The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 48,001-49,000 of 98,686 items.

Kᵢ Database

Reset Grid
Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
50749DORHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50750HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50751HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50752H1HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP1030Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50753H2HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP2126Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50754H3HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50755H4HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50756hERGHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50757KORHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50758HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50759HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50760MORHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50761NMDAHIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 28, 2025
50762Sigma 2HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP123Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50763VMAT1HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50764NTSR1HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50765I1HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50766HIPPOCAMPUSBOVINE3H-8-OH-DPAT[11C]MMP>10000Kumar JS et al., 2007Jan 15, 2025Jan 15, 2025
50767SLC6A3UNDEFINEDHUMANUNDEFINEDMETHYLPHENIDATE110Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50768SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine23Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50769SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine16Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50770SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine7.8Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50771SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine46Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50772SLC6A3UNDEFINEDHUMANUNDEFINED(RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine11Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50773SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine37Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50774SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine180Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50775SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate25Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50776SLC6A3UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50777SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine3.7Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50778SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine36Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50779SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine400Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50780SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine440Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50781SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine24Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50782SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine440Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50783SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine130Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50784SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine9.4Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50785SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine120Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50786SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine3.6Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50787SLC6A3UNDEFINEDHUMANUNDEFINED1-phenyl-1-(piperidin-2-yl)propan-2-one370Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50788SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine3300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50789SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine22Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50790SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine52Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50791SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine6.6Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50792SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine1Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50793SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine2.3Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50794SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine0.97Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50795SLC6A3UNDEFINEDHUMANUNDEFINEDmethyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate1.4Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50796SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50797SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine510Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50798SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine870Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50799SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine170Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50800SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine290Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50801SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50802SLC6A3UNDEFINEDHUMANUNDEFINED(RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine380Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50803SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine1800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50804SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine3900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50805SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate2000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50806SLC6A3UNDEFINEDHUMANUNDEFINEDmethyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate90Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50807SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine140Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50808SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine690Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50809SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine5700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50810SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine2900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50811SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50812SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine550Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50813SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine260Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50814SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine310Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50815SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine6500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50816SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine950Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50817SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine770Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50818SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine44Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50819SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine31Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50820SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine29Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50821SLC6A3UNDEFINEDHUMANUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine43Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50822SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDMETHYLPHENIDATE>10000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50823SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine2200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50824SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine5900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50825SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine4300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50826SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine5300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50827SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine2700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50828SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine7800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50829SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine4900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50830SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate6000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50831SLC6A4UNDEFINEDUNDEFINEDUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester340Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50832SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine3200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50833SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine5700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50834SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine3900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50835SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50836SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine640Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50837SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine1100Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50838SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50839SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine2900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50840SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine3900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50841SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine5000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50842SLC6A4UNDEFINEDUNDEFINEDUNDEFINED1-phenyl-1-(piperidin-2-yl)propan-2-one7800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50843SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine3300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50844SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine4200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50845SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine2800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50846SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine1300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50847SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine1600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50848SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine1300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50849SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine1800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50850SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDmethyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate1600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50851SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine3500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50852SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine6700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50853SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine3600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50854SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine4300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50855SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine4800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50856SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine3200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50857SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine4200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50858SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine9100Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50859SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate5900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50860SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine>10000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50861SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine3200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50862SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine4600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50863SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine4800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50864SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine1500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50865SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine1800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50866SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine4300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50867SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine3700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50868SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine3200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50869SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine1700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50870SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine3800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50871SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine950Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50872SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine1500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50873SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine450Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50874SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine1100Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50875SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine450Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50876SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDmethyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate2500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50877SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDMETHYLPHENIDATE660Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50878SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine160Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50879SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine840Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50880SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine230Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50881SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine810Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50882SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50883SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine360Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50884SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine360Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50885SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate110Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50886SLC6A2UNDEFINEDUNDEFINEDUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50887SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine23Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50888SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine380Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50889SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine970Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50890SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine490Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50891SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine1800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50892SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine2900Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50893SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine4200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50894SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine1700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50895SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine1400Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50896SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine830Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50897SLC6A2UNDEFINEDUNDEFINEDUNDEFINED1-phenyl-1-(piperidin-2-yl)propan-2-one2700Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50898SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine2500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50899SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine3800Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50900SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine3100Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50901SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine190Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50902SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine25Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50903SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine12Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50904SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine3.9Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50905SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDmethyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate14Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50906SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3,3-dimethylbutyl]-piperidine5500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50907SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-methylpentyl]piperidine>10000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50908SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)hexyl]piperidine1500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50909SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]piperodine4500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50910SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)pentyl]piperidine1600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50911SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RS/SR)-2-[1-(4-chlorophenyl)butyl]piperidine1400Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50912SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)propyl]piperidine9200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50913SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-(1-(4-chlorophenyl)ethyl)piperidine6300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50914SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-methyl 2-(4-chlorophenyl)-2-(piperidin-2-yl)acetate6100Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50915SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-methylpropyl]piperidine>10000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50916SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-chlorophenyl)-3-methylbutyl]piperidine340Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50917SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[(4-chlorophenyl)cyclopentylmethyl]-piperidine3300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50918SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-ethylbutyl]piperidine4300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50919SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-4-phenylbutyl]piperidine1500Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50920SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-3-phenylpropyl]piperidine2400Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50921SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-phenylethyl]piperidine4000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50922SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclohexylethyl]-piperidine4300Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50923SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-chlorophenyl)-2-cyclopentylethyl]-piperidine2600Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50924SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-isopropylphenyl)-3-methylbutyl]piperidine3200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50925SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3-methoxyphenyl)-3-methylbutyl]piperidine>10000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50926SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(4-methoxyphenyl)-3-methylbutyl]piperidine>10000Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50927SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-1-methylpiperidine660Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50928SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)-3-methylbutyl]-piperidine120Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50929SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)pentyl]piperidine31Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50930SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(RR/SS)-2-[1-(3,4-dichlorophenyl)butyl]piperidine30Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50931SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDmethyl 2-(3,4-dichlorophenyl)-2-(piperidin-2-yl)acetate4200Froimowitz M et al., 2007Jan 15, 2025Jan 15, 2025
50932GABRA2UNDEFINEDRATUNDEFINEDN-(4-ethylbenzyl)-2-(1H-indol-3-yl)-2-oxoacetamide1600Primofiore G et al., 2007Jan 15, 2025Jan 15, 2025
50933GABRA2UNDEFINEDRATUNDEFINEDN-isopropyl-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide175Primofiore G et al., 2007Jan 15, 2025Jan 15, 2025
50934GABRA2UNDEFINEDRATUNDEFINEDN-butyl-2-(5-nitro-1H-indol-3-yl)-2-oxoacetamide553Primofiore G et al., 2007Jan 15, 2025Jan 15, 2025
50935GABRA2UNDEFINEDRATUNDEFINEDN-(4-ethynylbenzyl)-2-(1H-indol-3-yl)-2-oxoacetamide414Primofiore G et al., 2007Jan 15, 2025Jan 15, 2025
50936GABRA2UNDEFINEDRATUNDEFINEDN-(4-bromobenzyl)-2-(1H-indol-3-yl)-2-oxoacetamide81Primofiore G et al., 2007Jan 15, 2025Jan 15, 2025
50937GABRA2UNDEFINEDRATUNDEFINEDZolpidem765Primofiore G et al., 2007Jan 15, 2025Jan 15, 2025
50938SLC6A2UNDEFINEDHUMANUNDEFINEDDESIPRAMINE1Schou M et al., 2007Jan 15, 2025Jan 15, 2025
50939SLC6A2UNDEFINEDHUMANUNDEFINED(S,S)-1-cyclopentyl-2-(5-fluoro-2-methoxy-phenyl)-1-morpholin-2-yl-ethanol10.8Schou M et al., 2007Jan 15, 2025Jan 15, 2025
50940SLC6A2UNDEFINEDHUMANUNDEFINED(R)-1-(10,11-dihydro-dibenzo[b,f]azepin-5-yl)-3-methylamino-propan-2-ol8.29Schou M et al., 2007Jan 15, 2025Jan 15, 2025
50941SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-methoxyphenoxy)(phenyl)methyl)morpholine7.93Schou M et al., 2007Jan 15, 2025Jan 15, 2025
50942MORUNDEFINEDHUMANUNDEFINED17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol0.23Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50943MORUNDEFINEDHUMANUNDEFINED(5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate0.43Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50944MORUNDEFINEDHUMANUNDEFINED17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate0.29Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50945MORUNDEFINEDHUMANUNDEFINED(5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate0.46Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50946MORUNDEFINEDHUMANUNDEFINEDNaloxone(-)0.79Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50947MORUNDEFINEDHUMANUNDEFINEDNaltrexone0.23Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50948MORUNDEFINEDHUMANUNDEFINEDNalbuphine0.89Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50949KORUNDEFINEDHUMANUNDEFINED17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol0.079Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50950KORUNDEFINEDHUMANUNDEFINED(5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate0.13Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50951KORUNDEFINEDHUMANUNDEFINED17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate0.12Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50952KORUNDEFINEDHUMANUNDEFINED(5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate0.34Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50953KORUNDEFINEDHUMANUNDEFINEDNaloxone(-)1.1Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50954KORUNDEFINEDHUMANUNDEFINEDNaltrexone0.25Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50955KORUNDEFINEDHUMANUNDEFINEDNalbuphine2.2Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50956DORUNDEFINEDHUMANUNDEFINED17-cyclobutylmethyl-(1R,9R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-4-ol5.9Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50957DORUNDEFINEDHUMANUNDEFINED(5alpha)-17-allylllyl-14-hydroxy-6-oxo-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate39Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50958DORUNDEFINEDHUMANUNDEFINED17-(cyclopropylmethyl)morphinan-3-yl(5alpha)-17-(cyclopropylmethyl)-14-hydroxy-6-oxo-4,5-epoxymorphiana-3-yl sebacoylate15Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50959DORUNDEFINEDHUMANUNDEFINED(5alpha,6alpha)-17-(cyclobutylmethyl)-6,14-dihydroxy-4,5-epoxymorphinan-3-yl-17-(cyclobutylmethyl)morphinan-3-yl sebacoylate28Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50960DORUNDEFINEDHUMANUNDEFINEDNaloxone(-)76Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50961DORUNDEFINEDHUMANUNDEFINEDNaltrexone38Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50962DORUNDEFINEDHUMANUNDEFINEDNalbuphine240Peng X et al., 2007Jan 15, 2025Jan 15, 2025
50963Gabra3UNDEFINEDRATUNDEFINED8-ethoxy-3-iodo-benzo[e]pyrazolo[5,1-c][1,2,4]triazine 5-oxide34Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50964Gabra3UNDEFINEDRATUNDEFINEDDIAZEPAM14Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50965Gabra3UNDEFINEDRATUNDEFINED3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine4-oxide12.3Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50966Gabra3UNDEFINEDRATUNDEFINED3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine133Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50967GABRA5UNDEFINEDRATUNDEFINED8-ethoxy-3-iodo-benzo[e]pyrazolo[5,1-c][1,2,4]triazine 5-oxide99Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50968GABRA5UNDEFINEDRATUNDEFINEDDIAZEPAM9.8Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50969GABRA5UNDEFINEDRATUNDEFINED3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine4-oxide70Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50970GABRA5UNDEFINEDRATUNDEFINED3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine95Guerrini G et al., 2007Jan 15, 2025Jan 15, 2025
50971TRPV1UNDEFINEDRATUNDEFINEDCHLORPROMAZINE1300Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50972TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]cyclopropyl}thiourea370Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50973TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-methyl-1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}thiourea2890Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50974TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}thiourea67Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50975TRPV1UNDEFINEDRATUNDEFINEDN-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-2-methoxy-phenyl}-methanesulfonamide51Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50976TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-methyl-1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea7700Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50977TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{[4-(methylsulfonylamino)-3-fluorophenyl](phenyl)methyl}thiourea100Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50978TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)-3-fluorophenyl]-2-phenylethyl}thiourea1740Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50979TRPV1UNDEFINEDRATUNDEFINEDN'-(4-tert-butylbenzyl)-N-{1-[4-(methylsulfonylamino)-3-fluorophenyl]-2-ethylpropyl}thiourea339Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50980TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)-3-fluorophenyl]propyl}thiourea230Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50981TRPV1UNDEFINEDRATUNDEFINED(S)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea2140Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50982TRPV1UNDEFINEDRATUNDEFINED(R)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea39.2Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50983TRPV1UNDEFINEDRATUNDEFINED1-(4-tert-butylbenzyl)-3-(1-(3-fluoro-4-(methylsulfonamido)phenyl)ethyl)thiourea54Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50984TRPV1UNDEFINEDRATUNDEFINEDN-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-2-fluoro-phenyl}-methanesulfonamide53.5Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50985TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)phenyl]cyclopropyl}thiourea171Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50986TRPV1UNDEFINEDRATUNDEFINEDN-(4-{(S)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide3950Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50987TRPV1UNDEFINEDRATUNDEFINEDN-(4-{(R)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide41Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50988TRPV1UNDEFINEDRATUNDEFINEDN-(4-{1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide59.3Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50989TRPV1UNDEFINEDRATUNDEFINEDN-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-phenyl}-methanesulfonamide63Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50990TRPV1UNDEFINEDRATUNDEFINEDCHLORPROMAZINE520Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50991TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]cyclopropyl}thiourea243Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50992TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-methyl-1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}thiourea663Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50993TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[3-methoxy-4-(methylsulfonylamino)phenyl]ethyl}thiourea28.6Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50994TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-methyl-1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea980Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50995TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{[4-(methylsulfonylamino)-3-fluorophenyl](phenyl)methyl}thiourea860Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50996TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)-3-fluorophenyl]-2-phenylethyl}thiourea700Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50997TRPV1UNDEFINEDRATUNDEFINEDN'-(4-tert-butylbenzyl)-N-{1-[4-(methylsulfonylamino)-3-fluorophenyl]-2-ethylpropyl}thiourea223Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50998TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)-3-fluorophenyl]propyl}thiourea54Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
50999TRPV1UNDEFINEDRATUNDEFINED(S)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea2670Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51000TRPV1UNDEFINEDRATUNDEFINED(R)-N-(4-tert-butylbenzyl)-N'-{1-[3-fluoro-4-(methylsulfonylamino)phenyl]ethyl}thiourea37Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51001TRPV1UNDEFINEDRATUNDEFINED1-(4-tert-butylbenzyl)-3-(1-(3-fluoro-4-(methylsulfonamido)phenyl)ethyl)thiourea9.2Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51002TRPV1UNDEFINEDRATUNDEFINEDN-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-2-fluoro-phenyl}-methanesulfonamide9.2Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51003TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-[4-(methylsulfonylamino)phenyl]cyclopropyl}thiourea60Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51004TRPV1UNDEFINEDRATUNDEFINEDN-(4-tert-butylbenzyl)-N'-{1-methyl-1-[4-(methylsulfonylamino)phenyl]ethyl}thiourea1800Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51005TRPV1UNDEFINEDRATUNDEFINEDN-(4-{(R)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide4.5Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51006TRPV1UNDEFINEDRATUNDEFINEDN-(4-{1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide14.7Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51007TRPV1UNDEFINEDRATUNDEFINEDN-{4-[3-(4-tert-Butyl-benzyl)-thioureidomethyl]-phenyl}-methanesulfonamide54Chung JU et al., 2007Jan 15, 2025Jan 15, 2025
51008CB1UNDEFINEDHUMANUNDEFINED1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid cyclohexylamide3.9Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51009CB1UNDEFINEDHUMANUNDEFINED1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide3.7Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51010CB1UNDEFINEDHUMANUNDEFINED5-bromo-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide19Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51011CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-isopropyl-1H-imidazole-4-carboxamide18Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51012CB1UNDEFINEDHUMANUNDEFINED5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide10Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51013CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide5.7Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51014CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide5Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51015CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-methyl-1H-imidazole-4-carboxamide6.9Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51016CB1UNDEFINEDHUMANUNDEFINEDrac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl)-1H-imidazole-4-carboxamide17Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51017CB1UNDEFINEDHUMANUNDEFINEDrac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl)-1H-imidazole-4-carboxamide41Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51018CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide18Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51019CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide6.3Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51020CB1UNDEFINEDHUMANUNDEFINEDrac-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide22Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51021CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide75Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51022CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide29Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51023CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide97Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51024CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide29Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51025CB1UNDEFINEDHUMANUNDEFINEDrac-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide22Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51026CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1R,2R)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide920Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51027CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1S,2S)-2-(methylamino)cyclohexyl)-1H-imidazole-4-carboxamide620Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51028CB1UNDEFINEDHUMANUNDEFINEDN-((1R,2R)-2-aminocyclohexyl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide940Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51029CB1UNDEFINEDHUMANUNDEFINEDN-((1S,2S)-2-aminocyclohexyl)-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazole-4-carboxamide270Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51030CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-N-cyclohexyl-1-(pyridin-3-yl)-1H-imidazole-4-carboxamide1100Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51031CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-N-methyl-1H-imidazole-4-carboxamide34Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51032CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohexyl)-1H-imidazole-4-carboxamide17Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51033CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-(2-methoxyphenyl)-1H-imidazole-4-carboxamide95Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51034CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-(2-ethylphenyl)-1H-imidazole-4-carboxamide39Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51035CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide21Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51036CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-N-cyclohexyl-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide20Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51037CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide9Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51038CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imidazole-4-carboxamide4.6Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51039CB1UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide2.2Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51040CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-difluorophenyl)-1H-imidazole-4-carboxamide36Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51041CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphenyl)-1H-imidazole-4-carboxamide7.2Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51042CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-phenyl-1H-imidazole-4-carboxamide130Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51043CB1UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-(2,5-dichlorophenyl)-1H-imidazole-4-carboxamide25Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51044CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-fluorophenyl)-1H-imidazole-4-carboxamide8.2Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51045CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl-2-(2,4-dichlorophenyl)-1-(4-methoxyphenyl)-1H-imidazole-4-carboxamide4.9Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51046CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl-2-(2,4-dichlorophenyl)-1-p-tolyl-1H-imidazole-4-carboxamide1.9Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51047CB1UNDEFINEDHUMANUNDEFINEDRimonabant1.1Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51048CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide7.8Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51049CB2UNDEFINEDHUMANUNDEFINED1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imidazole-4-carboxylic acid cyclohexylamide240Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51050CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl-1H-imidazole-4-carboxamide2300Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51051CB2UNDEFINEDHUMANUNDEFINED1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imidazole-4-carboxamide1000Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51052CB2UNDEFINEDHUMANUNDEFINEDrac-1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-(2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide1100Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51053CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide5300Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51054CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclopentyl)-1H-imidazole-4-carboxamide6300Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51055CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide1200Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51056CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl)-1H-imidazole-4-carboxamide5100Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51057CB2UNDEFINEDHUMANUNDEFINED1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide2700Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51058CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2-hydroxycyclohexyl)-5-propyl-1H-imidazole-4-carboxamide2700Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51059CB2UNDEFINEDHUMANUNDEFINED2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((1S,2S)-2-hydroxycyclohexyl)-1H-imidazole-4-carboxamide2300Smith RA et al., 2007Jan 15, 2025Jan 15, 2025
51060Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide14Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51061Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide2.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51062Alpha1AUNDEFINEDHUMANUNDEFINEDTamsulosin0.19Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51063Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide43Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51064Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide3.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51065Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide23Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51066Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide16Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51067Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide31Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51068Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide12Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51069Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide69Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51070Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide8.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51071Alpha1AUNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide38Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51072Alpha1AUNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide5.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51073Alpha1AUNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide12Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51074Alpha1AUNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide7Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51075Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide4.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51076Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide5.9Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51077Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide10Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51078Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide6.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51079Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide2.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51080Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51081Alpha1AUNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide21Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51082Alpha1AUNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide1.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51083Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide16Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51084Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide3.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51085Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide1.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51086Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide4.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51087Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide1.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51088Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51089Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide0.91Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51090Alpha1AUNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide1.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51091Alpha1AUNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51092Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide28Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51093Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide144Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51094Alpha1BUNDEFINEDHUMANUNDEFINEDTamsulosin2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51095Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide1487Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51096Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide299Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51097Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide639Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51098Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide690Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51099Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide681Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51100Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide300Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51101Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide4403Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51102Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide401Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51103Alpha1BUNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide302Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51104Alpha1BUNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide76Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51105Alpha1BUNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide355Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51106Alpha1BUNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide261Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51107Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide787Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51108Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide181Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51109Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide703Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51110Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide216Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51111Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide91Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51112Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide92Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51113Alpha1BUNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide368Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51114Alpha1BUNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide123Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51115Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide340Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51116Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide275Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51117Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide337Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51118Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide107Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51119Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide305Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51120Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide82Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51121Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide133Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51122Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide141Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51123Alpha1BUNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide1385Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51124Alpha1BUNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide470Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51125Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide148Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51126Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide0.77Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51127Alpha1DUNDEFINEDHUMANUNDEFINEDTamsulosin0.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51128Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide53Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51129Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide1.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51130Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide60Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51131Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide12Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51132Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide86Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51133Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide4.1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51134Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide49Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51135Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide5.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51136Alpha1DUNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide86Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51137Alpha1DUNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide2.7Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51138Alpha1DUNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide70Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51139Alpha1DUNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide5.9Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51140Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide44Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51141Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide0.98Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51142Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide36Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51143Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide1.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51144Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide26Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51145Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51146Alpha1DUNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide23Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51147Alpha1DUNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide2.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51148Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide57Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51149Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide13Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51150Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide32Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51151Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide2.1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51152Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide47Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51153Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide2.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51154Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide34Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51155Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51156Alpha1DUNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide87Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51157Alpha1DUNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide7.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51158Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide40Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51159D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide144Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51160D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide94Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51161D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(5-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide178Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51162D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide104Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51163D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(4-fluoro-2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide106Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51164D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide88Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51165D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2-difluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide276Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51166D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide284Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51167D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2-fluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide201Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51168D2UNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide104Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51169D2UNDEFINEDHUMANUNDEFINED4-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide154Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51170D2UNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide129Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51171D2UNDEFINEDHUMANUNDEFINED3-(difluoromethoxy)-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide85Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51172D2UNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide37Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51173D2UNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide78Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51174D2UNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide82Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51175D2UNDEFINEDHUMANUNDEFINED5-chloro-2-methoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide69Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51176D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide23Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51177D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-sulfonamide57Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51178D2UNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1r,4r)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide83Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51179D2UNDEFINEDHUMANUNDEFINED3,4-dimethoxy-N-((1s,4s)-4-(4-(2-(2,2,2-trifluoroethoxy)phenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide111Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51180D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide71Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51181D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzo[d][1,3]dioxole-5-sulfonamide66Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51182D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide159Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51183D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide187Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51184D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide154Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51185D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide129Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51186D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide133Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51187D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-cyclopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide144Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51188D2UNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide79Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51189D2UNDEFINEDHUMANUNDEFINED3,4-difluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)benzenesulfonamide79Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51190D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperidin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide55Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51191CHRNA4UNDEFINEDRATUNDEFINEDNicotine0.94Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51192CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-3-pyridinyl)-5,5-dimethyl-2,5-diazabicyclo-[2.2.1]heptanium iodide0.2Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51193CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-3-pyridinyl)-5-ethyl-2,5-diazabicyclo[2.2.1]-heptane34Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51194CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-3-pyridinyl)-5-methyl-2,5-diazabicyclo-[2.2.1]heptane1.3Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51195CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(4-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane5200Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51196CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane0.15Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51197CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(2-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane980Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51198CHRNA4UNDEFINEDRATUNDEFINED6-(6-chloro-3-pyridinyl)-2,6-diazabicyclo[3.2.1]octane2.8Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51199CHRNA4UNDEFINEDRATUNDEFINED2-(6-chloro-3-pyridinyl)-2,6-diazabicyclo[3.2.1]octane1.5Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51200CHRNA4UNDEFINEDRATUNDEFINED6-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane0.065Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51201CHRNA4UNDEFINEDRATUNDEFINED3-(3-pyridinyl)-3,6-diazabicyclo[3.2.1]octane0.047Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51202CHRNA4UNDEFINEDRATUNDEFINED2-(3-pyridinyl)-2,5-diazabicyclo[2.2.2]octane0.02Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51203CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.018Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51204CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.1Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51205CHRNA4UNDEFINEDRATUNDEFINEDEpibatidine0.047Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51206CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(6-chloro-5-methoxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane0.1Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51207CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(5,6-dichloro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.018Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51208CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(5-trifluoromethyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane490Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51209CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(6-chloro-5-methyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane0.014Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51210CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.12Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51211CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.53Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51212CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-5-hydroxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane0.17Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51213CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-5-hydroxy-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane1.6Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51214CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-[5-hydroxy-3-pyridinyl]-2,5-diazabicyclo[2.2.1]-heptane0.035Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51215CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-[5-hydroxy-3-pyridinyl]-2,5-diazabicyclo[2.2.1]-heptane4Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51216CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-aminomethyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane140Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51217CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(6-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.027Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51218CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-cyano-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane1.7Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51219CHRNA4UNDEFINEDRATUNDEFINED(S,S)-2-(6-aminopyridin-3-yl)-2,5-diazabicyclo[2.2.1]-heptane20Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51220CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-nitro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane110Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51221CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(6-methoxy-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.25Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51222CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-methyl-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane1.6Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51223CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-fluoro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.028Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51224CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-fluoro-3-pyridinyl)-2,5-diazabicyclo[2.2.1]-heptane0.17Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51225CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane0.018Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51226CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-aminocarbonyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane0.83Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51227CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-aminocarbonyl-3-pyridinyl)-2,5-diazabicyclo-[2.2.1]heptane24Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51228CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(2,5-diazabicyclo[2.2.1]hept-2-yl)-thieno[3,2-b]pyridine0.83Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51229CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-3-(2,5-diazabicyclo[2.2.1]hept-2-yl)-thieno[3,2-b]pyridine280Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51230CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(2-quinolinyl)-2,5-diazabicyclo[2.2.1]heptane4000Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51231CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-quinolinyl)-2,5-diazabicyclo[2.2.1]heptane17Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51232CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(2-thiazolyl)-2,5-diazabicyclo[2.2.1]heptane2300Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51233CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(3-methyl-(1,2,4)-thiadiazol-5-yl)-2,5-diazabicyclo-[2.2.1]heptane350Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51234CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-methylisothiazol-5-yl)-2,5-diazabicyclo[2.2.1]-heptane4.9Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51235CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane22Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51236CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptane250Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51237CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-nitrophenyl)-2,5-diazabicyclo[2.2.1]heptane600Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51238CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(4-nitrophenyl)-2,5-diazabicyclo[2.2.1]heptane67Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51239CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(phenyl)-2,5-diazabicyclo[2.2.1]heptane1000Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51240CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-1,3-pyrimidin-4-yl)-2,5-diazabicyclo[2.2.1]-heptane52Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51241CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(5-pyrimidinyl)-2,5-diazabicyclo[2.2.1]-heptane0.95Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51242CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(4-chloro-1-phthalazinyl)-2,5-diazabicyclo[2.2.1]-heptane1900Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51243CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloro-5-methyl-3-pyridazinyl)-2,5-diazabicyclo-[2.2.1]heptane3.8Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51244CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-pyridazinyl)-2,5-diazabicyclo[2.2.1]heptane120Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51245CHRNA4UNDEFINEDRATUNDEFINED2-(6-Chloro-pyridazin-3-yl)-2,5-diaza-bicyclo[2.2.1]heptane0.24Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51246CHRNA4UNDEFINEDRATUNDEFINED2-(6-Chloro-pyridazin-3-yl)-2,5-diaza-bicyclo[2.2.1]heptane8.8Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51247CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(6-chloropyridin-3-yl)-2,5-diazabicyclo[2.2.1]-heptanone>10000Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51248CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(6-chloropyridine-3-carbonyl)-2,5-diazabicyclo-[2.2.1]heptane590Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51249CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(5-bromo-6-chloropyridine-3-sulfonyl)-2,5-diazabicyclo[2.2.1]heptane17Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51250CHRNA4UNDEFINEDRATUNDEFINED(1R,4R)-2-(3-pyridinylmethyl)-2,5-diazabicyclo[2.2.1]-heptane56Bunnelle WH et al., 2007Jan 15, 2025Jan 15, 2025
51251SLC6A4UNDEFINEDRATUNDEFINEDFLUOXETINE2.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51252SLC6A4UNDEFINEDRATUNDEFINED1-(4-ethylphenyl)-3-methyl-6-(4-(4-(1-phenylvinyl)cyclohexyl)butyl)-1,2,3,4-tetrahydronaphthalene21Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51253SLC6A4UNDEFINEDRATUNDEFINED(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)(1-methyl-1H-pyrrol-2-yl)methanone8.4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51254SLC6A4UNDEFINEDRATUNDEFINED1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)-2-methylpropan-1-one15Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51255SLC6A4UNDEFINEDRATUNDEFINED1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)ethanone15Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51256SLC6A4UNDEFINEDRATUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline25Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51257SLC6A4UNDEFINEDRATUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(pyridin-4-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline5.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51258SLC6A4UNDEFINEDRATUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(thiazol-2-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline2.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51259SLC6A4UNDEFINEDRATUNDEFINED4-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)benzonitrile3.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51260SLC6A4UNDEFINEDRATUNDEFINED2-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)phenol5.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51261SLC6A4UNDEFINEDRATUNDEFINED7-(3-(4-cyclopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline10Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51262SLC6A4UNDEFINEDRATUNDEFINED7-(3-(4-isopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline1.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51263SLC6A4UNDEFINEDRATUNDEFINED7-(3-(4-ethylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline1.5Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51264SLC6A4UNDEFINEDRATUNDEFINEDN-cyclopropyl-N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine7.6Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51265SLC6A4UNDEFINEDRATUNDEFINEDN-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51266SLC6A4UNDEFINEDRATUNDEFINEDN,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine2.2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51267SLC6A4UNDEFINEDRATUNDEFINEDN-ethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine0.73Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51268SLC6A4UNDEFINEDRATUNDEFINED7-(3-(3,3-difluoropyrrolidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51269SLC6A4UNDEFINEDRATUNDEFINED7-(3-(3,3-difluoroazetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51270SLC6A4UNDEFINEDRATUNDEFINED7-(3-(azetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline1Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51271SLC6A4UNDEFINEDRATUNDEFINED7-[3-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-propoxy]-4-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydro-isoquinoline6.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51272SLC6A4UNDEFINEDRATUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(trifluoromethyl)piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline19Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51273SLC6A4UNDEFINEDRATUNDEFINED1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidine-4-carbonitrile5.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51274SLC6A4UNDEFINEDRATUNDEFINED(1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-yl)methanol2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51275SLC6A4UNDEFINEDRATUNDEFINED1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol1.4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51276SLC6A4UNDEFINEDRATUNDEFINED7-(3-(3,3-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline10Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51277SLC6A4UNDEFINEDRATUNDEFINED7-(3-(4,4-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline5.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51278SLC6A4UNDEFINEDRATUNDEFINED7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline1.6Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51279SLC6A4UNDEFINEDRATUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline4.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51280SLC6A4UNDEFINEDRATUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51281SLC6A4UNDEFINEDHUMANUNDEFINEDFLUOXETINE2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51282SLC6A4UNDEFINEDHUMANUNDEFINED1-(4-ethylphenyl)-3-methyl-6-(4-(4-(1-phenylvinyl)cyclohexyl)butyl)-1,2,3,4-tetrahydronaphthalene19Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51283SLC6A4UNDEFINEDHUMANUNDEFINED(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)(1-methyl-1H-pyrrol-2-yl)methanone8.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51284SLC6A4UNDEFINEDHUMANUNDEFINED1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)-2-methylpropan-1-one15Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51285SLC6A4UNDEFINEDHUMANUNDEFINED1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)ethanone42Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51286SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline33Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51287SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(pyridin-4-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51288SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(thiazol-2-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline5.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51289SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)benzonitrile8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51290SLC6A4UNDEFINEDHUMANUNDEFINED2-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)phenol7.2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51291SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(4-cyclopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline18Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51292SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(4-isopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline1.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51293SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(4-ethylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51294SLC6A4UNDEFINEDHUMANUNDEFINEDN-cyclopropyl-N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine9.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51295SLC6A4UNDEFINEDHUMANUNDEFINEDN-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine19.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51296SLC6A4UNDEFINEDHUMANUNDEFINEDN,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51297SLC6A4UNDEFINEDHUMANUNDEFINEDN-ethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine3.4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51298SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(3,3-difluoropyrrolidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline7.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51299SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(3,3-difluoroazetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline2.9Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51300SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(azetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline4.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51301SLC6A4UNDEFINEDHUMANUNDEFINED7-[3-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-propoxy]-4-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydro-isoquinoline12Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51302SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(trifluoromethyl)piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline14Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51303SLC6A4UNDEFINEDHUMANUNDEFINED1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidine-4-carbonitrile5.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51304SLC6A4UNDEFINEDHUMANUNDEFINED(1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-yl)methanol3.2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51305SLC6A4UNDEFINEDHUMANUNDEFINED1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol3.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51306SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(3,3-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline8.2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51307SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(4,4-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline6.5Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51308SLC6A4UNDEFINEDHUMANUNDEFINED7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline2.9Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51309SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline6.5Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51310SLC6A4UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline5.1Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51311H3UNDEFINEDHUMANUNDEFINEDFLUOXETINE7300Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51312H3UNDEFINEDHUMANUNDEFINED1-(4-ethylphenyl)-3-methyl-6-(4-(4-(1-phenylvinyl)cyclohexyl)butyl)-1,2,3,4-tetrahydronaphthalene2840Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51313H3UNDEFINEDHUMANUNDEFINED(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)(1-methyl-1H-pyrrol-2-yl)methanone2606Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51314H3UNDEFINEDHUMANUNDEFINED1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)-2-methylpropan-1-one509Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51315H3UNDEFINEDHUMANUNDEFINED1-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)ethanone267Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51316H3UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(4-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline1440Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51317H3UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(pyridin-4-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline3.3Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51318H3UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(thiazol-2-yl)piperazin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline268Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51319H3UNDEFINEDHUMANUNDEFINED4-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)benzonitrile144Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51320H3UNDEFINEDHUMANUNDEFINED2-(4-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperazin-1-yl)phenol1108Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51321H3UNDEFINEDHUMANUNDEFINED7-(3-(4-cyclopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline30Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51322H3UNDEFINEDHUMANUNDEFINED7-(3-(4-isopropylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline9.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51323H3UNDEFINEDHUMANUNDEFINED7-(3-(4-ethylpiperazin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline12Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51324H3UNDEFINEDHUMANUNDEFINEDN-cyclopropyl-N-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine7.4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51325H3UNDEFINEDHUMANUNDEFINEDN-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)cyclopropanamine38Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51326H3UNDEFINEDHUMANUNDEFINEDN,N-diethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine1.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51327H3UNDEFINEDHUMANUNDEFINEDN-ethyl-3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propan-1-amine47Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51328H3UNDEFINEDHUMANUNDEFINED7-(3-(3,3-difluoropyrrolidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline9.5Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51329H3UNDEFINEDHUMANUNDEFINED7-(3-(3,3-difluoroazetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline69Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51330H3UNDEFINEDHUMANUNDEFINED7-(3-(azetidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51331H3UNDEFINEDHUMANUNDEFINED7-[3-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-propoxy]-4-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydro-isoquinoline106Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51332H3UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(4-(trifluoromethyl)piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline40Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51333H3UNDEFINEDHUMANUNDEFINED1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidine-4-carbonitrile7.4Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51334H3UNDEFINEDHUMANUNDEFINED(1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-yl)methanol9.5Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51335H3UNDEFINEDHUMANUNDEFINED1-(3-(4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yloxy)propyl)piperidin-4-ol11Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51336H3UNDEFINEDHUMANUNDEFINED7-(3-(3,3-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline14Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51337H3UNDEFINEDHUMANUNDEFINED7-(3-(4,4-difluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline8.7Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51338H3UNDEFINEDHUMANUNDEFINED7-(3-(4-fluoropiperidin-1-yl)propoxy)-4-(4-methoxyphenyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51339H3UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-morpholinopropoxy)-1,2,3,4-tetrahydroisoquinoline3.8Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51340H3UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-2-methyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydroisoquinoline2Keith JM et al., 2007Jan 15, 2025Jan 15, 2025
51341M1UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((phenethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine220Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51342M1UNDEFINEDHUMANUNDEFINED7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine1.8Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51343M1UNDEFINEDHUMANUNDEFINED7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine36Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51344M1UNDEFINEDHUMANUNDEFINED(4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol18Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51345M1UNDEFINEDHUMANUNDEFINED4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexanol19Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51346M1UNDEFINEDHUMANUNDEFINED3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine140Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51347M1UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydro-2H-thiopyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine52Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51348M1UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydropyran-4-ylidene)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine86Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51349M1UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine58Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51350M1UNDEFINEDHUMANUNDEFINED{3-[(2-adamantan-1-yl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-dimethyl-amine5.9Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51351M1UNDEFINEDHUMANUNDEFINED3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine12Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51352M1UNDEFINEDHUMANUNDEFINED3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine18Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51353M1UNDEFINEDHUMANUNDEFINED3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine21Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51354M1UNDEFINEDHUMANUNDEFINED3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine31Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51355M1UNDEFINEDHUMANUNDEFINEDOxybutinin1Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51356M1UNDEFINEDHUMANUNDEFINED3-((2-fluorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine380Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51357M1UNDEFINEDHUMANUNDEFINED3-((2,6-dichlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine540Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51358M1UNDEFINEDHUMANUNDEFINED3-((4-isopropylphenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine200Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51359M1UNDEFINEDHUMANUNDEFINED3-((4-chlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine260Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51360M1UNDEFINEDHUMANUNDEFINEDdimethyl-{3-[(2-p-tolyl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-amine220Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51361M2UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((phenethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine90Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51362M2UNDEFINEDHUMANUNDEFINED7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine0.12Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51363M2UNDEFINEDHUMANUNDEFINED7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine5.1Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51364M2UNDEFINEDHUMANUNDEFINED(4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol1.8Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51365M2UNDEFINEDHUMANUNDEFINED4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexanol1.9Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51366M2UNDEFINEDHUMANUNDEFINED3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine12Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51367M2UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydro-2H-thiopyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine7.2Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51368M2UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydropyran-4-ylidene)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine8.8Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51369M2UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine6Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51370M2UNDEFINEDHUMANUNDEFINED{3-[(2-adamantan-1-yl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-dimethyl-amine0.66Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51371M2UNDEFINEDHUMANUNDEFINED3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine2Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51372M2UNDEFINEDHUMANUNDEFINED3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine6.2Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51373M2UNDEFINEDHUMANUNDEFINED3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine2.4Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51374M2UNDEFINEDHUMANUNDEFINED3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine12Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51375M2UNDEFINEDHUMANUNDEFINEDOxybutinin8.1Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51376M2UNDEFINEDHUMANUNDEFINED3-((2-fluorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine41Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51377M2UNDEFINEDHUMANUNDEFINED3-((2,6-dichlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine49Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51378M2UNDEFINEDHUMANUNDEFINED3-((4-isopropylphenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine44Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51379M2UNDEFINEDHUMANUNDEFINED3-((4-chlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine49Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51380M2UNDEFINEDHUMANUNDEFINEDdimethyl-{3-[(2-p-tolyl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-amine48Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51381M3UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((phenethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine20Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51382M3UNDEFINEDHUMANUNDEFINED7,8-dichloro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine0.22Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51383M3UNDEFINEDHUMANUNDEFINED7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine4.2Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51384M3UNDEFINEDHUMANUNDEFINED(4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexyl)methanol2.1Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51385M3UNDEFINEDHUMANUNDEFINED4-(2-((3-(dimethylamino)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl)methylamino)ethyl)cyclohexanol2.9Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51386M3UNDEFINEDHUMANUNDEFINED3-((2-(3,6-dihydro-2H-thiopyran-4-yl)ethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine5.8Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51387M3UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydro-2H-thiopyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine6.8Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51388M3UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydropyran-4-ylidene)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine14Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51389M3UNDEFINEDHUMANUNDEFINEDN,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine11Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51390M3UNDEFINEDHUMANUNDEFINED{3-[(2-adamantan-1-yl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-dimethyl-amine1.5Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51391M3UNDEFINEDHUMANUNDEFINED3-((2-cycloheptylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine2.7Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51392M3UNDEFINEDHUMANUNDEFINED3-((2-cyclohexylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine2.5Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51393M3UNDEFINEDHUMANUNDEFINED3-((2-cyclopentylethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine3.3Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51394M3UNDEFINEDHUMANUNDEFINED3-((cyclohexylmethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine4.9Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51395M3UNDEFINEDHUMANUNDEFINEDOxybutinin0.78Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51396M3UNDEFINEDHUMANUNDEFINED3-((2-fluorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine19Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51397M3UNDEFINEDHUMANUNDEFINED3-((2,6-dichlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine23Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51398M3UNDEFINEDHUMANUNDEFINED3-((4-isopropylphenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine56Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51399M3UNDEFINEDHUMANUNDEFINED3-((4-chlorophenethylamino)methyl)-N,N-dimethyl-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine20Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51400M3UNDEFINEDHUMANUNDEFINEDdimethyl-{3-[(2-p-tolyl-ethylamino)-methyl]-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-yl}-amine18Sonda S et al., 2007Jan 15, 2025Jan 15, 2025
51401D2UNDEFINEDUNDEFINEDUNDEFINED(R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine80Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51402D2UNDEFINEDUNDEFINEDUNDEFINEDHALOPERIDOL3.3Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51403D2UNDEFINEDUNDEFINEDUNDEFINED(S)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine70Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51404D2UNDEFINEDUNDEFINEDUNDEFINED(R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine46Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51405D2UNDEFINEDUNDEFINEDUNDEFINED(S)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine400Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51406D4UNDEFINEDHUMANUNDEFINED(R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine426Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51407D4UNDEFINEDHUMANUNDEFINEDHALOPERIDOL103Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51408D4UNDEFINEDHUMANUNDEFINED(S)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine225Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51409D4UNDEFINEDHUMANUNDEFINED(R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine507Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51410D4UNDEFINEDHUMANUNDEFINED(S)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine483Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51411D3UNDEFINEDHUMANUNDEFINED(R)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine2.1Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51412D3UNDEFINEDHUMANUNDEFINEDHALOPERIDOL6.4Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51413D3UNDEFINEDHUMANUNDEFINED(S)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine5.1Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51414D3UNDEFINEDHUMANUNDEFINED(R)-1-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)-4-(2-ethoxyphenyl)piperazine2.1Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51415D3UNDEFINEDHUMANUNDEFINED(S)-1-(bis(4-fluorophenyl)methyl)-4-(3-(3-(3,4-dimethoxyphenyl)-4,5-dihydroisoxazol-5-yl)propyl)piperazine20Jung JY et al., 2007Jan 15, 2025Jan 15, 2025
51416SLC6A4UNDEFINEDRATUNDEFINED2-[2-(hydroxymethyl)piperazin-1-yl]-6-nitroquinoline0.43Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51417SLC6A4UNDEFINEDRATUNDEFINEDFLUOXETINE8.7Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51418SLC6A4UNDEFINEDRATUNDEFINED6-Nitro-2-piperazin-1-yl-quinoline0.24Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51419SLC6A4UNDEFINEDRATUNDEFINED2-[(2-butoxymethyl)piperazin-1-yl]-6-nitroquinoline15.36Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51420SLC6A4UNDEFINEDRATUNDEFINED6-nitro-2-(2-propoxymethylpiperazin-1-yl)quinoline5.67Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51421SLC6A4UNDEFINEDRATUNDEFINED2-[2-(ethoxymethyl)piperazin-1-yl]-6-nitroquinoline0.43Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51422SLC6A4UNDEFINEDRATUNDEFINED2-[(2-methoxymethyl)piperazin-1-yl]-6-nitroquinoline0.68Lee JH et al., 2007Jan 15, 2025Jan 15, 2025
51423Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,2S,5S )-6-Benzyl-8-methyl-6,8-diazabicyclo-[3.2.2]nonan-2-ol2890Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51424Sigma2UNDEFINEDUNDEFINEDUNDEFINEDditolylguanidine63.9Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51425Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,5S )-6-benzyl-8-methyl-6,8-diazabicyclo[3.2.2]-nonane-2-one dimethyl acetal1830Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51426Sigma2UNDEFINEDUNDEFINEDUNDEFINED6-benzyl-2-(benzyloxy)-8-phenethyl-6,8-diaza-bicyclo[3.2.2]nonane628Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51427Sigma2UNDEFINEDUNDEFINEDUNDEFINED6-benzyl-2-(benzyloxy)-8-butyl-6,8-diaza-bicyclo[3.2.2]nonane820Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51428Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,2R,5S )-6-benzyl-2-benzyloxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane30.4Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51429Sigma2UNDEFINEDUNDEFINEDUNDEFINED6-benzyl-2-methoxy-8-phenethyl-6,8-diaza-bicyclo[3.2.2]nonane297Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51430Sigma2UNDEFINEDUNDEFINEDUNDEFINED6-benzyl-8-butyl-2-methoxy-6,8-diaza-bicyclo[3.2.2]nonane219Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51431Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,2R,5S )-6-benzyl-2-methoxy-8-methyl-6,8-diazabicyclo[3.2.2]nonane327Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51432Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,2R,5S )-6-benzyl-8-(2-phenylethyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol588Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51433Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,2S,5S )-6-Benzyl-8-(2-phenylethyl)-6,8-diazabidiazabicyclo343Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51434Sigma2UNDEFINEDUNDEFINEDUNDEFINED6-benzyl-8-butyl-6,8-diaza-bicyclo[3.2.2]nonan-2-ol447Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51435Sigma2UNDEFINEDUNDEFINEDUNDEFINED(1R,2R,5S )-6-benzyl-8-methyl-6,8-diazabicyclo[3.2.2]nonan-2-ol4180Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51436Sigma2UNDEFINEDUNDEFINEDUNDEFINEDHALOPERIDOL34.2Weigl M et al., 2007Jan 15, 2025Jan 15, 2025
51437Alpha1AUNDEFINEDHUMANUNDEFINEDTamsulosin0.19Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51438Alpha1AUNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide3.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51439Alpha1AUNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide14.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51440Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide13.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51441Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide4.9Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51442Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide5.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51443Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51444Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide3.9Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51445Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide1.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51446Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide36Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51447Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide19Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51448Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide189Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51449Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide45Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51450Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51451Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide61Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51452Alpha1AUNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51453Alpha1AUNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51454Alpha1AUNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide0.56Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51455Alpha1AUNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide12Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51456Alpha1AUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide1.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51457Alpha1AUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide4.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51458Alpha1AUNDEFINEDHUMANUNDEFINED3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide1.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51459Alpha1AUNDEFINEDHUMANUNDEFINED3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51460Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51461Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide4.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51462Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide25Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51463Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide36Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51464Alpha1AUNDEFINEDHUMANUNDEFINED5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide10Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51465Alpha1AUNDEFINEDHUMANUNDEFINED5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide1.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51466Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide3.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51467Alpha1AUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51468Alpha1AUNDEFINEDHUMANUNDEFINED5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51469Alpha1AUNDEFINEDHUMANUNDEFINED5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51470Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide0.9Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51471Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide18Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51472Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide17Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51473Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide8.7Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51474Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide23Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51475Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide1.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51476Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide100Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51477Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide17Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51478Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide7.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51479Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide4.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51480Alpha1AUNDEFINEDHUMANUNDEFINED4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide1.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51481Alpha1AUNDEFINEDHUMANUNDEFINED4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide5.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51482Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide20Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51483Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide14Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51484Alpha1AUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide0.73Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51485Alpha1AUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide3.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51486Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51487Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide6.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51488Alpha1AUNDEFINEDHUMANUNDEFINED2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide0.88Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51489Alpha1AUNDEFINEDHUMANUNDEFINED2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide5.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51490Alpha1AUNDEFINEDHUMANUNDEFINED2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide0.77Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51491Alpha1AUNDEFINEDHUMANUNDEFINED2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide9.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51492Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide2.7Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51493Alpha1AUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide13.7Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51494Alpha1BUNDEFINEDHUMANUNDEFINEDTamsulosin2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51495Alpha1BUNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide279Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51496Alpha1BUNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide125Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51497Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide268Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51498Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide169Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51499Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide192Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51500Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide400Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51501Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide200Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51502Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide82Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51503Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide952Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51504Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide601Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51505Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide364Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51506Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide1855Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51507Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide399Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51508Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide112Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51509Alpha1BUNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide243Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51510Alpha1BUNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide101Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51511Alpha1BUNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide348Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51512Alpha1BUNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide120Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51513Alpha1BUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide596Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51514Alpha1BUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide177Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51515Alpha1BUNDEFINEDHUMANUNDEFINED3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide193Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51516Alpha1BUNDEFINEDHUMANUNDEFINED3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide167Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51517Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide173Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51518Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide85Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51519Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide258Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51520Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide473Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51521Alpha1BUNDEFINEDHUMANUNDEFINED5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide131Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51522Alpha1BUNDEFINEDHUMANUNDEFINED5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide42Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51523Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide250Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51524Alpha1BUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide78Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51525Alpha1BUNDEFINEDHUMANUNDEFINED5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide714Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51526Alpha1BUNDEFINEDHUMANUNDEFINED5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide162Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51527Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide218Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51528Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide162Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51529Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide424Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51530Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide153Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51531Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide126Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51532Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide109Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51533Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide1254Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51534Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide174Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51535Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide392Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51536Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide195Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51537Alpha1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide301Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51538Alpha1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide150Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51539Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide334Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51540Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide222Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51541Alpha1BUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide545Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51542Alpha1BUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide108Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51543Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide236Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51544Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide201Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51545Alpha1BUNDEFINEDHUMANUNDEFINED2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide385Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51546Alpha1BUNDEFINEDHUMANUNDEFINED2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide103Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51547Alpha1BUNDEFINEDHUMANUNDEFINED2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide31Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51548Alpha1BUNDEFINEDHUMANUNDEFINED2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide217Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51549Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide487Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51550Alpha1BUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide111Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51551Alpha1DUNDEFINEDHUMANUNDEFINEDTamsulosin0.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51552Alpha1DUNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide14.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51553Alpha1DUNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide0.14Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51554Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide76Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51555Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide9.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51556Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide5.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51557Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide46Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51558Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide12Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51559Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide3.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51560Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide44Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51561Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide48Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51562Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide64Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51563Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide15Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51564Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide12Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51565Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide19Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51566Alpha1DUNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide19Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51567Alpha1DUNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide1.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51568Alpha1DUNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide24Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51569Alpha1DUNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide6.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51570Alpha1DUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide8.6Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51571Alpha1DUNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide0.64Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51572Alpha1DUNDEFINEDHUMANUNDEFINED3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide16Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51573Alpha1DUNDEFINEDHUMANUNDEFINED3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51574Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide22Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51575Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide2.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51576Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide15Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51577Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide14Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51578Alpha1DUNDEFINEDHUMANUNDEFINED5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide38Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51579Alpha1DUNDEFINEDHUMANUNDEFINED5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide0.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51580Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide11Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51581Alpha1DUNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide0.75Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51582Alpha1DUNDEFINEDHUMANUNDEFINED5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide66Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51583Alpha1DUNDEFINEDHUMANUNDEFINED5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51584Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide31Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51585Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide7Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51586Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide56Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51587Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide5.1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51588Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide24Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51589Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51590Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide111Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51591Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide2.1Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51592Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide22Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51593Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide3.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51594Alpha1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide36Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51595Alpha1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide4.8Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51596Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide35Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51597Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide1.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51598Alpha1DUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide24.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51599Alpha1DUNDEFINEDHUMANUNDEFINED3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide3.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51600Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide27Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51601Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide2.5Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51602Alpha1DUNDEFINEDHUMANUNDEFINED2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide30Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51603Alpha1DUNDEFINEDHUMANUNDEFINED2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide2.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51604Alpha1DUNDEFINEDHUMANUNDEFINED2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide3.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51605Alpha1DUNDEFINEDHUMANUNDEFINED2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide6.3Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51606Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide55Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51607Alpha1DUNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide5.2Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51608D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide191Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51609D2UNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide80Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51610D2UNDEFINEDHUMANUNDEFINED5-bromo-6-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide61Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51611D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide43Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51612D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methoxypyridine-3-sulfonamide92Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51613D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide55Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51614D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)pyridine-3-sulfonamide15Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51615D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide71Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51616D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)(phenyl)methanesulfonamide24Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51617D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-fluorobenzenesulfonamide425Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51618D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide588Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51619D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-(cyclopropylmethoxy)phenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide123Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51620D2UNDEFINEDHUMANUNDEFINED5-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide356Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51621D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide259Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51622D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide810Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51623D2UNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide42Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51624D2UNDEFINEDHUMANUNDEFINED4-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide130Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51625D2UNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide271Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51626D2UNDEFINEDHUMANUNDEFINED3-chloro-2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide198Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51627D2UNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide76Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51628D2UNDEFINEDHUMANUNDEFINED2,4-dichloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide42Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51629D2UNDEFINEDHUMANUNDEFINED3-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide52Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51630D2UNDEFINEDHUMANUNDEFINED3-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-methylbenzenesulfonamide60Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51631D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide18Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51632D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-nitrobenzenesulfonamide45Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51633D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide1.9Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51634D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-(trifluoromethyl)benzenesulfonamide194Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51635D2UNDEFINEDHUMANUNDEFINED5-bromo-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide36Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51636D2UNDEFINEDHUMANUNDEFINED5-bromo-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide37Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51637D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide78Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51638D2UNDEFINEDHUMANUNDEFINED5-chloro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide101Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51639D2UNDEFINEDHUMANUNDEFINED5-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide139Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51640D2UNDEFINEDHUMANUNDEFINED5-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxybenzenesulfonamide173Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51641D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide50Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51642D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-methoxy-5-methylbenzenesulfonamide110Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51643D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide62Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51644D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2,5-dimethoxybenzenesulfonamide81Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51645D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide62Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51646D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3,4-dimethoxybenzenesulfonamide94Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51647D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide58Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51648D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(trifluoromethoxy)benzenesulfonamide430Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51649D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide14Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51650D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-4-(methylsulfonyl)benzenesulfonamide122Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51651D2UNDEFINEDHUMANUNDEFINED4-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide27Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51652D2UNDEFINEDHUMANUNDEFINED4-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide69Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51653D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide39Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51654D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(trifluoromethyl)benzenesulfonamide118Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51655D2UNDEFINEDHUMANUNDEFINED3-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide64Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51656D2UNDEFINEDHUMANUNDEFINED3-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide74Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51657D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide86Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51658D2UNDEFINEDHUMANUNDEFINEDN-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-2-nitrobenzenesulfonamide51Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51659D2UNDEFINEDHUMANUNDEFINED2-fluoro-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide31Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51660D2UNDEFINEDHUMANUNDEFINED2-fluoro-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide149Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51661D2UNDEFINEDHUMANUNDEFINED2-cyano-N-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide2.4Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51662D2UNDEFINEDHUMANUNDEFINED2-cyano-N-((1s,4s)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide55Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
51663D2UNDEFINEDHUMANUNDEFINEDN-((1r,4r)-4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)benzenesulfonamide34Chiu G et al., 2007Jan 15, 2025Jan 15, 2025
516645-HT7UNDEFINEDRATUNDEFINED5-CT0.5Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516655-HT7UNDEFINEDRATUNDEFINED4-(2-pyridinyl-N-oxide)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide8027Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516665-HT7UNDEFINEDRATUNDEFINED4-(2-pyridinyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide278Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516675-HT7UNDEFINEDRATUNDEFINED4-(2-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide131Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516685-HT7UNDEFINEDRATUNDEFINED4-(2-methylsulfonamidophenyl)-N-(1,2,3,tetrahydronaphthalen-1-yl)-1-piperazinehexanamide4253Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516695-HT7UNDEFINEDRATUNDEFINED4-(2-acetylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide338Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516705-HT7UNDEFINEDRATUNDEFINED4-(2-aminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide8178Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516715-HT7UNDEFINEDRATUNDEFINED4-(2-methylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide25.4Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516725-HT7UNDEFINEDRATUNDEFINED4-(2-dimethylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide0.9Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516735-HT7UNDEFINEDRATUNDEFINED4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide0.13Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516745-HT7UNDEFINEDRATUNDEFINED4-[2-(1,1-dimethylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide538Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516755-HT7UNDEFINEDRATUNDEFINED4-[2-(1-methylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1.1Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516765-HT7UNDEFINEDRATUNDEFINED4-(2-butylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide2810Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516775-HT7UNDEFINEDRATUNDEFINED4-(2-propylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide49.6Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516785-HT7UNDEFINEDRATUNDEFINED4-(2-ethylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide7.1Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516795-HT1AUNDEFINEDHUMANUNDEFINED8-OH-DPAT2.1Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516805-HT1AUNDEFINEDHUMANUNDEFINED4-(2-pyridinyl-N-oxide)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide194Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516815-HT1AUNDEFINEDHUMANUNDEFINED4-(2-pyridinyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide36.4Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516825-HT1AUNDEFINEDHUMANUNDEFINED4-(2-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide29.2Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516835-HT1AUNDEFINEDHUMANUNDEFINED4-(2-acetylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide2500Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516845-HT1AUNDEFINEDHUMANUNDEFINED4-(2-aminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide415Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516855-HT1AUNDEFINEDHUMANUNDEFINED4-(2-methylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide133Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516865-HT1AUNDEFINEDHUMANUNDEFINED4-(2-dimethylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide112Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516875-HT1AUNDEFINEDHUMANUNDEFINED4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide60.9Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516885-HT1AUNDEFINEDHUMANUNDEFINED4-[2-(1,1-dimethylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1196Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516895-HT1AUNDEFINEDHUMANUNDEFINED4-[2-(1-methylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide167Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516905-HT1AUNDEFINEDHUMANUNDEFINED4-(2-butylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide60Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516915-HT1AUNDEFINEDHUMANUNDEFINED4-(2-propylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide168Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
516925-HT1AUNDEFINEDHUMANUNDEFINED4-(2-ethylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide79.2Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51693D2UNDEFINEDUNDEFINEDUNDEFINEDHALOPERIDOL2Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51694D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-pyridinyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51695D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-fluorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide292Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51696D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-methylsulfonamidophenyl)-N-(1,2,3,tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51697D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-acetylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51698D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-methylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide107Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51699D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-dimethylaminophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide32Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51700D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-diphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide224Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51701D2UNDEFINEDUNDEFINEDUNDEFINED4-[2-(1,1-dimethylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51702D2UNDEFINEDUNDEFINEDUNDEFINED4-[2-(1-methylethyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide15Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51703D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-butylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide60Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51704D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-propylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide123Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51705D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-ethylphenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide173Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51706D2UNDEFINEDUNDEFINEDUNDEFINED4-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51707D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-chlorophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide51Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51708D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-nitrophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide681Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51709D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-cyanophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide265Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51710D2UNDEFINEDUNDEFINEDUNDEFINED6-(4-(2-hydroxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide987Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51711D2UNDEFINEDUNDEFINEDUNDEFINED6-(4-(2-acetylphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide68Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51712D2UNDEFINEDUNDEFINEDUNDEFINEDN-(1,2,3,4-tetrahydronaphthalen-1-yl)-6-(4-o-tolylpiperazin-1-yl)hexanamide143Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51713D2UNDEFINEDUNDEFINEDUNDEFINED6-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide26.4Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51714D2UNDEFINEDUNDEFINEDUNDEFINED6-(4-(2-(methylthio)phenyl)piperazin-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)hexanamide7.3Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51715D2UNDEFINEDUNDEFINEDUNDEFINED4-[2-(methylsulfonyl)phenyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51716D2UNDEFINEDUNDEFINEDUNDEFINED4-(2-carboxamidophenyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-piperazinehexanamide1000Leopoldo M et al., 2007Jan 15, 2025Jan 15, 2025
51717NR3C1UNDEFINEDHUMANUNDEFINEDdexamethasone2.1Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51718NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline4.4Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51719NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline1.1Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51720NR3C1UNDEFINEDHUMANUNDEFINED(+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1.2Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51721NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-hydroxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline0.6Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51722NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1.4Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51723NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline0.2Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51724NR3C1UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline0.7Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51725PGRUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1400Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51726PGRUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline57Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51727PGRUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline38Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51728PGRUNDEFINEDHUMANUNDEFINED(+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline2290Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51729PGRUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-hydroxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline790Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51730PGRUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1780Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51731PGRUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline190Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51732NR3C2UNDEFINEDHUMANUNDEFINEDdexamethasone7.2Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51733NR3C2UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline42Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51734NR3C2UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline48Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51735NR3C2UNDEFINEDHUMANUNDEFINED(+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline410Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51736NR3C2UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-hydroxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline21Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51737NR3C2UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline670Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51738NR3C2UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline10Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51739NR3C2UNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline980Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51740ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-hydroxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline290Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51741ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(E-methylbutenyl)thienylmethylidene))-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]-quinoline346Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51742ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-methoxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline110Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51743ARUNDEFINEDHUMANUNDEFINED(+/-)-(Z)-5-(2'-(3'-(1''-hydroxyethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1530Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51744ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-((E)-1''-hydroxyiminoethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno-[3,4-f]quinoline290Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51745ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-(1''-hydroxy-2'',2'',2''-trifluoroethyl)thienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline1900Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51746ARUNDEFINEDHUMANUNDEFINED(Z)-5-(2'-(3'-methoxymethylthienylmethylidene))1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5H-chromeno[3,4-f]quinoline150Hudson AR et al., 2007Jan 15, 2025Jan 15, 2025
51747CHRNA4UNDEFINEDRATUNDEFINEDNicotine6.2Jensen AA et al., 2007Jan 15, 2025Jan 15, 2025
51748CHRNA4UNDEFINEDRATUNDEFINED(1R,9R,18S,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-phenyl-10,26-dioxa-8,15,24,31-tetraazaundecacyclo[29.5.2.0^{1,32}.0^{2,7}.0^{8,36}.0^{9,22}.0^{13,21}.0^{15,19}.0^{18,23}.0^{25,35}.0^{29,34}]octatriaconta-2,4,6,12,28-pentaene>10000Jensen AA et al., 2007Jan 15, 2025Jan 15, 2025