The database has 98685 Ki values for searching, and is growing. This list shows the Top 100 Receptors/Targets in Ki Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments. Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity. Anatomical profiling of GPCR expression is offered for selected targets.


Make a new search

Your search returned 65 results:

Download Data
IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEBIHot Ligand/AliasesSpeciesSourceReference
258 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 119.510000 PubChem-Compound N/A 3H-8-OH-DPAT  Aliases HUMAN CORTEX PIERCE & PEROUTKA, 1989
 
83205 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 450.000000 PubChem-Compound N/A 3H-8-OH-DPAT  Aliases HUMAN CLONED Janowsky A et al 2014
 
261 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 245.000000 PubChem-Compound N/A 3H-8-OH-DPAT  Aliases RAT CORTEX TAYLOR ET AL,. 1987
 
260 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 140.740000 PubChem-Compound N/A 3H-8-OH-DPAT  Aliases BOVINE HIPPOCAMPUS PEROUTKA, 1985
 
78869 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-WAY100635  Aliases HUMAN CLONED Ray TS 2010
 
1012 5-HT1B  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 2,200.000000 PubChem-Compound N/A 125I-CYP  Aliases RAT CORTEX OFFORD ET AL., 1988
 
78902 5-HT1B  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-5-CT  Aliases HUMAN CLONED Ray TS 2010
 
78933 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 93.000000 PubChem-Compound N/A 3H-5-CT  Aliases HUMAN CLONED Ray TS 2010
 
1259 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 270.000000 PubChem-Compound N/A 3H-5HT  Aliases HUMAN CORTEX PEROUTKA ET AL., 1989
 
1260 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 342.860000 PubChem-Compound N/A 3H-5HT  Aliases BOVINE STRIATUM PEROUTKA, 1985
1258 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 190.000000 PubChem-Compound N/A 3H-5HT  Aliases BOVINE STRIATUM HEURING & PEROUTKA, 1987
Average266.43 
1257 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 71.380000 PubChem-Compound N/A 3H-5HT  Aliases COW CAUDATE PIERCE & PEROUTKA, 1989
 
78966 5-HT1E  Aliases NCBI - UniGene N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 455.700000 PubChem-Compound N/A 3H-5-HT  Aliases HUMAN CLONED Ray TS 2010
 
83227 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 53.000000 PubChem-Compound N/A 125I-DOI  Aliases HUMAN CLONED Janowsky A et al 2014
83204 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 210.000000 PubChem-Compound N/A 125I-DOI  Aliases HUMAN CLONED Janowsky A et al 2014
Average131.50 
50490 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 42.000000 PubChem-Compound N/A 125I-DOI  Aliases RAT CORTEX MCKENNA & PEROUTKA, 1989
 
1847 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 462.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases HUMAN CORTEX SADZOT ET AL., 1989
 
78998 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 2,323.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases HUMAN CLONED Ray TS 2010
83232 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 175.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases HUMAN CLONED Janowsky A et al 2014
Average1249.00 
1852 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 1,200.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases RAT CORTEX LYON ET AL., 1988
1851 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 1,200.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases RAT CORTEX LYON ET AL., 1988
1849 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 558.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases RAT CORTEX TAYLOR ET AL,. 1987
1850 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 1,183.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases RAT CORTEX LYON ET AL., 1987
Average1035.25 
1845 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 230.270000 PubChem-Compound N/A 3H-SPIPERONE  Aliases HUMAN CORTEX PIERCE & PEROUTKA, 1989
 
1848 5-HT2B  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 550.000000 PubChem-Compound N/A 3H-KETANSERIN  Aliases BOVINE CORTEX MCKENNA & PEROUTKA, 1989
 
79031 5-HT2B  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 107.600000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
83203 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 166.000000 PubChem-Compound N/A 125I-DOI  Aliases HUMAN CLONED Janowsky A et al 2014
 
79062 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 334.600000 PubChem-Compound N/A 3H-MESULERGINE  Aliases HUMAN CLONED Ray TS 2010
 
80048 5-HT3  Aliases NCBI - UniGene N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-GR-65630  Aliases HUMAN CLONED Ray TS 2010
 
79093 5-HT5a  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 611.000000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
79124 5-HT6  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 487.400000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
4349 5-HT6  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 68.000000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED KOHEN R, ET AL., 1996
Average277.70 
79155 5-HT7  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 87.500000 PubChem-Compound N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
79344 alpha1A  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 1,745.000000 PubChem-Compound N/A 3H-PRAZOSIN  Aliases HUMAN CLONED Ray TS 2010
 
79374 alpha1B  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 973.700000 PubChem-Compound N/A 3H-PRAZOSIN  Aliases HUMAN CLONED Ray TS 2010
 
79399 Alpha2A  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 1,561.000000 PubChem-Compound N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Ray TS 2010
 
79424 Alpha2B  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 257.700000 PubChem-Compound N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Ray TS 2010
 
79449 Alpha2C  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 258.600000 PubChem-Compound N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Ray TS 2010
 
79474 Beta 1  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 125I-Pindolol  Aliases HUMAN CLONED Ray TS 2010
 
79505 Beta 2  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-CGP12177  Aliases HUMAN CLONED Ray TS 2010
 
80284 BZP Rat Brain  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A FNZ  Aliases RAT CORTICAL MEMBRANES Ray TS 2010
 
80005 Calcium channel  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-Nitrendipine  Aliases HUMAN CLONED Ray TS 2010
 
79962 CB1  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-CP55940  Aliases HUMAN CLONED Ray TS 2010
 
79983 CB2  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-CP55940  Aliases HUMAN CLONED Ray TS 2010
 
79780 Cholinergic, muscarinic M1  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79806 Cholinergic, muscarinic M2  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79832 Cholinergic, muscarinic M3  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79856 Cholinergic, muscarinic M4  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79880 Cholinergic, muscarinic M5  Aliases NCBI - UniGene Anatomical Profiling N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79187 D1  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 271.100000 PubChem-Compound N/A 3H-SCH23390  Aliases HUMAN CLONED Ray TS 2010
 
79220 D2  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-N-Methylspiperone  Aliases HUMAN CLONED Ray TS 2010
 
79252 D3  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-N-Methylspiperone  Aliases HUMAN CLONED Ray TS 2010
 
79284 D4  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-N-Methylspiperone  Aliases HUMAN CLONED Ray TS 2010
 
79317 D5  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-SCH23390  Aliases HUMAN CLONED Ray TS 2010
 
79565 DAT  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-WIN 35,428  Aliases HUMAN CLONED Ray TS 2010
 
80182 GABA A  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-MUSCIMOL  Aliases RAT CORTICAL MEMBRANES Ray TS 2010
 
79937 H2  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 125I-aminopotentidine  Aliases HUMAN CLONED Ray TS 2010
 
80076 H3  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-Alpha-methylhistamine  Aliases HUMAN CLONED Ray TS 2010
 
80099 H4  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-Histamine  Aliases HUMAN CLONED Ray TS 2010
 
79626 Imidazoline 1  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 650.300000 PubChem-Compound N/A 3H-CLONIDINE  Aliases HUMAN CLONED Ray TS 2010
 
79722 KOR  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-U69593  Aliases HUMAN CLONED Ray TS 2010
 
79596 Norepinephrine transporter  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-Nisoxetine  Aliases HUMAN CLONED Ray TS 2010
 
79534 SERT  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 3,742.000000 PubChem-Compound N/A 3H-CITALOPRAM  Aliases HUMAN CLONED Ray TS 2010
 
79648 Sigma-1  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 5,209.000000 PubChem-Compound N/A 3H-Pentazocine(+)  Aliases HUMAN CLONED Ray TS 2010
 
79670 Sigma-2  Aliases N/A N/A N,N-DIMETHYLTRYPTAMINE  Aliases 63795 > 10,000.000000 PubChem-Compound N/A 3H-DTG  Aliases HUMAN CLONED Ray TS 2010