The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 1-28 of 28 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
899965-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900215-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900465-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine16Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90071Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine580Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90095Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine260Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90120D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90145D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90170D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90195CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine120Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90220CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90245NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4300Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90270DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90295SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine8100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90320H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
899975-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900225-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1.1Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900475-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine6.4Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90072Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine340Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90096Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine360Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90121D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine4100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90146D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90171D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90196CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine90Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90221CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90246NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine3700Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90271DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine4800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90296SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine3200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90321H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1200Rickli A et al 2015Jan 15, 2025Jan 28, 2025