The database has 98685 Ki values for searching, and is growing. This list shows the Top 100 Receptors/Targets in Ki Please let us know if you feel we should add any papers or data. We welcome all feedback/suggestions/comments. Other features on Ki DB are: Download Ki, Data Mining, CDD Interface allows mining Ki database by structure, substructure or structure similarity. Anatomical profiling of GPCR expression is offered for selected targets.


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Your search returned 76 results:

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IDReceptor/AliasesUniGeneAnat. ProfilingTest Ligand Name/AliasesNCIKi (nM)PubChemChEBIHot Ligand/AliasesSpeciesSourceReference
89975 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 240.000000 N/A N/A 3H-8-OH-DPAT  Aliases HUMAN CLONED Rickli A et al 2015
94216 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 311.000000 N/A N/A 3H-8-OH-DPAT  Aliases HUMAN CLONED Kolaczynska KE et al 2019
Average275.50 
78868 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 240.800000 N/A N/A 3H-WAY100635  Aliases HUMAN CLONED Ray TS 2010
 
94057 5-HT1A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 311.000000 N/A N/A [3H]-8-OH-DPAT  Aliases HUMAN CLONED Luethi D et al 2018
 
78901 5-HT1B  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 104.400000 N/A N/A 3H-5-CT  Aliases HUMAN CLONED Ray TS 2010
 
78932 5-HT1D  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 26.300000 N/A N/A 3H-5-CT  Aliases HUMAN CLONED Ray TS 2010
 
78965 5-HT1E  Aliases NCBI - UniGene N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 119.500000 N/A N/A 3H-5-HT  Aliases HUMAN CLONED Ray TS 2010
 
90000 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 8.600000 N/A N/A 3H-KETANSERIN  Aliases HUMAN CLONED Rickli A et al 2015
78997 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 27.600000 N/A N/A 3H-KETANSERIN  Aliases HUMAN CLONED Ray TS 2010
94231 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 6.900000 N/A N/A 3H-KETANSERIN  Aliases HUMAN CLONED Kolaczynska KE et al 2019
Average14.37 
94073 5-HT2A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 6.900000 N/A N/A [3H]-ketanserin  Aliases HUMAN CLONED Luethi D et al 2018
 
79030 5-HT2B  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 13.500000 N/A N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
79061 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 89.500000 N/A N/A 3H-MESULERGINE  Aliases HUMAN CLONED Ray TS 2010
90025 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 47.000000 N/A N/A 3H-MESULERGINE  Aliases HUMAN CLONED Rickli A et al 2015
94246 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 43.000000 N/A N/A 3H-MESULERGINE  Aliases HUMAN CLONED Kolaczynska KE et al 2019
Average59.83 
94089 5-HT2C  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 43.000000 N/A N/A [3H]-mesulergine  Aliases HUMAN CLONED Luethi D et al 2018
 
80047 5-HT3  Aliases NCBI - UniGene N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-GR-65630  Aliases HUMAN CLONED Ray TS 2010
 
79092 5-HT5a  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
79123 5-HT6  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 319.900000 N/A N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
79154 5-HT7  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 209.500000 N/A N/A 3H-LSD  Aliases HUMAN CLONED Ray TS 2010
 
94291 adrenergic Alpha1A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 6,500.000000 N/A N/A 3H-PRAZOSIN  Aliases HUMAN CLONED Kolaczynska KE et al 2019
 
94306 adrenergic Alpha2A  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 15,000.000000 N/A N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Kolaczynska KE et al 2019
 
79343 alpha1A  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-PRAZOSIN  Aliases HUMAN CLONED Ray TS 2010
 
79373 alpha1B  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-PRAZOSIN  Aliases HUMAN CLONED Ray TS 2010
 
90075 Alpha2A  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 320.000000 N/A N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Rickli A et al 2015
79398 Alpha2A  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 308.800000 N/A N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Ray TS 2010
Average314.40 
79448 Alpha2C  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 103.300000 N/A N/A 3H-RAUWOLSCINE  Aliases HUMAN CLONED Ray TS 2010
 
79473 Beta 1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 125I-Pindolol  Aliases HUMAN CLONED Ray TS 2010
 
79504 Beta 2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-CGP12177  Aliases HUMAN CLONED Ray TS 2010
 
80283 BZP Rat Brain  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A FNZ  Aliases RAT CORTICAL MEMBRANES Ray TS 2010
 
79961 CB1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-CP55940  Aliases HUMAN CLONED Ray TS 2010
 
79982 CB2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-CP55940  Aliases HUMAN CLONED Ray TS 2010
 
79779 Cholinergic, muscarinic M1  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79805 Cholinergic, muscarinic M2  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79831 Cholinergic, muscarinic M3  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 821.600000 N/A N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79855 Cholinergic, muscarinic M4  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79879 Cholinergic, muscarinic M5  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-QNB  Aliases HUMAN CLONED Ray TS 2010
 
79186 D1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-SCH23390  Aliases HUMAN CLONED Ray TS 2010
90099 D1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 12,000.000000 N/A N/A 3H-SCH23390  Aliases HUMAN CLONED Rickli A et al 2015
 
79219 D2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 3,371.000000 N/A N/A 3H-N-Methylspiperone  Aliases HUMAN CLONED Ray TS 2010
 
90124 D2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 2,200.000000 N/A N/A 3H-SPIPERONE  Aliases HUMAN CLONED Rickli A et al 2015
94321 D2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 25,200.000000 N/A N/A 3H-SPIPERONE  Aliases HUMAN CLONED Kolaczynska KE et al 2019
Average13700.00 
79251 D3  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 7,116.000000 N/A N/A 3H-N-Methylspiperone  Aliases HUMAN CLONED Ray TS 2010
 
90149 D3  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 10,000.000000 N/A N/A 3H-SPIPERONE  Aliases HUMAN CLONED Rickli A et al 2015
 
79283 D4  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-N-Methylspiperone  Aliases HUMAN CLONED Ray TS 2010
 
79316 D5  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-SCH23390  Aliases HUMAN CLONED Ray TS 2010
 
94352 DAT  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 6,500.000000 N/A N/A 3H-WIN 35,428  Aliases HUMAN CLONED Kolaczynska KE et al 2019
79564 DAT  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-WIN 35,428  Aliases HUMAN CLONED Ray TS 2010
90249 DAT  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 30,000.000000 N/A N/A 3H-WIN 35,428  Aliases HUMAN CLONED Rickli A et al 2015
 
79691 DOR  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-DADLE  Aliases HUMAN CLONED Ray TS 2010
 
80297 EP3  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-PGE2  Aliases HUMAN CLONED Ray TS 2010
 
80181 GABA A  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-MUSCIMOL  Aliases RAT CORTICAL MEMBRANES Ray TS 2010
 
90299 H1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 14,000.000000 N/A N/A 3H-PYRILAMINE  Aliases HUMAN CLONED Rickli A et al 2015
79905 H1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-PYRILAMINE  Aliases HUMAN CLONED Ray TS 2010
 
79936 H2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 125I-aminopotentidine  Aliases HUMAN CLONED Ray TS 2010
 
80075 H3  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-Alpha-methylhistamine  Aliases HUMAN CLONED Ray TS 2010
 
80098 H4  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-Histamine  Aliases HUMAN CLONED Ray TS 2010
 
79625 Imidazoline 1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 2,155.300000 N/A N/A 3H-CLONIDINE  Aliases HUMAN CLONED Ray TS 2010
 
79721 KOR  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-U69593  Aliases HUMAN CLONED Ray TS 2010
 
79752 MOR  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-DAMGO  Aliases HUMAN CLONED Ray TS 2010
 
80022 NMDA  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-MK-801  Aliases RAT CORTICAL MEMBRANES Ray TS 2010
 
90224 Norepinephrine transporter  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 31,000.000000 N/A N/A 3H-Nisoxetine  Aliases HUMAN CLONED Rickli A et al 2015
79595 Norepinephrine transporter  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-Nisoxetine  Aliases HUMAN CLONED Ray TS 2010
 
94336 Norepinephrine transporter  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 30,500.000000 N/A N/A n-methyl-[3h]nisoxetine  Aliases HUMAN CLONED Kolaczynska KE et al 2019
 
94367 SERT  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 13,300.000000 N/A N/A 3H-CITALOPRAM  Aliases HUMAN CLONED Kolaczynska KE et al 2019
79533 SERT  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-CITALOPRAM  Aliases HUMAN CLONED Ray TS 2010
90274 SERT  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 9,700.000000 N/A N/A 3H-CITALOPRAM  Aliases HUMAN CLONED Rickli A et al 2015
Average11500.00 
79647 Sigma-1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-Pentazocine(+)  Aliases HUMAN CLONED Ray TS 2010
 
79669 Sigma-2  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-DTG  Aliases HUMAN CLONED Ray TS 2010
 
94276 TAAR1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 2,400.000000 N/A N/A 3H-RO5166017  Aliases MOUSE CLONED Kolaczynska KE et al 2019
 
94261 TAAR1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 370.000000 N/A N/A 3H-RO5166017  Aliases RAT CLONED Kolaczynska KE et al 2019
 
90199 trace amine-associated receptor  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 3,000.000000 N/A N/A 3H-RO5166017  Aliases MOUSE CLONED Rickli A et al 2015
 
90174 trace amine-associated receptor  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A 90.000000 N/A N/A 3H-RO5166017  Aliases RAT CLONED Rickli A et al 2015
 
80121 VASOPRESSIN V1  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-VASOPRESSIN  Aliases HUMAN CLONED Ray TS 2010
 
80140 VASOPRESSIN V2  Aliases NCBI - UniGene Anatomical Profiling 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-VASOPRESSIN  Aliases HUMAN CLONED Ray TS 2010
 
80160 Vasopressin V3  Aliases N/A N/A 4-Bromo-2,5-dimethoxyphenethylamine  Aliases N/A > 10,000.000000 N/A N/A 3H-VASOPRESSIN  Aliases HUMAN CLONED Ray TS 2010