidin-3-yl)isobutyramide (S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide (S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclopentanecarbonyl)pyrrolidine-2-carboxamide (S)-N-(2-oxo-2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (S)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide (S)-N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide (S)-N-(4-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)butyl)-2-naphthamide (S)-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide (S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide (S)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea (S)-N-isobutyl-2-isopropyl-N-(pyrrolidin-3-yl)benzamide (S)-N-methyl-3-(naphthalen-1-yl)-3-(thiophen-2-yl)propan-1-amine hydrochloride (S)-N-methyl-4-(naphthalen-1-yl)-4-(thiophen-2-yl)butan-1-amine hydrochloride (S)-N-Phenyl-3-(pyrrolidin-2-ylmethoxy)isoxazole-5-carbox-amide Hydrochloride (S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-2-yl)methyl)amino]benzenepropaneamide bis(trifluoroa... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-3-yl)methyl)amino]benzenepropaneamide bis(trifluoroa... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-1-(pyridin-4-yl)methyl)amino]benzenepropaneamide bis(trifluoroa... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-2-phenylethyl) amino]benzenepropaneamide bis-(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-dimethylbutyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-phenylprop- 2-enyl)amino]benzenepropaneamide bis(trifluoroace... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-3-phenylpropyl)amino]benzenepropaneamide bis-(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxo-cyclohexylmethyl)amino]benzenepropaneamide bis(trifluoroacetate... (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxobutyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxoethyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxohexyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxophenylmethyl)amino]benzenepropaneamide bis-(trifluoroacetate) (S)-N-[8-[(3-Aminopropyl)amino]octyl]-4-hydroxy-alpha-[(1-oxopropyl)amino]benzenepropaneamide bis(trifluoroacetate) (S)-N3-(1-(1-Naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (S)-N3-(1-(2-Naphthyl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (S)-N3-(1-Phenylethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide (S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide (S)-N6-(2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl)-N6-propyl4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine (S)-N6-Propyl-N6-(2-(4-(4-(pyridin-4-yl)phenyl)piperazin-1-yl)ethyl)-4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine (S)-N6-Propyl-N6-(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)-4, 5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine (S)-N6-Propyl-N6-(2-(4-(quinolin-5-yl)piperazin-1-yl)ethyl)-4, 5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine (S)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)-butyl]amide (S)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide (S)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}am... (S)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide (S)-Nicotine (S)-SIB-1508Y (S)-tert-butyl 1,5-dioxo-1,5-bis(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethylamino)pentan-2-ylcarbamate (S)-tert-butyl 3-(1H-indol-3-yl)-1-oxo-1-(2-(1,2,3,4-tetrahydroacridin-9-ylamino)ethylamino)propan-2-ylcarbamate (S)-tert-butyl 3-(1H-indol-3-yl)-1-oxo-1-(3-oxo-3-(1,2,3,4-tetrahydroacridin-9-ylamino)propylamino)propan-2-ylcarbamate (S)-Thio-ATPA (S)-Trihexyphenidyl (S)-UH-301 (S)-Zopiclone (S)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone (S)ACPA (S,E)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol (S,S)-1-cyclopentyl-2-(5-fluoro-2-methoxy-phenyl)-1-morpholin-2-yl-ethanol (S,S)-2-(6-aminopyridin-3-yl)-2,5-diazabicyclo[2.2.1]-heptane (Z)-2-amino-4-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one (Z)-2-amino-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one (Z)-2-amino-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one (Z)-2-amino-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-1H-imidazol-5(4H)-one (Z)-2-amino-5-((4-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one (Z)-2-amino-5-((5-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one (Z)-2-amino-5-((6-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one (Z)-2-amino-5-((7-bromo-1H-indol-3-yl)methylene)-1H-imidazol-4(5H)-one (Z)-3-Aminopropen-2-yl)methylphosphinic acid (Z)-4-((1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one (Z)-4-((1H-indol-3-yl)methylene)-2-amino-1-methyl-1H-imidazol-5(4H)-one (Z)-4-((4-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one (Z)-4-((5-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one (Z)-4-((6-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one (Z)-4-((7-bromo-1H-indol-3-yl)methylene)-1-methyl-2-(methylamino)-1H-imidazol-5(4H)-one (Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol (Z)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)benzene-1,2-diol and (Z)-4-(5-((2-amin... (Z)-5-((1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one (Z)-5-((1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one (Z)-5-((1H-indol-3-yl)methylene)-2-amino-1H-imidazol-4(5H)-one (Z)-5-((1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one (Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one (Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one (Z)-5-((4-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one (Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one (Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one (Z)-5-((5-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one (Z)-5-((6-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one (Z)-5-((6-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-(methylthio)-1H-imidazol-4(5H)-one (Z)-5-((7-bromo-1H-indol-3-yl)methylene)-2-thioxoimidazolidin-4-one (Z)-5-(2'-(3'-((E)-1''-hydroxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,... (Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,... (Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H... (Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quino... (Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline (Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline (Z)-CH2OCOC(CH3)3 (Z)-N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-4-phenylbut-3-en-1-amine (Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride ([Dmt1]DALDA) (±)-2-ethylamino-1-phenyl-propan-1-one (±)-nicotine )-5-((6-bromo-1H-indol-3-yl)methylene)-2-(methylamino)-1H-imidazol-4(5H)-one + 1 mM GTP +-(1H-Indol-2-yl)-(3-methyl-piperazin-1-yl)-methanone , 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine , 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine ,14-endoetheno – 7 a (1-(R)-hydroxy-1 methylbutyl)-tetrahydro-nororipavine . (2-Amino-4-(2,2-dimethylpropyl)-5-(4-(1-(methyl)ethyl) phenyl)thiophen-3-yl)(4-chlorophenyl)methanone . (2-Amino-4-(2,2-dimethylpropyl)-5-phenylthiophen-3-yl) (4-chlorophenyl)-methanone . 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl) butan-1-one 0-[(2-Methyl-lH-imidazol-l-yl)methyl]-5,6,8,9,10,llhexahydro-4H-pyrido[3^,l-ji]carbazol-1l-oneHydrochloride 1 1'-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one 1'-(2-(4-(4-fluorophenyl)-5,6-dihydropyridin-1(2H)-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one 1'-(o-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1'-(p-methylcinnamoyl)-[7alpha,8alpha:3',4']-pyrrolidino-6,14-endoethenotetrahydrooripavine 1'-Acetyle-(3R)-(4-Phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydrospiro[Beta-carboline-1,4'-piperidine] 1'-benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4'-piperidine] 1'-[2-(4-phenylpiperazin-1-yl)ethyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(4-chlorobenzoyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(4-chlorophenoxy)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(4-chlorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{2-[4-(4-fluorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1'-{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1, (S)-citalopram 1, 10-diamiodecane 1, 12-DB-3-4-3 1, 2, 3, 4,-tetrahydro-N-methyl)-1,6-naphhyridine 1, 2-Benzenediol, 4-(2-amino-1-hydroxyethyl)- 1, HENECA 1,1-Dibutyl-6-chloro(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline 1,1-Dibutyl-6-chloro-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline 1,1-dimethyl-2-quinolin-6-yl-pyrrolidinium iodide 1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium 1,1-dimethyl-4-phenylpiperazinium iodide 1,1-Dimethylethyl-alpha-(S)-[[[[3-[[(10(S)-cyclohexyl-8,11-dioxo-2-oxa-9,12-diazabicyclo[13.3.1]nonadeca-1(19),15,17-trien-13... 1,1-Dimethylethyl-alpha-(S)-[[[[3-[[(11(S)-cyclohexyl-2-oxa-10,13-diazabicyclo[14.3.1]eicosa-1(20),16,18-trien-14(S)-yl)carbo... 1,1-Dimethylethyl-alpha-(S)-[[[[3-[[(11(S)-cyclohexyl-2-oxa-10,13-diazabicyclo[14.3.1]eicosa-1(20),16,18-trien-14(S)-yl)carbo... 1,2,3,11b-Tetrahydro[1]benzothiopyrano[4,3,2-de]isoquinolin-8,9-diol 1,2,3,4,10,14b-hexahydro-2-methyl-6-triflouromethanesulfonoxydibenzo[c,f]pyrazino[1,2-a]azepin, (+/-) 1,2,3,4,10,14b-Hexahydro-6-hydroxy-2-methyldibenzo[c,f]pyrazino[1,2-a]azepin, (+/-) 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+) 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(+/-) 1,2,3,4,10,14b-hexahydro-6-methoxy-2-methyldibenzo[c,f]-pyrazino[1,2-a]azepin,(-) 1,2,3,4,5,6-Hexahydro-2-benzazocine 1,2,3,4-Tetrahydroisoquinoline 1,2,3,4-Tetrahydroisoquinoline, THIQ 1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1,2,3,7,8,9-Hexadropyrano[2,3-g], 1-(1-indolinyl)-2-propylamines 1,2,3.4-Tetrahydro[2,7]naphthyrldine oxalate 1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol 1,2-dimethoxy-4-propylbenzene; 2-(2H-1,3-benzodioxol-5-yl)ethan-1-amine; butylbenzene 1,2-dimethoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 1,2-dimethoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H-[1,3]dioxolo[4,5:4,5]benzo[1,2- g]benzo[de]quinoline 1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine 1,3,7-n-tripropylxantine 1,3,7-Trimethy1-8-(3-aminostyryl)xanthine 1,3,7-trimethyl 1,3,7-Trimethyl-8-(2,3-dimethoxystyryl)xanthine 1,3,7-Trimethyl-8-(2-methoxystyryl)xanthine 1,3,7-Trimethyl-8-(3,4-dimethoxystyryl)xanthine 1,3,7-Trimethyl-8-(3,5-dimethoxystyryl)xanthine 1,3,7-Trimethyl-8-(3-aminostyryl)xanthine 1,3,7-Trimethyl-8-(3-nitrostyryl)xanthine 1,3,7-Trimethyl-8-(4-methoxystyryl)xanthine 1,3,7-Trimethyl-8-[2-(3-aminophenyl)ethyl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-(benzyloxy)styryl]-xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-(benzyloxy)styryl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-[(4-amino-trans-butenyl)oxy]styryl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-[(4-aminobutyl)oxy]styryl]xanthine 1,3,7-Trimethyl-8-[3,5-dimethoxy-4-[[4-[[(tert-butyloxy)carbonyl]amino]butyl]oxy]styryl]xanthine 1,3,7-Trimethyl-8-[3-(4-phenyl-1-piperazinyl)- propylamino]-purine-2,6-dione hydrochloride 1,3,7-Trimethyl-8-[3-(acetylamino)styryl]xanthine 1,3,7-Trimethyl-8-[3-(trifluoromethyl)styryl]xanthine 1,3,7-Trimethyl-8-[3-[(3-carboxy-1-oxopropyl)amino]styryl]xanthine 1,3,7-Trimethyl-8-[3-[(tert-butyloxy)carbonyl]amino]-styryl]xanthine 1,3,7-Trimethyl-8-[3-[(tert-butyloxy)carbonyl]amino]styryl]xanthine 1,3,7-Trimethyl-8-[3-[bis[(tert-butyloxy)carbonyl]amino]-styryl]xanthine 1,3,7-Trimethyl-8-[3-[bis[(tert-butyloxy)carbonyl]amino]styryl]xanthine 1,3,9-trimethyl 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-bis(2-chloroethyl)-1-nitrosourea 1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}-5-methylbenzene 1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene 1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride 1,3-di-o-tolyl-guanidine 1,3-diallyl-7-methylxantine 1,3-Diallylxantine 1,3-dibenzylxantine 1,3-DibutylX-7-riboside 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1,3-Diethyl-3-(4-hydroxybutyl)-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1,3-Diethyl-7-methyl-8-(4-bromophenoxymethyl)xanthine 1,3-Diethyl-7-methyl-8-(4-chlorophenoxymethyl)xanthine 1,3-Diethyl-7-methyl-8-(4-fluorophenoxymethyl)xanthine 1,3-Diethyl-7-methyl-8-(4-methoxyphenoxymethyl)xanthine 1,3-Diethyl-7-methyl-8-(4-methylphenoxymethyl)xanthine 1,3-Diethyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(2-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(3-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-Diethyl-8-(4-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1,3-diethyl-8-phenyl 1,3-diethyl-8-phenylxanthine 1,3-diethyl-8phenyl 1,3-Diethylxanthine 1,3-diethylxantine 1,3-DihexylX 1,3-dihydro-1-[2-[4-[3-(trifluoromethyl)phenyl-1-piperazinyl]-ethyl]-2H-benzimidol-2-one 1,3-diisobutylxantine 1,3-dimethyl 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-7-n-butyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione hydrochloride 1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-dimethyl-7-[2-(4-phenylpiperazin-1-yl)ethyl]purine-2,6-dione 1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione 1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione 1,3-Dimethyl-8(3,4-dimethoxystyryl)xanthine 1,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)-5-methylthiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H... 1,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)thia-zol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-((2-(thiophen-2-yl)thiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochlo... 1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-8-((4-phenylisoxazol-3-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(2,3-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(2-(thiophen-2-yl)ethyl)-6,7,8,9-tetra-hydropyrazino[2,1-f]purine2,4-(1H,3H)-dione 1,3-Dimethyl-8-(2-methoxystyryl)xanthine 1,3-Dimethyl-8-(2-methyl-2-phenylethyl)-6,7,8,9-tetrahy-dropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 1,3-Dimethyl-8-(2-phenoxyethyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(3,4-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(3,5-dimethoxystyryl)xanthine 1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(3-aminostyryl)xanthine 1,3-Dimethyl-8-(3-nitrostyryl)xanthine 1,3-Dimethyl-8-(3-phenylpropyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(4-methoxystyryl)xanthine 1,3-Dimethyl-8-(naphtha-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 1,3-Dimethyl-8-(propyn-2-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-phenethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-dimethyl-8-phenyl 1,3-Dimethyl-8-phenyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-8-[3-(2-methoxy-2-oxoethoxy)-phenyl]xanthine 1,3-Dimethyl-8-[3-(trifluoromethyl)styryl]xanthine 1,3-Dimethyl-8-[3-methoxy-4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]-xanthine 1,3-Dimethyl-8-[3-methoxy-4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-methoxy-4-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[3-{2-(morpholin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine 1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine 1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine 1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]xanthine 1,3-Dimethyl-8-[4-(2-morpholin-4-ylethoxy)phenyl]xanthine 1,3-Dimethyl-8-[4-(2-piperidin-4-ylethoxy)phenyl]xanthine 1,3-Dimethyl-8-[4-(2-pyrrolidin-1-ylethoxy)phenyl]xanthine 1,3-Dimethyl-8-[4-(3-imidazol-1-ylpropoxy)phenyl]xanthine 1,3-Dimethyl-8-[4-(3-morpholinopropoxy)benzyl]xanthine 1,3-Dimethyl-8-[4-(dimethylamino)styryl]xanthine 1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2-oxo-ethoxy}-phenyl]-xanthine 1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-methoxy-3-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthin 1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthin 1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phenyl]xanthine 1,3-Dimethyl-8-[4-{3-(1,4-dioxa-8-azaspiro[4.5]decan-1-yl)- propoxy}benzyl]-xanthine 1,3-Dimethyl-8-[4-{3-(1H-imidazol-1-yl)propoxy}benzyl] xanthine 1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-oxo-ethoxy)-4-methoxy}-phenyl]-xanthine 1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine 1,3-Dimethyl-8-[{3-(2-(homoveratrylamino)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine 1,3-Dimethyl-8-[{3-(2-(imidazol-1-yl)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine 1,3-Dimethyl-8-[{3-(2-methoxy-2-oxoethoxy)-4-methoxy}-phenyl]xanthine 1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine 1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-3-methoxy}-phenyl]-xanthin 1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-3-methoxy}-phenyl]-xanthine 1,3-Dimethyl-8-[{4-(2-(homoveratrylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine 1,3-Dimethyl-8-[{4-(2-(imidazol-1-yl)-2-oxoethoxy)-3-methoxy}-phenyl]xanthine 1,3-Dimethyl-8-[{4-(2-methoxy-2-oxoethoxy)-3-methoxy}-phenyl]xanthine 1,3-dimethyl-8phenyl 1,3-Dimethyl-8[4-(dimethylamino)styryl]xanthine 1,3-dimethyl-9-(2-(p-tolyloxy)ethyl)-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-dimethyl-9-(2-(pyridin-2-yl)ethyl)-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6... 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-dimethyl-9-(pyridin-2-ylmethyl)-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-dipropyl 1,3-Dipropyl-7-methyl-8-styrylxanthine 1,3-Dipropyl-8-(4-hydroxyphenyl)xanthine 1,3-Dipropyl-8-(p-hydroxyphenyl)xanthine 1,3-Dipropyl-8-phenylxanthine 1,3-Dipropyl-8-[1-(1-p-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-3,7-dihydro-purine-2,6-dione 1,3-Dipropyl-8-{1-[1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-3,7-dihydro-purine-2,6-dione 1,3-Dipropyl-8-{1-[1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-3,7-dihydro-purine-2,6-dione 1,3-DipropylX-7-riboside 1,3-Dipropylxanthine 1,3-n-dipropyl-7-propargyl 1,3-n-dipropylxantine 1,4-bis[3-(1,2,3,4-Tetrahydroacridin-9-yl)aminopropyl]piperazine 1,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene 1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1Hpyrazole-3-carboxamide 1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole 1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione 1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1,7-dimethyl-3-isobutylxantine 1,7-dimethyl-3-n-propylxantine 1,7-Dimethylxanthine 1,9-DimethylX 1,N6-Ehteno-2-oxoado 1-( 2,5-Dimet hoxy-4-propionylphenyl)-2-aminopropane Hydrochloride 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-(3,3-dimethylbutyl)piperazine 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-(cyclopropylsulfonyl)piperazine 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-(methylsulfonyl)piperazine 1-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazine 1-((1-((1H-Imidazol-1-yl)methyl)cyclopropyl)methyl)-3-(3,4-dimethoxyphenyl)thiourea 1-((1H-Indol-3-yl)methyl)-4-(1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate)piperidin-4-ol oxalate 1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1-((2 ,6-dimethoxy-[1,1 -biphenyl]-3-yl)methyl)-4- methylpiperidine 1-((2 ,6-dimethoxy-[1,1 -biphenyl]-3-yl)methyl)-4-(2- methoxyphenyl)piperazine 1-((2 -methoxy-6-methyl-[1,1-biphenyl]-3-yl)methyl)-4- methylpiperidine 1-((2 -methoxy-6-methyl-[1,1-biphenyl]-3-yl)methyl)-4-(2- methoxyphenyl)piperazine 1-((2 -methoxy-[1,1-biphenyl]-3-yl)methyl)-4- methylpiperidine 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5R*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,5S*,6S*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,6R*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,6R*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,6R*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,6R*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 1-((2R*,6S*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,6S*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1-((2R*,6S*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,6S*)-6-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide and 1-((2R*,6R*)-6-(4-Benzylphenyl)- 1,4... 1-((2R*,6S*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R*,6S*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+) 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride 1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((5-bromopyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((5-ethynylpyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate 1-((6-bromopyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride 1-((6-bromopyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((6-Chloro-2 -methoxy-[1,1 -biphenyl]-3-yl)methyl)-4-(2- methoxyphenyl)piperazine 1-((6-Chloro-2-methoxy-[1,1-biphenyl]-3-yl)methyl)-4- methylpiperidine 1-((6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride 1-((6-chloropyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride 1-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-3-morpholinopropan2-ol 1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride 1-((7-(2-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)methyl)- 4-methylpiperidine 1-((R)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea 1-((S)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea 1-((S)-4-Fluoro-phenyl)-1-[(4aR,5S)-1-(4-fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-ethanol 1-(1,3-Benzodioxol-4-ylmethyl)-4-(2-methylphenyl)piperazine 1-(1,3-Benzodioxol-4-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperazine 1-(1,3-Benzodioxol-4-ylmethyl)-4-[4-(trifluoromethyl)phenyl]piperazine 1-(1,3-Benzodioxol-5-ylmethyl)-4-(2-methylphenyl)piperazine 1-(1,3-Benzodioxol-5-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperazine 1-(1,3-Benzodioxol-5-ylmethyl)-4-[4-(trifluoromethyl)phenyl]piperazine 1-(1,4-dioxaspiro[4,5]dec-2-ylmethyl)-4-(2-methoxyphenyl)piperazine 1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 1-(1-(2-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-(2-fluorophenyl)-2-(2-methoxyphenyl)ethyl)piperazine 1-(1-(3-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-(3-fluorophenyl)-2-(2-methoxyphenyl)ethyl)piperazine 1-(1-(4-(1H-Indol-3-yl)butyl)piperidin-4-yl)-5-chloro-1Hbenzo[d]imidazol-2(3H)-one 1-(1-(4-(Benzo[d]oxazol-2-yl)butyl)piperidin-4-yl)-5- chloro-1H-benzo[d]imidazol-2(3H)-one 1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone 1-(1-(4-fluorophenyl)-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-(4-fluorophenyl)-2-(2-methoxyphenyl)ethyl)piperazine 1-(1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo-[1,5-b]isoquinolin-6-yl)but-3-en-1-ol 1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one 1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 1-(1-adamantylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(1-Methoxy-9,10-dihydro-9-anthracenyl)methanamine 1-(1-Methyl-1H-pyrrol-2-yl)-2-(piperidin-1-yl)ethanols 1-(1-Methyl-1H-pyrrol-2-yl)ethanoneamines 1-(1-methylpyrrol-2-yl)-2-(3H-[1,2,4]triazolo[4,3-a]benzimidazol-1-ylsulfanyl)ethanone 1-(1-NAPHTHYL)PIPERAZINE 1-(1-phenyl-2-(2-(trifluoromethoxy)phenyl)ethyl)piperazine 1-(1-phenyl-2-(2-propoxyphenyl)ethyl)piperazine 1-(1H-indol-4-yloxy)-3-(cycloheptylamino)propan-2-ol 1-(1H-indol-4-yloxy)-3-(cyclohexylamino)propan-2-ol 1-(1H-indol-4-yloxy)-3-(cyclopentylamino)propan-2-ol 1-(1H-indol-4-yloxy)-3-(pentan-3-ylamino)propan-2-ol 1-(1H-indol-4-yloxy)-4-(cyclohexylamino)butan-2-ol 1-(1H-indol-5-yloxy)-3-(cyclohexylamino)propan-2-ol 1-(2 ,6-dimethoxy-[1,1 -biphenyl]-3-yl)-N,N-dimethylmethanamine 1-(2 ,6-dimethoxy-[1,1 -biphenyl]-3-yl)-N-methylmethanamine 1-(2 -methoxy-6-methyl-[1,1-biphenyl]-3-yl)-N,N-dimethylmethanamine 1-(2 -methoxy-[1,1 -biphenyl]-3-yl)-N-methylmethanamine 1-(2 -methoxy-[1,1-biphenyl]-3-yl)-N,N-dimethylmethanamine 1-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)-4,4-difluoropiperidine 1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-4-(4-fluoro-phenyl)-1,2,3,6-tetrahydro-pyridine 1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-piperidine 1-(2,3-Dichlorophenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine 1-(2,3-Dichlorophenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 1-(2,3-dimethoxyphenyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]methanamine 1-(2,4,5-trimethoxyphenyl)-2-aminopropane HCI 1-(2,4-Dichloro-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(2,4-dichlorophenyl)-4-(hydroxymethyl)-N-(piperidin-1-yl)-5-(4-(pyridin-3-yl)phenyl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-(fluoromethoxy)phenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-morpholino-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-morpholino-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(pyrrolidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-morpholino-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-N-piperidin-1-yl-1H-pyrazole-4-carboxamide 1-(2,4-Dichlorophenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,4-Difluorophenyl)-3-[4-(3-pyridylethynyl)-2-thiazolyl]urea 1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,4-Dimethyl-phenyl)-4-(2-phenyl-cyclopropylmethyl)-piperazine; hydrobromide 1-(2,4-dimethylphenyl)-4-(((1R,2S)-2-phenylcyclopropyl)methyl)piperazine 1-(2,4-dimethylphenyl)-4-(((1S,2R)-2-phenylcyclopropyl)methyl)piperazine 1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,5-dimethoxy-4-ethoxyphenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 1-(2,5-dimethoxy-4-fluorophenyl)-2-aminopropane HCI 1-(2,5-Dimethoxy-4-hydroxypheny1)-2-aminopropane Hydrogen Oxalate 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane, (+) 1-(2,5-dimethoxy-4-iodophenyl)-2-aminopropane, (-) 1-(2,5-dimethoxy-4-methylphenyl)-2-aminopropane 1-(2,5-dimethoxy-4-n-hexylphenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-n-propylphenyl)-2-aminopropane HCI 1-(2,5-dimethoxy-4-nitrophenyl)-2-aminopropane HCI 1-(2,5-Dimethoxy-4-octylphenyl)-2-aminopropane Hydrochloride 1-(2,5-dimethoxy-4-t-butylphenyl)-2-aminopropane HCI 1-(2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2,6-Dimethoxypyridin-3-yl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-(1H-Imidazol-1-yl)ethyl)-3-(3,4-dimethoxyphenyl)thiourea 1-(2-(2,3-dihydrobenzofuran-7-yl)-1-phenylethyl)piperazine 1-(2-(2-(cyclopropylmethoxy)phenyl)-1-phenylethyl)piperazine 1-(2-(2-(difluoromethoxy)-6-fluorophenyl)-1-phenylethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-(2-fluorophenyl)ethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-(3-fluorophenyl)ethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-(4-fluorophenyl)ethyl)piperazine 1-(2-(2-(difluoromethoxy)phenyl)-1-phenylethyl)piperazine 1-(2-(2-cyclopropoxyphenyl)-1-phenylethyl)piperazine 1-(2-(2-fluoro-6-methoxyphenyl)-1-phenylethyl)piperazine 1-(2-(2-isopropoxyphenyl)-1-phenylethyl)piperazine 1-(2-(2-methoxyphenyl)-1-phenylethyl)piperazine 1-(2-(3-fluoro-2-methoxyphenyl)-1-phenylethyl)piperazine 1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate 1-(2-Aminopropyl)-3-methyl-8,9-dihydropyranol[3,2-e]-indole Hydrochloride 1-(2-Aminopropyl)-8,9-dihydropyrano[3,2-e]indole Hydrochloride 1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 1-(2-bromo-2-phenylethyl)-6-(methylthio)-4-(pyrrolidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-bromo-2-phenylethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-bromo-2-phenylethyl)-N-(2-ethoxyethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-bromo-2-phenylethyl)-N-butyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-Bromo-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2-Bromo-4-isopropyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(2-bromophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2-Bromophenyl)-5-(4-methoxyphenyl)-N3-(piperidin-1-yl)-1H-pyrazole-3,4-dicarboxamide 1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-chlorophenyl)ethyl)-N,N-diethyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(2-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(3-fluorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-(4-fluorophenyl)ethyl)-N-(4-fluorobenzyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-Chloro-2-phenyl-ethyl)-6-methylsulfanyl-4-morpholin-4-yl-1H-pyrazolo[3,4-d]pyrimidine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-4-(piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-6-(methylthio)-N-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(ethylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-diethyl-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N,N-dimethyl-4-morpholino-1H-pyrazolo[3,4-d]pyrimidin-6-amine 1-(2-chloro-2-phenylethyl)-N-(2-fluorophenethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N-(3-fluorophenyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N-propyl-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1-(2-chloro-2-phenylethyl)-N6,N6-dimethyl-N4-propyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 1-(2-Chloro-4-cyanophenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-Chloro-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 1-(2-Chloro-4-methanesulfonylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-Chloro-4-methylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(1-cyclopropyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 1-(2-chlorophenyl)-5-(4-chlorophenyl)-3-(1-isopropyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-methyl-3-(1-(2-phenylpropan-2-yl)-1H-imidazol-4-yl)-1H-pyrazole 1-(2-chlorophenyl)-5-(4-chlorophenyl)-4-methyl-3-(1-phenyl-1H-imidazol-4-yl)-1H-pyrazole 1-(2-Dimethylaminoethyl)-4-hydroxyindole 1-(2-methoxy-6-methyl-[1,1-biphenyl]-3-yl)-N-methylmethanamine 1-(2-Methoxy-9,10-dihydro-9-anthracenyl)methanamine 1-(2-Methoxy-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(2-methoxyphenyl)-4-((7-(2-methoxyphenyl)benzo[d] [1,3]dioxol-5-yl)methyl)piperazine 1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine 1-(2-Methoxyphenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine 1-(2-Methoxyphenyl)-4-(4-(1-phenyl-1H-1,2,3-triazol-4-yl)butyl)piperazine 1-(2-Methoxyphenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine 1-(2-Methoxyphenyl)-4-(4-(4-phenyl-1H-1,2,3-triazol-1-yl)butyl)piperazine 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1-(2-Methoxyphenyl)-4-{1,4,8-trioxaspiro[4.5]decan-2-ylmethyl}piperazine 1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride 1-(2-Methoxyphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrotrifluoroacetate 1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide 1-(2-Methoxyphenyl)piperazine 1-(2-phenoxyphenyl)-3-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]urea 1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin 1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one 1-(2’-Butyl)-1H-benzotriazole-5-carboxylic acid 1-(2’-Ethoxy-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(2’-Ethylsulfanyl-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(2’-Methoxy-1’-methyl-ethyl)-1H-benzotriazole-5-carboxylic acid 1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperazine 1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperidine 1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4- one 1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4-ol 1-(3-(1H-Imidazol-1-yl)-propyl)-3-(4-methylsulfanyl-phenyl)-thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,3-dihydrobenzo[b][1,4]dioxin-7-yl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,4-dimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4,5-trimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxybenzyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)-1-methylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)urea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,5-dimethoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3-methoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(benzyloxy)phenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(dimethylamino)phenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-acetylphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-ethylphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-fluorophenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methoxyphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methylphenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-nitrophenyl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-(benzo[d][1,3]dioxol-6-yl)thiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-benzylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-butylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-cyclohexylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-isopropylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-methylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-naphthalen-1-ylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-phenylthiourea 1-(3-(1H-Imidazol-1-yl)propyl)-3-tert-butylthiourea 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol 1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidine-4-carbonitrile 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 1-(3-(Benzo[d]thiazol-2-yl)propyl)-4-(4-chlorophenyl) piperidin-4-ol hydrochloride 1-(3-(trifluoromethyl)phenyl)piperazine 1-(3-Chloro-4-fluorophenyl)-4-(morpholin-4-yl)-1,5-dihydro-pyrrole-2-one 1-(3-Chlorophenyl) piperazine 1-(3-chlorophenyl)-2-(cyclobutylamino)propan-1-one 1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(3-Hydroxypropyl)uracil 1-(3-Isopropoxypropyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(3-Methoxy-7,12-dihydro-12-tetraphenyl)methanamine 1-(3-Methoxy-9,10-dihydro-9-anthracenyl)methanamine 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 1-(3-Methoxyphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(3-Methylphenyl)-4-morpholin-1-yl-2,4-dihydro-pyrrol-2-one 1-(3-Phenoxypropyl)-4-phenylpiperazine 1-(3-tert-Butyldimethylsilyloxypropyl)uracil 1-(3-Triphenylsilyloxypropyl)uracil 1-(3-Tritylaminopropyl)uracil 1-(3-Trityloxypropyl)uracil 1-(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-heptan-1-one 1-(3’,5’-Difluorobenzyl)-1H-benzotriazole-5-carboxylic acid 1-(3’-Methoxybenzyl)-1H-benzotriazole-5-carboxylic acid 1-(3’-Pentyl)-1H-benzotriazole-5-carboxylic acid 1-(4,4-Bis(4-chlorophenyl)butyl)-4-(4-chlorophenyl)piperidin-4-ol Hydrochloride 1-(4,5-dimethyl-1H-benzimidazol-2-yl)-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)methanamine 1-(4,5-Dimethyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(4,5-Diphenyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(4-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazin-1-yl)-3,3-dimethylbutan-1-one 1-(4-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazin-1-yl)ethanone 1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2,3-dichlorophenyl)piperazine 1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2-methoxyphenyl)piperazine 1-(4-(1-pyrrolidinyl)-2-butynyl)-2-pyrrolidinone 1-(4-(1H-Imidazol-1-yl)butyl)-3-(3,4-dimethoxyphenyl)thiourea 1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(naphtha-len-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol 1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(quinolin-3-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol 1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-(2-methoxyphenyl)piperazin-1-yl)-2-(4-phenyl-6-(trifluoromethyl)pyrimidin-2-ylthio)propan-1-one 1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol 1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(quinolin-6-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol 1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)butan-2-ol 1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride 1-(4-(3-(2,4-dimethoxyphenyl)-1-m-tolyl-1H-pyrazole-5-carbonyl)piperazin-1-yl)ethanone 1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)-2-methylpropan-1-one 1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)ethanone 1-(4-(3-(piperidin-1-yl)propoxy)benzyl)piperidine 1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea 1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea 1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2,3-dichlorophenyl)piperazine 1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine 1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine 1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine 1-(4-(4-chlorophenyl)-5,6-dihydropyridin-1(2H)-yl)-3,3-diphenylpropan-1-one 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 1-(4-(Benzo[d]oxazol-2-yl)butyl)-4-(4-chlorophenyl) piperidin-4-ol 1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl) piperidin-4-ol 1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol 1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione 1-(4-(N-hydroxyl)aminobenzenesulfonyl)naphthalene 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-olol 1-(4-acetyl-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-amino-3-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one 1-(4-aminobenzenesulfonyl)naphthalene 1-(4-aminobenzyl)indene 1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-aminophenyl)-2-pyrrolidin-1-yl-pentan-1-one 1-(4-azio-3-iodophenyl)-2-pyrroldin-1-yl-pentan-1-one 1-(4-benzhydrylpiperazin-1-yl)-3-(3-methyl-1H-indol-4-yloxy)propan-2-ol 1-(4-benzyl-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-Benzyl-2,5-dimethoxyphenyl)-2-aminopropane Hydrochloride 1-(4-Biphenyl-4-y)-4-(4-chlorophenyl)butyl]-4-(4-chlorophenyl)piperidin-4-ol 1-(4-bromo-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-Bromophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 1-(4-Bromophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-(4-Carboxy-2,5-dimet hoxyphenyl)-2-aminopropane Hydrochloride 1-(4-chloro-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(4-Chloro-2,6-dimethylphenyl)-5-(1-methoxymethylpropyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochlorid... 1-(4-Chloro-2-cyanophenyl)-5-(1-ethylpropyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Chloro-2-cyanophenyl)-5-(1-methoxymethylpropyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Chloro-2-cyanophenyl)-5-(1-propylbutyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 1-(4-Chloro-2-cyanophenyl)-5-(2-methoxy-1-methoxy-methylethyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triaza-acenaphthylene 1-(4-Chloro-2-methylbenzyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid cyclohexylamide 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 1-(4-Chloro-phenyl)-5-(1-methoxymethyl-propyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one trifluoroacet... 1-(4-Chloro-phenyl)-5-cyano-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid piperidin-1-ylamide 1-(4-Chloro-phenyl)-7-methyl-5-(1-propylbutyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(ethylthio)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(hydroxymethyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfinyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylsulfonyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylthio)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylthio)-N-(pyrrolidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-fluoro-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-iodo-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(morpholin-4-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-(pyrrolidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-N-[4-(trifluoromethyl)benzyl]-1H-imidazole-4-carbox-amide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N,N-diethyl-5-methyl-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1R,2R)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1S,2S)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N-(hexahydrocyclopenta[c]pyrrol-2-(1H)yl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-N-(trans-4-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carbox-amide 1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-Chlorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione 1-(4-Chlorophenyl)-3-pyrrolidin-1-yl-pyrrole-2,5-dione 1-(4-chlorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride 1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one  1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl) butan-1-one hydrochloride 1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride 1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl 1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride 1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine 1-(4-Chlorophenyl)-4-azepan-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-azepan-1-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-piperidin-1-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-2,4-dihydro-pyrrol-2-one 1-(4-Chlorophenyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1-(4-Chlorophenyl)-4-{[1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Chlorophenyl)-4-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazine 1-(4-Chlorophenyl)-5-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-1,2,4-triazole-3-carboxamide Dihydrochloride 1-(4-Chlorophenyl)-5-cyano-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-N-cycloheptyl-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-N-cyclohexyl-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-difluorophenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2,5-dichlorophenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2-ethylphenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-(2-methoxyphenyl)-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide 1-(4-chlorophenyl)-N-cyclohexyl-2-phenyl-1H-imidazole-4-carboxamide 1-(4-Chlorophenyl)-N-cyclopentyl-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazole-4-carboxamide 1-(4-Cyan0-2,5-dimethoxyphenyl)-2-aminopropane Hydrochloride 1-(4-Cyano-4,4-diphenylbutyl)-4-phenylpiperidine-4-carbonitrile 1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Amide 1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Ethyl Ester Hydrochloride 1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Hydrochloride 1-(4-Ethoxy-phenyl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea 1-(4-ethylphenyl)-3-methyl-6-(4-(4-(1-phenylvinyl)cyclohexyl)butyl)-1,2,3,4-tetrahydronaphthalene 1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one 1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-(4-Fluorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione 1-(4-fluorophenyl)-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 1-(4-fluorophenyl)-4-(3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one 1-(4-fluorophenyl)-4-(4-(pyridin-2-yl)-1,4-diazepan-1-yl)butan-1- one oxime 1-(4-fluorophenyl)-4-(4-(pyrimidin-2-yl)-1,4-diazepan-1-yl)butan1-one oxime 1-(4-fluorophenyl)-4-(8-phenyl-3,8-diaza-bicyclo[3.2.1]octan-3-yl)butan-1-one 1-(4-Fluorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 1-(4-Fluorophenyl)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine 1-(4-Fluorophenyl)-4-{[1-(4-fluorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Fluorophenyl)-4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazine 1-(4-Hydroxyphenyl)-4-{[1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Iodophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-(4-Methanesulfonyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(4-Methoxy-2-methylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydromethanesulfonate 1-(4-Methoxy-9,10-dihydro-9-anthracenyl)methanamine 1-(4-Methoxy-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(4-Methoxycarbonyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(4-methoxyphenyl)-2-[4-[(3-methyl-1,2-oxazol-5-yl)methyl]piperazin-1-yl]ethanol 1-(4-Methoxyphenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one 1-(4-Methoxyphenyl)-4-{[1-(4-chlorophenyl)-1H-1,2,3-triazol-4-yl]methyl}piperazine 1-(4-Methylphenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 1-(4-Methylphenyl)-7-methyl-5-(1-propylbutyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide 1-(4-p-Tolyl-butyl)-piperidine 1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone 1-(4-Phenyl-1-piperazinyl)-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone 1-(4-Phenyl-1-piperazinyl)-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone 1-(4-Phenyl-1-piperazinyl)-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone 1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone 1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone 1-(4-Phenyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(4-tert-butylbenzyl)-3-(1-(3-fluoro-4-(methylsulfonamido)phenyl)ethyl)thiourea 1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 1-(4-{[4-(2,4-Diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanone 1-(4-{[4-(2,4-Diamino-6-ethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanol 1-(4-{[4-(2,4-Diamino-6-ethyl-pyrimidin-5-yl)-phenylamino]-methyl}-phenyl)-ethanone 1-(5,5-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl 1-(5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-yl)methyl)-fenchylamine 1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea 1-(5-Chloro-pyridin-2-yl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(5-Chloropyridin-2-yl)-2-(2,4-dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 1-(5-chloropyridin-2-yl)-4-(3-((4-fluorophenyl)thio) propyl)-1,4-diazepane hydrochloride 1-(5-chloropyridin-2-yl)-4-(4-(4-fluorophenyl)butyl)piperazine 1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201) 1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate 1-(5-Oxohexyl)theobromine (pentoxifylline) 1-(5-Phenyloxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(5-Triphenylsilyloxypentyl)uracil 1-(5-Tritylaminopentyl)uracil 1-(5-Trityloxypentyl)uracil 1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo [d]imidazol-2(3H)-one 1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-5,6- dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one 1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[cd] indol-2(1H)-one 1-(6-Chloro-2 -methoxy-[1,1-biphenyl]-3-yl)-N,N-dimethylmethanamine 1-(6-Chloro-2 -methoxy-[1,1-biphenyl]-3-yl)-N-methylmethanamine 1-(6-chloro-pyridin-3-yloxymethyl)-cyclopropylamine; hydrochloride 1-(6-Methoxy-pyridin-3-yl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1-(7-(2-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)-N,Ndimethylmethanamine 1-(7-(2-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)-N-methylmethanamine 1-(8-Bromo-2,3,6,7-tetrahydrobenzo[1,2-b;4,5-b′]difuran-4-yl)2-aminoethane 1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate 1-(adamantan-1-ylamino)-3-(1H-indol-4-yloxy)-propan-2-ol 1-(adamantan-1-ylamino)-3-(1H-indol-5-yloxy)-propan-2-ol 1-(adamantan-1-ylamino)-4-(1H-indol-4-yloxy)-butan-2-ol 1-(allyloxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 1-(allyloxy)-2-methoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H- [1,3]dioxolo[4,5:4,5]benzo[1,2-g]benzo[de]quinoline 1-(allyloxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine 1-(Aminomethyl)-6-hydroxynaphthalene 1-(Aminomethyl)-6-methoxynaphthalene 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one 1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one 1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(3-(4-chlorophenyl)-3- hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-pentan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one 1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(4-(bis(4-fluorophenyl) methyl)piperazin-1-yl)pentan-1-one dihydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride 1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride 1-(benzo[d]thiazol-2-yl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine 1-(benzo[d]thiazol-2-ylmethyl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine 1-(Bicyclo[2.2.1]hept-5-en-2-yl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea 1-(bis(4-chlorophenyl)methyl)-3-((3,5-difluorophenyl)(methylsulfonyl)methylene)azetidine 1-(cyano-2,5-dimethoxyphenyl)-2-aminopropane HCI 1-(cyclobutylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(cyclohexylcarbonyl)-4-(diphenylmethyl)-1,4-diazepane 1-(Cyclohexylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(cyclopentylcarbonyl)-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine 1-(cyclopropylmethoxy)-2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 1-(cyclopropylmethoxy)-2-methoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H- [1,3]dioxolo[4,5:4,5]benzo[1,2-g]benzo[de]quinolin... 1-(cyclopropylmethoxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 1-(hexyloxy)-2-methoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H- [1,3]dioxolo[4,5:4,5]benzo[1,2-g]benzo[de]quinoline 1-(Isopropoxymethyl)-9-(4-methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine 1-(oxazol-2-yl)-1-oxo-9(Z)-octadecene 1-(pyridin-3-yloxymethyl)-cyclopropylamine; hydrochloride 1-([1,1'-biphenyl]-2-yl)-4-(3,4-dichlorophenethyl)piperazine hydrochloride 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1) 1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1) 1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(4-[trifluoromethyl]-benzoyl)amino-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(alpha-toluenesulfonyl)amino-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-6-(4-n-propylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-6-(4-phenylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-4-phenyl-6-(phenylaminocarbonyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(2-furoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(2-[4-methoxyphenyl]ethylamino)carbonyl-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-chlorobenzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-tert-butylbenzyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-[2-phenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-[3-phenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(4-[4-tert-butylphenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-(tert-butoxymethylcarbonyl)aminophenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-6-phenylethoxy-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline 1-Acetyl-D-lysergic acid diethylamide 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 1-acetyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2,3-dihydroindole-5-carboxamide 1-Adrenaline 1-allyl-3,7-dimethylxantine 1-Amino-2-phenylethane 1-Benzhydryl-1H-benzotriazole-5-carboxylic acid 1-Benzoyl-4-cyclohexyl-1,4-diazaspiro[5.5]undecane-3,5-dione 1-Benzoyl-9-benzyl-4-cyclohexyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 1-Benzoyl-9-tert-butyl-4-cyclohexyl-1,4-diazaspiro[5.5]undecane-3,5-dione 1-Benzoylpiperazine 1-Benzyl-1H-benzotriazole-5-carboxylic acid 1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-Benzyl-2-pyridin-2-yl-1H-benzoimidazole 1-Benzyl-2-thiazol-4-yl-1H-benzoimidazole 1-benzyl-3-(N,N-dimethylaminoethyl)indene 1-Benzyl-4-(3-hydroxyphenyl)piperidine 1-benzyl-4-(4-methoxybenzyl)piperazine 1-benzyl-4-methyl-6-phenyl-3-(phenylsulfonyl)pyridin-2(1H)-one 1-Benzyl-4-[3-(methylsulfonyl)phenyl]piperazine 1-Benzyl-4-[3-(methylsulfonyl)phenyl]piperidine 1-Benzyl-4-{2-[2-(mesityloxy)ethoxy]ethyl}piperazine dihydrochloride 1-benzyl-5,6-dimethoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 1-Benzyl-N-(2-cyclohexylidene-2-fluoroethyl)-4-piperidinamine 1-Benzyl-N-(2-cyclopentylidene-2-fluoroethyl)-4-piperidinamine 1-Benzyl-N-(4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl)-1H-1,2,3-triazole-4-carboxamide 1-benzyl-N-cycloheptyl-4-oxo-1,4-dihydroquinoline-3-carboxamide 1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide 1-benzyl-N-cyclohexyl-7-methoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide 1-Benzylpiperazine 1-beta-hydroxyethyl-3-methylxantine 1-Butanoyl-d-lysergic acid diethylamide 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 1-butoxy-2-methoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H-[1,3]dioxolo[4,5:4,5]benzo[1,2- g]benzo[de]quinoline 1-Butyl-1H-benzotriazole-5-carboxylic acid 1-Butyl-4-(2-(2-fluoroethoxy)phenyl)piperazine 1-Butyl-4-(2-methoxyphenyl)piperazine 1-Butyl-8-(4-carboxy)phenylxanthine 1-Butyl-8-(4-carboxymethyloxy)phenylxanthine 1-Butyl-8-(4-sulfophenyl)xanthine 1-Butyl-8-phenylxanthine 1-Butyl-8-[4-((4-(2-metoxyphenyl-piperazin-1-yl)-2-oxoethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-acetyl-piperazin-1-yl)-2-oxoethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-benzyl-piperazin-1-yl)-2-oxoethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-benzyloxycarbonylpiperazin-1-yl)-2-oxoethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-carboxymethyl)phenylamino-2-oxoethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-ethoxycarbonyl-piperazin-1-yl)-2-oxo-ethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-ethylpiperazin-1-yl)-2-oxo-ethoxy)phenyl]xanthine 1-Butyl-8-[4-((4-phenylpiperazin-1-yl)-2-oxoethoxy)phenyl]xanthine 1-Butyl-8-[4-(carboxymethyl)phenyl]xanthine 1-Butylpsilocin 1-Butylpsilocybin 1-Butyltheobromine 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1-Cyclobutyl-1H-benzotriazole-5-carboxylic acid 1-Cyclohexyl-1H-benzotriazole-5-carboxylic acid 1-Cyclohexyl-3-(4-phenyl-1H-imidazol-2-yl)-9H-Beta-carboline 1-Cyclopentyl-1H-benzotriazole-5-carboxylic acid 1-Cyclopropyl-1H-benzotriazole-5-carboxylic acid 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 1-deaza-2-Cl-CHA (2c) 1-deaza-2-Cl-CPA (2b) 1-deaza-2-Cl-PIA (2a) 1-deazaadenosine 1-deazaCHA (3c) 1-deazaCPA (3b) 1-deazaNECA (10) 1-deazaPIA (3a) 1-Deoxysalvinorin A 1-ethoxy-2-methoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H-[1,3]dioxolo[4,5:4,5]benzo[1,2- g]benzo[de]quinoline 1-Ethoxy-4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-4-aza-tricyclo[5.2.2.0*2,6*]undecane-3,5,8-trione 1-ethyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1-ethyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin 1-Ethyl-1H-benzotriazole-5-carboxylic acid 1-ethyl-1H-benzo[d]imidazol-2(3H)-one 1-Ethyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-10-ol 1-Ethyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol 1-ethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 1-Ethyl-3,3-dimethyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1-ethyl-3-methylxantine 1-Ethyl-3-{(1,4-cis)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 1-Ethyl-3-{(1,4-trans)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 1-ethyl-5-methoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 1-Ethyl-8-(2,3-dimethoxyphenethyl)-3-propargyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-(2-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-(4-(4-(3-fluorobenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-fluorobenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-methoxybenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-methoxyphenyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-methylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(4-phenethylpiperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-(piperidine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 1-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione 1-ethyl-8-phenylxanthine 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 1-Ethyltheobromine 1-Hydroxy-1-[5-(2-pyridyl)oxazol-2-yl]-7-phenylheptane 1-Hydroxy-1-[5-(2-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1-hydroxyindane 1-Hydroxymethyl-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Isopropoxymethyl-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Isopropyl-1H-benzotriazole-5-carboxylic acid 1-isopropyl-4-(4-(3-((methylamino)methyl)-4-(4-(methylthio)phenoxy)phenyl)but-3-ynyl)piperazin-2-one 1-Isopropyl-5-Methoxytryptamine 1-Isopropyl-5-Methyltryptamine 1-Isopropyl-N-[[1-(2-morpholin-4-ylethyl]-4-piperidinyl]methyl]- 1H-indazole-3-carboxamide 1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide 1-Isopropyl-N-[[1-(2-pyridin-2-ylethyl)-4-piperidinyl]methyl]-1Hindazole-3-carboxamide 1-Isopropyl-N-[[1-[2-(4-hydroxyphenyl)ethyl]-4-piperidinyl]- methyl]-1H-indazole-3-carboxamide 1-Isopropyl-N-[[1-[2-(4-nitrophenyl)ethyl]-4-piperidinyl]methyl]- 1H-indazole-3-carboxamide 1-Isopropyl-N-[[1-[2-[(methylsulfonyl)amino]ethyl]-4- piperidinyl]methyl]-1H-indazole-3-carboxamide 1-Isopropyl-N-[[1-[3-(methylamino)-3-oxo-1-propyl]-4- piperidinyl]methyl]-1H-indazole-3-carboxamide 1-Isopropyltryptamine 1-Me-Tet-AMPA 1-Methoxy-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1-Methoxy-1,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene 1-Methoxy-4-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.2.0*2,6*]undec-8-ene-3,5-dione 1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-Methyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-10-ol 1-Methyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol 1-Methyl-2-(2,4,5-trimethoxy-phenyl)-ethylamine 1-Methyl-2-oxoado 1-methyl-2-phenylethylamine 1-Methyl-2-thiazol-4-yl-1H-benzoimidazol 1-Methyl-3-phenyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1-Methyl-4-(3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propyl)-1,4- diazepane 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepane TFA 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazine TFA 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazine TFA 1-Methyl-4-naphthalen-2-yl-piperidine-4-carbonitrile 1-Methyl-4-naphthalen-2-yl-piperidine-4-carboxylic Acid Ethyl Ester 1-methyl-4-phenylpyridinium ion 1-methyl-4-[1-(2-methylpropanesulfonyl)-4-(pyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate 1-methyl-4-[1-(2-methylpropanesulfonyl)-4-phenyl-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate 1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[2-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate 1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[3-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate 1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate 1-methyl-4-[4-(1-methyl-1H-pyrazol-4-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole 1-Methyl-5-(2-thioxo-1,2-dihydrospiro[3,1-benzoxazine-4,1'-cyclobutan]-6-yl)-1H-pyrrole-2-carbonitrile 1-methyl-5-(4-methyl-4-thien-3-yl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)- 1H-pyrrole-2-carbonitrile 1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole 1-methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g] quinoxalin-2(6H)-one HCl 1-Methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1-Methyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1-Methyl-9-(4-methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Methyl-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-methyl-N-(6-methylpyridin-2-yl)-1H-imidazole-2-carboxamide 1-methyl-N-(6-methylpyridin-2-yl)-1H-indole-2-carboxamide 1-methyl-N-(6-methylpyridin-2-yl)-1H-pyrrole-2-carboxamide 1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide 1-methyl-serotonin 1-Methylenoxime-9-(4-methylpiperazin-1-yl)pyrrolo- [2,1-b][1,3]benzothiazepine 1-Methylenoxime-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 1-Methylpsilocin 1-Methylpsilocybin 1-Methylxanthine 1-N-Allyl-7, 8-dihydro-14-hydroxymorphinone 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 1-N-methyl-1-N-[2-methyl-2-[[(1S)-1-phenylethyl]amino]propyl]cyclopropane-1,1-dicarboxamide 1-Naphthalenamine, 4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-, (1S-cis)- 1-Naphyrone 1-NP 1-oleoyl 2-acetyl glycerol 1-Oxo-1-[4-(2-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[4-(3-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[4-(4-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-furyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-oxazolyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-oxazolyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-pyrazinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-pyrazinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-10-phenyldecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-11-phenylundecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-2-phenylethane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-3-phenylpropane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-4-phenylbutane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-5-phenylpentane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-6-(phenyl)hex-5-yne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-6-heptyne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-6-phenylhexane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-7-(phenyl)hept-6-yne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-7-(trimethylsilyl)hept-6-yne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-8-phenyloctane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-decene 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-decyne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-octadecyne 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]-9-phenylnonane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]butane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]decane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]dodecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]ethane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]heptane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]hexadecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]hexane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]nonane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]octadecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]octane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]pentane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]propane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]tetradecane 1-Oxo-1-[5-(2-pyridyl)oxazol-2-yl]undecane 1-Oxo-1-[5-(2-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-pyrimidinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-thiazolyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-thiazolyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(2-thienyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(2-thienyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(3-pyridazinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(3-pyridazinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(3-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(3-thienyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(4-pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(4-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(4-pyrimidinyl)oxazol-2-yl]-9(Z)-octadecene 1-Oxo-1-[5-(5-pyrimidinyl)oxazol-2-yl]-7-phenylheptane 1-Oxo-1-[5-(phenyl)oxazol-2-yl]-7-phenylheptane 1-Pentyl-1H-benzotriazole-5-carboxylic acid 1-phenlsemicarbazide 1-phenyl-1-(piperidin-2-yl)propan-2-one 1-Phenyl-2-amino-athan (GERMAN) 1-phenyl-2-aminopropane 1-phenyl-2-aminopropane,(+) 1-phenyl-4-((1-phenyl-1H-1,2,3-triazol-4-yl)methyl)piperazine 1-phenyl-4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazine 1-Phenyl-4-(2-phenyl-3H-imidazol-4-ylmethyl)-piperazine 1-Phenyl-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 1-PP 1-propionyl-lysergic acid diethylamide 1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiaden-5-ol 1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene-5,6-diol 1-Propyl-1H-benzotriazole-5-carboxylic acid 1-Propyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-10-ol 1-Propyl-2,3,12,12a-tetrahydro-1H-7-oxa-1-aza-pleiaden-5-ol 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepane TFA 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazine TFA 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine TFA 1-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1-Propyl-8-(4-(4-(3-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Propyl-8-(4-(4-(4-trifluoromethylbenzyl)piperazine-1-sulfonyl)phenyl)-3,7-dihydropurine-2,6-dione 1-Propyl-8-{1-[3-(3-trifluoromethyl-phenyl)-prop-2-ynyl]-1H-pyrazol-4-yl}-3, 7-dihydro-purine-2, 6-dione 1-t-Butyl-1H-benzotriazole-5-carboxylic acid 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 1-thiocarbamoyl-3,5-di-(4-methylphenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydropyrazole 1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(4-methylphenyl)-5-(furan-2-yl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-chlorophenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-methylphenyl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(furan-2-yl)-4,5-dihydropyrazole 1-thiocarbamoyl-3-(thiopen-2-yl)-5-(thiopen-2-yl)-4,5-dihydropyrazole 1-TMT 1-[(1-(4-Chlorophenyl)-1H-1,2,3-triazol-4-yl)methyl]-4-phenylpiperazine 1-[(1-(4-Chlorophenyl)-1H-pyrazol-4-yl)methyl]-4-phenylpiperazine 1-[(1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazol-4-yl)carbonyl]-THIQ 1-[(1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazol-4-yl)carbonyl]piperidin-4-ol 1-[(1-(4-Fluorophenyl)-1H-pyrazol-4-yl)methyl]-4-phenylpiperazine 1-[(2,4-dichlorophenyl)(phenyl)methyl]-4-(piperidin-1-ylcarbonyl)piperazine 1-[(2,6-dichlorophenyl)methyl]-4-[[(2S)-oxolan-2-yl]methyl]piperazine 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-methyl-N-[[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl]methanamine 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine 1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-methylmethanamine 1-[(3-fluorophenyl)methyl]-4-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]piperazine 1-[(3-methylpyridin-2-yl)methyl]-4-[(2-phenyl-1H-imidazol-5-yl)methyl]piperazine 1-[(E)-4-trityloxy-2-butenyl]uracil 1-[(Z)-4-Trityloxy-2-butenyl]uracil 1-[1-(2,5-Dimethoxybenzenesulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(2-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol(HCl) 1-[1-(3-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol (HCl) 1-[1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(3-Fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(3-Fluorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(3-Methoxyphenyl)-2-(4-methyl-1-piperazinyl)ethyl]cyclohexanol Dihydrochloride 1-[1-(3-Methoxyphenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(4-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol (HCl) 1-[1-(4-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(4-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(4-Fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride 1-[1-(4-Fluorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(4-Methoxyphenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride 1-[1-(5-Bromo-2-methoxybenzenesulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(5-Dimethylaminonaphthalene-1-sulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(Benzo[b]thiophene-3-sulfonyl)-piperidin-4-yl]-8-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(Naphthalene-1-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[1-(Quinoline-8-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 1-[2-(3-fluorophenoxy)ethyl]-N-(5-methyl-1,2-oxazol-3-yl)piperidine-4-carboxamide 1-[2-(3-methyl-1,2-oxazol-5-yl)ethyl]piperidin-4-yl}(thiophen-2-yl)methanol 1-[2-(4-Benzoyl-1-piperazinyl)ethyl]-2-imidazolidinone 1-[2-(4-Benzyl-1-piperazinyl)ethyl]-2-imidazolidinone 1-[2-(Azidomethyl)-4-(trityloxy)butyl]uracil 1-[2-(Benzoyloxyethoxy)methyl]uracil 1-[2-(diethylamino)quinazolin-4-yl]-3-phenylurea 1-[2-(Hydroxymethyl)-4-(trityloxy)butyl]uracil 1-[2-(Trityloxy)ethoxymethyl]uracil 1-[2-Dimethylamino-1-(3-methoxy-phenyl)-ethyl]-cyclohexanol (HCl) 1-[2-Dimethylamino-1-(3-trifluoromethyl-phenyl)-ethyl]-cyclohexanol (HCl) 1-[2-[4-(1-Indanyl)-1-piperazinyl]ethyl]-2-imidazolidinone 1-[2-[[(1R)-1-(furan-2-yl)ethyl]-methylamino]acetyl]piperidine-4-carboxamide 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride 1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride 1-[3-(Methylsulfonyl)phenyl]-4-propylpiperazine 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1-[3-[N-(4-Bromobenzyl)-N-(pyrid-2-yl)amino]propyl]-3-[3-(1H-imidazol-4-yl)propyl]thiourea Dihydrochloride 1-[4-(2,5-dimethylthiophen-3-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Hydrobromide 1-[4-(2-chlorophenoxy)butyl]piperazine 1-[4-(2-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(2-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(2-Pyridyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(2-Pyrimidyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-(4-phenyl-1-piperazinyl)-1-propanone 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone 1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(1H-indol-3-yl)ethan-1-one 1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1- one 1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl) ethan-1-one 1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(6-fluoro-1H-indol-3-yl)ethan-1- one 1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-3-(1H-indol-3-yl)propan-1-one 1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-4-(1H-indol-3-yl)butan-1-one 1-[4-(4-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(4-ethylphenyl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Fumarate 1-[4-(4-methoxyphenyl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Fumarate 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 1-[4-(4-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone 1-[4-(4-methylcyclohexyl)butyl]alpha,alpha-diphenyl-4-piperdinemethanol 1-[4-(4-methylphenyl)butyl]-alpha,alpha-diphenyl-4-piperdine-methanol 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 1-[4-(dimethyl-1,2-oxazol-4-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Hydrobromide 1-[4-(tert-Butoxycarbonylamino)-3-(trityloxymethyl)butyl]-uracil 1-[4-Acetyloxy-3-(tritylaminomethyl)butyl]uracil 1-[4-Hydroxy-2-(trityloxymethyl)butyl]uracil 1-[4-Hydroxy-3-(tritylaminomethyl)butyl]uracil 1-[5-(1-Methylimidazol-2-yl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(1-Methylpyrrol-2-yl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(2-Furyl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(2-Pyridyl)oxazol-2-yl]-7-phenylheptane 1-[5-(2-Pyridyl)oxazol-2-yl]-9(Z)-octadecene 1-[5-(2-Pyrimidinyl)oxazol-2-yl]-7-phenylheptan-1-ol 1-[5-(3-Furyl)oxazol-2-yl]-1-oxo-9(Z)-octadecene 1-[5-(3-Pyridazinyl)oxazol-2-yl]-7-phenylheptan-1-ol 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-phenylpiperidin-4-amine 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime 1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride 1-[N2-[3,4-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]4-(4-pyridinyl)piperazine 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidal-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)pi... 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)... 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-4-phenyl-2(2H)-oxoimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyrid... 1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperazinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluor... 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)pi... 1-[N2-[3,5-Dibromo-N-[[4-[2(3H)-oxobenzoxazol-3-yl]-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis... 1-[N2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 1-[N2-[4-amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl-4-(4-pyridinyl)piperazine 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-(4-pyridinyl)piperazine 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-phenyl-piperazine Hydrobromide 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-piperazine Dihydrobromide 1-[N2-[N-[[4-[N-(Aminocarbonyl)phenylamino]-1-piperidinyl]carbonyl]-3,5-dibromo-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine... 1-[N2-[N[[4-[N-(Aminocarbonyl)phenylamino]-1-piperidinyl]carbonyl]-3,5-dibromo-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine ... 1-[[2,3-Dihydro-7-(3-pyridyl)benzofuran-5-yl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[2-Chloro-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[2-Fluoro-5-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[3-Fluoro-5-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid 1-[[4-Chloro-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[4-Chloro-3-(4-methyl-3pyridyl)phenyl]carbamoyl-5-methoxy-6-trifluoromethylindoline 1-[[4-Methoxy-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[4-tert-Butyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-(2,6-Difluorophenyl)-3-pyridyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-(3,5-Difluorophenyl)-3-pyridyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-Bromo-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-[[5-Ethyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 1-{1,4-Dioxa-8-thiaspiro[4.5]decan-2-ylmethyl}-4-(2-methoxyphenyl)piperazine 1-{2-(3-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride 1-{2-(3-Methylpiperazin-1-yl)-1-[3-(trifluoromethyl)phenyl]ethyl}cyclohexanol Dihydrocholoride 1-{2-(4-Methylpiperazin-1-yl)-1-[4-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride 1-{2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride 1-{2-Piperazin-1-yl-1-[3-(trifluoromethyl)phenyl]ethyl}cyclohexanol Dihydrochloride 1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride 1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride 1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{2-[4-(7-Chloro-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepin-9-yl)-1-piperazinyl]ethyl}-2-imidazolidinone 1-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-4-(3-phenyl-propyl)-piperazine 1-{3-[4-(1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{3-[4-(1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dion 1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion 1-{4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[3-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyr-rolidine-2,5-dione 1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione 1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion 1-{4-[4-(benzyloxy)phenyl]-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-methylpiperazine Fumarate 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid 1-{6-amino-4-thia-2-azatricyclo[7.3.0.0³,⁷]dodeca-1(9),2,5,7-tetraen-5-yl}ethan-1-one 1-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one 1-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{6-[4-(2-pyrimidinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1-{[1-(4-Chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methoxyphenyl)piperazine 1-{[1-(4-Fluorophenyl)-1H-1,2,3-triazol-4-yl]methyl}-4-phenylpiperazine 1-{[1-(4-Nitrophenyl)-1H-1,2,3-triazol-4-yl]methyl}-4-phenylpiperazine 1-{[5-(4-Chloro-3-methylphenyl)-1-(4-methylbenzyl)-1Hpyrrol-3-yl]methyl}-4-(3,4-dichlorophenyl)piperazine 1-{[5-(4-Chloro-3-methylphenyl)-1-(4-methylbenzyl)-1Hpyrrol-3-yl]methyl}-4-(4-chlorophenyl)piperazine 10 10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 10-(1-ethyl-1,2,3,6-tetrahydro-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin 10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-Butenyl)-11-hydroxy-N-propylnoraporphine 10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(2-Methylallyl)-11-hydroxy-N-propylnoraporphine 10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(3-Hydroxypropoxy)-3,9-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 10-(4-(5-(4-fluorobenzamido)-1H-indol-3-yl)piperidin-1-yl)decanoic acid 10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 10-(4-methylpiperazino)-5H-dibenz[b,f]oxepin 10-(Cyclopropylmethoxy)-3,9-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 10-(Hexyloxy)-3,9-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 10-Allyl-11-hydroxy-N-methylaporphine 10-Allyl-11-hydroxy-N-propylnoraporphine 10-amino-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-1-o 10-Butoxy-3,9-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 10-Ethoxy-3,9-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) 10-[1,2,3,6-tetrahydro-1(2-propenyl)-4-pyridinyl]-5H-dibenzo[a,d]cycloheptene 10-[1-methyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin 103 104 105 108 109 10a-homo-9,11-ethano PGH2 10alpha,11alpha-oxido PGA2 10S-hydroxylobel-7-ene 11 11(S)-Cyclohexyl-N-[1-[2-[[2-[[2-(dimethylamino)-2-oxo-1(S)-phenylethyl]amino]-2-oxoethyl]amino]-1,2-dioxo-ethyl]butyl]-9,12-... 11(S)-Cyclohexyl-N-[1-[2-[[2-[[2-(methylamino)-2-oxo-1(S)-phenylethyl]amino]-2-oxoethyl]amino]-1,2-dioxo-ethyl]butyl]-9,12-di... 11,9-epoxymethano PGH2 11-(1-Methylallyloxy)-N-methylaporphine 11-(2-Butynyloxy)-N-propylnoraporphine 11-(2-Hexyl-5-hydroxyphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(2-Hexyl-5-hydroxyphenoxy)undecanoic Acid (4-Hydroxyphenyl)amide 11-(2-Hexyl-5-hydroxyphenoxy)undecanoic Acid Cyclopropylamide 11-(3-Hydroxy-4-hexylphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(3-Hydroxy-4-hexylphenoxy)undecanoic Acid (4-Hydroxyphenyl)amide 11-(3-Hydroxy-4-hexylphenoxy)undecanoic Acid Cyclopropylamide 11-(3-Hydroxy-5-pentylphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(3-Hydroxy-5-pentylphenoxy)undecanoic Acid (4-Hydroxyphenyl)amide 11-(3-Hydroxy-5-pentylphenoxy)undecanoic Acid Cyclopropylamide 11-(3-Hydroxyphenoxy)undecanoic Acid (2-Hydroxyethyl)amide 11-(3-Hydroxyphenoxy)undecanoic Acid (4-Hydroxy-phenyl)amide 11-(3-Hydroxyphenoxy)undecanoic Acid Cyclopropilamide 11-(4-Methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 11-(Piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 11-Allyloxy-N-methylaporphine 11-Amino-9,10-dihydro-9,10-ethanoanthracene Oxalate 11-Hydroxy-N-propylnoraporphine 11-Propargyloxy-N-methylaporphine 11-Propargyloxy-N-propylnoraporphine 11-valeryloxynoraporphine 110 111 112 113 116 117 118 119 11f 11Z,14Z,17Z-eicosatrienoic acid 12 12'-hydroxy-2',5'-diisopropyl-3',6',18-trioxoergotaman 12(R)-HETE 12-Deoxyphorbol 13-phenylacetate 12-METHOXYIBOGAMINE 12-oxo-LTB4 120 121 122 1229U91 124 125I-NCQ 298 127 128 12a 12b 12c 13 13,14,15,16-Tetrahydrosalvinorin A 130 134 136 137 138 13a 13b 13c 13d 13e 14 14-Benzyloxymetopon 14-ethoxy-3-hydroxy-5-methyl- 17-(2-phenylethyl)morphinan-6-one 14-Hydroxydihydromorphinone 14-methoxymetopon 14-O-(1-naphthylmethyl)oxymorphone 14-O-(2,6-dichlorobenzyloxy)oxymorphone 14-O-Allyloxymorphone 14-O-Benzyloxymorphone 14-O-methyloxymorphone 14-O-phenylpropylnaltrexone 14-phenylpropoxymetopon 14a 14b 14beta-(2'-chlorocinnamoylamino)-7,8-dihydromorphinone 14beta-(p-chlorocinnamoylamino)-7,8-dihydrocodeinone 14Beta-(p-nitrocinnamoylamino)-7,8-dihydrocodeinone 14c 14d 14e 14f 14g 14h 14i 14j 14k 14l 15 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one 15-(2-hydroxyethyl)-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one 15-ethyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl PGF2alpha 15-methyl-N-(1,3,4-thiadiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl-N-(4-methyl-1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15-methyl-N-(5-methyl-1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 15a 15b 15c 15d 15e 15f 15g 15h 16 16,16-dimethyl PGF2alpha 16-(2-Hexyl-5-hydroxyphenoxy)hexadecanoic Acid (4-Hydroxyphenyl)amide 16-(2-Hexyl-5-hydroxyphenoxy)hexadecanoic Acid Cyclopropylamide 16-(3-Hydroxy-4-hexylphenoxy)hexadecanoic Acid (4-Hydroxyphenyl)amide 16-(3-Hydroxy-5-pentylphenoxy)hexadecanoic Acid (2-Hydroxyethyl)amide 16-(3-Hydroxy-5-pentylphenoxy)hexadecanoic Acid (4-Hydroxyphenyl)amide 16-(3-Hydroxy-5-pentylphenoxy)hexadecanoic Acid Cyclopropylamide 16-(3-Hydroxyphenoxy)hexadecanoic Acid (2-Hydroxy-ethyl)amide 16-(3-Hydroxyphenoxy)hexadecanoic Acid (4-Hydroxy-phenyl)amide 16-(3-Hydroxyphenoxy)hexadecanoic Acid Cyclopropylamide 16-epi-Leoleorin F (9,13:15,16-diepoxylabdane-6β,16α-diol 16a 16b 16c 17 17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate 17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(2',3',4',6'-tetra-O-benzyl-D-glucopyranosyl)acetamido]morp... 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3'-methoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(D-glucopyranosyl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(thiophen-2'-yl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzylacetamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(cinnamoylacetamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(D-glucopyranosyl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)phenylacetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-nitro)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-amino)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carboxy)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-methoxy)benzylacetamido]morphinan ( 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-tert-butoxycarbonylamino)benzamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(thiophen-2'-yl)acetamido]morphinan 17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-[(3'-dimethylamino)benzamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-bromo)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-iodo)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-methyl)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-t-butyl)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-epoxy-6beta-[(4'-trimethylfluoro)benzamido]morphinan-oxalate 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-naphthalyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(2'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-isoquinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(3'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6alpha-[(4'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(2'-naphthalyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(2'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-isoquinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(3'-quinolyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5r-epoxy-6beta-[(4'-pyridyl)acetamido]morphinan 17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan 17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphina... 17-Cyclopropylmethyl-6,7-didehydro-4,5-alpha-epoxy-5'-guanidinyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-4-chlorobenzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphi... 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-4-nitrobenzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphin... 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-(N'-benzyl)guanidinylethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 17-Cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-5'-guanidinylmethyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 17-deoxysalvinorin A 17-Hydroxy-13-methyl-10-(4-methyl-benzyl)-17-prop-1-ynyl-1,2,6,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-cyclopenta[a]phen... 17a 17b 17beta-Estradiol 18 18-MC 18F-Mefway 19 19a 19b 19c 1alpha H, 3 alpha, 5 alpha H-tropan-3-yl-3,5dichlorobenzoate 1b 1c 1d 1DMe-Y8Fa 1e 1H-Benzimidazol-2-yl-thiourea 1H-indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide 1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 1H-Indole-3-carboxylic acid [5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]amide 1H-indole-3-carboxylic acid [6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]amide 1H-indole-3-carboxylic acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide 1H-indole-3-carboxylic acid [8-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)octyl]amide 1H-Methylindole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide 1R)-1-(3,4-dimethylphenyl)-2-[4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl]ethanol 1R,3R-ACPD 1R,3S-ACPD 1S, 3R-ACPD 1S, 3S-ACPD 1S,2R,3S,4R,5S)-2,3-Dihydroxy-N-methyl-4-(4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-1-carboxamide 1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbox... 2 2 (BCCT) 2',3'-Dihydro-(3R)-(4-Phenyl-1H-imidazol-2-yl)spiro[Beta-carboline-1,2'-1H-indene] 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 2'-Deoxy-N6-methylado 2'-Deoxyadenosine 2'-O-Methyladenosine 2'-Oxopyrrolidino-1-pyrrolidino-4-butyne 2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one 2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone 2,2,6,6-Tetramethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine 2,2,6,6-Tetramethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 2,2,6,6-Tetramethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine 2,2,6,6-Tetramethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 2,2-Dimethyl-1-(oxazol-2-yl)-1-oxo-9(Z)-octadecene 2,2-Dimethyl-propionic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-(2,2-dimethyl-propionyloxymethyl)-propyl Ester 2,2-Dimethyl-propionic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phosphono-oxymethyl-propyl Ester, Ammonium Salt 2,2-Dimethyl-propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3... 2,2-Diphenyl-ethylamine 2,2-diphenylethylamine 2,3,4,5-Tetrahydro-1H-2-benzazepine 2,3,4,5-tetrahydro-1H-[1,4]diazepinol[1,7-a]indole 2,3,4,5-Tetrahydro-5H-1,4-benzothiazepine 2,3,4,5-Tetrahydro-5H-1,4-benzoxazepine 2,3,7,11b-Tetrahydrodibenzo[d,e,h]isoquinoline Oxalate 2,3-dichloro-alpha-methyl benzylamine 2,3-Difluoro-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzamide 2,3-Dihydro-5,6-dimethoxy-N-(2-phenylethyl)-N-propyl-1H-inden-2-amine 2,3-Dihydro-5,6-dimethoxy-N-(3-phenylpropyl)-N-propyl-1H-inden-2-amine 2,3-Dihydro-5,6-dimethoxy-N-propyl-N-[2-[4-(trifluoromethyl)phenyl]ethyl]-1H-inden-2-amine 2,3-Dihydro-5,6-dimethoxy-N-[2-(4-methoxyphenyl)ethyl]-N-propyl-1H-inden-2-amine 2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-1H-benzimidazole-1-carboxamide 2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-6-methoxy-1H-benzimidazole-1-carboxylate 2,3-dihydroamentoflavone 2,3-dihydrohinokiflavone 2,3-Dihydroisoindole 2,3-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 2,3-DIMETHYLPHENYLPIPERAZINE 2,3-O-(4 benzoylbenzoyl)-ATP 2,4,5-TMA 2,4,5-Trimethoxamphetamine 2,4,5-trimethoxyamphetamine 2,4,9-trimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione 2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione 2,4-Diaminobutyric acid 2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine 2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2,4-dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione 2,4-DIMETHYLPHENYLPIPERAZINE 2,4-Diphenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 2,4-Diphenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 2,4-DMA 2,4‐dichloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline 2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine 2,5,7-Trimethyl-3-[4-(phenylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine 2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione 2,5-bis(GSyl)-alpha-MethylDopamine 2,5-Difluoro-N-{1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 2,5-Difluoro-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 2,5-Dihydro-6-methoxy-2-(2-methoxyphenyl)-5-[2-(4-morpholinyl)ethyl]-1H-pyrido[4,3-b]indol-1-one 2,5-Dihydro-6-methoxy-5-[2-(4-morpholinyl)ethyl]-2-[(1S,2S)-1,33-trimethylbicyclo[2.2.1]heptan-2-yl]-1H-pyrido[4,3-b]indol-1-... 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine 2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine 2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine 2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine 2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine 2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine 2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine 2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine 2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine 2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine 2,5-dimethoxy-4-allylthiophenethylamine 2,5-dimethoxy-4-benzylthiophenethylamine 2,5-dimethoxy-4-benzylthiophenethylamine, 2,5-Dimethoxy-4-bromoamphetamine 2,5-Dimethoxy-4-bromoamphetamine, benzyloxy 2,5-Dimethoxy-4-bromoamphetamine, R(-) 2,5-Dimethoxy-4-bromoamphetamine, S(+) 2,5-Dimethoxy-4-ethoxyamphetamine 2,5-dimethoxy-4-ethoxyphenethylamine 2,5-Dimethoxy-4-ethyl-amphetamine,(+/-) 2,5-DIMETHOXY-4-ETHYLAMPHETAMINE 2,5-DIMETHOXY-4-ETHYLAMPHETAMINE, (-) 2,5-DIMETHOXY-4-IODOAMPHETAMINE , (+) 2,5-DIMETHOXY-4-IODOAMPHETAMINE , (-) 2,5-dimethoxy-4-isobutylthiophenethylamine 2,5-dimethoxy-4-isopropoxyamphetamine 2,5-dimethoxy-4-isopropylthiophenethylamine 2,5-dimethoxy-4-methallyloxyamphetamine 2,5-dimethoxy-4-methallyloxyphenethylamine 2,5-Dimethoxy-4-methylamphetamine 2,5-Dimethoxy-4-methylamphetamine, R(-) 2,5-dimethoxy-4-methylphenylisopropylamine 2,5-dimethoxy-4-methylthiophenethylamine 2,5-dimethoxy-4-n-butylthiophenethylamine 2,5-dimethoxy-4-propylthiophenethylamine 2,5-Dimethoxy-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide 2,5-dimethoxyphenethylamin 2,5-dimethoxyphenethylamine 2,5-dimethyoxy-4-iodophenylisopropylamine 2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine 2,6-bis(2-fluorophenyl)pyrimidin-4-amine 2,6-bis(2-methoxyphenyl)pyrimidin-4-amine 2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine 2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine 2,6-bis(4-acetylphenyl)pyrimidin-4-amine 2,6-bis(4-chlorophenyl)pyrimidin-4-amine 2,6-bis(4-fluorophenyl)pyrimidin-4-amine 2,6-bis(4-methoxyphenyl)pyrimidin-4-amine 2,6-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}pyridine 2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine 2,6-di(furan-2-yl)pyrimidin-4-amine 2,6-di(furan-3-yl)pyrimidin-4-amine 2,6-di(thiophen-2-yl)pyrimidin-4-amine 2,6-di(thiophen-3-yl)pyrimidin-4-amine 2,6-di-p-tolylpyrimidin-4-amine 2,6-Difluorobenzoic Acid 2-(2,6-difluorobenzoyloxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester 2,6-Dimethyl-4-(5-methyl-3-phenyl-isoxazol-4-yl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 2,6-dimethyl-4-(5-methyl-3-phenyl-isoxazol-4-yl)-pyridine-3,5-dicarboxylic acid diethyl ester 2,6-diphenyl-8-propan-2-yl-7H-purine 2,6-diphenylpyrimidin-4-amine 2,6-distyrylpyrimidin-4-amine 2,8-Dimethyl-3-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl... 2,N,N-TMT 2,N,N-TRIMETHYLTRYPTAMINE 2-((2,5-Dimethoxy-4-(trifluoromethyl)phenethylamino)methyl)phenol hydrochloride 2-((2,5-Dimethoxy-4-methylphenethylamino)methyl)phenol hydrochloride 2-((2,5-Dimethoxy-4-propylphenethylamino)methyl)phenol hydrochloride 2-((2-(2-fluorophenyl)-7-methoxybenzofuran-4-yl)methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline 2-((2-(furan-2-yl)-7-methoxybenzofuran-4-yl)methyl)-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline 2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one 2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 2-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 2-((3R)-3-Methyl-4-{[(2S)-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}pipera-zin-1-yl)quinoline-6-carbonitril... 2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethanamine 2-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 2-((4-Ethyl-2,5-dimethoxyphenethylamino)methyl)phenol hydrochloride 2-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 2-((5-((3-Chlorophenoxy)methyl)isoxazol-3-yl)oxy)-N-(cyclo-propylmethyl)-N-methylethan-1-amine Hydrochloride 2-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hy-drochloride 2-((5-Methoxy-1H-indol-3-yl)methyl)-5-methyloxazole 2-((5-Methoxy-1H-indol-3-yl)methyl)5-1,3,4-oxadiazole 2-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)thio) benzo[d]oxazole 2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)acetic acid 2-(-3-pyridinyl)-1-azabicyclo[2.2.2]octane 2-(1,3-benzodioxol-5-yl)guanidine 2-(1-(3,5-diethoxy-4-(1H-pyrrol-1-yl)benzyl)piperidin-4-ylamino)-N,N-dimethylbenzo[d]oxazole-5-sulfonamide 2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-carboxamide 2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-carboxylic acid 2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)-N,N-dimethylbenzo[d]oxazole-5-sulfonamide 2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide 2-(1-(4-(4-chlorophenyl)-2,2,4-trimethyl-3,4-dihydroquinolin-1(2H)-yl)-1-oxopropan-2-yl)hexahydro-1H-isoindole-1,3(2H)-dione 2-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-sulfonamide 2-(1-(4-chloro-3,5-diethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-5-carboxylic acid 2-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-carboxylic acid 2-(1-Methyl-2-phenylethyl)-4,5-dihydro-1H-imidazole Oxalate 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethanone 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone O-benzyloxime 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone O-methyloxime 2-(1H-benzimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxyphenyl)ethanone oxime 2-(1H-Benzoimidazol-2-yl)-phenol 2-(1H-Benzoimidazol-2-yl)-pyridin-3-ol 2-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 2-(1H-Indol-3-yl)-2-oxo-N-(1-phenyl-ethyl)-acetamide 2-(1H-indol-3-yl)-N,N -dimethylethanamine 2-(1H-Indol-3-yl)-N-(4-methoxy-benzyl)-2-oxo-acetamide 2-(1H-Indol-3-yl)-N-(4-nitro-benzyl)-2-oxo-acetamide 2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 2-(2,4-Dichlorophenyl)-1-(4-fluorophenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 2-(2,4-Dichlorophenyl)-1-(4-methoxyphenyl)-5-methyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 2-(2,4-Dichlorophenyl)-4-methyl-6-(1-propylbutyl)-2,6,7,8-tetrahydro-1,2,3,6-tetraazaacenaphthylene 2-(2,4-Dichlorophenyl)-5-methyl-N-(piperidin-1-yl)-1-(4-(trifluoromethyl)phenyl)-1H-imidazole-4-carbox-amide 2-(2,5- dimethoxy-4-nitro)ethanamine 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(2,5-dimethoxy-4-methyl) ethanamine 2-(2,5-dimethoxy-4-methyl) ethanamine-(4-chloro-2,5-dimethoxy)ethanamine 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 2-(2,5-dimethoxy-4-nitrophenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 2-(2,5-dimethoxy-4-propylphenyl)ethanamine; 2-(2,5-Dimethoxy-phenyl)-1-methyl-ethylamine 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(2,6-bis(2-(diethylamino)ethoxy)phenoxy)-N,N-diethylethanamine 2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline 2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride 2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one, 2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline 2-(2-(4-(2,3-Dichlorophenyl)piperazin-1-yl)ethyl)-6-methoxyisoindolin-1-one 2-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2-azaspiro[4.5]decane-1,3-dione 2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole 2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4- tetrahydroisoquinoline hydrochloride 2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 2-(2-(5-Methoxy-1H-indol-3-yl)ehtyl)-1,3,4-oxadiazole 2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyl-1,3,4-oxadiazole 2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyloxazole 2-(2-benzylphenyl)-ethylamine 2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-isopropyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-N-methyl-1H-imidazole-4-carboxamide 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-chlorophenyl)-3-(4-chlorophenyl)-5-methyl-6-(2,2,2-trifluoroethyl)-2H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2,2,2-trifluoroethyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoropropyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-c]pyridine hydrochloride 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2,2-difluoropropyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-(2-methoxy-2-methylpropyl)-5,6-dihydro-2H-pyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-cyclopentyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-ethyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-isobutyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-6-isopropyl-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohexyl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-(pyridin-3-yl)-1H-imidazole-4-carboxamide 2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imidazole-4-carboxamide 2-(2-Dimethylaminomethyl-phenylsulfanyl)-5-methyl-phenylamine 2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 2-(2-fluorophenyl)-1-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]ethanone 2-(2-methoxyphenyl)-8-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-2,8-diazaspiro[4.5]decane 2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 2-(2-phenylethenyl)-3,1-benzoxazin-4-one  2-(2-Phenylpropyl)-4,5-dihydro-1H-imidazole Maleate 2-(2-Thiazolyl)ethanamine 2-(2-thiazolyl)ethylamine (TEA) 2-(2-{4-[2-(Mesityloxy)ethyl]piperazin-1-yl}ethoxy)ethanol dihydrochloride 2-(3,4-Dichloro-phenyl)-N-methyl-N-(2-pyrrolidin-1-yl-cyclohexyl)-acetamide 2-(3,4-dihydro-1H-isoquinolin-2-yl)-N-[3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propyl]acetamide 2-(3,4-dimethoxyphenyl)quinazolin-4(3H)-one 2-(3,5-Difluorophenyl)-4-(3-fluorophenylethynyl)thiazole 2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(4-chloro-2-fluorophenyl)- amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-Drib... 2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(±)-endo-norbornyl-9H-(5- (3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl... 2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(R)-3-tetrahydrofuranyl-9H- (5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranos... 2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine 2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline 2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)acetamide 2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-isopropoxyphenyl)piperazin-1-yl)ethyl)acetamide 2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)acetamide 2-(3-(2-(cyclopropylamino)pyrimidin-4-yl)piperidin-1-yl)-1-(1H-indol-3-yl)ethanone 2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide 2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-5,6-dimethoxyisoindolin-1-one 2-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propyl)-6-methoxyisoindolin-1-one 2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole 2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride 2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 2-(3-Biphenylylethynyl)-6-methylpyridine 2-(3-Bromophenyl)histamine 2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide 2-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate 2-(3-Chlorophenyl)histamine 2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 2-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 2-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine 2-(3-Hydroxy-2-methoxybenzyl)-6-methoxy-1-methyl-1,2,3,4-tetrahydroisoquinolin-7-ol 2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate 2-(3-Iodophenyl)histamine 2-(3-methoxyphenoxy)ethanimidamide 2-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate 2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 2-(3-Methoxyphenyl)-N-methylethan-1-amine 2-(3-methoxyphenyl)ethanimidamide 2-(3-pyridinyl)-2,5-diazabicyclo[2.2.2]octane 2-(4'-Methylaminophenyl)Benzothiazole 2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide 2-(4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxy-5-fluorophenoxy)ethanol 2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)ac... 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)ac... 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetam... 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamid... 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)ace... 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl... 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)pr... 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acet... 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)a... 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetami... 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamid... 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)ac... 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-y... 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-... 2-(4-(2-(benzylamino)ethyl)phenoxy)isonicotinamide 2-(4-(2-(benzylamino)ethyl)phenoxy)nicotinamide 2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione 2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline1,3-dione 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 2-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)phenol 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine 2-(4-(3-(tert-butylamino)-2-hydroxypropoxy)-1H-indol-3-yl)acetamide 2-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one 2-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one 2-(4-(4-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)piperazin-1-yl)butyl)-6-(1H-imidazol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)piperazin-1-yl)butyl)-6-(1H-indol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)-4-oxobutyl)-6-(1H-imidazol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)butyl)-6-(1H-imidazol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-ethoxyphenyl)piperazin-1-yl)butyl)-6-(1H-indol-1-yl)pyridazin-3(2H)-one 2-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one 2-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one 2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole 2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole 2-(4-(4-(Bis(4-fluorophenyl)methyl)piperazin-1-yl)butyl) benzo[d]thiazole dihydrochloride 2-(4-(4-(Pyridin-2-yl)piperazin-1-yl)butyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-1-one 2-(4-(4-(Pyridin-2-yl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one 2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride 2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride 2-(4-(5-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3- yl)propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)phenyl)oxazole 2-(4-(5-(aminomethyl)pyridin-2-yloxy)phenyl)-N-benzylethanamine 2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 2-(4-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- butyl)isoindoline-1,3-dione 2-(4-(benzyloxy)phenyl)-3-(2-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta... 2-(4-(benzyloxy)phenyl)-3-(8-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta... 2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride 2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione 2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione 2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline1,3-dione 2-(4-([1,1'-biphenyl]-2-yl)piperazin-1-yl)-1-(3,4-dichlorophenyl)ethanol hydrochloride 2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate 2-(4-bromo-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamin 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(4-bromo-2,5-dimethoxyphenyl)ethanamine 2-(4-Bromobenzyl)-3-{4-[2-(4-(dimethylamino)phenyl)vinyl]phenoxy}propan-1-ol 2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-bromophenyl)-2-phenylethanamine 2-(4-bromophenyl)-4H-3,1-benzoxazin-4-one 2-(4-bromophenyl)ethylamine 2-(4-bromophenyl)quinazolin-4(3H)-one 2-(4-Chloro-1,3-dihydro-isoindol-2-ylamino)-4,5-dihydro-3H-imidazol-1-ium 2-(4-chloro-2,5-dimethoxy)ethanamine 2-(4-chloro-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one 2-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-chlorophenyl)-3,1-benzoxazin-4-one 2-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 2-(4-Chlorophenyl)-5-phenyl-4-isoxazolin-3-one 2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine 2-(4-chlorophenyl)quinazolin-4(3H)-one 2-(4-ethoxyphenyl)-3,1-benzoxazin-4-one 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(4-Fluoro-phenyl)-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-acetamide 2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide 2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide 2-(4-fluorophenyl)-3,1-benzoxazin-4-one 2-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 2-(4-Fluorophenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-(4-fluorophenyl)quinazolin-4(3H)-one 2-(4-Hexyl-2,5-dimethoxy-phenyl)-1-methyl-ethylamine : (Hydrochloride) 2-(4-hexylphenyl)-2-phenylethanamine 2-(4-hexylphenyl)ethanamine 2-(4-Hydroxyphenyl)-1-p-tolyl-3H-inden-5-ol 2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol 2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-Hydroxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-methoxyphenyl)-4H-3,1-benzoxazin-4-one 2-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 2-(4-Methoxyphenyl)ado (CV-1674) 2-(4-methoxyphenyl)quinazolin-4(3H)-one 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamin 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-methylphenyl)-3,1-benzoxazin-4-one  2-(4-methylphenyl)quinazolin-4(3H)-one 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(4-Nitro-phenyl)-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-acetamide 2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2-(4-{2-[2-(2,3,5-Trimethylphenoxy)ethoxy]ethyl}piperazin-1-yl)ethanol dihydrochloride 2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}-1,4-diazepan-1-yl)-quinoline-6-carbonitrile 2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile 2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)quino-line-6-carboxamide 2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,4-diol 2-(5-benzyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)-N-isopropylpropanamide 2-(5-Bromo-1H-indol-3-yl)-N,N-dimethylethanamine 2-(5-Bromo-1H-indol-3-yl)-N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]acetamide 2-(5-Bromo-7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethan-1-one 2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8atetrahydro-2H-phthalazin-1-one 2-(5-Chloro-1H-indol-3-yl)-N,N-dimethylethanamine 2-(5-fluoro-4-((R)-1-(3-fluorophenyl)ethoxy)pyrimidin-2-yl)-2,7-diazaspiro[4.4]nonane 2-(5-fluoro-4-((R)-1-(4-fluorophenyl)ethoxy)pyrimidin-2-yl)-2,7-diazaspiro[4.4]nonane 2-(5-Iodo-1H-indol-3-yl)-N,N-dimethylethanamine 2-(5-Nitro-1H-indol-3-yl)-2-oxo-N-(1-phenyl-ethyl)-acetamide 2-(5-{2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethoxy}-1H-indol-3-yl)-ethylamine 2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine 2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(4-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo[de] isoquinoline-1,3(2H)-dione 2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-[1,2,4] triazolo[4,3-a]pyridin-3(2H)-one 2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)–2H-naphtho [1,8-cd]isothiazole 1,1-dioxide 2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)isoindoline1,3-dione 2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(pyrimidin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide 2-(6-Bromo-3-pyridinyl)-N-ethyl-N-methylethanamine 2-(6-chloro-3-pyridinyl)-2,6-diazabicyclo[3.2.1]octane 2-(6-Chloro-3-pyridinyl)-N-ethyl-N-methylethanamine 2-(6-chloro-4-methylpyridin-3-yl)-7-azabicyclo[2.2.1]heptane 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-azabicyclo[2.2.1]heptane 2-(6-Chloro-5-phenyl-3-pyridinyl)-7-methyl-7-azabicyclo[2.2.1]heptane 2-(6-Chloro-pyridazin-3-yl)-2,5-diaza-bicyclo[2.2.1]heptane 2-(6-chloropyridin-3-yl)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene 2-(6-chloropyridin-3-yl)-2,7-diazaspiro[4.4]nonane 2-(6-Fluoro-5-phenyl-3-pyridinyl)-7-azabicyclo[2.2.1]heptane 2-(6-fluoro-5-phenylpyridin-3-yl)-1,2,3,4-tetrahydro-1,4-epiminonaphthalene 2-(6-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane 2-(6-Phenylpyridazin-4-yl)benzonitrile 2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,3-d]pyrimidin-4-ylthio)-N-(2-methoxyphenyl)propanamide 2-(8-Ethoxycarbonyl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin5-ylamino)-ethyl-amine hydrochloride 2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine 2-(9-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- 3,9-diazaspiro[5.5]undecan-3-yl)phenol 2-(Aminoethyl)-5-(2'-methoxy-5'-fluorophenethyl)tetrahydrofuran 2-(Aminomethyl)-4-hydroxy-3-methyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one hydrochloride 2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 2-(benzo[d][1,3]dioxol-5-yl)-N-(3,4-dimethoxyphenethyl)-N-phenethylethan-1-amine 2-(benzo[d][1,3]dioxol-5-yl)-N-benzyl-N-(3,4-dimethoxyphenethyl)ethan-1-amine 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide 2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide 2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate 2-(Dimethylamino)-2-oxoethyl 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate 2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-bi... 2-(dimethylamino)-6-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-3H-pyrrolo[2,3-d]pyrimidin-4(7H)-one 2-(Dimethylamino)tetralin 2-(furan-2-yl)-4H-3,1-benzoxazin-4-one 2-(furan-2-yl)-5-methyl-4-[[4-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]piperazin-1-yl]methyl]-1,3-oxazole 2-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 2-(furan-2-yl)quinazolin-4(3H)-one 2-(methylamino)-1-(4-methylphenyl)propan-1-one 2-(methylamino)-N6-(3-Iodobenzyl)adenosine-5'-N-methyluronamide 2-(methylthio)-N6-(3-Iodobenzyl)adenosine-5'-N-methyluronamide 2-(N,N-Diethylamino)-3'-chloropropiophenone 2-(N,N-Dimethylamino)-3'-chloropropiophenone 2-(N-(2-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-(4-chlorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-(4-fluorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-(4-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 2-(N-Cyclopentylamino)-3'-chloropropiophenone 2-(N-Cyclopropylamino)-3-chloropropiophenone 2-(N-dipropylamino)quinoline 2-(N-Isopropylamino)-3'-chloropropiophenone 2-(N-Methyl-N-tert-butylamino)-3'-chloropropiophenone 2-(N-Propylamino)-3'-chloropropiophenone 2-(N-tert-Butylamino)-1-(2'-thienyl)-1-propanone 2-(N-tert-Butylamino)-3',4'-dichloropropiophenone 2-(N-tert-Butylamino)-3'-bromopropiophenone 2-(N-tert-Butylamino)-3'-chloro-4'-methylpropiophenone 2-(N-tert-Butylamino)-3'-chlorobutyrophenone 2-(N-tert-Butylamino)-3'-chloroheptanophenone 2-(N-tert-Butylamino)-3'-chlorohexanophenone 2-(N-tert-Butylamino)-3'-chlorooctanophenone 2-(N-tert-Butylamino)-3'-chloropentanophenone 2-(N-tert-Butylamino)-3'-chlorophenyl-4-cyclohexylbutanophenone 2-(N-tert-Butylamino)-3'-chlorophenyl-4-methylpentanophenone 2-(N-tert-Butylamino)-3'-methylpropiophenone 2-(N-tert-Butylamino)-4'-bromo-5'-methylpropiophenone 2-(N-tert-Butylamino)-4'-bromopropiophenone 2-(N-tert-Butylamino)-4'-chloropropiophenone 2-(N-tert-Butylamino)-4'-methylpropiophenone 2-(N-tert-Butylamino)propiophenone 2-(Naphthalen-1-yloxalylamino)benzoic Acid 2-(Naphthalen-2-yloxalylamino)benzoic Acid 2-(Phenylamino)ado (CV-1808) 2-(pyridin-3-yl)-2,7-diazaspiro[4.4]nonane 2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 2-(tert-Butylamino)-3',4'-dichlorobutyrophenone 2-(tert-Butylamino)-3',4'-dichloropentanophenone 2-(tert-Butylamino)-3',5'-dichloropropiophenone 2-(tert-Butylamino)-3',5'-difluoropropiophenone 2-(tert-Butylamino)-3'-fluoropropiophenone 2-(tert-butylamino)-7-chloro-3,4-dihydronaphthalen-1(2H)-one 2-(thiophen-2-yl)-4H-3,1-benzoxazin-4-one 2-(thiophen-2-yl)quinazolin-4(3H)-one 2-(Trifluoromethanesulfonyloxy)-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 2-(Trifluoromethanesulfonyloxy)-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 2-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 2-1sopropyl-l.2,3,4-tetrahydro[2.7]naphthyridine oxalate 2-AG 2-amino-2-(3-hydoxy-5-methylisoxazol-4-yl)acetic acid, (RS) 2-amino-2-(3-hydoxy-5-methylisoxazol-4-yl)propionic acid 2-Amino-3-(4-bromo-3-hydroxyisothiazol-5-yl)-propionic Acid Hyrochloride 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 2-amino-3-phosphonopropionate 2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate 2-Amino-4-(2,2-dimethylpropyl)-5-(pyridin-3-yl) thiophen-3-yl)(4-chlorophenyl)-methanone 2-Amino-4-(3-difluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-fluorophenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-hydroxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-methoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-methylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-trifluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(3-trifluoromethylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-(dimethylamino)phenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-difluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-fluorophenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-hydroxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-methoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-methylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-trifluoromethoxyphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-(4-trifluoromethylphenyl)-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-benzo[1,3]dioxol-5-yl-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-amino-4-oxo-6-methyl-5-substituted pyrrolo[2,3-d]pyrimidine 2-Amino-4-phenyl-6-(2-hydroxyethylsulfanyl)pyridine-3,5-dicarbonitrile 2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (3,4-dichlorophenyl)methanone 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (3-chlorophenyl)methanone 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (3-trifluoromethylphenyl)methanone 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (4-chlorophenyl)methanone 2-Amino-5-(2,2-dimethylpropyl)thiophen-3-yl] (4-methylphenyl)methanone 2-Amino-5-bromo-4-methylthiophen-3-yl)(4-chlorophenyl)methanone 2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate 2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 2-amino-6-(2-ethoxyphenyl)-N-(pyridin-2-ylmethyl)pyrimidine-4-carboxamide 2-Amino-6-(3-hydroxy-5-methylisoxazol-4-yl)hexanoic Acid 2-Amino-6-ethyl-5-[(1'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(2',6'-dimethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(2'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3',4'-dichlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3',5'-trifluoromethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]p-yrimidine 2-Amino-6-ethyl-5-[(3'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(3'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-fluorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-ethyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-6-methyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2-Amino-N-(2,3-dihydro-5,6-dimethoxy-1H-inden-2-yl)-N-propyl-4-thiazoleethanamine 2-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 2-Amino-N6- (3-iodobenzyl)-adenosine 2-amino-suberic acid 2-Aminoethyl-5-(3'-(2''-methoxy-5''-fluorophenyl)-1'-propyl)tetrahydrofuran 2-Aminoindan 2-Aminoquinoline 2-Arachidonyl glycerol + PMSF 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 2-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-7-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-3-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-(2-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-ethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-Benzylcarbamyl-5-carboethoxy-1-[4-chlorophenyl]pyrrolidine 2-Biphenyl-2-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-Biphenyl-4-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-Br LSD 2-Bromo-3-(2(S)-azetidinylmethoxy)pyridine 2-Bromo-3-ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Bromo-4-(3-fluorophenylethynyl)thiazole 2-Bromo-4-hydroxy-3-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Bromo-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Bromo-5-(1-methyl-2-pyrrolidinyl)pyridine 2-Bromo-alpha-ergocryptine 2-Bromomelatonin 2-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenyl... 2-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenyl... 2-Butyl-7-(2-methoxyphenyl)-2,7-diazaspiro[4.4]nonane 2-CADO 2-carboxymethylbenzenesfulfonamide 2-CH3-5-HT 2-Chloro-3-(2(S)-azetidinylmethoxy)pyridine 2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(R)-pyrrolidinyl)methoxy)pyridine 2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine 2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine 2-Chloro-3-cyclohexyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-cyclopropyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-cyclopropyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-ethyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-hexyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-Chloro-4-hydroxy-3-hydroxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-isopropyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-isopropyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-thione 2-Chloro-4-hydroxy-3-isopropyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-isopropyl-5-phenylthieno[2,3-b]pyridin-6(7H)-thione 2-Chloro-4-hydroxy-3-methoxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-methyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-3-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-5-(3-phenoxyphenyl)-3-propylthieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 2-Chloro-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine 2-Chloro-5'-methylthioado 2-chloro-5,5a,6,7,8,10-hexahydro-5,8-methanopyrrolo[2,1-g][1,7]naphthyridine 2-Chloro-5-(1-methyl-2-pyrrolidinyl)pyridine 2-chloro-5-(2-prpylidene)-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 2-Chloro-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-chloro-5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine 2-chloro-5′-chloro-5′-deoxyN6 -(±)-endo-norbornyl-adenosine 2-Chloro-9-methyladenines 2-Chloro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-benzamide 2-Chloro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)acetamide 2-Chloro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-7-yl)-benzamide 2-chloro-N-(2,6-dimethylphenyl)-N-(2-morpholino-2-(4-nitrophenyl)acetyl)benzamide 2-chloro-N-[3-(4-ethylpiperazin-1-yl)propyl]-4-fluorobenzamide 2-chloro-N-[[2-(4-methylpiperazin-1-yl)phenyl]methyl]benzamide 2-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine 2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine 2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-chloro-5- deoxy-β-D-ribofuranosyl)adenine 2-Chloro-N6 -(±)-endo-norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine 2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine 2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-Dribofuranosyl)adenine 2-Chloro-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine 2-Chloro-N6-(3-iodobenzyl)-adenosine 2-Chloro-N6-(3-iodobenzyl)adenosine-5'-N-methyluronamide 2-chloro-N6-cyclopentyladenosine 2-Chloroadenosine 2-Chloroado 2-Chloroethyldibenzylamine 2-Chloromelatonin 2-CI Adenosine 2-CI-DPH 2-Cl-CPA 2-Cl-diphenidine 2-CPP 2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-cyclohexyl-3-(4-methoxyphenyl)-N-(6-methylpyridin-2-yl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-4-carboxamide 2-cyclohexyl-5-(2-morpholinoethyl)-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 2-cyclohexyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-7-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-cyclohexyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-(2-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... 2-cyclohexyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-(4-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbo... 2-cyclohexyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-7-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2-cyclohexylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.... 2-debromo-2-chloro-psammopemmin A 2-dimethylamino-2-(3-hydroxy-5-methyl-isoxazol-4-yl)acetic acid zwitterion monohydrate, (RS) 2-dimethylamino-2-(3-hydroxy-5-methyl-isoxazol-4-yl)acetic acid zwitterion monohydrate, (RS) 2-dimethylamino-3-(3-hydroxy-5-methyl-isoxalzol-4-yl)-propionic acid zwitterion 2-ethoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 2-Ethoxy-N-{1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl}benzamide 2-Ethoxy-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzamide 2-Ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 2-Ethyl-7-(3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Ethyl-l,2,3,4-tetrahydro[2,7]naphthyrtdme oxalate 2-Ethynyl-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-Ethynyl-4-(3-fluorophenylethynyl)thiazole 2-exo-(5-(6-Hydroxy-1-hexynyl)-3-pyridyl)-7-azabicyclo[2.2.1]heptane 2-exo-norbornyl isomer 2-Fluoro-2-[(2-methoxyphenyl-1-piperazinyl)-methyl]-HEAT HCl 2-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 2-Fluoro-5'-MethylthioAdo 2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine 2-Fluoro-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-fluoro-6-[4-[(2R)-1-methoxypropan-2-yl]piperazin-1-yl]benzonitrile 2-Fluoro-HEAT HCl 2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 2-FluoroAdo 2-Fluorobenzoic Acid 2-(2-fluorobenzoyloxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester 2-Fluoromethyl-3-{4-[2-(4-methylaminophenyl)vinyl]phenoxy}propan-1-ol 2-fluoronorepinehprine 2-furan-2-yl-5-methylamino- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid N0 -phenylhydrazide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (1,1-dimethyl-2-phenyl-ethyl)-amide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (2-phenoxy-ethyl)-amide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3,4-dimethoxy-benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid phenethyl-amide 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid [2-(3,4-dimethoxy-phenyl)-ethyl]-amide 2-Hydrazinobenzenesulfonamide 2-Hydroxy-11-(4-methylpiperazine)-5H-dibenzo[b,e][1,4]diazepine 2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 2-hydroxy-N-[[(3R)-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]methyl]acetamide 2-hydroxydibenzodiazepine 2-hydroxyethyl (S)-7-(buta-1,3-diyn-1-yl)-9-oxo-12,13,13a,14-tetrahydro-9H,11H-benzo[f]imidazo[5,1-d]pyrrolo[1,2-a][1,5]diazo... 2-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 2-Iodomelatonin 2-Iodophenyl-[2-methyl-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone 2-Isopropyl-4-[[1-(2-phenylethyl)-4-piperidinyl]methoxy]-2Hpyrrolo[3,4-c]quinoline 2-Me-Tet-AMPA 2-Methoxy-10-allyl-11-hydroxy-N-methylaporphine 2-Methoxy-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 2-Methoxy-11-allyloxy-N-methylaporphine 2-methoxy-11-hydroxy-N-propylnoraporphine 2-Methoxy-11-hydroxyaporphine 2-Methoxy-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-methoxy-4-amino-5-chlorobenzoic acid 2-(diethylamino)ethyl ester 2-Methoxy-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 2-methoxy-6-methyl-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine 2-methoxy-6-methyl-10-nitro-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 2-methoxy-6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-1-ol 2-methoxy-6-methyl-4-phenyl-1-propoxy-5,6,6a,7-tetrahydro-4H- [1,3]dioxolo[4,5:4,5]benzo[1,2-g]benzo[de]quinoline 2-methoxy-6-methyl-4-phenyl-5,6,6a,7-tetrahydro-4H-[1,3]dioxolo[4,5:4,5]benzo[1,2- g]benzo[de]quinolin-1-ol 2-Methoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 2-methoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 2-methoxy-diphenidine 2-methoxyapomorphine 2-methoxydibenzodiazepine 2-MethoxyethylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate 2-METHOXYPHENYLPIPERAZINE 2-Methyl 5-HT 2-Methyl- 2.3-dihydro-l H-pyrrolo[3,4-c]pyrMine oxalate 2-Methyl-1-(oxazol-2-yl)-1-oxo-9(Z)-octadecene 2-Methyl-3-(4-phenylpiperazinylmethyl)imidazo[1,2-a]-pyridine 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 2-Methyl-3-[4-(4-chlorophenyl)piperazinylmethyl]imidazo-[1,2-a]-pyridine 2-Methyl-4-(2-thienylethynyl)thiazole 2-Methyl-4-(3-thienylethynyl)thiazole 2-methyl-4-(4-(methylthio)phenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 2-Methyl-4-(4-piperidinylmethoxy)-2H-pyrrolo[3,4-c]quinoline 2-Methyl-4-(m-tolylethynyl)thiazole 2-Methyl-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2-methyl-4-phenyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 2-Methyl-4-[4-(3-methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine 2-Methyl-4-[[1-(2-morpholin-4-ylethyl)-4-piperidinyl]methoxy]- 2H-pyrrolo[3,4-c]quinoline 2-Methyl-4-[[1-(2-phenylethyl)-4-piperidinyl]methoxy]-2Hpyrrolo[3,4-c]quinoline 2-Methyl-4-[[3-(trifluoromethoxy)phenyl]ethynyl]thiazole 2-Methyl-4-[[3-(trifluoromethyl)phenyl]ethynyl]thiazole 2-Methyl-5-(1-methyl-2-pyrrolidinyl)pyridine 2-Methyl-5-(2-pyrimidinyl)-1,3-benzothiazole 2-Methyl-5-(6-methyl-2-pyridinyl)-1,3-benzothiazole 2-Methyl-5-phenyl-benzothiazole 2-Methyl-6-[(5-phenyl-3-pyridinyl)ethynyl]pyridine 2-Methyl-6-{[3-(2-thienyl)phenyl]ethynyl}pyridine 2-Methyl-6-{[5-(2-thienyl)-3-pyridinyl]ethynyl}pyridine 2-Methyl-7-(2-hydroxy-3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(2-morpholinoethoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(2-pyrazinyl)quinoline 2-Methyl-7-(2-pyridinyl)quinoline 2-Methyl-7-(2-pyrimidinyl)quinoline 2-Methyl-7-(2-thienyl)quinoline 2-Methyl-7-(3-(2-methylpiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(2-methylpyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(3-hydroxypyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(4-ethylpiperazin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(4-hydroxypiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(4-methylpiperazin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(4-methylpiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(4-oxopiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(diethylamino)propoxy)- 3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-(pyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(4-morpholinobutoxy)-3,4-dihydroisoquinolin-1(2H)-one 2-Methyl-7-(5-methyl-2-pyridinyl)quinoline 2-Methyl-7-phenylquinoline 2-Methyl-l,2,3.4-tetrahydro[2,7]naphthyridine oxalate 2-Methyl-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzamide 2-methyl-serotonin 2-methylhistamine 2-METHYLPHENYLPIPERAZINE 2-Methylsulfonyloxy-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 2-Methylsulfonyloxy-11-(4-methyl-1-piperazinyl)-dibenz[b,f][1,4]oxazepine 2-Methylthiazole-4-carboxylic Acid 3-Fluorophenylamide 2-Methylthiazole-4-carboxylic Acid 3-Pyridylamide 2-methylthio-ATP 2-MPP 2-MsO-11-(4-methl-1-piperazinyl)-5H-dibenzo [b,e] [1,4]diazepine 2-MsO-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 2-MsO-11-(4-methyl-1-piperazinyl)-dibenz[b,f][1,4]oxazepine 2-MXP 2-n-propoxy-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g] quinoxaline HCl 2-NAP 2-NP 2-O-(20 ,30 -dimethylacryloyl)salvinorin B 2-O-(20 -methyl-30 -butenoyl)salvinorin B 2-O-(200,400-dimethoxycinnamoyl)salvinorin B 2-O-(200,500-dimethoxycinnamoyl)salvinorin B 2-O-(200-methoxycinnamoyl)salvinorin B 2-O-(200-nitrocinnamoyl)salvinorin B 2-O-(200-trifluoromethylcinnamoyl)salvinorin 2-O-(200-trifluoromethylcinnamoyl)salvinorin B 2-O-(30 ,30 -dimethylacryloyl)salvinorin B 2-O-(30 -butenoyl)salvinorin B 2-O-(30 -methylbut-30 -enoyl)salvinorin B 2-O-(300,400,500-trimethoxycinnamoyl)salvinorin B 2-O-(300,400-dioxymethylenecinnamoyl)salvinorin B 2-O-(400-methoxycinnamoyl)salvinorin B 2-O-(400-nitrocinnamoyl)salvinorin B 2-O-(400-trifluoromethylcinnamoyl)salvinorin B 2-O-acryloylsalvinorin B 2-O-cinnamoylsalvinorin B 2-O-crotonoylsalvinorin B 2-O-methacryloylsalvinorin B 2-O-[200,500-bis(trifluoromethyl)cinnamoyl]salvinorin B 2-O-[30 -(300-pyridyl)acryloyl]salvinorin B 2-O-[30 -(300-thiophenyl)acryloyl]salvinorin B 2-Oxoado (isoguanosine) 2-Oxoquazepam 2-Phenethylamine 2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167) 2-phenyl-3,1-benzoxazin-4-one 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-(trifluoromethyl)- pyrimidine 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-propylpyrimidine 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-(trifluoromethyl)-pyrimidine 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-propylpyrimidine 2-phenyl-4-[[4-(1,3-thiazol-2-yl)-1,4-diazepan-1-yl]methyl]-1,3-oxazole 2-phenyl-4H-3,1-benzoxazin-4-one 2-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine 2-phenyl-N,N-diallyltryptamine 2-phenylethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]... 2-Phenylethylamine 2-Phenylmelatonin 2-phenylquinazolin-4(3H)-one 2-Piperidino-3'-chloropropiophenone 2-Propyl-l,2,3,4-tetrahydro[2,7]naphthyrMme oxalate 2-Pyrazin-2-yl-1H-benzoimidazol 2-Pyridin-2-yl-1H-benzoimidazol 2-Pyridin-2-yl-3H-benzoimidazol-5-ylamine 2-Pyridin-2-yl-3H-benzoimidazole-5-carbonitrile 2-Pyridin-3-yl-1H-benzoimidazol 2-Pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane 2-Pyrrolidinone, {1-[4-(1-pyrrolidinyl)-2-butynyl]-} 2-Sulfamoylbenzoic acid hydrazide 2-tert-butyl-3-methyl-2,3-dihydroisoquinolin-4(1H)-one 2-tert-butyl-4-[[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl]-1,3-thiazole 2-tert-Butylamino-3',4'-difluoropropiophenone 2-Thio-3-propylX 2-Thiophen-2-yl-1H-benzoimidazol 2-[ [ 4-(2-Carbomethoxyethyl)phenethyl]amino]-adenosine-5’-N-ethylcarboxamide Hydrochloride 2-[(1R,11S,13S,17S,18R,20R,27S,29R,30R,31S,35E)-19-phenyl-21-oxa-8,14,19,26-tetraazadecacyclo[24.5.2.2^{11,14}.0^{1,27}.0^{2,... 2-[(1R,2S)-2-(5-{[(2S)-azetidin-2-yl]methoxy}pyridin-3-yl)cyclopropyl]ethan-1-ol 2-[(1R,2S)-2-(5-{[(2S)-azetidin-2-yl]methoxy}pyridin-3-yl)cyclopropyl]ethyl N-methylcarbamate 2-[(1S)-cyclopent-2-en-1-yl]-1-{4-[(1S,2R)-2-hydroxycyclopentyl]piperazin-1-yl}ethan-1-one 2-[(2,3-Dimethylphenyl)oxalylamino]benzoic Acid 2-[(2-Amino-4-fluoro-5-methylphenyl)thio]-N,N-dimethylbenzenemethanamine 2-[(2-Amino-4-fluoromethylphenyl)thio]-N,N-dimethylbenzenemethanamine 2-[(2-Amino-4-fluorophenyl)thio]-N,N-dimethylbenzenemethanamine 2-[(2-Amino-4-methylphenyl)thio]-N,N-dimethylbenzenemethanamine 2-[(2-Amino-4-methylphenyl)thio]-N-(2-fluoroethyl)benzenemethanamine 2-[(2-Amino-4-methylphenyl)thio]-N-(3-fluoropropyl)-benzenemethanamine 2-[(2-Amino-4-methylphenyl)thio]-N-ethylbenzenemethanamine 2-[(2-Amino-4-methylphenyl)thio]-N-propylbenzenemethanamine 2-[(2-Amino-4-methylphenyl)thio]benzenemethanamine 2-[(2-Benzylphenyl)oxalylamino]benzoic Acid 2-[(2-butoxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[(2-Ethylphenyl)oxalylamino]benzoic Acid 2-[(2-Isopropylphenyl)oxalylamino]benzoic Acid 2-[(2-methoxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[(2-Methyl-4-thiazolyl)ethynyl]pyrazine 2-[(2R)-4-[(5-methyl-2-naphthalen-2-yl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]ethanamine 2-[(3'-Methoxy-3-biphenylyl)ethynyl]-6-methylpyridine 2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]acetic acid bis(tetrafluoroborate) 2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]acetic acid bis(tetrafluoroborate) 2-[(7-Hydroxynaphthalen-1-yl)oxalylamino]benzoic Acid 2-[(E)-2-phenylethenyl]quinazolin-4(3H)-one 2-[(Z)-1-chloro-2-(3-hydroxy-4-methoxyphenyl)ethenyl]-8-methyl-3H-quinazolin-4-one 2-[1-(2-Bromophenyl)methylidene]-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-[1-(2-Bromophenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 2-[1-(4-Hydroxyphenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 2-[2,4-Dioxo-5-phenyl-3-[(1H-pyrazolo[3,4-b]pyridin-4-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-... 2-[2,4-Dioxo-5-phenyl-3-[(4,5,6,7-tetrahydro-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropy... 2-[2,5-Dimethoxy-4-(3-phenyl-propyl)-phenyl]-1-methyl-ethylamine 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamin 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine; 2-[2-(2,4,6-Trimethyl-phenoxy)-acetylamino]-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid (1,1-dioxo-tetrahydro-1lam... 2-[2-(4-Chlorophenyl)ethyl]-5-(1-methyl-2-pyrrolidinyl)pyridine 2-[2-(4-Methoxyphenyl)ethyl]-5-(1-methyl-2-pyrrolidinyl)pyridine 2-[2-(4’-Butoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-N,N-diethylacetamide 2-[2-(4’-Ethoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl]-N,N-diethylacetamide 2-[2-(4’-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl]-N,N-diethylacetamide 2-[2-(ethoxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[2-(hydroxymethyl)piperazin-1-yl]-6-nitroquinoline 2-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(2-methoxyphenyl)... 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(3-methoxyphenyl)... 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[3,4-(methylenedi... 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[4-(trifluorometh... 2-[3-(1H-Indazol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-meth... 2-[3-(1H-Indazol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-terahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methox... 2-[3-(1H-Indol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)ac... 2-[3-(1H-Indol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methox... 2-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxy... 2-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)ethanone 2-[3-(Benzo[d]isoxazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyp... 2-[3-[(1-Benzyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-met... 2-[3-[(4-Fluoro-1H-indazol-3-yl)methyl]methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl... 2-[3-[(5-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-iso... 2-[3-[(6-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-iso... 2-[3-[(7-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-met... 2-[3-[(N-Methylindol-3-yl)methyl]-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-... 2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole 2-[4-(1H-benzimidazol-2-ylamino)-6-methyl-1,3,5-triazin-2-yl]phenol 2-[4-(2,3-Dimethyl-1H-imidazolium-1-yl)-2-butynyl]isoxazolidin-3-one iodide 2-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]isoxazolidin-3-one sesquifumarate 2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole  2-[4-(3-Phenyl-propyl)-phenyl]-ethylamine 2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole 2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-fluoro-1H-indole 2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole 2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methyl-1H-indole 2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile 2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one 2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride 2-[4-[(2R)-2-(3,4-dimethylphenyl)-2-hydroxyethyl]piperazin-1-yl]pyridine-3-carbonitrile 2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dion 2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione 2-[4-[5-(4-methylpyrazol-1-yl)pentyl]piperazin-1-yl]pyridine-4-carbonitrile 2-[5,7-Dimethyl-2-(4-(prop-2-yn-1-yloxy)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-N,N-diethylacetamide 2-[5,7-Dimethyl-2-(4’-propoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]-N,N-diethylacetamide 2-[5-(1-Methyl-2-pyrrolidinyl)-2-pyridinyl]-1-phenylethanol 2-[5-(3,4-Dichlorophenyl)-6-fluoro-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[5-(4-Chlorophenyl)-6-fluoro-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[5-(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxoacetamide 2-[5-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-diethyl-2-oxoacetamide 2-[5-(6-Chloroimidazo[2,1-b][1,3]thiazole-5-sulfonylamino)-1H-indol-3-yl]-N,N-dimethyl-2-oxoacetamide 2-[6-Chloro-5-(4-methoxyphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[6-Chloro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[6-Fluoro-5-(3-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[6-Fluoro-5-(4-fluoro-3-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[6-Fluoro-5-(4-fluorophenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[6-Fluoro-5-(4-methylphenyl)-3-pyridinyl]-7-azabicyclo[2.2.1]heptane 2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline 2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]isoindoline 2-[Oxalyl(2-piperidin-1-ylphenyl)amino]benzoic Acid 2-[Oxalyl-(5,6,7,8-tetrahydronaphthalen-1-yl)amino]- benzoic Acid 2-[p-(2-carboxyethyl)-phenethylamino]-5'-N-ethylcarboxamido adenosine 2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-mesitylenepiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-naphthalen-1-ylpiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-o-tolylpiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-(4-o-xylylpiperazin-1-yl)ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-[(2,3-dimethoxyphenyl)piperazin-1-yl]ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-[4-(benzodioxan-5-yl)piperazin-1-yl]ethanone 2-[[1-(4-Methylpiperazin-1-yl)naphthalen-7-yl]oxy]-1-[4-(o-cyanophenyl)piperazin-1-yl]ethanone 2-[[2-Amino-4-(2-fluoroethyl)phenyl]thio]-N,N-dimethylbenzenemethanamine 2-[[2-Amino-4-(3-fluoropropyl)phenyl]thio]-N,N-dimethylbenzenemethanamine 2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]1H-benzimidazole 2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]benzothiazole 2-[[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]thio]benzoxazole 2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]1H-benzimidazole 2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]benzothiazole 2-[[2-[4-(2-Nitrophenyl)-1-piperazinyl]ethyl]thio]benzoxazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]-1-methyl-1H-benzimidazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]1H-benzimidazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(2-Methoxyphenyl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]1H-benzimidazole 2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(2-Nitrophenyl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(Pyridin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzothiazole 2-[[3-[4-(Pyrimidin-2-yl)-1-piperazinyl]propyl]thio]benzoxazole 2-[[4-(2-Carboxyethyl)phenethyl]amino]adenosine-5'-N-ethylcarboxamide Hydrochloride 2-[[4-(2-Carboxyethyl)phenethyl]amino]adenosine-5'-N-ethylcarboxamide Hydrochloride 2-[[4-(2-phenylethyl)piperazin-1-yl]methyl]indolizine-1-carbonitrile 2-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methylsulfanyl]-N-(2-methylphenyl)acetamide 2-[[4-[4-(2-Methoxyphenyl)-1-piperazinyl]butyl]thio]benzothiazole 2-[[4-[4-(2-Methoxyphenyl)-1-piperazinyl]butyl]thio]benzoxazole 2-[[6-[4-(2-Methoxyphenyl)-1-piperazinyl]hexyl]thio]benzothiazole 2-[[6-[4-(2-Methoxyphenyl)-1-piperazinyl]hexyl]thio]benzoxazole 2-{(1H-Pyrrolo[2,3-b]pyridin-3-yl)methyl}-5-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane 2-{1-[2,5-Di(trifluoromethyl)phenyl]methylidene}-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 2-{1-[4-(Dimethylamino)phenyl]methylidene}-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(3,4-dihydroisoquinoline) 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2'-pyrimidil)piperazine 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3'-chlorophenyl)piperazine 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3'-trifluoromethyl)piperazine 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(N-methyl)piperazine 2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-2-aza-spiro[4.5]decane-1,3-dione 2-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol 2-{4-[2-(4-Methylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol 2-{4-[4-(3-Methoxyphenyl)-1-piperazinyl]butyl}-4-methyl-1,2,4-triazine-3,5(2H,4H)-dione 2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione 2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-methyl-amine 2-{6-[2-(4-Chlorophenyl)ethyl]-3-pyridinyl}-N-ethyl-N-methylethanamine 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione 2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione 2-{[2-(2-Carbamoylvinyl)-4-(2-(S)-methanesulfonylamino-2-pentylcarbamoylethyl)phenyl]oxalylamino}- benzoic Acid 2-{[2-(2-Carbamoylvinyl)phenyl]oxalylamino}benzoic Acid 2-{[2-(2-Hydroxyethyl)phenyl]oxalylamino}benzoic Acid 2-{[3-(2-Furyl)phenyl]ethynyl}-6-methylpyridine 2-{[4-((S)-2-tert-Butoxycarbonylamino-2-pentylcarbamoylethyl)phenyl]oxalylamino}benzoic Acid 2-{[4-(2-(S)-Acetylamino-2-pentylcarbamoylethyl)- phenyl]oxalylamino}benzoic Acid 2-{[4-(2-(S)-Amino-2-pentylcarbamoylethyl)phenyl]- oxalylamino}benzoic Acid 2-{[4-(2-(S)-Methanesulfonylamino-2-pentylcarbamoylethyl)phenyl]oxalylamino}benzoic Acid 2-{[4-(2-Acetylamino-2-pentylcarbamoylethyl)-2- ethylphenyl]oxalylamino}benzoic Acid 2-{[4-(2-Acetylamino-2-pentylcarbamoylethyl)-2-piperidin-1-ylphenyl]oxalylamino}benzoic Acid 2-{[4-(2-Acetylamino-2-pentylcarbamoylethyl)naphthalen-1-yl]oxalylamino}benzoic Acid 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l4-thiaspiro[4.5]decan-8-one 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l6-thiaspiro[4.5]decane-8,8-dione 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyridin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-phenyl-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane 2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-N-phenyl-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide 2-{[5-(2-Furyl)-3-pyridinyl]ethynyl}-6-methylpyridine 2-{[5-(3-Methoxyphenyl)-3-pyridinyl]ethynyl}-6-methylpyridine 20 20-COOH-LTB4 20-OH-LTB4 20a 20b 21 21-nitro-7alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 21-nitro-8alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 21a 21b 21c 22 22-nitro-7apha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 22-nitro-8alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 227I-BOP 22a 22b 23 24 24c 25 25CN-NBOH 26 26A 26B 26c 27 27 (6-PBC) 27a 27b 28 28g 28h 28i 28j 28k 28l 29 29a 29b 2a 2alpha,3alpha-Di(4-methylphenyl)tropane 2alpha,3alpha-Diphenyltropanes 2‐methyl‐5‐(2‐phenylethyl)‐1H,2H,3H,4H,5H‐pyrido[4,3‐b]indole 2′′-F-DPPy 2″-glucosylvitexin 2b 2beta,3beta-Di(4-methylphenyl)tropane 2beta,3beta-Diphenyltropanes 2beta-(4-Fluorophenyl)-3beta-(4-methylphenyl)tropane 2C-B, 4-bromo-2,5-dimethoxyphenethylamine 2C-BI-1 2C-BI-10 2C-BI-11 2C-BI-12 2C-BI-2 2C-BI-3 2C-BI-4 2C-BI-5 2C-BI-7 2C-BI-8 2e 2f 2g 2Me4CPG 2R)-1-(4-methylphenoxy)-3-[4-(pyrazol-1-ylmethyl)piperidin-1-yl]propan-2-ol 2R, 4R-APDC 2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide 2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide 2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2'-methoxyphenyl)piperazine 2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(4'-fluorophenyl)piperazine 3 3 (BCCE) 3 EBC 3 PBC 3'-(3-Aminophenyl)epibatidine 3'-(3-Bromophenyl)epibatidine 3'-(3-Chlorophenyl)epibatidine 3'-(3-Dimethylaminophenyl)epibatidine 3'-(3-Fluorophenyl)epibatidine 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 3'-(3-nitrophenyl)epibatidine 3'-(4-Aminophenyl)epibatidine 3'-(4-Chlorophenyl)epibatidine 3'-(4-fluorophenyl)deschloroepibatidine 3'-(4-Methoxylphenyl)epibatidine 3'-(4-Nitrophenyl)epibatidine 3'-(7-Methyl-imidazo[1,2-b]pyridazin-3-yl)-biphenyl-2-carbonitrile 3'-Amino-N-(1-benzyl-3-pyrrolidinyl)-4-biphenylcarboxamide 3'-Deoxyadenosine (cordycepin) 3(R)-Amino-2-(R,S)-hydroxybutyl)phosphinic Acid 3, 4-Dihydroxyphenethylamine 3, {4-Dihydroxy-alpha-[(methylamino)methyl]benzyl} alcohol 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3,4,5-Trimethoxyphenethylami 3,4,5-Trimethoxyphenethylamine 3,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}furan 3,4-dichloro amphetamine 3,4-dichloro-N-(4-phenyl-1,3-thiazol-2-yl)benzamide 3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7... 3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-Difluoro-N-{1-[2-(3-fluorophenoxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 3,4-Difluoro-N-{1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl} benzenesulfonamide 3,4-Difluoro-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 3,4-Dihydro-2-[4-(3,4-dihydro-6-methoxypyrazino[1,2-a]indol-2(1H)-yl)butyl]pyrazino[1,2-a]indol-1(2H)-one 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one 3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one 3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 3,4-Dihydroxyphenylethylamine 3,4-Dimethoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)-oxy]morphinan-6-one 3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3,4-Dimethoxy-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide 3,4-Dimethoxy-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide 3,4-DNH 3,4CTMP 3,5-DHPG 3,5-dihydroxyphenylglycine 3,5-Dimethyl-2-phenyl-3H-imidazo[4,5-b]pyridine 3,5-diphenylpyridazine 3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 3,6-diacetyldihydromorphine 3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine 3,7-dimethyl-1-n-propylxantine 3,7-dimethyl-1-proporgylxantine 3,7-Dimethyl-8-(m-hydroxystyryl)-1-propargylxanthine 3,7-dimethylxanthine 3,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine 3,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine 3,9,10-Trimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 3,9-Dimethoxy-10-(pentyloxy)-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 3,9-Dimethoxy-10-propoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-2-ol 3,9-DimethylX 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine 3-(((4-Hydroxy-3-methoxyphenethyl)(methyl)amino)methyl)-2-methoxyphenol 3-((1-(pyrrolidin-1-yl)cyclopropyl)methoxy)pyridine 3-((1-Methyl-2(R)-azetidinyl)methoxy)pyridine Dihydrochloride 3-((1-Methyl-2(R)-pyrrolidinyl)methoxy)pyridine Dihydrochloride 3-((1-Methyl-2(S)-azetidinyl)methoxy)pyridine Dihydrochloride 3-((1-Methylpiperidin-4-yl)methoxy)-5-(phenoxymethyl)-isoxazole Hydrochloride 3-((1H-Pyrrole-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol 3-((2,2-Dimethylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((2,6-dichlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-fluorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((2-hydroxyethoxy)methyl)-6,9-dimethyl-5,6-dihydrobenzo[g]imidazo[1,5-a][1,5]diazocin-7(4H)-one 3-((2-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3,3-Difluoroazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3,3-Dimethylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propyl)thio)-5-phenyl-4H-1,2,4-triazol-4-amine 3-((3-Methylazetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((3R,4R)-1-((S)-3-cyclohexyl-3-hydroxypropyl)-3,4-dimethylpiperidin-4-yl)phenol 3-((4-chlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((4-isopropylphenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)propan-1-amineHydrochloride 3-((5-Methoxy-1H-indol-3-yl)methyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one 3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-N,N-dipropylpropan-1- amine 3-((Acetoxy)-1-methylpropyl)dimethylammonium Oxalate 3-((Azetidine-1-carbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((Benzoyloxy)-1-methylpropyl)dimethylammonium Chloride 3-((Cyclobutanecarbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 3-((Cyclopropanecarbonyloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((Ethyl(4-hydroxy-3-methoxyphenethyl)amino)methyl)-2-methoxyphenol 3-((Isobutyryloxy)-1-methylpropyl)dimethylammonium Oxalate 3-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonit... 3-((S)-1-Azetidin-2-ylmethoxy)-2-fluoro-pyridine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 3-(1-Methyl-2-pyrrolidinyl)-4-pyridinamine 3-(1-Methyl-2-pyrrolidinyl)-5-propylpyridine 3-(1-methyl-2-pyrrolidinyl)pyridine 3-(1-methyl-2-pyrrolidinyl)pyridine, (+) 3-(1-methyl-2-pyrrolidinyl)pyridine, (-) 3-(1-methyl-2-pyrrolidinyl)pyridine, (S) 3-(1-methyl-2-pyrrolidinyl)pyridine-6-acetamide 3-(1-methyl-2-pyrrolidinyl)pyridine-6-carboxamide oxalate 3-(1-Methylcyclopropyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine1,1-Dioxide 3-(1-{17-[4-({[5-(Ethoxycarbonyl)-2,6-dimethyl-4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-1,4-dihydropyridin-3-yl]carbonyloxy}meth... 3-(1-{2-[2-(2-{4-[({4-[3-(4-Bromophenyl)-5-methyl-1,2-oxazol-4-yl]-5-(ethoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridin-3-yl}ca... 3-(1H-Indol-3-yl)-N-[5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]propionamide 3-(2(R)-Azetidinylmethoxy)pyridine Dihydrochloride 3-(2(R)-Pyrrolidinylmethoxy)pyridine Dihydrochloride 3-(2(s)-Azetidinylmethoxy) Pyridine 3-(2,4-Difluorophenyl)-5-[3-(3,5-difluoropyridin-2-yl)-4-fluorophenyl]pyridazine 3-(2,4-Dimethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2,4-dithioxo-1,3-thiazolidin-3-yl)propanoic acid 3-(2,6-Difluorophenyl)-5-[4-fluoro-3-(3-fluoropyridin-2-yl)-phenyl]pyridazine 3-(2-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9- diazaspiro[5.5]undecane 3-(2-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-yl)eth... 3-(2-(2-Fluoroethoxy)phenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4- triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one 3-(2-(allylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(benzylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(5-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(butylamino)ethyl)-8-(6,7-dichloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-... 3-(2-(butylamino)ethyl)-8-(6-chloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-on... 3-(2-(butylamino)ethyl)-8-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclobutylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclohexylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclohexylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-... 3-(2-(cyclopentylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclopropylmethylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(cyclopropylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4... 3-(2-(diisopropylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-(S)-Pyrrolidinylmethoxy)pyridine Fumarate 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide 3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(2-Aminoethyl)-2-chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one hydrochloride 3-(2-Aminoethyl)-2-chloro-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one hydrochloride 3-(2-aminoethyl)-8-(bis(2-chlorophenyl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 3-(2-Chlorophenoxycarbonylmethyl)-8-chloropyrazolo-[5,1-c][1,2,4]benzotriazine 5-oxide 3-(2-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(2-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 3-(2-Dimethylaminoethyl)-4-hydroxy 2-methylindole 3-(2-Dimethylaminoethyl)-6-hydroxyindole 3-(2-DIMETHYLAMINOETHYL)INDOL-5-OL 3-(2-Ethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Fluoro-4-(trifluoromethyl)phenyl)-9-(3-((4-methyl-5-phenyl4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(2-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 3-(2-Fluorophenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 3-(2-Furylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 5-oxide 3-(2-Hydroxyethyl)-8-(m-methoxystyryl)-7-methyl-1-propargylxanthine 3-(2-Methoxy-phenyl)-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-acrylamide 3-(2-Methoxybenzyloxycarbonyl)-8-chloro pyrazolo-[5,1-c][1,2,4]benzotriazine 3-(2-Methoxyphenoxycarbonylmethyl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide 3-(2-Methoxyphenyl)-9-(2-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)ethyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methoxyphenyl)-9-(3-((1-methyl-5-phenyl-1H-imidazol-2- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-(4-(thiophen-3-yl)- phenyl)-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]- und... 3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-(pyridin-3-yl)-4H-1,2,4- triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane 3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)propyl)-3,9-diazaspiro[5.5]undec-1-ene 3-(2-Methoxyphenyl)-9-(3-((5-(2-methoxyphenyl)-4-methyl-4H1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methoxyphenyl)-9-(3-((5-phenyl-1H-imidazol-2-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methoxyphenyl)-9-(3-((5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methoxyphenyl)-9-(4-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)butyl)-3,9-diazaspiro[5.5]undecane 3-(2-Methyl-1,3-benzothiazol-5-yl)benzonitrile 3-(2-Methyl-7-quinolinyl)benzonitrile 3-(2-Thienylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 3-(2-Thienylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 5-oxide 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)-8-methylpyrimido[5,4-c]quinolin-4(3H)-one 3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)-9-methylpyrimido[5,4-c]quinolin-4(3H)-one 3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)pyr-imido[5,4-c]equinolin-4(3H)-one 3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 3-(3,5-Difluoropyridin-4-yl)-5-[4-fluoro-3-(3-fluoropyridin-2- yl)phenyl]pyridazine 3-(3-((4-Ethyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-9-(2- methoxyphenyl)-3,9-diazaspiro[5.5]undecane 3-(3-((5-(2-Fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane 3-(3-((5-(4-Fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane 3-(3-((5-Cyclohexyl-4-methyl-4H-1,2,4-triazol-3-yl)thio)propyl)- 9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane 3-(3-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(3-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 3-(3-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(3-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 3-(3-Furylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 5-oxide 3-(3-hydroxypentyl)-N-(1-propyl)piperidine 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate 3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide 3-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane 3-(3-Thienylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-1,2,4]benzotriazine 5-oxide 3-(3-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}propyl)pyrimido[5,4-c]quinolin-4(3H)-one 3-(4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxybenzofuran-2-yl)-N-(2-(dimethylamino)ethyl)benzamide 3-(4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-ylamino)propan-1-ol 3-(4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl)benzoic acid 3-(4-(3,4-dichlorophenethyl)piperazin-1-yl)benzo[d]isothiazole hydrochloride 3-(4-(3-(methoxymethyl)-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-(4-fluorophenyl)naphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-(4-hydroxyphenyl)naphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-(4-methoxyphenyl)naphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-butyl-6-hydroxy-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(3-cyclopropyl-6-hydroxy-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(4-cyclohexylpiperazin-1-yl)butyl)benzo[d]thiazole-2(3H)-thione 3-(4-(6-hydroxy-3-isobutyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(6-hydroxy-3-octyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-(6-hydroxy-3-pentyl-2-phenylnaphthalen-1-yloxy)phenyl)acrylic acid 3-(4-aminobenzyl)indene 3-(4-aminobenzyl)indole 3-(4-aminophenethyl)-7-(2-(ethyl(2-hydroxyethyl)amino)ethyl)-1-propyl-1H-purine-2,6(3H,7H)-dione 3-(4-Benzyl-piperazin-1-yl)-phenol 3-(4-benzylpiperazin-1-yl)-N-(1,3-thiazol-2-yl)propanamide 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(4-Chlorophenyl)-1-(1H-indol-3-ylmethyl)pyrrolidin-3-ol 3-(4-Chlorophenyl)-1-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrrolidin-3-ol 3-(4-Chlorophenyl)-1-[2-(1H-indol-3-yl)ethyl]pyrrolidin-3-ol 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2,2-trifluoroethyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2-difluorobutyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-(2,2-difluoropropyl)-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-2-(2-chlorophenyl)-7-isopropyl-6,7-dihydro-2H,5H-4-oxa-1,2,7-triazulen-8-one 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 3-(4-Chlorophenyl)-5-morpholin-4-yl-1,2,4-oxadiazole 3-(4-Chlorophenyl)-8-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-Chlorophenyl)-8-(4-fluorobenzyl)-8-azabicyclo[3.2.1]octan-3-ol 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-(2-hydroxy-2-methylpropyl)-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidin... 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[3-(dimethylamino)propyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine... 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(methyl)-piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidi... 3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(pyrrolidin-1-yl)butyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidin... 3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide 3-(4-chlorophenyl)deschloroepibatidine 3-(4-Fluoro-2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 3-(4-Fluorophenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-(4-fluorophenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(4-Methoxyphenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-(4-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane 3-(4-methylphenyl)tropane-2-carboxylic acid methyl ester 3-(4-Methylpiperazin-1-yl)-5-(phenoxymethyl)isoxazole Hy-drochloride 3-(4-Propyl-1-piperazinyl)phenol 3-(4-Pyridylmethoxycarbonyl)-8-chloropyrazolo[5,1-c]-[1,2,4]benzotriazine 5-oxide 3-(4-tert-butylbenzoyl)-2-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)thiazolidine-4-carboxamide 3-(4-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}butyl)pyrimido[5,4-c]quinolin-4(3H)-one 3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid 3-(5-Benzoyl-2-isobutoxyphenyl)propionic Acid 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluor... 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Cyano-6-(propylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 3-(5-Methyl-2-phenyl[1,3]thiazolo[4,5-b]pyridin-6-yl)benzonitrile 3-(5-Phenylpyridazin-3-yl)benzonitrile 3-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d] oxazol-2(3H)-one 3-(6-Ethoxypyridazin-4-yl)benzonitrile 3-(6-ethylaminopyridazin-4-yl)-benzonitrile 3-(6-methylpyridin-2-ylcarbamoyl)phenyl methanesulfonate hydrobromide 3-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester 3-(6-Phenyl-pyridazine-4-yl)-benzoic acid methyl ester 3-(6-Phenylpyridazin-4-yl)benzonitrile 3-(8-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-yl)oct... 3-(8-(3,4-dichlorophenyl)-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)-N,N-diethylpropan-1-amine 3-(8-(3,4-dichlorophenyl)-6-methyl-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)-N,N-diethylpropan-1-amine 3-(Anilinomethyl)-5-[(2(S)-azetidinyl)methoxy]isoxazole 3-(azepan-1-yl)-N,5-dicyclopropyl-2-methylbenzenamine 3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate 3-(benzo[d][1,3]dioxol-5-yl)-N-(2-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-2-oxo-1-p-tolylethyl)-N-methylacrylamide 3-(Benzyloxy)-5-(3-bromophenyl)pyridazine 3-(Benzyloxy)-5-(3-cyanophenyl)pyridazine 3-(benzyloxy)-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-(chloromethyl)-6,9-dimethyl-5,6-dihydrobenzo[g]imidazo[1,5-a][1,5]diazocin-7(4H)-one 3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 3-(dimethylamino) butyl pyrrolidine-1-carboxylate 3-(dimethylamino)butyl dimethylcarbamate 3-(dimethylamino)butyl methylcarbamate 3-(dimethylamino)butyl piperidine-1-carboxylate 3-(Dimethylamino)fluoranthene 3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole 3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole 3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole 3-(m-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepin 3-(m-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 3-(methoxymethyl)-6,9-dimethyl-5,6-dihydrobenzo[g]imidazo[1,5-a][1,5]diazocin-7(4H)-one 3-(N-Cyclopropyl-N-methylaminornethyl)pyrMine oxalate 3-(N-ethyl-N-n-methylaminomethyl)pyridine; 3-(N-Formylcarbamoyl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-(N-Methyl-N-n-peno, laminomethyl)pyrtdine oxalate 3-(N-methyl-N-n-propylaminomethyl)pyridine 3-(N-Methyl-N-n-propylaminomethyl)pyridine oxalate 3-(N-Methyl-N-n-propylammomethyl)-2-methylpyridine oxalate 3-(N-n-Butyl-N-methylaminornethyl)pyridine oxalate 3-(N-propylpiperidin-4-yl)phenol 3-(o-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(oxolan-2-ylmethyl)-8-phenyl-1-propyl-7H-purine-2,6-dione 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 3-(Phenoxymethyl)-5-[(2(S)-pyrrolidinyl)methoxy]isoxazole 3-(Phenylmethyl)-1-(4-phenyl-1-piperazinyl)propan-1-one 3-(Phenylsulfonyl)-4-(2-piperidin-1-ylethyl)-1H-indole 3-(Phenylsulfonyl)-4-(2-pyrrolidin-1-ylethyl)-1H-indole 3-(Phenylsulfonyl)-4-(3-piperidin-1-ylpropyl)-1H-indole 3-(piperazin-1-yl)-N-(m-tolyl)propanamide 3-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 3-(pyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane 3-(Pyrrol-1-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-(tert-butylamino)-1-(3-chlorophenyl)-2-methylpropan-1-one 3-(Tetrahydro-3-furylmethoxycarbonyl)-8-chloropyrazolo[5,1-c][1,2,4]benz otriazine 5-oxide 3-(Thien-2-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-(Thien-3-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)benzonitrile 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyrazine-2-carbonitrile 3-allyl-8-benzhydryl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 3-Amino-5-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carbothioamide 3-amino-6-ethyl-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propylthio)thieno[2,3-d]pyrimidin-4(3H,4aH,7aH)-one 3-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 3-Aminofluoranthene 3-AMTBI 3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester 3-benzyl-5-cyclopentyl-1-propylxanthine 3-Benzyl-5-methyl-2-phenyl-3H-imidazo[4,5-b]pyridine 3-Benzyl-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 3-Benzyl-8-[4-chlorophenyl]-3,8-diazabicyclo[3.2.1]octane-2,4-dione 3-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3-benzyl-N1-(N,N-dimethylaminoethyl)indole 3-Benzylamino-6-chloro-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 3-beta-hydroxyethyl-1-methylxantine 3-Bromo-5-(1-methyl-2-pyrrolidinyl)pyridine 3-Bromo-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-bromo-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-bromoboldine 3-Butoxycarbonyl-4-quinolone 3-Butoxycarbonyl-6-ethyl-4-quinolone 3-Butyl-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane 3-Butylaminocarbonyl-6-ethyl-4-quinolone 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 3-Carboethoxy-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 3-Carboxy-6-ethyl-4-quinolone 3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]piperidin-4-yl}benzenesulfonamide 3-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide 3-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3-chloro-5,7,8,9,9a,10-hexahydro-7,10-methanopyrrolo[1,2-b][2,6]naphthyridine 3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide 3-Chloro-N-(1,2,3,4-tetrahydro-1,3,4-trioxoisoquinolin-6-yl)propanamide 3-Chloro-N-(1-{2-[(propan-2-yl)-phenyloxy]ethyl} pyrrolidin-3-yl)benzenesulfonamide 3-chloro-N-(4-methylthiazol-2-yl)benzamide hydrobromide 3-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide 3-chloro-N-(6-chloropyridin-2-yl)benzamide hydrobromide 3-Chloro-N-(6-methyl-2-pyridinyl)benzamide 3-chloro-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-Chloro-N-({1-[2-(2-methylsulfanylphenoxy)ethyl] piperidin-4-yl}methyl) benzenesulfonamide 3-Chloro-N-({1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl}methyl)benzenesulfonamide 3-Chloro-N-({1-[2-(methylsulfanyl)phenyloxy]ethyl}pyrrolidin-3-yl)benzenesulfonamide 3-Chloro-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide 3-chloro-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-4-hydroxybenzamide 3-Chloro-N-{[1-(2-(2-methoxyphenoxy)ethyl)piperidin4-yl]methyl}benzenesulfonamide 3-chlorophenyl (±)-(4aR,8S,8aR)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 3-chlorophenyl (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 3-chlorophenyl (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 3-CPP 3-Cyano-N-(6-methyl-2-pyridinyl)benzamide 3-cyano-N-(6-methylpyridin-2-yl)benzamide 3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one 3-Cyclopentoxycarbonyl-6-ethyl-4-quinolone 3-Cyclopropyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 3-cyclopropyl-N-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-amine 3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 3-Deoxy-1,2-O-isopropylidene-D-glucose 3-desoxy-3-carboxamidonaltrexone 3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine 3-Ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene 3-Ethoxycarbonyl-4-quinolone 3-Ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone 3-Ethoxycarbonyl-6-ethyl-4-quinolone 3-Ethoxycarbonyl-6-i-propyl-4-quinolone 3-Ethoxycarbonyl-6-propyl-4-quinolone 3-Ethyl-1-methyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3-Ethyl-1-methyl-8-(4-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3-ethyl-1-NP 3-ethyl-2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-1H-benzimidazole-1-carboxamide 3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxylic acid (8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-amide 3-Ethyl-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 3-Ethyl-4-hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 3-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione 3-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione 3-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 3-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3-Ethyl-8-(4-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3-Ethyl-8-{1-[1-(3-fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione 3-Ethyl-8-{1-[1-(4-fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione 3-Ethyl-8-{1-[1-(4-methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione 3-Ethyl-8-{1-[5-oxo-1-(3-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dio... 3-Ethyl-8-{1-[5-oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dion... 3-Ethyl-8-{1-[5-oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dion... 3-ethyl-THIQ 3-Ethynyl-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine 3-F-DPPy 3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile 3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 3-Fluoromethyl-7-bromo-THIQ 3-Fluoromethyl-7-cyano-THIQ 3-Fluoromethyl-7-N-(4-chlorophenyl)aminosulfonyl-THIQ 3-Fluoromethyl-7-nitro-THIQ 3-fluoromethyl-THIQ 3-Heptanone, 6-(dimethylamino)-4,4-diphenyl-, (+-)- 3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid, (RS) 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3-Hydroxy-9-aminomethyl-9,10-dihydroanthracene 3-Hydroxymethyl-7-nitro-THIQ 3-Hydroxymethyl-THIQ 3-Hydroxytyramine 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine4-oxide 3-iodo-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-Iodoboldine 3-Iodophenyl-[2-methyl-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone 3-isobutyl-1-methyl 3-isobutyl-1-methyl-7-n-propylxantine 3-isobutyl-1-methyl-7-propargylxantine 3-Isobutyl-1-methylxanthine 3-isobutyl-1-methylxantine 3-isopropyl-1-methyl 3-isopropyl-2,3-dihydro-N-[endo-8-methyl-8-azabicylclo(3.2.1)oct-3-yl]-2-oxo-1H-benzimidazole-1-carboxamide 3-Isopropylcarbonyl-8-chloropyrazolo[5,1-c][1,2,4]-benzotriazine 5-oxide 3-methoxy-4-((S)-((S)-morpholin-2-yl)(phenyl)methoxy)benzonitrile 3-Methoxy-5-(1-methyl-2-pyrrolidinyl)pyridine 3-methoxy-9-aminomethyl-9,10-dihydroanthracene 3-methoxy-dibenz[d,g]azecine 3-methoxy-diphenidine 3-methoxy-N-(4-methylthiazol-2-yl)benzamide hydrobromid 3-methoxy-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-methoxyeticyclidine hydrochloride 3-Methoxymethyl-THIQ 3-methoxyphencyclidine hydrochloride 3-METHOXYPHENYLPIPERAZINE 3-Methyl-1,2,3,4,8,13-hexahydropyrido[4,3:2,3]indolo[1,7-bc][2]benzazepine 3-Methyl-1,2,3,4,8,9-hexahydropyrido[4,3:2,3]indolo[1,7-ab][1]benzazepine 3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 3-Methyl-2-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-benzonitrile 3-Methyl-2-((R)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)-phenol 3-methyl-2-(4-(3-(pyrrolidin-1-yl)propoxy)phenyl)quinazolin-4(3H)-one 3-Methyl-2-morpholin-4-yl-7-[(4-phenylpiperazin-1-yl)methyl]-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 3-Methyl-5-(1-methyl-2-pyrrolidinyl)pyridine 3-Methyl-5-[(2(S)-pyrrolidinyl)methoxy]isoxazole 3-Methyl-6-phenyl-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole 3-methyl-6-phenyl-1,5-dihydropyrrolo[3,2-d]pyrimidin-2,4-dione 3-Methyl-7-nitro-THIQ 3-Methyl-7-[(4-phenylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 3-Methyl-7-[(4-pyridin-2-ylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 3-methyl-N-(6-methylpyridin-2-yl)benzamide hydrobromide 3-Methyl-N-phenyl-N-(3-(piperidin-1-yl)propyl)benzofuran-2-carboxamide (KSCM-5) 3-methyl-THIQ 3-methylbutyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]... 3-MXP 3-N,N-dimethylaminobutyl-N,N-dimethylcarbamate 3-n-Hexyl-6-methoxy-9-aminomethyl-9,10-dihydroanthracene 3-n-Pentyloxy-9-aminomethyl-9,10-dihydroanthracene fumarate 3-PBC 3-Phenyl-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 3-phenyl-1,4-benzoxazin-2-one  3-phenyl-1-NP 3-Phenyl-2-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-propionic acid te... 3-Phenyl-4-N-phenylamino-1-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrazolo[3,4-d]pyrimidine 3-Phenyl-4-N-phenylamino-1-alpha-L-lyxofuranosylpyrazolo[3,4-d]pyrimidine 3-Phenyl-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 3-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine 3-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine 3-Phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 3-phenylchromen-2-one 3-phenylisochromen-1-one 3-phenylisoquinolin-1(2H)-one 3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0... 3-Propylxanthine (enprofylline) 3-Tert-butoxy-N-{1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}propanamide 3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)urea 3-tert-Butyl-2-chloro-4-hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]-pyridin-6(7H)-one 3-Trifluoromethylphenylpiperazine 3-[((1S,2S,5R)-3-Azabicyclo[3.1.0]hexan-2-yl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(1,4-cis)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-cis)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-cis)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-trans)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-trans)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1,4-trans)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[(1-Ethyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-((1S,2S)-2-ethylcyclopropyl)-pyridine trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 3-[(2(S)-Azetidinyl)methoxy]-5-isoxazolylmethanol 3-[(2(S)-Azetidinyl)methoxy]-5-methylisoxazole 3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2,2-difluoroethyl)-cyclopropyl]pyridine trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperidin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-fluoroethyl)-cyclopropyl]pyridine trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate 3-[(2(S)-Azetidinyl)methoxy]-5-[(cyclopropylmethoxy)methyl]isoxazole 3-[(2(S)-Azetidinyl)methoxy]-5-[(hexyloxy)methyl]isoxazole 3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 3-[(2,4-dimethoxy)benzylidene]-anabaseine 3-[(2,5-Dimethyl-4-thiazolyl)ethynyl]pyridine 3-[(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)carbamoyl]benzenesulfonyl fluoride 3-[(2-Methyl-4-oxazolyl)ethynyl]pyridine 3-[(2-Methyl-4-thiazolyl)ethynyl]-5-vinylpyridine 3-[(2-Methyl-4-thiazolyl)ethynyl]benzamide 3-[(2-Methyl-4-thiazolyl)ethynyl]benzonitrile 3-[(2-Methyl-4-thiazolyl)ethynyl]phenol 3-[(2-Methyl-4-thiazolyl)ethynyl]quinoline 3-[(2-Methyl-5-phenyl-4-thiazolyl)ethynyl]pyridine 3-[(3(R)-Pyrrolidinyl)oxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridineTrifluoroacetate 3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[(5-Ethyl-2-methyl-4-thiazolyl)ethynyl]pyridine 3-[1-(17-{4-[({4-[3-(m-bromophenyl)-5-methyl-1,2-oxazol-4-yl]-5-(ethoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridin-3-yl}carbony... 3-[1-(17-{4-[({4-[3-(o-Bromophenyl)-5-methyl-1,2-oxazol-4-yl]-5-(ethoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridin-3-yl}carbony... 3-[1-(17-{4-[({4-[3-(p-Bromophenyl)-5-methyl-1,2-oxazol-4-yl]-5-(ethoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridin-3-yl}carbony... 3-[1-(2-{2-[2-(2-{4-[({4-[3-(p-Bromophenyl)-5-methyl-1,2-oxazol-4-yl]-5-(ethoxycarbonyl)-2,6-dimethyl-1,4-dihydropyridin-3-yl... 3-[2-(1,3-dihydroisoindol-2-yl)ethyl]-1-methyl-1-[(1-methylpyrazol-4-yl)methyl]urea 3-[2-(4-Pyrimidin-2-ylpiperazin-1-yl)ethyl]pyrimido[5,4-c]quinolin-4(3H)-one 3-[2-(DIMETHYLAMINO)ETHYL]-2-METHYLINDOLE 3-[2-(DIMETHYLAMINO)ETHYL]-2-METHYLINDOLE 3-[2-(Isopropylamino)ethoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate 3-[2-Benzyloxy-5-(4-isobutoxybenzoyl)phenyl]propionic Acid 3-[2-Isobutoxy-5-(3-isobutoxybenzoyl)phenyl]propionic Acid 3-[2-Isobutoxy-5-(4-isobutoxybenzoyl)phenyl]propionic Acid 3-[2-Isobutoxy-5-(4-propoxybenzoyl)phenyl]propionic Acid 3-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3-[2-[Diphenethylamino]ethyl]phenol 3-[3-(4-Isobutoxybenzoyl)phenyl]propionic Acid 3-[3-(4-Phenylpiperazin-1-yl)propyl]-8-methylpyrimido[5,4-c]quinolin-4(3H)-one 3-[3-(4-Phenylpiperazin-1-yl)propyl]-9-methylpyrimido[5,4-c]quinolin-4(3H)-one 3-[3-(4-Phenylpiperazin-1-yl)propyl]pyrimido[5,4-c]quino-lin-4(3H)-one 3-[3-(4-Pyrimidin-2-ylpiperazin-1-yl)propyl]pyrimido[5,4-c]quinolin-4(3H)-one 3-[3-(Imidazol-4(5)-yl)propyl]-1-[3-[N-(4-bromobenzyl)-N-(pyrid-2-yl)amino]propyl]-S-methylisothiourea Hydroiodide Dihydrochl... 3-[3-[[[(3R)-oxolan-3-yl]amino]methyl]indol-1-yl]propanamide 3-[4-(2,3-Dimethyl-1H-imidazolium-1-yl)-2-butynyl]oxy-delta2-isoxazoline iodide 3-[4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl]benzoic acid methyl ester 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxy-delta2-isoxazoline sesquifumarate 3-[4-(2-Methyl-1H-imidazol-1-yl)-2-butynyl]oxyisoxazole sesquifumarate 3-[4-(2-Methyl-3-(4-bromobenzyl)-1H-imidazolium-1-yl)-2-butynyl]oxyisoxazole bromide 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(3-Aminopropoxy)-3-bromophenyl]-N-[2-(4-chlorophenyl)ethyl]-2- hydroxyiminopropanamide 3-[4-(3-Fluorophenylethynyl)-2-thiazolyl]-2-propyn-1-ol 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Es... 3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylami... 3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole 3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-4-methoxy-1H-indole 3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole 3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-7-methoxy-1H-indole 3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 3-[4-(4-Phenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quino-lin-4(3H)-one 3-[4-(4-Pyrimidin-2-ylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-cyclohexyl]-1H-indole-5-carbonitrile 3-[4-(methylsulfonyl)phenyl]-5-(trifluoromethyl)(2-pyridyl) phenyl ketone 3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 3-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butoxy]isoquinoline 3-[5-(4-Isobutoxybenzoyl)-2-propoxyphenyl]propionic Acid 3-[5-[(2-Methyl-4-thiazolyl)ethynyl]-3-pyridyl]-2-propyn-1-ol 3-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyloxy]isoquinoline 3-[6-(2,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[6-(2-Fluorophenyl)-pyridazin-4-yl]benzonitrile 3-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[6-(4-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclo-hexyl]-1H-indole 3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclohexyl]-2-methyl-1H-indole 3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-1H-indole 3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-2-methyl-1H-indole 3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine 3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine 3-[[3-(5-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide 3-[[3-(7-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide 3-[[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl]-1H-indole 3-[[4-[[(2S)-1-(1,2,4-triazol-1-yl)propan-2-yl]amino]piperidin-1-yl]methyl]phenol 3-{(1,4-cis)-4-[(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine 3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-isopropyl-1H-indole-5-carbonitrile 3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile 3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile 3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-pipera-zin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile 3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile 3-{(1,4-trans)-4-[4-(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine 3-{(4-(Pyrimidin-2-yl)piperazin-1-yl)methyl}-1H-pyrrolo[2,3-b]pyridine 3-{(Cyclopropylmethyl)[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Cyclopropylmethyl)[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Cyclopropylmethyl)[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Cyclopropylmethyl)[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid 3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid Methyl Ester 3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(3,4-dihydroisoquinoline) 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(2'-methoxyphenyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(2'-pyrimidyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3'-chlorophenyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3'-methyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3'-trifluoromethylphenyl)piperazine 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(4'-fluorophenyl)piperazine 3-{2-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]ethyl}-1H-indole 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide 3-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl}-3,4-dihydro-1(2H)-naphthalenone 3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(2-Methylphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 3-{2-[4-(2-Pyridinyl)-1-piperazinyl]ethyl}-3,4-dihydro-1(2H)-naphthalenone 3-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(3-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 3-{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]ethyl}-2-methyl-1H-indole 3-{2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}-8-methylpyr-imido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{2-[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]ethyl}-3,4-dihydro-1(2H)-naphthalenone 3-{2-[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]ethyl}-7-methoxy-3,4-dihydro-1(2H)-naphthalenone 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-4-fluoro-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-5-fluoro-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-5-methoxy-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-5-methyl-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-6-fluoro-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-7-fluoro-1H-indole 3-{3-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-7-methyl-1H-indole 3-{3-[4-(2-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8-meth-ylpyrimido[5,4-c]-quinolin-4(3H)-one 3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-9-meth-ylpyrimido[5,4-c]-quinolin-4(3H)-one 3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(2-Methylphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(3-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]propyl}-1H-indole 3-{3-[4-(4-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(4-Fluorophenyl)piperazin-1-yl]propyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(4-Fluorophenyl)piperazin-1-yl]propyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(4-Fluorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{3-[4-(4-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-Amino-5-[4-(3-m-tolylureido)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N,N-dimethylpropionamide 3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N-methylpropanamide 3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}propanamide 3-{4-[(1,4-cis)-4-(1H-Indol-4-yl)-pipera-zinyl-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile 3-{4-[(1,4-trans)-4-(1H-indol-4-yl)-pipera-zinyl-1-yl]cyclohexyl}-1H-indole-5-carbonitrile 3-{4-[2-(4-Aminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol 3-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol 3-{4-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]butyl}-1H-indole 3-{4-[4-(2-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(2-Methylphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]-8-methylpyr-imido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]-9-methylpyr-imido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]butyl}-1H-indole 3-{4-[4-(4-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{4-[4-(4-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one 3-{5-[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]pentyl}-1H-indole 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N,N-dimethylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-isopropylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-propylchromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxylic Acid 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-(cyclopropylmethyl)-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopentyl-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopropyl-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-ethyl-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide 3-{Cyclobutyl[3-(5-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(6-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[3-(7-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{Cyclobutyl[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide 3-{[(1S)-1-(4-Bromophenyl)ethyl]amino}-6-chloro-4H-thieno-[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 3-{[(1S)-2-(4,5-diphenyl-1,3-oxazol-2-yl)-2-cyclohexen-1-yl]methyl}benzoic acid 3-{[3-(5-Fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide 3-{[4-(2,3-Dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]methyl}-1H-indole 3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine 3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-5,7-dimethylimidazo[1,2-c]pyrimidine 3-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole 3-{[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]methyl}-1Hpyrrolo[2,3-b]pyridine 3-{[4-(4-Chlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine 3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}2,5,7-rimethylimidazo[1,2-c]pyrimidine 3-{[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]methyl}-3,4-dihydro-1(2H)-naphthalenone 3-{[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]methyl}-6,7-dimethoxy-3,4-dihydro-1(2H)-naphthalenone 3-{[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]methyl}-6-methoxy-3,4-dihydro-1(2H)-naphthalenone 3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3- carbonyl]-amino}-butyric acid 1-ethyl-1-me... 3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid 1-ethyl-1-m... 3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid 1-isobutyl-... 3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid ethyl ester 3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-propionic acid tert-butyl ... 30 30a 30b 30m 30n 30o 30p 31 31 (ZK 93423) 31a 31b 32 32 (abecarnil) 32a 32b 32D-W-NPY 33 33a 33b 33bMet 34 34a 34b 35 36 37 38 39 3a 3alpha-(4-Methoxyphenyl)-2alpha-(4-methylphenyl)tropane 3alpha-(4-Methylphenyl)-2beta-(3,4-dimethoxyphenyl)tropane 3alpha-Hydroxy-3beta-octyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-phenyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-phenylethyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-phenylmethyl-5alpha-androstan-17-one 3alpha-Hydroxy-3beta-propyl-5alpha-androstan-17-one 3alpha-Phenyl-2alpha-(4-methylphenyl)tropane 3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline 3′′-F-DPPy 3b 3b-(4-chlorophenyl)-2b-[3-(4-methylphenyl)-isoxazol-5-yl]tropane 3b-(4-methylphenyl)-2b-[3-(4-chlorophenyl)-isoxazol-5-yl]tropane 3beta-(4'-Methylphenyl)-2beta-(3,4-dimethoxyphenyl)tropane 3beta-(4-Methoxyphenyl)-2beta-(4-methylphenyl)tropane 3beta-(p-chlorophenyl)tropane-2beta-carboxylic acid methyl ester 3beta-(p-methylphenyl)tropane-2beta-carboxylic acid methyl ester 3beta-4-ChloroBZT 3beta-Cyclohexyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-Cyclohexylethyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-Cyclohexylmethyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-n-Butyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-n-Hexyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-Phenyl-2beta-(4-methylphenyl)tropane 3beta-s-Butyl-3alpha-hydroxy-5alpha-androstan-17-one 3beta-tert-Butyl-3alpha-hydroxy-5alpha-androstan-17-one 3c 3C4HPG 3CTMP 3CTMPNMe 3d 3e 3f 3FLB 3g 3h 3H-GR113808 3HPG 3i 3j 3k 3l 3m 3PPP(+/-) 3PPP,(+) 3PPP,(-) 3PPP,(R) 3PPP,(S) 3R)-1-[(2R)-2-(4-phenylpiperazin-1-yl)propanoyl]piperidine-3-carboxamide 4 4 (3EBC) 4'deoxy EM-A enolether 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 4, 9-DB-3-4-3 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 4,4'-DifluoroBZT 4,4-Dimethyl-1-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)- thio)propyl)piperidine 4,5-Dimethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 4,5-Dimethyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 4,5a-Epoxy-3-methoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)oxy]morphinan-6-one 4,5a-Epoxy-5Beta,17-dimethyl-14Beta-[(3-phenylpropyl)oxy]3-[(prop-2-ynyl)oxy]morphinan-6-one 4,5alpha-Epoxy-3-hydroxy-5beta,17-dimethyl-14beta-[(3-phenylpropyl)oxymorphinan-6-one 4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine 4,6-bis(2-fluorophenyl)pyrimidin-2-amine 4,6-bis(2-methoxyphenyl)pyrimidin-2-amine 4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine 4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine 4,6-bis(4-chlorophenyl)pyrimidin-2-amine 4,6-bis(4-fluorophenyl)pyrimidin-2-amine 4,6-bis(4-methoxyphenyl)pyrimidin-2-amine 4,6-bis(acetylphenyl)pyrimidin-2-amine 4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine 4,6-di(furan-2-yl)pyrimidin-2-amine 4,6-di(furan-3-yl)pyrimidin-2-amine 4,6-di(thiophen-2-yl)pyrimidin-2-amine 4,6-di(thiophen-3-yl)pyrimidin-2-amine 4,6-di-p-tolylpyrimidin-2-amine 4,6-diphenylpyrimidin-2-amine 4,6-distyrylpyrimidin-2-amine 4-((1-Bromo-2-naphthyl)methyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid 4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxyphenol 4-((4-Chlorophenyl)(2,4-dichlorophenyl)methyl)-N-cyclohexylpiperazine-1-carboxamide 4-((5S)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-8-yl)morpholine 4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxy-N-(quinuclidin-3-yl)benzofuran-2-carboxamide 4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-N-(2-(dimethylamino)ethyl)-7-methoxybenzofuran-2-carboxamide 4-((6aS,10aR)-4,5,7,8,10,10a-Hexahydro-6aH-pyrido[4,3-b]pyrrolo[3,2,1-hi]indol-9-yl)-1-(4-Fluoro-phenyl)-butan-1-one 4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one 4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one ( 4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-thia-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)-butan-1-one 4-((6bR,10aS)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone 4-((6bR,10aS)-3-benzyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1... 4-((6bR,10aS)-3-benzyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1... 4-((6bR,10aS)-3-Butyl-2,3,6b,9,10,10ahexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-b... 4-((6bR,10aS)-3-Ethyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-... 4-((6bR,10aS)-3-Isopropyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl... 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4,4-difluoro-piper... 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-b... 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-phenyl-butan-1-one 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-phenyl-butan-1-one ... 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-ph... 4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fl... 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-( 4-pyridinyl)-1-b... 4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-( 4-pyridinyl)-1-b... 4-((6bR,10aS)-5-Bromo-3-methyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorop... 4-((6bR,10aS)-5-Methoxy-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluor... 4-((6bS,10aR)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone 4-((6bS,10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-bu... 4-((6bS,10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-bu... 4-((7aR,11aS)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-buta... 4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-buta... 4-((8aS,12aR)-4,5,6,7,9,10,12,12a-Octahydroazepino[3,2,1-hi]pyrido[4,3-b]-indol-11(8aH)-yl)-1-(4-fluorophenyl)-1-butanone 4-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonit... 4-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-6-ylcarbamoyl)-butyric acid 4-(1-(1-(1H-indol-3-yl)propan-2-yl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(2-methoxyethyl)pyrimidin-2-amine 4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(3-methoxypropyl)pyrimidin-2-amine 4-(1-(2-(1H-pyrazol-4-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(5-chloro-1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-(benzo[b]thiophen-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine 4-(1-(2-bromo-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 4-(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 4-(1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)morpholine 4-(1-hydroxy-2-(4-(4-hydroxyphenyl)butan-2-ylamino)ethyl)phenol 4-(1-hydroxy-2-(methylamino)ethyl)-1,2-benzenediol 4-(1-phenylcyclohexyl)morpholine 4-(1H-Benzimidazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)butan-1-one 4-(1H-imidazol-1-yl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzamide 4-(1H-indol-4-yloxy)-1-(cyclohexylamino)butan-2-ol 4-(1H-indol-4-yloxy)-1-(isopropylamino)butan-2-ol 4-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)morpholine 4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine 4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine 4-(2,2-Diphenyl-1-ethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-(2,2-Diphenylethyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(2,4-Dichloro-5-methoxyanilino)-7-methoxy-8-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyanilino)-8-methoxy-7-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyphenylamino)-7-[2-(4-hydroxypiperidin-1-yl)ethoxy]-8-methoxybenzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloro-5-methoxyphenylamino)-8-[2-(4-hydroxypiperidin-1-yl)ethoxy]-7-methoxybenzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloroanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,4-Dichloroanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2,5-dichlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide 4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexanol 4-(2-((4-fluoro-2-methoxybenzyl)amino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride 4-(2-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-morpholine Hydrochloride 4-(2-((6-Methyl2-phenylpyrimidin-4-yl)oxy)ethyl)morpholine 4-(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-ylsulfonyl)morpholine 4-(2-(2-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)ethoxy)ethyl)- morpholine 4-(2-(2-Hydroxybenzylamino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride 4-(2-(3,4-Dimethylphenylamino)ethyl)-1H-imidazole 4-(2-(3-tert-Butylphenylamino)ethyl)-1H-imidazole 4-(2-(4-Cyclohexylphenylamino)ethyl)-1H-imidazole 4-(2-(4-Methoxyphenylamino)ethyl)-1H-imidazole 4-(2-(4-Methylphenylamino)ethyl)-1H-imidazole 4-(2-(4-tert-Butylphenylamino)ethyl)-1H-imidazole 4-(2-(4-Trifluoromethylphenylamino)ethyl)-1H-imidazole 4-(2-(Benzo[d][1,3]dioxol-4-ylmethylamino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride 4-(2-(Cyclohexylamino)ethyl)-1H-imidazole 4-(2-(Phenylamino)ethyl)-1H-imidazole 4-(2-acetylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-amino-1-hydroxyethyl)-1,2-benzenediol 4-(2-Amino-propyl)-2,5-dimethoxy-phenol 4-(2-aminoethyl)-1,2-benzenediol 4-(2-Aminoethyl)pyrocatechol 4-(2-aminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Azepan-1-ylethyl)-3-(phenylsulfonyl)-1H-indole 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 4-(2-Biphenyl)-N-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-piperazinehexanamide 4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 4-(2-butylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-carboxamidophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Chloro-4-fluoro-5-methoxyanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2-Chloro-5-methoxy-4-methylanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(2-Chloro-5-methoxy-4-methylanilino)-8-[2-(4-hydroxypiperidin-1-yl)ethoxy]-7-methoxybenzo[g]quinoline-3-carbonitrile 4-(2-chlorobenzoyl)-1H-pyrrole-2-carboxamide 4-(2-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(2-chlorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(2-chlorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(2-chlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(2-chlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(2-chlorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 4-(2-cyanophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-dimethylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-(2-ethylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-fluorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(2-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(2-fluorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(2-fluorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(2-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 4-(2-Fluorophenylethynyl)-2-methylthiazole 4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-(2-methoxyphenyl)-N-(6-methylpyridin-2-yl)picolinamide 4-(2-Methoxyphenylethynyl)-2-methylthiazole 4-(2-methylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-methylsulfonamidophenyl)-N-(1,2,3,tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-(2-Naphthylmethyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(2-Naphthylmethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-(2-nitrophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)cyclohexanol 4-(2-Phenylethyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(2-propylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-pyridinyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(2-pyridinyl-N-oxide)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-(3′-Fluorophenethyl)-4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecan-3-ol 4-(3′-Fluorophenyl)methyl-4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecan-3-ol 4-(3,3-Diphenyl-1-propyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-(3,3-Diphenylpropyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(3,4-Dichlorophenyl)-1-methylpiperidine-4-carbonitrile 4-(3,4-Dichlorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(3,4-dichlorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dichlorophenyl)-7-((1-isopropylpiperidin-4-yl)methoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dichlorophenyl)-7-((1-isopropylpiperidin-4-yl)methoxy)-2-methyl-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-dichlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(3,4-dichlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl) butan-1-one hydrochloride 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl) butan-1-one hydrochloride 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride, 4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one 4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one 4-(3,4-dimethoxyphenyl)-2-(5-((R)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1... 4-(3,4-dimethoxyphenyl)-2-(5-((S)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1... 4-(3,5-difluorophenyl)-N-(6-methylpyridin-2-yl)picolinamide 4-(3,5-Difluorophenylethynyl)-2-methylthiazole 4-(3- f 4-[2-(2-Fluoroethoxy)-phenyl]-piperazin-1-yl g -propoxy)-4- aza-tricyclo[5.2.1.02,6]dec-8-ene-3,5-dion 4-(3- f 4-[2-(3-Fluoroethoxy)-phenyl]-piperazin-1-yl g -propoxy)-4- aza-tricyclo[5.2.1.02,6]dec-8-ene-3,5-dion 4-(3- f 4-[2-(4-Fluoroethoxy)-phenyl]-piperazin-1-yl g -propoxy)-4- aza-tricyclo[5.2.1.02,6]dec-8-ene-3,5-dion 4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)propyl)-2-methoxyphenol 4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)propyl)benzene-1,2-diol 4-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)morpholine 4-(3-(3,5-Dimethylpiperidin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 4-(3-(4-(piperidin-1-yl)but-1-ynyl)benzyl)morpholine 4-(3-(4-Boc-piperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 4-(3-(4-Ethylpiperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 4-(3-chloro-4-methoxyphenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(3-chlorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3-chlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 4-(3-Chlorophenylethynyl)-2-methylthiazole 4-(3-cyanophenyl)-N-(6-methylpyridin-2-yl)picolinamide 4-(3-fluorophenyl)-N-(6-methylpyridin-2-yl)picolinamide 4-(3-Fluorophenylethynyl)-2-methylthiazole 4-(3-Fluorophenylethynyl)-2-thiazolylamine 4-(3-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 4-(3-methoxyphenyl)-N-(6-methylpyridin-2-yl)picolinamide 4-(3-Methoxyphenylethynyl)-2-methylthiazole 4-(3-Phenylpropyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester 4-(3-piperidin-1-yl-propoxy)-benzonitrile 4-(3-piperidin-1-ylpropoxy)benzonitrile 4-(3-Pyridylethynyl)-2-thiazolylamine 4-(4,4-Diphenylbutyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(4-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)piperazin-1-yl)indolin-2-one 4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)butyl)morpholine 4-(4-((phenethylamino)methyl)phenoxy)benzamide 4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Ac... 4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid 4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid 4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid 4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate 4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid 4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol 4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 4-(4-(2-Methoxyphenyl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide 4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile 4-(4-(3-((methylamino)methyl)-4-(4-(methylthio)phenoxy)phenyl)but-3-ynyl)piperazin-2-one 4-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)benzonitrile 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 4-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-1-phenylbutan-1-one 4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(4-chloropyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid 4-(4-(5-chloropyridin-2-yl)piperazin-1-yl)-1-(4-fluorophenyl)butan1-one 4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 4-(4-(difluoromethoxy)phenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(4-(pyridine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(pyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(pyrimidine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid 4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol 4-(4-([1,1’-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol 4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-N-phenylbenzamide 4-(4-aminobenzenesulfonyl)-1-NP 4-(4-Bromo-2-chlorophenylamino)-5,6-dichloro-N-(2-hydroxyethoxy)nicotinamide 4-(4-Bromo-2-chlorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-6-methoxynicotinamide 4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-5-fluoro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 4-(4-chloro-3-fluorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Chloro-5-methoxy-2-methylanilino)-7-methoxy-8-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-5-methoxy-2-methylanilino)-7-methoxy-8-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-5-methoxy-2-methylanilino)-8-methoxy-7-[2-(4-methyl-1-piperazinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-5-methoxy-2-methylanilino)-8-methoxy-7-[2-(4-morpholinyl)ethoxy]benzo[g]quinoline-3-carbonitrile 4-(4-Chloro-phenyl)-1-(1H-indol-3-ylmethyl)-piperidin-4-ol 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(3-phenoxypropyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4,4-diphenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-(3,4-dichlorophenyl)-4-phenylbutyl)piperidin-4-ol Hydrochloride 4-(4-Chlorophenyl)-1-(4-(4-chlorophenyl)-4-phenylbutyl)piperidin-4-ol 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-(4-methoxyphenyl)-4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-cyano-4,4-diphenylbutyl)-4-hydroxy-1-methylpiperidinium Iodide 4-(4-Chlorophenyl)-1-(4-hydroxy-4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-(4-phenyl-4-m-tolylbutyl)piperidin-4-ol Hydrochloride 4-(4-Chlorophenyl)-1-(4-phenyl-4-p-tolylbutyl)piperidin-4-ol Hydrochloride 4-(4-Chlorophenyl)-1-(4-phenylbutyl)piperidin-4-ol 4-(4-Chlorophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Chlorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-Chlorophenyl)-1-pyrid-2-yl-pyrazole 4-(4-chlorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion 4-(4-chlorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(4-chlorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(4-Chlorophenyl)-5-(2,4-dichlorophenyl)-N-(piperidin-1-yl)thiazolecarboxamide 4-(4-chlorophenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(4-chlorophenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Chlorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 4-(4-ethoxyphenyl)-7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinoline 4-(4-Fluorophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Fluorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Easter 4-(4-Fluorophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-fluorophenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion 4-(4-fluorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(4-fluorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione 4-(4-Fluorophenyl)-N-[4-methoxy-3-(4-methyl-1-piperazinyl)phenyl]-1-piperazinecarboxamide 4-(4-Fluorophenylethynyl)-2-methylthiazole 4-(4-Idophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 4-(4-Iodophenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Iodophenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)ethyl)azetidin-2-one 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(pyridin-4-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(thiazol-2-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(trifluoromethyl)piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline 4-(4-methoxyphenyl)-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-methoxyphenyl)-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine 4-(4-Methylphenyl)-1-methylpiperidine-4-carbonitrile 4-(4-Methylphenyl)-1-methylpiperidine-4-carboxylic Acid Ethyl Ester 4-(4-Phenylbenzyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol 4-(5-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)-N,N-dimethylanil... 4-(5-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)pentyl)morpholine 4-(5-(Phenoxymethyl)isoxazol-3-yl)morpholine Hydrochlor-ide 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepane TFA 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazine TFA 4-(5-Methyl-7-oxo-6,7-dihydro-thiazolo[5,4-d]pyrimidin-2- yl)-benzoic acid 4-(6-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)hexyl)-2-methoxyphenol 4-(6-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)hexyl)morpholine 4-(6-(4-chlorophenyl)-2,6-diazabicyclo[2.2.1]heptan-2-yl)-1-(4-fluorophenyl)butan-1-one 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzamide 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoic Acid 4-(6-methoxy-2-(4-methoxyphenyl)benzofuran-3-carbonyl)benzonitrile 4-(6-Phenylpyridazin-4-yl)benzonitrile 4-(7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-1,2,3,4-tetrahydroisoquinolin-4-yl)benzonitrile 4-(8-benzyl-5-cyano-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-propylpiperazine-1-carboxamide 4-(8-Chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-1-ethylpiperazine N-oxide 4-(8-Chloro-5H-dibenzo[b,e][1,4]diazepin-11-yl)-1-isopropylpiperazine N-oxide 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine TFA 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazine TFA 4-(9-Anthracylmethyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(adamantan-1-ylamino)-1-(1H-indol-4-yloxy)-butan-2-ol 4-(Bis(2-bromoethyl)amino)-2,3,5-trifluorobenzoic Acid 4-(Bis(2-bromoethyl)amino)-3,5-difluorobenzoic Acid 4-(Bis(2-chloroethyl)amino)-2,3,5,6-tetrafluorobenzoic Acid 4-(Bis(2-chloroethyl)amino)-2,3,5-trifluorobenzoic Acid 4-(Bis(2-chloroethyl)amino)-3,5-difluorobenzoic Acid 4-(Bis(2-iodoethyl)amino)-2,3,5,6-tetrafluorobenzoic Acid 4-(Bis(2-iodoethyl)amino)-2,3,5-trifluorobenzoic Acid 4-(Bis(2-iodoethyl)amino)-3,5-difluorobenzoic Acid 4-(Cyclohexylmethyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(Diacetylamino)-l-ethyl-[ 1,2,4]triazolo[4,3-a]quinoxaline 4-(diethylamino) [ 1,2,4]triazolo[4,3-a]quinoxaline 4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 4-(Dimethylamino)-N-(4-(9-(2-methoxyphenyl)-3,9-diazaspiro- [5.5]undecan-3-yl)butyl)benzamide 4-(Dimethylaminomethyl)-6-methoxy-1,2,3,4-tetrahydrocarbazole Oxalate 4-(Diphenylmethyl)-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzamide 4-(N-(2-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(3,4-dichlorophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-acetylphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-benzyloxyphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-biphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-bromophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-chlorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-ethyloxycarbonylphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfona mide 4-(N-(4-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-nitrophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-(4-phenoxyphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-fluorenylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(N-phenylsulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide 4-(naphthalen-1-yl)-N-(6-methylpyridin-2-yl)picolinamide 4-(naphthalen-2-yl)-N-(6-methylpyridin-2-yl)picolinamide 4-(rel-(6bR, 10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoropheny... 4-(rel-(6bS,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl... 4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile 4-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)isoquinoline 4-({4-(2-[4-(2,3-Dichlorophenyl)iperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline 4-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl) isoquinoline 4-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline 4-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline 4-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline 4-({4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazin-1-yl}carbonyl)morpholine 4-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)isoquinoline 4-({[4-(2,4-Diamino-6-ethylpyrimidin-5-yl)phenyl]amino}methyl)benzonitrile 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 4-acetoxy-N,N-diallyltryptamine 4-allyloxy-2,5-dimethoxyamphetamine 4-allyloxy-2,5-dimethoxyphenethylamine 4-Amino Phosphonobutyrate 4-Amino-1-(2-hydroxy-3-nonyl)pyrazolo[3,4-d]pyrimidine 4-Amino-1-(beta-hydroxyethyl)pyrazolo[3,4-d]pyrimidine 4-amino-2-decylpyrazolo[3,4-d]pyrimidine 4-Amino-3-bromo-1-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrazolo[3,4-d]pyrimidine 4-Amino-3-bromo-1-alpha-L-lyxofuranosylpyrazolo[3,4-d]pyrimidine 4-Amino-4'-hydroxystilbene 4-Amino-5-bromo-7-(5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-bromo-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(4'-C-spirocyclopropyl-beta-D-erythro-pentofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(5-O-methyl-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-Amino-5-iodo-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine 4-Amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-Aminobutanoic acid 4-aminobutanoic acid 4-Aminobutyric acid 4-ARA-127 4-benzenesulfonyl-1-NP 4-benzhydryl-N-butylpiperazine-1-carboxamide 4-benzhydryl-N-cyclohexylpiperazine-1-carbothioamide 4-benzhydryl-N-cyclohexylpiperazine-1-carboxamide 4-benzoyl-1-NP 4-benzyl-1-NP 4-Benzyl-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-Benzyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-benzyloxy-2,5-dimethoxyphenethylamine 4-bromo-1-NP 4-Bromo-2,5-dimethoxyphenethylamine 4-Butyl-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-carboxybenzenesulfonamide 4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine 4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine 4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine 4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine 4-chloro-3-(trifluoromethyl)phenyl (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-c... 4-chloro-3-(trifluoromethyl)phenyl (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-benzyl-1-oxo-7-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-benzyl-7-(2-methoxyphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-benzyl-7-ethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-benzyl-7-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-cyclohexyl-1-oxo-7-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-cyclohexyl-7-(2-methoxyphenyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylat... 4-chloro-3-(trifluoromethyl)phenyl 2-cyclohexyl-7-ethyl-6-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-cyclohexyl-7-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 2-cyclohexyl-7-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 3-benzyl-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 3-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 7-(2-methoxyphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 7-(4-methoxyphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 7-ethyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 7-isopropyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-(trifluoromethyl)phenyl 7-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-chloro-3-hydroxy-dibenz[d,g]azecine 4-Chloro-3-{3-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 4-Chloro-N-(1,2,3,4-tetrahydro-1,3,4-trioxoisoquinolin-6-yl)butanamide 4-chloro-N-(6-methylpyridin-2-yl)picolinamide 4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-10,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}... 4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide 4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl]-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptylamino]-methy... 4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl][4-(1,2,3,4-tetrahydroacridin-9-ylamino)butylamino]methylen... 4-ChloroBZT 4-Cl-KYNA 4-CPP 4-cyano-1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 4-Cyano-N-ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]benzamide 4-Cyclohexyl-1-(2,4-dimethoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione 4-Cyclohexyl-1-(4-methoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione 4-Cyclohexyl-1-(4-methylbenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione 4-Cyclopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 4-Cyclopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 4-DAMP 4-diphenylacetoxy-N-methyl-piperadine 4-Ethyl 2-methyl 3-methyl-5-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)thiophene-2,4-dicarboxylate 4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-((4-methoxyphenyl)amino) thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate 4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate 4-Ethyl-2,5-dimethoxyphenethylamine 4-Ethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 4-Ethyl-2-phenyl6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 4-Ethyl-3-((5-methoxy-1H-indol-3-yl)methyl)1H-1,2,4-triazol-5(4H)-thione 4-Ethyl-3-(2-(5-methoxy-1H-indol-3-yl)ethyl)-1H-1,2,4-triazol-5(4H)-thione 4-Ethyl-5-(4-piperidyl)-3-isoxazolol 4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210) 4-Ethylthio-2,5-dimethoxyphenethylamine 4-Ethylthio-2,5-dimethoxyphenylbutylamine 4-F-DPPy 4-Fluoro-(R)-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 4-Fluoro-(S)-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 4-fluoro-2,3,7,11b-tetrahydro-1H-pyrido[3,4,5-k]acridin-8,9-diol 4-Fluoro-3-(2-dimethylaminoethyl)indole 4-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 4-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 4-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenylthio)benzylamine 4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 4-Fluoro-N-(1-{2-[(propan-2-yl)phenoxy]ethyl}piperidin-4- yl) benzenesulfonamide 4-Fluoro-N-(1-{2-[2-(methylsulfanyl)phenoxy]ethyl} pyrrolidin-3-yl)benzenesulfonamide 4-fluoro-N-(3-(1-(2-(piperidin-1-yl)ethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide 4-fluoro-N-(3-(1-(2-hydroxyethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide 4-fluoro-N-(3-(1-octylpiperidin-4-yl)-1H-indol-5-yl)benzamide 4-fluoro-N-(3-{1-[(2E)-4-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)but-2-en-1-yl]piperidin-4-yl}-1H-indol-5... 4-fluoro-N-(3-{1-[10-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)decyl]piperidin-4-yl}-1H-indol-5-yl)benzamid... 4-fluoro-N-(3-{1-[11-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)undecyl]piperidin-4-yl}-1H-indol-5-yl)benzam... 4-fluoro-N-(3-{1-[12-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)dodecyl]piperidin-4-yl}-1H-indol-5-yl)benzam... 4-fluoro-N-(3-{1-[2-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethoxy)ethyl]piperidin... 4-fluoro-N-(3-{1-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)benzamide 4-fluoro-N-(3-{1-[3,3,3-trifluoro-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-ind... 4-fluoro-N-(3-{1-[3-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-indol-5-yl)benzamid... 4-fluoro-N-(3-{1-[6-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)hexyl]piperidin-4-yl}-1H-indol-5-yl)benzamide 4-fluoro-N-(3-{1-[7-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)heptyl]piperidin-4-yl}-1H-indol-5-yl)benzamid... 4-fluoro-N-(3-{1-[9-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)nonyl]piperidin-4-yl}-1H-indol-5-yl)benzamide 4-Fluoro-N-({1-[2-(3-fluorophenoxy)ethyl]piperidin-4-yl}methyl) benzenesulfonamide 4-Fluoro-N-({1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl} methyl) benzenesulfonamide 4-Fluoro-N-[(1-{2-[2-(propan-2-yl)phenoxy]ethyl}piperidin-4-yl)methyl] benzenesulfonamide 4-Fluoro-N-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-be... 4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-benzamide 4-Fluoro-N-{1-[2-(5,6,7,8-tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 4-Fluoro-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 4-Fluoro-N-{1-[2-(phenoxy)ethyl]pyrrolidin-3-yl}benzenesulfonamide 4-fluoro-N-{3-[1-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethyl)piperidin-4-yl]-1H-... 4-fluoro-N-{3-[1-({3-[(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)methyl]phenyl}methyl)piperidin-4-yl]-1H-ind... 4-Fluoro-N-{[1-(2-(2-isopropoxyphenoxy)ethyl)piperidin-4-yl]methyl}benzenesulfonamide 4-fluorodinapsoline hydrobromide 4-Hexyl-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-HPCA 4-HT 4-Hydrazino-3-chlorobenzenesulfonamide 4-Hydrazino-3-fluorobenzenesulfonamide 4-Hydroxy-1-methylgramine 4-Hydroxy-2,3-dimethyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-2-methyl-5-(2-thienyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-2-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-(2-dimethylaminopropyl)indole 4-Hydroxy-3-(2-pyrrolidin-1-ylethyl)indole 4-Hydroxy-3-(2-thienyl)-5,6,7,8-tetrahydrobenzo[b]thieno[2,3-b]pyridin-2(1H)-one 4-Hydroxy-3-(2-[N-1,2,3,4 tetrahydroquinolino]ethyl)indole 4-Hydroxy-3-(2-[N-methylpiperazino]ethyl)indole 4-Hydroxy-3-(3-dimethylaminopropyl)indole 4-Hydroxy-3-(3-phenoxyphenyl)-1,5,6,7-tetrahydrocyclopenta[4,5]thieno[2,3-b]pyridin-2-one 4-Hydroxy-3-(3-phenoxyphenyl)-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-b]pyridin-2(1H)-one 4-Hydroxy-3-isopropyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methoxymethyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methyl-5-(2-thienyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methyl-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-methyl-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-3-phenylquinolin-2(1H)-one 4-Hydroxy-3-phenylthieno[3,4-b]pyridin-2(1H)-one 4-Hydroxy-5-(3-phenoxyphenyl)thieno[2,3-b]pyridin-6(7H)-one 4-Hydroxy-5-phenylthieno[2,3-b]pyridin-6(7H)-one 4-hydroxy-N,N-diallyltryptamine 4-Hydroxy-N,N-dimethyltryptamine 4-hydroxydinapsoline hydrobromide 4-hydroxyduloxetine 4-hydroxyduloxetine glucuronide 4-hydroxyduloxetine glucuronide 4-Hydroxygramine 4-hydroxytamoxifen 4-iodo-2,5-dimethoxyphenethylamine 4-Iodo-2,5-dimethoxyphenylisopropylamine 4-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide 4-Iodonaphthalen-1-yl-[1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone 4-Iodophenyl-[2-methyl-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]methanone 4-Isopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 4-Isopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 4-MB-3-3 4-Methoxy-2-(dipropylamino)indan 4-Methoxy-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 4-Methoxy-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 4-Methoxy-3-(1-methyl-2-pyrrolidinyl)pyridine 4-methoxy-diphenidine 4-METHOXY-N,N-DIMETHYLTRYPTAMINE 4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benzamide 4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide 4-methoxy-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide 4-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 4-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide 4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide 4-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 4-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide 4-Methoxy-N-[4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-benzamide 4-Methoxy-N-[4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-benzamide 4-methoxybenzyl (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-methoxybenzyl (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-methoxymeridianin A 4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081) 4-Methoxyphencyclidine 4-methoxyphenyl (±)-(4aR,8S,8aR)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 4-METHOXYPHENYLPIPERAZINE 4-Methyl-1-[2-(4-chlorophenoxy)ethyl]piperidine hydrochloride 4-Methyl-1-[3-(4-chlorophenoxy)propyl]piperidine hydrochloride 4-Methyl-2-phenyl-6-(3-(2,2,6,6-tetramethylpiperidin-1-yl)- propoxy)pyrimidine 4-Methyl-2-phenyl-6-(3-(4-phenylpiperazin-1-yl)propoxy)- pyrimidine 4-Methyl-2-phenyl-6-(3-(piperazin-1-yl)propoxy)pyrimidine 4-Methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 4-Methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 4-Methyl-3-phenyl-5-(propylthio)-4H-1,2,4-triazole 4-methyl-3-phenyl-pyrrolidine 4-Methyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 4-Methyl-6-(3-(4-methylpiperazin-1-yl)propoxy)-2-phenylpyrimidine 4-Methyl-6-(3-(4-methylpiperidin-1-yl)propoxy)-2-phenylpyrimidine 4-methylcyclohexylpiperidine 4-methylhistamine 4-methyl[1]benzofuro[3,2-g]quinolin-2-ol 4-MXP 4-N,N'-Dimethylamino-4'-hydroxystilbene 4-N-(2-Methoxyphenyl)amino-5-(4-ethoxyphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3,4-Ethylenedioxyphenyl)amino-5-(2-methylphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3,4-Ethylenedioxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3-Ethoxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(3-Pyridyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Bromophenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Chlorophenyl)amino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Chlorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-(4-chlorophenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-(4-ethoxyphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-(4-methoxyphenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Cyanophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Ethoxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-(3-aminophenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-(4-fluorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(4'-C-spirocyclopropyl-beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Fluorophenyl)amino-5-phenyl-7-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine 4-N-(4-Hydroxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Hydroxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methoxyphenyl)amino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methoxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methoxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(4-Methylphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-(Cyanoyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Benzylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Benzylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Cyclohexylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Cyclohexylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Methylamino-4'-hydroxystilbene, SB-13 4-N-Phenylamino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-iodo-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(2,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(2-deoxy-beta-D-erythropentofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(3,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5'-deoxy-4'-C-methyl-beta-D-ribo-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5-amino-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5-azido-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-5-phenyl-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 4-N-Phenylamino-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 4-N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]piperidine-1,4-dicarboxamide 4-OH-TRYPTAMINE 4-Oxo-4-piperidin-1-yl-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-butyramide 4-oxo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)chromene-2-carboxamide 4-P-ADOT 4-P-CADOT 4-P-PDOT 4-phenyl-1-NP 4-phenyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydro-2,6-naphthyridine 4-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-phenylpiperidine 4-PIOL 4-Piperazino[ 1,2,4]triazolo[4,3-a ]quinoxaline 4-quinolone 4-Sulfamoylbenzoic acid hydrazide 4-TrifluoromethylBZT 4-[(1-Butyl-4-piperidinyl)methoxy]-2-methyl-2H-pyrrolo[3,4-c]- quinoline 4-[(1E)-3-({2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(1-pyrrolidinyl)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl}amino)-3-oxo... 4-[(1E)-3-[[2-[2,4-Dichloro(methyl)-3-({[2-methyl-4-(2-pyridinylmethoxy)-8-quinolinyl]oxy}methyl)anilino]-2-oxoethyl]amino]-3... 4-[(2,4-Dichlorophenyl)(p-tolyl)methyl]-N-piperidin-1-ylpiperazine-1-carboxamide 4-[(2,4-Dichlorophenyl)(phenyl)methyl]-N-piperidin-1-ylpiperazine-1-carboxamide 4-[(2-chloro-4-fluorophenyl)(phenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(2-fluoro-4-chlorophenyl)(phenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(2-fluorophenyl)methyl]-1-[2-(3-methylpyrazol-1-yl)ethyl]piperidine 4-[(2R)-2-hydroxy-3-[4-(pyrazol-1-ylmethyl)piperidin-1-yl]propoxy]benzonitrile 4-[(2R)-2-hydroxy-3-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]propoxy]benzonitrile 4-[(3-chlorophenyl)(2,4-dichlorophenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(3-Fluorophenyl)ethynyl]-2-methyloxazole 4-[(3R)-piperidin-3-yl]oxypyridine 4-[(4-bromo-2-fluorophenyl)(phenyl)methyl]-N-cyclohexylpiperazine-1-carboxamide 4-[(5-Amino-1-benzoyl-1H-1,2,4-triazol-3-yl)amino]-benzenesulfonamide 4-[(Indol-3-yl)methyl]-2-methyl-thiazole 4-[(Indol-3-yl)methyl]thiazole 4-[1-(1,3-benzodioxol-5-yl)cyclohexyl]morpholine 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine 4-[1-(2-methoxyphenyl)cyclohexyl]morpholine 2Me0 4-[1-(3-Methoxyphenyl)cyclohexyl]morpholine 4-[1-(3-methylphenyl)cyclohexyl]morpholine 4-[1-(4-methoxyphenyl)cyclohexyl]morpholine 4-[2-(1,1-dimethylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-[2-(1-methylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide 4-[2-(1-Naphthyl)ethyl]-5-(4-piperidyl)-3-isoxazolol Hydrobromide 4-[2-(1-Pyrrolidinyl)ethyl]-imidazole 4-[2-(1H-Benzimidazol-2-ylsulfanyl)-1-hydroxyethyl]-2-chlorophenol 4-[2-(2-Methylpiperidin-1-yl)ethyl]-3-(phenylsulfonyl)-1H-indole 4-[2-(3,4-Dichloro-phenyl)-acetyl]-3-pyrrolidin-1-ylmethyl-piperazine-1-carboxylic acid methyl ester(GR89696) 4-[2-(3-Methylpiperidin-1-yl)ethyl]-3-(phenylsulfonyl)-1H-indole 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 4-[2-(6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl)ethoxy]benzenesulfonamide 4-[2-(methylsulfonyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-(1-pyrrolidinyl)pyridine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-fluoropyridine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-methylpyridine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine 4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine 4-[2-[(2,3-Dihydro-5,6-dimethoxy-1H-inden-2-yl)propylamino]ethyl]benzamide 4-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 4-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzenemethanol 4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid 4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]phenylacetamide 4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid 4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 4-[3-(2,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 4-[3-(4-Benzhydryl-piperazin-1-yl)-2-hydroxy-propoxy]-1H-indole-2-carbonitrile 4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one 4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one 4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)-1-butanone 4-[3-(4-Phenylpiperazin-1-yl)propoxy]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[3-(4-Phenylpiperazin-1-yl)propoxy]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[3-(4-Phenylpiperazin-1-yl)propyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[3-(4-Phenylpiperazin-1-yl)propyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[3-(m-Bromo-phenyl)-5-methyl-isoxazol-4-yl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 4-[3-(Methylsulfonyl)phenyl]-1-propylpiperidine 4-[3-(o-Bromo-phenyl)-5-methyl-isoxazol-4-yl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 4-[3-(p-Bromo-phenyl)-5-methyl-isoxazol-4-yl]-2,6-dimethyl-1,4-dihydro-pyridine 3,5-dicarboxylic acid 3-ethyl ester 5-(1-phen... 4-[3-(p-bromo-phenyl)-5-methyl-isoxazol-4-yl]-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid diethyl ester 4-[3-[4-( o -Methoxyphenyl)piperazin-1-yl]propoxy]-4-aza-tricyclo- [5.2.1.02,6]dec-8-ene-3,5-dione 4-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-morpholine 4-[4-(2,4-Diamino-6-benzyloxymethyl-pyrimidin-5-yl)-phenoxymethyl]-benzonitrile 4-[4-(2-Pyrimidine)piperazin-1-yl]-1-(4-fluorophenyl)butan-1-one 4-[4-(3-Methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine 4-[4-(4-Benzylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[4-(4-Benzylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one 4-[4-(4-Phenylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-[4-(4-Phenylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-[4-(4-Phenylpiperazinilmetil)-1H-1,2,3-triazol-4-yl]acetamide 4-[4-[4-[hydroxy(diphenyl)methyl]-1-piperidinyl]butyl]benzoic acid 4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one 4-[5-(7-Azabicyclo[2.2.1]hept-2-yl)-2-fluoro-3-pyridinyl]benzonitrile 4-[5-Amino-1-(2,6-difluoro-benzenesulfonyl)-1H-[1,2,4]triazol-3-ylamino]-benzenesulfonamide 4-[5-Amino-1-(2,6-difluoro-benzoyl)-1H-[1,2,4]triazol-3-ylamino]-N-(2-dimethylaminoethyl)-benzenesulfonamide 4-[5-Amino-1-(2,6-difluoro-benzyl)-1H-[1,2,4]triazol-3-ylamino]-benzenesulfonamide 4-[5-trans-hydroxy-5-cis-(4′-chlorophenyl)-2-azabicyclo[3.2.1]octanyl]-4″-fluorobutyrophenone 4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzonitrile Hydrobromide 4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenol Fumarate 4-[6-fluoro-2,2-bis-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-ylmethyl]-morpholine 4-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-6H-pyridazin-1-yl]-butyric acid 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2,4-difluorophenyl)piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2-fluorophenyl)piperazine-1- carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2-fluorophenyl)piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(3,4-difluorophenyl)piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(4-fluorophenyl)piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(cyclohexylmethyl)piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(pyridin-2-yl)piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclohexylpiperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclopentylpiperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-phenylpiperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[(2- fluorobenzene)sulfonyl]piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[1-(trifluoromethyl)cyclopentyl]-piperazine-1-carboxamide 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[6-(difluoromethoxy)pyridin-3-yl]piperazine-1-carboxamide 4-[[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]carbamoylamino]benzamide 4-[[(3R)-3-methoxypiperidin-1-yl]methyl]-5-methyl-2-(3-phenoxyphenyl)-1,3-oxazole 4-[[(3R)-3-phenylpyrrolidin-1-yl]methyl]-2-propan-2-yl-1,3-thiazole 4-[[(3R)-3-phenylpyrrolidin-1-yl]methyl]-2-propyl-1,3-thiazole 4-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methoxy]-2-methyl2H-pyrrolo[3,4-c]quinoline 4-[[1-[2-[4-(Methoxymethyl)phenyl]ethyl]-4-piperidinyl]- methoxy]-2-methyl-2H-pyrrolo[3,4-c]quinoline 4-[[2-[(Dimethylamino)methyl]phenyl]thio]-3-nitrobenzenemethanol 4-[[3-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-5-yl]amino]-benzenesulfonamide 4-[[3-[(dimethylamino)methyl]phenyl]methyliminomethyl]-3-hydroxy-2H-isoquinolin-1-one 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 4-[[5-Amino-1-(2,3,6-trifluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2,6-difluoro-3-methylbenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-(2-thienylcarbonyl)-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-[(3,5-dimethyl-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-[(3-fluoro-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[5-Amino-1-[(3-methyl-2-thienyl)carbonyl]-1H-1,2,4-triazol-3-yl]amino]-benzenesulfonamide 4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]-1- methyl-1-(2-phenylethyl)piperidinium Iodide 4-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}butyric Acid Methyl Ester 4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2'-pyrimidyl)piperazine 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3'-trifluoromethylphenyl)piperazine 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(N-methyl)piperazine 4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(2-Pyridyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{4-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-pyrazol-1-ylmethyl]-2-oxo-pyrrolidin-1-yl}-benzoic acid 4-{4-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-pyrazol-1-ylmethyl]-2-oxo-pyrrolidin-1-yl}-benzonitrile 4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate 4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione 4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate 4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)] undecane-3,5,8-trione 4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate 4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole 4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole 4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-methyl-1H-benzimidazole 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole 4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]piperazin-1-yl}-2-methyl-1H-benzimidazole 4-{[(4-Iodobenzyl)sulfanyl]methyl}-1H-imidazole 4-{[(4-{2,4-Diamino-6-[(benzyloxy)methyl]pyrimidin-5-yl}phenyl)amino]methyl}benzonitrile 4-{[4-(3-{4-[(Benzyl{2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)butanoyl]amino}butanoic Acid 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 40 3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one 40 40 (DMCM) 41 42 43 43a 43b 44 44a 44b 44c 44d 44e 44f 45 45a 45b 46 47 48 49 4a 4a-Benzyl-2-chloroethynyl-1,2,3,4,4a,9,10,10a-octahydro-phenanthrene-2,7-diol(CP-394531) 4a-Benzyl-7-hydroxy-3,4,4a,9,10,10a-hexahydro-1H-phenanthren-2-one 4aH-8, {9c-Iminoethanophenanthro[4,5-bcd]furan-5(6H)-one,} N-allyl-7,7a,8, 9-tetrahydro-3,7a-dihydroxy- 4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aR,9aS-(+)-cis-4a-Ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro-[2,3-c]pyridin-6-ol 4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4aS,9aR-(-)-cis-4a-Ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro-[2,3-c]pyridin-6-ol 4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol 4ATMP 4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline 4‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline 4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic A... 4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-c... 4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-ca... 4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-car... 4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxyli... 4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid 4′′-F-DPPy 4b 4c 4C3HPG 4CPG 4d 4e 4f 4FTMP 4g 4h 4i 4j 4k 4MeTMP 4MeTMPNMe 4OHBA 4OHMNA 4Z,7Z,10Z,13Z,16Z,19Z-Docosahexaenoic acid 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(3,4-dihydroisoquinoline) 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2'-methoxyphenyl)piperazine 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3'-trifluoromethylphenyl)piperazine 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(4'-fluorophenyl)piperazine 5 5'-(Dimethylamino)methyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 5'-(N-ethyl-carbamoyl)adenosine 5'-(N-ethylcarboxamido)adenosine 5'-(Trimethylammonium)methyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]-morphinan Iodi... 5'-Amidinomethyl-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 5'-amino-5'-deoxy- 5-iodotubercidin 5'-benzyl-12'-hydroxy-2'-isopropyl-3',6',18-trioxoergotaman 5'-benzyl-12'-hydroxy-2'-methyl-3',6',18-trioxoergotaman 5'-ChloroAdo 5'-Deoxy-5'-aminoadenosine 5'-Deoxy-5'-iodoado 5'-Deoxy-5'-isobutylthioadenosine 5'-deoxy-5-iodotubercidin 5'-Deoxyadenosine 5'-guanidinonaltrindole 5'-Methylthioado 5'-N-Biguanidino-17-cyclopropylmethyl-6,7-didehydro-4,5alpha-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan 5'-O-Acetylado 5'-O-Nitroado 5(S)-HETE 5, 6-Dehydroarachidonic acid 5,5-Bis-(4-bromo-phenyl)-3-(2-morpholin-4-yl-ethyl)-imidazolidine-2,4-dione 5,5a,6,7,8,10-hexahydro-5,8-methanopyrrolo[2,1-g][1,7]naphthyridin-2-amine 5,6,7,9-Tetrahydro-8H-pyrldo[3,4-c]azepine oxalate 5,6-DHT 5,6-difluoroindol-methylethylamine 5,6-DIHYDROXY TRYPTAMINE 5,6-dihydroxy-2-(N,N-di-n-propylamino)tetralin ((-)-5,6-diOH-DPAT 5,6-DIHYDROXY-DPAT 5,6-Dihydroxyduloxetine glucuronide 5,6-Dihydroxytryptamine 5,6-dimethoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5,6-dimethoxy-1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5,6-dimethoxy-1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5,6-dimethoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)isoindolin-1-one 5,6-Dimethoxy-2-(dibutylamino)indan 5,6-Dimethoxy-2-(dipropylamino)indan 5,6-Dimethoxy-2-[(3-fluoropropyl)propylamino]indan 5,6-Dimethoxy-2-[(butyl)propylamino]indan 5,6-Dimethoxy-2-[(methylcyclopropyl)propylamino]indan 5,6-Dimethoxy-3-methyl-N-phenyl-N-(3-(piperidin-1-yl)propyl)benzofuran-2-carboxamide (KSCM-1) 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone 5,6-Dimethyl-2-pyridin-2-yl-1H-benzoimidazole 5,6-Dimethyl-2-thiazol-4-yl-1H-benzoimidazole 5,6-methylenedioxy-2-aminoindan 5,7,8,9,9a,10-hexahydro-7,10-methanopyrrolo[1,2-b][2,6]naphthyridin-3-amine 5,7-DCKA 5,7-DHT 5,7-diethyl-2-phenylthieno[2,3-d]pyridazin-4(5H)-one 5,7-DIHYDROXY TRYPTAMINE 5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine 5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-N,N,6-trimethyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine 5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazol-2(3H)-one 5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazole-2(3H)-thione 5-((5-Methoxy-1H-indol-3-yl)methyl)-3-methyl-1,2,4-oxadiazole 5-(1,2,3,4-Tetrahydro-acridin-9-ylamino)-pentanoic acid [3-(acridin-9-ylsulfanyl)-propyl]-amide 5-(1,4,4-trimethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1H- pyrrole-2-carbonitrile 5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole 5-(1-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole 5-(1-Ethyl-propyl)-1-(4-methoxy-2-methyl-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5-(1-Ethyl-propyl)-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5-(1-Ethyl-propyl)-7-methyl-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5-(1-Ethylpropyl)-7-methyl-1-(2-methyl-4-trifluoromethoxyphenyl)-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene Hydrochloride 5-(1-Ethynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(1-Hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(1-Methoxymethyl-propyl)-1-(4-methoxyphenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5-(1-Methyl-2-pyrrolidinyl)-2-(2-phenylethyl)pyridine 5-(10-Hydroxy-1-decynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (1,5-dimethyl-hexyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (1-methyl-hexyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (2-diisopropylcarbamoyl-1-methy... 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (3,3-dimethyl-butyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid (3-tert-butoxy-propyl)-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid diisobutylamide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid isobutyl-amide 5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carboxylic acid isobutyl-methyl-amide 5-(2,2,2-Trifluoroacetyl)-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide 5-(2-(5-Methoxy-1H-indol-3-yl)-3-methyl-1,2,4-oxadiazole 5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazol-2(3H)-one 5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazole-2(3H)-thione 5-(2-Azetidnylmethoxy)-2-Chloropyridine, (R) 5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl 5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5-(2-isopropylidene)-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 5-(2-methoxyphenyl)-N-(6-methylpyridin-2-yl)picolinamide 5-(2-morpholinoethyl)-2-phenyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 5-(2-Phenyl-1-ethynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole 5-(2-tert-butoxycarbonylamino-ethylamino)-2- furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid 5-(2-tert-Butoxycarbonylamino-ethylamino)-2-furan-2-yl-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxylic acid ethyl ester 5-(3,4-dimethoxy-benzylamino)-2-furan-2-yl- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid benzhydryl-amide 5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 5-(3,5-dimethyl-piperidine-1-sulfonyl)-3-methyl-benzofuran-2-carboxylic acid 4-methyl-benzylamide 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzofuran-2-carboxamide 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide 5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethyl-N-phenethylbenzofuran-2-carboxamide 5-(3-Bromophenyl)-3-ethoxy pyridazine 5-(3-Bromophenyl)-3-isopropoxypyridazine 5-(3-Bromophenyl)-3-methoxypyridazine 5-(3-Bromophenyl)-3-phenyl pyridazine 5-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine 5-(3-Chlorophenyl)-2-methyl-1,3-benzothiazole 5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 5-(3-cyanophenyl)-N-(6-methylpyridin-2-yl)picolinamide 5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 5-(3-Hydroxy-1-propargyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(3-Hydroxy-3-methyl-1-butynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 5-(3-Methoxyphenyl)-2-methyl-1,3-benzothiazole 5-(3-methoxyphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine   5-(4,4-diethyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile 5-(4,4-Dimethyl-2-thioxo-1,4-dihydro-2H-3, 1-benzoxazin-6-yl)-1H-pyrrole-2-carbonitrile 5-(4-((phenethylamino)methyl)phenoxy)picolinamide 5-(4-(3,4-Dichlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one, 5-(4-(3-Chloro-4-trifluoromethylphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole 5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole 5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline 5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid 5-(4-(4-Bromophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Chlorophenyl)piperazin-1-yl)-2,2-diphenypentanenitrile 5-(4-(4-Chlorophenyl)piperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(4-Methoxyphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-(Diphenylmethylene)piperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Aminophenyl)-6-methylthieno[2,3-d]pyrimidin-4-amine 5-(4-Benzyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Bromophenyl)-1-(2,4-dichlorophenyl)-N-(4-methylpiperazin-1-yl)-1H-pyrazole-4-carboxamide 5-(4-Bromophenyl)-N-cycloheptyl-1-(2,4-dichlorophenyl)-1H-pyrazole-4-carboxamide 5-(4-Bromophenyl)-N-cyclopropyl-1-(2,4-dichlorophenyl)-1H-pyrazole-4-carboxamide 5-(4-Butyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide 5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide 5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide 5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(1-isopropyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(1-isopropyl-5-methyl-1H-imidazol-4-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(2-isopropyl-1H-imidazol-5-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-(5-isopropyl-1H-imidazol-2-yl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4,5-dihydro-1H-pyrazole-3-carboxylic acid morpholin-4-ylamide bisulphate salt 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylsulfinyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylthio)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylthio)-N-(pyrrolidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-(1-(2-phenylpropan-2-yl)-1H-imidazol-4-yl)-1H-pyrazole 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(7-(N-(1-phenethylpiperidin-4-yl)propionamido)heptyl)-1H-pyrazole-3-carb... 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(4-methylpiperazin-1-yl)-1H-pyrazole-4-carboxamide 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-1,2,4-triazole-3-carboxamide Dihydrochloride 5-(4-chlorophenyl)-3-(1-cyclobutyl-1H-imidazol-4-yl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole 5-(4-chlorophenyl)-3-(1-cyclohexyl-1H-imidazol-4-yl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole 5-(4-Chlorophenyl)-4-(2,4-dichlorophenyl)-N-(piperidin-1-yl)thiazolecarboxamide 5-(4-chlorophenyl)-4-cyano-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide 5-(4-Chlorophenyl)-N-cyclopropyl-1-(2,4-dichlorophenyl)-1H-pyrazole-4-carboxamide 5-(4-ethyl-4-methyl-2-thioxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile 5-(4-Fluorophenyl)-2-methyl-1,3-benzothiazole 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Hydroxy-4-p-tolylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride 5-(4-Hydroxy-4-phenylpiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-Hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile 5-(4-Methoxy-2-pyrimidinyl)-2-methyl-1,3-benzothiazole 5-(4-Piperidyl)-4-(1-naphthylmethyl)-3-isoxazolol Hydrobromide 5-(4-Piperidyl)-4-octyl-3-isoxazolol Hydrobromide 5-(4-Piperidyl)-4-propyl-3-isoxazolol Hydrobromide 5-(4-Piperidyl)-4-propylisothiazol-3-ol Hydrobromide 5-(4-Piperidyl)-4-[2-(2-naphthyl)ethyl]-3-isoxazolol Hydrobromide 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis... 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (tra... 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 5-(4-{[3,5-Difluoro-4-(methylsulfonyl)benzyl]amino}phenyl)-6-ethylpyrimidine-2,4-diamine 5-(5-methylthiophen-2-yl)-N-(4-morpholin-4-ylbutyl)-1H-pyrazole-3-carboxamide 5-(6-Fluoro-1-hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(6-Hydroxy-1-hexynyl)-3-(1-methyl-2(S)-pyrrolidinylmethoxy)pyridine 5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5-(GSyl)-alpha-MethylDopamine 5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methyl-2-butenyl)dihydro-2(3H)-furanone 5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methylbutyl)dihydro-2(3H)-furanone 5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5-(N-Ethyl)amino-5,0,7,8-tetrahydroquinoline maleate 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 5-(Phenoxymethyl)-3-(piperazin-1-yl)isoxazole Hydrochlor-ide 5-(Phenoxymethyl)-3-(piperidin-1-yl)isoxazole Hydrochlor-ide 5-(Phenoxymethyl)-3-(piperidin-4-ylmethoxy)isoxazole Tri-fluoroacetate 5-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-(2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-(2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline 5-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)quinoline 5-2-Azetidnylmethoxy)-2-Chloropyridine, (R) 5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-6-oxa-1-aza-chrysene-9-carboxylic acid methyl ester 5-Amino-2-thiazol-4-yl-1H-benzimidazol 5-amino-3-(N-methylpiperidin-4-yl)-1H-indole 5-Amino-3-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carboamide 5-Amino-3-[[4-(aminosulfonyl)phenyl]amino]-N-(2,6-difluorophenyl)-1H-1,2,4-triazole-1-carbothioamide 5-Amino-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-Amino-7-(thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-Amino-7-(thiophen-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-aminomethyl-(5H)-dibenzo[a,d]-cycloheptenehydrochloride 5-aminomethyl-10,11-dihydro-5(H)-dibenzo[a,d]-cycloheptadiene 5-Aminosalicylic acid 5-APB 5-APT 5-Benzoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-Benzoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-benzyl-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 5-benzyl-7-chloro-2-cyclohexyl-2H-pyrazolo[4,3-c]quinolin-3(5H)-one 5-Benzyloxytryptamine 5-Br-T 5-Br-T, 1-Isopropyl 5-Bromo-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 5-bromo-2-(((1R)-3-bromo-2,2-dimethyl-6-methylenecyclohexyl)methyl)-4-methoxyphenol 5-bromo-2-(((1S)-3-bromo-2,2-dimethyl-6-methylenecyclohexyl)methyl)-4-methoxyphenol 5-Bromo-2-((R)-2,2-dimethyl-6-methylene-cyclohexylmethyl)-4-methoxy-phenol 5-bromo-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 5-Bromo-3-(1-methyl-2-pyrrolidinyl)pyridine 5-Bromo-3-(2(S)-azetidinylmethoxy)pyridine 5-bromo-4-methoxy-2-(((1S)-2,2,5-trimethyl-6-methylenecyclohexyl)methyl)phenyl acetate 5-Bromo-4-methoxy-2-((1S,4R)-2,2,4-trimethyl-6-methylene-cyclohexylmethyl)-phenol 5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide 5-bromo-N,N-diallyltryptamine 5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-Bromotryptamine 5-Butyl-1-(4-chloro-2-cyanophenyl)-7-methyl-1,3,4,5-tetrahydro-1,5,8-triazaacenaphthylene 5-Butyl-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide 5-BZT 5-carboxamidotryptamine 5-Carboxyamido Tryptamine 5-Carboxyamido Tryptamine, Dipropyl 5-carboxyl-2,4-di-benzamidobenzoic acid 5-Chlor-2-thiazol-4-yl-1H-benzimidazol 5-Chloro-(R)-N-(1-{2-[(propan-2-yl)-phenyloxy]ethyl} pyrrolidin-3-yl)thiophene-2-sulfonamide 5-Chloro-(R)-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3- yl}thiophene-2-sulfonamide 5-Chloro-(S)-N-(1-{2-[(propan-2-yl)-phenyloxy]ethyl} pyrrolidin-3-yl)thiophene-2-sulfonamide 5-Chloro-(S)-N-{1-[2-(biphenyl-2-yloxy)ethyl]pyrrolidin-3- yl}thiophene-2-sulfonamide 5-Chloro-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide 5-Chloro-1H-indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide 5-Chloro-2,4-dimethyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 5-chloro-2-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide 5-chloro-2-(1-(3-ethoxy-4-fluorobenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide 5-chloro-2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazole-6-sulfonamide 5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride 5-Chloro-2-(3,4-dichlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine 5-Chloro-2-(3,4-difluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride 5-Chloro-2-(4-chlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 5-Chloro-2-(4-fluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 5-Chloro-2-(4-methoxyphenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine 5-Chloro-2-cyclopropyl-4-methyl-6-(3-(piperidin-1-yl)propoxy)-pyrimidine 5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide 5-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]piperidin-4-yl}benzenesulfonamide 5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide 5-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide 5-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide 5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide 5-Chloro-2-pyridin-2-yl-1(3)H-benzoimidazole 5-Chloro-2-[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]thio]benzothiazole 5-Chloro-2-[[3-[4-(2-methoxyphenyl)-1-piperazinyl]propyl]thio]benzoxazole 5-Chloro-3-(2(S)-azetidinylmethoxy)pyridine 5-Chloro-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole 5-Chloro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-Chloro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-Chloro-3-{3-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 5-Chloro-4-methyl-2-(naphthalen-2-yl)-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 5-Chloro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 5-Chloro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(4- (trifluoromethyl)phenyl)pyrimidine 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(p-tolyl)-pyrimidine 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine 5-Chloro-N-(1-{2-[(propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)thiophene-2-sulfonamide 5-Chloro-N-(1-{2-[2-(methylsulfanyl)phenoxy]ethyl}pyrrolidin-3-yl)thiophene-2-sulfonamide 5-Chloro-N-({1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl}methyl)thiophene-2-sulfonamide 5-Chloro-N-{1-[2-(2,3-dichlorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 5-Chloro-N-{1-[2-(2,5-dichlorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 5-Chloro-N-{1-[2-(biphenyl-2-yloxy)ethyl]piperidin-4-yl}thiophene-2-sulfonamide 5-Chloro-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}thiophene-2-sulfonamide 5-Chloro-N-{1-[2-(phenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide 5-Chlorotryptamine 5-Cl-T 5-CT 5-CT,DP 5-CT,N,N-DiMe 5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methoxy)-benz... 5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-(prop-2-ynyloxy)benzamide 5-cyano-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-6-methylpyridine-2-carboxamide 5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 5-dimethoxy-4-(b-methallyl)thio-phenethylamine 5-ethyl-1-hydroxy-3-(3-prop-2-enoxyphenyl)imidazo[5,1-a]phthalazin-6-one 5-ethyl-3-(1-methyl-2-pyrrolidinyl)pyridine 5-Ethyl-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-Ethyl-7-(thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-Ethyl-7-(thiophen-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-Ethyl-7-phenylthieno[2,3-d]pyridazin-4(5H)-one 5-F-6-F3C, 1-(1-indolinyl)-2-propylamines 5-F-6-I, 1-(1-indolinyl)-2-propylamines 5-F-T 5-Fluor-2-thiazol-4-yl-1H-benzimidazol 5-Fluoro-2-[(2-methyl-4-thiazolyl)ethynyl]pyridine 5-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 5-Fluoro-3-[(1,4-cis)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole 5-Fluoro-3-[(1,4-trans)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole 5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole 5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole 5-Fluoro-3-{cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole 5-Fluoro-3-{trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole 5-fluoro-4-((R)-1-(3-fluorophenyl)ethoxy)-N-((R)-pyrrolidin-3-yl)pyrimidin-2-amine 5-fluoro-4-((R)-1-(3-fluorophenyl)ethoxy)-N-((S)-pyrrolidin-3-yl)pyrimidin-2-amine 5-fluoro-4-((R)-1-(4-fluorophenyl)ethoxy)-N-((R)-pyrrolidin-3-yl)pyrimidin-2-amine 5-Fluoro-4-((R)-1-(4-fluorophenyl)ethoxy)-N-((S)-pyrrolidin-3-yl)pyrimidin-2-amine 5-Fluoro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 5-Fluoro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine 5-fluoro-4-[(4-fluorophenyl)methoxy]-2-[(2R)-2methylpiperazin-1-yl]pyrimidine 5-fluoro-N,N-diallyltryptamine 5-Fluoro-N,N-dimethyl-2-(2-amino-4-methylphenoxy)benzylamine 5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide 5-Fluorotryptamine 5-Fluorowillardiine-(S) 5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-HMMP 5-HPCA 5-HT 5-HT, alpha,Omega-dimethyl 5-HT,1-Me 5-HT,2-Me 5-HT,20Me 5-HT,a-Me 5-HT,a-Me-,S(+) 5-HT,b-Me 5-HT,N,N-DIMETHYL 5-HT,N,N-DIPROPYL 5-HT,N-ACETYL 5-HT,o-N 5-HT,omega-N-Me 5-HT,x-Me 5-HT7 5-HTP dipeptide 5-HTQ 5-Hydroxy Tryptamine 5-HYDROXY TRYPTAMINE, 1-Me 5-Hydroxy Tryptamine, 2-Me 5-Hydroxy Tryptamine, Alpha-methyl 5-HYDROXY TRYPTAMINE, b-Me 5-HYDROXY TRYPTAMINE, Omega-N-Me 5-Hydroxy-6-(3-phenoxyphenyl)-3,4-dihydro-2H,8H-1,9-dithia-8-azafluoren-7-one 5-hydroxy-6-methoxyduloxetine 5-hydroxy-6-methoxyduloxetine glucuronide 5-hydroxy-6-methoxyduloxetine sulfate 5-Hydroxy-N,N-dimethyl-1-(benzenesulfonyl)tryptamine 5-HYDROXY-N,N-DIMETHYLTRYPTAMINE 5-hydroxyduloxetine 5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isobutyl-5-methyl-hexanoyloxymethyl)tetrahydro-2-furanone 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 5-hydroxypentanoic acid 5-I-aminoindane 5-iod-2-aminoindane 5-iodo-2-aminoindane 5-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 5-Isopropyl-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5-Isopropyl-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 5-M-DMT 5-M-N,N-DMT 5-MCA-NAT 5-ME-URAPIDIL 5-MeO-TMT 5-MeOT 5-MeOT,N,N tryptamine 5-MeOT,N,N-DIPROPYL 5-MeOT-N-butanyl 5-MeOT-N-hexanyl 5-MeOT-N-pentanyl 5-MeOT-N-propionyl 5-MET 5-methoxy-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5-Methoxy-1-(2-propyl)-DMT Maleate 5-methoxy-1-methyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5-methoxy-1-propyl-1,2,3,7,12,12a-hexahydro-1-aza-pleiadene 5-Methoxy-1-[(5-phenyl-3-pyridyl)carbamoyl-6-triflouromethylindoline 5-Methoxy-1-[[2-methyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[2-[(3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(2,4-dimethyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(2-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(2-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[3-(4-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[4-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[4-(4-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[4-methyl-3-(3-pyridyl)phenyl]carbamoyl]-5-methoxy-6-trifluoromethylindoline 5-Methoxy-1-[[4-methyl-3-(4-methyl-3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(4-fluorophenyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(4-methyl-3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-(4-pyridyl)-3-pyridyl]carbamoyl-6-trifluoromethylindoline 5-Methoxy-1-[[5-fluoro-4-methyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[5-phenyl-3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-1-[[6-(3-pyridyl)-3-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate 5-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one 5-Methoxy-2-(dipropylamino)indan 5-Methoxy-2-aminoindan 5-methoxy-2-fluoro-N,N-diallyltryptamine 5-methoxy-2-methyl-N,N-diallyltryptamine 5-Methoxy-2-n-propyl-DMT Oxalate 5-Methoxy-2-phenyl-DMT Oxalate 5-Methoxy-3-(di-n-propylamino)chroman 5-METHOXY-3-[2-(DIMETHYLAMINO)ETHYL]INDOLE 5-Methoxy-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-Methoxy-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole 5-methoxy-6-methyl-2-aminoindan 5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 5-methoxy-N,N-diallyltryptamine 5-Methoxy-N,N-diethyl-1-(4-acetamidobenzenesulfonyl)tryptamine 5-Methoxy-N,N-diethyl-1-(4-aminobenzenesulfonyl)tryptamine 5-Methoxy-N,N-diethyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N,N-diisopropyltryptamine 5-Methoxy-N,N-dimethyl-1-(4-acetamidobenzenesulfonyl)tryptamine 5-Methoxy-N,N-dimethyl-1-(4-aminobenzenesulfonyl)tryptamine 5-Methoxy-N,N-dimethyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N,N-Dimethyltryptamine 5-Methoxy-N-benzyl-N-methyl-1-(4-aminobenzenesulfonyl)tryptamine 5-Methoxy-N-benzyl-N-methyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N-methyl-1-(benzenesulfonyl)tryptamine 5-Methoxy-N-methyl-N-isopropyltryptamine 5-Methoxytryptamine 5-Methyl-(3R)-3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-hexanoic aci... 5-Methyl-(3S)-3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-hexanoic aci... 5-Methyl-1-[[2-{(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-6-trifluoromethylindoline 5-methyl-10-(1,2,3,6-tetrahydro-1-methyl-4-pyridinyl)-5H-dibenzo[a,d]cycloheptene 5-methyl-10-(4-methylpiperazino)-5H-dibenzo[a,d]cycloheptene 5-Methyl-2,6-diphenyl[1,3]thiazolo[4,5-b]pyridine 5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-on 5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 5-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 5-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-phenyl-1H-imidazo[4,5-b]pyridine 5-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one 5-Methyl-2-phenyl[1,3]thiazolo[4,5-b]pyridine 5-Methyl-2-pyridin-2-yl-1(3)H-benzoimidazol 5-Methyl-2-thiazol-4-yl-1(3)H-benzoimidazole 5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 5-Methyl-3-{[5-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}-hexanoic acid ter... 5-Methyl-4,5,6,7,9,10-hexahydropyrido[4,3:2,3]indolo[7,1-ab][3]benzazepine 5-Methyl-N,N-Dimethyltryptamine 5-methyl-N-[3-[4-(3-methylphenyl)piperazin-1-yl]propyl]-1H-pyrazole-4-carboxamide 5-methyl-urapidil 5-Methylthio-1-[[3-(3-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methylthio-1-[[3-(4-pyridyl)phenyl]carbamoyl]-6-trifluoromethylindoline 5-Methyltryptamine 5-Methylurapidil 5-MOT 5-MPEP 5-MT 5-NH2T 5-Nitro-2-pyridin-2-yl-1(3)H-benzoimidazol 5-Nitro-2-thiazol-4-yl-1(3)H-benzoimidazole 5-Nitro-N-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-isophthalamic acid methyl ester 5-OBzlTRYPTAMINE 5-OH-DMT 5-OH-ME-Nw Tryptamine 5-OME-3-ADTN 5-Phenyl-4-N-phenylamino-7-(5-amino-5-deoxy-alpha-L- lyxofuranosylpyrrolo[2,3-d]pyrimidine 5-Phenyl-4-N-phenylamino-7-(5-deoxy-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine 5-Phenyl-4-N-phenylamino-7-(5-O-methyl-alpha-L-lyxofuranosyl)pyrrolo[2,3- d]pyrimidine 5-Phenyl-4-N-phenylamino-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine 5-Propyl-5-normetazocine 5-tert-Butyl-2-pyridin-2-yl-1H-Benzoimidazole 5-tert-Butyl-2-thiazol-4-yl-1H-benzimidazol 5-[(2(S)-Azetidinyl)methoxy]-3-(fluoromethyl)isoxazole Trifluoroacetate 5-[(2(S)-Azetidinyl)methoxy]-3-(phenoxymethyl)isoxazole 5-[(2(S)-Azetidinyl)methoxy]-3-isoxazolylmethanol 5-[(2(S)-Azetidinyl)methoxy]-3-methylisoxazole 5-[(2(S)-Azetidinyl)methoxy]-3-[(4-fluoroanilino)methyl]isoxazole 5-[(2(S)-Azetidinyl)methoxy]-3-[(N-cyclopentylcarbamoyloxy)methyl]isoxazole 5-[(2(S)-Azetidinyl)methoxy]-3-[(N-ethylcarbamoyloxy)methyl]isoxazole 5-[(2(S)-Azetidinyl)methoxy]-3-[(N-phenylcarbamoyloxy)methyl]isoxazole 5-[(2-Methyl-4-thiazolyl)ethynyl]-1H-indole 5-[(2-Methyl-4-thiazolyl)ethynyl]-2-vinylpyridine 5-[(2-Methyl-4-thiazolyl)ethynyl]pyrimidine 5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(Z)-3-isobutyl-5 -methylhexylidene]tetrahydro-2-furanone 5-[(Z)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine 5-[3-(3,5-Difluoropyridin-2-yl)-4-fluorophenyl]-3-(2,4,6-trifluorophenyl)pyridazine 5-[3-(3,5-Difluoropyridin-2-yl)-4-fluorophenyl]-3-(3-fluoropyridin-2-yl)pyridazine 5-[3-(3,5-Difluoropyridin-2-yl)-4-fluorophenyl]-3-(3-fluoropyridin-4-yl)pyridazine 5-[3-(3,5-Difluoropyridin-2-yl)-4-fluorophenyl]-3-(4-fluorophenyl)pyridazine 5-[3-(3,5-Difluoropyridin2-yl)-4-fluorophenyl]-3-(2-fluorophenyl)pyridazine 5-[3-Bromo-4-(4-methanesulfonyl-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 5-[3-Chloro-4-(4-methanesulfonyl-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 5-[3-[3-(3,5-dimethylpyrazol-1-yl)azetidin-1-yl]propyl]-3-phenyl-1,2,4-oxadiazole 5-[4-(1,3-Benzoxazol-2-ylamino)phenyl]-6-methylthieno[2,3-d]pyrimidin-4-amine 5-[4-(2-Amino-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(2-Bromo-ethyl)-piperazin-1-yl]-5-[4-(4-bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-5-[4-(4-iodo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-5-[4-(4-methoxy-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-piperazin-1-yl-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-carboxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-2-thioxo-dihydro-pyrimidine-4,6-dione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(3-iodo-benzoyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-fluoro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-iodo-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-nitro-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(4-trimethylsilyl-phenyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-5-[4-(isopropyl)-piperazin-1-yl]-pyrimidine-2,4,6-trione 5-[4-(4-Bromo-phenoxy)-phenyl]-pyrimidine-2,4,6-trione 5-[4-(4-Chloro-benzylamino)-phenyl]-6-ethyl-pyrimidine-2,4-diamine 5-[4-(4-Chloro-benzylamino)-phenyl]-6-phenethyl-pyrimidine-2,4-diamine 5-[4-(Benzylamino)phenyl]-6-[(benzyloxy)methyl]pyrimidine-2,4-diamine 5-[4-Fluoro-3-(3,5-difluoropyridin-2-yl)-phenyl]-3-(3,5-difluoropyridin-4-yl)pyridazine 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3,5-difluoropyridin-2-yl)pyridazine 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3,5-difluoropyridin-2-yl)pyridazine5-[4-Fluoro-3-(3,5-difluoropyridin-2-yl)-p... 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3-fluoropyridin-2-yl)pyridazine 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)-phenyl]-3-(3-fluoropyridin-4-yl)pyridazine 5-[4-Fluoro-3-(3-fluoropyridin-2-yl)phenyl]-3-(2-fluorophenyl)- pyridazine 5-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2-dihydropyridin-2-one Hydrobromid... 5-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-indole Hydrochloride 5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid 5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-(3,4-dihydroisoquinoline) 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2'-methoxyphenyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2'-pyrimidyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(3'-chlorophenyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(4'-fluorophenyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(N-methyl)piperazine 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 5-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline 5-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline 5-{4-[(2-Chloro-pyridin-4-ylmethyl)-amino]-phenyl}-6-ethyl-pyrimidine-2,4-diamine 5-{4-[(5-Chloro-thiophen-3-ylmethyl)-amino]-phenyl}-6-ethyl-pyrimidine-2,4-diamine 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (ci... 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (tr... 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid 5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester 50 50a 50b 51 51a 51b 52 52a 52b 53 53a 53b 54 54a 54b 55 55a 55b 56 56a 56b 57 58 5a 5’-Bromo-4’-OMethyl-HEAT HCl 5’-Iodo-HEAT HCl 5′-Chloro-5′- deoxy-N6 -(±)-endo-norbornyl-adenosine 5′-Chloro-5′- deoxy-N6 -(±)-endo-norbornyl-adenosine (5′Cl5′d-(±)-ENBA 5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine 5b 5c 5d 5e 5f 5g 5h 5i 5j 5k 5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol 5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16-triol 5Z,8Z,11Z,14Z,17Z-eicosapentaenoic acid 6 6'-methylepibatidine 6, PHPNECA 6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 6,7 di-Chloro-2-methylmelatonin 6,7,8,9-Tetrahydro-2-methoxy-10-(N,N-dimethylaminoethyl)pyrido[1,2-a] indole Oxalate 6,7-Di(1H-imidazol-1-yl)-2,3(1H,4H)-quinoxalinedione 6,7-dichloro-3-(hydroxyimino)indolin-2-one 6,7-Didehydro-4,5alpha-epoxy-5'-guanidinyl-17-methyl-3,14-dihydroxyindolo[2',3':6,7]morphinan 6,7-dimethoxy-2-((7-methoxy-2-(2-(trifluoromethyl)phenyl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 6,7-dimethoxy-2-((7-methoxy-2-(3-methoxyphenyl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 6,7-dimethoxy-2-((7-methoxy-2-(pyridin-2-yl)benzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 6,7-dimethoxy-2-((7-methoxy-2-phenylbenzofuran-4-yl)methyl)-1,2,3,4-tetrahydroisoquinoline 6-(((6-chloro-4H-1,3-benzodioxin-8-yl)methyl)thio)-3-(cyclopropylmethyl)-1,2,3,4-tetrahydro-1,3,5-triazine 6-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)oxy)- 3,4-dihydroquinolin-2(1H)-one 6-(1,2,3,4-Tetrahydro-acridin-9-ylamino)-hexanoic acid [3-(acridin-9-ylsulfanyl)-propyl]-amide 6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline 6-(1H-1,2,4-Triazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-2-Ethylimidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-2-Methylimidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-4,5,6,7-Tetrahydrobenzimidazol-1-yl)-7-nitro-2,3-(1H,4H)-quinoxalinedione 6-(1H-4-Methylimidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-4-Nitroimidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-4-Phenylimidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-Benzimidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-Benzoimidazol-2-yl)-pyridin-2-ol 6-(1H-imidazol-1-yl)-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)-4-oxobutyl)pyridazin-3(2H)-one 6-(1H-imidazol-1-yl)-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-imidazol-1-yl)-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)-4-oxobutyl)pyridazin-3(2H)-one 6-(1H-imidazol-1-yl)-2-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-imidazol-1-yl)-2-(4-(4-(pyrimidin-2-yl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-Imidazol-1-yl)-7-(trifluoromethyl)-2,3(1H,4H)-quinoxalinedione 6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-Imidazol-1-yl)-8-nitro-2,3(1H,4H)-quinoxalinedione 6-(1H-Imidazol-4-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione Hydrochloride 6-(1H-indol-1-yl)-2-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-indol-1-yl)-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-indol-1-yl)-2-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-indol-1-yl)-2-(4-(4-(pyrimidin-2-yl)piperazin-1-yl)butyl)pyridazin-3(2H)-one 6-(1H-Pyrazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione 6-(2,3-Cl2-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2,3-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2,3-Difluorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2,3-F2-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2,4-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2,4-Difluorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2,5-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2,6-Cl2-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2,6-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2-(2-ethylbutyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(2-morpholinoethyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(3,3-dimethylbutyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(3-cyclohexylpropyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(3-morpholinopropyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(3-phenylpropyl)-1,2,3,4-tetrahydroisoquinolin-6-yloxy)nicotinamide 6-(2-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-amine 6-(2-(4-methylpentyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-(5-methylhexyl)-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-benzyl-1,2,3,4-tetrahydroisoquinolin-6-yloxy)nicotinamide 6-(2-benzyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)nicotinamide 6-(2-benzylisoindolin-5-yloxy)nicotinamide 6-(2-Bromobenzenesulfonyl)-2H-pyridazin-3-one 6-(2-butyl-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-CF3-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2-Chloro-4-fluorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2-Chlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2-Cl-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2-F-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2-Fluorobenzenesulfonyl)-2H-pyridazin-3-one 6-(2-hexyl-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-Hexyl-5-hydroxyphenoxy)hexanoic Acid (2-Hydroxyethyl)amide 6-(2-Hexyl-5-hydroxyphenoxy)hexanoic Acid Cyclopropylamide 6-(2-isopentyl-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-pentyl-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-phenethyl-1,2,3,4-tetrahydroisoquinolin-6-yloxy)nicotinamide 6-(2-phenethyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)nicotinamide 6-(2-phenethyl-2,3,4,5-tetrahydro-1H-benzo[c]azepin-7-yloxy)nicotinamide 6-(2-phenethylisoindolin-5-yloxy)nicotinamide 6-(2-Phenylethyl)nicotine 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 6-(2Cl,6F-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2F,3-CF3-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2F,3-Cl-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(2F,4Br-phenylmethanesulfonyl)-2H-pyridazin-3-one 6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene 6-(3,5-Dimethylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(3-benzyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)nicotinamide 6-(3-CF3-phenylmethanesulfonyl-2H-pyridazin-3-one 6-(3-Chlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(3-Chlorophenyl)-5-methyl-2-phenyl[1,3]thiazolo[4,5-b]pyridine 6-(3-Hydroxy-4-hexylphenoxy)hexanoic Acid (2-Hydroxyethyl)amide 6-(3-Hydroxy-4-hexylphenoxy)hexanoic Acid Cyclopropylamide 6-(3-Hydroxy-5-pentylphenoxy)hexanoic Acid Cyclopropylamide 6-(3-Methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(3-phenethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)nicotinamide 6-(3-Phenylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane 6-(3-Trifluoromethylbenzenesulfonyl)-2H-pyridazin-3-one 6-(3-[4-Fluorophenyl]benzofuran-2-methylsulfonyl)-2H-pyridazin-3-one 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6-(4-((benzylamino)methyl)phenoxy)nicotinamide 6-(4-((phenethylamino)methyl)phenoxy)nicotinamide 6-(4-((phenethylamino)methyl)phenoxy)pyridine-3-sulfonamide 6-(4-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenoxy)nicotinamide 6-(4-(2-(3-phenylpropylamino)ethyl)phenoxy)nicotinamide 6-(4-(2-(benzylamino)ethyl)phenoxy)nicotinamide 6-(4-(2-(benzylamino)ethyl)phenoxy)nicotinic acid 6-(4-(2-(benzylamino)ethyl)phenoxy)nicotinonitrile 6-(4-(2-(benzylamino)ethyl)phenoxy)picolinamide 6-(4-(2-(methylthio)phenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 6-(4-(2-(phenethylamino)ethyl)phenoxy)nicotinamide 6-(4-(2-acetylphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 6-(4-(2-hydroxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 6-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide 6-(4-(3-(benzylamino)propyl)phenoxy)nicotinamide 6-(4-(3-(phenylamino)propyl)phenoxy)nicotinamide 6-(4-(3-phenylpropylamino)phenoxy)nicotinamide 6-(4-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butoxy)phenyl)-5,6-dihydroimidazo[2,1-b]thiazole 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6-(4-Bromo-2-fluorobenzenesulfonyl)-2H-pyridazin-3-one 6-(4-Bromobenzenesulfonyl)-2H-pyridazin-3-one 6-(4-Chlorobenzenesulfonyl)-2H-pyridazin-3-one 6-(4-Fluorobenzenesulfonyl)-2H-pyridazin-3-one 6-(4-Fluorophenyl)-5-methyl-2-phenyl[1,3]thiazolo[4,5-b]pyridine 6-(4-Methoxybenzenesulfonyl)-2H-pyridazin-3-one 6-(4-Trifluoromethylbenzenesulfonyl)-2H-pyridazin-3-one 6-(5,6-Methylenedioxyindole-2-sulfonyl)-2H-pyridazin-3-one 6-(5,7-Dichlorobenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5,7-Dichloroindole-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chloro-3-ethylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chloro-3-isopropylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chloro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chloro-3-methylbenzothiophene-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chloro-3-phenylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chlorobenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Fluoro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Methoxybenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(5-Methylbenzothiophene-2-sulfonyl)-2H-pyridazin-3-one 6-(6-Chloro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(6-chloro-3-pyridinyl)-2,6-diazabicyclo[3.2.1]octane 6-(6-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one 6-(6-chloropyridin-3-yl)-1,6-diazaspiro[3.4]octane 6-(6-Fluoroindole-2-sulfonyl)-2H-pyridazin-3-one 6-(7-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one 6-(alpha-Naphthylmethylbenzenesulfonyl)-2H-pyridazin-3-one 6-(Benzofuran-2-sulfonyl)-2H-pyridazin-3-one 6-(Benzothiazole-2-sulfonyl)-2H-pyridazin-3-one 6-(Benzothiophene-2-sulfonyl)-2H-pyridazin-3-one 6-(beta-Naphthylmethylbenzenesulfonyl)-2H-pyridazin-3-one 6-(Biphenylyl-2-sulfonyl)-2H-pyridazin-3-one 6-(cyclopropylmethyl)-1,2-dimethoxy-4-phenyl-5,6,6a,7-tetrahydro-4H- [1,3]dioxolo[4,5:4,5]benzo[1,2-g]benzo[de]quinoline 6-(Indole-2-sulfonyl)-2H-pyridazin-3-one 6-(morpholine-4-carbonyl)-2,2-diphenyl-benzo[1,3]dioxole-5-carbonitrile 6-(N,N-di-n-propylamino)-3,4,5,6,7,8-hexahydro-2H-naphthalen-1-one 6-(N,N-Di-n-propylamino)-3,4,5,6,7,8-hexahydro-2H-naphthalen-1-one O-Methyloxime 6-(N,N-Di-n-propylamino)-3,4,5,6,7,8-hexahydro-2H-naphthalen-1-one Oxime 6-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)-5,6, 7,8-tetrahydronaphthalen-1-ol 6-(pyridin-3-yl)-1,6-diazaspiro[3.4]octane 6-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 6-AcDHM 6-allyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-one 6-amino-1-(2-phenylethyl)-2-thioxo-2,3-dihydro-4(1H)-pyrimidinone 6-amino-1-[(3-methoxyphenyl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione 6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 6-aminonicotine 6-APB 6-APT 6-Benzoyl-9-cyclohexyl-6,9-diazaspiro[4.5]decane-8,10-dione 6-benzyl-2-(benzyloxy)-8-butyl-6,8-diaza-bicyclo[3.2.2]nonane 6-benzyl-2-(benzyloxy)-8-phenethyl-6,8-diaza-bicyclo[3.2.2]nonane 6-benzyl-2-methoxy-8-phenethyl-6,8-diaza-bicyclo[3.2.2]nonane 6-Benzyl-3-ethoxycarbonyl-4-quinolone 6-Benzyl-3-propoxycarbonyl-4-quinolone 6-Benzyl-3-propylaminocarbonyl-4-quinolone 6-benzyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-one 6-benzyl-8-butyl-2-methoxy-6,8-diaza-bicyclo[3.2.2]nonane 6-benzyl-8-butyl-6,8-diaza-bicyclo[3.2.2]nonan-2-ol 6-Benzyloxymethyl-5-[4-(4-chloro-benzylamino)-phenyl]-pyrimidine-2,4-diamine 6-Benzyloxymethyl-5-[4-(4-trifluoromethyl-benzylamino)-phenyl]-pyrimidine-2,4-diamine 6-Benzyloxymethyl-5-{4-[(4-chloro-phenylamino)-methyl]-phenyl}-pyrimidine-2,4-diamine 6-Benzyloxymethyl-5-{4-[(5-chloro-thiophen-2-ylmethyl)-amino]-phenyl}-pyrimidine-2,4-diamine 6-Benzyloxymethyl-5-{4-[(5-chloro-thiophen-3-ylmethyl)-amino]-phenyl}-pyrimidine-2,4-diamine 6-Benzyloxymethyl-5-{4-[(quinolin-3-ylmethyl)-amino]-phenyl}-pyrimidine-2,4-diamine 6-Benzylthioinosine 6-Bromo-3-(1-methylcyclopropyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Bromo-3-ethoxycarbonyl-2-methyl-4-quinolone 6-Bromo-3-ethoxycarbonyl-4-quinolone 6-Bromo-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 6-Bromo-5-methyl-2-phenyl[1,3]thiazolo[4,5-b]pyridine 6-Bromonicotine 6-Chloro-2-methylmelatonin 6-Chloro-3-(1-methyl-1-phenylethyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Chloro-3-(1-methylcyclopropyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Chloro-3-(1-phenylcyclopropyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Chloro-3-(2,2,2-trifluoroethyl)amino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Chloro-3-(N-ethyl-N-methyl)aminomethylpyridine oxalat 6-chloro-3-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine 6-Chloro-3-isopropylamino-4H-thieno[2,3-e]-1,2,4-thiadiazine1,1-Dioxide 6-Chloro-3-[1-(3-chlorophenyl)cyclobutylamino]-4H-thieno-[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Chloro-3-[1-(4-methoxyphenyl)cyclopropyl]amino-4H-thieno-[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-Chloro-3-{3-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 6-Chloro-3-{[1-(trifluoromethyl)cyclopropyl]amino}-4H-thieno-[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide 6-chloro-4-N-[1-[(2-fluorophenyl)methyl]piperidin-4-yl]pyrimidine-2,4-diamine 6-Chloro-5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]indoline 6-Chloro-5-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-1,... 6-chloro-N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]thiazol-2-amine 6-chloro-N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine 6-chloro-N-[(2R)-2-(4-phenylpiperazin-1-yl)propyl]pyrazin-2-amine 6-chloro-N-[2-[4-(3-methylphenyl)piperazin-1-yl]ethyl]pyrazin-2-amine 6-chloro-N-[2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl]pyrazin-2-amine 6-chloro-N-[3-(4-phenylpiperazin-1-yl)propyl]pyrazin-2-amine 6-chloro-N-[3-[4-(2-fluorophenyl)piperazin-1-yl]propyl]pyrazin-2-amine 6-chloro-N-[4-(4-phenylpiperazin-1-yl)butyl]pyrazin-2-amine 6-Chloromelatonin 6-Cl, 1-(1-indolinyl)-2-proylamines 6-Cl-5-F, 1-(1-indolinyl)-2-propylamines 6-cyanonicotine 6-desoxonaltrexone 6-desoxycodeine 6-desoxymorphine 6-Dimethylamino-4,4-diphenyl-3-heptanone 6-dimethylamino-4,4-diphenyl-heptan-3-one 6-dimethylamino-4,4-diphenyl-heptan-3-one, (-) 6-ethyl-1,2-dimethoxy-4-phenyl-5,6,6a,7-tetrahydro-4H-[1,3]dioxolo[4,5:4,5]benzo[1,2- g]benzo[de]quinoline 6-ethyl-3-(1-methyl-2-pyrrolidinyl)pyridine hydrochloride 6-Ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone 6-Ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 6-Ethyl-3-(3-pentoxycarbonyl)-4-quinolone 6-Ethyl-3-(4-methyl-2-pentoxycarbonyl)-4-quinolone 6-Ethyl-3-i-propoxycarbonyl-4-quinolone 6-Ethyl-3-pentoxycarbonyl-4-quinolone 6-Ethyl-3-propoxycarbonyl-4-quinolone 6-Ethyl-3-propylaminocarbonyl-4-quinolone 6-Ethyl-5-(4-{methyl[4-(methylsulfonyl)benzyl]amino}phenyl)pyrimidine-2,4-diamine 6-Ethyl-5-(4-{[(4-nitro-phenyl)amino]methyl}phenyl)pyrimidine-2,4-diamine 6-Ethyl-5-(4-{[4-(methylsulfonyl)benzyl]amino}phenyl)pyrimidine-2,4-diamine 6-Ethyl-5-[4-(4-trifluoromethanesulfonyl-benzylamino)-phenyl]-pyrimidine-2,4-diamine 6-Ethyl-5-[4-({[4-(methylsulfonyl)phenyl]amino}methyl)phenyl]pyrimidine-2,4-diamine 6-Ethyl-5-{4-[(4-nitrobenzyl)amino]phenyl}pyrimidine-2,4-diamine 6-ethylamino-3-(1-methyl-2-pyrrolidinyl)pyridine oxalate 6-ethyldinapsoline hydrobromide 6-EtS, 1-(1-indolinyl)-2-propylamines 6-Ets-5-F, 1-(1-indolinyl)-2-propylamines 6-Fluoro-2-pyridin-2-yl-1H-benzoimidazole 6-Fluoro-3-( l-methyl-2-pyrrohdinyl )pyridme maleate 6-Fluoro-3-(2(S)-azetidinylmethoxy)pyridine 6-Fluoro-3-(N-ethyl-N-methyl)aminomethylpyridine oxalate 6-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]cyclohexyl]-1H-indole 6-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-pipera-zinyl]cyclohexyl]-1H-indole 6-Fluoro-5’Iodo-HEAT HCl 6-fluoro-DMT: 6-Fluoro-N,N-dimethyltryptamine 6-Fluoro-HEAT HCl 6-Fluoro-N,N-dimethyltryptamine 6-fluoronorepinehprine 6-formylnicotine 6-HT 6-Hydroxy-2,5,7,9-tetramethyl-9H-beta-carbolin-2-ium 6-Hydroxy-2,5,7-trimethyl-9H-beta-carbolin-2-ium 6-Hydroxy-2-[1-(4-hydroxyphenyl)methylidene]-3,4-dihydro-2H-naphthalen-1-one 6-hydroxy-3-(1-methyl-2-pyrrolidinyl)pyridine hydrochloride 6-Hydroxy-5,7,9-trimethyl-beta-carboline 6-Hydroxy-5,7-dimethyl-beta-carboline 6-hydroxy-5-methoxyduloxetine 6-hydroxy-5methoxyduloxetine 6-hydroxyduloxetine 6-hydroxyduloxetine glucuronide 6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-hexanoyloxymethyl-tetrahydro-2-pyranone 6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-octanoyloxymethyl-tetrahydro-2-pyranone 6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone 6-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone 6-Iodo-3-(2(S)-azetidinylmethoxy)pyridine 6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene 6-Iodo-4'-dimethyaminoflavone 6-Iodo-4'-hydroxyflavone 6-Iodo-4'-methoxyflavone 6-Iodo-4'-methyaminoflavone 6-Iodo-HEAT HCl 6-MeOT 6-MeS, 1-(1-indolinyl)-2-propylamines 6-Metho,D'-3-(N-ethyl-N-methylamtnomethyl)pyndine oxalate 6-methoxy-2-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)isoindolin-1-one 6-Methoxy-2-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)isoindolin-1-one 6-Methoxy-2-naphthylacetic acid 6-Methoxy-2-[1-(2-methylphenyl)methylidene]-3,4-dihydro-2H-naphthlalen-1-one 6-Methoxy-3-methyl-N-phenyl-N-(3-(piperidin-1-yl)propyl)benzofuran-2-carboxamide (KSCM-11) 6-Methoxy-5-methyl-2-phenyl[1,3]thiazolo[4,5-b]pyridine 6-methoxynicotine 6-Methyl-1,1-dipentyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carboline 6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol 6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ylamine 6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ylamine 6-Methyl-1-(2,4-dichlorophenyl)-N-(homopiperidinyl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 6-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 6-Methyl-1-(2,4-dichlorophenyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 6-Methyl-1-(2,4-dichlorophenyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 6-Methyl-1-(2,4-dichlorophenyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 6-Methyl-1-(4-methylbenzyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 6-methyl-10-nitro-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline 6-Methyl-2-{2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}nicotinonitrile 6-Methyl-3-(1 -methyl-2-pyrrohdmyl)pyridme dthydrochlortde 6-Methyl-3-(N-ethyl-N-methylammomethyl)pyridme oxalate 6-Methyl-3-bromoflavone 6-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine 6-Methyl-5'-[(6-methyl-2-pyridinyl)ethynyl]-2,3'-bipyridine 6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-amine 6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol 6-n-Propyl-3-(1-methyl-2-pyrrolidinyl)pyridine hydrochloride 6-nitro-2-(2-propoxymethylpiperazin-1-yl)quinoline 6-Nitro-2-piperazin-1-yl-quinoline 6-Nitro-7-(3-pyridyl)-2,3(1H,4H)-quinoxalinedione 6-Nitronicotine 6-PBC 6-phenyl-3-propyl-1,5-dihydropyrrolo[3,2-d]pyrimidin-2,4-dione 6-phenylsulfonylpyridazin-2H-3-one 6-Propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol 6-Propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-2,10,11-triol 6-Sulfonamido-3-(1-methyl-2-pyrrolidinyl)pyridine hydrochloride 6-tert-Butyl-2-(2-chlorophenyl)-3-(4-chlorophenyl)-5,6-dihydro-2Hpyrazolo[3,4-c]pyridin-7(4H)-one 6-Thioguanosine 6-Thiopurine riboside 6-TMT 6-[((2S)-2-[(1-benzofuran-2-ylcarbonyl)amino]-5-{[(benzyloxy)carbonyl]amino} pentanoyl)amino]hexanoic acid 6-[(2-Hydroxy-5-nitrobenzyl)thio]inosine 6-[(2-Methyl-4-thiazolyl)ethynyl]quinoxaline 6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-N-(4-fluorophenyl)-1,3,5-triazine-2,4-diamine 6-[(Benzyloxy)methyl]-5-(4-{[(2-chloropyridin-4-yl)methyl]amino}phenyl)pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-(4-{[(4-nitro-phenyl)amino]methyl}phenyl)pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-(4-{[4-(methylsulfonyl)benzyl]amino}phenyl)pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-(4-{[4-(methylsulfonyl)benzyl]oxy}phenyl)pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-[4-(neopentylamino)phenyl]pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-[4-({4-[(trifluoromethyl)sulfonyl]benzyl}amino)phenyl]pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-{4-[(4-methoxybenzyl)amino]phenyl}pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-{4-[(4-nitrobenzyl)amino]phenyl}pyrimidine-2,4-diamine 6-[(Benzyloxy)methyl]-5-{4-[(pyridin-4-ylmethyl)amino]phenyl}pyrimidine-2,4-diamine 6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole 6-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine 6-[4-(phenethylamino-methyl)-phenoxy]-nicotinamidine 6-[4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl]pyridine-3-carboxamide 6-[Me2]N-HEAT HCl 61 62 69 6a 6a,7,8,12b-Tetrahydro-6H-chromeno[3,4-c]isoquinoline-2,3-diol 6b 6c 6d 6MNA 6R, (R)-PHPNECA 6S, (S)-PHPNECA 7 7 (3PBC) 7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 7,8-dihydro-3,6-didesoxymorphine 7,8-dihydro-3-desoxyheterocodeine 7,8-dihydro-3-desoxymorphine 7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(2-phenoxyethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 7,8-Dimethoxy-3-[4-(quinolin-6-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole 7,8-Dimethoxy-5-methyl-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isox... 7-((1-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)piperidin-4-yl)methoxy)benzo[d]oxazol-2(3H)-one 7-((1-(2-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)ethyl)piperidin-4-yl)methoxy)benzo[d]oxazol-2(3H)-one 7-((1-isopropylpiperidin-4-yl)methoxy)-4-(4-methoxyphenyl)-1,2,3,4-tetrahydro-2,6-naphthyridine 7-((1-isopropylpiperidin-4-yl)methoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydro-2,6-naphthyridine 7-((1R,4R)-5-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl)benzo[d]oxazol-2(3H)-o... 7-((2-(4-(Isoquinolin-1-yl)piperazin-1-yl)ethyl)(propyl)amino)5,6,7,8-tetrahydronaphthalen-2-ol 7-((2-(4-(Naphthalen-1-yl)piperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-o 7-((2-(4-(Naphthalen-1-yl)piperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-2-ol 7-((2-(4-(Naphthalen-2-yl)piperazin-1-yl)ethyl)(propyl)amino)5,6,7,8-tetrahydronaphthalen-2-ol 7-((4-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)piperazin-1-yl)methyl)benzo[d]oxazol-2(3H)-one 7-((N-(Methylsulfonyl)amino)methyl)-1,2,3,4-tetrahydroisoquinoline 7-((N-Methylamino)sulfonyl)-1,2,3,4-tetrahydroisoquinoline 7-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine 7-(1-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)piperidin-4-yloxy)benzo[d]oxazol-2(3H)-one 7-(1-(2-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)ethyl)piperidin-4-yloxy)benzo[d]oxazol-2(3H)-one 7-(1-hydroxy-1-methylethyl)-3-[4-fluoro-3-(pyridine-3-yl)phenyl derivative 7-(2-Chloroethyl)theophylline 7-(2-Dimethylaminoethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c... 7-(2-Methoxyethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ymethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxaz... 7-(3-(3,3-difluoroazetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(3,3-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(3,3-difluoropyrrolidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4,4-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate 7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 7-(3-(4-cyclopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-ethylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(3-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylsulfonyl)phenyl)-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(methylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(trifluoromethyl)phenyl)-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-(4-(trifluoromethylthio)phenyl)-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-p-tolyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-2-methyl-4-phenyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(3-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(4-isopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propoxy)-3,4-dihydroquinolin-2(1H)-one 7-(3-(azetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline 7-(3-morpholinopropoxy)-4-phenyl-1,2,3,4-tetrahydro-2,6-naphthyridine 7-(4,6-Dimethoxy-2-pyrimidinyl)-2-methylquinoline 7-(4,6-Dimethyl-2-pyrimidinyl)-2-methylquinoline 7-(4-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)methyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 7-(4-((6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 7-(4-(2-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 7-(4-(3-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)propyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 7-(4-(3-(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-2-yl)propyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate 7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)butyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 7-(4-Methoxy-2-pyrimidinyl)-2-methylquinoline 7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate 7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate 7-(5-Fluoro-2-pyrimidinyl)-2-methylquinoline 7-(6-chloropyridin-3-yl)-1,7-diazaspiro[4.4]nonane 7-(allyl)-theophylline 7-(benzyl)-theophylline 7-(beta-acetoxyethyl)-theophylline 7-(beta-chloroethyl)-theophylline 7-(beta-hydroxyethyl)-theophylline 7-(diethylaminomethyl)-5-nitrosoquinolin-8-ol 7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol 7-(N,N-Bis(methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline 7-(N-(Methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline 7-(n-propyl)-theophylline 7-(propargyl)-theophylline 7-(Propyl(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)amino)-5,6, 7,8-tetrahydronaphthalen-2-ol 7-(Propyl(2-(4-(quinolin-5-yl)piperazin-1-yl)ethyl)amino)-5,6, 7,8-tetrahydronaphthalen-2-ol 7-(pyridin-3-yl)-1,7-diazaspiro[4.4]nonane 7-(Thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one 7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 7-allyl-1,3-n-dipropylxantine 7-allyl-3-isobutyl-1-methylxantine 7-amino-1-benzyl-N-cyclohexyl-4-oxo-1,4-dihydro-1,8-naphthyridine-2-carboxamide 7-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine 7-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine 7-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines 7-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine 7-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 7-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 7-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 7-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-benzylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 7-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 7-Aminosulfonyl-3-hydroxymethyl-THIQ 7-benzoyl-11-(4-(diethylamino)phenyl)-3,3-dimethyl-2,3,4,5,10,11-hexahydro-1H-dibenzo[b,e][1,4]diazepin-1-one 7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride 7-benzyl-1,3-dipropylxanthine 7-benzyl-1,3-n-dipropylxantine 7-benzyl-3-isobutyl-1-methylxantine 7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride 7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 7-benzyl-IBMX 7-benzyltheophylline 7-Bromo-9-(4-methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine 7-Bromo-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 7-bromo-eudistomin D 7-CH3-methyl-1,3-n-dipropyl-xantine 7-chloro-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide 7-Chloro-1-(methoxymethyl)-9-(4-methyl-1-piperazinyl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine 7-Chloro-3-[(4-phenylpiperazin-1-yl)methyl]-1Hpyrrolo[2,3-c]pyridine 7-Chloro-3-{3-[4-(2,3-dihydro-1,4-benzodioxin-5-yl)-1-piperazinyl]propyl}-1H-indole 7-Chloro-9-(4-methyl-1,4-diazepan-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 7-Chloro-9-(4-methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine 7-Chloro-9-(4-methylhexahydro-1H-1,4-diazepin-1-yl)pyrrolo[2,1-b][1,3] benzothiazepine 7-Chloro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 7-Cl-4-hydroxy-3-phenylquinolin-2(1H)-one 7-Cl-KYNA 7-Cyano-6-(1H-imidazol-1-yl)-2,3(1H,4H)-quinoxalinedione 7-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 7-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 7-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 7-Cyclopentyloxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol... 7-Cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine 7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine 7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine 7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine 7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine 7-Ethyl-1,3-trimethyl-8-(3,4,5-trimethoxystyryl)xanthine 7-ethyl-10-hydrocamptothecin 7-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine 7-ethyl-N,N-diallyltryptamine 7-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 7-Fluoro-9-(4-methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine 7-Fluoro-9-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine 7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine 7-Hydroxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole 7-Hydroxy-6-phenylthieno[3,2-b]pyridin-5(4H)-one 7-iodo-THIQ 7-methoxy-1-naphthylpiperazine 7-Methoxy-1-[2-(4-morpolinyl)ethyl]-N-[(1S,2S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl)-1H-indazol-3-carboxamide 7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one 7-Methoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole 7-Methoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole 7-Methoxy-3-{2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl}-3,4-dihydro-1(2H)-naphthalenone 7-Methoxy-3-{2-[4-(2-pyridinyl)-1-piperazinyl]ethyl}-3,4-dihydro-1(2H)-naphthalenone 7-Methoxy-8-[2-(4-methyl-1-piperazinyl)ethoxy]-4-(3,4,5-trimethoxyanilino)benzo[g]quinoline-3-carbonitrile 7-Methoxy-8-[2-(4-morpholinyl)ethoxy]-4-(3,4,5-trimethoxyanilino)benzo[g]quinoline-3-carbonitrile 7-METHOXY-Beta-CARBOLINE 7-Methoxy-N,N-Dimethyltryptamine 7-Methoxy-N-[(2-methoxyphenyl)methyl]-1-[2-(4-morpholinyl)ethyl]-1H-indazol-3-carboxamide 7-Methoxy-N-[phenyl(2-pyridinyl)methyl]-1-[2-(4-morpholinyl)ethyl]-1H-indazol-3-carboxamide 7-Methyl-1-(2,4-dichlorophenyl)-N-(homopiperidinyl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(2,4-dichlorophenyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(2,4-dichlorophenyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-methyl-1-(2,4-dichlorophenyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(2,4-dichlorophenyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(2,4-dichlorophenyl)-N-morpholinyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-(homopiperidin-yl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-1-(4-methylbenzyl)-N-morpholinyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide 7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide 7-Methyl-3-[3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]imidazo-[1,2-a]pyridine 7-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 7-methyl-6,7,8,9,14,15-hexahydro-5 H-benz[d]indolo[2,3-g]azecine 7-Methylsulfonyl-3-hydroxymethyl-THIQ 7-MethylX 7-nitro-THIQ 7-OH-CHLORPROMAZINE 7-OH-DPAT 7-OH-DPAT,(+) 7-OH-DPAT,(-) 7-Propyl-6a,7,8,12b-tetrahydro-6H-chromeno[3,4-c]isoquinoline-2,3-diol 7-tert-butyl-5-(4-chlorophenyl)-6,7-dihydro-5H-pyrazolo[3,4-d]pyrimidin-4-amine 7-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 7-Thia-9deazaado 7-trifluoromethyl-3-(2'-cyano-2,4'-difluorobiphenyl-5-yl) analogue 7-[2-(2-Ethoxyethoxy)ethoxy]-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,... 7-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione  7-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione   7-[3-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-propoxy]-4-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydro-isoquinoline 7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride 7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione 7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione 7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride 7-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyloxy]quinoline 7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione 7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione 7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride 7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride 7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride 7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride 7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chlorid... 7-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 7-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one 70 74 75 76 77 78 79 7a 7alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(2'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(2'-methoxycinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(2'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(2'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(4'-chlorocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(4'-chlorocinnamyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(4'-chlorocinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(4'-methoxycinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(4'-methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(4'-Methylcinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(4'-nitrocinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(cinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(cinnamoyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrooripavine 7alpha-[(cinnamyl)-aminomethyl]-6,14-endoethanotetrahydrothebaine 7b 7HCCMA 8 8,15-dimethyl-N-(1,3,4-thiadiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 8,15-dimethyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide 8,17-didehydro-17-deoxysalvinorin A 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 8-((1,3-Dimethyl-1H-pyrazol-5-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-((2-(3-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-((2-(4-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochlorid... 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochlor... 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochlori... 8-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-2-(furan-2-yl)-[1,2,4]triazolo[1,5-f]pyrimidin-5-amine 8-(1-((4-Chlorophenyl)-1H-2,1,3-triazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]pur-ine-2,4(1H,3H)-dione 8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-3-ethyl-1-propyl-1H-purine-2,6(3H,7H)-dione 8-(1-Benzylpiperidin-4-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(1-Buten-3-yl)-11-hydroxy-N-propylnoraporphine 8-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)-1,3-dipropylxanthine 8-(1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)-1,3-dipropylxanthine 8-(1-{1-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dion... 8-(1-{2-Hydroxy-2-[5-oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purin... 8-(1-{2-Oxo-2-[4-(3-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-(1-{2-Oxo-2-[4-(4-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-(1-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-(1-{2-[4-(3-Chloro-4-fluoro-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-(1-{2-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dion... 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2,3-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,3-Dihydro-1H-inden-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,4,6-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,4-Diaminophenyl)-1,3-dipropylxanthine 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(2,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2,4-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2,6-dichloro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-dichlorobenzyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-dichlorobenzyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-dichlorobenzyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(2,6-Dichlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(2,6-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-yl)eth... 8-(2-(1H-indol-3-yl)ethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol 8-(2-(1H-Pyrrol-1-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-(2,3-Dimethoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-(2-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-(3,4-Dimethoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2-(3-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-(5-Bromo-2-methoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-(Benzo[d][1,3]dioxol-5-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Amino-4-chlorophenyl)-1,3-dipropylxanthine 8-(2-Aminophenyl)theophylline 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione ( 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(2-Bromobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(2-Bromophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione 8-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)purine  8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-(4-pentanoylpiperazin-1-yl)-9H-purine 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(piperidin-1-yl)-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2,3-dihydro-1,4-benzodioxin-2-ylcarbonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2-phenylpropanoyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(3,3-dimethylbutanoyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(butylsulfonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclopentylacetyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclopropylsulfonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(ethoxyacetyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(ethylsulfonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(methylsulfonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(piperidin-1-ylacetyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(propylsulfonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(tetrahydro-2H-thiopyran-4-ylcarbonyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(tetrahydrofuran-3-ylacetyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(trifluoroacetyl)piperazin-1-yl]-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(1-methylethyl)sulfonyl]piperazin-1-yl}-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(2-methylpropyl)sulfonyl]piperazin-1-yl}-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(3,3,3-trifluoropropyl)sulfonyl]piperazin-1-yl}-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(cyclohexylmethyl)sulfonyl]piperazin-1-yl}-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(pyrrolidin-1-yl)carbonyl]piperazin-1-yl}-9H-purine 8-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(tetrahydro-2H-pyran-4-ylmethyl)sulfonyl]piperazin-1-yl}-9H-purine 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Fluoro-5-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Fluorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2-Furyl)theophylline 8-(2-Hydroxy-2-phenylethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione 8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(2-Methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(2-Methoxyphenyl)-2-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)propyl)-2,8-diazaspiro[4.5]decane 8-(2-Methyl-2-buten-4-yl)-11-hydroxy-N-propylnoraporphine 8-(2-Thienyl)theophylline 8-(3,4,5-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,4,5-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione 8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(3,4-Dichlorobenzyl)-1-cyclopropyl-3-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3,4-Difluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3,4-Dimethoxyphenyl)-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,5-Bis(trifluoromethyl)benzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,5-bis(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,5-Bis(trifluoromethyl)benzyl)-3-ethyl-1-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3,5-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(1H-Imidazol-1-yl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(1H-Pyrrol-1-yl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-(3,4-Dichlorophenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(3-Bromophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-(3-Chlorophenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(3-Methoxyphenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 8-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)pperidin-1-yl)-1-hydroxypropyl)-5,6-dihydro-1Hpyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(3-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(3-(4-(6-Fuorobenzo[d]isoxazol-3-yl)- piperidin-1-yl) propyl)-5,6-dihydro-1H-pyrrolo [3,2,1-ij]quinolin4(2H)-one 8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(3-(4-Chlorophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3-Bromophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Bromophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Chloro-5-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Chlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Chlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Fluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Fluorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Fluorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Furyl)theophylline 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(3-Methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Methoxyphenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(3-Phenylpropyl)-1,3,7-triethylxanthine 8-(3’-Fluorobenzyl)amino-4-oxapentacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecane 8-(3’-Fluorophenethyl)amino-4-oxapentacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecane 8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(4,5-Difluoro-2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 8-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(1-(4-(5-chlorobenzo[d]thiazol-2-yl)piperazin-1-yl)-2-methyl-1-oxopropan-2-yloxy)phenyl)-1,3-dimethyl-1H-purine-2,6(3H,7... 8-(4-(1H-Indol-3-yl)butyl)-1-phenyl-1,3,8-triazaspiro[4.5] decan-4-one 8-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione 8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(4-(4-(3-Chlorobenzyl)piperazine-1-sulfonyl)phenyl)-1-ethyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(3-Chlorobenzyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(3-Fluorobenzyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1-ethyl-1H-purine-2,6(3H,7H)-dione 8-(4-(4-(4-chlorobenzyl)piperazin-1-ylsulfonyl)phenyl)-1-propyl-1H-purine-2,6(3H,7H)-dione 8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-ethyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-prop-2-ynyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-Chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-Fluorobenzyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-Methoxybenzyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-Methoxyphenyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(4-Methylbenzyl)piperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-sulfonyl)phenyl)-1-ethyl-3,7-dihydropurine-2,6-dione 8-(4-(4-Benzo[1,3]dioxol-5-ylmethylpiperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(4-benzylpiperazin-1-ylsulfonyl)phenyl)-1-ethyl-1H-purine-2,6(3H,7H)-dione 8-(4-(4-Phenethylpiperazine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-(5-Chlorobenzo[d]thiazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one 8-(4-(Benzo[d]oxazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one 8-(4-(Benzo[d]thiazol-2-yl)butyl)-1-phenyl-1,3,8- triazaspiro[4.5]decan-4-one 8-(4-(benzo[d]thiazol-2-yl)butyl)-3-(4- chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol hydrochloride 8-(4-(Piperidine-1-sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-Acetoxyphenyl)theophylline 8-(4-Aminophenyl)theophylline 8-(4-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Bromophenoxymethyl)caffeine 8-(4-Bromophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(4-Bromophenyl)-1,3-dipropylxanthine 8-(4-Bromophenyl)-1-butylxanthine 8-(4-Bromophenyl)-1-propargylxanthine 8-(4-Bromophenyl)-1-propylxanthine 8-(4-Carboxymethyloxyphenyl)-1-propylxanthine 8-(4-Carboxyphenyl)theophylline 8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Chloro-2-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 8-(4-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(4-Chlorophenoxymethyl)caffeine 8-(4-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(4-Chlorophenyl)theophylline 8-(4-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Fluorophenoxymethyl)caffeine 8-(4-Fluorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(4-Hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione 8-(4-hydroxyphenyl)theophylline 8-(4-Iodophenyl)-1,3-dipropylxanthine 8-(4-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 8-(4-Methoxycarbonylmethoxy)phenyl-1-propylxanthine 8-(4-Methoxyphenoxymethyl)caffeine 8-(4-Methoxyphenyl)theophylline 8-(4-Methylcarboxyethylidene)phenyl-3-propylxanthine 8-(4-Methylphenoxymethyl)caffeine 8-(4-Nitrophenyl)theophylline 8-(4-Sulfophenyl)theophylline 8-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 8-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(5-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)pentyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(6-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)hexanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 8-(6-Carboxynaphth-2-yl)-1-propylxanthine 8-(8-((8R,9S,13S,14S,17S)-3,17-dihydroxy-13-methyl-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthren-17-yl)oct... 8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxa... 8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 8-(Benzo[d][1,3]dioxol-5-ylmethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(piperidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(3-(pyrrolidin-1-yl)propyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(butylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylmethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(diisopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(dimethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-(2-methoxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(bis(2-chlorophenyl)methyl)-3-isopentyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine 8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-methyl-1-propyl-3,7-dihydro-purine-2,6-dione 8-(m-Aminostyryl)-3,7-dimethyl-1-propargylxanthine 8-(m-Bromostyryl)-3-(2-hydroxyethyl)-7-methyl-1-propargylxanthine 8-(m-Bromostyryl)-3-(3-hydroxypropyl)-7-methyl-1-propargylxanthine 8-(p-Hydroxyphenyl)theophylline 8-(p-sulfophenyl)theophylline 8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 8-benzhydryl-1-phenyl-3-(prop-2-ynyl)-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-(cyclobutylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-(cyclohexylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-(cyclopropylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-isopropyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one 8-Benzoyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 8-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione 8-Benzyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine 8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 8-Bromoadenosine 8-Butyl-2-(2-methoxyphenyl)-2,8-diazaspiro[4.5]decane 8-CAC 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide 8-Chloro-11-(4-ethylpiperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 8-Chloro-11-(4-isopropylpiperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine 8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine 8-Chloro-11-[4-(1,1-dideutrioethyl)piperazin-1-yl]-5H-dibenzo[b,e][1,4]diazepine 8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine 8-Chloro-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-chromane-5-carboxamide 8-ChloroT 8-Cinnamyl-1-propylxanthine 8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-cyclopentyl-1,3-dipropylxanthine 8-cyclopentyl-1,3-dipropylxanthine 8-Cyclopentyl-1-propylX 8-Cyclopentyl-1-propylxanthine 8-Cyclopentyl-3-(1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-ylmethyl)-1-propylxanthine 8-Cyclopentyltheophylline (CPT) 8-ethoxy-3-iodo-benzo[e]pyrazolo[5,1-c][1,2,4]triazine 5-oxide 8-Fluoro-3-[[4-(4-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide 8-Fluoro-3-[[4-(5-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide 8-Fluoro-3-[[4-(6-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide 8-Fluoro-3-[[4-(7-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide 8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}-N-methylchromane-5-carboxamide 8-Fluoro-l-hydroxy-4-(isopropylamino)-[ 1,2,4]triazolo[4,3-a ]quinoxaline Hydrobromide Hydrate 8-Fluoro-N-isopropyl-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide 8-Fluoro-N-phenyl-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide 8-Fluoro-N-propyl-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide 8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine 8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 8-hydroxy-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 8-Hydroxy-5,7,9-trimethyl-delta-carboline 8-Hydroxy-5-[(R)-1-hydroxy-2-(4,7-diethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-di-n-butylindan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-di-n-propylindan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-diethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-dimethoxyindan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-dimethylindan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-5-[(R)-1-hydroxy-2-(indan-2-ylamino)-ethyl]-1H-quinolin-2-one 8-Hydroxy-7,9-dimethyl-delta-carboline 8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 8-Hydroxyamoxapine 8-hydroxydibenzazepine 8-hyroxy-2-(di-n-propylaminotetralin 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione 8-M-ADOT 8-M-CADOT 8-M-PDOT 8-MeO-C1EPAT 8-MeO-DPAT 8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane 8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 8-methoxy-11-(4-methylpiperazino)-5H-dibenzo[b,e][1,4]diazepine 8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate 8-Methoxy-7-[2-(4-methyl-1-piperazinyl)ethoxy]-4-(3,4,5-trimethoxyanilino)benzo[g]quinoline-3-carbonitrile 8-Methoxy-7-[2-(4-morpholinyl)ethoxy]-4-[(3,4,5-trimethoxyanilino)benzo[g]quinoline-3-carbonitrile 8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 8-Methoxy-N-methylquipazine 8-methoxydibenzodiazepine 8-Methoxyquipazine 8-Methyl-1-[1-(naphthalene-1-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 8-Methyl-1-[1-(quinoline-8-sulfonyl)-piperidin-4-yl]-1,4-dihydro-benzo[d][1,3]oxazin-2-one 8-Methyl-5.6,7,9-tetrahydro-8H-pyrido[3,4-c]azepine oxalate 8-Methylsulfonyloxy-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 8-MsO-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 8-OH-AT 8-OH-DPAT 8-OH-DPAT,(+) 8-OH-DPAT,(-) 8-Oxa-norcocaine 8-Phenyl-1-propylxanthine 8-Phenyltheophylline 8-phenylxanthine 8-Propyltheophylline 8-SPT 8-TfO-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 8-trifluoromethylsulfonyloxy-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine 8-[1-(5-Oxo-1-m-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-[1-(5-Oxo-1-p-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-[2-(4-Oxo-1,2,3,4-tetrahydro-2-naphthalenyl)ethyl]-1,3,8-triazaspiro[4.5]decan-4-one 8-[2-(4-Oxo-1,2,3,4-tetrahydro-2-naphthalenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione 8-[2-(6-Methoxy-4-oxo-1,2,3,4-tetrahydro-2-naphthalenyl)ethyl]-1,3,8-triazaspiro[4.5]decan-4-one 8-[2-(6-Methoxy-4-oxo-1,2,3,4-tetrahydro-2-naphthalenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione 8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine 8-[4-(((1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)amino)-2-oxoethoxy)phenyl]-1-propylxanthine 8-[4-((2-Aminoethylamino)-2-oxoethoxy)phenyl]-1-propylxanthine 8-[4-((2-Hydroxyethylamino)-2-oxoethoxy)phenyl]-1-propylxanthine 8-[4-(2-Diethylaminoethoxy)phenyl]-1,3-dimethylxanthine 8-[4-(2-Dimethylaminoethoxy)phenyl]-1,3-dimethylxanthine 8-[4-(3-Chloropropoxy)benzyl]-1,3-dimethylxanthine 8-[4-(3-Chloropropoxy)phenyl]-1,3-dimethylxanthine 8-[4-(4-benzylpiperazide-1-sulfonyl)phenyl]-1-propylxanthine 8-[4-(Cyclopentyloxy)phenyl]-1,3-dimethylxanthine 8-[4-[(Carboxymethyl)oxy]phenyl]-1,3-dimethylxanthine 8-[4-[(Carboxymethyl)oxy]phenyl]-1,3-dipropylxanthine Ethyl Ester 8-[4-[(Carboxymethyl)oxy]phenyl]-l,3-dipropylxanthine 8-[4-[(Carboxymethyl)oxy]phenyl]-l,3-dipropylxanthine N-Hydroxy-succinimide Ester 8-[4-[[(p-Toluidinocarbonyl)methyl]oxy]phenyl]-l,3-dipropylxanthine 8-[4-[[[(4-Hydroxyanilino)carbonyl]methyl]oxy]-phenyl]-1,3-dipropylxanthine 8-[4-[[[[(2- Aminoethyl)amino]carbonyl]methyl]oxy]-phenyl]-1,3-dipropylxanthine 8-[4-[[[[[2-(Biotinylamino)ethyl]amino]carbonyl]-methyl]oxy]phenyl]-l,3-dipropylxanthine 8-[4-[[[[[2-[ Ethyl(4-hydroxybenzyl)ammonio]ethyl]-amino]carbonyl]methyl]oxy]phenyl]-1,3-dipropylxanthine Acetate 8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine 8-[4-{3-(4-(2-Chlorobenzyl)piperazin-1-yl)propoxy}phenyl]- 1,3-dimethylxanthine 8-[bis-(2-chloro-phenyl)-methyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 8-[{3-(2-(Diethylaminoethylamino)-2-oxoethoxy)-4-meth-oxy}phenyl]-1,3-dimethylxanthine 8-[{4-(2-(Diethylaminoethylamino)-2-oxoethoxy)-3-meth-oxy}-phenyl]-1,3-dimethyl-xanthine 8-{1-[1-(2,4-Difluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(3-Fluoro-phenyl)-2-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(3-Methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(3-Methoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(4-Methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[1-(4-Methoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[2-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[2-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[2-Oxo-2-(4-p-tolyl-piperazin-1-yl)-ethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[5-Oxo-1-(3-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[5-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{1-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{3-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{3-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{3-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{3-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline 8-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline 8-{4-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{4-[1-(4-Fluorophenyl)-5-oxo-pyrrolidin-3-ylmethoxy]phenyl}-1,3-dipropyl-3,7-dihydropurine-2,6-dione 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2,2-dimethyl-2H-1,4-benzoxazin-3(4H)-one 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2,4-dimethyl-2H-1,4-benzoxazin-3(4H)-one 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2-methyl-2H-1,4-benzoxazin-3(4H)-one 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-2H-1,4-benzoxazin-3(4H)-one 8-{4-[3-(1H-Indol-3-yl)propyl]-1-piperazinyl}-3,4-dihydro-2H-1,4-benzoxazine 8-{4-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{4-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{4-[N-(3-Dimethylaminopropyl)-sulfonamido]phenyl}-1,3-Dipropylxanthine (PD 113,297) 8-{6-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{6-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{6-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 8-{6-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione 80 81 82 83 84 85 86 87 88 89 8a 8alpha-phenyl-6alpha,14alpha-endo-Ethenotetrahydrothebaine 8b 8PST 8PT 8R-hydroxylobel-9-ene 8R-lisuride 8Z,11Z,14Z-eicosatrienoic acid 9 9, PENECA 9,10-Didehydro-N,N-diethyl-6-methylergoline-8ß-carboxamide 9,11-azo PGH2 9,11-epoxymethano PGH2 9,11-ethano PGH2 9,13-epoxy-15,16-dihydroxylabd-5-en-7-one 9,13-epoxy-6-hydroxylabdan-15,16-olide 9,13-epoxylabd-5-en-7-on-15,16-olide 9,13-epoxylabd-5-ene-7 b,15,16-triol 9,13-epoxylabd-5-ene-7 b,15,16-triol, 9,13-epoxylabd-5-ene-7 β,15,16-triol 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(1H-indol-2-yl)-acetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimeth... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(2,3-dichloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-di... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(2,4-dichloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-di... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(2,5-dichloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-di... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(2-chloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimeth... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(2-hydroxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimet... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-2-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-2-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-2-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-3-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-3-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4,5-trimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-4-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4-dichloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-di... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,4-dimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-d... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,5-di-tert-butyl-4-hydroxy)phenylacetate]-5,6,9,10,11,12,13,13a-o... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3,5-dimethoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-d... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(3-chloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimeth... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(4-bromo)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimetho... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(4-chloro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimeth... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(4-diethylamino)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(4-ethyl)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimetho... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(4-fluoro)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimeth... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-(4-methoxy)phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimet... 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxo-phenylacetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimethoxy 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxofuran-2-yl-acetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimethoxy 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxopyridin-3-yl-acetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimethoxy 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxopyridin-4-yl-acetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimethoxy 9,13-Imino-8H-azocino [2,1-a] isoquinolin-8-one,14-[2-oxothiophen-2-yl-acetate]-5,6,9,10,11,12,13,13a-octahydro-1,3-dimethoxy 9,13:15,16-diepoxylabdane-6b,15a-diol 9,13:15,16-diepoxylabdane-6b,16a-diol 9,13:15,16-diepoxylabdane-6b,16b-diol 9,13:15,16-diepoxylabdane-6β,15α-diol 9,13:15,16-diepoxylabdane-6β,16α-diol 9,13:15,16-diepoxylabdane-6β,16β-diol 9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one 9-(1-Aminoethyl)-9,10-dihydroanthracene Hydrochloride 9-(2',2',2'-Trifluoroethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-(2'-Methoxyethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-(1H-indol-3-yl)ethyl)-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-(2,4-dichlorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(2-(4-chlorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-(4-fluorobenzyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-(benzylamino)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-(benzyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-aminoethyl)-9,10 dihydroanthracene oxalate) 9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(2-Hydroxyethyl)adenines 9-(2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(2-Tetrahydrofuryl)adenines 9-(3,4-dimethoxyphenethyl)-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(6-fluoro benzo[d]isoxazol-3-yl)piperidin-1-yl)- 1-hydroxypropyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on... 9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one 9-(3-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- propanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(Benzo[d]thiazol-2-yl)piperidin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(Pyridin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-(Pyrimidin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-(4-Phenylpiperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(3-chlorobenzyl)-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(2,3-Dimethylphenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl)butanoyl)-1-methyl-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-... 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on 9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(4-chlorobenzyl)-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine 9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(piperidin-1-yl)-9H-purine 9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-9H-purin-6-amine 9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophenyl)-9H-purin-6-amine 9-(4-hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-(4-Methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine 9-(4-Methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine-1,10-dicarbaldehyde 9-(4-Methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepine-1-carbaldehyde 9-(4-Methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine-1,10-dicarbaldehyde 9-(4-Methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepine-1-carbaldehyde 9-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one 9-(5-Amino-5-deoxy-alpha-L-lyxofuranosyl)adenine 9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(Aminomethyl)-9,10-dihydroanthracene 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-(Methylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-(N,N,-Dimethyl-N-oxyamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-(N,N-Dimethyl-N-oxyamino)-3-(N-hexamethyleneiminyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one 9-(N,N-Ethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-alpha-L-Lyxofuranosyladenine 9-aminoacridine 9-Aminomethyl-9(H)-thioxantheneoxalate 9-Aminomethyl-9(H)-xanthene 9-Benzyl-4-cyclohexyl-1-(4-methoxybenzoyl)-1,4,9-triazaspiro[5.5]undecane-3,5-dione 9-Benzyl-4-cyclohexyl-1-(4-methylbenzoyl)-1,4,9-triazaspiro[5.5]undecane-3,5-dione 9-benzyl-9-azabicyclo[3.3.1]nonan-3-yl 2-methoxy-5-methylphenylcarbamate 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4,5,6,7-tetrahydro-1H-benzo[7,8]cycloocta[1,2-c]pyrazole-3-carboxamide 9-chloro-7-(2-ethoxyphenyl)azepino[1,7-a]indole 9-Cyclohexyl-6-(4-methoxybenzoyl)-6,9-diazaspiro[4.5]decane-8,10-dione 9-Cyclohexyl-6-(4-methylbenzoyl)-6,9-diazaspiro[4.5]decane-8,10-dione 9-Cyclopentyladenine 9-Cyclopropylamino-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Deazaado 9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(1-adamantyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(1H-indazol-6-yl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(2'-methoxy-5'-pyridyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(2,4-dichlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(2,4-dimethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(2-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(2-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(3-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(3-n-pentyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4'-ethylphenyl)-3H-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4'-methyl-1'-cyclohexyl)-3H-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-cyclohexylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-cyclopropylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one 9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3-diazafluoren-4-one 9-Dimethylamino-3-(4-isopropylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-methylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one 9-Dimethylamino-3-(4-n-propylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(4-tert-butylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(N-hexamethyleneiminyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(o-hydroxyphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(p-bromophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(p-chlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(p-fluorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(p-tolyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-(p-trifluoromethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-benzyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclobutyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclohexyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclooctyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclopentyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclopentylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cyclopropyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-cycoheptyl-3H-5-thia-1,3,6-triazafluoren-4-one 9-Dimethylamino-3-hydrogen-3H-5-thia-1,3,6-triazafluoren-4-one 9-Erythro-(2-hydropy-3-monyl) adenine 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Ethyladenine 9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-Methyladenine 9-MethylX 9-N-Azetidinyl-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one 9-OH-risperidone 9-pentyl-N-(piperazin-1-ylmethyl)-9H-carbazole-3-carboxamide 9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[1,2-a]purine-2,4(1H,3H)-dione 9-Phenyladenines 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 9-tert-Butyl-4-cyclohexyl-1-(4-methoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione 9-THA 9-[(1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]-3-(4-chlorophenyl)-3,9-diazabicyclo[4.2.1]nonane 93 96 97D76 98 99 9a 9b a A 348441 A 35043 A 36569 A 37843 A 37850 A 38120 A 98593 A(pF-F)R(ChA)(hR)(I-Y)-NH2 A, 2, 3-dihydroamentoflavone A-151892 A-159470 A-304121 A-312110 A-317344 A-317491 A-317920 A-331440 A-349821 A-54741 A-57282 A-70874 A-71623 A-80426 A-81754 A-84543 A-85380 A-85380,5-Iodo A-85380-I A-86929 A-94224 A-98795 A68930 A77636 AB-MECA AB-NECA ABA Abecarnil ABHD-I ABT-089 ABT-229 ABT-239 ABT-418 ABT-594 ABT-702 AC 915‚HCl AC-90179 Ac-c[Cys-Glu-His-D(2')Nal-Arg-Trp-Gly-Cys]-Pro-Pro-Lys-Asp-NH2 Ac-c[Cys-Gly-Gln-Leu-Ala-Asp-Gly-Cys]-NH2 Ac-DPhe-Leu-Arg-Ile-Arg-Pro-Arg-OH Ac-DPhe-Leu-Arg-Ile-Arg-Pro-Lys-OH Ac-DPhe-Nle-Arg-Nle-Arg-Pro-Arg-OH Ac-Nle-c[Asp-Acpc-DNal(2') Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Aic-DNal(2')Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Che-DNal(2') Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Cpe-DNal(2') Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-His-DNal(2')Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Hyp-DNal(2')Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Ioc-DNal(2')Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Oic-DNal(2') Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Pro-DNal(2'Arg-Trp-Lys]-NH2 Ac-Nle-c[Asp-Tic-DNal(2')Arg-Trp-Lys]-NH2 Ac-Phe-Leu-Arg-Ile-Arg-Pro-Arg-OH Ac-Phe-Leu-Arg-Ile-Arg-Pro-DLys-OH Ac-Phe-Leu-Arg-Ile-Arg-Pro-Lys-OH Ac-Phe-Nle-Arg-Nle-Arg-Pro-Arg-OH Ac-pTyr-Cha-Pro-Gln-Thr-NH2 Ac-pTyr-Ile-Pro-Gln-Thr-NH2 Ac-pTyr-Leu-1Ac6c-Gln-Thr-NH2 Ac-pTyr-Leu-4-hydroxy-Pro-Gln-Thr-NH2 Ac-pTyr-Leu-alphaMe-Pro-Gln-Thr-NH Ac-pTyr-Leu-Azt-Gln-Thr-NH2 Ac-pTyr-Leu-cis-3,4-methanoPro-Gln-Thr-NH2–1 Ac-pTyr-Leu-cis-3,4-methanoPro-Gln-Thr-NH2–2 Ac-pTyr-Leu-Cmpi-Gln-Thr-NH2 Ac-pTyr-Leu-D-Pro-Gln-Thr-NH2 Ac-pTyr-Leu-Inp-Gln-Thr-NH2 Ac-pTyr-Leu-Nip-Gln-Thr-NH2-1 Ac-pTyr-Leu-Nip-Gln-Thr-NH2-2 Ac-pTyr-Leu-Pip-Gln-Thr-NH2 Ac-pTyr-Leu-Pro-3-carboxamidoanilide Ac-pTyr-Leu-Pro-3Ac6c-NH2 Ac-pTyr-Leu-Pro-Ahx Ac-pTyr-Leu-Pro-Cmpi-NH2 Ac-pTyr-Leu-Pro-Gaba Ac-pTyr-Leu-Pro-Gln(Me2)-Thr-NH2 Ac-pTyr-Leu-Pro-Gln-N-MeThr-NH2 Ac-pTyr-Leu-Pro-Gln-NH2 Ac-pTyr-Leu-Pro-Gln-OH Ac-pTyr-Leu-Pro-Gln-Thr-NH2 Ac-pTyr-Leu-Pro-Gln–NEt2 Ac-pTyr-Leu-Pro-Gln–NH(R)CHMePh Ac-pTyr-Leu-Pro-Gln–NH(S)CHMePh Ac-pTyr-Leu-Pro-Gln–NHBn Ac-pTyr-Leu-Pro-Gln–NHMe Ac-pTyr-Leu-Pro-Gln–NMe2 Ac-pTyr-Leu-Pro-Gln–piperidine Ac-pTyr-Leu-Pro-Gln–pyrrolidine Ac-pTyr-Leu-Pro-Glu(Me)-Thr-NH2 Ac-pTyr-Leu-Pro-Inp-NH2 Ac-pTyr-Leu-Pro-Met(O)-Thr-NH2 Ac-pTyr-Leu-Pro-Met(O2)-Thr-NH2 Ac-pTyr-Leu-Pro-Nip-NH2 Ac-pTyr-Leu-Pro-PyA-NH2 Ac-pTyr-N-MeLeu-Pro-Gln-Thr-NH2 Ac-pTyr-Nle-Pro-Gln-Thr-NH2 Ac-pTyr-Phe-Pro-Gln-Thr-NH2 Ac-pTyr-Phe2Ala-Pro-Gln-Thr-NH2 Ac-pTyr-Val-Pro-Gln-Thr-NH2 Ac-RYYKWK-NH2 Ac-RYYKWR-NH2 Ac-RYYRIK-NH2 Ac-RYYRWK-NH2 Ac-RYYRWR-NH2 Acamprosate acebutolol aceclidine,R(-) aceclidine,S(+) Aceperone acetaminophen acetazolamide Acetic acid (R)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester acetic acid (R)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester Acetic Acid 1-acetoxymethyl-4-(2-chloro-6-methylamino-purin-9-yl)-bicyclo[3.1.0]hex-2-yl Ester Acetic Acid 2-acetoxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester Acetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl... Acetic acid 4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-8,8-dimethyl-3,5,11-trioxo-4-aza-tricyclo[5.2.2.0*2,6*]undec-1-... ACETOPHENAZINE Acetyl Beta-methylcholine Acetyl-His1-PACAP-27 Acetyl-His1-VIP Acetyl-L-Carnitine HCl Acetylcholine Acetylenic GABA-7 Acetylsalicylic acid Acetylthiocholine Ach AcNH-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH2 AcNH-4-NO2-Phe-c[D-Cys-Tyr-D-Trp-Lys-Thr-Cys]-Tyr-NH2 ACP-103 ACPA ACPA Acrylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-y... ACT-058362 ACTH-(1-10) ACTH-(1-39) ACTH-(4-10) AD-5423 ADAM adamantan-1-yl-[3-(1H-indol-4-yloxy)-2-methoxy-propyl]-amine Adamantane-1-carboxylic acid ((S)-1-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-2,5-dioxo-pyrrolidin-3-yl)-amide Adenine-beta-D-arabinofuranoside Adenosine monophosphate Adenosine triphosphate adenosine-5'-N-ethyluronamide Adenosine-N1-oxide Adinazolam Ado-5'-(2-hydroxyethyl)carboxamide Ado-5'-carboxamide Ado-5'-cyclohexylcarboxamide Ado-5'-cyclopropylcarboxamide Ado-5'-ethylcarboxylate Ado-5'-methylcarboxamide ADP ADP, alpha beta-me ADP, Beta S ADPD ADR40-43, CGRP30-34, ADR50-52 ADR40-43, CGRP30-37 ADR40-49, CGRP35-37 Adrenaline Adrenaline, (-) Adrenaline,(+) Adrenaline,(R),(-) Adrenomedullin ADT ADTN ADTN 5,6 ADTN 6,7 ADTN DIMETHYL 5,6 ADTN DIMETHYL 6,7 ADTN DIPROPYL 6,7 ADTN, (+) AF-DX 116 AF-DX 116,(+/-) AF-DX 250 AF-DX 384 AF2 Agmatine AGN 190910 AGN 190911 AGN 191088 AGN 191365 AGN 191366 AGN 191995 AGN 192151 AGN 194394 Agomelatine AH-13205 AH-23848 AH-23848,(-) AH-6809 AI-OH-DP,(+) AI-OH-DP,(-) AIDA AIDC AJ119,(+) AJ76 AJ76(+) AKUAMMIGINE AL-37350A Ala11-SRIF-14-amide Ala6-SRIF-14-amide Ala7-SRIF-14-amide Ala8,Ava14,15 Alanine-beta Alaproclate Albendazole Albuterol Alcuronium alcuronium Alfuzosin Alinidine Allopregnanolone Alloxazine Allylnormetazocine, (+) almokalant ALNESPIRONE Alniditan alpha MSH alpha, beta methylene adenosine triphosphate alpha,O-di-methyl-5-hydroxytryptamine alpha-(-)-Acetylmethadol alpha-(S)-[[[[3-[[(10(S)-Cyclohexyl-8,11-dioxo-2-oxa-9,12-diazabicyclo[13.3.1]nonadeca-1(19),15,17-trien-13(S)-yl)carbonyl]am... alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionic acid alpha-Amino-3-hydroxy-5-tert-butyl-4-isoxazolepropionate Alpha-BGT Alpha-Btx Alpha-bungarotoxin Alpha-Cobratoxin Alpha-Conotoxin MII alpha-ddCHA Alpha-Dimethylhistane-alpha alpha-Ergocryptine alpha-Estradiol alpha-fluoro phosphonate Alpha-Helical CRF alpha-keto phosphonate alpha-M-5-HT Alpha-methyl p tyrosine alpha-Methyl-(+)norepinephrine,(+/-) alpha-Methyl-(+/-)norepinephrine,(+/-) alpha-Methyl-(-)norepinephrine,(+/-) alpha-methyl-5-hydroxytryptamine alpha-Methylbenzeneethanamine alpha-Methylbenzeneethanamine,(+) alpha-methylene phosphonate alpha-methylhistamine Alpha-Methylhistamine-R Alpha-Methylhistamine-S Alpha-Methylhistane-R Alpha-Methylphenethylamine Alpha-methyltryptamine, (+) alpha-MSH, [Nle4, D-Phe7] alpha-MSH, [Nle4] Alpha-Neoendorphin alpha-OH biphosphonate alpha-tetrahydropyran-beta-sulfone Alpidem Alprazolam ALPRENOLOL ALPRENOLOL,(+) ALPRENOLOL,(-) alsterpaullone ALTANSERIN Alytesin AM 251 AM2233 AM3661 AM3677 AM630 AMAA Amantadine Ambenyl AMDA Amentoflavone AMESERGIDE AMFONELIC ACID AMI-098 AMI-193 Amiloride amino-norchloro-epibatidine aminoacetic acid Aminoclonidine, p Aminoethanoic acid Aminoethylpyridine-2 Aminoguanidine aminopotentidine Aminopropanesulfonic-3 Aminopropyl-cyclohexylamine Aminorex Aminotetralin-6,7-dihydroxy-(+) Aminotetralin-6,7-dihydroxy-(-) aminotetralin-6,7-diol Amiodarone Amisulpride AMITRIPTYLINE amlodipine AMN107 AMOA AMOXAPINE AMOXIPINE AMP AMPA AMPEROZIDE Amphetamine AMPHETAMINE, (D) Amphetamine,(+) Amphetamine,(-) Ampyrone amrinone amselamine AMT,(+) AMT,(-) amthamine Anabaseine Anabasine Anabasine, (+/-) ANANDAMIDE Anandamide + PMSF Anatoxin-a Anatoxin-A (+) Anatoxin-a (+_) Anatoxin-A,(+) androsterone Ang II 4-NH2-Phe6 Ang II Ile8, Sar1 Ang II Sar1 Ang II Thr8, Sar1 Ang III Ang IV Ang IV D-Val1 Ang IV Nor1 Ang(1-7) Ang(1-7) D-Ala7 Ang(2-7) Ang(3-10) Ang(3-11) Ang(3-4) Ang(3-5) Ang(3-6) Ang(3-7) Ang(3-9) Ang(4-8) Angiotensin II Anpirtoline Ant-CH2 (3,3)d Ant-CH2 (4,4) Ant-CH2CH2 (4,4) Ant-CH2CH2CH2 (4, 4) Antalarmin Antazoline Anti-endo-MPDC Antmethyl (3,3) Antmethyl(4,4) Aoct8,9,10 AP2A AP3A AP4A AP5A AP6A APEC APNEA APOMORPHINE Apomorphine,(+) Apomorphine,(-) Aprophen AQ-RA 741 Arachidonic acid Arachidonyl cyclopropylamide Arachidonyl-2-chloro-ethylamide arachidonylcyclopropylamide ARC-239 Arcaine Arecoline Arginine vasopressin ARIPIPRAZOLE Arodyn Arotinolol Arpromidine Arterenol Artrenolol ARVANIL AS-19 Asenapine Asperlicin ASTEMIZOLE Astressin ATC0065 ATC0175 ATENOLOL ATIPAMEZOLE Atomoxetine Atorvastatin Atorvastatin lactone Atosiban ATP ATP, 2-meS ATP, alpha, beta methylene ATP, Bz ATP,2',3'-dideoxy ATP,2'-deoxy ATP,3'-deoxy ATP,Beta Gamma-me ATP,Gamma S ATP,TNP ATPA ATPA-R ATPA-S ATR Atracurium Atracurium ATROPINE Atropine,(-) AUKAMMIGINE Ava14,15 Ava9,10 Ava9,10,Ava14,15 AVP Azabicyclo[2.2.1]heptane AZAPERONE AZAPETINE azatidine azepan-1-yl(5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-yl)methanone azepinoindoline azepino[4,5-b]indole azetidine azimilide ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate ±)-(4aS,8R,8aS)-(4aS,8R,8aS)-2-benzyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide ±)-(4aS,8R,8aS)-1-oxo-2-(4-(trifluoromethyl)benzyl)-N-(4-(trifluoromethyl)phenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-... ±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide ±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid ±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-8-(piperidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one ±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS... ±)-(4aS,8R,8aS)-2-benzyl-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one ±)-(4aS,8R,8aS)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one ±)-(4aS,8R,8aS)-N,2-dibutyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide ±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide ±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamid... ±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-o... ±)-(4aS,8R,8aS)-N-(thiazol-2-yl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (Â... ±)-2,5-Dimethoxy-4-bromoamphetamine ±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate b-FNA-HCl B-HT 920 B-NECA B8-DL-B8 B8-DL-B8 (low PS) Baclofen Baclofen, (R)(-) Baclofen, (S)(+) BAM 1303 BANISTERINE banyu 6 basilen blue Bay 36-7620 BAY 38-7271 BAY 59-3074 Bay k 8644 BAY u9773 BAY X 9228 BAY-43-9006 BAY36-7620 BCCE BCCt BCTC BD1008 BDF6143 BE-2254 BE2254 BE4444 Benoxathian BENPERIDOL Benzamidine Benzamil Benzedrone Benzeneethanamine, alpha-methyl-, (±)- Benzeneethanamine, alpha-methyl-, (S)- Benzhexol Benzofuran-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-propyl-amino]-ethyl}-cyclohexyl)-amide benzofuranyl Benzoic Acid 2-acetoxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester Benzoic Acid 2-benzoyloxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester Benzoic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonooxymethyl-propyl Ester, Ammonium Salt benzooxazol-2-yl-[1-(3-isobutoxy-4-methoxy-benzyl)-piperidin-4-yl]-amine Benzotript Benzoxacole N-methylation Benzoyl-pTyr-Leu -Pro-Gln-Thr-NH2 Benzo[1,3]dioxole-5-carboxylic Acid {(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethy... Benzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol Benzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide Benzo[g]quinoline-1-propyl-7,8-diol-trans(+-) Benzquinamide BENZTROPINE benzyl ((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate(±)-((4aS,8R,8aS)-2-... benzyl ((4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate(±)-((4aS,8R,... benzyl ((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate(±)-((4aS,8R,8aS)-2-(3,... benzyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-... benzyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalaninate benzyl (±)-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate benzyl (±)-((4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalaninate benzyl (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalaninate benzyl (±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalaninate Benzyl 1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-Beta-carbolin-6-yl Ether Benzyl 4-[(2-cyclohexylidene-2-fluoroethyl)amino]-1-piperidinecarboxylate Benzyl-NECA benzylamine Benzyloxycarbonyl CCK(27-32)NH2 Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate Bepridil BERAPROST Beta C N A Beta CCE Beta CCM Beta CCP Beta MSH beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl) beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-L-3(phenylmethyl) Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl) Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-( 1-S- trans) Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are tran... Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1-R-trans) Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans) Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1S-trans) Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring centers are trans (... beta-aminopropylbenzene beta-Casomorphin Beta-CCT Beta-CDIT Beta-CIT beta-D-Psicofuranosyladenine Beta-Endorphin Beta-Endorphin (6-31) Beta-Endorphin, des-Tyr beta-funaltrexamine Beta-Funeltrexamine Beta-L-adenosine Beta-LT beta-methyl-APB Beta-Methylhistamine Beta-Neoendorphin Beta-PEA Beta-Phenethylamine Beta-Phenylaethylamin (GERMAN) Beta-Phenylethylamine BETAXOLOL Bethanechol BHT-933 BIBO3304 BIBP3226 bicalutamide Bicuculline Bicuculline methochloride,(+/-) Bicuculline,(+) bifeprunox Bifeprunox BIIE0246 BIIL-260 BIIL-284 BIIL-315 BIM 23003 BIM 23014 BIM 23023 BIM 23027 BIM 23030 BIM 23034 BIM 23042 BIM 23049 BIM 23050 BIM 23051 BIM 23052 BIM 23053 BIM 23055 BIM 23056 BIM 23057 BIM 23058 BIM 23059 BIM 23060 BIM 23063 BIM 23064 BIM 23065 BIM 23066 BIM 23067 BIM 23068 BIM 23069 BIM 23070 BIM 23073 BIM 23197 BIM 23268 BIM 23295 BIM 23313 BIM-23190 BIM-23208D BIM-23745 BIM-23926 BIMT 17 BIMU 1 BIMU 8 Bip-Ala-Thr-Pro-Lys-Thr(OBzl)-Gly Bip-Tyr(3'Bzl)-Thr-Pro-Lys-Thr Bip-Tyr-Ala-Pro-Lys-Thr(OBzl)-Gly Bip-Tyr-Thr(OBzl)-Pro-Lys-Thr-Gly Bip-Tyr-Thr-Ala-Lys-Thr(OBzl)-Gly Bip-Tyr-Thr-Ala-Thr(OBzl)-Gly Bip-Tyr-Thr-Pro-Ala-Thr(OBzl)-Gly Bip-Tyr-Thr-Pro-Lys-Thr Bip-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly Bip-Tyr-Thr-Pro-Phe Bip-Tyr-Thr-Pro-Thr(OBzl)-Gly Biperiden Biperidine Biphalin Biphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide BIRB-796 Biscaline Bismuth subsalicylate Bisoprolol BL 6341A Blephamide Blonanserin BM 13177 BM 13505 BM 573 BM 613 BMS181,101 BMY 13980 BMY 14802 BMY 7378 BN 52021 BNTX Boc-CCK-4 BOL 146 boldine Bombesin Bombesin, SAP Bombesin,Phe13 BOSENTAN Botiacrine BP-897 Bpa-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly Br-6-APT Br-HIBO Br-HIBO,(R) Br-HIBO,(RS) Br-HIBO,(S) Bradykinin Brassinin Bremazocine BREMAZOCINE(-) Bretazenil Brexpiprazole Brimonidine AppNHp Brimonidine ATP Brimonidine GppNHp Brimonidine GTP brinzolamide BRL 15572 BRL 24682 BRL 24924 BRL 34778 BRL 37344 BRL 43694 BRL 47204 BRL44408 Bromanyl bromo-norchloro-epibatidine BROMOCRIPTINE Bromocriptine+ (GTP+) Bromocriptine+ (GTP-) BROMOCRIPTINE,(+) Bromodiphen-hydramine Bromoperidol BROMPERIDOL Brompheniramine Bromphenol blue Brophenol Blue Brotizolam Broxaterol BS-DMPX BTM1086 BTS 54 354 BTS 54 505 BU 46 BU 47 BU 61 BU 95 BU 96 BU-E 47 Bu-HIBO Budesonide BUDIPINE BUFOTENINE BUFOTENINE METHYL ETHER BULBOCAPNINE Bungarotoxin Neuronal Bungarotoxin,Alpha BUPRENORPHINE Buprenorphine(+) Buprenorphine(-) BUPROPION Burimamide BUSPIRONE But-2-enoic Acid 2-but-2-enoyloxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester butabindide BUTACLAMOL BUTACLAMOL, (-) BUTACLAMOL,(+) BUTACLAMOL,d- Butanoic acid, 4-amino- Butanserin BUTAPROST Butaprost (Free Acid) Butaprost (Methyl Ester) Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpr... Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpr... Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpr... Butorphanol Butorphanol Butoxamine butriptyline butylamide benzthiophene Butylone Butyric acid, 4-amino- Butyrylfentanyl BW-1 BW-723C86 BW-A1433 BW245C BW284C51 BW373U86 BW501 BW868C BWA1433 BWA868C C-(3-Bromo-9,10-dihydro-anthracen-9-yl)-methylamine C-(3-Hexyl-9,10-dihydro-anthracen-9-yl)-methylamine C-(9,10-Dihydro-anthracen-9-yl)-methylamine C-[3-(2-Dimethylamino-ethyl)-1H-indol-5-yl]-N-[4-({[3-(2-dimethylamino-ethyl)-1H-indol-5-ylmethanesulfonyl]-methyl-amino}-met... C-[3-(3-Phenyl-propyl)-9,10-dihydro-anthracen-9-yl]-methylamine C1 C1-HIBO C1-IB-MECA C10H14BrNO3 C12H11FN2O·C4H4O4 C12H12N2O·C4H4O4 C12H12N4 C12H14N2O2·C4H4O4 C12H18ClNO3 C13H14F2N2·0.5C4H4O4 C13H14N2·C4H4O4 C13H14N2O·C4H4O4 C13H15FN2·0.5C4H4O4 C13H16ClNO3 C13H16N2·0.5C4H4O4 C13H16N2O·C4H4O4 C14H14N2·C4H4O4 C14H15ClN2·C4H4O4 C14H15FN2·C4H4O4 C14H16N4 C14H16N4O2 C14H22ClNO3 C15H15F3N2·C4H4O4 C15H16N2·C4H4O4 C15H16N2O·C4H4O4 C15H18N2·C4H4O4 C15H18N2O·C4H4O4 C15H18N402 C15H19N5O4 C15H20N2·C4H4O4 C15H22ClNO3 C16H15ClN5O4H2O C16H17BrClNO3 C16H17ClINO3-0.25H2O C16H18ClNO3 C16H18ClNO4-0.25H2O C16H20N2·0.5C4H4O4 C16H21N5O4 C16H23ClNO4 C16H24ClNO3 C16H26ClNO3-0.3H2O C17H14N40 C17H20ClNO3 C17H20ClNO4 C17H20ClNO4-0.5H2O C17H22N402 C17H22N6O4 C17H23N5O4 C18H15N9O3 C18H16N2O·C4H4O4 C18H22ClNO3 C18H22ClNO4 C18H25N5O4 C18H28ClNO3 C19H17N9O3 C19H18N40z*3/zHz C19H21ClN5O4 C19H23ClN2S dimaleate (54) C19H23ClN2S hemifumarate (54, +) C19H23ClN2S hemifumarate (54, -) C19H23N7O4 C19H24C1N7O4 C19H26ClNO3 C19H28ClNO3 C19H30ClNO4-.05H2O C2 c2,2′(Dmt-DCys-Gly-Phe)2-cystamine c2,2′(Dmt-DCys-Gly-Phe)2-piperazine c2,2′(Tyr-DCys-Gly-Phe)2-cystamine c2,2′(Tyr-DCys-Gly-Phe)2-piperazine c2,2′(Tyr-DPen-Gly-Phe)2-piperazine c2,2′(Tyr-DPen-Gly-Phe-NH-)2 c2,2′(Tyr-DPen-Gly-Phe-NH-)2. C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester C20H24FN704 C20H24FN7O4 C20H25Cl2N7O4 C20H25ClN2S 2HCl 0.7H2O (55) C20H25N7O4 C20H28ClNO3 C20H30ClNO3 C21H24ClFN2 dimaleate (27) C21H24ClFN2 fumarate (41, +) C21H24ClFN2 fumarate (41, -) C21H24ClFN2 hemifumarate (41) C21H26ClN7O4 C21H27CIN7O4 C21H27ClN7O4 C22H24F4N2 (43) C22H26BrFN2 1.5fumarate (42) C22H26C1N7O6 C22H26Cl2N2 dioxalate 0.5H2O (53) C22H26ClFN2 (48) C22H26ClFN2 1.3oxalate (49) C22H26ClFN2 dihydrochloride (28, +) C22H26ClFN2 dihydrochloride (28, -) C22H26ClFN2 dimaleate (26) C22H26ClFN2 dimaleate (51) C22H26ClFN2 dimaleate (52) C22H26ClFN2 dioxalate (25) C22H26ClFN2 dioxalate (47) C22H26ClFN2 maleate (28) C22H26F2N2 dimaleate (40) C22H26F2N2 fumarate (40, +) C22H26F2N2 fumarate (40, -) C22H26F2N2 oxalate (50) C22H27ClN2 1.5maleate (38) C22H27ClN2 fumarate (38, +) C22H27ClN2 fumarate (38, -) C22H27FN2 (45) C22H27FN2 dimaleate (39) C22H27FN2 fumarate (39, +) C22H27FN2 fumarate (39, -) C22H28CIN7O7 C22H28ClN7O6 C22H28N2 dimaleate (37) C23H24ClNO3 C23H26ClFN2 dihydrochloride 0.5H2O (33) C23H26ClFN2 dimaleate (24) C23H26F4N2 (44) C23H28ClFN2O (30) C23H29FN2 (46) C23H30ClNO3 C24H28ClFN2 dihydrochloride (34, - ) C24H28ClFN2 dihydrochloride (34, -) C24H28ClFN2 dihydrochloride 0.4H2O (34, +) C24H28ClFN2 fumarate (34) C24H30ClFN2 dioxalate (29, -) C24H30ClFN2 dioxalate 0.8H2O (29) C24H30ClFN2 oxalate (32) C24H30ClFN2O dioxalate (31) C24H30CLlFN2 dioxalate (29, +) C24H30CLlFN2 dioxalate (29, -) C25H30ClFN2 dihydrochloride (36) C25H30ClFN2O 1.8hydrochloride (35) C25H30ClFN2O dihydrobromide 0.6H2O (35, +) C25H30ClFN2O dihydrobromide 0.6H2O (35, -) C25H30CLlFN2 dihydrochloride (36) C28H32NClO C29H41N11O5S2 C3 C30H36NO3 C30H43N11O5S2 C31H43N11O5 C32H46N11O5 C33H47N11O5 C36H50Cl2N6O9•0.75H2O), C, H, N C37H49N11O6S2 C38H51N11O6S2 C39H51N11O6 C4 C42H62Cl2N6O8•0.75H2O), C, H, N C44H54N11O10 C45H56N11O10 C49H63N12O11 C5 C50H65N12O11 C51H67N12O11 C54H76NO5 C54H76NO6 C54H76NO7 C54H80NO8 C55H74N2O9 C55H77N2O8 C55H77NO7 C55H78NO7 C56H79N2O8 C56H80N3O7 C56H80NO8 C56H81N2O8S C56H81N2O9S C57H79N2O9 C57H79N2O9Na C57H81N2O7 C6 C7 C8 Cabergoline CACA CaCl2 CACO Caerulein caffeine Caffeine (1,3,7-trimethylxanthine) CAM Camel Snus extract Camptosar camptothecin CANDESARTAN Cannabinol Capsaicin capsazepine captopril CARAMIPHEN CARAZOLOL CARBACHOL CARBACYCLIN CARBAMAZEPINE Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexy... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexy... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexy... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl... Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl... carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]- cyclohexyl ester carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]-2-chlorocyclohexyl ester trans (+/-) Carbamoyl-des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS(sst3-ODN-8) Carbamylcholine Carbendazim CARBETAPENTANE Carbinoxamine Carbonic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phenoxycarbonyloxy-methyl-propyl Ester Phenyl Ester Carbonic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonooxymethyl-propyl Ester Ethyl Ester, Ammonium Salt Carboperamide Cariprazine carmoterol Carpipramine Carprofen Cartazolate Carvedilol catechin Cathinone Cathinone, (-) CBD CBD, abnormal Cbz-pTyr-Leu -Pro-Gln-Thr-NH2 Cc-25,(+/-) Cc-34,(+/-) CCDC 710249, HCl salt CCI19234 CCK CCK-(26-29)-tetrapeptide CCK-(30-32)-tripeptide CCK-8 CCK2 CCK3 CCK33 CCK4 CCK4 acid CCK8 CCK8 acid CCPA CD CD-214 CDP 840 CELECOXIB Cerivastatin Cetapred Cetirizine Cetirizine (+) isomer Cetirizine (-) isomer CF 25-397 CF3-5-APT CF3-6-APT CFR (12-41),DPhe12,Nle21,38-r/h CFR (9-41),Alpha-helical CFR,r/h CFT CGP 12177 CGP 20712 CGP 20712-A CGP 23996 CGP 361A CGP 42112 CGP 71683A CGP 71863 CGP27492 CGP34938 CGP35024 CGP35348 CGP35582 CGP35832 CGP36216 CGP36742 CGP38593 CGP44530 CGP47656 CGP49713 CGP70522 CGP70523 CGP71683A CGRP 27-37 CGRP Ac-27-37 CGRP Y0-28-37 CGRP Y0-29-37 CGRP Y0-30-37 CGRP26-29, ADR44-49, CGRP35-37 CGRP26-29, ADR44-52 CGRP26-34, ADR50-52 CGRP26-34, IAPP35-37 CGS 12066A CGS 12066B CGS 15943 CGS 19755 CGS 20625 CGS 21577 CGS 21680 CGS 23113 CGS 23114 CGS 23130 CGS 23131 CGS 23167 CGS 23356 CGS 24115 CGS 25019 C CGS 8216, 1 CGS 9895 CGS 9896 CGS10746B CGS19281A CGS21680 CGS8216 CGS9895 CGS9896 CH275 CH2OCOC(CH3)3 CHA Chantix Chelerytherine Chlorcyclizine CHLORDIAZEPOXIDE CHLORETHYLCLONIDINE CHLORIMIPRAMINE Chlorisondamine chloronicotine-6 Chloroptic-p s.o.p. Chloroquine CHLORPHENIRAMINE CHLORPHENIRAMINE-d chlorpheniramine-l Chlorphentermine chlorproethazine CHLORPROMAZINE chlorpromazine CHLORPROMAZINE-N-OXIDE CHLORPROTHIXENE Chlorprothixene (cis) Choline CHPG CHPG(RS) CHPG(S) CI 218872 CI-1015 CI-1033 CI-988 CI-996 CI-IB-MECA CI9Hl8N4O2H Cibacron blue CICAPROST ciclesonide cilanseton cilansetron Cilomilast Cimbi-712 Cimbi-717 Cimbi-772 Cimbi-775 Cimbi‐701 CIMETIDINE CINANSERIN cinnarizine CINUPERONE Cipralisant Ciproxifan cirazoline Cirazoline cis 1-hydroxyindane CIS PIFLUTIXOL cis piflutixol-(Z) CIS TEFLUTIXOL cis-(+/-)-2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one Cis-(+/-)-2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-propyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl-4a,5,8,8a-tetrahydro-2H-phtha... cis-(+/-)-2-{5-[3-(5-fluoro-2-methoxyphenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl]-4,5,8,8a-tetrahydro-2H-phthala... cis-(3'R)-Quinuclidin-3'-yl 4-Hydroxy-1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine cis-1,2-bis(4-chlorophenyl)-5-(3,4-difluorobenzyl)piperidine cis-1,6-bis(4-chlorophenyl)-3-(3,4-difluorobenzyl)piperidin-2-one cis-1-(Aminomethyl)-3-cyclohexyl-3,4-dihydro-5,6-dihydroxy-1H-2-benzopyran Hydrochloride cis-1-methyl-1-phenyl-3-(dimethylamino)tetralin cis-1-[(Allylamino)methyl]-3-cyclohexyl-3,4-dihydro-5,6-dihydroxy-1H-2-benzopyran Hydrochloride cis-2,5-Dicarboethoxy-1-[4-chlorophenyl]pyrrolidine cis-2,6-Dimethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine cis-2,6-Dimethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine cis-2,6-Dimethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine cis-2,6-Dimethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine cis-2-(3-Pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-(5-(Benzyloxy)pyridin-3-yl)octahydropyrrolo[3,4-c]pyrrole cis-2-(5-Bromopyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate cis-2-(5-Ethoxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-(5-Hydroxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-(5-Methoxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-(5-Phenyl-pyridin-2-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate cis-2-(5-Phenylpyridin-3-yl)-5-methyl-octahydro-pyrrolo[3,4-c]-pyrrole Sesqui-fumarate cis-2-(5-Phenylpyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bistrifluoroacetate cis-2-(6-Biphenyl-3-yl-pyridin-3-yl)-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole p-Toluenesulfonate cis-2-(6-Chloro-3-pyridinyl)-5-methyloctahydropyrrolo[3,4-c]-pyrrole cis-2-(6-Chloro-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Hydrochloride cis-2-(6-Phenyl-pyridazin-3-yl)-5-methyloctahydro-pyrrolo[3,4-c]-pyrrole cis-2-(6-Phenyl-pyridazin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate cis-2-(6-Phenyl-pyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate cis-2-(Pyridin-2-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate cis-2-(Pyridin-4-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate cis-2-Biphenyl-4-yl-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-Biphenyl-4-yl-octahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate cis-2-Ethyl-5-(6-phenyl-pyridazin-3-yl)-octahydro-pyrrolo[3,4-c]-pyrrole Bis-p-toluenesulfonate cis-2-Methyl-5-(3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-Methyl-5-(5-phenyl-pyridin-2-yl)-octahydro-pyrrolo[3,4-c]pyrrole 4-Toluenesulfonate cis-2-Methyl-5-(6-(2-methylphenyl)pyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole Bis-L-tartrate cis-2-Methyl-5-(6-(3-methylphenyl)pyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-Methyl-5-(6-(4-methylphenyl)pyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-Methyl-5-(6-m-tolyl-pyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-L-tartrate cis-2-Methyl-5-(6-phenyl-pyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole L-Tartrate cis-2-Methyl-5-[6-(3-nitrophenyl)-pyridin-3-yl]-octahydro-pyrrolo[3,4-c]pyrrole p-toluenesulfonate cis-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol cis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 4-hydroxy piperid-1-yl] 5-fluoroindan-1-01 cis-2-[6-(3,5-(Dimethylphenyl)pyridazin-3-yl]-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole Dihydrochloride cis-2-[6-(3-Methoxy-phenyl)-pyridin-3-yl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole Bis-L-tartrate cis-2-[6-(4-Methoxy-phenyl)-pyridazin-3-yl]-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole p-Toluenesulfonate cis-2a cis-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile cis-3-(5-Isopropyloxy-3-pyridinyl)-3,7-diazabicyclo[3.3.0]octane Semi(fumarate) cis-3-(5-Propyloxy-3-pyridinyl)-3,7-diazabicyclo[3.3.0]octane Semifumarate cis-3-aminocyclopentane-1-carboxylic acid,(+/-) cis-3-Cyclohexyl-3,4-dihydro-5,6-dihydroxy-1-(methylamino)methyl-1H-2-benzopyran Hydrochloride cis-3-[6-(5-Methyl-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl)-pyridazin-3-yl]-phenol dihydrochloride cis-4-(5-(Hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)pyridin-3-yl)morpholine Sesqui-fumarate cis-4-aminocrotonic acid cis-4-[6-(5-Methyl-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl)-pyridazin-3-yl]-phenol Bis-p-toluenesulfonate cis-5-(6-Bromo-pyridin-3-yl)-hexahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate cis-5-(6-Chloropyridin-3-yl)-2,2-dimethyloctahydropyrrolo[3,4-c]-pyrrol-2-ium Iodide cis-5-(6-Phenylpyridazin-3-yl)-2,2-dimethyloctahydropyrrolo[3,4-c]pyrrol-2-ium Iodide cis-5-[6-(5-Methyl-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl)-pyridazin-3-yl]-1H-indole Bis-p-toluenesulfonate cis-benzocycloheptyl-PAT cis-Clopenthixol cis-CPCA, - cis-flupenthixol cis-H2-PAT(+) cis-H2-PAT(+/-) cis-H2-PAT(-) cis-methyl-{1-[3-(pyridin-3-yloxy)-propenyl]-cyclopropyl}-amine; hydrochloride cis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine cis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine cis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine cis-N-Benzyl-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1′-cyclohexan]-4′-amine cis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine cis-N-Benzyl-3-methoxy-N-methyl-3,4-dihydrospiro-[[2]benzopyran-1,1′-cyclohexan]-4′-amine Cis-N-Methyl-2'-methyl-2',3'-dihydrofuro[m]aporphine cis-N-oleoylcyclopropanolamide cis-PAB cis-phenyl-2-aminotetralins cis-Thiothixene CISAPRIDE Cismethyl-dioxolane(+) CIT CITALOPRAM citansetron CK 204-933 CL-5-APT CL-6-APT Cl-diazepam,4 CL218,872 Cl5HI8N4O Cl7HI4N4O2H CLEBOPRIDE Clemastine clemizole Clenbuterol CllH10N40 Clobazam Clobenpropit clocinnamox CLOFLUPEROL CLOMIPRAMINE CLOMIPRIMINE Clonazepam CLONIDINE Cloperatine CLOPIMOZIDE CLOPIPAZAN CLOPROSTENOL CLORGYLINE CLOROTEPINE (+) CLOROTEPINE(-) CLOTHIAPINE Clovoxamine CLOZAPINE Clozapine N-oxide CLOZAPINE-N-OXIDE CM-A-82a CM-A-87 CM-A100 CM-A49 (R) CM-A50 (S) CM-A57 CM-A58 CM-A64 CM-A77 CM-A82a CM-A87 CM-B01 CM-B31c CM-B34 CM-B3li (ss) CM-B44 (ss) CM-B45 CM-B47 CM-C28 (SR) CM-D44 CM-D45 CM-D45 C19H21N3O4 CM-E09a CM-E09b CM-E10 CM-E11 CMA57 Cn4c(=O)c3c(nc2CN(Cc1ccc(Cl)c(Cl)c1)CCn23)n(C)c4=O Cn4c(=O)c3c(nc2CN(Cc1ccccc1)CCn23)n(C)c4=O CNQX Co 2-6749 COCAINE Cocaine (-) Codeine Codeine CODEINE SULFATE codeine-6-methyl ether codeinone Codrix Compound 1 Compound 2 compound 25 Compound 3 compound 33 Compound 4 compound 42 compound 43 Compound 5 Compound 6 COMPOUND I COMPOUND II Congo Red Cortalone Cortan CorticotropinReleasing Factor (12-41),DPhe12,Nle21,38-r/h CorticotropinReleasing Factor (9-41),Alpha-helical CorticotropinReleasing Factor,r/h Cortistatin cortistatin14 CORYNANTHINE cotinine Cotinine fumarate CP 122288 CP 154,526 CP 166866 CP 55,940 CP 62508 CP 93129 CP 99994 CP-101,606 CP-132,484 CP-132,484(4b) CP-24441 CP-394531 CP-409069 CP-409069 CP-465021 CP-465022 CP-471236 CP-471237 CP-51973 CP-52002 CP-52003 CP-526427 CP-55244 CP-55940 [(-)-AC],XIV CP-56667 [(+)-AC],XV CP-66,713 CP-68,247 CP-96,345 CP53261 CP55940 CP732925 CP760524 CP781214 CP8816 CP8863 CPA CPAP4 CPCA, + CPCCOEt CPG(S) CPP CPPG CPT CPW399, S CPX CPZ CR 1409 CRA1000 CRA1001 Crinone CROMAKALIM (-) CSC CST14 CST14-Tyr10 CST17 CTA2 CTAP CTAP-NH2 CTOP Curare CV 1808 CV-3988 CV-6209 CXCL10 CXCL11 CXCL9 Cyamemazine cyanogen bromide, CNBr CYANOPINDOLOL CYANOPINDOLOL(+) CYANOPINDOLOL(+/-) CYANOPINDOLOL(-) Cyclazocine Cyclazocine (+) CYCLAZOCINE (-) cyclo(-Nal-Gly-D-Tyr-Ala-Arg-) cyclo(-Nal-Gly-D-Tyr-Asn-Arg-) cyclo(-Nal-Gly-D-Tyr-cis-4-guanidino-Pro-Arg-) cyclo(-Nal-Gly-D-Tyr-D-Ala-Arg-) cyclo(-Nal-Gly-D-Tyr-D-MeAla-Arg-) cyclo(-Nal-GLy-D-Tyr-D-Pro-Arg-) cyclo(-Nal-Gly-D-Tyr-Dab-Arg-) cyclo(-Nal-Gly-D-Tyr-g-Dab-Arg-) cyclo(-Nal-Gly-D-Tyr-g-Lys-Arg-) cyclo(-Nal-Gly-D-Tyr-Gln-Arg-) cyclo(-Nal-Gly-D-Tyr-Glu-Arg-) cyclo(-Nal-Gly-D-Tyr-Lys-Arg-) cyclo(-Nal-Gly-D-Tyr-MeAla-Arg-) cyclo(-Nal-Gly-D-Tyr-Orn-Arg-) cyclo(-Nal-Gly-D-Tyr-Pro-Arg-) cyclo(-Nal-Gly-D-Tyr-trans-4-guanadino-Pro-Arg-) cyclo(6beta-10-)(succinyl6-D-(2')Nal7-Arg8-Trp9-Lys10)-NH2 Cyclo-(CH2-CO-Adi-Leu-(3'-CO2H-Tyr)- Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Adi-Leu-(3'-CO2H-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Adi-Leu-(3'-CO2H-Tyr)-Ac6c-Asn-Ava-Cys)-amide Cyclo-(CH2-CO-Adi-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Adi-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Adi-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Ava-Cys)-amide Cyclo-(CH2-CO-Adi-Leu-(3'-NO2-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Adi-Leu-(3'-NO2-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Adi-Leu-(3'-NO2-Tyr)-Ac6c-Asn-Ava-Cys)-amide Cyclo-(CH2-CO-Adi-Leu-(3'-OH-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Adi-Leu-(3'-OH-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Adi-Leu-(3'-OMe-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Adi-Leu-(3'-OMe-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Adi-Leu-(3'-OMe-Tyr)-Ac6c-Asn-Ava-Cys)-amide Cyclo-(CH2-CO-Adi-Leu-Tyr-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Adi-Leu-Tyr-Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Adi-Leu-Tyr-Ac6c-Asn-Ava-Cys)-amide Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)- Ac6c-Asn -Cys)-amide Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (R) Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Ava-Cys (O))-amide (S) Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Ava-Cys)-amide Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-beta-Ala-Cys (O))-amide (S) Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-beta-Ala-Cys(O))-amide (R) Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-beta-Ala-Cys)-amide Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Cys (O))-amide (R) Cyclo-(CH2-CO-Gla-Leu-(3'-NH2-Tyr)-Ac6c-Asn-Cys (O))-amide (S) cycloantagonist SA Cyclobenzaprine Cyclobutyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate Cyclobutylmethyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate Cyclohexanecarboxylic acid (1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-amide Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide cyclohexyl (±)-(4aR,8S,8aR)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate cyclohexyl (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate cyclohexyl (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate Cyclohexyl-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone Cyclohexyl-NECA Cyclopentamine Cyclopentolate Cyclopentyltheophylline Cyclopropanecarboxylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3... cyclopropyl-(4-(3-1H-imidazol-4-yl)propyloxy)phenyl) ketone Cyclorphan Cyclorphan,(-) Cyclosporin A Cyclo[(diaminoethylcarbamoyl)HyPro-Arg-D-Trp-Lys-Tyr(Bzl)-Phe] Cyclo[(diaminoethylcarbamoyl)HyPro-His-D-Trp-Lys-Tyr(Bzl)-Phe] Cyclo[(diaminoethylcarbamoyl)HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe] Cyclo[(diaminoethylcarbamoyl)HyPro-Phg-D-Trp-Lys-Tyr(Bzl)-Phe] Cyclo[(diaminoethylcarbamoyl)HyPro-Tyr-D-Trp-Lys-Tyr(Bzl)-Phe] Cyclo[(diaminopentylcarbamoyl)HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe] Cyclo[(N,N-dimethyldiaminoethylcarbamoyl)HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe cyclo[Ahep-Phe-DTrp-Lys-Thr(Bzl)] Cyclo[HyPro-Phe-D-Trp-Lys-Tyr(Bzl)-Phe] CYN-15486 Cyprodime CYPROHEPTADINE CYPROHEPTIDINE Cytidine Cytisine Cytisine-(-) d(CH2)5Tyr(Me)AVP D,L Kavain d,l-Bromopheniramine D,L-Trimipramine D-(S)-Amphetamine D-237 D-264 D-315 D-366 D-367 D-578 D-Ala2-MePhe4-Met(0)5-enkephalin-ol D-AP4 D-AP5 D-APB D-APV D-Arg6,Ava14,15 D-Arg6,Ava9,10 D-Arg6,Ava9,10,Ava14,15 D-Aspartate d-brompheniramine d-Butaclamol d-Chlorpheniramine D-Cys7,Ava14,15 D-cystine d-Fenfluramine D-Glu D-Glutamate D-homocysteic acid D-homocysteine sulfinic acid D-homocysteine thiolactone d-Isolysergic acid amide d-Lysergic acid amide D-lysergic acid diethylamide D-lysergic acid diethylamide (LSD) d-Methamphetamine D-methionine d-Metoprolol d-Nantradol d-Norfenfluramine D-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2 D-Phe-D-Phe-D-Nle-D-Arg-NH2 D-PheCRF D-PIA d-sotalol d-TA-3090 D-Thr6-D-Trp8,9)-galanin (1-5)ol D-Trimipramine D-Trp8 SST-14 D-Trp8-SRIF-14 d-Tubocurarine D600 D609 D888,(+) D888,(-) DABDMA DADLE DADLE-OH DAGO DALDA DALEA DALLE DAMGO Darifenacin DASB DAU 6215 DAU 6236 DAU 6285 DAU 6287 DB-10 DB-3-3 DB-7 DC-23-99 DC-25-100 DC-25-12 DC-25-20 DC23-60 DCG-IV DCUK-Ome DCUKA dDAVP ddCHA DDMV Decamethonium dechloroepibatidine-(+) dechloroepibatidine-(-) Dehydrocorybulbine, (2,9,10-Trimethoxy-13-methyl-6,7-dihydro-5H-isoquinolino[2,1-b] isoquinolin-7-ium-3-one Delta 103-104 Delta 105-110 Delta 111C Delta 13-16 Delta 17-20 Delta 2-4 Delta 21-24 Delta 25C Delta 26-28 Delta 29 Delta 30C Delta 31-32 Delta 328-330 Delta 33-36 Delta 331-332 Delta 5-8 Delta 9-12 Delta 9-THC delta MSH Delta-cortef Delta-Dome delta9 -tetrahydrocannabinol (THC) Delta9 -tetrahydrocannabinol (THC)) Delta9-Tetrahydro-6,6,9-trimethyl-3-pentyl-6H-dibenzo[b,d]pyran-1-ol Delta9-tetrahydrocannabinol Deltasone Deltorphin I Deltorphin II, ile(5,6)- DELTORPHIN-II Demethyl-ACPA Demethyl-AMPA DEPRENYL Dequalinium Dequalinium chloride Dermatop Dermorphin des(Ac-Arg6),Ava14,15 des-AA 1,2,4,5,12,13[D-2Nal8]-SS (ODN-8) des-AA 1,2,4,5,12,13[D-Cys3, D-Agl8(Me,2-naphthoyl)]-SS des-AA 1,2,4,5,12,13[D-Cys3,Tyr7, D-Agl8(Me,2-naphthoyl)]-SS des-AA 1,2,4,5,12,13[D-Trp8]-SS (ODT-8) des-AA 1,2,4,5,12,13[DAgl8(2-naphthoyl)]-SS des-AA 1,2,4,5,12,13[DAgl8(Me,2-naphthoyl)]-SS des-AA 1,2,4,5,12,13[Tyr7, D-Agl8(Me,2-naphthoyl)]-SS Des-AA10-17[Cys7,21, Pro34]-NPY Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26, Pro34]-NPY Des-AA11-18[Cys7,21,D-Lys9 (Ac), D-His26]-NPY Des-AA11-18[Cys7,21,D-Lys9 (Ac), Pro34]-NPY Des-AA11-18[Cys7,21,D-Lys9 (Ac)]-NPY des-CIC Des-His1-[Glu3]PACAP(1-38) desacetyl-alpha-MSH desArg6,Ava14,15 Desaza1TRH DESIPRAMINE Desmethylcitalopram Desmethyldesipramine Desmethylimipramine Desmethylpiclamilas Desmethylsertraline Desonate Desonide Desowen Desoxy-HEAT HCl desoxy-nor-ephedrine Desoxypipradol Desoxypipradrol Despiramine Desulfated CCK8 Desvenlafaxine DET,4-OH DET,5-MeO Devazepide dexamethasone dexchlorpheniramine dexefaroxan Dexetimide Dexmedetomidine Dexoxadrol Dextrallorphan Dextroamphetamine Dextromethorphan Dextromoramide Dextrorphan DFP DHA DHBA DHbetaE DHBetaE,D-Beta-E DHC DHE DHKA DHL DHPG DHX (+) Di(s)BT,4-OH DIAZEPAM diazoxide Dibenamine Dibenzepine Dibenzylamine, N-(2-chloroethyl)- Dibozane DIBT,4-OH Dibutyryl cGMP Dibutyryl-cGMP Dichloroisoproterenol,(+/-) Dichlorphenamide Diclofenac sodium salt Diclofensine DICLOFENSINE,(+) DICLOFENSINE,(-) Dicyclomine Dieldrin diethyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-glutamate diethyl (±)-((4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-glutamate diethyl (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-glutamate diethyl (±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-glutamate diethylpropion Diflunisal DIHETE 12(s), 5(s) dihomo-gamma-linolenic acid Dihydrexidine Dihydrexidine, 2-methyl Dihydrexidine, 4-methyl Dihydrexidine, 4-methyl-N-propyl Dihydrexidine, DHX Dihydrexidine, N-propyl Dihydro-14-hydroxymorphinone Dihydro-alpha-ergocryptine Dihydro-Beta-erythroidine Dihydroalprenolol,(+/-) dihydrobilobetin Dihydrocinnamoyl-pTyr-Leu-Pro-Gln-Thr-NH2 Dihydroergocornine Dihydroergocristine dihydroergocryptine DIHYDROERGOCRYPTINE Dihydroergotamine dihydroetorphine Dihydroheroin Dihydrokainate DIHYDROMORPHINE dihydroMotu (3,3) dihydroMotu (3,3)c dihydroMotu (4,4) Diisopropyl fluorophosphate diisopropyl-fluorophosphate DILTIAZEM Dimaprit Dimetane-DC Dimethindene dimethyl-phenyl-piperazinium dimethyl-[1-(pyridin-3-yloxymethyl)-cyclopropyl]-amine; hydrochloride dimethyl-{3-[(2-p-tolyl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-amine dimethylamino-norchloro-epibatidine Dimethylamylamine Dimethylhistaprodifen Dinapsoline, (+/-) Dinapsoline, (R)(+) Dinapsoline, (S)(-) Dinapsoline,(+/-)-4-Methyl Dinapsoline,(+/-)-4-Methyl-N-allyl Dinapsoline,(+/-)-4-Methyl-N-propyl Dinapsoline,(+/-)-6-Methyl Dinapsoline,(+/-)-N-allyl Dinapsoline,(+/-)-N-propyl Diphenhydramine Diphenidine Diphenyl-piperidin-4-yl-methanol Diphenyl-[1-(2-p-tolyl-ethyl)-piperidin-4-yl]-methanol Diphenyl-[1-(3-p-tolyl-propyl)-piperidin-4-yl]-methanol Diphenylpyraline Dipicolinate DiPOA Diprenorphine DIPRENORPHINE-HCl Diprophylline dipropyltryptamine DIPT,5-OH Dipyridamole Dithiocarbonic Acid S-benzyl Ester O-[2-benzylsulfanylthiocarboxyoxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl] Este... ditolylguanidine Divalinal Ang IV dizocilpine DKR-1677 dl-2-amino-4-(methylphosphino)butanoic acid dl-alpha-methylphenethylamine DL-AMPB DL-AP7 DL-homocysteic acid DL-homocysteine dl-Norepinephrine DL-TBOA DL-TBzOAsp DL-THA DM 1451 DM 236 DM 286 DM-139 DM-146 DM-173 DM-215 DM-239 DM-I-81 DM-II-20 DM-II-30 DM-II-30 (C20H13N3O2BrF3) DM-II-33 DM-II-72 DM-II-72 (C15H10N20BrCl) DM-II-90 DM-II-90 (C17H12N4BrCl) DM-III-01 DM-III-01 (C18H12N3O2Br) DMA DMA,2,4- DMA,2,5- DMAB DMAC DMCAE DMCC DMCM DMH-D-053 DMHP, 1', 2' DMP696 DMP904 DMPP DMT DMT,2-Me DMT,2-Me-5-methoxy DMT,4-MeO DMT,5-Me DMT,5-MeO DMT,5-MeO-7-M DMT,5-OH DMT,6-MeO DMT,7-Br DMT,7-MeO DMT,7-OH Dmt-d-Ala-Phe-Phe-NH2 Dmt-d-Arg-Phe-A2pr-NH2 Dmt-d-Arg-Phe-Orn-NH2 dmt1 DALDA DMT: 6-Fluoro-N,N-dimethyltryptamine DMXB Dnal,Cys,Tyr,DTrp,Lys,Val,Cys,Nal-nh2 DNQX DOAc DOB DOB,BENZYLOXY- DOB,OH- DOB,R(-) DOB,S(+) DOBU DOBz DOC DOCN docosanoic acid (R)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester DOET DOET,(-) DOF dofetilide DOHx DOI DOI,(+) DOI,(-) DOM DOM,iso DOM,R(-) Domoate domoic acid DOMPERIDONE DON Donepezil DOPAMINE Dopamine + GPP(NH)p Dopamine D2, High Dopamine D2, low Dopamine+ (GTP+) Dopamine+ (GTP-) Dopamine+GTP Dopamine, D2 high Dopamine, D2 low Dopargimine DOPR dorzolamide DOTB Dotheipin Dothiepin Doxazosin DOXEPIN Doxepine DP-5-CT dp-ADTN DPAT DPCPX DPDPE DPDPE-Cl DPDPE-OH DPH Dphe12-Bn DPhe6,12,Leu14-Bn DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14) DPhe6,Leu13,Psi(CH2NH),Cpa14-Bn(6-14) DPhe6-Bn(1-13)NH2 DPhe6-Bn(6-13)hexylamide DPhe6-Bn(6-13)hydrazide DPhe6-Bn(6-13)methylester DPhe6-Bn(6-13)NH2 DPhe6-Bn(6-13)NHN(ME)2 DPhe6-Bn(6-13)propylamide DPhe6-Bn[6-14) DPI-3290 DPI-5201 DPI-5336 DPI-5337 DPI-5402 DPI-5701 DPI-5702 DPI-673 DPPy DPSPX DPX DR4004 DROPERIDOL DSLET DSLET-OH DTG DTyr6,DAla11-Bn(6-13)butylamide DU125530 Duloxetine duloxetine-5,6-diol I duloxetine-5,6-diol II DuP 532 DUP 734 DXM DXO DynA-(2-13) DynA-(3-10) DynA-(3-11) DynA-(3-13) DynA-(3-6) DynA-(3-7) DynA-(3-8) DynA-(3-9) DynA-(4-11) DynA-(4-13) DynA-(5-11) DynA-(5-12) DynA-(5-13) Dynorphin A Dynorphin A (1-13) Dynorphin A (1-13) NH2 Dynorphin A (1-17) Dynorphin A(1-10)-NH2, [Pro3,Arg10] Dynorphin A(1-10)-NH2, [Pro3] Dynorphin A(1-10)-NH2,[Pro3] Dynorphin A(1-10)-NH2[Pro3,Arg10] Dynorphin A(1-10)-OH Dynorphin A(1-11)-NH2 Dynorphin A(1-11)-NH2, [Pro3,Arg10] Dynorphin A(1-11)-NH2, [Pro3,Arg8] Dynorphin A(1-11)-NH2, [Pro3] Dynorphin A(1-11)-NH2,[Pro3] Dynorphin A(1-11)-OH, [Pro3] Dynorphin A(1-11)-OH,[Pro3] Dynorphin A(1-13)-OH Dynorphin A(1-5)-NH2, [Pro3] Dynorphin A(1-5)-OH (Leu-Enk) Dynorphin A(1-6)-NH2, [Pro3] Dynorphin A(1-6)-OH Dynorphin A(1-7)-NH2, [Pro3,Nle6] Dynorphin A(1-7)-NH2, [Pro3] Dynorphin A(1-7)-NH2,[Pro3] Dynorphin A(1-7)-OH Dynorphin A(1-8)-NH2, [Pro3,Arg8] Dynorphin A(1-8)-NH2,[Pro3] Dynorphin A(1-8)-OH Dynorphin A(1-9)-NH2,[Pro3] Dynorphin A(1-9)-OH Dynorphin A, (1-9)-NH2[Pro3] Dynorphin B Dynorphin B (1-13) DYNORPHIN B-OH DYNORPHIN(1-11)-OH DYNORPHIN(1-13)-OH DYNORPHIN(1-17)-OH DYNORPHIN(1-8)-OH Dysiherbaine d^/-10-[(2-Methyl-lH-imidazol-l-yl)methyl]-5,6,8,9,10,llhexahydro-4i7-pyrido[3,2,l-/A]carbazol-ll-one E 2020 E 3174 E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinoli... E-4031 EAA-090 EAB-318 EB ebastine EC5-21 Econopred EDC-I-071 EDC-I-093 EDC-II-044 efaroxane Efavirenz EGLU EHNA EHNA, (+) EKB-569 EKC EKC(-) Elacridar eledoisin Eliprodil Eltoprazine EM-A enolether EM-B enolether EM523 EMDT EN 1530 base Enadoline endo-8-(1H-Indol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo-[3.2.1]octan-3-ol endo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene endo-8-Dimethylaminomethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene endo-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-3-ethyl-2-ox Endometrin Endomorphin 1 Endomorphin 2 Enkephalin, Ala(2)-MePhe(4)-Gly(5)- Enprofylline ENPROSTIL ent-UB-165 EP011 EP045 EPA Ephedrine,(+) Ephedrine,(+/-) Ephedrine,(-) Ephendine Ephenidine Epibatidine Epibatidine, (+/-) Epibatidine, (+/-) Epibatidine-(+) Epibatidine-(-) Epibatidine-I,(+/-) EPIDEPRIDE epigallocatechin Epigallocatechin 3-gallate epinastine EPINEPHRINE Epinephrine, (R) EPINEPHRINE,(+) EPINEPHRINE,(-) EPINEPHRINE-l Epinine Eplivanserin Ergine Ergocornin Ergocornine Ergocristine Ergocryptine, beta Ergocrystine ERGOMETRINE ERGONOVINE Ergotaman-3',6',18-trione, 12'-hydroxy-2',5'-bis(1-methylethyl)-, (5'alpha)- Ergotaman-3',6',18-trione, 12'-hydroxy-2'-(1-methylethyl)-5'-(phenylmethyl)-, (5'alpha)- Ergotaman-3',6',18-trione, 12'-hydroxy-2'-methyl-5'-(phenylmethyl)-, (5'alpha)- ERGOTAMINE erythro-Phenyl-2-piperidyl-carbinol,(-) erythromycin Erythromycin A 6,9-enolether erythromycin-A Erythromycin-A enol ether Erythromycin-B Erythromycin-B enol ether Escitalopram Eserine Estradiol eszopiclone Eszopiclone ET-18-OCH3 Etamiphylline Etazocine ETE-12-Oxo ETE-5-Oxo Ethanamine, 2-phenyl- ethopropazine Ethosuximide ethoxzolamide ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyl... ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate and et... ethyl (1S)-2-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexan... ethyl (1S)-2-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyl... Ethyl (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9yl)-2,3-dihydroxybicyclo[3.1.0]hexane-... Ethyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbox... Ethyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-(dimethylamino)-9H-purin9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate Ethyl (1S,2R,3S,4R,5S)-4-(5-((5-Chlorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-2,3-dihydroxybicy... ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-... ethyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1... ethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicycl... ethyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-methioninate ethyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-valinate ethyl (±)-((4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-methioninate ethyl (±)-((4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-valinate ethyl (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-methioninate ethyl (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-valinate ethyl (±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-methioninate ethyl (±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-valinate ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate Ethyl 2-(2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate Ethyl 2-(2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate Ethyl 2-(4-(dimethylamino)-2-((methoxycarbonyl)amino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylat... Ethyl 2-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate Ethyl 2-(4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate Ethyl 2-(4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate Ethyl 2-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate Ethyl 2-(5-((2-ethoxy-2-oxoethyl)amino)-2-(furan-2-yl)-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxamido)acetate ethyl 2-(6-bromo-2-(4-fluorophenyl)-4-phenyl-1,2-dihydroquinazolin-3(4H)-yl)acetate Ethyl 2-(furan-2-yl)-5-(2-phenylhydrazinyl)-[1,2,4]triazolo[1,5-c] pyrimidine-8-carboxylate Ethyl 2-(furan-2-yl)-5-(piperazin-1-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride Ethyl 2-(furan-2-yl)-5-hydrazinyl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate ethyl 2-[2-(4-chlorophenyl)-5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate ethyl 2-[5-methyl-2-(4-methylphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate ethyl 4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2,6-diethoxybenzoate ethyl 4-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate ethyl 4-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)benzoate ethyl 4-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate ethyl 4-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate ethyl 4-(3-(2-chlorophenyl)-1-(2,4-dimethylphenyl)-1H-pyrazole-5-carbonyl)piperazine-1-carboxylate Ethyl 5-(2-(tert-butoxycarbonyl)hydrazinyl)-2-(furan-2-yl)-[1,2,4triazolo[1,5-c]pyrimidine-8-carboxylate Ethyl 5-(3-(4-((benzo[d][1,3]dioxol-5-yl)methyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate Ethyl 5-(3-(4-(2-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate Ethyl 5-(3-(4-(2-cyanophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate ethyl 5-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate Ethyl 5-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate Ethyl 5-(3-(4-(3-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate Ethyl 5-(3-(4-(4-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate Ethyl 5-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate Ethyl 5-(3-(4-o-tolylpiperazin-1-yl)propoxy)-1H-indole-2-carboxylate Ethyl 5-(4-(tert-butoxycarbonyl)piperazin-1-yl)-2-(furan-2-yl)- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate Ethyl 5-(4-chlorobenzoyl)-4-phenylthiazol-2-ylcarbamate Ethyl 5-(4-methoxybenzoyl)-4-phenylthiazol-2-ylcarbamate Ethyl 5-benzoyl-4-phenylthiazol-2-ylcarbamate Ethyl 5-ethoxy-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylate ethyl 5-methoxy-2-[(propan-2-ylamino)methyl]-1-benzofuran-3-carboxylate ethyl 5-methoxy-2-{[(propan-2-yl)amino]methyl}-1-benzofuran-3-carboxylate ethyl 5-[(3,4-dimethoxyphenyl)methylamino]-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate ethyl 6'-amino-1-benzyl-5',5',7'-tricyano-2-oxo-5',8a'-dihydro-1'H-spiro[indoline-3,8'-isoquinoline]-2'(3'H)-carboxylate Ethyl 7-Oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate Ethyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-acetic acid hydrochloride Ethyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-butyric acid Ethyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate Ethyl {4-[(3-{[({(2E)-3-[6-(Acetylamino)-3-pyridinyl]-2-propenoyl}amino)acetyl](methyl)amino}-2,6-dichlorobenzyl) Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carbox... Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hex... Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]h... Ethyl(1S,2R,3S,4R,5S)-4-(2-((5-bromothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxyb... Ethyl(1S,2R,3S,4R,5S)-4-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,3-dihydroxy... Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyc... Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]... Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocy... Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-((5-chlorothiophen-2-yl)- ethynyl)-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- 2,2-dimet... Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]c... ethyl-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoyl}amino)... Ethyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate Ethyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate Ethyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate Ethyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate Ethyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate Ethyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate Ethyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate Ethyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate Ethyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate Ethyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate Ethyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate Ethyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate Ethyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate Ethyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate Ethyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate Ethyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate ethyladenosin-5'-uronamide Ethylone ETICLOPRIDE ETICLOPRIDE,S(-) Etodolac Etofylline ETONITAZENE Etoperidone ETORICOXIB Etorphine ETORPHINE - HCI Etoxadrol Eucatropine EW5182 exo-8-Benzyloxymethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene exo-8-Dimethylaminomethyl-3-ethoxycarbonyl-4-hydroxy-1-azabicyclo[3.3.1]non-3-ene EXP3174 EXP655 F106A F17464 F332A F33A famotidine Fananserin FAUC 3019 FE200041 FECIMBI-36 Femoxetine FEMPT Fenbendazole FENDOLOPAM Fenfluramine Fenfluramine (+) Fenfluramine (+/-) Fenfluramine (-) Fenobam FENOLDOPAM Fenoprofen Fenoterol Fentanyl FENTANYL-HCl Fernisolone-P Fernisone Fexofenadine FG 5803 FG 5893 FG 7142 FG 8205 FG8205 Fiduxosin Finazine FK 1052 FK 224 FK 888 FK-453 FK480 FK881 Flavopiridol Flephedrone FLESINOXAN FLUANISONE Flubiprofen Flufenamate Flufylline flumazenil Flunitrazepam fluoro-norchloro-epibatidine Fluorocarazolol,(R) Fluorocarazolol,(S) Fluorolintane (2-F-DPPy) Fluorowillardiine FLUOXETINE Fluoxetine-R-(-) Fluoxetine-S-(+) Fluparoxan Flupenthixol FLUPENTHIXOL, Alpha Flupenthixol, Beta FLUPENTHIXOL, CIS Flupenthixol, trans Flupenthixol, Trans-(E) FLUPENTHIXOL,a- FLUPERLAPINE FLUPHENAZINE Fluphenthixol Fluprofylline FLUPROSTENOL FLUSPIPERONE FLUSPIRILENE Fluticasone Fluvastatin Fluvoxamine FMRFamide FMS586 formic acid (R)-2-fluoro-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester Formoterol Fostedil FR72112 FSLLRN-NH2 Fuberidazole Furan-2-carboxylic acid (4-phenyl-5-pyridin-2-yl-thiazol-2-yl)-amide Furan-2-carboxylic acid (4-phenyl-5-pyridin-4-yl-thiazol-2-yl)-amide Furan-2-carboxylic acid [4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-amide Furan-2-carboxylic acid [5-(4-amino-5,6,7,8-tetrahydro-benzo[4,5]thieno[2,3-d]pyrim-idin-2-yl)-4-phenyl-thiazol-2-yl]-amide Furan-2-carboxylic acid [5-(4-amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide Furan-2-carboxylic acid [5-(4-oxo-3,4-dihydro-quinazolin-2-yl)-4-phenyl-thiazol-2-yl]-amide Furan-2-carboxylic acid [5-(5,6-dimethyl-4-oxo-3,4-dihydro-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide Furan-2-carboxylic-acid [4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-amide G107A G36A GABA GABA, 2-methylthienyl GABA, m-chlorophenyl Gal(1-13)-BK (2-29) Gal(1-13)-Std I Gal-(1-15)-ol,[d-Thr6,d-Trp8,9] Galanin (-7 +29), porcine Galanin (-7 to+29), porcine Galanin (1-13)-bradikinin(2-9) Galanin (1-13)-bradykinin (2-29) Galanin (1-13)-SP-(5-11) Galanin (1-13)-spantide Galanin (1-15) Galanin (1-15)-ol,[Ala6,D-trp8] Galanin (1-16) Galanin (1-16), porcine Galanin (1-16), rat Galanin (1-19), rat Galanin (1-29), porcine Galanin (1-29), rat Galanin (1-29),[D-Trp2] Galanin (10-29), rat Galanin (2-29), rat Galanin (3-29), porcine Galanin (3-29), rat Galanin Porcine 2-29 Galanin rat Galanin [-7 to +29], porcine Galanin [D-Trp2], porcine Galanin, Human Galanin, Porcine Galantide Galantide (M15) Gallamine Gallamine Gallopamil Galnon Gamma-Aminobutanoic acid Gamma-Aminobutyric acid GAMMA-MANGOSTIN gamma-methyl-APB Gamma1-MSH Gamma2-MSH Gamma3-MSH GAMS Gastrin Gastrin I Gastrin Releasing Peptide Gastrin-17 Gastrin-I-(1-17) Gastrin-I-(4-17) Gastrin-I-(5-17) GBR-12909 GBR-12935 GBR-13,069 Gbu6,Ava14,15 GDP GDP[S] GEPIRONE GHB Gitoxigenin Glaucine HBr Glaucium fl. extract Glaxo 1192U90 Gleevec glibenclamide Glivec Glutamate glutamate-AMPA GLYCINE GM 611 GMAP (1-41) GMAP (44-59) GMC 1-116 GMC1-169 GMC2-83 GMC3-06 GMC61-39 GMP GNF-Pf-1694 GNTI GP 515 GPA 2163 GPP(NH)P(+) GPP(NH)p(-) Gpr6,Ava14,15 GR 103691 GR 113808 GR 125487 GR 127935 GR 128107 GR 135533 GR 168320 GR 196429 GR 231118 GR 32191 GR 38032 GR 38032F GR 63799 GR 63799X GR 65630 GR-103545 GR-89696 GR-NH2 GR125,743 GR218231 GR231118 GR46,611 GR85,548 GR89696 GRANISETRON grepafloxacin GRP GRP-10,frog GS39783 GT 2016 GT 2130 GT 2136 GT 2140 GT 2142 GT 2146 GT 2148 GT 2174 GT 2227 GT 2228 GT 2231 GT 2260 GT 2286 GT 2287 GT 2288 GT 2293 GT 2321 GT 2327 GT 2331 GTI GTP GTP[S] GTS-21 Guanabenz Guanfacine Guanidine, N-cyano-N'-(1,1-dimethylpropyl)-N''-3-pyridinyl Guanidinoproprionic-beta Guanosine Guanosine 5'-[gamma-thio]triphosphate tetralithium salt Guanylyl imidodiphosphate GuoPP[NH]P Gva6,Ala12,Ava14,15 Gva6,Ala8,Ava14,15 Gva6,alphaAbu8,Ava14,15 Gva6,Ava14,15 Gva6,Ava14,15, OH Gva6,Ava9,10 Gva6,Ava9,10,Ava14,15 Gva6,betaAla14,15 Gva6,cisAcx14,15 Gva6,D-Cys7,Ava14,15 Gva6,desLeu9,Ava14,15 Gva6,gammaAbu14,15 Gva6,Gly14,15 Gva6,Nle8,Ava14,15 GW-2016 GW501516 GW5823 GYKI-52466 h alpha-CGRP h alpha-CGRP8-37 H-2Fpa-cyclo[DCys-His-DTrp-Lys-Val-Cys]-2Fpa-NH2 H-2Fpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-2Fpa-NH2 H-3Fpa-cyclo[DCys-His-DTrp-Lys-Val-Cys]-3Fpa-NH2 H-3Fpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-3Fpa-NH2 H-Ala-Ala-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Ala-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Ala-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Ala-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Ala-Trp-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Ala-Lys-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Ala-Thr-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Ala-Phe-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Ala-Thr-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ala-Ser-Cys}-NH2 H-Ala-Gly-{Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ala-Cys}-NH2 h-alpha-CGRP h-alpha-CGRP (reduced) h-alpha-CGRP 8-37 H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Leu-OH H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH H-Asp-C[Cys-Phe-DTrp-Lys-Tyr-Cys]Val-OH H-Asp-C[Cys-Phe-DTrp-Orn-Tyr-Cys]Val-OH H-Asp-C[Cys-Phe-Trp-Orn-Tyr-Cys]Val-OH H-Asp-C[DPen-Phe-DTrp-Orn-Tyr-Cys]Val-OH H-Asp-C[Pen-Phe-DTrp-DOrn-Tyr-Cys]Val-OH H-Asp-C[Pen-Phe-DTrp-Lys-Tyr-Cys]Val-OH H-Asp-C[Pen-Phe-DTrp-Orn-Tyr-Cys]Val-OH H-Asp-C[Pen-Phe-Trp-Orn-Tyr-Cys]Val-OH H-Bip-cyclo[DCys-Tyr-DTrp-Lys-Ile-Cys]-Bip-NH2 H-Bpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Bpa-NH2 H-Cpa-cyclo[DCys-2Pal-DTrp-Lys-Thr-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-D2Pal-DTrp-Lys-Thr-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-Pal-DTrp-Lys-Tba-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-Pal-DTrp-Lys-Thr-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-Cpa-NH2 H-Cpa-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Cpa-NH2 H-Cpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-Phe-DTrp-Lys-Thr-Cys]-Nal-NH2 H-Cpa-cyclo[DCys-Tyr-DTrp-Lys-Thr-Cys]-Nal-NH2 H-D-Phe-c[-N-epsilon-Lys-Tyr(3-tBu)-beta-Ala-] H-DCpa-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-DCpa-NH2 H-DFpa-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-Nal-NH2 H-DFpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-DFpa-NH2 H-Dmt-D-Arg-Phe-A2bu-NH2 H-Dmt-D-Arg-Phe-Orn-NH2 H-Dmt-Tic-NH2 H-Dmt-Tic-OH H-Fpa-cyclo[DCys-His-DTrp-Lys-Val-Cys]-Fpa-NH2 H-Fpa-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-Nal-NH2 H-Fpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Fpa-NH2 H-Fpa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Nal-NH2 H-Hmt-D-Arg-Phe-Lys-NH2 I H-Hmt-D-Arg-Phe-Lys-NH2 II H-Igl-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Igl-NH2 H-Iph-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Iph-NH2 H-Mmt-D-Arg-Phe-Lys-NH2 H-Nal-cyclo[DCys-3ITyr-DTrp-Lys-Val-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Bta-DTrp-Lys-Val-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Ala-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Gly-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Ile-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Leu-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Nle-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-DDip-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Fpa-NH2 H-Nal-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Nal-NH2 H-Nal-cyclo[DCys-Tyr-DTrp-Lys-Val-Cys]-DDip-NH2 H-P5U-Asp-C[Pen-Phe-Trp-Lys-Tyr-Cys]Val-OH H-Pfp-cyclo[DCys-2Pal-DTrp-Lys-Val-Cys]-Pfp-NH2 H-Pfp-cyclo[DCys-D2Pal-DTrp-Lys-Val-Cys]-Pfp-NH2 H-Pfp-cyclo[DCys-His-DTrp-Lys-Val-Cys]-Pfp-NH2 H-Pfp-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Pfp-NH2 H-Phe-Ala-Arg-Ala-Arg-Pro-Arg-OH H-Phe-c[-N-epsilon-D-Lys-Tyr(3-tBu)-beta-Ala-] H-Phe-c[-N-epsilon-Lys-D-Tyr(3-tBu)-beta-Ala-] H-Phe-c[-N-epsilon-Lys-Tyr(3,5-di-tBu)-beta-Ala-] H-Phe-c[-N-epsilon-Lys-Tyr(3-tBu)-4-aminobutyric acid-] H-Phe-c[-N-epsilon-Lys-Tyr(3-tBu)-6-Aminohexanoic acid-] H-Phe-c[-N-epsilon-Lys-Tyr(3-tBu)-beta-Ala-] H-Phe-c[-N-epsilon-Lys-Tyr(3-tBu)-Gly-] H-Phe-c[-N-epsilon-Lys-Tyr(O-secBu)-beta-Ala-] H-Phe-c[-N-epsilon-Lys-Tyr(O-tBu)-beta-Ala-] H-Phe-c[-N-epsilon-Lys-Tyr-beta-Ala-] H-Phe-Leu-Arg-Arg-Ile-Arg-Arg-Pro-Lys-OH H-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-NH2 H-Phe-Leu-Arg-Ile-Arg-Pro-Arg-OH H-Phe-Leu-Arg-Ile-Erg-Pro-Lys-OH H-Phe-Nle-Arg-Nle-Arg-Pro-Arg-OH H-Tic-cyclo[DCys-Tyr-DTrp-Lys-Val-Cys]-Tic-NH2 H-Trp-cyclo[DCys-Pal-DTrp-Lys-Tle-Cys]-Nal-NH2 H-Tyr-D-Ala-Gly-Phe-NH-NH-(NMe)Phe-Asp-Lys(Cpac)-Trp-Ac H-Tyr-Pro-Phe-Phe-NH2 H-U-II(4-11)-Asp-C[Cys-Phe-Trp-Lys-Tyr-Cys]Val-OH H-Ypa-cyclo[DCys-Pal-DTrp-Lys-Val-Cys]-Ypa-NH2 H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 H2N-4-NO2-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2 H2N-4-NO2-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-Nh2 H7 H89 HA-1077 hAc-MCH(6-16)-NH2 Haldol HALOPERIDOL HARMINE haTRAP hCS 13 hCS 15 hCS 17 HE-NECA Helodermin Hemicholinium-3 HENECA HETE-(+/-)5 HETE-15(S) HETE-20 HETE-5(S) HETE-8(R ) heterocodeine Hexahydro-sila-dilfenidol Hexahydrodifenidol hexahydrosiladifenidol HEXAMETHONIUM Hexocyclium HHC, 9 beta-OH HHC. 9 alpha-OH HHD hhs HHSiD HIBO HIMBACINE HIS HISTAMINE histaprodifen Histidine HJ-I-037 HMA hMCH Homatropine homo-AMPA homohistamine Homoibotenic acid Homoibotenic acid, (R) Hoodia Extract HP 873 hPTH(1-34) hrCRF HS,(+/-) HS378 HS414 HS464 HS510A HS531 HS595 hsd HTQZ HU-210 Human U-II huprine X HX Hydeltra-Tba Hydralazine Hydrocodone Hydromorphine hydromorphone hydroxy-norchloro-epibatidine Hydroxyamphetamine,(+/-) Hydroxybenzylpindolol,(+/-) Hydroxybupropion Hydroxynefazodone Hydroxytyramin Hydroxyzine Hydroxyzine, (R) Hyperforin Hypericin hypericin Hyperoside Hypoxanthine Hz148 I I-ABA I-ABOPX I-APE I-BOP I-Naphyrone I-PTA-OH I-RTX I-TBZ I31,G34-PP,human I4AA IAB-MECA IAPP26-34, CGRP30-37 IB-MECA ibipinabant IBMX IBOGAINE Ibotenate Ibotenic acid ibuprofen ibuprofen solid, (S)-(+) ICI 106270 ICI 118,115 ICI 118,551 ICI 169,369 ICI 198615 ICI 63, 197 ICI 79939 ICI 86,406 ICI 89,406 ICI-174864 ICS 205-930 ICS 205-930, Q ICS 205930 ICYANOPINDOLOL IDAZOXAN IDORENATE Ifenprodil Ifenprodil,(+/-) II III III-BTD ILOPERIDONE ILOPROST IMAFEN,(+) IMAFEN,(-) imbutamine Imetit Imidazenil Imidazole Imidazole-4-acetic acid IMILOXAN IMIPRAMINE Immepip immethridine Impentamine Impromidine Indacaterol INDALPINE Indatraline Indinavir sulphate Indiplon Indirubin-3monoxime indisulam INDOL-5-OL, 3-[2-(DIMETHYLAMINO)ETHYL] INDOLE, 3-[2-(DIMETHYLAMINO)ETHYL]-2-METHYL INDOLE, 5-METHOXY-3-[2-(DIMETHYLAMINO)ETHYL] Indomethacin Indoramin INDORAMINE INDORENATE Inosine iodo-βCCE iodo-βCCt Iodoclonidine-p Iodophenpropit Iodoproxyfan Iodosulpride iperoxo IPH IPP Ipratropium IPRINDOLE Iproniazid IPSAPIRONE Ipsapirone IPT Iressa irindalone Irinotecan Irinotecan ISAM-134 ISAM-140 ISAM-141 ISAM-142 ISAMOLTANE Iso-nicotine (+/-) ISOCARBACYCLIN ISOCLOZAPINE Isoflurane isoginkgetin Isoguvacine Isoloxapine Isomenthol-(+) Isonicotinic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazo... ISOPRENALINE Isopropamide Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate Isopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate Isoproterenol Isoproterenol (-) Isoproterenol,(+) Isoproterenol-l ISOPROTERONOL Isoquercitrin Isoquinoline-1,3,4-trione Istradefylline ISVY071 ISVY074 ISVY127 ISVY130 ISVY133 ISVY169 IT-290, (+) IT-290, (-) IV IX βCCE βCCt J-104132 J-113397 Janty EC Liquid JBR-313 JBR-321 JBR-73 JC184 JC184 C13H9BrN2OS JC208 JC208 C15H10N2OS JC221 ANX1 JC222 JCF109 JDTic JF-1 JNJ 7777120 JNJ-5207852 JTE-522 JTE-907 JVW-1034 JWH-015 JWH-030 JWH-031 JWH-032 JWH-036 JWH-044 JWH-045 JWH-051 JWH-073 JWH-133 JWH-391 JYI-01 JYI-01 (c19H20N3O3Br) JYI-03 JYI-03 (C21H21N3O3) JYI-04 JYI-04 (C12H23N3O3) JYI-06 JYI-06 (C23H23N3O4) JYI-10 JYI-11 JYI-11 (C22H22N3O3F3Si) JYI-12 JYI-12 (C19H16N3O3F3) JYI-13 JYI-13 (C21H16N3O4F3) JYI-14 JYI-15 JYI-19 JYI-19 (C23H23N3O3S) JYI-32 JYI-32 (C2OH15N3O2BrF) JYI-42 JYI-47 JYI-48 JYI-49 JYI-49 (C20H12N3O2F4Br) JYI-54 JYI-54 (C24H15N3O3F4) JYI-55 JYI-57 JYI-59 JYI-59 (C22H13N3O2F4) JYI-60 JYI-60 (C17H11N2OF JYI-60 (C17H11N2OF) JYI-64 JYI-64 (C17H12N4FBr) JYI-70 JYI-70 (C19H13N4F) JYI-72 JYI-72 (C22H21N4SiF) JYL1421 K117 K368,374C K376 K604 KA Kadsurenone Kainate kassinin KE108 KE119 kenpaullone Ketamine KETANSERIN Ketoconazole Ketoprofen Ketorolac tris salt KETOTIFEN KJM429 KN-62 Kodiak extract KRH-594 KUR-1246 KYMVm-NH2 Kynurenate L 745,870 L(+)-2-amino-3-phosphonopropionic acid L(+)-2-amino-4-phosphonobutyric acid l-(2,3-Dihydropyrrolo[l,2,3-de][l,4]benzothiazin-6-yl)-3-(5-methylimidazol-4-yl)propan-l-one Hydrochloride l-(2,5-Dimethoxy-4-hexylphenyl)-2-aminopropane Hydrochloride L-054,522 l-1-(3, 4-Dihydroxyphenyl)-2-methylaminoethanol L-152,804 L-158,809 L-159,530 L-159,689 L-159,882 L-159,913 L-161,274 L-161,276 L-161,713 L-161,865 L-161,948 L-162,193 L-2-amino-3-phosphonopropionate L-2-amino-4-phosphonobutyrate L-361,301 L-362,823 L-362,855 L-362,862 L-363,301 L-363,301 HyPro L-363,301 Pro L-363,376 L-363,377 L-363,572 L-364,718 L-365,209 L-365,260 L-366,670 L-366,682 L-366,706 L-366,811 L-366,875 L-366,948 L-630,571 L-639,019 L-644,763 L-652731 L-654,284 L-657,743 L-657925 L-657926 L-659,989 L-659,989, (+) L-659,989, (-) L-662,418 L-701,324 L-737,415 L-740,093 L-741,626 L-745,870 L-745870 L-745870 L-779,976 L-796,778 L-797,591 L-803,087 L-817,818 L-826,141 L-amino-4-phosphonobutyrate L-AP3 L-AP4 L-APB L-Aspartate l-Brompherinamine L-Carnitine L-CCG-I L-CCG-IV L-CCGI l-Chlorpheniramine L-cysteic acid L-cysteine L-cysteine sulfinic acid L-cystine L-DOPA l-Fenfluramine L-GDEE L-Glu L-Glutamate L-glutamate tetrazole L-glutamic acid L-homocysteic acid L-homocysteine sulfinic acid L-homocysteine thiolactone L-Isoleucyl-L-prolinamide trifluoroacetate L-Leucyl-L-prolinamide trifluoroacetate L-methionine l-Metoprolol l-Nantradol l-Norepinrpherine l-norfenfluramine L-Norleucyl-L-prolinamide hydrogen oxalate hemihydrate L-Norvalyl-L-prolinamide trifluoroacetate hemihydrate L-pGlu-(2-cyclohexyl)-L-His-L-Pro-NH2 L-pGlu-(2-cyclopropyl)-L-His-L-Pro-NH2 L-pGlu-(2-isopropyl)-L-His-L-Pro-NH2 L-pGlu-(2-propyl)-L-His-L-Pro-NH2 L-pGlu-(2-tert-butyl)-L-His-L-Pro-NH2 L-pGlu-[2-(adamantan-1-yl)]-L-His-L-Pro-NH2 L-Phenylalanyl-L-prolinamide trifluoroacetate L-PIA L-SOP l-TA-3090 L-Trimipramine L-Valyl-L-prolinamide trifluoroacetate L-Valyl-L-proline benzylamide hydrogen oxalate L-Valyl-L-proline cyclohexylmethylamide hydrogen oxalate L-Valyl-L-Proline hexylamide hydrogen oxalate L-Valyl-L-proline piperidinylamide hydrogen oxalate hemihydrate L-Valyl-L-proline-N- β-naphthylamide trifluroacetate l-[2,5-Dimethoxy-4-(3-phenylpropyl)phenyl]-2-aminopropane Hydrochloride L109A L110A L31,P34-NPY,human L35A L694,247 L741,626 L745,337 L775,606 LA-Iii LAAM LABETALOL Lanreotide LATANOPROST (Free Acid) Latanoprost (Isopropyl Ester) LATANOPROST (PHXA41) LE300 LE301 LE302 LE304 LE400 Lecozotan Lensiprazine LERGOTRILE LESOPITRON Leu-ENKEPHALIN Leu13,Psi(CH2NH),Leu14-BN Leu5-Enkephalin Leu8, D-Trp22, Tyr25 SST-28 Leu8-phyllolitorin LEUCOHARMINE Levallorphan Levcromakalim Levetimide Levlofexidine LEVO-BC-2627 Levocabastine Levocetirizine Levomepromazine Levomethorpan Levonantradol Levorphanol LEVORPHANOL-tartarate Levoxadrol Liarozole Lidoflazine lipoxin-A4 LISURIDE lisuride, (S) lisuride, R Lithocholylcholine Lithocholylglycine Lithocholyltaurine Litorin LJD-III-15E lobelane Lobelane Lobeline Lobeline, (-) Lobeline,Alpha Lofepramine Loperamide loratidine Losartan LOXAPINE Loxiglumide LP-211 LSD LSD, IODO LSD,(+) LSD,(-) LSD,2-Bromo LSD,2-iodo LSD,l- LSD-25 LTA3-ME LTA4-ME LTA5-ME LTB4 LTB4-14,15-dehydro LTB4-20-carboxy LTB4-20-hydroxy LTB4-3-aminopropylamide LTB4-6-trans LTB5 LTC3 LTC4 LTC5 LTD3 LTD4 LTD5 LTE3 LTE4 LTF4 LTT-SRIF28 LTT-SST-28 LU 19,005 Lu 2-098 Lumateperone Lunesta LUPITIDINE Lurasidone Lurasidone HCl Luzindole Luzindole,5-Methoxy Luzindole,N-butanoyl Luzindole,N-hexanoyl Luzindole,N-pentanoyl Luzindole,N-propanoyl LY 063518 LY 108742 LY 110140 LY 134046 LY 139603 LY 17883 LY 193525 LY 197541 LY 211000 LY 215840 LY 225297 LY 254239 LY 258458 LY 266097 LY 278584 LY 278989 LY 293111 LY 293284 LY 293558 LY 294486 LY 302679 LY 314228 LY 320950 LY 320951 LY 320954 LY 334359 LY 334362 LY 335102 LY 344864 LY 382884 LY 457691 LY 458545 LY 466195 LY 467711 Ly 5182 LY 525327 LY 53857 LY 86057 LY 97241 LY-171555 LY-255582 LY-333531 LY-334370 LY-364947 LY135252 LY139602 LY170053 LY23728 LY248685 LY248686 LY307452 LY341495 LY354740 LY366563 LY367385 LY379268 LYS170 LYS201 LYS227 LYS231 LYS322 LYS328 LYS401 LYS402 LYS403 Lysergamide LYSERGIC ACID LYSERGOL lysergsaure diethylamid Lysophosphatidic Acid M&B-28767 M- (3-Iodoben zy1)adenosine- N-methyluronamide M-154 m-chloro-phenyl-biguanide m-chlorophenylpiperazine M-MPEP M100907 M32 M35 M40 M6G M99 MA-3-PROPOXYL MADAM MAP4 MAPPINE MAPROTILINE mazapertine MAZINDOL MB-3 MBDB MC-CAM MC-CAM MCC MCCG MCCG-I MCH MCH6-17 MCL-101 MCL-133 MCL-134 MCL-135 MCL-136 MCL-139 MCL-140 MCL-141 MCL-142 MCL-143 MCL-144 MCL-145 MCL-145 MCL-153 MCL-154 MCL-176 MCL-177 MCL-178 MCL-179 MCL-201 MCL-202 MCL-203 MCL-204 MCL-205 MCL-206 MCL-207 MCL-209 MCL-210 MCL-211 MCL-212 MCL-213 MCL-214 MCL-215 MCL-216 MCL-217 MCL-218 MCL-230A MCL0129 McN-5652-15 McN-5652-W-68 McN-5652-X-68 McN-5652-Z-14 McN-5652-Z-68 McN-A-343 MCPG MCPG(RS) mCPP MDA MDA, (R,S) MDA,R(-) MDA,S(+) MDEA MDL 100907 MDL 103,392A racemate MDL 104,335 (S)-enantiomer MDL 105,212 (R)-enantiomer MDL 105,212A (R)-enantiomer MDL 11,939 MDL 72222 MDL 72832 MDL 72832, (+) MDL 72832, (-) MDL 73005 EF MDMA MDMA, R(-) MDMA,S(+) MDPV ME36 ME4 ME523 Mebendazole MECA Mecamylamine Meclizine Meclofenamate medroxyprogesterone acetate Mefenamic acid MEGY MELATONIN melatonin, 6-Chloro melatonin, 6-Hydroxy melatonin, 6-Methoxy Melatonin,2-Bromo Melatonin,2-Chloro Melatonin,2-Iodo Melatonin,2-Phenyl Melatonin,6,7 di-cl-2-Me Melatonin,6-Cl Melatonin,6-Cl-2-Me Melatonin,6-Hydroxy Melatonin,6-Methoxy Melatonin,6-OH Mellpaladine A Mellpaladine B Meloxicam sodium MELPERONE Melperone HCl MEM Memantine Menthol-(+) Menthol-(-) Meperidine mephedrone Mephentermine MEPYRAMINE Mequitazine meridianin A MESCALINE Mescaline-NBOMe MESORIDAZINE mesotransdiene MESULERGINE Met-enkephalin Met5-Enkephalin Met5-enkephalin-Arg-Phe Metazocine METERGOLINE Methacholine Methadone Methadone,(R)(-) Methadone,(S)(+) Methadone-HCL,(-) Methamphetamine METHAMPHETAMINE (+) METHAMPHETAMINE (-) Methanandamide Methanesulfonic Acid 3-[(2-Methyl-4-thiazolyl)ethynyl]-2-pyridyl Ester Methanesulfonic Acid 5-[(2-Methyl-4-thiazolyl)ethynyl]-2-pyridyl Ester Methapyrilene methazolamide Methcathinone Methcathinone, (-) Methdilazine METHERGINE methimmepip Methiopropamine METHIOTHEPIN methiothepine METHOCTRAMINE Methotrimeprazine METHOXAMINE METHOXETAMINE Methoxyacetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxaz... methoxymethyl-MTEP Methoxynaltrexone,3 Methsergide Methyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbo... methyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-bromothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1... Methyl (2S,4aR,6aR,7R,9R,10aS,10bR)-2-(3-furyl)-6a,10b-dimethyl-4,10-dioxo-9-sulfanyldodecahydro-2H-benzo[f]isochromene-7-car... Methyl (2S,4aR,6aR,7R,9R,10aS,10bR)-9-(acetylsulfanyl)-2-(3-furyl)-6a,10b-dimethyl-4,10-dioxododecahydro-2H-benzo[f]isochrome... Methyl (2S,4aR,6aR,7R,9S,10aS,10bR)-2-(3-furyl)-6a,10b-dimethyl-4,10-dioxo-9-sulfanyldodecahydro-2H-benzo[f]isochromene-7-car... Methyl (2S,4aR,6aR,7R,9S,10aS,10bR)-9-(acetylsulfanyl)-2-(3-furyl)-6a,10b-dimethyl-4,10-dioxododecahydro-2H-benzo[f]isochrome... methyl (6Z)-6-(2,2'-bithiophen-5-ylmethylidene)octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(2'-fluorobiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(2'-methoxybiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(3',4'-difluorobiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(3',5'-difluorobiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(3'-fluorobiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(3'-methoxybiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-[(4'-fluorobiphenyl-4-yl)methylidene]octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-{[3'-(trifluoromethyl)biphenyl-4-yl]methylidene}octahydro-3,7-methanoindolizine-8-carboxylate methyl (6Z)-6-{[4'-(methylsulfanyl)biphenyl-4-yl]methylidene}octahydro-3,7-methanoindolizine-8-carboxylate Methyl (9Z)-9-({5-[4-(methylsulfanyl)phenyl]-2-thienyl}methylene)-7-azatricyclo[4.3.1.03,7]decane-2-carboxylate methyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-alaninate methyl (±)-((4aS,8R,8aS)-2-(4-chlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-alaninate methyl (±)-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-alaninate methyl (±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-alaninate methyl (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate methyl (±)-(S)-2-((4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)-2-phen... methyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate methyl 2-(8-(bis(2-chlorophenyl)methyl)-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl)acetate Methyl 3-(1, 2, 3, 4-tetrahydro-1, 3, 4-trioxoisoquinolin-6-ylcarbamoyl)-5-nitro-benzoate Methyl 3-(1-methyl-2-pyrrolidinyl)pyridine-6-carboxylate hydrochloride methyl 3-amino-6-methoxy-1H-indole-2-carboxylate Methyl 3-[({[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]amino}carbonyl)amino]benzoate methyl 4-(4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butyl)benzoate methyl 4-(4-(9H-fluoren-9-yl)piperazin-1-ylsulfonyl)-2,5-dimethylfuran-3-carboxylate Methyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate methyl 4-[4-[[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methyl-methylamino]methyl]-5-methyl-1,3-oxazol-2-yl]benzoate Methyl 4′-((tert-Butoxycarbonyl)amino)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-... Methyl Beta-carboline-3 carboxylate methyl N-4-(5-(thiophen-2-yl)-3-(trifluoromethyl)-1H-pyrazol-1-yl)phenylsulfonylpyrrolidine-1-carbimidothioate methyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen... Methyl-((E)-4-pyridin-3-yl-but-3-enyl)-amine methyl-3-(1-methyl-2-pyrrolidinyl)pyridine -6-carboxylate hydrochloride methyl-3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H--1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoate acetate Methyl-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxylate methyl-6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate methyl-[1-(2-pyridin-3-yl-vinyl)-cyclopropyl]-amine fumarate methyl-{1-[2-(pyridin-3-yloxy)-ethyl]-cyclopropyl}-amine fumarate methyl-{1-[3-(pyridin-3-yloxy)-propyl]-cyclopropyl}-amine fumarate methylcaconitine Methylcarbamylcholine Methylenedioxy-aminoindane Methylenedioxy-aminotetralin Methylenedioxy-N-benzylcathinone Methylenedioxyaminoindane Methylenedioxyaminotetralin methylenedioxybenzedrone METHYLERGONOVINE Methylethcathinone Methylhistamine-1,4 Methylhistamine-4 Methylhistaprodifen Methyllycaconitine Methylone METHYLPHENIDATE Methylphenidate-d METHYSERGIDE Meti-derm Metiamide Meticortelone Metimyd METITEPIN METOCLOPRAMIDE Metopimazine metoprolol mexiletine Mezerein MG624 MGBG MgCl2 MH.MZ MIANSERIN MIANSERIN (+) MIANSERIN (-) mianserine mibefradil Midazolam mifentidine Milnacipran Milrinone Minoxidil MIP-1Alpha Miquelianin miquelianin mirtazapine mirtazepine mirtazepine(+) mirtazepine(-) MISOPROSTOL MISOPROSTOL (Free Acid) MISOPROSTOL (Methyl Ester) Mitragynine mizolastine MJ-1998,(+/-) MJ-9184-1,(+/-) MK 212 MK 571 MK 678 MK-056 MK-329 MK-499 MK-801 MK-801,(+) MK-801,(-) MK-886 MK-912 ml-toxin 3 ML10302 ML10375 MLA MLN-518 MLT MLT-I-70 MLT-II-16 MLT-II-18 MLT-II-34 MMB-II-74 MMB-II-87 MMB-II-90 MMB-III-016 MMB-III-018 MMB-III-14 MMB-III-16 moclobemide, MCL MOLINDONE Montelukast MOPERONE Morphiceptin Morphiceptin [Val4] Morphinan-3,6 alpha-diol, 4, 5 alpha-epoxy-17-methyl- Morphinan-3,6-diol, 4, 5-epoxy-17-methyl-, (5alpha,6alpha)- Morphinan-6-one, 17-allyl-4,5alpha-epoxy-3,14-dihydroxy- Morphinan-6-one, 4,5-epoxy-3, 14-dihydroxy-17-methyl-, (5alpha)- Morphinan-6-one, 4,5alpha-epoxy-3, 14-dihydroxy-17-methyl- Morphine Morphine 6-glucuronide Morphine,(+) Morphine,(-) MORPHINE-SULFATE morphinone Morpholin-4-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone Morpholine-4-carboxylic Acid (2-Hydroxyethyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid (3-Cyanopropyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Butyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Ethyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Heptyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Hexyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Methyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Octyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Pentyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Phenethyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Morpholine-4-carboxylic Acid Propyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide Mosapride Motilin moxifloxacin Moxonidine Mpa MPC-MECA MPC-NECA MPEP MPP+ MPPG MPR-178 MPR-179 MPV 295 MR2034 MR2035 Mr2266 MRE 3008F20 MRE 3010F20 MRE 3046F20 MRE 3048F20 MRE 3055F20 MRE 3062F20 MRP3160 MRP3172 MRP3175 MRP3200 MRP3201 MRP3215 MRP4264 MRP4268 MRP4269 MRP4270 MRP5022 MRP5028 MRP5057 MRP5063 MRP5067 MRP5069 MRP5099 MRS1067 MRS1097 MRS1191 MRS3558 MRS5202 MRS5474 MRS5474 33618 MRS5676 MRS5678 MRS5697 MRS5697 33654 MRS5698 MRS5698 33655 MRS5755 MRS5755 33620 MRS5914 MRS5914 33653 MRS5917 MRS5917 33621 MRS5923 MRS5930 MRS5979 MRS5980 MRS7112 NS MRS7115 33740 MRS7119 33738 MRS7138 33736 MS-429 MS-449 MS-DMPX MSA-IV-35 MSPG MSR-I-032 MSX-2 MT-1 MT-2 MT-3 MT-4 MT-45 MT-5 MT-6 MT-7 MT-alpha MT-beta MTEP MTHPI MTPG MTX Muscimol MW011 Mybanil Myristicin n -Butyl 2,5-Dimethoxy-4-(2-aminopropyl)benzoate Hydrogen Oxalate n -Propyl 2,5-Dimethoxy-4-(2-aminopropyl)benzoate Hydrogen Oxalate N 0840 N 0889 N 0890 N 0891 N'-(4-tert-butylbenzyl)-N-{1-[4-(methylsulfonylamino)-3-fluorophenyl]-2-ethylpropyl}thiourea N,15-dimethyl-N-(1,3-thiazol-2-yl)tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-pheny... N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine N,N(CH3)2-Dmt-Tic-NH2 N,N,-di-propyl-5-carboxamido-tryptamine N,N,N-trimethyl-1-(4-bromo-2,5-dimethoxyphenyl)-2-aminopropane iodide N,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate N,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate N,N,O-TMS N,N,O-TRIMETHYLSEROTONIN N,N-(CH3)2-5-MeOT N,N-Bis[3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl]-N-allylamine N,N-Bis[3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl]-N-ethylamine N,N-Bis[3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl]-N-hydroxyethylamine N,N-di-n-Propyldopamine N,N-diallyl-Tyr-Aib-Aib-Phe-Leu N,N-diallyltryptamine N,N-dibenzyl-2-chloroethanamine N,N-Diethyl-1-(4-acetamidobenzenesulfonyl)tryptamine N,N-Diethyl-1-(4-aminobenzenesulfonyl)tryptamine N,N-Diethyl-2-oxo-2-[5-(quinoline-8-sulfonylamino)-1H-indol-3-yl]-acetamide N,N-Diethyl-2-[5-(naphthalene-1-sulfonylamino)-1H-indol-3-yl]-2-oxoacetamide N,N-Diethyl-2-{2-[4-(2-fluoroethoxy)phenyl]-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}acetamide N,N-Diethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan-1- amine N,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine N,N-diethyl-3-(6-methyl-8-phenyl-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)propan-1-amine N,N-diethyl-3-(8-(4-methoxyphenyl)-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)propan-1-amine N,N-diethyl-3-(8-(4-methoxyphenyl)-6-methyl-5,6,7,8-tetrahydro-2,6-naphthyridin-3-yloxy)propan-1-amine N,N-diethyllysergamide N,N-Diisobutyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide N,N-Diisopropyltryptamine N,N-DIISOPROPYLTRYPTAMINE, 5-HO N,N-DIISOPROPYLTRYPTAMINE, 5-HYDROXY N,N-DIISOPROPYLTRYPTAMINE, 5-OH N,N-dimethyl derivative N,N-dimethyl-1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride N,N-Dimethyl-1-(4-acetamidobenzenesulfonyl)tryptamine N,N-Dimethyl-1-(4-aminobenzenesulfonyl)tryptamine N,N-dimethyl-1-(4-bromo-2,5-dimethoxyphenyl)-2-aminopropane HBr N,N-dimethyl-1-(benzenesulfonyl)tryptamine N,N-Dimethyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)-ethan-1-amine Hydrochloride N,N-Dimethyl-2-(2'-amino-4'-(2-fluoroethyl)phenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-(3-fluoropropyl)phenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-(ethan-2-ol)phenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-(propan-3-ol)phenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-ethenylphenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-ethylphenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-hydroxymethylphenylthio)benzylamine N,N-dimethyl-2-(2'-amino-4'-iodophenylthio)benzylamine N,N-Dimethyl-2-(2'-amino-4'-methylphenylthio)benzylamine N,N-Dimethyl-2-(2'-aminophenylthio)benzylamine N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine N,N-dimethyl-3-((2-(tetrahydro-2H-thiopyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine N,N-dimethyl-3-((2-(tetrahydropyran-4-ylidene)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine N,N-Dimethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan1-amine N,N-dimethyl-3-((phenethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine N,N-Dimethyl-4-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine N,N-Dimethyl-4-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine N,N-Dimethyl-5-(2-fluoroethoxy)-2-(2-amino-4-methylphenoxy)benzylamine N,N-Dimethyl-5-(3-fluoropropoxy)-2-(2-amino-4-methylphenoxy)benzylamine N,N-Dimethyl-5-(4-fluorobutoxy)-2-(2-amino-4-methylphenoxy)benzylamine N,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine   N,N-dimethyl-AMAA N,N-dimethyl-AMPA N,N-Dimethyl-N-{2-[3-(phenylsulfonyl)-1H-indol-4-yl]ethyl}amine N,N-dimethylcarbamoyl-N,N-dimethylaminoethanol N,N-dimethylcarbamoylcholine N,N-Dimethylserotonin N,N-DIMETHYLTRYPTAMINE N,N-Dipropylserotonin N,N-Dipropyltryptamine N,omega-Methyltryptamine N,S-Dimethyl-N-phenethyldithiocarbamate N- Ethyl-1-deoxy-1-[e-amino-2- [ (1 -naphthyDethynyl] - 9H-purin-9-yl]-Beta-D-ribofuranuronamide N-(((3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)cyclopropanesulfonamide N-(((3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)naphthalene-1-sulfonamide N-(((3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)propane-1-sulfonamide N-(((3R,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)pyridine-3-sulfonamide N-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)-4-cyanobenzamide N-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)cyclopropanecarboxamide N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-ethylacetamide N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-pentylacetamide N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-propylacetamide N-((1-(2-(tert-Butylamino)-2-oxoethyl)piperidin-4-yl)methyl)-9- pentyl-9H-carbazole-3-carboxamide N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-(cyclohexylmethyl)acetamide N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-ethylacetamide N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-pentylacetamide N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-propylacetamide N-((1-benzylpiperidin-4-yl)methyl)-N-(cyclohexylmethy)acetamide N-((1-benzylpiperidin-4-yl)methyl)-N-butylacetamide N-((1-benzylpiperidin-4-yl)methyl)-N-ethylacetamide N-((1-benzylpiperidin-4-yl)methyl)-N-pentylacetamide N-((1-benzylpiperidin-4-yl)methyl)-N-propylacetamide N-((1R,2R)-2-aminocyclohexyl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide N-((1r,4r)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1r,4r)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1S,2S)-2-aminocyclohexyl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide N-((1s,4s)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide N-((5E,13E)-(3S,4R,11S,12R)-11-Toluenesulfonamide-4,12-dimethyl-8,16-dioxo-1,9dioxa-cyclohexadeca-5,13-dien-3-yl)-toluenesulf... N-((S)-1-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-3-yl)cyclohexanecarboxamide N-((S)-3-(1-hydroxy-1-phenyl)propylpiperidin-4-yl)-1-naphthamide N-(1)-(S)-Fenchyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-(1)-(S)-fenchyl-6-chloro-2,5-dimethyl-1-(4- methylbenzyl)-1,4-dihydroindeno[1,2-b]pyrrole-3-carboxamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-yl)-2-methoxybenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-yl)-2-phenylacetamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-yl)-4-fluorobenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-yl)-4-nitrobenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-5-yl)cyclopropanecarboxamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-6-yl)-2-methoxybenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-6-yl)-2-nitrobenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-6-yl)-3-nitrobenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-6-yl)-4-nitrobenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-6-yl)propionamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-7-yl)-2-methoxybenzamide N-(1,2,3,4-Tetrahydro-1,3,4-trioxoisoquinolin-7-yl)-4-nitrobenzamide N-(1,2,3,4-Tetrahydroacridin-9-yl)-9-[(1,2,3,4-tetrahydro-9-yl)thio]nonan-1-amine N-(1,2,3,4-Tetrahydroacridin-9-yl)-N-(3-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)propyl)-1,4-butanediamine N-(1,2,3,4-Tetrahydroacridin-9-yl)-N-[8-(1,2,3,4-tetrahydroacridin-9-yl)oct-1-yl]amine N-(1,2,3,4-tetrahydronaphthalen-1-yl)-6-(4-o-tolylpiperazin-1-yl)hexanamide N-(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl) N-(1,2-dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-2-chlorobenzamide N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-3-nitrobenzamide N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-acetamide N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-5-yl)-benzamide N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-benzamide N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamic acid N-(1,3,4-Trioxo-1,2,3,4-tetrahydro-isoquinolin-7-yl)-benzamide N-(1,3-Benzodioxol-5-ylmethyl)-2-cyclohexylidene-2-fluoroethanamine N-(1-((5-ethoxy-6-methoxypyridin-3-yl)methyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide N-(1-(2,3,4,5,6-F-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(2-((N-Methylsulfonyl)amino)ethyl)piperidin-4-yl)-1-isopropylindazole-3-carboxamide Maleate N-(1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl) quinoline-8-sulfonamide N-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide N-(1-(2-Cl-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(2-Cl-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(2-Me-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(2-Me-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(2-Pyridyl)-piperidin-4-yl)-2-naphthamide N-(1-(3,4-dimethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3,5-diethoxy-2-fluorobenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3,5-diisopropoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-(2-fluoroethoxy)-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-(cyclopentyloxy)-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-(ethylamino)-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-Br-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(3-Br-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(3-CF3-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(3-CF3-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(3-Cl-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(3-Cl-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(3-ethoxy-4-(trifluoromethyl)benzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-fluorobenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-isopropoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)-5-(ethylsulfonyl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)-5-(trifluoromethoxy)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)-5-nitrobenzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)oxazolo[4,5-b]pyridin-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)oxazolo[5,4-b]pyridin-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)oxazolo[5,4-c]pyridin-2-amine N-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-yl)thiazolo[5,4-b]pyridin-2-amine N-(1-(3-ethoxy-4-methoxyphenyl)piperidin-4-yl)benzo[d]thiazol-2-amine N-(1-(3-ethoxy-4-methylbenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-5-(tetrahydro-2H-pyran-4-yloxy)benzyl)piperidin-4-yl)-5-(ethylsulfonyl)benzo[d]oxazol-2-amine N-(1-(3-ethoxy-5-(tetrahydro-2H-pyran-4-yloxy)benzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(3-Me-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(3-Me-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(3-MeO-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(3-MeO-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(3-Phenylbutyl)piperidin-4-yl)-2-naphthamide N-(1-(3-Phenylpropyl)piperidin-4-yl)-2-naphthamide N-(1-(3-Pyridyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-amino-3,5-diethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(4-Br-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(4-Br-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-CF3-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(4-CF3-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-chloro-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(4-Cl-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(4-Cl-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-cyclopropoxy-3-ethoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(4-Me-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(4-Me-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-MeO-benzyl)-piperidin-4-yl)-1-naphthamide N-(1-(4-MeO-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-methoxy-3-propoxybenzyl)piperidin-4-yl)benzo[d]oxazol-2-amine N-(1-(4-NO2-benzyl)-piperidin-4-yl)-2-naphthamide N-(1-(4-Pyridyl)-piperidin-4-yl)-2-naphthamide N-(1-(allyloxy)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide N-(1-Benzyl-3-pyrrolidinyl)-2'-formyl-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-3'-fluoro-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-3-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-4'-(methylsulfanyl)-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-4'-(trifluoromethyl)-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-4'-chloro-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-4'-fluoro-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-4'-formyl-4-biphenylcarboxamide N-(1-Benzyl-3-pyrrolidinyl)-4-(2-thienyl)benzamide N-(1-Benzyl-3-pyrrolidinyl)-4-(3-thienyl)benzamide N-(1-Benzyl-3-pyrrolidinyl)-4-biphenylcarboxamide N-(1-Benzylpiperidin-4-yl)-1-isopropylindazole-3-carboxamide Hydrochloride N-(1-Benzylpiperidin-4-yl)-1-naphthamide N-(1-Benzylpiperidin-4-yl)-2-naphthamide N-(1-Benzylpiperidin-4-yl)-4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)benzenesulfonamide N-(1-Phenylethylpiperidin-4-yl)-1-naphthamide N-(1-Phenylethylpiperidin-4-yl)-2-naphthamide N-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)-8-quinolinesulfonamide N-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)quinoline-2-carboxamide N-(1-{2-[(Propan-2-yl)-phenyloxy]ethyl}pyrrolidin-3-yl)thiophene-2-sulfonamide N-(11-Amino-5,6-dihydro-7-thia-8,10-diazabenzo[c]fluoren-3-yl)-N'-(3-methylphenyl)urea N-(1H-benzimidazol-2-yl)-3-(4-oxo-3H-quinazolin-2-yl)propanamide N-(1H-imidazol-2-yl)-15-methyltetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamide N-(1R,2R,3R,5S)-Isopinocampheyl-5-(4-chloro-3- methylphenyl)-1-(4-methylbenzyl)-1H-pyrrole-3-carboxamide N-(1S,2R)-Myrtanyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride N-(2,3-Dihydro-5,6-dimethoxy-1H-inden-2-yl)-N-propyl-2-thiopheneethanamine N-(2,3-Dihydro-5,6-dimethoxy-1H-inden-2-yl)-N-propyl-3-pyridineethanamine N-(2,3-Dihydro-5,6-dimethoxy-1H-inden-2-yl)-N-propyl-3-thiopheneethanamine N-(2,3-Dihydro-5,6-dimethoxy-1H-inden-2-yl)-N-propyl-3-thiophenemethanamine N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide N-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide N-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide N-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide N-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide N-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide N-(2,6-di-p-tolylpyrimidin-4-yl)butyramide N-(2,6-di-p-tolylpyrimidin-4-yl)propionamide N-(2,6-diisopropylphenyl)-4-(3-(4-methylbenzyl)-1,2,4-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide N-(2,6-diphenylpyrimidin-4-yl)acetamide N-(2,6-diphenylpyrimidin-4-yl)butyramide N-(2,6-diphenylpyrimidin-4-yl)propionamide N-(2,6-distyrylpyrimidin-4-yl)acetamide N-(2,6-distyrylpyrimidin-4-yl)butyramide N-(2,6-distyrylpyrimidin-4-yl)propionamide N-(2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethyl)-4-cyanobenzamide N-(2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethyl)-4-cyanobenzenesulfonamide N-(2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethyl)acetamide N-(2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethyl)cyclopropanesulfonamide N-(2-((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethyl)pyridine-3-sulfonamide N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro... N-(2-((5-((3-Chlorophenoxy)methyl)isoxazol-3-yl)oxy)ethyl)-N-methylcyclohexanamine Hydrochloride N-(2-((5-((3-Fluorophenoxy)methyl)isoxazol-3-yl)oxy)ethyl)-N-methylcyclohexanamine Hydrochloride N-(2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazol-5-yl)-1-methyl-1H-imidazole-4-sulfonamide N-(2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazol-5-yl)acetamide N-(2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazol-5-yl)benzenesulfonamide N-(2-(1-(3-ethoxy-4-methoxybenzyl)piperidin-4-ylamino)benzo[d]oxazol-5-yl)cyclobutanecarboxamide N-(2-(1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)ethyl)cyclopropanesulfonamide N-(2-(2-Me-benzyl)-piperidin-4-yl)-2-naphthamide N-(2-(2-phenyl-6-(4-(3-phenylpropyl)piperazine-1-carbonyl)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)ethyl)acetamide N-(2-(4-((Benzyloxycarbonyl)amino)-1-piperidinyl)-ethyl)-1-isopropylindazole-3-carboxamide Oxalate N-(2-(4-(1-Adamantylcarboxamido)-1-piperidinyl)ethyl)-1-isopropylindazole-3-carboxamide Oxalate N-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) picolinamide N-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-N-(pyridin-2-yl)cyclohexanecarboxamide trihydrochloride N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide N-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl) picolinamide N-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propyl) picolinamide N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) picolinamide N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide N-(2-(4-(4-fluorophenyl)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-2-oxoethyl)-N-isobutylfuran-2-carboxamide N-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(4-fluorophenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)-N-isopropyl-3,3-dimethylbutanamide N-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) picolinamide N-(2-(4-(furoyl)piperazin-1-yl)ethyl)isonicotinamide N-(2-(4-(furoyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(o-tolyl)piperazin-1-yl)ethyl)isonicotinamide N-(2-(4-(piperonyl)piperazin-1-yl)ethyl)isonicotinamide N-(2-(4-(piperonyl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide N-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl) isonicotinamide N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide N-(2-(4-phenylpiperazin-1-yl)ethyl)isonicotinamide N-(2-(4-phenylpiperazin-1-yl)ethyl)picolinamide N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-4-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-fluorophenyl)-N-(3,4- dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2,5-dimethoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(2-methoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3,4,5-trimethoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(3-methoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-(4-methoxyphenyl)propan-1-amine N-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-N-(3,4-dimethoxyphenethyl)-3-phenylpropan-1-amine N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)a... N-(2-amino-2-methylpropyl)-4-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyl)-7-methoxybenzofuran-2-carboxamide N-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(2-Bromobenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(2-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(2-chlorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-(2-chloroethyl)icosa-5,8,11,14-tetraenamide N-(2-Cyanoethyl)-N-ethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide N-(2-Cyclohexylidene-2-fluoroethyl)- 4-piperidinamine N-(2-Cyclohexylidene-2-fluoroethyl)-1-adamantanamine N-(2-Cyclohexylidene-2-fluoroethyl)-N-(2-phenylethyl)amine N-(2-Cyclohexylidene-2-fluoroethyl)-N-(4-fluorobenzyl)amine N-(2-Cyclohexylidene-2-fluoroethyl)-N-(4-methoxybenzyl)amine N-(2-Cyclohexylidene-2-fluoroethyl)-N-[3-(trifluoromethyl)benzyl]amine N-(2-Cyclohexylidene-2-fluoroethyl)aniline N-(2-Cyclohexylidene-2-fluoroethyl)cyclohexanamine N-(2-Cyclopentylidene-2-fluoroethyl)-N-(2-phenylethyl)amine N-(2-Cyclopentylidene-2-fluoroethyl)-N-(2-pyridinylethyl)amine N-(2-Cyclopentylidene-2-fluoroethyl)-N-(4-fluorobenzyl)amine N-(2-Cyclopentylidene-2-fluoroethyl)-N-(4-methoxybenzyl)amine N-(2-Cyclopentylidene-2-fluoroethyl)cyclohexanamine N-(2-Dimethylaminoethyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-(2-ethoxybenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-(2-fluoro-4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide N-(2-fluoro-5-(2-(4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide N-(2-fluoro-5-(2-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide N-(2-fluoro-5-(2-(8-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-3-azabicyclo[3.2.1]octan-3-yl)ethoxy)phenyl)methanesulfon... N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate N-(2-hydroxyethyl)-2-(4-(1-methyl-2,4-dioxo-3-propyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide N-(2-Hydroxyethyl)-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine N-(2-Hydroxyethyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-(2-methoxy-6-methyl-1-(prop-2-yn-1-yloxy)-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide N-(2-Methoxy-phenyl)-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-(2-Methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(2-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine hydrochloride N-(2-methoxybenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-(2-methoxyethyl)-2-[4-(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-5-yl)piperazin-1-yl]acetamide N-(2-methoxyethyl)-N-[1-(2-thiophen-2-ylethyl)piperidin-4-yl]acetamide N-(2-Methyl-2-propanyl)-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide N-(2-Methylphenyl)-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-(2-Phenylethylpiperidin-4-yl)-1-naphthamide N-(3,3-Diphenyl)propyl-2,2-diphenylacetamide N-(3,3-Diphenyl)propyl-2-(4-bromophenyl) acetamide N-(3,3-Diphenyl)propyl-2-(4-chlorophenyl)acetamide N-(3,3-Diphenyl)propyl-2-chloro-2,2-diphenylacetamide N-(3,3-Diphenyl)propyl-2-hydroxy-2,2-diphenylacetamide N-(3,3-Diphenyl)propyl-2-methyl-2,2-diphenylacetamide N-(3,3-Diphenyl)propyl-2-phenylacetamide N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide N-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride N-(3-((3-ethoxy-4-methoxyphenylamino)methyl)phenyl)benzo[d]thiazol-2-amine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro... N-(3-(1-(3-(dimethylamino)propyl)piperidin-4-yl)-1H-indol-5-yl)-4-fluorobenzamide N-(3-(1-benzylpiperidin-4-yl)-1H-indol-5-yl)-4-fluorobenzamide N-(3-(1H-Imidazol-1-yl)propyl)-1-(3,4-dimethoxyphenyl)cyclopropanecarbothioamide N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-chlorophenyl)cyclobutanecarbothioamide N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-chlorophenyl)cyclopentanecarbothioamide N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-methoxyphenyl)cyclohexanecarbothioamide N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-methoxyphenyl)cyclopropanecarbothioamide N-(3-(1H-Imidazol-1-yl)propyl)-2,2-diphenylethanethioamide N-(3-(1H-Imidazol-1-yl)propyl)-2-(3,4-dimethoxyphenyl)ethanethioamide N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)pheno... N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phen... N-(3-(1H-Imidazol-1-yl)propyl)-5,6-dimethoxybenzo[d]thiazol-2-amine N-(3-(1H-Imidazol-1-yl)propyl)-6-chlorobenzo[d]thiazol-2-amine N-(3-(1H-Imidazol-1-yl)propyl)-6-methoxybenzo[d]thiazol-2-amine N-(3-(1H-imidazol-1-yl)propyl)benzo[d]thiazol-2-amine N-(3-(1H-indol-4-yloxy)-2-methoxypropyl)cyclohexanamine N-(3-(1H-indol-4-yloxy)propyl)cyclohexanamine N-(3-(1H-indol-4-yloxy)propyl)cyclopentanamine N-(3-(2-(4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide N-(3-(2-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide N-(3-(2-(8-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-3-azabicyclo[3.2.1]octan-3-yl)ethoxy)phenyl)methanesulfonamide N-(3-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide N-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) picolinamide N-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) picolinamide N-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) picolinamide N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide N-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine N-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) picolinamide N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide N-(3-(4-(furoyl)piperazin-1-yl)propyl)isonicotinamide N-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(o-tolyl)piperazin-1-yl)propyl)isonicotinamide N-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide N-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide N-(3-(4-phenylpiperazin-1-yl)propyl)isonicotinamide N-(3-(4-phenylpiperazin-1-yl)propyl)picolinamide N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxam... N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenox... N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)pheno... N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)... N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt N-(3-Bromobenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(3-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamide N-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide N-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide N-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-methyl-2-(p-tolylamino)thiazole-5-carboxamide N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide N-(3-Chlorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamide N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4- (dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamide N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide N-(3-Ethoxy-phenyl)-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol N-(3-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane N-(3-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol N-(3-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decane N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide N-(3-Iodobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-iodoprop-2E-enyl)-2B-carbomethoxy-3B-(3',4'-dichlorophenyl)nort.. N-(3-Methoxy-phenyl)-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-(3-Methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(3-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol N-(3-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decane N-(3-Methylbenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide N-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride N-(3-Methylthiobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-Phenyl)propyl-2,2-diphenylacetamide N-(3-Phenyl)propyl-2-(4-bromophenylacetamide) N-(3-Phenyl)propyl-2-(4-chlorophenyl)-2-phenylacetamide N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine N-(3-Phenylpropylpiperidin-4-yl)-1-naphthamide N-(3-Propoxy-phenyl)-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-(3-Trifluoromethylbenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(3-TrifluoroMethylPhenyl) PIPERAZINE N-(3-{1-[2-carbamoyl-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)-4-flu... N-(3-{[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-methylamino}propyl)-3-(1H-indol-3-yl)propionamide N-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide N-(4,5-dimethyl-1,3-thiazol-2-yl)-15-methyltetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2,4,6,9(14),10,12-hexaene-15-carboxamid... N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide N-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide N-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide N-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide N-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide N-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide N-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide N-(4,6-di-tolylpyrimidin-2-yl)propionamide N-(4,6-dip-tolylpyrimidin-2-yl)acetamide N-(4,6-dip-tolylpyrimidin-2-yl)butyramide N-(4,6-diphenylpyrimidin-2-yl)acetamide N-(4,6-diphenylpyrimidin-2-yl)butyramide N-(4,6-diphenylpyrimidin-2-yl)propionamide N-(4,6-distyrylpyrimidin-2-yl)acetamide N-(4,6-distyrylpyrimidin-2-yl)butyramide N-(4,6-distyrylpyrimidin-2-yl)propionamide N-(4,6-dithiophen-2-ylpyrimidin-2-yl)propanamide N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro... N-(4-(2-(1,3-dimethyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[1,2-a]purin-9(6H)-yl)ethoxy)phenyl)acetamide N-(4-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethoxy)phenyl)acetamide N-(4-(2-Chlorophenyl)piperazin-1-yl)-(5-(4-chloro-3- methylphenyl)-1-(4-methylbenzyl)-1H-pyrrole-3-carboxamide N-(4-(3-((methylamino)methyl)-4-(4-(methylthio)phenoxy)phenyl)but-3-ynyl)cyclopropanamine N-(4-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propoxy)phenyl)acetamide N-(4-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)acetamide N-(4-(3-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)phenyl) Acetamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-2-hydroxypropoxy)phenyl)acetamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)-2-methylphenyl)acetamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)benzyl)acetamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) benzamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) propionamide N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)-N-methylacetamide N-(4-(3-(4-(benzo[b]thiophen-4-yl)piperazin-1-yl)propoxy)phenyl)acetamide N-(4-(3-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)propoxy)phenyl) acetamide N-(4-(3-(4-(pyridin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide N-(4-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-7-methoxybenzofuran-2-carboxamide N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(2-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)benzo[c][1,2,5]oxadiazole-5-carboxamide N-(4-(4-(2-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal N-(4-(4-(2-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(2-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(3,4-dichlorophenoxy)-3-((methylamino)methyl)phenyl)but-3-ynyl)-N-methylcyclopropanamine N-(4-(4-(3,4-dichlorophenoxy)-3-((methylamino)methyl)phenyl)but-3-ynyl)cyclopropanamine N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(3-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide)benzamide N-(4-(4-(3-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(3-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(3-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt: N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide N-(4-(4-(4-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(4-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(4-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(4-(4-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt N-(4-(4-(4-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt: N-(4-(4-(m-Tolyl)piperazin-1-yl)butyl)benzo[b]furan-2-carboxamide N-(4-(4-phenylpiperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1H-1,2,3-triazole-4-carboxamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-2-methoxy-5-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-... N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-(2-fluoroethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)-be... N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-fluoroethoxy)ethyl)-1H-1,2,3-triazol-4-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(4-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzam... N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((2-(2-fluoroethoxy)ethoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-m... N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-(2-fluoroeth... N-(4-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- butyl)-4-(thiophen-3-yl)benzamide N-(4-Acetamidophenyl)indomethacinamide N-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt N-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide N-(4-bromobenzyl)-2-(1H-indol-3-yl)-2-oxoacetamide N-(4-Bromobenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(4-Bromobenzyl)-2-(5-methoxy-1H-indol-3-yl)N-(3-Fluorobenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide N-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide N-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide N-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide N-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide N-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide N-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide N-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide N-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide N-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide N-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide N-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide N-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl) benzamide N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide N-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide N-(4-chloro-3-(trifluoromethyl)phenyl)-2,7-dibenzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide N-(4-chloro-3-(trifluoromethyl)phenyl)-3-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide N-(4-chloro-3-(trifluoromethyl)phenyl)-7-(2-methoxyphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxami... N-(4-chloro-3-(trifluoromethyl)phenyl)-7-isopropyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide N-(4-chloro-3-(trifluoromethyl)phenyl)-7-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide N-(4-Chlorobenzhydryl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide N-(4-Chlorobenzyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(4-Chlorobenzyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-Chlorobenzyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(4-Chlorobenzyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-Chlorobenzyl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(4-Chlorobenzyl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-Chlorophenyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(4-Chlorophenyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-Chlorophenyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(4-Chlorophenyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-Chlorophenyl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(4-Chlorophenyl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(4-Cyanobutyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-(4-cyanophenyl)-2-(4-(2,4-dioxo-1,3-dipropyl-2,3,4,5-tetrahydro-1H-pyrrolo[3,2-d]pyrimidin-6-yl)phenoxy)acetamide N-(4-Cyanophenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide N-(4-Cyanophenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide N-(4-Cyanophenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide N-(4-Cyanophenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide N-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide N-(4-Dipropylaminobutyl)-4-biphenylcarboxamide N-(4-ethylbenzyl)-2-(1H-indol-3-yl)-2-oxoacetamide N-(4-ethynylbenzyl)-2-(1H-indol-3-yl)-2-oxoacetamide N-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride (3) N-(4-Fluoro-benzyl)-2-(1H-indol-3-yl)-2-oxo-acetamide N-(4-Fluoro-phenyl)-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-(4-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol N-(4-Fluorobenzyl)-2-azatricyclo[3.3.1.13,7]decane N-(4-fluorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-(4-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol N-(4-Fluorophenethyl)-2-azatricyclo[3.3.1.13,7]decane N-(4-Fluorophenyl)-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyla... N-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide N-(4-Methanesulfonyloxyphenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide N-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide N-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide N-(4-Methanesulfonyloxyphenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide N-(4-Methoxy-benzyl)-2-(5-nitro-1H-indol-3-yl)-2-oxo-acetamide N-(4-Methoxy-phenyl)-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-(4-Methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride N-(4-Methoxybenzyl)-2-(5-methoxy-1H-indol-3-yl)ethan-1-amine maleate N-(4-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decan-1-ol N-(4-Methoxybenzyl)-2-azatricyclo[3.3.1.13,7]decane N-(4-methylthiazol-2-yl)benzamide hydrobromide N-(4-Nitro-benzyl)-2-(5-nitro-1H-indol-3-yl)-2-oxo-acetamide N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide N-(4-Phenylbutylpiperidin-4-yl)-1-naphthamide N-(4-Propylaminobutyl)-4-biphenylcarboxamide N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide N-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide N-(4-tert-butylbenzyl)-N'-{1-methyl-1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-methyl-1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-methyl-1-[4-(methylsulfonylamino)phenyl]ethyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]cyclopropyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)-3-fluorophenyl]-2-phenylethyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)-3-fluorophenyl]propyl}thiourea N-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)phenyl]cyclopropyl}thiourea N-(4-tert-butylbenzyl)-N'-{[4-(methylsulfonylamino)-3-fluorophenyl](phenyl)methyl}thiourea N-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine-1(2H)-carboxamide N-(4-{(R)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide N-(4-{(S)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide N-(4-{1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide N-(4-{2-[((S)-2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-propyl-amino]-ethyl}-cyclohexyl)-3-phenyl-acrylamide N-(4-{4-Amino-6-[(4-methylpiperazin-1-yl)methyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea N-(4-{4-Amino-6-[(dimethylamino)methyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea N-(4-{4-Amino-6-[2-(dimethylamino)ethyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide N-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide N-(5-(2-Amino-1-(4-(trifluoromethyl)phenyl)-1H-imidazole5-carbonyl)-4IJdimethylamino)thiazol-2-yl)benzamide N-(5-(2-Amino-1-(4-chlorophenyl)-1H-imidazole-5-carbonyl)-4-(dimethylamino)thiazol-2-yl)benzamide N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide N-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-(4-(Methylsulfonyl)benzoyl)-4-phenylthiazol-2-yl)benzamide N-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methoxybenzamide N-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methylbenzamide N-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide N-(5-(4-Chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methylbenzamide N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide N-(5-(4-Chlorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-(4-Methoxybenzoyl)-4-phenylthiazol-2-yl)benzamide N-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-(4-Methylbenzoyl)-4-phenylthiazol-2-yl)benzamide N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide N-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide N-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide N-(5-Benzoyl-4-phenylthiazol-2-yl)-4-methylbenzamide N-(5-Benzoyl-4-phenylthiazol-2-yl)benzamide N-(5-Benzoyl-4-phenylthiazol-2-yl)furan-2-carboxamide N-(5-methyl-1,2-oxazol-3-yl)-3-[4-[(1S)-1-pyridin-3-ylethyl]piperazin-1-yl]propanamide N-(5-methyl-1,2-oxazol-3-yl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,2-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2-phenylacetamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-3-phenylpropanamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)furan-2-carboxamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isoxazole-5-carboxamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide N-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide N-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) benzenesulfonamide N-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-1-sulfonamide N-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-2-sulfonamide N-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-4- methyl-N-phenylbenzenesulfonamide N-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-N-(3- (trifluoromethyl)phenyl)benzenesulfonamide N-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzamide N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide N-(6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-yl)-acetamide N-(6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-yl)-acetamide N-(6-Methyl-2-pyridinyl)-1-naphthamide N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)acetamide N-(6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-10-yl)butamide N-(6-methylpyridin-2-yl)-1-naphthamide hydrobromide N-(6-methylpyridin-2-yl)-1H-indole-2-carboxamide N-(6-methylpyridin-2-yl)-2,3'-bipyridine-6'-carboxamide N-(6-methylpyridin-2-yl)-2-phenylthiazole-4-carboxamide N-(6-methylpyridin-2-yl)-3-(trifluoromethyl)benzamide hydrobromide N-(6-methylpyridin-2-yl)-3-phenethoxybenzamide hydrobromide N-(6-methylpyridin-2-yl)-3-phenoxybenzamide hydrobromide N-(6-methylpyridin-2-yl)-4-(pyrimidin-2-yl)picolinamide N-(6-methylpyridin-2-yl)-4-(thiophen-2-yl)picolinamide N-(6-methylpyridin-2-yl)-5-(thiophen-2-yl)picolinamide N-(6-methylpyridin-2-yl)-5-phenylpicolinamide N-(6-methylpyridin-2-yl)benzamide hydrobromide N-(6-methylpyridin-2-yl)benzofuran-2-carboxamide N-(6-methylpyridin-2-yl)benzo[b]thiophene-2-carboxamide N-(6-methylpyridin-2-yl)biphenyl-3-carboxamide hydrobromide N-(6-methylpyridin-2-yl)isoquinoline-1-carboxamide N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide N-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide N-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide N-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide N-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide N-(9,10-Dihydro-9-anthracenylmethyl)-2-phenylethanamine N-(9,10-Dihydro-9-anthracenylmethyl)-3-phenyl-1-propanamine N-(9,10-Dihydro-9-anthracenylmethyl)-4-phenyl-1-butanamine N-(Adamant-1-yl)-1-allyl-5,8-dimethoxy-4-oxo-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-4-oxo-1-pentyl-6-(phenylthio)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-4-oxo-1-pentyl-6-(trifluoromethyl)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-4-oxo-1-pentyl-6-phenyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-4-oxo-1-pentyl-7-(phenylsulfinyl)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-4-oxo-1-pentyl-7-(phenylsulfonyl)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-4-oxo-1-pentyl-7-(phenylthio)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-5,8-dimethoxy-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-6-(3-chloro-4-fluorophenoxy)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-6-bromo-1-(but-3-en-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-6-bromo-4-oxo-1-(pent-4-en-1-yl)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-6-bromo-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-6-fluoro-4-oxo-1-pentyl-7-(1H-pyrrol-1-yl)-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-6-isopropyl-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-7-chloro-8-methyl-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)-7-fluoro-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N-(Adamant-1-yl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-(Adamant-1-yl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-(Adamant-2-yl)-S-methyl-dithiocarbamate N-(Adamantan-1-yl)-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride N-(Azepan-1-yl)-1-(4-Chlorophenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxamide N-(azepan-1-yl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(methylthio)-1H-imidazole-4-carboxamide N-(azepan-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methylthio)-1H-pyrazole-3-carboxamide N-(benzo[d]thiazol-2-yl)-1-(3-ethoxy-4-methoxybenzyl)piperidine-4-carboxamide N-(benzo[d]thiazol-2-yl)-4-(3-ethoxy-4-methoxyphenyl)piperazine-1-carboxamide N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(2,5-dimethoxy-4-(methylthio)phenyl)ethanamine hydrochloride N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(2,5-dimethoxy-4-(propylthio)phenyl)-ethanamine hydrochloride N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(2,5-dimethoxy-4-(trifluoromethyl)phenyl)- ethanamine hydrochloride N-(Benzo[d][1,3]dioxol-4-ylmethyl)-2-(4-(ethylthio)-2,5-dimethoxyphenyl)-ethanamine hydrochloride N-(benzyloxy)-3-{[(1S)-2-(4,5-diphenyl-1,3-oxazol-2-yl)-2-cyclohexen-1-yl]methyl}benzamide N-(benzylsulfonyl)-3-{[(1S)-2-(4,5-diphenyl-1,3-oxazol-2-yl)-2-cyclohexen-1-yl]methyl}benzamide N-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine N-(cyclohexylmethyl)-N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)acetamide N-(Cyclopropylmethyl)-2-((5-((3-fluorophenoxy)methyl)-isoxazol-3-yl)oxy)-N-methylethan-1-amine Hydrochloride N-(Cyclopropylmethyl)-N-methyl-2-((5-(phenoxymethyl)-isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride N-(Endo-[2.2.1]bicyclohept-2-yl)-1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazole-4-carboxamide N-(furan-2-ylmethyl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]prop-2-yn-1-amine N-(Indan-2-yl)-S-methyl-dithiocarbamate N-(m-trifluoromethylphenyl)piperazine N-(Naphthalen-1-yl)-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-(pyridin-2-yl)benzamide hydrobromide N-(R)-()-Cyclohexylethyl-5-(4-chloro-3-methylphenyl)-1- (4-methylbenzyl)-1H-pyrrole-3-carboxamide N-(R)-(þ)-Bornyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-(S)-(þ)-Cyclohexylethyl-5-(4-chloro-3-methylphenyl)-1- (4-methylbenzyl)-1H-pyrrole-3-carboxamide N-(Tert-butoxy)-1-(4-Chlorophenyl)-2-(2,4-dichloro-phenyl)-5-methyl-1H-imidazole-4-carboxamide N-({1-[2-(3-Fluorophenoxy)ethyl]piperidin-4-yl}methyl)thiophene-2-sulfonamide N-0434 N-0437 N-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-3,4-dichlorobenzyl 1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-3,4-dichlorobenzyl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-3,4-dichlorobenzyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-3,4-dichlorobenzyl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-3,4-dichlorobenzyl 1-(4-chlorophenyl)-3-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-4-carboxamide N-3,4-dichlorobenzyl 4-cyano-1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-3,4-dihlorobenzyl 1-(2,4,6-trichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-4-Fluorophenethyl-S-methyl-dithiocarbamate N-Acetyl-2-hydrazinobenzenesulfonamide N-Acetyl-4-[(carboxycarbonyl)(2-carboxyphenyl)- amino]-N-pentyl-3-(2-hydroxyethane)phenylalaninamide N-Acetyl-4-[(carboxycarbonyl)(2-carboxyphenyl)amino]-3-isopropyl-N-pentylphenylalaninamide N-acetyl-5-hydroxytryptamine N-Acetylhistamine N-Acetyltryptamine N-Acetyltryptamine,5-Benzyloxy N-Acetyltryptamine,5-Hydroxy N-Acetyltryptamine,5-Methyl N-Adamantylmethane-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-Allyl-2-(5-methoxy-1H-indol-3-yl)acetamide N-Allyl-2-[(2-amino-4-methylphenyl)thio]-benzenemethanamine N-Allyl-3-(5-methoxy-1H-indol-3-yl)propanamide N-Allyl-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-Allyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine n-Allylnoroxymorphone N-Allynormetazocine N-alpha-methylhistamine N-arachidonylethanolamine N-benzhydryl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-2-fluorobenzamide N-benzhydryl-6-(2,6-dimethylmorpholino)-5-nitropyrimidin-4-amine N-Benzoyl-N-(4-chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-Benzoyl-N-(4-chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-Benzoyl-N-(4-chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-Benzoyl-N-(4-chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide N-Benzo[1,3]dioxol-5-yl-2-[5-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1-methyl-1H-pyrazol-3-yloxy]-acetamide N-benzyl-1-(2-bromo-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-benzyl-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-benzyl-1-(2-chloro-2-phenylethyl)-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-Benzyl-1-(9,10-dihydro-9-anthracenyl)methanamine N-Benzyl-1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-methylpiperidin-4-amine N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide N-Benzyl-2-azatricyclo[3.3.1.13,7]decan-1-ol N-Benzyl-2-azatricyclo[3.3.1.13,7]decane N-Benzyl-2-cyclohexylidene-2-fluoroethanamine N-Benzyl-2-cyclopentylidene-2-fluoroethanamine N-Benzyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide N-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide N-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide N-Benzyl-4-(2-methylthiophenyl)-1-piperazinehexanamide N-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide N-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethylbenzofuran-2-carboxamide N-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N-ethyl-3-methylbenzofuran-2-carboxamide N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine N-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine N-benzyl-8-bromo-9-propyl-9H-purin-6-amine N-benzyl-9-propyl-9H-purin-6-amine N-Benzyl-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-benzyl-N-methyl-2-[4-(1H-pyrazol-5-yl)piperidin-1-yl]acetamide N-Benzyl-N-methyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide N-Benzyl-N-[4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]amine N-Benzyl-N-[4-[4-(3-methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]amine N-Benzyl-S-methyl-dithiocarbamate N-butanyl-5 methoxy tryptamine N-butyl-1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-butyl-1-(2-chloro-2-(4-fluorophenyl)ethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-butyl-1-(2-chloro-2-phenylethyl)-6-(methylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-butyl-1-(2-chloro-2-phenylethyl)-6-(propylthio)-1H-pyrazolo[3,4-d]pyrimidin-4-amine N-butyl-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide N-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide N-Butyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide N-Butyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-butyl-4-(diphenylmethyl)-1,4-diazepane-1-carboxamide N-Butyl-4-[(2,4-dichlorophenyl)(phenyl)methyl]piperazine-1-carboxamide N-butyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-Butyl-8-fluoro-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-butyl-N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)acetamide N-butyl-N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)acetamide N-Butyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-CBCPT N-CHO-4,4'-diFBZT N-CPM-CACO N-Cyclobutyl-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]-amino}-8-fluorochromane-5-carboxamide N-Cycloheptyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cycloheptyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-Cycloheptyl-1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-1H-pyrazole-4-carboxamide N-Cycloheptyl-1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cycloheptyl-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-cycloheptyl-1-(2-morpholinoethyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide N-Cycloheptyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cycloheptyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(2,4,6-trichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-cyclohexyl 1-(4-chlorophenyl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cyclohexyl({1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}amino)sulfonamide N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide N-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide N-cyclohexyl-2-(2,4-dichlorophenyl)-1-p-tolyl-1H-imidazole-4-carboxamide N-cyclohexyl-2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-methylpyrimidin-4-amine N-Cyclohexyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide N-Cyclohexyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-cyclohexyl-4-((2,5-dichlorophenyl)(phenyl)methyl)piperazine-1-carboxamide N-cyclohexyl-4-((3,4-dichlorophenyl)(phenyl)methyl)piperazine-1-carboxamide N-cyclohexyl-4-(diphenylmethyl)-1,4-diazepane-1-carbothioamide N-cyclohexyl-4-(diphenylmethyl)-1,4-diazepane-1-carboxamide N-cyclohexyl-4-[(2,4-dichlorophenyl)(4-fluorophenyl)methyl]piperazine-1-carboxamide N-cyclohexyl-4-[(2,4-dichlorophenyl)(4-methoxyphenyl)methyl]piperazine-1-carboxamide N-cyclohexyl-4-[(2,4-dichlorophenyl)(4-phenoxyphenyl)methyl]piperazine-1-carboxamide N-Cyclohexyl-4-[(2,4-dichlorophenyl)(p-tolyl)methyl]piperazine-1-carboxamide N-Cyclohexyl-4-[(2,4-dichlorophenyl)(phenyl)methyl]-piperazine-1-carbothioamide N-Cyclohexyl-4-[(2,4-dichlorophenyl)(phenyl)methyl]-piperazine-1-carboxamide N-cyclohexyl-4-[(2,6-dichlorophenyl)(phenyl)methyl]piperazine-1-carboxamide N-cyclohexyl-4-{(2,4-dichlorophenyl)[4-(trifluoromethyl)phenyl]methyl}piperazine-1-carboxamide N-cyclohexyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-Cyclohexyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-cyclohexyl-7-(dimethylamino)-1-(2-morpholinoethyl)-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide N-cyclohexyl-7-methoxy-1-(2-morpholinoethyl)-4-oxo-1,4-dihydroquinoline-3-carboxamide N-Cyclohexyl-8-fluoro-3a,9b-dihydro-3H-thiochromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-cyclohexylmethyl 1-(4-chlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cyclopentyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cyclopentyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-Cyclopentyl-1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cyclopentyl-1-(2,4-sifluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-Cyclopentyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-Cyclopentyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-Cyclopentyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-(4-methoxy... N-Cyclopentyl-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine N-cyclopentyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide N-Cyclopropyl-1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-1H-pyrazole-4-carboxamide N-Cyclopropyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacet... N-cyclopropyl-4-(1-(2-((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine N-cyclopropyl-4-(1-(2-(2,3-dihydro-1H-inden-2-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine N-cyclopropyl-4-(1-(2-(5-fluoro-1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine N-cyclopropyl-4-(1-(2-(6-fluoro-1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine N-cyclopropyl-4-(1-(2-(7-fluoro-1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine N-cyclopropyl-4-(1-(2-(thiazol-4-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine N-cyclopropyl-N-(2-oxo-2-(4-p-tolylpyrrolo[1,2-a]quinoxalin-5(4H)-yl)ethyl)cyclopentanecarboxamide N-cyclopropyl-N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine N-Cyclopropylmethyl-14beta-4'-chlorocinnamoyloxy-7,8-dihydrocodeinone N-Cyclopropylmethyl-14beta-4'-methylcinnamoyloxy-7,8-dihydrocodeinone N-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone N-cyclopropylmethylnor-14beta-(p-chlorocinnamoylamino)-7,8-dihydrocode N-cyclopropylmethylnor-14Beta-(p-nitrocinnamoylamino)-7,8-dihydrocodei N-dealkylated Diethylpropion N-Decyl-3-(3-hydroxyphenyl)pyrrolidine N-Desalkylquetiapine N-DESMETHYLCLOZAPINE N-dipropyltryptamine, 1-Isopropyl-5-hydroxy N N-dipropyltryptamine, 5-Hydroxy-N N-EthyI-l-deoxy-l-[6-amino-2-(5-phenyl-l-pentyn-lyl)-9H-purin-9-yl]-beta-D-ribofuranuronamide N-EthyI-l-deoxy-l-[6-amino-2-[(2-formylphenyl)- ethynyl]-9H-purin-9-yl]-Beta)-D-ribofuranuronamide N-EthyI-l-deoxy-l-{6-amino-2-[[4-(3-fert-butoxy-3- oxopropenyl)phenyl]ethynyI]-9H-purin-9-yl}-Beta-D-ribofuranuronamide N-ethyl N-methyl EM-A N-ethyl N-methyl EM-A enolether N-ethyl, N-Methyl Erythromycin-A N-ethyl, N-methyl Erythromycin-A enol ether N-ethyl,N-methyl 4''deoxy EM-B enolether N-Ethyl- l-deoxy-1- [6-amino-2- [ (4-hydroxyphenyl)- ethynyl]-9H-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl- l-deoxy-1- [6-amino-2-[(2-thienyl)ethynyl] - 9H-purin-9-yl]-beta-D-ribofuranuronamide N-ethyl-1-((pyridin-3-yloxy)methyl)cyclopropanamine N-Ethyl-1-deoxy-1- [6-amino-2-(phenylethynyI)-9Hpurin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-1-deoxy-1- [6-amino-2-[ (2-pyridyl)ethynyl] - 9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-1-deoxy-1- [6-amino-2-[(4-pyridyl)ethynyl]- 9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-1-deoxy-1-( 6-amino-2-ethynyl-9H-purin-9-yl)-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(3-hydroxy-1-pentyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(3-hydroxy-1-propyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(3-hydroxy-3,5-dimethyl-l-hexyn-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(3-hydroxy-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(4-hydroxy-1-butyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(4-hydroxy-1-pentyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(5-hydroxy-1-pentyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-1-[6-amino-2-(6-hydroxy-1-hexyn-1-y1)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-1-deoxy-l-[6-amino-2-(3-N-piperidyl-l-propynl-yl)-9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-1-deoxy-l-[6-amino-2-[(2-furyl)ethynyl]-9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-1-deoxy-r-{6-amino-2-[(4-carboxamidophenyl)- ethynyl]-9H-purin-9-yl}-Beta-D-ribofuranuronamide N-Ethyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride N-Ethyl-2-(3-pyridinyl)ethanamine N-Ethyl-2-(4-hydroxyphenyl)-norapomorphine hydrochloride N-Ethyl-2-methylnorapomorphine hydrochloride N-Ethyl-2-phenylnorapomorphine hydrochloride N-Ethyl-2-{6-[2-(4-methoxyphenyl)ethyl]-3-pyridinyl}-N-methylethanamine N-ethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine N-Ethyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide N-Ethyl-5-((5-methoxy-1H-indol-3-yl)methyl)-1,3,4-thiadiazol-2-amine N-ethyl-6-(4-((phenethylamino)methyl)phenoxy)nicotinamide N-Ethyl-l-deoxy-1-[6-amino-2-(1-cyclohexenylethyny1)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(3,3-diethoxy-1-propyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(3-amino-1-propyn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(3-hydroxy-3-phenyl-1-butyn-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(3-hydroxy-3-phenyl-l-propyn-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(3-methylbut-3-en-1-yn-1-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(3-phenyl-l-propyn-lyl)-9H-purin-9-yI]-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(5-chloro-l-pentyn-l-yl)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(5-cyano-1-pentyn-1-y1)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-(cyclohexylethyny1)-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-[2-(1-aminocyclohexy1)-ethynyl]-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-[2-(1-hydroxycyclopenty1)-ethynyl]-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-[3-(N,N-dimethylamino)-l-propyn-l-yl]-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-1-[6-amino-2-[4-(2-tetrahydro-2H-pyrany1oxy)-l-butyn-l-yl]-9H-purin-9-yl]-B-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-(3-N-imidazolyl-l-propyn-l-yl)-9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-(3-N-morpholinyl-l-propyn-l-yl)-9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-(4-phenyl-l-butyn-l-yl)- 9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-(4-tolylethynyl)-9ifpurin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(2-thiazolyI)ethynyI]-9H-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(3-formylphenyl)- ethynyl]-9H-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(3-pyridyl)ethynyl]- 9H-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(4-acetyIphenyl)- ethynyl] -9H-purin-9-yl] -Beta-D-ribofiiranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(4-aminophenyl)- ethynyl]-9H-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(4-fluorophenyl)- ethynyl]-977-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(4-formylphenyl)- ethynyl]-9H-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(4-methoxyphenyl)- ethynyl]-9i-purin-9-yl]-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-amino-2-[(4-nitrophenyl)ethynyl]- 9jH-purin-9-yl]-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-[6-ammo-2-(3-N-thiomorpholinyI-1-propyn-1 -yl)-9H-purin-9-yl] -beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-{6-amino-2-[3-(4-methyl-N-piperazinyl)-l-propyn-l-yl]-9H-purin-9-yl}-beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-{6-amino-2-[[4-(2-carboxyethyl)- phenyl]ethynyl]-9H-purin-9-yl}-Beta-D-ribofuranuronamide N-Ethyl-l-deoxy-l-{6-amino-2-[[4-(cyanomethyl)- phenyl]ethynyl]-9f-purin-9-yl}-D-ribofuranuronamide N-Ethyl-l-deoxy-l-{6-amino-2-[[4-(trifluoromethyl)- phenyl]ethynyl]-9f-purin-9-yl}-Beta-D-ribofuranuronamide N-Ethyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine N-ethyl-N-Antmethyl (4,4) N-Ethyl-N-methyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)-ethan-1-amine Hydrochloride N-Ethyl-N-methyl-2-(3-pyridinyl)ethanamine N-Ethyl-N-methyl-2-(5-propyl-3-pyridinyl)ethanamine N-Ethyl-N-methyl-2-(6-methyl-3-pyridinyl)ethanamine N-Ethyl-N-methyl-2-[6-(2-phenylethyl)-3-pyridinyl]ethanamine N-Ethyl-N-methyl-3-[3-(phenylsulfonyl)-1H-indol-4-yl]propan-1-amine N-Ethyl-N-methyl-N-{2-[3-(phenylsulfonyl)-1H-indol-4-yl]ethyl}amine N-Ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-Ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isonicotinamide N-Ethyl-N-{2-[3-(phenylsulfonyl)-1H-indol-4-yl]ethyl}amine N-ethylcarboxiamidoadenosine N-ethylpyridinium iodide N-formylnormorphine N-Heptyl-3-(3-hydroxyphenyl)pyrrolidine N-hexanyl-5 methoxy tryptamine N-Hexyl-3-(3-hydroxyphenyl)pyrrolidine N-Homopiperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride N-isopropyl-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide N-Isopropyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide N-Isopropyl-3-[3-(phenylsulfonyl)-1H-indol-4-yl]propan-1-amine N-Isopropyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-isopropyl-6-(4-((phenethylamino)methyl)phenoxy)nicotinamide N-isopropyl-N-(2-(4-(4-methoxyphenyl)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-2-oxoethyl)cyclohexanecarboxamide N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]dia... N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[... N-Me-Arg11 N-Me-Arg14 N-Me-bicuculline N-Me-Gly10 N-Me-Leu9 N-Me-Nle8 N-Menthyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-Met N-methepibatidine N-Methoxy-N-methyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide N-methyl(2-(3-methyl-4-(methylthio)phenoxy)-5-(4-morpholinobut-1-ynyl)phenyl)methanamine N-methyl(2-(4-(methylthio)phenoxy)-4-(4-morpholinobut-1-ynyl)phenyl)methanamine N-methyl(2-(4-(methylthio)phenoxy)-5-(4-(piperidin-1-yl)but-1-ynyl)phenyl)methanamine N-methyl(2-(4-(methylthio)phenoxy)-5-(4-(piperidin-1-yl)but-1-ynyl)phenyl)methanamine N-methyl(2-(4-(methylthio)phenoxy)-5-(4-thiomorpholinobut-1-ynyl)phenyl)methanamine N-methyl(2-(4-(methylthio)phenoxy)-5-(4-thiomorpholinobutyl)phenyl)methanamine N-methyl(5-(4-morpholinobut-1-ynyl)-2-(4-(trifluoromethyl)phenoxy)phenyl)methanamine N-methyl(5-(4-morpholinobut-1-ynyl)-2-phenoxyphenyl)methanamine N-methyl-1-((1R,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride N-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride N-methyl-1-((1S,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride N-methyl-1-((5-vinylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride N-methyl-1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride N-methyl-1-((pyridin-3-yloxy)methyl)cyclopropanamine hydrochloride N-methyl-1-(2-(pyridin-3-yl)ethyl)cyclopropanamine hydrochloride N-Methyl-2'-methyl-2',3'-dihydrofuro[m]aporphine N-Methyl-2'-methyl-furo[m]aporphine N-Methyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride N-Methyl-2-(2'-amino-4'-ethylphenylthio)benzylamine N-Methyl-2-(2'-amino-4'-hydroxymethylphenylthio)benzylamine N-Methyl-2-(2'-nitrophenylthio)benzamide N-Methyl-2-(4'-methyl-2'-nitrophenylthio)benzamide N-Methyl-2-hydroxy-2'-methyl-2',3'-dihydrofuro[m]aporphine N-Methyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide N-methyl-6-(4-((phenethylamino)methyl)phenoxy)nicotinamide N-methyl-6-[4-(phenethylamino-methyl)-phenoxy]-nicotinamidine N-methyl-AMAA N-methyl-AMPA N-methyl-laudanosine N-Methyl-N'-(1,2,3,4-tetrahydro-acridin-9-yl)-N-[3-(1,2,3,4-tetrahydro-acridin-9-ylamino)-propyl]-propane-1,3-diamine N-Methyl-N'-(1,2,3,4-tetrahydroacridin-9-yl)-N-[3-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)propyl]-1,3-propanediamine N-Methyl-N'-(1,2,3,4-tetrahydroacridin-9-yl)-N-[4-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)butyl]-1,3-propanediamine N-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclobutanamine Hydrochloride N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclohexanamine Hydrochloride N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclopentanamine Hydrochloride N-methyl-N-(4-(3-((methylamino)methyl)-4-(4-(methylthio)phenoxy)phenyl)but-3-ynyl)cyclopropanamine N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide N-Methyl-N-phenethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide N-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isonicotinamide N-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]nicotinamide N-Methyl-N-{2-[3-(phenylsulfonyl)-1H-indol-4-yl]ethyl}amine N-methylazabicyclo[2.2.1]heptane N-methylcarbamoylcholine N-methylcarbamylcholine N-methylepibatidine N-methylhistamine N-Methylpiperidine N-methylpyridinium iodide N-methylpyrrolidine N-methylquipazine n-methylscopolamine N-morpholin-4-yl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-n-butylpyridinium iodide N-n-decylpyridinium iodide N-n-dodecylpyridinium iodide N-n-eicosylpyridinium iodide N-n-heptylpyridinium iodide N-n-hexylpyridinium iodide N-n-nonylpyridinium iodide N-n-octylpyridinium iodide N-n-pentadecylpyridinium iodide N-n-pentylpyridinium iodide N-n-propyl-1-(4-bromo-2,5-dimethoxyphenyl)-2-aminopropane HCI N-n-propyldihydrexidine, N-Pr-DHX N-n-propylpyridinium iodide N-n-undecylpyridinium iodide N-Nonyl-3-(3-Hydroxyphenyl)Pyrrolidine N-Octyl-3-(3-hydroxyphenyl)pyrrolidine N-oleoylethanolamine N-omega-MT N-pentanyl-5 methoxy tryptamine N-Pentyl-3-(3-hydroxyphenyl)pyrrolidine N-Phenethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide N-phenethyl-9-propyl-9H-purin-6-amine N-Phenethyl-S-methyl-dithiocarbamate N-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide N-Phenyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-Phenyl-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-phenyl-N-(1-(phenylcarbamoyl)cyclohexyl)-4-(1H-tetrazol-1-yl)benzamide N-phenylmethyl-3-[(phenylmethyl)amino]propanamide N-Phenylmethyl-3-[4-(phenylmethyl)-1-piperazinyl]propanamide N-piperidin-1-yl 1-(2,4,6-trichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(2,4,6-trichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(4-chlorophenyl)-3-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide N-piperidin-1-yl 1-(4-chlorophenyl)-4-cyano-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(4-chlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 1-(4-chlorophenyl)-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide N-piperidin-1-yl 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-piperidin-1-yl 4-cyano-1-phenyl-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide N-piperidin-1-yl 4-methyl-1-phenyl-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide N-Piperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide N-Piperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide N-piperidinyl-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide N-piperidinyl-[8-chloro-1-(2,4-dichlorophenyl)-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide] N-Propargyl-2-(5-methoxy-1H-indol-3-yl)acetamide N-Propargyl-3-(5-methoxy-1H-indol-3-yl)propanamide N-propionyl-5 methoxy tryptamine N-propionyl-5-MeOT N-Propyl-2',2'-bismethyl-2',3'-dihydrofuro[m]noraporphine N-Propyl-2',3'-bismethyl-2',3'-dihydrofuro[m]noraporphine N-Propyl-2',3'-bismethyl-furo[m]noraporphine N-Propyl-2'-methyl-2',3'-dihydrofuro[m]noraporphine N-Propyl-2'-methyl-furo[m]noraporphine N-Propyl-2-(4-hydroxyphenyl)-norapomorphine hydrochloride N-Propyl-2-methylnorapomorphine hydrochloride N-Propyl-2-phenylnorapomorphine hydrochloride N-Propyl-3a,9b-dihydro-3H-chromeno[4,3-c][1,2]oxazole-1(4H)-carboxamide N-propyl-dihydrexidine N-Propyl-N'-(1,3,4-trioxo-1,2,3,4-tetrahydro-isoquinolin-6-yl)-succinamide N-Propyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-propylapomorphine,(-) N-propylnorapomorphine N-propylnorapomorphine-(+) N-propylnorapomorphine-(-) N-Propylquipazine N-Pyrrolidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide N-tert-Butyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylaceta... N-tert-Butyl-2-[4-(9-pentyl-9H-carbazole-3-carbonyl)piperazin-1- yl]acetamide N-tert-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide N-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide N-[(1R)-3-[(2R)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]-3-oxo-1-phenylpropyl]acetamide N-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-cyclohexylcarbamoyl-2-hydroxypropyl]-2,4,6-trifluorobenzamide N-[(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-cyclohexylcarbamoyl-2-hydroxy-propyl]-2,4,6-trifluoro-benzamide N-[(1S,2S)-3-Cyclohexylcarbamoyl-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl]-2,4,6-trifluoro-benzamide N-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-p... N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](2-naphthyl)amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](3-phenylpropyl)amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]benzylamine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(1-naphthyl)ethyl]amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(2,4-dichlorophenyl)ethyl]amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(3,4-dichlorophenyl)ethyl]amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-bromophenyl)ethyl]amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-chlorophenyl)ethyl]amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-methoxyphenyl)ethyl]amine N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-nitrophenyl)ethyl]amine N-[(2-Chloro-6flurophenyl)methyl]-7methoxy-N-(1-methylethyl)-1-[2-(4-morpholinyl)ethyl]-1H-indazol-3-carboxamide N-[(2-cyclopentyl-1,3-thiazol-4-yl)methyl]-N-ethyl-2-pyridin-2-ylethanamine N-[(2-Naphthyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea N-[(2-Triphenylmethyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-5-phenyl-1H-pyrazole-4-carboxamide N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-... N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-... N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-... N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-... N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-... N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-... N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl... N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl... N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-... N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-... N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-... N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-... N-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide N-[(3R)-1-Benzyl-3-pyrrolidinyl]-3-(3-thienyl)benzamide N-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(2-thienyl)benzamide N-[(3R)-1-Benzyl-3-pyrrolidinyl]-4-(3-thienyl)benzamide N-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(2-thienyl)benzamide N-[(3S)-1-Benzyl-3-pyrrolidinyl]-3-(3-thienyl)benzamide N-[(3S)-1-Benzyl-3-pyrrolidinyl]-4-(3-thienyl)benzamide N-[(3S)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide N-[(3S)-1-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide N-[(4-Chlorophenyl)-DL-a-methyltryptophanyl][(2phenylethyl)amino]urea N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide N-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide N-[(4-Phenyl-1-piperazinyl)-propyl-3-(4-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride N-[(4-Phenyl-1-piperazinyl)-propyl]-3,3- diphenyl-pyrrolidine-2,5-dione dihydrochloride N-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride N-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-chlorophenyl)-pyrrolidine-2,5-dione dihydrochloride N-[(4-Phenyl-1-piperazinyl)-propyl]-3-(4-fluorophenyl)-pyrrolidine-2,5-dione dihydrochloride N-[(4-Phenyl-1-piperazinyl)-propyl]-3-phenylpyrrolidine-2,5-dione dihydrochloride N-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-4-oxo-1H-quinoline-3-carboxamide N-[(Indol-3-yl)methyl]propanethioamide N-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide N-[(Naphth-2-yl)methyl]-S-methyl-dithiocarbamate N-[1-(1-Phenyl)ethyl]1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[1-(2-Diethylaminoethyl)-1H-indol-5-yl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-[1-(2-Diethylaminoethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide N-[1-(2-Diethylaminoethyl)-1H-indol-5-yl]naphthalene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-4-yl]naphthalene-1-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-4-yl]naphthalene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-5-yl]-1-phenylmethanesulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-5-yl]-4-phenylbenzenesulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-5-yl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-5-yl]naphthalene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-6-yl]-2-(naphthalen-1-yl)-ethanesulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-6-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-6-yl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-6-yl]naphthalene-1-sulfonamide N-[1-(2-Dimethylaminoethyl)-1H-indol-6-yl]naphthalene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-2-methyl-1H-indol-4-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-2-methyl-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[1-(2-Dimethylaminoethyl)-2-methyl-1H-indol-5-yl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-[1-(2-Dimethylaminoethyl)-2-methyl-1H-indol-5-yl]naphthalene-1-sulfonamide N-[1-(2-Dimethylaminoethyl)-2-methyl-1H-indol-5-yl]naphthalene-2-sulfonamide N-[1-(2-Phenoxyethyl)piperidin-4-yl]thiophene-2-sulfonamide N-[1-(2-pyridin-2-ylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)acetamide N-[1-(Indol-3-yl)ethyl]-N'-methyl-thiourea N-[10-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)decyl]-3-(1H-indol-3-yl)propionamide N-[2-(1,3-dihydroisoindol-2-yl)ethyl]-3-(methoxymethyl)benzamide N-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(3,4-Dimethoxyphenyl)ethyl]-2,3-dihydro-5,6-dimethoxy-N-propyl-1H-inden-2-amine N-[2-(3-(2-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Acetylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Aminomethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Aminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Bromomethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Dimethylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Ethoxycarbonylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Formylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl] acetamide N-[2-(3-(3-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]butyramide N-[2-(3-(3-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]cyclobutyl carboxamide N-[2-(3-(3-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]propionamide N-[2-(3-(3-Iodomethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Methoxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(3-Methylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-(4-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide N-[2-(3-Aminophenyl)ethyl]-2,3-dihydro-5,6-dimethoxy-N-propyl-1H-inden-2-amine N-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamid... N-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamid... N-[2-(3-fluorophenyl)ethyl]-2,3-dihydro-5,6-dimethoxy-N-propyl-1H-inden-2-amine N-[2-(3-phenyl-7-methoxynaphth-1-yl)ethyl] acetamide N-[2-(4-Bromophenyl)ethyl]-2,3-dihydro-5,6-dimethoxy-N-propyl-1H-inden-2-amine N-[2-(4-Chlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(4-Chlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(4-Chlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(4-Chlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(4-Chlorophenyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide N-[2-(4-Chlorophenyl)ethyl]1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide N-[2-(4-Phenyl-1,2,3,6-tetrahydropyridin-1-yl) ethyl]-2-quinoline Carboxamide N-[2-(4-Phenyl-1,2,3,6-tetrahydropyridin-1-yl) ethyl]-3-quinoline Carboxamide N-[2-(4-Phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-2-quinoxaline Carboxamide N-[2-(4-Phenylpiperazin-1-yl)ethyl]-2-quinoline Carboxamide N-[2-(4-Phenylpiperazin-1-yl)ethyl]-2-quinoxaline Carboxamide N-[2-(4-Phenylpiperazin-1-yl)ethyl]-3-methoxybenzamide N-[2-(4-Phenylpiperazin-1-yl)ethyl]-3-quinoline Carboxamide N-[2-(Benzo[b]thiophen-3-yl)ethyl]-S-methyl-dithiocarbamate N-[2-(Indol-3-yl)ethyl]-S-benzyl-dithiocarbamate N-[2-(Indol-3-yl)ethyl]-S-methyl-dithiocarbamate N-[2-(Indol-3-yl)ethyl]-S-[(naphth-2-yl)methyl]dithiocarbamate N-[2-(Indol-3-yl)ethyl]-S-[(pyrid-3-yl)methyl]dithiocarbamate N-[2-(Indol-3-yl)ethyl]-S-[(pyrid-4-yl)methyl]dithiocarbamate N-[2-[(2-hydroxycyclohexyl)amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamic Acid Tricyclo[3.3.1.1]dec-2-yl Ester N-[2-[4-(1-Naphthalenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl]pyrazolo[1,5-a]pyridine-2-carboxamide N-[2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl]pyrazolo[1,5-a]pyridine-3-carboxamide N-[2-[4-(2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(4-Chloro-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(4-Methyl-2-pyridinyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-[4-(4-Methylphenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide N-[2-{4-(2-Methoxyphenyl)-piperazin-1-yl}-ethyl]-3-cyclohexyl-pyrrolidine-2,5-dione N-[2-{4-(2-Methoxyphenyl)-piperazin-1-yl}-ethyl]-pyrrolidine-2,5-dione N-[2-{4-(3-Chlorophenyl)-piperazin-1-yl}-ethyl]-3-cyclohexyl-pyrrolidine-2,5-dione N-[2-{4-(3-Chlorophenyl)-piperazin-1-yl}-ethyl]-pyrrolidine-2,5-dione N-[3-(1,2,3,4-Tetrahydroacridin-9-ylamino)propyl]-N'-[3-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)propyl]acetamide N-[3-(1,2,3,4-Tetrahydroacridin-9-ylamino)propyl]-N'-[4-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)butyl]acetamide N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]-4-phenylbenzenesulfonamide N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]-5-chlorothiophene-1-sulfonamide N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]-5-chlorothiophene-2-sulfonamide N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]naphthalene-1-sulfonamide Hydrochloride N-[3-(1-Methylpiperidin-4-yl)-1H-indol-5-yl]quinolyl-2-sulfonamide N-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide N-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide N-[3-(2-Dibutylaminoethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide N-[3-(2-Diethylaminoethyl)-1-methyl-1H-indol-5-yl]naphthalene-2-sulfonamide N-[3-(2-Diethylaminoethyl)-1H-indol-5-yl]-3,5-dichlorobenzenesulfonamide N-[3-(2-Diethylaminoethyl)-1H-indol-5-yl]-4-phenylbenzenesulfonamide N-[3-(2-Diethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[3-(2-Diethylaminoethyl)-1H-indol-5-yl]-5-chloronaphthalene-1-sulfonamide N-[3-(2-Diethylaminoethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide N-[3-(2-Diethylaminoethyl)-1H-indol-5-yl]naphthalene-2-sulfonamide N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-4-phenylbenzenesulfonamide N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-5-chloronaphthalene-2-sulfonamide N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-[3-(2-Dimethylaminoethyl)-1H-indol-5-yl]naphthalene-1-sulfonamide N-[3-(2-Dipropylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[3-(2-Dipropylaminoethyl)-1H-indol-5-yl]naphthalene-2-sulfonamide N-[3-(3-Diethylaminopropyl)-1H-indol-5-yl]naphthalene-2-sulfonamide N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-1H-quinoline-2-carboxamide N-[3-(Acridin-9-ylsulfanyl)-propyl]-N''-(1,2,3,4-tetrahydro-acridin-9-yl)-pentane-1,5-diamine N-[3-(Indol-3-yl)propyl]-S-methyl-dithiocarbamate N-[3-Dimethylaminomethyl-1H-indol-5-yl]-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-[3-[(2-Methyl-4-thiazolyl)ethynyl]phenyl]acetamide N-[3-[4-(2,3-Dichlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide N-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-3-methoxybenzamide N-[3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl]pyrazolo[1,5-a]pyridine-2-carboxamide N-[3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl]pyrazolo[1,5-a]pyridine-3-carboxamide N-[3-[4-(4-Chlorophenyl)piperazin-1-yl]propyl]-3-methoxybenzamide N-[4-(1,2,3,4-Tetrahydro-5-methoxy--carbolin-2-yl)butyl]isoquinoline-3-carboxamide N-[4-(1,2,3,4-Tetrahydroacridin-9-ylamino)butyl]-2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-1H-imidazole-4-carboxamide N-[4-(1H-Tetrazol-5-yl)butyl]-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide N-[4-(2-Ethyl-4-phenyl-1,3-thiazol-5-yl)-2-pyridyl]benzamide N-[4-(3,4-Dihydro-6-methoxypyrazino[1,2-a]1ndol-2(1H)-yl)-butyl]isoquinoline-3-carboxamide N-[4-(3-Pyridylethynyl)-2-thiazolyl]acetamide N-[4-(3-Pyridylethynyl)-2-thiazolyl]benzamide N-[4-(4-Amino-6-benzylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-cyclohexylurea N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea N-[4-(4-Amino-6-isopropylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-1H-indole-2-carboxamide N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-2-(3-methylphenyl)acetamide N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-3-methylbenzamide N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N' '-cyano-N'-(3-methylphenyl)guanidine N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-chlorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-fluoro-5-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-fluorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-methoxyphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3,5-dichlorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3,5-dimethylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-bromophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-chlorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-fluorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methoxyphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)thiourea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-bromophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-chlorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-fluorophenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-methoxyphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-benzylurea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-cyclohexylmethylurea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-methyl-N'-(3-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-phenylurea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[2-fluoro-5-(trifluoromethyl)phenyl]urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[4-(trifluoromethyl)phenyl]urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N-methyl-N'-(3-methylphenyl)urea N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]benzenesulfonamide N-[4-(4-Amino-6-propylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-chlorophenyl]-N'-(3-methylphenyl)urea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-fluorophenyl]-N'-(3-methylphenyl)urea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-methoxyphenyl]-N'-(3-methylphenyl)urea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-chlorophenyl)urea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-butylurea N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-isobutylurea N-[4-(4-methylpiperazin-1-yl)butyl]imidazo[1,2-a]pyridine-2-carboxamide N-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine N-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-4-(2-methoxyphenyl)-1-piperazinecarboxamide N-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-4-[4-(trifluoromethyl)phenyl]-1-piperazinecarboxamide N-[4-[(2-amino-6-ethyl-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidin-5-yl)thio]benzoyl]-L-glutamic acid N-[4-[2-Ethyl-4-(2-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Ethyl-4-(3-methoxyphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-2-phenylacetamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-3-phenylpropionamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(2-phenylethyl)amine N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(3-phenylpropyl)amine N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-methylbenzamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]acetamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]butyramide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]cyclohexanecarboxamide N-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]propionamide N-[4-[2-Ethyl-4-(4-fluorophenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Ethyl-4-(4-methoxyphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Ethyl-4-(4-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Ethyl-4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[2-Methyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[3-(2-Methoxyphenyl)piperazin-1-yl]propyl]-2,1,3-benzoxadiazole-5-carboxamide N-[4-[3-(3-Methoxyphenyl)piperazin-1-yl]propyl]-4-(1Himidazol-1-yl)benzamide N-[4-[4-(1,2-Benzisoxazol-3-yl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(1-Isoquinolyl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(1-Naphthalenyl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-(1,1'-biphenyl)-4-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-methoxy-2-naphthalenecarboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indazole-3-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indole-2-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1H-indole-3-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-benzofurancarboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-benzofurancarboxamide36 N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-2-naphthalenecarboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-bromo-1-methoxy-2-naphthalenecarboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-4-quinolinecarboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-7-methoxy-2-benzofurancarboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]tellurophene-2-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide N-[4-[4-(2,3-Dimethylphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(2,4-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one N-[4-[4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl]butyl]-2,1,3-benzoxadiazole-5-carboxamide N-[4-[4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl]butyl]-4-(1H-imidazol-1-yl)benzamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]benzo[b]tellurophen-2-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]benzo[b]thiophene-2-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-3-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-4-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-5-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-7-carboxamide N-[4-[4-(2-Methoxyphenyl)piperazin]1-yl]butyl]pyrazolo[1,5-a]pyridine-6-carboxamide N-[4-[4-(3-(2-Fluoroethoxy)phenyl)piperazin-1-yl]butyl]-2,1,3-benzoxadiazole-5-carboxamide N-[4-[4-(3-(2-Fluoroethoxy)phenyl)piperazin-1-yl]butyl]-4-(1H-imidazol-1-yl)benzamide N-[4-[4-(3-Chlorophenyl)-2-ethyl-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[4-(3-Chlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide N-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one N-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide N-[4-[4-(3-Fluoro-5-methoxyphenyl)piperazin-1-yl]butyl]-2,1,3-benzoxadiazole-5-carboxamide N-[4-[4-(3-Fluoro-5-methoxyphenyl)piperazin-1-yl]butyl]-4-(1H-imidazol-1-yl)benzamide N-[4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl]-2,1,3-benzoxadiazole-5-carboxamide N-[4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl]-4-(1Himidazol-1-yl)benzamide N-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-2-phenylacetamide N-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(2-phenylethyl)amine N-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[4-(3-Methylphenyl)-2-propyl-1,3-thiazol-5-yl]-2-pyridyl]benzamide N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine N-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine N-[4-[4-(4-Chlorophenyl)piperazin-1-yl]butyl]-3-methoxybenzamide N-[4-[4-(4-Methoxyphenyl)piperazin-1-yl]butyl]-2,1,3-benzoxadiazole-5-carboxamide N-[4-[4-(4-Methoxyphenyl)piperazin-1-yl]butyl]-4-(1Himidazol-1-yl)benzamide N-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide N-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide N-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide N-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide N-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide N-[5-(4-Amino-6-dimethylamino-[1,3,5]triazin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)propionamide N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-3-(1H-indol-3-yl)propionamide N-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-4-(1H-indol-3-yl)butyramide N-[5-pyridin-4-yl-4-(3,4,5-trimethoxyphenyl)thiazol-2-yl]acetamide N-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide N-[5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide N-[5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl]pyrazolo[1,5-a]pyridine-2-carboxamide N-[5-[4-(2-Methoxyphenyl)piperazin-1-yl]pentyl]pyrazolo[1,5-a]pyridine-3-carboxamide N-[5-[4-(4-Chlorophenyl)piperazin-1-yl]pentyl]-3-methoxybenzamide N-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)acrylamide N-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(5-cyano-1H-indol-3-yl)propionamide N-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-4-(1H-indol-3-yl)butyramide N-[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl]-2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-1H-imidazole-4-carboxamide N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-2-(1H-indol-3-yl)acetamide N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide N-[7-[(1S)-1-(3-methoxyphenoxy)ethyl]-1H-[1,2,4]triazolo[1,5-a]pyrimidin-8-ium-2-yl]-N,N-dimethylmethanimidamide N-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(2-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide N-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(3-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide N-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide N-[8-(4-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide N-[8-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)octyl]-3-(1H-indol-3-yl)propionamide N-[9-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)nonyl]-3-(1H-indol-3-yl)propionamide N-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide N-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide N-[N'-Propyl-N'-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide N-[N-[(2-Adamantyloxy)carbonyl]-D-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine N-[N-[(2-Adamantyloxy)carbonyl]-D-tryptophanyl]-N-(2-phenylethyl)glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(1-naphthyl)alaninyl]-N-(2-phenylethyl)glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(2-naphthyl)alaninyl]-N-(2-phenylethyl)glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(4-bromophenyl)alaninyl]-N-(2-phenylethyl)glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methylphenyl-alaninyl]-N-(2-phenylethyl)glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-2-phenylethylamine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)-3-aminopropionic Acid N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(2,4-dichlorophenyl)ethyl]glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]aniline N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]glycine N-[N-[(2-Adamantyloxy)carbonyl]-L-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine N-[[1-(2-Cyclohexylethyl)-4-piperidinyl]methyl]-1-isopropyl-1Hindazole-3-carboxamide N-[[1-(2-Phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide N-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide N-[[1-[3-(Dimethylamino)propyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide N-[[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-1-[(2S)-2,3-dihydro-1-benzofuran-2-yl]-N-methylmethanamine N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide N-[[[[4-(1,3-Dipropyl-8-xanthinyl)phenyl]oxy]methyl]-carbonyl]-N,N'-dicyclohexylurea N-{(1S,2S)-1-(4-Benzo[1,3]dioxol-5-yl-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-h... N-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-2-hydroxy-3-[2-(3-methoxyphenyl)ethylcarbamoyl]propyl}-2,4,6-tri-fluorobenzamide N-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethylcarbamoyl]-2-hydroxypropyl}-2,4,6... N-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethylcarbamoyl]-2-hydroxypropyl}-3,4-d... N-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-2-hydroxy-3-[2-(3-methoxy-phenyl)-ethylcarbamoyl]-propyl}-2,4,6-trifluoro-benzamide N-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propyl... N-{(1S,2S)-2-Hydroxy-3-[2-(3-methoxy-phenyl)-ethylcarbamoyl]-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl}-2,4,6-trifluoro-benz... N-{1-[2-(2-Isopropoxyphenoxy)ethyl]piperidin-4-yl} quinoline-8-sulfonamide N-{1-[2-(2-Isopropoxyphenoxy)ethyl]pyrrolidin-3-yl} isoquinoline-4-sulfonamide N-{1-[2-(2-Methoxyphenoxy)ethyl]piperidin-4-yl}isoquinoline-4-sulfonamide N-{1-[2-(3-Fluorophenoxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide N-{1-[2-(5,6,7,8-Tetrahydronaphthalen-1-yloxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide N-{1-[2-(Biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}quinoline-2-carboxamide N-{1-[2-(Biphenyl-2-yloxy)ethyl]pyrrolidin-3-yl}thiophene-2-sulfonamide N-{1-[2-(Piperidin-1-yl)ethyl]-1H-indol-5-yl}-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-{1-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-5-yl}-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-{1-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-6-yl}-2-(naphthalen-1-yl)-ethanesulfonamide N-{1-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-6-yl}-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-{1-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-6-yl}-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-{1-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-6-yl}naphthalene-1-sulfonamide N-{1-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-6-yl}naphthalene-2-sulfonamide N-{1-[3-(Piperidin-1-yl)propyl]-1H-indol-5-yl}-6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2,4-difluorobenzamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2,4-difluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-phenylpropanamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3,3-trifluoropropane-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3-dimethylbutanamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}cyclohexanesulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pentylsulfonamide N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pyridin-2-amine N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}tetrahydro-2H-thiopyran-4-carboxamide N-{1-[8-(2-Chlorophenyl)-9-(4-fluorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-(5-methyl-1,2-oxazol-3-yl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamid N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}benzamide N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide N-{2-[(4-methoxypyrimidin-2-yl)(methyl)amino]ethyl}acetamide N-{2-[3-(Phenylsulfonyl)-1H-indol-4-yl]ethyl}-N-propylamine N-{2-[3-(Phenylsulfonyl)-1H-indol-4-yl]ethyl}cyclopentanamine N-{2-[3-(Phenylsulfonyl)-1H-indol-4-yl]ethyl}propan-2-amine N-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(2-Methylphenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(2-Methylphenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(2-Methylphenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(3-Methoxyphenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(3-Methoxyphenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(3-Methoxyphenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(3-Methylphenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(3-Methylphenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(3-Methylphenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(3-Trifluoromethylphenyl)piperazin-1-yl] ethyl}-2-quinoline Carboxamide N-{2-[4-(3-Trifluoromethylphenyl)piperazin-1-yl] ethyl}-3-quinoline Carboxamide N-{2-[4-(3-Trifluoromethylphenyl)piperazin-1-yl]ethyl}-2-quinoxaline Carboxamide N-{2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{2-[4-(4-Methylphenyl)piperazin-1-yl]ethyl}- 2-quinoline Carboxamide N-{2-[4-(4-Methylphenyl)piperazin-1-yl]ethyl}- 2-quinoxaline Carboxamide N-{2-[4-(4-Methylphenyl)piperazin-1-yl]ethyl}- 3-quinoline Carboxamide N-{3-[2-(Morpholin-4-yl)ethyl]-1H-indol-5-yl}-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-{3-[2-(Morpholin-4-yl)ethyl]-1H-indol-5-yl}naphthalene-1-sulfonamide N-{3-[2-(Morpholin-4-yl)ethyl]-1H-indol-5-yl}naphthalene-2-sulfonamide N-{3-[2-(Morpholin-4-yl)ethyl]-1H-indol-5-yl}quinolyl-8-sulfonamide N-{3-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-5-yl}-5-chloro-3-methyl-benzo[b]thiophene-2-sulfonamide N-{3-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-5-yl}naphthalene-1-sulfonamide N-{3-[2-(Pyrrolidin-1-yl)ethyl]-1H-indol-5-yl}naphthalene-2-sulfonamide N-{4-[(1,2,3, 4-Tetrahydroacridin-9-yl)amino]butyl}-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)sulfanyl]propyl}acetamide N-{4-[(1,2,3,4-Tetrahydroacridin-9-yl)amino]butyl}-N{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}acetamide N-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-2-fluoro-phenyl}-methanesulfonamide N-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-2-methoxy-phenyl}-methanesulfonamide N-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-phenyl}-methanesulfonamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-chlorobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-fluorobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-hydroxy-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-iodobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-methoxy-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-nitrobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-chlorobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-fluorobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-iodobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-methoxy-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-nitrobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-(1H-imidazol-2-yl)-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-chlorobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-fluorobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-hydroxy-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-iodobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-methoxy-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-nitrobenzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-4-yl-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyrimidin-2-yl-benzamide N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-nicotinamide N-{4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl}(9-oxofluoren-4-yl)carboxamide N-{4-[4-Amino-6-(2-hydroxyethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea N-{4-[4-Amino-6-(2-methoxyethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea N-{4-[4-Amino-6-(3-hydroxypropyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea N-{4-[4-Amino-6-(morpholin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea N-{4-[4-Amino-6-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea N-{4-[4-Amino-6-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea N-{[(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0... N-{[1-(2-(2-Isopropoxyphenoxy)ethyl)piperidin-4-yl] methyl}quinoline-8-sulfonamide N-{[1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl] methyl}isoquinoline-4-sulfonamide N-{[1-(2-methylpyrimidin-4-yl)piperidin-2-yl]methyl}acetamide N1,N1-diethyl-N4-(2-methoxy-9-acridinyl)-1,4-pentanediamine N1,N10-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)decanediamide N1,N11-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)undecanediamide N1,N13-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tridecanediamide N1,N14-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tetradecanediamide N1,N15-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)pentadecanediamide N1,N16-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)hexadecanediamide N1,N3-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)malonamide N1,N5-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)glutaramide N1,N8-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)octanediamide N1-(2-Cyclohexylidene-2-fluoroethyl)-N3,N3-dimethyl-1,3-propanediamine N1-(2-Cyclopentylidene-2-fluoroethyl)-N3,N3-dimethyl-1,3-propanediamine N1-(benzo[d]thiazol-2-yl)-N4-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine N1-(benzo[d]thiazol-2-ylmethyl)-N4-(3-ethoxy-4-methoxyphenyl)cyclohexane-1,4-diamine N1-dansyl-spermidine N1-DnsSpm N1-ethyl-N1-Ant-CH2 (3,3) N1-ethyl-N1-Ant-CH2 (4,4) N1-n-octanesulfonyl-spermine N1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt N1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine N2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine N2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine N2 -benzyl-9-propyl-9H-purine-2,6-diamine N2 -phenethyl-9-propyl-9H-purine-2,6-diamine N2-(3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide hydrobromide N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamide N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamine N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide Hydrobromide N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-L-lysine-2-phenethylamide N2-[3,5-Dibromo-N-(4-phenyl-1-oxybutyl)-L-tyrosyl]-L-lysine-2-phenethylamide N2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysine-2-phenethylamide N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysine-phenylamide Hydrobromide N2-[4-Amino-3,5-dibromo-N-(3-phenyl-1-oxopropyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrochloride N2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide N3-(1-(3,5-Dimethyl)adamantyl)-4-oxo-1-benzyl-1,4-dihydroquinoline-3-carboxamide N3-(1-(3,5-Dimethyl)adamantyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(1-adamantyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(1-Naphthyl)-1-butyl-4-oxo-1,4-dihydroquinoline-3-carboxamide N3-(1-Naphthyl)-1-hexyl-4-oxo-1,4-dihydroquinoline-3-carboxamide N3-(1-Naphthyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(2-(Benzo[1,3]dioxol-5-yl)ethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(2-Adamantyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(3,4-Dichlorophenyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(3-Phenylpropyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(4-Cyanophenyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(Benzyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N3-(Phenethyl)-4-oxo-1-pentyl-1,4-dihydroquinoline-3-carboxamide N4-benzyl-1-(2-chloro-2-phenylethyl)-N6,N6-dimethyl-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine N4-Deazaquipazine N6 - 2 - (4 - aminophenyl)ethyladenosine N6 -(4-Chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine N6 -(4-Chloro-2-fluorophenyl)amino-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine N6 -(±)-endo-Norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine N6 -(R)-3-Tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1- yl)-5-deoxy-β-D-ribofuranosyl)adenine N6 -Cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β- D-ribofuranosyl)adenine N6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide N6-( 3-Aminobenzyl)adenosine-5-N-methyluronamide N6-( 3-Aminobenzyl)adenosine-N-methyluronamide N6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt N6-( 4-Sulfobenzyl)adenosine-5-N-methyluronamide N6-(2-endo-norbornyl)-adenosine N6-(2-Hydroxyethyl)ado N6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide N6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide N6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide N6-(3-Hydroxypropyl)ado N6-(3-Iodobenzyl)-adenosine N6-(3-iodobenzyl)-adenosine-5'-N-methyluronamide N6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide N6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide N6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide N6-(R)-3-Tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine N6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide N6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide N6-1-phenyl-2(R)-propyl-2-chloro-9-methyladenines N6-1-phenyl-2(R)-propyl-9-Methyladenines N6-1-phenyl-2(R)-propyl-9-phenyladenines N6-1-phenyl-2(S)-propyl-2-chloro-9-methyladenines N6-1-phenyl-2(S)-propyl-9-Methyladenines N6-1-phenyl-2(S)-propyl-9-phenyladenines N6-2-(4-aminophenyl)ethyl-adenosine N6-Benzyl-N6-methyladenosine N6-Benzyladenosine-5-N-cyclopropyluronamide N6-Benzyladenosine-N1-oxide N6-benzylado N6-BenzylNECA N6-c-C6H11-9-Ethyladenines N6-c-C6H11-9-Methyladenines N6-cyclohexyl adenosine N6-Cyclohexylado (CHA) N6-CyclohexylNECA N6-Cyclopentyl-2-Chloro-9-methyladenines N6-Cyclopentyl-2-chloroAdo N6-Cyclopentyl-5'chloroAdo N6-cyclopentyl-9-(2-Hydroxyethyl)adenines N6-Cyclopentyl-9-Cyclopentyladenines N6-cyclopentyl-9-ethyladenines N6-Cyclopentyl-9-Methyladenines N6-cyclopentyl-9-phenyladenines N6-cyclopentyladenosine N6-CyclopentylAdo N6-Cyclopentylado (CPA) N6-Cylcopentyl-9-(2-Tetrahydrofuryl)adenines N6-Methylado N6-phenyl-2-chloro-9-methyladenines N6-phenyl-9-Methyladenines N6-Phenyl-9-Phenyladenines N6-phenyladenosine N6-Phenylado N6-[(R)-1-Methyl-2-phenylethyl]ado (R-PIA) N6-[(S)-1-Methyl-2-phenylethyl]ado (S-PIA) N6-[3-(4-Chlorophenyl)bicyclo[2.2.2]oct-2-yl]ado (EMD 28422) NAAG Nabilone Nabumetone NAD-299 NAE-086 NAE-111 NAEPA naftopidil Nal1-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly Nal2-Tyr-Thr-Pro-Lys-Thr(OBzl)-Gly Nalbuphine NALBzoH Nalfurafine nalmefene Nalmefene NALMEFENE-HCl Nalmetrene Nalorphine NALORPHINE - HCI Naloxonazine NALOXONE Naloxone(+) Naloxone(-) Naltrexone Naltrexone methiodide Naltrexone-6-alpha-ol Naltrexone-6-beta-ol NALTREXONE-HCl NALTRINDOLE Naltrindole CNG Naltrindole G NAMH NAN-190 Nantenin nantentine Napamezole Naphazoline naphazoline Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073) Naphthalen-2-yl(4-(3-Phenylpropylamino)piperidin-1-yl)methadone Naphthalen-2-yl(4-(Phenylamino)piperidin-1-yl)methadone Naphthalene Naphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-(2-cyclohexyl-ethyl)-amino]-ethyl}-cy... Naphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-(3-methyl-butyl)-amino]-ethyl}-cycloh... Naphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-butyl-amino]-ethyl}-cyclohexyl)-amide Naphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-propyl-amino]-ethyl}-cyclohexyl)-amid... Naphthalene-2-carboxylic acid {4-[2-((R)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-cyclohexyl}-am... Naphthalene-2-carboxylic acid {4-[2-((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-ylamino)-ethyl]-cyclohexyl}-amide Naphthalene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide Naphyrone Naproxen Naproxen sodium,(-) Naratriptan naringenin NAS native GnRH N‐[2‐(diethylamino)ethyl]‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐2‐methyl‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐3‐fluoro‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐3‐methoxy‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐3‐methyl‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐4‐methoxy‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)‐4‐(trifluoromethyl)aniline N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine N‐[3‐(dimethylamino)propyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline N‐[3‐(dimethylamino)propyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline N‐[3‐(dimethylamino)propyl]‐N‐(2‐phenylethyl)aniline NB-Benzyladenosine-5-N-methyluronamide NBEP NBI 27914 NBI 35965 NBI-42902 NBI-55886 NBI-56297 NBI-56453 NBI-58702 NBI-58704 NBI-74330 NBQX NC4-28B NC8-12 NCS-382 NDMNEP NDP-MSH Nebivolol NECA NECA (5'-(N-ethylcarboxamido)adenosine) NECA, 2-heptynyl NECA, 2-hexynyl NECA, 2-octynyl NECA-N1-oxide NECI Nefazodone Nefopam Nelfinavir mesylate NEMONAPRIDE Neo-Delta-Cortef Neomenthol-(+) Neomenthol-(-) Neomycin NEP Nepinalone NEUROKININ A Neurokinin alpha NEUROKININ B Neuromedin B Neuromedin C neuromedin K Neuromedin N Neuropeptide Y Neuropeptide Y, Human Neuropeptide Y, human, rat Neuropeptide Y, porcine Neurotensin Neurotensin 2 Nevirapine NF023 NF279 NFEP NGB 2904 NGB2904 NGD 94-1 Nic-Tyr-Lys(Z-Arg)-His-Pro-Ile NICERGOLINE Nicotine Nicotine Free Janty EC Liquid Nicotine Free NicVape EC Liquid Nicotine-(+) nicotine-(-) nicotine-(S) Nicotine-D salicylate Nicotine-L (base) Nicotine-L salicylate NicVape EC Liquid NIFEDIPINE Niflumic acid Niguldipine(+) nimesulide Nimodipine NIPBF,NM Nipecotic NIPT,4-OH-NM NIPT,5,6-DiMeO-NM NIPT,5-Me-NM NIPT,5-MeO-NM NIPT,5MeO NIPT,6-MeO-NM NIPT,NM Nisoldipine Nisoxetine Nisoxetine Inhibitor Nitrazepam NITRENDIPINE NKA NKB NKB [MePhe7] Nle8,18,Tyr34-bPTH(1-34) Nle8,18,Tyr34-bPTH(3-34) NleYI-6-hexamide NLX-101 NMB NMCC NMDA NMS NMS,(-) NN-DIPROP-5-CT NNC 11-1314 NNC 11-1585 NNC 11-1607 NNC 26-9100 NNC-112 NNC-112,(-) NNC-687 NNC-756 NNEP Nociceptin Nociceptin-CONH2, [Aib11] Nociceptin-CONH2, [Aib15] Nociceptin-CONH2, [Aib7,Aib11] Nociceptin-CONH2, [Aib7] Nociceptin-CONH2, [MeAla11] Nociceptin-CONH2, [MeAla7] Nociceptin-CONH2,[MeAla15] Nociceptin-COOH, [Aib11] Nociceptin-COOH, [Aib15] Nociceptin-COOH, [Aib7] Nociceptin-COOH, [MeAla11] Nociceptin-COOH, [MeAla15] Nociceptin-COOH, [MeAla7] Nociceptin/Orphanin FQ NOHEP Noladin Ether, NE NOMIFENSINE Nor-binaltorphimine Nor-BNI NOR-BNI (HCI)2 Nor-d-fenfluramine nor-nicotine (+/-) Noradrenaline Noradrenaline,(+) NORADRENALINE,(-) Norbinaltorphimine norbinaltorphimine Norchloro-epibatidine Norclozapine Norephedrine, (+) Norephedrine, (-) NOREPINEPHRINE Norepinephrine,(+) Norfenfluramine Norfenfluramine (+) Norfenfluramine (+/-) Norfenfluramine (-) NORFLUOXETINE noribogaine Normorphine NORMORPHINE-HClO4 Normorphinone, N-allyl-dihydro-14-hydroxy- nornicotine northiaden Nortiptyline nortriptyline NORTRYPTYLINE NORTRYPTYLINE Norzimelidine NPA NPA+ (GTP+) NPA,(+) NPA,(-) NPA-11-OH-R,(+) NPA-11-OH-R,(-) NPFF NPFF-OH Nphe NPS 2390 NPSF NPY NPY 13-36 NPY 13-36, human NPY 13-36, human, rat NPY 18-36 NPY 28-36, [P30, Y32, L34] NPY 3-36, human NPY 3-36, porcine NPY D-Trp32 NPY D-Trp32, human NPY D-Trp32, human, rat NPY D-Trp32, porcine NPY Leu31, Pro34, human NPY Leu31, Pro34, human, rat NPY mod28-36, porcine NPY [Ala31, Aib32], porcine NPY [hPP(1-17), Ala31,Aib32], human NPY [Leu31, Pro34], human NPY, C2 NPY, C2, porcine NPY, free acid, human NPY, human NPY, human, rat NPY, LP, porcine NPY, porcine NPY, zebrafish NPY,[Leu31,Pro34] NPY,[leu31,Pro34], porcine NPY13-36 NPY13-36, porcine NPY16-36, porcine NPY18-36 NPY18-36, porcine NPY2-36 NPY2-36, human NPY2-36, porcine NPY2-36, rat, human NPY20-36, porcine NPY22-36, porcine NPY22-36, rat, human NPY26-36, porcine NPY3-36 NPY5-24, Ahx NPY8-20, Ahx NPY8-20, Pro34, Ahx NS-2710 NS102 NS1209 NS257 NS3763 NS3768 NS398 NT(1-13) NT(8-13) NTB NTEP Numorphan O-1986 O-1987 O-1988 O-2093 O-2094 O-2095 O-2109 O-2142 O-2154 O-2155 O-4331 O-4332 O-4333 O-4334 O-4335 O-4336 O-4337 O-4338 O-4339 O-4371 O-4372 O-4373 O-4423 O-4424 O-610 O-6211 O-6212 O-6213 O-6214 O-6215 O-6617 O-6618 O-6629 O-6658 O-6659 O-6668 O-6729 O-6730 O-6731 O-6740 O-680 O-687 O-689 O-Demethyl-18-deoxysalvinorin A O-desmethyl tramadol O-Desmethylvenlafaxine O-METHYLBUFOTENINE O2-(Acetylsalicyloyloxymethyl)-1-(N,N-dimethylamino)diazen-1-ium-1,2-diolate O2-(Acetylsalicyloyloxymethyl)-1-(pyrrolidin-1-yl)diazen-1-ium-1,2-diolate O2-[2-(1-(4-Chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl)acetoxymethyl]-1-(dimethylamino)diazen-1-ium-1,2-diolate O2-[2-(1-(4-Chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl)acetoxymethyl]-1-(pyrrolidin-1-yl)diazen-1-ium-1,2-diolate O2-[2-(4-(Isobutyl)phenyl)propanoyloxymethyl]-1-(N,N-dimethylamino)diazen-1-ium-1,2-diolate O2-[2-(4-(Isobutyl)phenyl)propanoyloxymethyl]-1-(pyrrolidin-1-yl)diazen-1-ium-1,2-diolate OAG Ocaperidone OCH3-5-APT OCH3-6-APT OCRF OCTOCLOTHEPIN OCTOCLOTHEPIN,(+) OCTOCLOTHEPIN,(-) OCTOCLOTHEPIN-R OCTOCLOTHEPIN-S Octopamine,(+/-) octreotide octreotide amide octreotide-Tyr3 of 8-{1-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione OFQ 1-17 OFQ II 1-17 OFQ II 1-28 OFQ/N OFQ/N (1-11) OFQ/N (1-11), Iodo[Tyr10] OFQ/N (1-11),[Tyr10] OFQ/N (1-7) OFQ/N UFP-102 OFQ/N,Iodo[Tyr14] OFQ/N,[Tyr14] OFQ/N-NH2,[(pF)Phe4,Arg14,Lys15] OHT OLANZAPINE olanzapine, 2-hydroxymethyl olanzapine, 4'-N-Oxide olanzapine, N-desmethyl Olvanil OMB OMB-18 OMB-19 OMO5-057 ONDANSETRON Ondansetron HCl Ondansetron HCl ONDANSETRON,R- ONDANSETRON,S- ONO 11,113 ONO 4057 ONO-1301 OPC-14597 OPC-18790 OPC-21268 OPC-28326 OPC-31260 OPC-41061 OPC-4392 opipramol ORF-11676 Org 3770,(+) Org 3770,(+-) Org 3770,(-) ORG GC94 ORG-12962 ORG-37684 ORG-3770 ORG-5222 ORG2766 oripavine Orphenadrine Oseltamivir Acid - tamiflu metabolite Oseltamivir PO4 - Tamiflu Otenabant oxaprosin Oxaprotiline Oxazepam OXIPEROMIDE OXO-M Oxotremorin Oxotremorine OXPRENOLOL Oxybutinin oxybutynin oxycodone OXYMETAZOLINE oxymetazoline Oxymorphine Oxymorphone Oxytocin Oxytremorine Oxytyramine p-AMINOCLONIDINE p-aminophenylethyl-m-trifluoromethylphenylpiperazine p-chlorophenyl moiety p-F-HHSiD p-FHSD p-iodoclonidine p-MPPI P103A P1075 P108A P242 P34-PYY,human P34A P4S P5 P5-NH2 P51 P513 P517 P518 P52 P550 P552 P88-8991 P95-12113 PACAP PACAP(1-23) PACAP(1-23,VIP28) PACAP(1-27) PACAP(1-33,Cys34) PACAP(1-38) PACAP(10-38) PACAP(11-27) PACAP(11-38) PACAP(2-27) PACAP(2-38) PACAP(3-25) PACAP(3-27) PACAP(3-38) PACAP(4-27) PACAP(4-38) PACAP(5-27) PACAP(5-38) PACAP(6-27) PACAP(6-31) PACAP(6-35) PACAP(6-38) PACAP(7-27) PACAP(7-38) PACAP(8-28) PACAP(8-38) PACAP(9-27) PACAP(9-38) PACAP-27 PACAP-38 PACAP-VIP PACPX PAF Pafenolol Paliperidone Palmidrol palmitoylethanolamide pancreatic polypeptide pancreatic polypeptide, bovine pancreatic polypeptide, human pancreatic polypeptide, rat Pancuronium Papaverine PAPP para-fluoro-hexahydro-sila-dilfenidol Paracetamol Paracort Paramorfan Paramorphan Paraxanthine PARECOXIB Pargyline PAROXETINE PARTHENOLIDE PAT paxilline PB-28 pb12 PBR28 PCCG-IV PCP PCP,m-NH2 PCP,m-OH pCPP PD 123177 PD 128,907 PD 166866 PD 81,723 PD116948 PD117302 PD156707 PDDF pdspTestCompound1 pdspTestCompound2 pdspTestCompound3 pdspTestCompound4 PE2I PEA Pemetrexed PENBUTOLOL(-) PENFLURIDOL Pentagastrin Pentamidine Pentanoic acid (R)-2-methoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester Pentazocine PENTAZOCINE (+) PENTAZOCINE (-) Pentazocine,(+/-) Pentobarbital Pentoxifylline penucuronium peptide histidine isoleucinamide-(1-27) perazine PERGOLIDE PERLAPINE Perospirone PERPHENAZINE PG 13,14-dihydro-15-keto-D2 PG Thromboxane B2 PG-L PG648 PGA2 PGB2 PGD1 PGD2 PGD2-methyl ester PGE1 PGE1, 13,14-dihydro PGE1, 8-iso PGE1,1-OH PGE1,11-DEOXY PGE2 PGE2 13,14-dihydro PGE2, 13,14-dihydro15-oxo PGE2, 15-epi PGE2, 5,6-trans PGE2,16,16-DIMETHYL PGE2,17-Phenyl PGE2,19R(OH) PGF1 alpha 6-keto PGF1alpha PGF1alpha, 6-oxo PGF2 Alpha, 1-isopropyl ester PGF2Alpha PGF2Alpha,16-Phenoxy PGF2Alpha,17-phenyl PGF2Alpha,8-Iso PGH2 PGH2, 9,11 azo- PGI1, 6beta PGI2 PGI2 Ph3COH Ph3SiOH PhAR PhAR, 5-I PhAR, 6-I PhAR, Cycloproyl PhAR, Di-hydro PhAR, ent PhAR, epoxy Phe-Phe-Tyr-Thr-Pro-Lys-Thr Phe2TRH Phenazocine PHENCYCLIDINE Phencyclidine HCl Phendimetrazine Phendimetrazine-(+) Phendimetrazine-(-) Phenelzine Phenethylamine Phenethylamine, alpha-methyl-, (+)- Phenindamine pheniramine Phenmetrazine Phenobarbitol sodium salt Phenothiazine PHENOXYBENZAMINE Phentermine PHENTOLAMINE phentolamine phenyl (±)-((4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-prolinate phenyl (±)-(4aR,8S,8aR)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate phenyl (±)-(4aR,8S,8aR)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate phenyl (±)-(4aR,8S,8aR)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate Phenyl (S)-3-(Pyrrolidin-2-ylmethoxy)isoxazole-5-carboxy-late Hydrochloride Phenyl(4-phenyl-2-(phenylamino)thiazol-5-yl)methanone Phenyl-(2-pyridin-2-yl-3H-benzoimidazol-5-yl)-methanone Phenyl-(2-thiazol-4-yl-1H-benzoimidazol-5-yl)-methanone Phenyl-carbamic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phosphonooxy-methyl-propyl Ester, Ammonium Salt Phenyl-[1-(4-p-tolyl-butyl)-piperidin-4-yl]-methanol Phenylacetic Acid 2-acetoxymethyl-3-(2-chloro-6-methylamino-purin-9-yl)-propyl Ester Phenylacetic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phenylacetoxymethyl-propyl Ester PHENYLBIGUANIDE Phenylbutanoylhistamine Phenylcarbamic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-phenylcarbamoyl-oxymethyl-propyl Ester PHENYLEPHRINE Phenylephrine,(+) Phenylephrine,(+/-) Phenylephrine,(-) Phenylethanolamine Phenylethylamine phenylpiperazine phenylpiperazine chromen-2-one phenylpiperidine dimethyl-substituted PHI PHNO PHNO,(+) PHNO,(-) Phosphinothricin phosphothioate PHXA85 Phyllolitorin physalaemin Physostigmine PIB piboserod Piclamilast Picrotoxin Pifluthixol Piflutixol Pilocarpine PIMOZIDE PINACIDIL PINDOBIND-5-HT1A PINDOLOL,(+) PINDOLOL,(+/-) PINDOLOL,(-) PIPAMPERONE Piperazine piperazinoindole Piperidin-1-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone Piperidine Piperidolate PIPEROXAN Pipotiazine pipridine PIRENPERONE PIRENZEPINE Piribedil Piroxicam Pitavastatin Pitavastatin lactone PIZOTIFEN Pizotyline PK11195 PL-3-016 PL-3-017 PL-3-025 PL-3-048-4 PL017 PNU-96415E PNU109,291 Poly-Pred PP 31-36, acid free, human PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human PP [Ile31,Gln34], human PP, BOVINE PP, chicken PP, guinea pig PP, human PP, rat PP,FROG PP,SALMON PP1 PP13-36, HUMAN PP2 PP2-36, HUMAN PP3 PP31-36, HUMAN PPADS PPAP, (-) PPG PPOM PPP, (+) PPP, R(+)-3 PPP, S(-)-3 PRACTOLOL Practolol,(+) Practolol,(-) Pramipexole Pranlukast Pravastatin Pravastatin lactone PRAZOSIN PrBCh Pred-G Predamide predicentrine Prednicarbate Prednicen-M prednisolone Prednisolone Prednisone Predsulfair Preladenant (SCH420814) Prelone Prenylamine Preprogalanin-(1-30) Procainamide PROCHLORPERAZINE Procyclidine Progestasert progesterone Progesterone Proglumide PROMAZINE PROMETHAZINE Prometrium propan-2-yl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]he... propan-2-yl (2S)-2-[(5-cyano-6-oxo-4-phenyl-1H-pyrimidin-2-yl)sulfanyl]propanoate propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate   PROPANOLOL(-) Propanolol,(+/-) PROPERICIAZINE Propionic Acid 3-(2-chloro-6-methylamino-purin-9-yl)-2-propionyloxymethyl-propyl Ester Propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7... Propionyl-pTyr-Leu -Pro-Gln-Thr-NH2 propofol Propoxyphene,(+/-) Propoxyphene-d PROPRANOLOL PROPRANOLOL, d PROPRANOLOL, dl PROPRANOLOL, l- PROPRANOLOL, S PROPRANOLOL,(+) PROPRANOLOL,(-) proptriptyline Propyl (1S,2R,3S,4R,5S)-4-(2-Chloro-6-((dicyclopropylmethyl)- amino)-9H-purin-9-yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carbo... propyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-... Propyl 2-methyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate Propyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate Prostacyclin Prostaglandin F2Alpha Prostaglandin F2Alpha, 1-isopropyl ester Prostaglandin F2Alpha, 17-phenyl Prostaglandin I2 Prostratin Protheobromine Prothipendyl Protriptyline Protryptyline proxyfan Proxyfylline Proxyphylline Prozac PrRP20 PrRP24-31 PrRP31 Prucalopride PS-1-34B PS-1-34B C20H17N4BrO PS-1-35 psammopemmin A PSB-1115 PSB-36 Pseudoephedrine, (-) Pseudoephedrine,(+) Pseudoephedrine,(+/-) Pseudohypericin Pseudonorephedrine, (+) [cathine, (+)] Pseudonorephedrine, (-) [cathine, (-)] Pseudophenmetrazine PSILOCIN PSILOCYBIN PTA2 PTH(7-34),[D-Trp12,Tyr34] PTHrP(1-34) PTHrP(7-34) PTT(-) PTZ Purealidin A Purealin purvalanol A PW-007A PWZ-0071 PWZ-007A PWZ-009A1 PWZ-029 PWZ-085 PWZ-096 Pyr3TRH Pyrathiazine Pyridine-2-carboxylic Acid ((R)-1-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethylc... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(3-bromo-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-eth... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(4-Benzo[1,3]dioxol-5-yl-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-but... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethylc... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(biphenyl-3-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-1-Benzyloxymethyl-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)ethylcarbamoyl]... Pyridine-2-carboxylic Acid ((S)-1-{(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methylbutylcarbamoyl)ethylcarbamoyl]-2-hydroxy-1-phene... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Benzo[1,3]dioxol-5-yl-benzyloxymethyl)-3-butylcarbamoyl-2-hydroxy-propylcarba... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromo-benzyloxymethyl)-2-hydroxy-3-[2-(3-methoxyphenyl)ethylcarbamoyl]propylc... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromo-benzyloxymethyl)-3-cyclohexylcarbamoyl-2-hydroxypropylcarbamoyl]-2-meth... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-2-hydroxy-3-(2-phenylaminoethylcarbamoyl)propylcarbamoy... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-2-hydroxy-3-(3-methoxypropylcarbamoyl)propylcarbamoyl]-... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-bromobenzyloxymethyl)-2-hydroxy-3-(3-phenylpropylcarbamoyl)propylcarbamoyl]-2... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-(4-cyanobenzylcarbamoyl)-2-hydroxypropylcarbamoyl]-2-... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-(cyclohexylmethylcarbamoyl)-2-hydroxypropylcarbamoyl]... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(4-Bromobenzyloxymethyl)-3-butylcarbamoyl-2-hydroxypropylcarbamoyl]-2-methylprop... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-1-(Biphenyl-4-ylmethoxymethyl)-3-butylcarbamoyl-2-hydroxy-propylcarbamoyl]-2-methy... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-3-Butylcarbamoyl-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propylcarbamoyl]-2-... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(3-... Pyridine-2-carboxylic Acid {(S)-1-[(1S,2S)-3-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(4-... Pyridine-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide Pyridine-4-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide pyridoxal-phosphate-6-azophenyl-2',4'-disulfonic acid PYRILAMINE pyrovalerone Pyrrolidin-1-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone Pyrrolidine PYRROLYLTRYP,DiMe PYY PYY 3-36 PYY 3-36, porcine PYY 3-36, rat PYY Pro34, Human PYY, chicken PYY, human PYY, N-alpha-Ac, 22-36 PYY, N-alpha-Ac, 25-36 PYY, porcine PYY, rat PYY, zebrafish PYY,[leu31,Pro34], human PYY13-36, porcine PYY13-36, rat PYY3-36, human Pyz11-D-Trp8-SRIF Pyz6-D-Trp8-SRIF Pyz7-D-Trp8-SRIF PZII-028 PZII-029 pzp QDOB QH-146 QH-II-063 QH-II-066 QH-II-067a QH-II-075 QH-II-077 QH-II-080b QH-II-082 QH-II-085 QH-II-090 QH-II-090 (CGS-8216) QH-II-092 QHII-066 QMDP(+) QNB Quercetin Quercitrin Quetiapine Quinelorane Quinerolane Quinidine Quinine Quinolinate Quinolinic acid Quinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide QUINPIROLE Quinpirole,(+) Quinpirole,(-) quinuclidin-3-yl benzhydrylcarbamate Quinuclidine Quinuclidinyl benzilate QUIPAZINE QUIPAZINE,8-Me Quisqualate Quisqualate, L Quisqualic acid R 115866 R 214127 R 34 427 R 43,448 R 48 800 R 50 890 R 50 970 R 51 562 R 51 703 R 52 368 R 52 981 R 56413 R(+)-3-(3-Hydroxyphenyl)-N-propylpiperidine hydrochloride R(+)-3-PPP hydrochloride R(+)-TMQ R(-)-2-methoxy-11-acetyloxy-N-n-propylnoraporphine R(-)-3-Methyl-1,2,3,4-tetrahydroisoquinoline R(-)NPA R)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) r, h, m MCH R,R-2b R,S-PHPNECA R-(+) staurosine R-(+)-3-Chloromethyl-7-nitro-THIQ R-(+)-3-Chloromethyl-THIQ R-(+)-3-Fluoromethyl-7-bromo-THIQ R-(+)-3-Fluoromethyl-7-cyano-THIQ R-(+)-3-Fluoromethyl-7-N-(4-chlorophenyl)aminosulfonyl-THIQ R-(+)-3-Fluoromethyl-7-nitro-THIQ R-(+)-3-fluoromethyl-THIQ R-(+)-3-Hydroxymethyl-7-bromo-THIQ R-(+)-3-Hydroxymethyl-7-nitro-THIQ R-(+)-3-Hydroxymethyl-THIQ R-(-)-2,3:[4,5-b]-2'-Aminothiazolo-10,11-dihydroxyaporphine R-(-)-3-methyl-7-nitro-THIQ R-(-)-3-methyl-THIQ R-3-methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole hydrochloride R-41-468 R-alpha-methylhistamine R-citalopram R-N6-(2-phenylisopropyl) adenosine R-nisoxetine R-PHPNECA R-PIA R121919 R214127 RA-7 rac, anti-7,9-difluoro-5-(3-methylcyclohex-2-en-1-yl)-2,2,4-trimethyl 2,5-dihydro-(1H)6-oxa-1-aza-chrysen rac, syn-5-(cyclohex-2-en-1-yl)-7,9-difluoro-2,2,4-trimethyl 2,5-dihydro-(1H)6-oxa-1-azachrysen rac, syn-7,9-difluoro-5-(3-methylcyclohex-2-en-1-yl)-2,2,4-trimethyl 2,5-dihydro-(1H)6-oxa-1-aza-chrysen rac-(1S,2R,4S)-2-bromo-N-[1-(3-bromobenzyl)-6-(2,4-dichlorophenyl)-4-(4-fluorobenzenesulfonyl)-2-hydroxyhexyl]-4,5-dimethoxyb... rac-(1S,2R,4S)-N-[1-(3-Bromobenzyl)-2-hydroxy-4-(3-methylbutane-1-sulfonyl)pentyl]-3-methanesulfonylpropionamide rac-(1S,2R,4S)-N-[1-(3-Bromobenzyl)-4-(4-fluorobenzenesulfonyl)-2-hydroxy-6-methylheptyl]-2-(2,6-dimethylphenoxy)acetamide rac-(1S,2R,4S)-N-[1-(3-bromobenzyl)-6-(2,4-dichlorophenyl)-4-(4-fluorobenzenesulfonyl)-2-hydroxyhexyl]-2-(2,4-dichlorophenoxy... rac-(1S,2R,4S)-N-[1-Bromobenzyl)-2-hydroxy-6-methyl-4-(4-methylaminobenzenesulfonyl)heptyl]-2-(2,6-dimethylphenoxy)acetamide rac-(1S,2R,4S)-N-[1-Bromobenzyl)-4-(4-(dimethylamino)benzenesulfonyl)-2-hydroxy-6-methylheptyl]-2-(2,6-dimethylphenoxy)acetam... rac-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide rac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl)-1H-imidazole-4-carboxamide rac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl)-1H-imidazole-4-carboxamide rac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide rac-2-(5-(3-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(5-(4-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(6-fluoro-5-(3-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(6-fluoro-5-(3-methoxyphenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(6-fluoro-5-(3-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(6-fluoro-5-(4-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(6-fluoro-5-(4-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-2-(6-fluoro-5-phenylpyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride rac-3'-(3-aminophenyl)deschloroepibatidine trihydrochloride rac-3'-(3-chlorophenyl)deschloroepibatidine dihydrochloride rac-3'-(3-fluorophenyl)deschloroepibatidine dihydrochloride rac-3'-(3-nitrophenyl)deschloroepibatidine dihydrochloride rac-3'-(4-nitrophenyl)deschloroepibatidine dihydrochloride rac-3-(3-methoxyphenyl)deschloroepibatidine dihydrochloride rac-3-(4-aminophenyl)deschloroepibatidine trihydrochloride rac-3-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride rac-3-phenyldeschloroepibatidine dihydrochloride rac-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide rac-4-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride rac-6-(1-methylpyrrolidin-2-yl)quinoline rac-8-fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide rac-cis-N-((2-hydroxycyclopropyl)palmitamide rac-cis-N-arachidonoylcyclopropanolamide rac-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine rac-N-{[(1R,2R)-2-(3-methoxyphenyl)cyclopropyl]methyl}ethanediamide rac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine rac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine rac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine rac-trans N-arachidonoylcyclopropanolamide rac-trans-N-oleoylcyclopropanolamide rac-[3-(5-fluoro-1H-indol-3-yl)-propyl]-(5-methoxy-chroman-3-yl)-propyl-amine Racemate RACLOPRIDE raloxifene raltitrexed RAMH Ranatensin RANITIDINE RAUBASINE RAUWOLSCINE RC 160 RC 160II RC-121 rCST-29 Reboxetine Rec 15/3079 Rec 27/0074 Rec 27/0224 rel-(2R,6R,11R)-6,11-Dimethyl-3-(3-methyl-but-2-enyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid ami... rel-3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)benzamide Remoxapride REMOXIPRIDE RENZAPRIDE RESERPINE Resiniferatoxin Resveratrol Revex RFRP-1 RFRP-3 Rhodamine123 Rhodei-Litorin RILAPINE rilmenidine Rilmenidine RIMCAZOLE Rimonabant Rinvanil Rinvanil, Acetyl Rinvanil, Benzoil Rinvanil, Phenyl-propionyl RISPERIDONE RIT-70 RITANSERIN Ritonavir RJR-2429 RMI 81,582 RN 76186 Ro 04-5595 Ro 04-6790 RO 19-3704 Ro 19-4603 RO 20-1724 Ro 25-1392 Ro 25-1553 Ro 25-6981 Ro 48-8071 Ro 48-8587 Ro 60-0175 Ro 600332 Ro 600869 Ro-15-4513 Ro-4864 Ro15-1788 Ro15-4513 Ro15-4513 Ro5-4864 Ro65-6570 ROFECOXIB Roflumilast Rohdei-litorin rolipram Ropinirole Roscovitine Rosuvastatin Roxindole RP 58467 RP 59227 RP 59228 RP 67,580 RP 73870 RS 100235 RS 23597 RS 23597/190 RS 39604 RS 57639 RS 67333 RS 67506 RS 67532 RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine (2) RS-(+/-)-Sulpriride RS-100975 RS-102221 RS-127445 RS-127445-190 RS-17053 RTI-106 RTI-110 RTI-111 RTI-112 RTI-113 RTI-114 RTI-116 RTI-117 RTI-118 RTI-12 RTI-120 RTI-121 RTI-122 RTI-127 RTI-128 RTI-129 RTI-13 RTI-133 RTI-134 RTI-135 RTI-14 RTI-146 RTI-147 RTI-149 RTI-15 RTI-150 RTI-156 RTI-160 RTI-183 RTI-186 RTI-190 RTI-191 RTI-192 RTI-193 RTI-196 RTI-198 RTI-203 RTI-204 RTI-205 RTI-206 RTI-207 RTI-208 RTI-209 RTI-210 RTI-211 RTI-212 RTI-213 RTI-214 RTI-215 RTI-221 RTI-222 RTI-226 RTI-227 RTI-228 RTI-229 RTI-258 RTI-29 RTI-31 RTI-32 RTI-49 RTI-51 RTI-52 RTI-53 RTI-55 RTI-59891 RTI-598923 RTI-598925 RTI-66 RTI-74 RTI-88 RU 24213 RU 24926 RU 24969 RU 27849 RU 28253 RU 28306 RU 38486 RU-43044 RU-486 Rutin RWAY,(-) RWJ-377796 RX 811033 RX811012 RX811022 RX811046 RX811055 RX811059 RX821002 RX821008 RX821010 RX821022 RX831001 RX831003 RX841047 RX851057 RX851062 RXFP1/2 RXFP2/1 RY 24 RY 80 RY-008 RY-023 RY-023 C22H27N3O3Si RY-024 RY-024 C19H19N3O3 RY-031 RY-033 RY-047 RY-053 RY-054 RY-057 RY-058 RY-059 RY-061 RY-062 RY-066 RY-067 RY-068 RY-069 RY-071 RY-072 RY-073 RY-076 RY-079 RY-080 RY-080 C17H15N3O3 RY-098 RY-A100 RY-I-28 RY-I-29 RY-I-31 S 1033 S 132 S 14489 S 145 S 15535 S 15931 S 20098 S 20499 S(+)-3-Methyl-1,2,3,4-tetrahydroisoquinoline S(-)-4-{4-[2-(isochroman-1-yl)ethyl]piperazin-1yl}benzenesulfonamide S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline S)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one S)-N6-Propyl-N6-(2-(4-(quinolin-4-yl)piperazin-1-yl)ethyl)-4, 5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine S,S-2c S,S-Hydroxybupropion S-(+)-3-methyl-7-nitro-THIQ S-(+)-3-methyl-THIQ S-(-)-3-Chloromethyl-7-nitro-THIQ S-(-)-3-Chloromethyl-THIQ S-(-)-3-Fluoromethyl-7-bromo-THIQ S-(-)-3-Fluoromethyl-7-cyano-THIQ S-(-)-3-Fluoromethyl-7-N-(4-chlorophenyl)aminosulfonyl-THIQ S-(-)-3-Fluoromethyl-7-nitro-THIQ S-(-)-3-fluoromethyl-THIQ S-(-)-3-Hydroxymethyl-7-bromo-THIQ S-(-)-3-Hydroxymethyl-7-nitro-THIQ S-(-)-3-Hydroxymethyl-THIQ S-(-)-3-PPP S-(-)-3-PPP Preclamol S-(-)-Sulpride S-(R)-1-((2S,3R)-1-(4-fluorophenyl)-2-(4-hydroxyphenyl)-4-oxoazetidin-3-yl)-3-phenylpropyl ethanethioate S-145,(+) S-34324 S-5751 S-Adenosylmethionine S-Allyl-brassinin S-Benzyl-brassinin S-Beta-Dimethylhistamine-R-alpha s-Duloxetine S-Hexyl-brassinin S-isomer S-L-365,260 S-N6-(2-phenylisopropyl) adenosine S-phenyl (±)-(4aS,8R,8aS)-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbothioate S-PHPNECA S-PIA S14297 S16924 S18127 S18616 S1P S31411 (+-) S32504 S32504 (+) S32601 (-) S33005 S33084 S33526 S38093 SA sakurantin Salbutamol,(+/-) Salicin Salicylaldehyde salicylic acid Salmeterol Salmon MCH salsalate Salvinorin A Salvinorin A lactol Salvinorin A, 8-epi Salvinorin B formate Salvinorin C Salvinorin D Salvinorin E Saquinavir mesylate Saralasin SAS-0132 SAS-1121 Sauvagine SB 200646 SB 206553 SB 207266 SB 209670 SB 216641 SB 217242 SB 221284 SB 223412 SB 234551 SB 235375 SB 242084 SB 277011 SB-214111 SB-215505 SB-224289 SB-258510 SB-258585 SB-258719 SB-269970 SB-271046 SB-277011-A SB-357134 SB200646a SB202190 SB203186 SB203580 SB204070 SB204741 SB205149 SB207710 SB242087 SC 53606 SC-46275 SC-51089 SC-51322 SC19220 SC241 SC49518 SC53116 SC58125 SCH 206272 SCH 23388 SCH 23388 (S-enantiomer) SCH 23390 SCH 23390 (R-enantiomer) SCH 23390,R(+) SCH 39166 SCH 79687 SCH58261 SCOPOLAMINE SDZ 205557 SDZ 206-792 SDZ 206-830 SDZ 21-009 SDZ 21-009,(+) SDZ 21-009,(-) SDZ 210-204 SDZ 210-205 SDZ 216,525 SDZ GLC 756 SDZ GLC 756 (+) SDZ SER-082 SDZ-HDC-912 SDZ-HTF919 Secoverine Secretin securinine seglitide selegiline, SEL Senktide SEPTOPERONE SER-084 Sergolexole seroquel Serotonin Serotonin,N-acetyl SERTINDOLE SERTRALINE Servisone SETOPERONE SFLLR SFLLR-NH2 SFLLR-OH SFLLRN-NH2 SFLLRN-OH SFLLRNPNDKYEPF-OH SH-053-2F SH-053-2F-S-CH3 SH-I-02B SH-I-030 SH-I-04 SH-I-047 SH-I-048A SH-I-085 SH-I-75 SH-I-89S SH-I-S66 SH-I89S SH-O53-5-CH3-2F SH-TS-CH3 SH-TSC-1 SH-TSC-2 SH-TSC-2 (BCCT) SHU-1-19 SHU-221-1 SHX SIB-1508Y SIB-1757 SIB-1765F SIB-1893 sibutramine Silahexocyclium sildenafil Simvastatin acid Simvastatin lactone sinoacutine SIOM SK&F 83822 SK&F 83959 SK-896 SKF 10,047 (+) SKF 10,047 (-) SKF 10047 SKF 10047 (+/-) SKF 104078 SKF 104856 SKF 108566 SKF 24260 SKF 29661 SKF 38393 SKF 38393 (+) SKF 38393 (+/-) SKF 64139 SKF 75670 SKF 77434 SKF 81297 SKF 82957 SKF 82958 SKF 83566 SKF 83566,R- SKF 86466 SKF-38393 SKF-76783 SKF-82526, (+) SKF-82526, (-) SKF-83959 SKF38393 SKF91581 SKI-606 SL 651498 SL-NH2 SL650155 SL651498 SLIGKV-NH2 SLIGR-NH2 SLIGRL-NH2 SM 13496 SMM-189 SMS 201-995 SN003 SNC-80 sodium 4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)benzenesulfonate Sodium salicylate Somatostatin Somatostatin response inhibitory factor 14 Somatostatin response inhibitory factor 28 Somatostatin-14 somatostatin-28 sopromidine, R(-) sopromidine, S(+) sorbinil Sotalol Sotalol,(+) Sotalol,(-) SP600125 SpAMDA sparfloxacin Spectramide Spermidine Spermine SPH-121 SPH-165 SPH-195 SPH-38 SPIPERONE SPIPERONE,N-Me Spiradoline Spiroperidol SPIROXATRINE SPIROXATRINE,(+) SPIROXATRINE,(-) Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate Spiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate SQ 28668 SQ 29548 SQ 30741 SR 120819A SR 121463B SR 140333 SR 141716A SR 142801 SR 142806 SR 142948A SR 144528 SR 147778 SR 27897 SR 46349B SR 48527 SR 48692 SR 48968 SR 49059 SR 49711 SR 57746 A SR 59230A SR 95531 SR144528 SR95531 SRI 63-441 SRI-22138 srif SRIF-D-Trp8 SRIF-[Des-Ala1,des-Gly2,His4,5,D-Trp8] srif14 srif28 SRIF28-Leu8,D-Trp22,Tyr25 ss-14 SS-22 SS-25 ss-28 SSR125543A SSR149415 SSR181507 SSR240600 SSR591813 sst-14 sst-28 St-600 ST-91 ST1460 ST1469 ST1615 ST1622 ST1899 STA2 Stadol Staurosporine Stavudine stepholidine Sterane Strychnine SU11248 Suberyldicholine Substance K Substance P Substance P [Sar9,Met(O2)11] Substance P(4-11),[Dpro4,Dtrp7,9,10] Substance P,[DArg1,DTrp7,9,Leu11] Succinic Acid mono-[2-(3-carboxy-propionyloxymethyl)-3-(2-chloro-6-methylamino-purin-9-yl)-propyl] Ester Succinylcholine Sufentanyl Sufugolix Sulfasalazine sulfated CCK(26-33) sulforidazine suliforidazine Sulindac Sulindac Sulfide Sulindac sulphide Sulphrin Sulpirid SULPIRIDE SULPIRIDE,(+) SULPIRIDE,(-) Sulpiride-d Sulpiride-high,(-) Sulpiride-l Sulpiride-low,(-) Sulpiride-R Sulpiride-S SULPROSTONE Sultopride SUMATRIPTAN Suprofen Suramin Suramin sodium SVO-8-14 SVO-8-20 SVO-8-30 SVO-8-67 SYA013 SYA16263 Symbicort Sympatholytin synaptic 34 Synephrine,(+/-) t-2,4-PDC T-226296 T-7-Riboside t-ADA t-PDC TACA Tacrine tacrine homodimer tadalafil TAK-013 Talipexole Talsupram Tamoxifen Tamoxifen, 4-hydroxy Tamsulosin Tanaproget Tapentadol TAPS Taranabant Tarceva Tasimelteon TB-3-4 TC-2429 Tc-LIGRLO-NH2 tc-NH2 TC-YT-II-76 TCMDC-124076 TCP TDBMSOH tefludazine Teflutixol TELENZEPINE TELEPATHINE Temelastine Tenidap TENILAPINE Tenofovir Terazosin Terbutaline Terbutaline,(+/-) Terfenadine Terfenadine, R(+) Terfenadine, S(-) TERGURIDE tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate tert-Butyl 1-(4-Chlorophenyl)-2-(2,4-dichlorophenyl)-5-methyl-1H-imidazole-4-carboxylate tert-butyl 4-(((3S,6S)-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)piperidin-3-yl)methyl)piperazine-1-carboxylate tert-butyl 4-((9-pentyl-9H-carbazole-3-carboxamido)methyl)piperidine-1-carboxylate Tert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate tert-butyl 4-(9-pentyl-9H-carbazole-3-carbonyl)piperazine-1-carboxylate tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate tert-Butyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate tert-Butyl 9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undec-7-ene3-carboxylate tert-butyl(3S)-3-[({(5S)-5- [2,2.2-trifluro-1-hydroy-1-(trifluoromethyl)ethyl]-4.5-dihydroisoxazol- 3yl}carbonyl)amino] butan... tert-Butyl-(3R)-3-[({(5R)-5-[2,2.2-trifluro-1-hydroy-1-(trifluoromethyl)ethyl]-4.5- dihydro-isoxazol-3yl}carbonyl)amino]butan... tert-Butyl-(3R)-3-[({(5S)-5- [2,2.2-trifluro-1-hydroy-1-(trifluoromethyl)ethyl]-4.5-dihydroisoxazol- 3yl}carbonyl)amino] buta... tert-Butyl-(3R)-3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}butanoate tert-Butyl-(3S)-3-[({(5R)-5-[2,2.2-trifluro-1-hydroy-1-(trifluoromethyl)ethyl]-4.5- dihydroisoxazol-3yl}carbonyl)amino]butano... tert-Butyl-(3S)-3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}butanoate tert-Butyl-3-{[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydroisoxazole- 3-carbonyl]-amino}butanoate TERTATOLOL(-) testosterone tetrabenazine TETRAETHYLAMMONIUM Tetrahydroalstonine tetrahydroamentoflavone Tetrahydrocannabinol tetrahydronaphthalene Tetrahydronicotyrine, DL- Tetrahydrozoline Tetramethylammonium tetrodotoxin TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-NMePhe-Asp-Yyy-Trp-Ac TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-1-Adoc TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-2-Adoc TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-Boc TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-D-Trp-H TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-Trp-Ac TFA·H-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-Nle-Trp-Boc TFMPP TG-4-29 TG-4-39 TG-II-82 THC THC, 1-O-(2-morpholinoethyl) THC, 1-O-(3-Aminopropyl) THC, 1-O-(4-Aminobutyl) THC, 1-O-(4-Phthalimidobutyl THC, 1-O-(6-Aminohexyl) THC, 1-O-biphenylmethyl-delta 8 THC, 1-O-biphenylmethyl-delta 9,11 THC, 1-O-Carbamoyl THC, 1-O-Methyl-3-(norpentyl)-3-propyl THC, 1-O-Methyl-delta 8 THC, 1-O-methyl-delta 9 THC, 1-O-methyl-delta 9,11 THC, 11-F THC, 11-OH-5'-TMA THC, 11-OH-delta 8 THC, 11-OH-delta 9 THC, 2-I THC, 2-I-delta 8 THC, 3-(Norpentyl)-3-propyl THC, 5'-Br THC, 5'-F THC, 5'-F3 THC, 5'-I THC, 5'-OH THC, 8 beta-OH THC, 8-(N-morpholino)-amino THC, 9-Nor-9-carboxy-delta 8 THC, 9-Nor-9-carboxy-delta 9 THC, delta 8 THC, delta 9 THC, delta 9, 11 THC, O, 10-Methano THC, O, 2-propano THC-DMH THC-DMH, (+)-11-OH THC-DMH, (-)-11-OH thebaine Theobromine theophylline Theophylline (1,3-dimethylxanthine) Thiabendazole Thio-4-PIOL thio-AMPA Thio-ATPA Thio-ATPA-R Thio-ATPA-S thio-Cl-IB-MECA thioflavin T thiol phosphoric acid Thiomuscimol Thioperamide Thioproperazine THIORIDAZINE THIOTHIXENE THIOTHIXENE,cis- THIOTHIXENE,trans- Thiothixene-cis THIP THIP, Aza- THIP, Iso- THIQ THIQ, 7-Aminosulfonyl-3-fluoromethyl THIQ-7-Br THIQ-7-CF3 THIQ-7-CH2NH2 THIQ-7-CH2NHSO2CH3 THIQ-7-CH2OH THIQ-7-CN THIQ-7-CO2H THIQ-7-COCF3 THIQ-7-COCH3 THIQ-7-CONH2 THIQ-7-I THIQ-7-N-(SO2CH3)2 THIQ-7-NH2 THIQ-7-NHCO2CH3 THIQ-7-NHSO2CH3 THIQ-7-NO2 THIQ-7-OCH3 THIQ-7-SCH3 THIQ-7-SO2CCl3 THIQ-7-SO2CH2CH=CH2 THIQ-7-SO2Ph THP Threohydrobupropion Thujone thyl (1S)-2-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyla... Thymeleatoxin Thymeleatoxin (low PS) Thymidine thyrotropin-releasing hormone Tianeptine Tiapamil Tiapride Ticlopidine TICP -psi Tilozepine TIMOLOL TIOSPERONE TIOSPIRONE Tiotidine tiotixene TIP39(7-39) TIPP TIPPpsi TIZANIDINE TJH-IV-43 TJH-IV-51 TJH-V-88 TL304 TL99 TMA TMA,2,3,5- TMA,2,4,5- TMA,3,4,5- TMP TMPNBn TMPNMe TMQ, (+/-)-8-Fluoro TMQ, 3',5'-Diiodo TMQ, 3'-Amino TMQ, 3'-Iodo TMQ, 3'-Nitro TMQ, 5,8-Difluoro TMQ, 5-Fluoro TMQ, 5-Iodo TMQ, 5-TrifluoroMe TMQ, 8-Iodo TMQ, Amidine TMQ, Cyclic sulfite TMQ, N-amino-benzyl TMQ, N-benzyl TMQ, N-chloro-benzyl TMQ, N-dichlorobenzyl TMQ, N-hydroxyethyl TMQ, N-methoxybenzyl TMQ, N-methyl TMQ, N-nitro-benzyl TMQ, R-(+) TMQ, R-(-)-8-Fluoro TMQ, Racemic TMQ, S-(+)-8-Fluoro TMQ, S-(-) Tmt-D-Arg-Phe-Lys-NH2 Tol2Gdn TOLAZOLINE Tolmetin toloxatone, TOL Toluene-4-sulfonic Acid 3-{4-[2-(4-(Dimethylamino)phenyl)vinyl]phenoxy}-2-hydroxymethylpropyl Ester Tomoxetine Tomoxiprol Tonapofylline topiramate Topotecan toxiferine TP-680 Tracazolate Tracrium Tramadol(+-) Tramadol,(+) Tramadol,(-) Tramazoline trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine trans -2-Amino-4,4a,5,6,7,8,8a,9-octahydro-5-propylthiazolo[4,5-g]quinoline Difumarate 2C4H4O4 trans 1-hydroxyindane trans piflutixol-(E) trans-(3'R)-Quinuclidin-3'-yl 4-Hydroxy-1-Phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate trans-(3R, 6S)-6-benzhydryl-tetra-hydropyran-3-yl ester trans-1,2-bis(4-chlorophenyl)-5-(3,4-difluorobenzyl)piperidine trans-1,6-bis(4-chlorophenyl)-3-(3,4-difluorobenzyl)piperidin-2-one trans-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-5-(3,4-difluorobenzyl)piperidine trans-1-(4-chlorophenyl)-6-(2,4-dichlorophenyl)-3-(3,4-difluorobenzyl)piperidin-2-one trans-1-methyl-1-phenyl-3-(dimethylamino)tetralin trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2(lH)-pyrimidinone trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinone trans-2-(2-phenylcyclopropyl)imidazoline trans-2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-5-(3,4-difluorobenzyl)piperidine trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperid-1-yl] indan-1-01 trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) piperid-1-yl] 6-nitroindan-1-01 trans-3-(2-(1-(4-(1-Naphthalenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((1-Naphthalenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((3-(2,6-Difluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(2-(4-Methyloxazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(2-(5-Methyloxazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzaze... trans-3-(2-(4-((3-(2-(5-Methyloxazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(2-Cyanophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepi... trans-3-(2-(4-((3-(2-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazep... trans-3-(2-(4-((3-(2-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benza... trans-3-(2-(4-((3-(2-Methoxyphenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(2-pyrimidinyl)phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((3-(3,5-Difluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))phenyl)-carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1... trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H... trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro... trans-3-(2-(4-((3-(3-Cyanophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepi... trans-3-(2-(4-((3-(3-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazep... trans-3-(2-(4-((3-(3-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benza... trans-3-(2-(4-((3-(3-Methoxyphenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(4-Cyanophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepi... trans-3-(2-(4-((3-(4-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazep... trans-3-(2-(4-((3-(4-Fluorophenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benza... trans-3-(2-(4-((3-(4-Methoxyphenyl)prop-2-enyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(5-(1-Methylpyrazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzaz... trans-3-(2-(4-((3-(5-(2-Methyloxazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzaze... trans-3-(2-(4-((3-(5-(2-Methyloxazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(2-(4-((3-(5-(3-Methylisoxazolyl))phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benza... trans-3-(2-(4-((3-(N-Pyrrolyl)phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((4-(2-Methylquinolinyl))carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((5-(2-Methylquinolinyl))carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((5-(2-Methylquinolinyl))carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-((5-(8-Fluoro-2-methylquinolinyl))carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzaz... trans-3-(2-(4-((5-Quinolinyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benzazepine trans-3-(2-(4-(3-(5-(3-Methylisoxazolyl)phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyloxy-2,3,4,5-tetrahydro-1H-3-benz... trans-3-(4-(6-(3-fluoropropoxy)-3,4-dihydroisoquinolin-2(1H)-yl)cyclohexyl)-1H-indole-5-carbonitrile trans-3-aminocyclopentane-1-carboxylic acid,(+/-) trans-4-aminocrotonic acid trans-azetidine-2, 4-dicarboxylate trans-Clopenthixol trans-H2-PAT(+) trans-H2-PAT(+/-) trans-H2-PAT(-) trans-methyl-{1-[3-(pyridin-3-yloxy)-propenyl]-cyclopropyl}-amine; hydrochloride trans-N, N-Dimethylphenylcyclopropylamine trans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine trans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine trans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine trans-N-Benzyl-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1′-cyclohexan]-4′-amine trans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine trans-N-Benzyl-3-methoxy-N-methyl-3,4-dihydrospiro-[[2]benzopyran-1,1′-cyclohexan]-4′-amine trans-N-Methyl-2'-methyl-2',3'-dihydrofuro[m]aporphine trans-N-Methylphenylcyclopropylamine trans-PAT trans-Thiothixene TRANYLCYPROMINE Tranylcypromine,(+) Tranylcypromine,(-) TRAZODONE Tremorine, oxo- Treprostinil Trequinsin TRH Triacin-C Triamcinolone (Fluoxyprednisolone) Triazolam Triazoledione Triciribine Tricyclo[3.3.1.1-3,7]dec-1- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate Tricyclo[3.3.1.1-3,7]dec-1-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoeth... Tricyclo[3.3.1.1-3,7]dec-2- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate Tricyclo[3.3.1.1-3,7]dec-2-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoeth... Tridesilon Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane TRIFLUOPERAZINE Trifluopromazine trifluoromethanesulfonate-norchloro-epibatidine TRIFLUORPERIDOL Trifluperazine Trifluperidol Triflupromazine Trihexyphenidyl Trimeprazine Trimethaphan Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane trimethyl({20-[(trimethylazaniumyl)methyl]-3,13-diazapentacyclo[11.7.0.0^{3,11}.0^{4,9}.0^{14,19}]icosa-1(20),4,6,8,10,14(19)... trimethyl-(4-quinolin-6-yl-but-3-ynyl)-ammonium iodide Trimipramine Tripelennamine TRIPITRAMINE Triprolidine Triton,(+) Triton,(-) TRK-820 TROHNBn TROMeNBn Tropanyl-3,5 dichlorobenzoate TROPICAMIDE TROPISETRON TRYPTAMINE TRYPTAMINE, 2,N,N-TRIMETHYL TRYPTAMINE, 4-METHOXY-N,N-DIMETHYL TRYPTAMINE, 5-HYDROXY-N,N-DIMETHYL tryptamine, 5-Methoxy Tryptamine, 5-methoxy-2me TRYPTAMINE,5-MeO,a- TRYPTAMINE,a-Me TRYPTAMINE,a-Me(+) TRYPTAMINE,a-Me(-) TRYPTAMINE,a-MeISO tryptophol, 5-Methoxy Tryptophol,5-Methoxy TS-011 Tuaminoheptane Tubocurarine Tubocurarine,d TXA2 Tyr-Asn-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-d-Ala-Phe-Phe-NH2 Tyr-d-Arg-Phe-A2pr-NH2 Tyr-d-Arg-Phe-Orn-NH2 Tyr-D-Asn-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-D-Lys-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-D-Met-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-D-Ser-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-lys-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-Met-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-Ser-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys-Dynorphin A (1-13) Tyr-tic-phe-phe-OH Tyr-W-Mif 1 Tyr10-cortistatin Tyr10-CST Tyr36-PTHrP(1-36) Tyramine Tyramine, m Tyramine, p U-101387 U-47700 U-50488H U-75302 U-97018 U-II (H-Glu-Thr-Pro-Asp-cyclo[Cys-Phe-Trp-Lys-Tyr-Cys]-Val-OH) U44069 U46619 U50,488 U50,488H U69,593 UB-165 UB-165 (+_) ucb 29992, (R) ucb 29993, (S) UCL 1684 UCL-1848 Ucn,r UF-021 UH232 UH232(+) UK-14,304 UK14304 UKH-1114 Ultracet UMB58 UMB68 UMB75 UPF 523 UR-AK22 UR-AK24 UR-AK26 UR-AK41 UR-AK46 UR-AK49 UR-AK51 UR-AK57 UR-AK59 UR-AK62 UR-AK64 UR-AK67 UR-AK68 URAPIDIL Urapidil-5-methyl URB 597 Uridine Urocortin Urotensin I, sf UTP V V105A Val-D-Pro-NHBu VALDECOXIB valeryl salicylate Valium Vanoxerine Vapreotide vardenafil varenicline Varenicline Vasoactive intestinal polypeptide Vasocidin Vatalanib Vecuronium Venlafaxine VER-3323 VER-5384 VER-5593 VERAPAMIL Verdeso VI vicenin-2 VII VIII Vilazodone Viloxazine Vinblastine Vinpocetine vip VIP Ala1 VIP Ala10 VIP Ala11 VIP Ala12 VIP Ala13 VIP Ala14 VIP Ala15 VIP Ala16 VIP Ala17 VIP Ala19 VIP Ala2 VIP Ala20 VIP Ala21 VIP Ala22 VIP Ala23 VIP Ala24 VIP Ala25 VIP Ala26 VIP Ala27 VIP Ala28 VIP Ala3 VIP Ala5 VIP Ala6 VIP Ala7 VIP Ala8 VIP Ala9 VIP [D- Ala18] VIP [D- Arg14] VIP [D- Asn24] VIP [D- Asn28] VIP [D- Gln16] VIP [D- Ile26] VIP [D- Leu23] VIP [D- Leu27] VIP [D- Lys15] VIP [D- Lys20] VIP [D- Lys21] VIP [D- Met 17] VIP [D- Ser25] VIP [D- Tyr22] VIP [D- Val19] VIP [D-Ala18] VIP [D-Ala4] VIP [D-Arg12] VIP [D-Arg14] VIP [D-Asn24] VIP [D-Asn28] VIP [D-Asn9] VIP [D-Asp3] VIP [D-Asp8] VIP [D-Gln16] VIP [D-His1] VIP [D-Ile26] VIP [D-Leu13] VIP [D-Leu23] VIP [D-Leu27] VIP [D-Lys15] VIP [D-Lys20] VIP [D-Lys21] VIP [D-Met17] VIP [D-Phe6] VIP [D-Ser25] VIP [D-Ser2] VIP [D-Thr11] VIP [D-Thr7] VIP [D-Tyr10] VIP [D-Tyr22] VIP [D-Val19] VIP [D-Val5] VIP(2-28) VIP(3-28) VIP(4-28) VIP-PACAP voacangine Vortioxetine VUF4614 VUF4616 VUF4617 VUF4681 VUF4682 VUF4683 VUF4686 VUF4687 VUF4742 VUF4903 VUF4904 VUF5202 VUF5207 VUF5300 VUF8328 VUF9153 VX-745 W104A WA-13 WAY 100,135 WAY 100,635 WAY 211686 WAY 212922 WAY 213394 WAY 213613 WAY 629 WAY-100635 WAY-855 WAY-865 WAY-879 WB 4101 WDYMVm-NH2 WEB2086 WEYMVm-NH2 WF-23 WF-31 WF-60 WHYMVm-NH2 WIN 35,065-2 WIN 35,428 WIN 44,441(-) WIN 52664 WIN 53024 WIN 53782 WIN 55,212-2 WIN 55212-2 WIN, 55-212 WKDMVm-NH2 WKEMVm-NH2 WKFMVm-NH2 WKHMVm-NH2 WKWMVm-NH2 WKYM(F/W)m-NH2 WKYMVm-NH2 WKYMYm-NH2 WRYMVm-NH2 WY 26392 WY 27127 WY 47384 WY-45030 WY-45651 WY-45655 WY-A-99-2 WY-B-08 WY-B-09-1 WY-B-14 WY-B-15 WY-B-20 WY-B-23-1 WY-B-23-2 WY-B-25 WY-B-26-2 WY-B-27-2 WY-B-99-1 WY-B-99-2 WY-S-2 WY-S-6 WY-TSC-4 WY-TSC-4 (WYS8) WY26703 WYB14 WYB27-1 WYB27-2 WYB29-2 WYS10 WYS10 C14H9F3N2O2 WYS12 WYS13 WYS13-C20H18N2O3 WYS15 WYS15 C22H20N2O2 WYS19 WYS8 WYS9 WYSC1 WYSC2 WYSCI C16H16N2O2 WZ-069 WZ-070 WZ-113 X XAC xanomeline Xanthine Xanthine Amine Congener Xanthosine Xenopus NMB XHE-I-037B (S-enriched) XHE-I-038 XHE-I-051 XHE-I-065 XHE-I-093 XHE-II-002 XHE-II-006a XHE-II-006b XHE-II-011 XHE-II-012 XHE-II-017 XHE-II-024 XHE-II-053 XHE-II-053-ACID XHE-II-065 XHE-II-073A (R Enriched) XHE-II-073B (S enriched) XHE-II-073B (S-ENRICHED) XHE-II-13 XHE-II-73A (R ENRICHED) XHE-II-O53-ACID XHE-III-04 XHE-III-06a XHE-III-06b XHE-III-13 XHE-III-14 XHE-III-24 XHE-III-49 XHE-III-74 XI XII XIII XLI-093 XLI-210 XLI-286 XLI-2TC XLI-317 XLI-347 XLI-348 XLi-350 C17H11ClN2O XLi-356 XLI-381 XLI-8TC XLi-JY-DMH ANX3 XLi-JY-DMH-ANX3 XLi093 XLi223 XLi223 C22H20BrN3O2 XLi268 XLi268 C17H13BrN4 Xli269 XLi270 XLi343 XLi343 C20H19ClN2OSi XLi350 XLi350 C17H11ClN2O XLi351 XLi351 C21H21ClN2OSi XLi352 XLi352 C18H13ClN2O XLi356 Xli366 Xorphanol XVI XYLAMIDINE Xylazine Xylometazoline Y-27632 Y-931 Y331A YAGEINE YaGF-NH2 YCT-5 YCT-7A YGGFMRF-amide YM 11170 YM-09151-2 YM-09538 YM022 YM087 YM12167 YM348 YM580 YM796 YM796(+) YM796(-) YM90k YMVm-NH2 YNT-1369 YNT-707 YNT-816 YNT-817 YOHIMBINE Yohimbine Hydrochloride YT-5 YT-6 YT-I-38 YT-II YT-II-76 YT-II-83 YT-III-23 YT-III-231 YT-III-25 YT-III-271 YT-III-272 YT-III-31 YT-III-38 YT-III-42 YT-TC-3 Z-Tyr-D-Ala-Gly-Phe-NH-NH-Phe-Asp-NMeNle-D-Trp-Boc ZACOPRIDE ZACOPRIDE,R ZACOPRIDE,RS ZACOPRIDE,S Zafirlukast Zalcitabine Zaleplon Zaprinast ZD 6169 ZD-6474 ZD6021 ZG 234 ZG 63 ZG-168 ZG-208 ZG-213 ZG-224 ZG-234 ZG-63A ZG-69a (Ro15-1310) ZG69A Zidovudine Zimeldine ZIMELIDINE Zimelidine (E-isomer) Zimelidine (Z-isomer) Ziprasidone ZK 91296 ZK 93423 ZK110841 ZK118182 ZM 241385 ZM-241385 ZM241385 zm244085 ZM253,270 Zolpidem Zomepirac zopolrestat ZOTEPINE ZP120 [ (R)-Atc4 ,D-Ala8]Dyn A-(1-11)NH2 [ (S)-Atc4 , D-Ala8]Dyn A-(1-11)NH2 [ (S)-Atc4 ,D-Ala8]Dyn A-(1-11)NH2 [ D-Ala8]Dyn A-(1-11)NH2 [ D-Phe4 ,D-Ala8]Dyn A-(1-11)NH2 [(1‐cyclohexylpiperidin‐4‐yl)methyl](2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)a... [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1R,2R,6R,10S,11R,15S,17R)-13-benzyl-6-hydroxy-4,17-dimethyl-5-oxo-15-(prop-1-en-2-yl)-12,14,18-trioxapentacyclo[11.4.1.0^{1... [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34,F35]-h-alpha-CGRP 8-37 [(20-{[dimethyl(prop-2-en-1-yl)azaniumyl]methyl}-3,13-diazapentacyclo[11.7.0.0^{3,11}.0^{4,9}.0^{14,19}]icosa-1(20),4,6,8,10,... [(3S)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl]-pyridin-2-ylmethanone [(4-Amino)-D-Phe1-(3-iodo)-Tyr3-Thr8] [(4-Amino)-D-Phe1-Asp8] [(4-Amino)-D-Phe1-D-Asp8] [(4-Amino)-D-Phe1-D-Thr8] [(4-Amino)-D-Phe1-Thr8] [(4-Amino-3-iodo)-D-Phe1-(3-iodo)-Tyr3-Asp8] [(4-Amino-3-iodo)-D-Phe1-(3-iodo)-Tyr3-Thr8] [(4-Amino-3-iodo)-D-Phe1-Asp8] [(4-Amino-3-iodo)-D-Phe1-Thr8] [(5-methyl-1H-imidazol-4-yl)methyl]-N-[(5-methylthiophen-2-yl)methyl]prop-2-en-1-amine [(5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol [(8-{[2,6-Dichloro-3-(methyl{[((2E)-3-{4-[(methylamino)-carbonyl]phenyl}-2-propenoyl)amino]acetyl}amino)benzyl] [(8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one [(E)-3-amino-1-propenyl]phosphinic acid [(R)-Atc4D-Ala8] Dyn A (1-11) NH2 [(S)-Atc4D-Ala8] Dyn A (1-11) NH2 [1-(1,2-Dimethyl-1H-imidazole-4-sulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid [1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]naphthalen-1-ylmethanone [1-(1-phenoxypropan-2-yl)piperidin-3-yl]-pyridin-3-ylmethanone [1-(2,5-Dichloro-benzenesulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid [1-(2-Chloro-2-phenyl-ethyl)-6-methylsulfanyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-(2-ethoxy-ethyl)-amine [1-(4-Chloro-benzenesulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid [1-(4-Methyl-benzyl)-piperidin-4-yl]-diphenyl-methanol [1-(5-bromo-pyridin-3-yloxymethyl)-cyclopropyl]-dimethyl-amine; hydrochloride [1-(Butane-1-sulfonyl)-5-fluoro-2-methyl-1H-indol-3-yl]-acetic acid [1-[2(methylsulphonylamino)ethyl]4-piperidinyl]methyl-1-methyl-indole-3-carboxylate [1-[2(methylsulphonylamino)ethyl]4-piperidinyl]methyl-5-fluoro-2-methoxy-1-H--indole-3-carboxylate [11C]CUMI [11C]MMP [125I]1-(2-iodophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxylate [125I]Iodopindolol [18F]MH.MZ [2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate [2-(4-Phenylpiperazin-1-yl)ethyl]pyrimido[5,4-c]quinolin-4(3H)-one [2-(5-methoxy-1H-indol-3-yl)ethyl]urea [2-(5-Methoxyindol-3-yl)ethyl]dimethylazan [22(R)-hydroxycholesterol [3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine [3-(2,2-Diphenylethylsulfanylmethyl)benzofuran-7-yloxy]acetic Acid [3-(2-Benzhydrylsulfanylethyl)-2-hydroxymethylbenzofuran-7-yloxy]acetic Acid [3-(2-Benzhydrylsulfanylethyl)benzofuran-7-yloxy]acetic Acid [3-(2-Chloro-6-methylamino-purin-9-yl)-2-phosphonomethyl-propyl]-phosphonic Acid [3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine [3-(3,3-Diphenylpropylsulfanylmethyl)benzofuran-7-yloxy]acetic Acid [3-(3-Benzhydrylsulfanylpropyl)benzofuran-7-yloxy]acetic Acid [3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-[4-(1,1-dioxothiomorpholinyl)methylene]-4-chlorobenzenesulfonamide [3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-{[2-(dimethylamino)ethylpiperazin-4-yl]methylene}-4-chlorobenzenesu... [3-Amino-1(R,S)-(trifluoromethyl)propyl]methylphosphinic acid [3-Amino-2(R,S)-(4-chlorophenyl)-2-hydroxypropyl]m-ethylphosphinic Acid [3-Amino-2(R,S)-(4-chlorophenyl)-2-hydroxypropyl]n-butylphosphinic Acid [3-Amino-2(R,S)-(4-chlorophenyl)propyl](diethoxymethyl)phosphinic Acid [3-Amino-2(R,S)-(4-chlorophenyl)propyl]methylphosphinic Acid [3-Benzhydrylsulfanylmethylbenzofuran-7-yloxy]acetic Acid [3-cyclohexyl-N-[3-(1H-imidazol-1-yl)propyl] propanic amide] [3-[2-(1,1-Diphenylbutylsulfanyl)ethyl]-2-hydroxymethylbenzofuran-7-yloxy]acetic Acid Sodium Salt [3-[2-(1,1-Diphenylethylsulfanyl)-ethyl]-2-(2-hydroxyethyl)benzofuran-7-yloxy]acetic Acid [3-[2-(1,1-Diphenylethylsulfanyl)ethyl]-2-(3-hydroxypropyl)benzofuran-7-yloxy]acetic Acid [3-[2-(1,1-Diphenylethylsulfanyl)ethyl]-2-hydroxymethylbenzofuran-7-yloxy]acetic Acid [3-[2-(1,1-Diphenylpropylsulfanyl)ethyl]-2-hydroxymethylbenzofuran-7-yloxy]acetic Acid Sodium Salt [3H] LSD [3H]N-methylspiperone [4-(2-Chloro-6-methylamino-purin-9-ylmethyl)-7-phosphono-heptyl]-phosphonic Acid, Sodium Salt [4-(3-Pyridylethynyl)-2-thiazolyl]carbamic Acid Methyl Ester [5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine [5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine [5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine [5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]carbamic acid 2-(1H-indol-3-yl)ethyl Ester [5-Fluoro-1-(3-fluoro-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid [5-Fluoro-1-(4-fluoro-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic-acid [5-Fluoro-1-(4-methoxy-benzenesulfonyl)-2-methyl-1H-indol-3-yl]-acetic acid [5-Fluoro-2-methyl-1-(4-methanesulfonyl-benzenesulfonyl)-1H-indol-3-yl]-acetic acid [5-Fluoro-2-methyl-1-(toluene-4-sulfonyl)-1H-indol-3-yl]-acetic acid [6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]carbamic acid 2-(1H-indol-3-yl)ethyl ester [6-Iodo-1-(1-methylpiperidin-2-ylmethyl)-1H-indol-3-yl]naphthalen-1-ylmethanone [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]carbamic acid 2-(1H-indol-3-yl)ethyl ester [7-Chloro-9-(4-methyl-1-piperazinyl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepin-1-yl]methanol [9-(4-Methyl-1-piperazinyl)pyrrolo[2,1-b][1,3]benzothiazepin-1-yl]methanol [a,d]dibenz-fused cycloheptane [a-MePhe4D-Ala8] Dyn A (1-11) NH2 [A27]CGRP 27-37 [A28]CGRP Y0-28-37 [A29,D31,p34,F35]-h-alpha-CGRP 27-37 [A31]CGRP Y0-28-37 [A34]CGRP Y0-28-37 [A35]CGRP Y0-28-37 [a36]CGRP Y0-28-37 [AcHis1,DPhe2]PACAP(1-27) [AcHis1,DPhe2]PACAP(1-38) [AcHis1,Phe2]PACAP(1-27) [AcHis1,Phe2]PACAP(1-38) [AcHis1]PACAP(1-27) [Aib29,D31,p34,F35]-h-alpha-CGRP 27-37 [Aic4D-Ala8] Dyn A (1-11) NH2 [ala1,leu13]pMOT(1-14) [ala10,leu13]pMOT(1-14) [ala11,leu13]pMOT(1-14) [ala12,leu13]pMOT(1-14) [ala13,leu13]pMOT(1-14) [ala14,leu13]pMOT(1-14) [Ala2]PACAP(1-27) [Ala2]PACAP(1-38) [ala3,leu13]pMOT(1-14) [Ala37]h alpha-CGRP8-37 [ala4,leu13]pMOT(1-14) [ala5,leu13]pMOT(1-14) [ala6,leu13]pMOT(1-14) [ala7,leu13]pMOT(1-14) [ala8,leu13]pMOT(1-14) [ala9,leu13]pMOT(1-14) [Arg2]PACAP(1-27) [Arg2]PACAP(1-38) [Asn3]PACAP(1-27) [Bpa5,Ile13]Motilin [C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline [C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline [C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline [C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline [C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline [C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline [Cha37]h alpha-CGRP8-37 [Cys(ACM)2,7]h alpha-CGRP [D-Ala2, Leu5] enkephalin amide [D-Ala2-D-Leu5]enkephalin [D-Ala8] Dyn A-(1-11)NH2 [D-Ala8]Dyn A (1-11) NH2 [D-Arg25, D-His26]-NPY [D-Arg25]-NPY [D-Bpa5,Ile13]Motilin [D-His25]-NPY [D-His26]-NPY [D-Homophe4 D-Ala8] Dyn A (1-11) NH2 [D-Pen2,7]h alpha-CGRP [D-Phe1-Asp8] [D-Phe2]PACAP-27 [D-Phe2]PACAP-38 [D-Phe4 , D-Ala8]Dyn A-(1-11)NH2 [D-Phe4D-Ala8] Dyn A (1-11)NH2 [D-Phe4D-Ala8] Dyn A (1-11) NH2 [D-Pro4]morphiceptin [D-Tyr6,(R)-Apa11,Phe13,Nle14]Bn(6-14) [D-Tyr6,(R)-Apa11-2Cl,Phe13,Nle14]Bn(6-14) [D-Tyr6,(R)-Apa11-3Cl,Phe13,Nle14]Bn(6-14) [D-Tyr6,(R)-Apa11-4Cl,Phe13,Nle14]Bn(6-14) [D-Tyr6,(S)-Apa11,Phe13,Nle14]Bn(6-14) [D-Tyr6,(S)-Apa11-2Cl,Phe13,Nle14]Bn(6-14) [D-Tyr6,(S)-Apa11-3Cl,Phe13,Nle14]Bn(6-14) [D-Tyr6,(S)-Apa11-4Cl,Phe13,Nle14]Bn(6-14) [D-Tyr6,Beta-Ala11,Phe13,Beta-Dap(Pr)14]Bn(6-14) [D-Tyr6,Beta-Ala11,Phe13,Nle14]Bn(6-14) [D-Tyr6,Beta-Asp(BzlAmd)11,Phe13,Nle14]Bn(6-14) [D-Tyr6,Beta-Asp11,Phe13,Nle14]Bn(6-14) [D-Tyr6,Beta-Dap11,Phe13,Nle14]Bn(6-14) [D-Tyr6,NAlpha-acetyl-Dap11,Phe13,Nle14]Bn(6-14) [D-Tyr6,NAlpha-benzoyl-Dap11,Phe13,Nle14]Bn(6-14) [D31,(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 [D31,(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34,F35]-h-alpha-CGRP 27-37 [D31,(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 [D31,(1S,2S,3S)-beta-aminocyclopropane carboxylic acid, F35]-h-alpha-CGRP 8-37 [D31,A34,F35]-h-alpha-CGRP 27-37 [D31,A34,F35]CGRP 27-37 [D31,A34,F35]CGRP 28-37 [D31,A34,F35]CGRP 29-37 [D31,A34,F35]CGRP Ac-27-37 [D31,A34,F35]CGRP Ac-28-37 [D31,A34,F35]CGRP Ac-29-37 [D31,A34,H35]CGRP 27-37 [D31,Acp34,F35]CGRP 27-37 [D31,Aib34,F35]CGRP 27-37 [D31,Hop34,F35]CGRP 27-37 [D31,Hyp34,F35]CGRP 27-37 [D31,p34,F35]-h-alpha-CGRP 27-37 [D31,P34,F35]CGRP 27-37 [D31,P34]CGRP 27-37 [D31,Pac34,F35]CGRP 27-37 [D31,Q35]CGRP 27-37 [D31,Tic34,F35]-h-alpha-CGRP 27-37 [D31,Tic34,F35]CGRP 27-37 [D31]CGRP 27-37 [D31]CGRP Y0-28-37 [DAla2]PACAP(1-27) [DAla2]PACAP(1-38) [DArg2]PACAP(1-27) [DArg2]PACAP(1-38) [Des-His1,Asn3]PACAP-27 [Des-His1,Glu3]PACAP-38 [Dmt1]DALDA [DPhe2]PACAP(1-27) [DPhe2]PACAP(1-38) [F28]CGRP Y0-28-37 [F29]CGRP Y0-28-37 [F31]CGRP Y0-28-37 [F35]CGRP Y0-28-37 [G36]CGRP Y0-28-37 [H35]CGRP Y0-28-37 [His5,D-Tyr6]GnRH [Homophe4 D-Ala8] Dyn A (1-11) NH2 [Hop29,D31,p34,F35]-h-alpha-CGRP 27-37 [Hyp29,D31,p34,F35]-h-alpha-CGRP 27-37 [Hyp29]CGRP Y0-28-37 [K35]CGRP 27-37 [K35]CGRP Y0-28-37 [L-Bpa5,Ile13]Motilin [L31]CGRP Y0-28-37 [L35]CGRP Y0-28-37 [Leu13]motilin [leu13]pMOT(1-11) [leu13]pMOT(1-14) [leu13]pMOT(1-16) [leu13]pMOT(1-19) [leu13]pMOT(1-22) [leu13]pMOT(1-5) [leu13]pMOT(1-7) [leu13]pMOT(1-9) [Lys15, Arg16, Leu27]VIP(1-7)GRF(8-27) [Mox3,6]-CCK8 [Mox3]-CCK8 [Mox6]-CCK8 [N-acetyl]h alpha-CGRP8-37 [N-benzol]h alpha-CGRP8-37 [N-MePhe4D-Ala8] Dyn A (1-11) NH2 [n31]CGRP Y0-28-37 [Nle13]-Motilin [NLeu2]-CCK4 [P28]CGRP 27-37 [p29]CGRP Y0-28-37 [P30]CGRP 27-37 [P31]CGRP 27-37 [P32]CGRP 27-37 [P33]CGRP 27-37 [P34]CGRP 27-37 [P35]CGRP 27-37 [P36]CGRP 27-37 [Phe13,Tyr19]-MCH [Phe13,Tyr19]MCH [Phe1]PACAP(1-27) [Phe1]PACAP-27 [Phe1]VIP [Phe2]PACAP(1-27) [Phe2]PACAP(1-38) [Pro14]h alpha-CGRP [Pro34,Phe35]h alpha-CGRP27-37 [propionyl-K24]-h-alpha-CGRP 8-37 [Q31]CGRP Y0-28-37 [Q35]CGRP Y0-28-37 [S30]CGRP Y0-28-37 [s34]CGRP Y0-28-37 [Ser9,Tyr13]VIP [Ser9]VIP [Tic29,D31,p34,F35]-h-alpha-CGRP 27-37 [Tic4D-Ala8] Dyn A (1-11) NH2 [Tyr13]VIP [v28]CGRP Y0-28-37 [Y37]CGRP Y0-28-37 [[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-... {(3-Phenylpropionyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid {(3-Phenylpropionyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester {(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester {1-[4-(1-Pyrrolidinyl)-2-butynyl]-2-pyrrolidinone} {2-Hydroxymethyl-3-[2-(2,2,2-trifluoro-1,1-diphenylethylsulfanyl)ethyl]benzofuran-7-yloxy}acetic Acid {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(2-nitrophenyl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(3-nitropyridin-2-yl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitropyridin-2-yl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitrothiazol-2-yl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrazin-2-ylamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-2-ylamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-5-ylamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(2-nitrophenyl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(3-nitropyridin-2-yl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-trifluoromethylpyridin-2-yl)amine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrazin-2-ylamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-2-ylamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-5-ylamine {2-[2-(2-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(4-nitrophenyl)amine {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate {2-[3-(Phenylsulfonyl)-1H-indol-4-yl]ethyl}amine {2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indol-7-yl}azinic acid {3-[(2-adamantan-1-yl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-dimethyl-amine {3-[2-(1,1-Diphenylethylsulfanyl)ethyl]benzofuran-7-yloxy}acetic Acid {3-[2-(2,2-Diphenylethylsulfanyl)ethyl]benzofuran-7-yloxy}acetic Acid {3-[2-(3,3-Diphenylpropylsulfanylmethyl)ethyl]benzofuran-7-yloxy}acetic Acid {3-[2-(Diphenylethanesulfinyl)ethyl]-2-hydroxymethylbenzofuran-7-yloxy}acetic Acid {3-[2-(Diphenylethanesulfonyl)ethyl]-2-hydroxymethylbenzofuran-7-yloxy}acetic Acid {3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine {3-[3-(2,2-Diphenylethylsulfanyl)propyl]benzofuran-7-yloxy}acetic Acid {3-[3-(3,3-Diphenylpropylsulfanyl)propyl]benzofuran-7-yloxy}acetic Acid {4-[Bis(2-bromoethyl)amino]-2,3,5,-trifluorobenzoyl}-L-glutamic Acid {4-[Bis(2-bromoethyl)amino]-3,5-difluorobenzoyl}-L-glutamic Acid {4-[Bis(2-chloroethyl)amino]-2,3,5,-trifluorobenzoyl}-L-glutamic Acid {4-[Bis(2-chloroethyl)amino]-2,3,5,6-tetrafluorobenzoyl}-L-glutamic Acid {4-[Bis(2-chloroethyl)amino]-3,5-difluorobenzoyl}-L-glutamic acid {4-[Bis(2-iodoethyl)amino]-2,3,5,-trifluorobenzoyl}-L-glutamic Acid {4-[Bis(2-iodoethyl)amino]-2,3,5,6-tetrafluorobenzoyl}-L-glutamic Acid {5-Amino-3-[4-(piperidine-1-sulfonyl)-phenylamino]-[1,2,4]triazol-1-yl}-(2,6-difluorophenyl)-methanone {Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid {Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester {[20-({dimethyl[(4-nitrophenyl)methyl]azaniumyl}methyl)-3,13-diazapentacyclo[11.7.0.0^{3,11}.0^{4,9}.0^{14,19}]icosa-1(20),4,... {[5-(2,2,2-Trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-4,5-dihydro-isoxazole-3-carbonyl]-amino}-acetic acid ethyl ester

Compound List: