The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 50,001-51,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
52749SLC6A4UNDEFINEDRATUNDEFINED1,6-Dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol28Zhang A et al., 2007Jan 15, 2025Jan 15, 2025
52750SLC6A4UNDEFINEDRATUNDEFINED6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol100Zhang A et al., 2007Jan 15, 2025Jan 15, 2025
52751SLC6A4UNDEFINEDRATUNDEFINED6-Methyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylen-1-ol14Zhang A et al., 2007Jan 15, 2025Jan 15, 2025
52752SLC6A4UNDEFINEDRATUNDEFINED(R)-5a,6-dimethyl-1,5,5a,6,7,8-hexahydro-6-aza-benzo[mno]aceanthrylene7Zhang A et al., 2007Jan 15, 2025Jan 15, 2025
52753D2UNDEFINEDHUMANUNDEFINEDZiprasidone5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52754D2UNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52755D2UNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide10Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52756D2UNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide15Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52757D2UNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide8Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52758D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isoxazole-5-carboxamide3Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52759D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)furan-2-carboxamide5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52760D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-3-phenylpropanamide33Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52761D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2-phenylacetamide26Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52762D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide6Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52763D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide6Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52764D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52765D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide15Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52766D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide22Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52767D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide67Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52768D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide21Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52769D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide27Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52770D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide34Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52771D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide22Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52772D2UNDEFINEDHUMANUNDEFINED6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-amine21Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52773D2UNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide10Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527745-HT2AUNDEFINEDHUMANUNDEFINEDZiprasidone0.08Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527755-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide0.68Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527765-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide1.65Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527775-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide0.65Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527785-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide0.45Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527795-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide0.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527805-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide0.25Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527815-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide0.33Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527825-HT2AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide0.15Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527835-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isoxazole-5-carboxamide0.08Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527845-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)furan-2-carboxamide0.55Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527855-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-3-phenylpropanamide0.95Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527865-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2-phenylacetamide0.04Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527875-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide0.95Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527885-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide2.45Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527895-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide0.1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527905-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide3Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527915-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide4.75Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527925-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide0.75Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527935-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide0.3Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527945-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide0.45Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527955-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide0.01Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527965-HT2AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide0.01Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527975-HT2AUNDEFINEDHUMANUNDEFINED6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-amine0.09Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527985-HT1AUNDEFINEDHUMANUNDEFINEDZiprasidone4Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
527995-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide7.7Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528005-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide7.8Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528015-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide2Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528025-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide2Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528035-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide2Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528045-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide1.1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528055-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528065-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isoxazole-5-carboxamide6.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528075-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)furan-2-carboxamide7.9Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528085-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-3-phenylpropanamide37.2Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528095-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2-phenylacetamide20.9Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528105-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)nicotinamide4.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528115-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-fluorobenzamide66.7Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528125-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-chlorobenzamide56Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528135-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-4-methylbenzamide28.1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528145-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)benzamide41.8Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528155-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide12Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528165-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)cyclopropanecarboxamide12Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528175-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)butyramide5.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528185-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)propionamide5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528195-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)acetamide7.5Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528205-HT1AUNDEFINEDHUMANUNDEFINED6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-amine2Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528215-HT1AUNDEFINEDHUMANUNDEFINEDN-(6-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)-2,2,2-trifluoroacetamide4.9Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
528225-HT1AUNDEFINEDHUMANUNDEFINEDN-(5-(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-2,3-dihydro-1H-inden-1-yl)isobutyramide1Graham JM et al., 2008Jan 15, 2025Jan 15, 2025
52823CHRNA4UNDEFINEDRATUNDEFINED3-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine2950Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52824CHRNA4UNDEFINEDRATUNDEFINEDNicotine7Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52825CHRNA4UNDEFINEDRATUNDEFINED2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine10Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52826CHRNA4UNDEFINEDRATUNDEFINED2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine251Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52827CHRNA4UNDEFINEDRATUNDEFINED(+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridine16Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52828CHRNA4UNDEFINEDRATUNDEFINED(S)-6-fluoro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine1995Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52829CHRNA4UNDEFINEDRATUNDEFINED(R)-6-fluoro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine316Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52830CHRNA4UNDEFINEDRATUNDEFINED(R)-6-bromo-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine691Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52831CHRNA4UNDEFINEDRATUNDEFINED(S)-6-chloro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine3715Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52832CHRNA4UNDEFINEDRATUNDEFINED(R)-6-chloro-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine147Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52833CHRNA4UNDEFINEDRATUNDEFINED(S)-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine2750Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52834CHRNA4UNDEFINEDRATUNDEFINED(R)-2-(pyrrolidin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine125Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52835CHRNA4UNDEFINEDRATUNDEFINED(+)-6-chloro-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine3460Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52836CHRNA4UNDEFINEDRATUNDEFINED(-)-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine1995Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52837CHRNA4UNDEFINEDRATUNDEFINED(+/-)-2-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine>10000Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52838CHRNA4UNDEFINEDRATUNDEFINED6-chloro-3-(piperidin-3-yl)-1H-pyrrolo[2,3-b]pyridine2950Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52839CHRNA4UNDEFINEDRATUNDEFINED(R)-2-((1-methylpyrrolidin-2-yl)methyl)-1H-pyrrolo[2,3-b]pyridine2511Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52840CHRNA4UNDEFINEDRATUNDEFINED(S)-2-((1-methylpyrrolidin-2-yl)methyl)-1H-pyrrolo[2,3-b]pyridine691Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52841CHRNA4UNDEFINEDRATUNDEFINEDMethyl-((E)-4-pyridin-3-yl-but-3-enyl)-amine26Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52842CHRNA4UNDEFINEDRATUNDEFINED(S)-5-(5-methoxypyridin-3-yl)-N-methylpent-4-en-2-amine11Stoit AR et al., 2008Jan 15, 2025Jan 15, 2025
52843CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52844CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 4-cyano-1-phenyl-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52845CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 4-methyl-1-phenyl-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52846CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 4-cyano-1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide280Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52847CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1600Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52848CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide2800Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52849CB1UNDEFINEDHUMANUNDEFINEDN-morpholin-4-yl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52850CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2800Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52851CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide14Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52852CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide280Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52853CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide28Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52854CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide5.6Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52855CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide35Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52856CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide30Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52857CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide42Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52858CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide28Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52859CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide38Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52860CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide56Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52861CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide37Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52862CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1850Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52863CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(4-chlorophenyl)-3-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-4-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52864CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-3-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52865CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-4-cyano-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52866CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexylmethyl 1-(4-chlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide110Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52867CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide110Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52868CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(4-chlorophenyl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide280Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52869CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide2820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52870CB1UNDEFINEDHUMANUNDEFINEDSR 1445282820Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52871CB1UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide2.3Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52872CB1UNDEFINEDHUMANUNDEFINEDRimonabant12Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52873CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4,6-trichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide28Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52874CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4,6-trichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide110Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52875CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dihlorobenzyl 1-(2,4,6-trichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide280Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52876CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4,6-trichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide1800Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52877CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide35Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52878CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide35Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52879CB1UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide1600Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52880CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52881CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 4-cyano-1-phenyl-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52882CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 4-methyl-1-phenyl-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52883CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 4-cyano-1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52884CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide65Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52885CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide390Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52886CB2UNDEFINEDHUMANUNDEFINEDN-morpholin-4-yl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52887CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2400Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52888CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide1.3Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52889CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide1370Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52890CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide29Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52891CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1.7Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52892CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide150Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52893CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide20Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52894CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide87Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52895CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52896CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide980Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52897CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide64Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52898CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide510Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52899CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1730Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52900CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(4-chlorophenyl)-3-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-4-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52901CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-3-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-4-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52902CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-4-cyano-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52903CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexylmethyl 1-(4-chlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide390Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52904CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2180Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52905CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(4-chlorophenyl)-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1750Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52906CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(4-chlorophenyl)-5-(1H-pyrrol-1-yl)-1Hpyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52907CB2UNDEFINEDHUMANUNDEFINEDSR 1445285.4Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52908CB2UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide112Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52909CB2UNDEFINEDHUMANUNDEFINEDRimonabant790Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52910CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4,6-trichlorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide390Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52911CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4,6-trichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52912CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dihlorobenzyl 1-(2,4,6-trichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52913CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4,6-trichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52914CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide570Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52915CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52916CB2UNDEFINEDHUMANUNDEFINEDN-piperidin-1-yl 1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1Hpyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2008Jan 15, 2025Jan 15, 2025
52917D1UNDEFINEDRATUNDEFINEDAPOMORPHINE1010Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52918D1UNDEFINEDRATUNDEFINED(R)-(-)-N-butyl-2-methoxy-11-hydroxynoraporphine>10000Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52919D1UNDEFINEDRATUNDEFINED2-methoxy-11-hydroxy-N-propylnoraporphine1690Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52920D1UNDEFINEDRATUNDEFINED(R)-(-)-N-ethyl-2-methoxy-11-hydroxynoraporphine130Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52921D1UNDEFINEDRATUNDEFINED2-Methoxy-11-hydroxyaporphine46Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52922D1UNDEFINEDRATUNDEFINED11-Hydroxy-N-propylnoraporphine699Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52923D1UNDEFINEDRATUNDEFINED(R)-6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol26.5Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52924D1UNDEFINEDRATUNDEFINED2-methoxyapomorphine>10000Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52925D1UNDEFINEDRATUNDEFINED2-Methoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol6450Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52926D1UNDEFINEDRATUNDEFINEDNPA3410Si YG et al., 2008Jan 15, 2025Jan 15, 2025
52927SRCUNDEFINEDHUMANUNDEFINEDN-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide2900Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52928SRCUNDEFINEDHUMANUNDEFINEDGleevec>10000Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52929SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide272Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52930SRCUNDEFINEDHUMANUNDEFINEDN-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide1137Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52931SRCUNDEFINEDHUMANUNDEFINEDN-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide169Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52932SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide900Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52933SRCUNDEFINEDHUMANUNDEFINEDN-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide334Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52934SRCUNDEFINEDHUMANUNDEFINEDN-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide247Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52935SRCUNDEFINEDHUMANUNDEFINEDN-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide718Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52936SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide522Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52937SRCUNDEFINEDHUMANUNDEFINEDN-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide64Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52938SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide170Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52939SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide263Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52940SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide199Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52941SRCUNDEFINEDHUMANUNDEFINEDN-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide569Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52942SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide200Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52943SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide165Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52944SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide221Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52945SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide219Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52946SRCUNDEFINEDHUMANUNDEFINEDN-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide195Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52947SRCUNDEFINEDHUMANUNDEFINEDN-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide464Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52948SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide217Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52949SRCUNDEFINEDHUMANUNDEFINEDN-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide354Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52950SRCUNDEFINEDHUMANUNDEFINED2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide2000Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52951ABL1UNDEFINEDHUMANUNDEFINEDGleevec13Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52952ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide1260Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52953ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide920Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52954ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide760Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52955ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide406Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52956ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide400Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52957ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide369Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52958ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide272Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52959ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide225Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52960ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide217Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52961ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide210Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52962ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide195Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52963ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-methoxybenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide189Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52964ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(3-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide167Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52965ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide104Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52966ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide92Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52967ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide89Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52968ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-nitrobenzylthio)-1,3,4-thiadiazol-2-yl)-2-chlorobenzamide83Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52969ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(3-chlorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide73Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52970ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(benzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide70Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52971ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-bromobenzylthio)-1,3,4-thiadiazol-2-yl)-4-chlorobenzamide47Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52972ABL1UNDEFINEDHUMANUNDEFINEDN-(5-(4-fluorobenzylthio)-1,3,4-thiadiazol-2-yl)-4-fluorobenzamide44Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52973ABL1UNDEFINEDHUMANUNDEFINED2-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide1300Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52974ABL1UNDEFINEDHUMANUNDEFINED4-iodo-N-(5-phenethyl-1,3,4-thiadiazol-2-yl)benzamide400Radi M et al., 2008Jan 15, 2025Jan 15, 2025
52975CB1UNDEFINEDHUMANUNDEFINEDRimonabant1.8Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52976CB1UNDEFINEDHUMANUNDEFINEDibipinabant4.1Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52977CB1UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N-ethyl-3-methylbenzofuran-2-carboxamide92Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52978CB1UNDEFINEDHUMANUNDEFINEDazepan-1-yl(5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-yl)methanone193Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52979CB1UNDEFINEDHUMANUNDEFINED5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethyl-N-phenethylbenzofuran-2-carboxamide172Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52980CB1UNDEFINEDHUMANUNDEFINED5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide198Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52981CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide108Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52982CB1UNDEFINEDHUMANUNDEFINEDN-butyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide94Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52983CB1UNDEFINEDHUMANUNDEFINEDN-cyclopentyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide90Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52984CB1UNDEFINEDHUMANUNDEFINEDN-(4-fluorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide62Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52985CB1UNDEFINEDHUMANUNDEFINED5-(3,5-dimethyl-piperidine-1-sulfonyl)-3-methyl-benzofuran-2-carboxylic acid 4-methyl-benzylamide79Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52986CB1UNDEFINEDHUMANUNDEFINEDN-(2-ethoxybenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide97Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52987CB1UNDEFINEDHUMANUNDEFINEDN-(2-methoxybenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide58Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52988CB1UNDEFINEDHUMANUNDEFINEDN-(2-chlorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide58Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52989CB1UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethylbenzofuran-2-carboxamide59Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52990CB1UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide77Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52991CB1UNDEFINEDHUMANUNDEFINED5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzofuran-2-carboxamide5Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52992CB2UNDEFINEDHUMANUNDEFINEDRimonabant554Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52993CB2UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N-ethyl-3-methylbenzofuran-2-carboxamide3100Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52994CB2UNDEFINEDHUMANUNDEFINEDazepan-1-yl(5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-yl)methanone4900Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52995CB2UNDEFINEDHUMANUNDEFINED5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-phenethylbenzofuran-2-carboxamide6000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52996CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide>10000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52997CB2UNDEFINEDHUMANUNDEFINEDN-butyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide9400Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52998CB2UNDEFINEDHUMANUNDEFINEDN-cyclopentyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide7400Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
52999CB2UNDEFINEDHUMANUNDEFINEDN-(4-fluorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide4000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53000CB2UNDEFINEDHUMANUNDEFINED5-(3,5-dimethyl-piperidine-1-sulfonyl)-3-methyl-benzofuran-2-carboxylic acid 4-methyl-benzylamide>10000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53001CB2UNDEFINEDHUMANUNDEFINEDN-(2-ethoxybenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide9900Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53002CB2UNDEFINEDHUMANUNDEFINEDN-(2-methoxybenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide>10000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53003CB2UNDEFINEDHUMANUNDEFINEDN-(2-chlorobenzyl)-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide4800Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53004CB2UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N,3-dimethylbenzofuran-2-carboxamide6600Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53005CB2UNDEFINEDHUMANUNDEFINEDN-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methylbenzofuran-2-carboxamide6600Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53006CB2UNDEFINEDHUMANUNDEFINED5-(3,5-dimethylpiperidin-1-ylsulfonyl)-3-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzofuran-2-carboxamide>10000Foloppe N et al., 2008Jan 15, 2025Jan 15, 2025
53007MORUNDEFINEDHUMANUNDEFINEDNaltrexone0.3Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53008MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(thiophen-2'-yl)acetamido]morphinan0.38Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53009MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(thiophen-2'-yl)acetamido]morphinan0.43Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53010MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-methoxy)benzylacetamido]morphinan (0.27Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53011MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzylacetamido)morphinan0.16Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53012MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)phenylacetamido]morphinan0.13Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53013MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan0.12Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53014MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(cinnamoylacetamido)morphinan0.06Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53015MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carboxy)benzamido]morphinan10.08Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53016MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-[(3'-dimethylamino)benzamido]morphinan1.2Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53017MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-tert-butoxycarbonylamino)benzamido]morphinan0.92Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53018MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)benzamido]morphinan0.12Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53019MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-amino)benzamido]morphinan0.43Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53020MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan0.31Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53021MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan0.26Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53022MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan0.21Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53023MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan0.21Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53024MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan0.19Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53025MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-nitro)benzamido]morphinan0.19Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53026MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan0.18Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53027MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3'-methoxy)benzamido]morphinan0.16Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53028MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan0.13Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53029MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan0.1Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53030MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan0.05Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53031MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(D-glucopyranosyl)acetamido]morphinan0.64Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53032MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(D-glucopyranosyl)acetamido]morphinan0.67Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53033MORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(2',3',4',6'-tetra-O-benzyl-D-glucopyranosyl)acetamido]morphinan1.49Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53034MORUNDEFINEDHUMANUNDEFINEDnalmefene0.91Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53035DORUNDEFINEDHUMANUNDEFINEDNaltrexone16.31Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53036DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(thiophen-2'-yl)acetamido]morphinan2.07Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53037DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(thiophen-2'-yl)acetamido]morphinan32.4Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53038DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-methoxy)benzylacetamido]morphinan (19.91Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53039DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzylacetamido)morphinan28Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53040DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)phenylacetamido]morphinan15.8Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53041DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan12.2Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53042DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(cinnamoylacetamido)morphinan8.22Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53043DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carboxy)benzamido]morphinan79.23Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53044DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-[(3'-dimethylamino)benzamido]morphinan8.5Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53045DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-tert-butoxycarbonylamino)benzamido]morphinan25.29Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53046DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)benzamido]morphinan3.8Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53047DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-amino)benzamido]morphinan36.52Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53048DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan56.3Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53049DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan17.59Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53050DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan27.18Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53051DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan12.4Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53052DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan6.83Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53053DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-nitro)benzamido]morphinan4.23Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53054DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan9.72Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53055DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3'-methoxy)benzamido]morphinan5.82Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53056DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan2.73Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53057DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan0.79Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53058DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan1.4Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53059DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(D-glucopyranosyl)acetamido]morphinan99Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53060DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(D-glucopyranosyl)acetamido]morphinan36.94Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53061DORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(2',3',4',6'-tetra-O-benzyl-D-glucopyranosyl)acetamido]morphinan24.52Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53062DORUNDEFINEDHUMANUNDEFINEDnalmefene13.26Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53063KORUNDEFINEDHUMANUNDEFINEDNaltrexone0.81Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53064KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(thiophen-2'-yl)acetamido]morphinan2.74Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53065KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(thiophen-2'-yl)acetamido]morphinan1.2Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53066KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-methoxy)benzylacetamido]morphinan (0.42Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53067KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzylacetamido)morphinan0.43Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53068KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)phenylacetamido]morphinan0.45Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53069KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(hydroxycinnamoylacetamido)morphinan0.09Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53070KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(cinnamoylacetamido)morphinan0.91Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53071KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carboxy)benzamido]morphinan150.61Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53072KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-[(3'-dimethylamino)benzamido]morphinan1.7Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53073KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-tert-butoxycarbonylamino)benzamido]morphinan0.79Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53074KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-methoxy)benzamido]morphinan0.24Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53075KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-amino)benzamido]morphinan0.4Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53076KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(2'-pyridyl)acetamido]morphinan0.39Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53077KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',5'-dimethoxy)benzamido]morphinan0.29Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53078KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-carbomethoxy)benzamido]morphinan0.73Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53079KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-(benzamido)morphinan0.78Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53080KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3', 5'-dimethoxy)benzamido]morphinan2.41Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53081KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-nitro)benzamido]morphinan0.28Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53082KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(benzamido)morphinan0.16Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53083KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(3'-methoxy)benzamido]morphinan0.72Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53084KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3'-hydroxy)benzamido]morphinan0.06Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53085KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(3',4'-dichloro)benzamido]morphinan0.1Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53086KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-[(4'-chloro)benzamido]morphinan0.37Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53087KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-beta-(D-glucopyranosyl)acetamido]morphinan4.5Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53088KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(D-glucopyranosyl)acetamido]morphinan2.03Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53089KORUNDEFINEDHUMANUNDEFINED17-cyclopropylmethyl-3,14-beta-dihydroxy-4,5-alpha-epoxy-6-alpha-[(2',3',4',6'-tetra-O-benzyl-D-glucopyranosyl)acetamido]morphinan0.51Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53090KORUNDEFINEDHUMANUNDEFINEDnalmefene1.03Ghirmai S et al., 2008Jan 15, 2025Jan 15, 2025
53091CB1UNDEFINEDHUMANUNDEFINED(R)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone3.3Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53092CB1UNDEFINEDHUMANUNDEFINED1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-4-(4-fluoro-phenyl)-1,2,3,6-tetrahydro-pyridine13Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53093CB1UNDEFINEDHUMANUNDEFINED(6-methyl-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone509Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53094CB1UNDEFINEDHUMANUNDEFINED6-(morpholine-4-carbonyl)-2,2-diphenyl-benzo[1,3]dioxole-5-carbonitrile277Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53095CB1UNDEFINEDHUMANUNDEFINED(6-bromo-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone873Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53096CB1UNDEFINEDHUMANUNDEFINED(6-chloro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-yl-methanone216Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53097CB1UNDEFINEDHUMANUNDEFINED4-[6-fluoro-2,2-bis-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-ylmethyl]-morpholine1000Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53098CB1UNDEFINEDHUMANUNDEFINED1-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)-4,4-difluoropiperidine3Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53099CB1UNDEFINEDHUMANUNDEFINED4-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-ylsulfonyl)morpholine25Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53100CB1UNDEFINEDHUMANUNDEFINED4-(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-ylsulfonyl)morpholine9Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53101CB1UNDEFINEDHUMANUNDEFINED(2-(2,4-dichlorophenyl)-6-fluoro-2-(2-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone4Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53102CB1UNDEFINEDHUMANUNDEFINED(6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone18Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53103CB1UNDEFINEDHUMANUNDEFINED(S)-(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(2-methoxypyrrolidin-1-yl)methanone46Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53104CB1UNDEFINEDHUMANUNDEFINED(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(4,4-difluoropiperidin-1-yl)methanone6Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53105CB1UNDEFINEDHUMANUNDEFINED(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(morpholino)methanone7Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53106CB1UNDEFINEDHUMANUNDEFINED[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone4Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53107CB1UNDEFINEDHUMANUNDEFINED(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone4Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53108CB1UNDEFINEDHUMANUNDEFINED(2,2-bis(2,4-difluorophenyl)-6-fluorobenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone1Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53109CB1UNDEFINEDHUMANUNDEFINED(2-(2,4-dichlorophenyl)-6-fluoro-2-(4-methoxyphenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone2Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53110CB1UNDEFINEDHUMANUNDEFINED(6-fluoro-2,2-bis(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone7Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53111CB1UNDEFINEDHUMANUNDEFINED(6-fluoro-2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone11Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53112CB1UNDEFINEDHUMANUNDEFINED(6-fluoro-2,2-diphenyl-benzo[1,3]dioxol-5-yl)-morpholin-4-ylmethanone15Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53113CB1UNDEFINEDHUMANUNDEFINED(2,2-diphenyl-[1,3]dioxolo[4,5-c]pyridin-6-yl)-piperidin-1-ylmethanone13Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53114CB1UNDEFINEDHUMANUNDEFINED(2-(2,4-dichlorophenyl)-2-(4-fluorophenyl)benzo[d][1,3]dioxol-5-yl)(morpholino)methanone30Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53115CB1UNDEFINEDHUMANUNDEFINED(2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(morpholino)methanone50Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53116CB1UNDEFINEDHUMANUNDEFINED(2,2-diphenylbenzo[d][1,3]dioxol-5-yl)(piperidin-1-yl)methanone28Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53117CB1UNDEFINEDHUMANUNDEFINED1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-piperidine38Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53118CB1UNDEFINEDHUMANUNDEFINED(S)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone35Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53119CB1UNDEFINEDHUMANUNDEFINEDRimonabant6Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53120CB1UNDEFINEDHUMANUNDEFINED(S)-3-(4-chlorophenyl)-N-(4-chlorophenylsulfonyl)-N'-methyl-4-phenyl-4,5-dihydropyrazole-1-carboxamidine8Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53121CB1UNDEFINEDHUMANUNDEFINED(6-(methylsulfonyl)-1-pentyl-1H-indol-3-yl)(naphthalen-2-yl)methanone110Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53122CB1UNDEFINEDHUMANUNDEFINED1-(4-(4-chlorophenyl)-5,6-dihydropyridin-1(2H)-yl)-3,3-diphenylpropan-1-one1500Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53123CB2UNDEFINEDHUMANUNDEFINED(R)-[2-(2,4-dichloro-phenyl)-6-fluoro-2-(4-fluoro-phenyl)-benzo[1,3]dioxol-5-yl]-morpholin-4-yl-methanone3Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53124CB2UNDEFINEDHUMANUNDEFINED1-(2,2-diphenyl-benzo[1,3]dioxole-5-sulfonyl)-4-(4-fluoro-phenyl)-1,2,3,6-tetrahydro-pyridine>10000Alig L et al., 2008Jan 15, 2025Jan 15, 2025
53125CHRNA4UNDEFINEDRATUNDEFINEDN-methyl-1-((pyridin-3-yloxy)methyl)cyclopropanamine hydrochloride3Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53126CHRNA4UNDEFINEDRATUNDEFINED1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride110Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53127CHRNA4UNDEFINEDRATUNDEFINED[1-(5-bromo-pyridin-3-yloxymethyl)-cyclopropyl]-dimethyl-amine; hydrochloride273Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53128CHRNA4UNDEFINEDRATUNDEFINED1-((6-bromopyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride394Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53129CHRNA4UNDEFINEDRATUNDEFINED1-(6-chloro-pyridin-3-yloxymethyl)-cyclopropylamine; hydrochloride98Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53130CHRNA4UNDEFINEDRATUNDEFINED1-((6-chloropyridin-3-yloxy)methyl)-N,N-dimethylcyclopropanamine hydrochloride304Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53131CHRNA4UNDEFINEDRATUNDEFINED1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride266Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53132CHRNA4UNDEFINEDRATUNDEFINEDN,N-dimethyl-1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride1090Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53133CHRNA4UNDEFINEDRATUNDEFINEDN-methyl-1-((5-vinylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride70.1Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53134CHRNA4UNDEFINEDRATUNDEFINED1-((5-ethynylpyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride6.56Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53135CHRNA4UNDEFINEDRATUNDEFINED1-((5-bromo-6-chloropyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride5.37Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53136CHRNA4UNDEFINEDRATUNDEFINED1-((5-bromopyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride1.07Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53137CHRNA4UNDEFINEDRATUNDEFINED1-((6-bromopyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride38.8Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53138CHRNA4UNDEFINEDRATUNDEFINED1-((6-chloropyridin-3-yloxy)methyl)-N-methylcyclopropanamine hydrochloride13Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53139CHRNA4UNDEFINEDRATUNDEFINEDN-methyl-1-((6-methylpyridin-3-yloxy)methyl)cyclopropanamine hydrochloride40Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53140CHRNA4UNDEFINEDRATUNDEFINED3-((1-(pyrrolidin-1-yl)cyclopropyl)methoxy)pyridine1610Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53141CHRNA4UNDEFINEDRATUNDEFINEDN-ethyl-1-((pyridin-3-yloxy)methyl)cyclopropanamine1010Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53142CHRNA4UNDEFINEDRATUNDEFINED1-(pyridin-3-yloxymethyl)-cyclopropylamine; hydrochloride34Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53143CHRNA4UNDEFINEDRATUNDEFINEDdimethyl-[1-(pyridin-3-yloxymethyl)-cyclopropyl]-amine; hydrochloride95Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53144CHRNA4UNDEFINEDRATUNDEFINEDmethyl-{1-[2-(pyridin-3-yloxy)-ethyl]-cyclopropyl}-amine fumarate109Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53145CHRNA4UNDEFINEDRATUNDEFINEDcis-methyl-{1-[3-(pyridin-3-yloxy)-propenyl]-cyclopropyl}-amine; hydrochloride2280Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53146CHRNA4UNDEFINEDRATUNDEFINEDtrans-methyl-{1-[3-(pyridin-3-yloxy)-propenyl]-cyclopropyl}-amine; hydrochloride1100Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53147CHRNA4UNDEFINEDRATUNDEFINEDmethyl-{1-[3-(pyridin-3-yloxy)-propyl]-cyclopropyl}-amine fumarate2460Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53148CHRNA4UNDEFINEDRATUNDEFINEDmethyl-[1-(2-pyridin-3-yl-vinyl)-cyclopropyl]-amine fumarate1160Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53149CHRNA4UNDEFINEDRATUNDEFINEDN-methyl-1-(2-(pyridin-3-yl)ethyl)cyclopropanamine hydrochloride251Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53150CHRNA4UNDEFINEDRATUNDEFINEDNicotine4Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53151CHRNA4UNDEFINEDRATUNDEFINEDAcetylcholine39Charton Y et al., 2008Jan 15, 2025Jan 15, 2025
53152A1UNDEFINEDHUMANUNDEFINED2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione379Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53153A1UNDEFINEDHUMANUNDEFINEDXAC9Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53154A1UNDEFINEDHUMANUNDEFINEDCaffeine (1,3,7-trimethylxanthine)>10000Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53155A1UNDEFINEDHUMANUNDEFINED7-bromo-eudistomin D7370Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53156A1UNDEFINEDHUMANUNDEFINED2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione>10000Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53157A1UNDEFINEDHUMANUNDEFINED2,4-dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione>10000Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53158A2AUNDEFINEDHUMANUNDEFINED2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione893Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53159A2AUNDEFINEDHUMANUNDEFINEDCGS 2168046.2Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53160A2AUNDEFINEDHUMANUNDEFINEDCaffeine (1,3,7-trimethylxanthine)>10000Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53161A2AUNDEFINEDHUMANUNDEFINED2,4,9-trimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione4190Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53162A2AUNDEFINEDHUMANUNDEFINED7-bromo-eudistomin D4920Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53163A2AUNDEFINEDHUMANUNDEFINED2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione6940Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53164A2AUNDEFINEDHUMANUNDEFINED2,4-dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione>10000Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53165A3UNDEFINEDHUMANUNDEFINEDNECA20Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53166A3UNDEFINEDHUMANUNDEFINED2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione13.9Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53167A3UNDEFINEDHUMANUNDEFINED2,4,9-trimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione3190Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53168A3UNDEFINEDHUMANUNDEFINED7-bromo-eudistomin D2050Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53169A3UNDEFINEDHUMANUNDEFINED2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione332Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53170A3UNDEFINEDHUMANUNDEFINED2,4-dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione526Ohshita K et al., 2007Jan 15, 2025Jan 15, 2025
53171SLC6A4UNDEFINEDRATUNDEFINED3-(4-(4-cyclohexylpiperazin-1-yl)butyl)benzo[d]thiazole-2(3H)-thione1402Mésangeau C et al., 2008Jan 15, 2025Jan 15, 2025
53172Alpha1AUNDEFINEDHUMANUNDEFINEDTamsulosin0.19Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53173Alpha1AUNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea11Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53174Alpha1AUNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea82Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53175Alpha1AUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea6.5Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53176Alpha1AUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea51Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53177Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea6.2Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53178Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea33Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53179Alpha1AUNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea3.6Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53180Alpha1AUNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea51Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53181Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea5.3Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53182Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea52Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53183Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea1.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53184Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea26Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53185Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea3.1Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53186Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea14Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53187Alpha1AUNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea34Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53188Alpha1AUNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea101Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53189Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea74Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53190Alpha1AUNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea110Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53191Alpha1AUNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea5.1Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53192Alpha1AUNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea22Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53193Alpha1AUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea38Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53194Alpha1AUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea155Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53195Alpha1AUNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea11Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53196Alpha1AUNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea48Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53197Alpha1BUNDEFINEDHUMANUNDEFINEDTamsulosin2Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53198Alpha1BUNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea69Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53199Alpha1BUNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea706Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53200Alpha1BUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea112Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53201Alpha1BUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea483Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53202Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea50Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53203Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea289Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53204Alpha1BUNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea60Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53205Alpha1BUNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea963Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53206Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea36Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53207Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea299Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53208Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea36.4Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53209Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea259Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53210Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea76Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53211Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea475Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53212Alpha1BUNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea81Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53213Alpha1BUNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea207Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53214Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea214Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53215Alpha1BUNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea475Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53216Alpha1BUNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea71Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53217Alpha1BUNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea277Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53218Alpha1BUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea107Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53219Alpha1BUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea223Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53220Alpha1BUNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea39Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53221Alpha1BUNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea373Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53222Alpha1DUNDEFINEDHUMANUNDEFINEDTamsulosin0.2Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53223Alpha1DUNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea15Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53224Alpha1DUNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea62Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53225Alpha1DUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea3.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53226Alpha1DUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea25Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53227Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea2.6Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53228Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea16Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53229Alpha1DUNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea1.6Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53230Alpha1DUNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea72Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53231Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea4.8Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53232Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea92Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53233Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea1.2Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53234Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea52Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53235Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea2.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53236Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea26.5Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53237Alpha1DUNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea2.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53238Alpha1DUNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea64Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53239Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea20Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53240Alpha1DUNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea92Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53241Alpha1DUNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea1.5Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53242Alpha1DUNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea29Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53243Alpha1DUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea8.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53244Alpha1DUNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea73Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53245Alpha1DUNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea3Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53246Alpha1DUNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea46Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53247D2UNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea120Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53248D2UNDEFINEDHUMANUNDEFINED1-(3-fluorobenzyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea183Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53249D2UNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea6.5Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53250D2UNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2,4,6-trichlorophenyl)urea103Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53251D2UNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea4.7Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53252D2UNDEFINEDHUMANUNDEFINED1-(2,6-dichlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea55Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53253D2UNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea54Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53254D2UNDEFINEDHUMANUNDEFINED1-(3,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea127Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53255D2UNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea2.4Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53256D2UNDEFINEDHUMANUNDEFINED1-(2,6-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea22Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53257D2UNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea0.46Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53258D2UNDEFINEDHUMANUNDEFINED1-(2,5-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea199Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53259D2UNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea0.69Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53260D2UNDEFINEDHUMANUNDEFINED1-(2,4-difluorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea35.5Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53261D2UNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea1.2Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53262D2UNDEFINEDHUMANUNDEFINED1-(5-chloro-2-methoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea99Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53263D2UNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea892Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53264D2UNDEFINEDHUMANUNDEFINED1-(2,4-dimethoxyphenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea288Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53265D2UNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea84Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53266D2UNDEFINEDHUMANUNDEFINED1-(3-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea108Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53267D2UNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea921Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53268D2UNDEFINEDHUMANUNDEFINED1-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-3-(2-methoxyphenyl)urea390Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53269D2UNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea33Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53270D2UNDEFINEDHUMANUNDEFINED1-(2-chlorophenyl)-3-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)urea878Chiu G et al., 2008Jan 15, 2025Jan 15, 2025
53271CHRNA4UNDEFINEDRATUNDEFINEDEpibatidine0.026Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53272CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(6-fluoro-5-(3-methoxyphenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.12Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53273CHRNA4UNDEFINEDRATUNDEFINEDrac-3-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride0.16Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53274CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(6-fluoro-5-(3-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.053Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53275CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(6-fluoro-5-(4-nitrophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.009Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53276CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(6-fluoro-5-(3-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.087Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53277CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(6-fluoro-5-(4-fluorophenyl)pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.029Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53278CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(5-(3-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.073Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53279CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(5-(4-chlorophenyl)-6-fluoropyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.044Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53280CHRNA4UNDEFINEDRATUNDEFINEDrac-2-(6-fluoro-5-phenylpyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane hydrochloride0.24Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53281CHRNA4UNDEFINEDRATUNDEFINEDrac-3-(3-methoxyphenyl)deschloroepibatidine dihydrochloride0.43Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53282CHRNA4UNDEFINEDRATUNDEFINEDrac-3'-(3-aminophenyl)deschloroepibatidine trihydrochloride1.16Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53283CHRNA4UNDEFINEDRATUNDEFINEDrac-3-(4-aminophenyl)deschloroepibatidine trihydrochloride0.34Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53284CHRNA4UNDEFINEDRATUNDEFINEDrac-3'-(3-nitrophenyl)deschloroepibatidine dihydrochloride0.17Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53285CHRNA4UNDEFINEDRATUNDEFINEDrac-3'-(4-nitrophenyl)deschloroepibatidine dihydrochloride0.34Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53286CHRNA4UNDEFINEDRATUNDEFINEDrac-3'-(3-fluorophenyl)deschloroepibatidine dihydrochloride0.2Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53287CHRNA4UNDEFINEDRATUNDEFINED3'-(4-fluorophenyl)deschloroepibatidine0.15Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53288CHRNA4UNDEFINEDRATUNDEFINEDrac-3'-(3-chlorophenyl)deschloroepibatidine dihydrochloride0.17Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53289CHRNA4UNDEFINEDRATUNDEFINED3-(4-chlorophenyl)deschloroepibatidine0.21Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53290CHRNA4UNDEFINEDRATUNDEFINEDrac-3-phenyldeschloroepibatidine dihydrochloride0.5Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53291CHRNA4UNDEFINEDRATUNDEFINEDvarenicline0.12Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53292CHRNA4UNDEFINEDRATUNDEFINEDNicotine1.5Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53293CHRNA4UNDEFINEDRATUNDEFINED2-(6-Fluoro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]heptane0.027Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53294CHRNA4UNDEFINEDRATUNDEFINED2-Pyridin-3-yl-7-aza-bicyclo[2.2.1]heptane0.02Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53295CHRNA4UNDEFINEDRATUNDEFINEDrac-4-(5-(7-aza-bicyclo[2.2.1]heptan-2-yl)-2-fluoropyridin-3-yl)benzenamine hydrochloride0.095Ivy Carroll F et al., 2008Jan 15, 2025Jan 15, 2025
53296MORUNDEFINEDHUMANUNDEFINEDNaloxone(-)3.7Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53297MORUNDEFINEDHUMANUNDEFINED(S)-6-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)hexanoic acid0.5Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53298MORUNDEFINEDHUMANUNDEFINED(S)-5-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanoic acid0.41Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53299MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanedioic acid11Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53300MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)succinic acid7.3Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53301MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-4-phenylbutanoic acid4.7Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53302MORUNDEFINEDHUMANUNDEFINED(S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid11Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53303MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-2-yl)propanoic acid2Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53304MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-1-yl)propanoic acid2.7Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53305MORUNDEFINEDHUMANUNDEFINED(S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-3-biphenyl-4-yl-propionic acid1.9Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53306MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-phenylpropanoic acid1.7Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53307MORUNDEFINEDHUMANUNDEFINED(R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid2.9Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53308MORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid0.63Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53309MORUNDEFINEDHUMANUNDEFINED(S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid15Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53310MORUNDEFINEDHUMANUNDEFINED(S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionyl}-amino)-3-phenyl-propionic acid74Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53311MORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenethylpropanamido)-3-phenylpropanoic acid66Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53312MORUNDEFINEDHUMANUNDEFINED(S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid23Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53313MORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenylpropanamido)-3-phenylpropanoic acid32Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53314MORUNDEFINEDHUMANUNDEFINED(S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid22Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53315MORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-isobutylpropanamido)-3-phenylpropanoic acid28Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53316MORUNDEFINEDHUMANUNDEFINED(S)-2-(N-ethyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid19Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53317MORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-methylpropanamido)-3-phenylpropanoic acid66Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53318MORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-4-phenylbutanoic acid58Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53319MORUNDEFINEDHUMANUNDEFINED(S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-propionic acid80Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53320MORUNDEFINEDHUMANUNDEFINED(S)-3-cyclohexyl-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)propanoic acid20Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53321MORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid36Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53322MORUNDEFINEDHUMANUNDEFINED2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)acetic acid0.47Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53323KORUNDEFINEDHUMANUNDEFINEDNaloxone(-)9.2Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53324KORUNDEFINEDHUMANUNDEFINED(S)-6-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)hexanoic acid580Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53325KORUNDEFINEDHUMANUNDEFINED(S)-5-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanoic acid200Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53326KORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-4-phenylbutanoic acid510Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53327KORUNDEFINEDHUMANUNDEFINED(S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid720Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53328KORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-2-yl)propanoic acid240Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53329KORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-1-yl)propanoic acid83Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53330KORUNDEFINEDHUMANUNDEFINED(S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-3-biphenyl-4-yl-propionic acid160Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53331KORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-phenylpropanoic acid250Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53332KORUNDEFINEDHUMANUNDEFINED(R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid910Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53333KORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid67Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53334KORUNDEFINEDHUMANUNDEFINED(S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid460Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53335KORUNDEFINEDHUMANUNDEFINED(S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionyl}-amino)-3-phenyl-propionic acid230Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53336KORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenethylpropanamido)-3-phenylpropanoic acid1200Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53337KORUNDEFINEDHUMANUNDEFINED(S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid550Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53338KORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenylpropanamido)-3-phenylpropanoic acid1400Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53339KORUNDEFINEDHUMANUNDEFINED(S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid2200Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53340KORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-isobutylpropanamido)-3-phenylpropanoic acid2200Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53341KORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-4-phenylbutanoic acid690Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53342KORUNDEFINEDHUMANUNDEFINED(S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-propionic acid1100Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53343KORUNDEFINEDHUMANUNDEFINED2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)acetic acid100Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53344DORUNDEFINEDHUMANUNDEFINEDNaloxone(-)33Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53345DORUNDEFINEDHUMANUNDEFINED(S)-6-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)hexanoic acid1500Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53346DORUNDEFINEDHUMANUNDEFINED(S)-5-amino-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanoic acid510Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53347DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)pentanedioic acid360Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53348DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)succinic acid500Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53349DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-4-phenylbutanoic acid10Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53350DORUNDEFINEDHUMANUNDEFINED(S)-3-cyclohexyl-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid15Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53351DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-2-yl)propanoic acid3.2Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53352DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-(naphthalen-1-yl)propanoic acid31Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53353DORUNDEFINEDHUMANUNDEFINED(S)-2-{(S)-2-benzyl-3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-3-biphenyl-4-yl-propionic acid8.3Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53354DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)-3-phenylpropanoic acid15Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53355DORUNDEFINEDHUMANUNDEFINED(R)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid74Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53356DORUNDEFINEDHUMANUNDEFINED(S)-2-((S)-2-(((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)methyl)-3-phenylpropanamido)propanoic acid22Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53357DORUNDEFINEDHUMANUNDEFINED(S)-2-(N-(3-chlorobenzyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid24Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53358DORUNDEFINEDHUMANUNDEFINED(S)-2-(biphenyl-4-ylmethyl-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionyl}-amino)-3-phenyl-propionic acid52Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53359DORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenethylpropanamido)-3-phenylpropanoic acid63Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53360DORUNDEFINEDHUMANUNDEFINED(S)-2-(N-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid39Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53361DORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-phenylpropanamido)-3-phenylpropanoic acid67Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53362DORUNDEFINEDHUMANUNDEFINED(S)-2-(N-(cyclopropylmethyl)-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid100Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53363DORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-isobutylpropanamido)-3-phenylpropanoic acid29Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53364DORUNDEFINEDHUMANUNDEFINED(S)-2-(N-ethyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid510Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53365DORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)-N-methylpropanamido)-3-phenylpropanoic acid620Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53366DORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-4-phenylbutanoic acid360Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53367DORUNDEFINEDHUMANUNDEFINED(S)-3-biphenyl-4-yl-2-{3-[(3R,4R)-4-(3-hydroxy-phenyl)-3,4-dimethyl-piperidin-1-yl]-propionylamino}-propionic acid160Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53368DORUNDEFINEDHUMANUNDEFINED(S)-3-cyclohexyl-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)propanoic acid170Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53369DORUNDEFINEDHUMANUNDEFINED(S)-2-(3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)-3-phenylpropanoic acid990Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53370DORUNDEFINEDHUMANUNDEFINED2-((S)-2-benzyl-3-((3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethylpiperidin-1-yl)propanamido)acetic acid12Le Bourdonnec B et al., 2008Jan 15, 2025Jan 15, 2025
53371MORUNDEFINEDHUMANUNDEFINEDMorphine4Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53372MORUNDEFINEDHUMANUNDEFINEDsinoacutine>10000Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53373MORUNDEFINEDHUMANUNDEFINEDthebaine7400Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53374MORUNDEFINEDHUMANUNDEFINEDCodeine6300Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53375MORUNDEFINEDHUMANUNDEFINEDcodeinone459Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53376MORUNDEFINEDHUMANUNDEFINEDoripavine286Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53377MORUNDEFINEDHUMANUNDEFINEDmorphinone146Nikolaev VO et al., 2007Jan 15, 2025Jan 15, 2025
53378CB1UNDEFINEDUNDEFINEDUNDEFINEDRimonabant1.98Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53379CB1UNDEFINEDUNDEFINEDUNDEFINED1-(2,4-dichlorophenyl)-4-(hydroxymethyl)-N-(piperidin-1-yl)-5-(4-(pyridin-3-yl)phenyl)-1H-pyrazole-3-carboxamide5.8Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53380CB1UNDEFINEDUNDEFINEDUNDEFINED5,5-Bis-(4-bromo-phenyl)-3-(2-morpholin-4-yl-ethyl)-imidazolidine-2,4-dione70.3Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53381CB1UNDEFINEDUNDEFINEDUNDEFINED1-(bis(4-chlorophenyl)methyl)-3-((3,5-difluorophenyl)(methylsulfonyl)methylene)azetidine100Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53382CB1UNDEFINEDUNDEFINEDUNDEFINED4-(6-methoxy-2-(4-methoxyphenyl)benzofuran-3-carbonyl)benzonitrile141Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53383CB1UNDEFINEDUNDEFINEDUNDEFINEDibipinabant7.8Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53384CB1UNDEFINEDUNDEFINEDUNDEFINED8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide0.00035Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53385CB2UNDEFINEDUNDEFINEDUNDEFINEDRimonabant1000Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53386CB2UNDEFINEDUNDEFINEDUNDEFINED1-(2,4-dichlorophenyl)-4-(hydroxymethyl)-N-(piperidin-1-yl)-5-(4-(pyridin-3-yl)phenyl)-1H-pyrazole-3-carboxamide2312Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53387CB2UNDEFINEDUNDEFINEDUNDEFINED4-(6-methoxy-2-(4-methoxyphenyl)benzofuran-3-carbonyl)benzonitrile>10000Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53388CB2UNDEFINEDUNDEFINEDUNDEFINEDibipinabant7943Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53389CB2UNDEFINEDUNDEFINEDUNDEFINED8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide21Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53390CB1UNDEFINEDHUMANUNDEFINED(3R,4S)-3-(benzofuran-2-ylmethyl)-4-(4-methoxyphenyl)-1-phenylazetidin-2-one839Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53391CB1UNDEFINEDHUMANUNDEFINEDS-(R)-1-((2S,3R)-1-(4-fluorophenyl)-2-(4-hydroxyphenyl)-4-oxoazetidin-3-yl)-3-phenylpropyl ethanethioate52.8Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53392CB1UNDEFINEDHUMANUNDEFINED(3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-one301.4Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53393CB1UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)ethyl)azetidin-2-one451.5Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53394CB1UNDEFINEDHUMANUNDEFINED(3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin-3-yl)propyl)azetidin-2-one243.8Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53395CB1UNDEFINEDHUMANUNDEFINEDRimonabant2.4Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53396CB2UNDEFINEDHUMANUNDEFINED(3R,4S)-3-(benzofuran-2-ylmethyl)-4-(4-methoxyphenyl)-1-phenylazetidin-2-one194.2Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53397CB2UNDEFINEDHUMANUNDEFINEDS-(R)-1-((2S,3R)-1-(4-fluorophenyl)-2-(4-hydroxyphenyl)-4-oxoazetidin-3-yl)-3-phenylpropyl ethanethioate282Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53398CB2UNDEFINEDHUMANUNDEFINED(3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3-hydroxypropyl)-4-(4-hydroxyphenyl)azetidin-2-one1818.2Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53399CB2UNDEFINEDHUMANUNDEFINED4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)ethyl)azetidin-2-one1242.8Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53400CB2UNDEFINEDHUMANUNDEFINED(3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin-3-yl)propyl)azetidin-2-one1090.5Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53401CB2UNDEFINEDHUMANUNDEFINEDRimonabant560Wang H et al., 2008Jan 15, 2025Jan 15, 2025
53402SLC6A4UNDEFINEDHUMANUNDEFINEDDuloxetine5Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53403SLC6A4UNDEFINEDHUMANUNDEFINEDReboxetine1400Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53404SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(p-tolyl)methyl)morpholine88Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53405SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(m-tolyl)methyl)morpholine69Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53406SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(o-tolyl)methyl)morpholine70Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53407SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(4-fluorophenyl)methyl)morpholine62Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53408SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(3-fluorophenyl)methyl)morpholine58Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53409SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(2-fluorophenyl)methyl)morpholine70Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53410SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-chloro-4-methoxyphenoxy)(phenyl)methyl)morpholine96Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53411SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-methoxy-4-(trifluoromethyl)phenoxy)(phenyl)methyl)morpholine41Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53412SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-bromo-2-methoxyphenoxy)(phenyl)methyl)morpholine30Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53413SLC6A4UNDEFINEDHUMANUNDEFINED3-methoxy-4-((S)-((S)-morpholin-2-yl)(phenyl)methoxy)benzonitrile110Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53414SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-dichlorophenoxy)(phenyl)methyl)morpholine100Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53415SLC6A4UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine20Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53416SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine1800Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53417SLC6A4UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine12Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53418SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine3390Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53419SLC6A4UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine34Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53420SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine185Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53421SLC6A4UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine20Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53422SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine260Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53423SLC6A4UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine22Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53424SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine740Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53425SLC6A4UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine11Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53426SLC6A4UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine110Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53427SLC6A4UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine85Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53428SLC6A4UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine28Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53429SLC6A4UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine220Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53430SLC6A4UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine60Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53431SLC6A4UNDEFINEDHUMANUNDEFINEDrac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine340Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53432SLC6A4UNDEFINEDHUMANUNDEFINEDrac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine240Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53433SLC6A2UNDEFINEDHUMANUNDEFINEDDuloxetine45Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53434SLC6A2UNDEFINEDHUMANUNDEFINEDReboxetine5Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53435SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(p-tolyl)methyl)morpholine180Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53436SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(m-tolyl)methyl)morpholine16Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53437SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(o-tolyl)methyl)morpholine84Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53438SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(4-fluorophenyl)methyl)morpholine29Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53439SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(3-fluorophenyl)methyl)morpholine9Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53440SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(2-fluorophenyl)methyl)morpholine22Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53441SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-chloro-4-methoxyphenoxy)(phenyl)methyl)morpholine28Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53442SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-methoxy-4-(trifluoromethyl)phenoxy)(phenyl)methyl)morpholine160Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53443SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-bromo-2-methoxyphenoxy)(phenyl)methyl)morpholine12Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53444SLC6A2UNDEFINEDHUMANUNDEFINED3-methoxy-4-((S)-((S)-morpholin-2-yl)(phenyl)methoxy)benzonitrile210Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53445SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-dichlorophenoxy)(phenyl)methyl)morpholine17Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53446SLC6A2UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine350Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53447SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine12Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53448SLC6A2UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine130Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53449SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine10Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53450SLC6A2UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine860Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53451SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine18Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53452SLC6A2UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine830Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53453SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine12Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53454SLC6A2UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine610Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53455SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine6Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53456SLC6A2UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine420Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53457SLC6A2UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine8Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53458SLC6A2UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine320Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53459SLC6A2UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine36Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53460SLC6A2UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine390Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53461SLC6A2UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine15Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53462SLC6A2UNDEFINEDHUMANUNDEFINEDrac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine1490Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53463SLC6A2UNDEFINEDHUMANUNDEFINEDrac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine275Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53464SLC6A3UNDEFINEDHUMANUNDEFINEDDuloxetine435Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53465SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(p-tolyl)methyl)morpholine1650Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53466SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(3-fluorophenyl)methyl)morpholine>10000Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53467SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-chloro-4-methoxyphenoxy)(phenyl)methyl)morpholine1090Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53468SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-dichlorophenoxy)(phenyl)methyl)morpholine420Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53469SLC6A3UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine5750Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53470SLC6A3UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine380Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53471SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine2600Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53472SLC6A3UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine950Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53473SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine1250Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53474SLC6A3UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine760Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53475SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine1170Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53476SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine3080Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53477SLC6A3UNDEFINEDHUMANUNDEFINED(R)-2-((R)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine1790Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53478SLC6A3UNDEFINEDHUMANUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine1570Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53479SLC6A3UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine2200Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53480SLC6A3UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine5050Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53481SLC6A3UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine1670Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53482SLC6A3UNDEFINEDHUMANUNDEFINEDrac-syn-2-((4-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine1540Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53483SLC6A3UNDEFINEDHUMANUNDEFINEDReboxetine>10000Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53484SLC6A3UNDEFINEDHUMANUNDEFINEDrac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine>10000Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53485SLC6A3UNDEFINEDHUMANUNDEFINEDrac-syn-2-((3-chloro-2-ethoxyphenoxy)(phenyl)methyl)morpholine>10000Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53486H1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-((R)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine26Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53487H1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-((R)-(4-fluoro-2-methoxyphenoxy)(phenyl)methyl)morpholine10Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53488H1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-((R)-(2,3-dihydrobenzofuran-7-yloxy)(phenyl)methyl)morpholine10Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53489H1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-((R)-(2,3-difluorophenoxy)(phenyl)methyl)morpholine10Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53490H1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-((R)-(4-fluoro-2-methylphenoxy)(phenyl)methyl)morpholine10Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53491H1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-((R)-(2-chloro-4-fluorophenoxy)(phenyl)methyl)morpholine10Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53492SLC6A4UNDEFINEDRATUNDEFINED(S)-2-((S)-(4-chloro-2-methoxyphenoxy)(phenyl)methyl)morpholine59Fish PV et al., 2008Jan 15, 2025Jan 15, 2025
53493MORUNDEFINEDUNDEFINEDUNDEFINED6-desoxycodeine305Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53494MORUNDEFINEDUNDEFINEDUNDEFINED6-desoxymorphine2.1Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53495MORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3-desoxyheterocodeine524Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53496MORUNDEFINEDUNDEFINEDUNDEFINEDcodeine-6-methyl ether1910Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53497MORUNDEFINEDUNDEFINEDUNDEFINEDheterocodeine1.1Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53498MORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3-desoxymorphine122Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53499MORUNDEFINEDUNDEFINEDUNDEFINEDCodeine727Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53500MORUNDEFINEDUNDEFINEDUNDEFINEDMorphine1.7Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53501MORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3,6-didesoxymorphine22.9Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53502DORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3-desoxymorphine5250Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53503DORUNDEFINEDUNDEFINEDUNDEFINEDCodeine>10000Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53504DORUNDEFINEDUNDEFINEDUNDEFINEDMorphine104.57Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53505DORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3,6-didesoxymorphine241Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53506DORUNDEFINEDUNDEFINEDUNDEFINED6-desoxycodeine4520Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53507DORUNDEFINEDUNDEFINEDUNDEFINED6-desoxymorphine11.8Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53508DORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3-desoxyheterocodeine8830Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53509DORUNDEFINEDUNDEFINEDUNDEFINEDcodeine-6-methyl ether4410Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53510DORUNDEFINEDUNDEFINEDUNDEFINEDheterocodeine65.8Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53511KORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3,6-didesoxymorphine589Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53512KORUNDEFINEDUNDEFINEDUNDEFINED6-desoxycodeine3090Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53513KORUNDEFINEDUNDEFINEDUNDEFINED6-desoxymorphine45.5Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53514KORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3-desoxyheterocodeine>10000Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53515KORUNDEFINEDUNDEFINEDUNDEFINEDcodeine-6-methyl ether5430Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53516KORUNDEFINEDUNDEFINEDUNDEFINEDheterocodeine22.8Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53517KORUNDEFINEDUNDEFINEDUNDEFINED7,8-dihydro-3-desoxymorphine4910Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53518KORUNDEFINEDUNDEFINEDUNDEFINEDCodeine>10000Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53519KORUNDEFINEDUNDEFINEDUNDEFINEDMorphine65.5Cunningham CW et al., 2008Jan 15, 2025Jan 15, 2025
53520SLC6A2UNDEFINEDHUMANUNDEFINEDVenlafaxine385Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53521SLC6A2UNDEFINEDHUMANUNDEFINED1-{2-Piperazin-1-yl-1-[3-(trifluoromethyl)phenyl]ethyl}cyclohexanol Dihydrochloride58Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53522SLC6A2UNDEFINEDHUMANUNDEFINED1-{2-(3-Methylpiperazin-1-yl)-1-[3-(trifluoromethyl)phenyl]ethyl}cyclohexanol Dihydrocholoride61Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53523SLC6A2UNDEFINEDHUMANUNDEFINED(+)-1-{(1S)-2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride117Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53524SLC6A2UNDEFINEDHUMANUNDEFINED(-)-1-{(1R)-2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride544Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53525SLC6A2UNDEFINEDHUMANUNDEFINED1-{2-Piperazin-1-yl-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrochloride140Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53526SLC6A2UNDEFINEDHUMANUNDEFINED(-)-1-{(1S)-2-(4-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride50Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53527SLC6A2UNDEFINEDHUMANUNDEFINED(+)-1-{(1R)-2-(4-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride785Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53528SLC6A2UNDEFINEDHUMANUNDEFINED1-{2-(3-Methylpiperazin-1-yl)-1-[3-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride91Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53529SLC6A2UNDEFINEDHUMANUNDEFINED1-{2-(4-Methylpiperazin-1-yl)-1-[4-(trifluoromethoxy)phenyl]ethyl}cyclohexanol Dihydrocholoride417Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53530SLC6A2UNDEFINEDHUMANUNDEFINED(+)-1-[(1S)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride17Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53531SLC6A2UNDEFINEDHUMANUNDEFINED(-)-1-[(1R)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride214Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53532SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride18Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53533SLC6A2UNDEFINEDHUMANUNDEFINED(-)-1-[(1S)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride14Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53534SLC6A2UNDEFINEDHUMANUNDEFINED(+)-1-[(1R)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride187Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53535SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride46Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53536SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(4-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride717Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53537SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(4-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride1220Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53538SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Fluorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride368Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53539SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride364Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53540SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(4-Fluorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride1034Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53541SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(4-Fluorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride1376Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53542SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Methoxyphenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride745Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53543SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Methoxyphenyl)-2-(4-methyl-1-piperazinyl)ethyl]cyclohexanol Dihydrochloride514Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53544SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(4-Methoxyphenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride519Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53545SLC6A2UNDEFINEDHUMANUNDEFINED(+)-1-[(1S)-1-(3-Chlorophenyl)-2-(dimethylamino)ethyl]cyclohexanol339Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53546SLC6A2UNDEFINEDHUMANUNDEFINED(-)-1-[(1R)-1-(3-Chlorophenyl)-2-(dimethylamino)ethyl]cyclohexanol41Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53547SLC6A2UNDEFINEDHUMANUNDEFINED1-[2-Dimethylamino-1-(3-trifluoromethyl-phenyl)-ethyl]-cyclohexanol (HCl)21Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53548SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(2-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol(HCl)125Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53549SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(3-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol (HCl)149Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53550SLC6A2UNDEFINEDHUMANUNDEFINED1-[1-(4-Chloro-phenyl)-2-dimethylamino-ethyl]-cyclohexanol (HCl)249Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53551SLC6A2UNDEFINEDHUMANUNDEFINED1-[2-Dimethylamino-1-(3-methoxy-phenyl)-ethyl]-cyclohexanol (HCl)316Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53552SLC6A2UNDEFINEDHUMANUNDEFINEDDESIPRAMINE2.1Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53553SLC6A3UNDEFINEDHUMANUNDEFINED1-[1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride53Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53554SLC6A3UNDEFINEDHUMANUNDEFINED(+)-1-[(1S)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride135Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53555SLC6A3UNDEFINEDHUMANUNDEFINED(-)-1-[(1R)-1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride340Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53556SLC6A3UNDEFINEDHUMANUNDEFINED1-[1-(3-Chlorophenyl)-2-piperazin-1-ylethyl]cyclohexanol Dihydrochloride45Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53557SLC6A3UNDEFINEDHUMANUNDEFINED(-)-1-[(1S)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride73Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53558SLC6A3UNDEFINEDHUMANUNDEFINED(+)-1-[(1R)-1-(3-Chlorophenyl)-2-(4-methylpiperazin-1-yl)ethyl]cyclohexanol Dihydrocholoride235Mahaney PE et al., 2008Jan 15, 2025Jan 15, 2025
53559SLC6A4UNDEFINEDRATUNDEFINEDFLUOXETINE2.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53560SLC6A4UNDEFINEDRATUNDEFINED5-Fluoro-3-[(1,4-cis)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole640Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53561SLC6A4UNDEFINEDRATUNDEFINED3-[(1,4-trans)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile13.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53562SLC6A4UNDEFINEDRATUNDEFINED3-[(1,4-cis)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile1.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53563SLC6A4UNDEFINEDRATUNDEFINED3-[(1,4-trans)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile20Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53564SLC6A4UNDEFINEDRATUNDEFINED3-[(1,4-cis)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile1.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53565SLC6A4UNDEFINEDRATUNDEFINED8-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline39.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53566SLC6A4UNDEFINEDRATUNDEFINED8-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline4.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53567SLC6A4UNDEFINEDRATUNDEFINED3-[(1,4-trans)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile4.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53568SLC6A4UNDEFINEDRATUNDEFINED3-[(1,4-cis)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile3.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53569SLC6A4UNDEFINEDRATUNDEFINED5-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline73Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53570SLC6A4UNDEFINEDRATUNDEFINED5-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline13.8Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53571SLC6A4UNDEFINEDRATUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole75Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53572SLC6A4UNDEFINEDRATUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole105Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53573SLC6A4UNDEFINEDRATUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]piperazin-1-yl}-2-methyl-1H-benzimidazole115Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53574SLC6A4UNDEFINEDRATUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-methyl-1H-benzimidazole61Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53575SLC6A4UNDEFINEDRATUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole75Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53576SLC6A4UNDEFINEDRATUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole13Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53577SLC6A4UNDEFINEDRATUNDEFINED3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-isopropyl-1H-indole-5-carbonitrile38.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53578SLC6A4UNDEFINEDRATUNDEFINED3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-pipera-zin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile62.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53579SLC6A4UNDEFINEDRATUNDEFINED3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile26.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53580SLC6A4UNDEFINEDRATUNDEFINED1-Ethyl-3-{(1,4-trans)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile58.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53581SLC6A4UNDEFINEDRATUNDEFINED1-Ethyl-3-{(1,4-cis)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile13.4Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53582SLC6A4UNDEFINEDRATUNDEFINED3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile102Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53583SLC6A4UNDEFINEDRATUNDEFINED3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile3.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53584SLC6A4UNDEFINEDRATUNDEFINED3-{4-[(1,4-trans)-4-(1H-indol-4-yl)-pipera-zinyl-1-yl]cyclohexyl}-1H-indole-5-carbonitrile8.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53585SLC6A4UNDEFINEDRATUNDEFINED3-{4-[(1,4-cis)-4-(1H-Indol-4-yl)-pipera-zinyl-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile1.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53586SLC6A4UNDEFINEDRATUNDEFINED6-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]cyclohexyl]-1H-indole12.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53587SLC6A4UNDEFINEDRATUNDEFINED5-Fluoro-3-{trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole67.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53588SLC6A4UNDEFINEDRATUNDEFINED5-Fluoro-3-{cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole11.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53589SLC6A4UNDEFINEDRATUNDEFINED3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-1H-indole155Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53590SLC6A4UNDEFINEDRATUNDEFINED3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclo-hexyl]-1H-indole38Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53591SLC6A4UNDEFINEDRATUNDEFINED5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole48.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53592SLC6A4UNDEFINEDRATUNDEFINED5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole5.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535935-HT1AUNDEFINEDHUMANUNDEFINEDCyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide0.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535945-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-trans)-4-[4-(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine7.8Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535955-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-cis)-4-[(1H-Indole-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-pyrrolo[2,3-b]pyridine15.8Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535965-HT1AUNDEFINEDHUMANUNDEFINED5-Fluoro-3-[(1,4-trans)-4-(4-naphthalen-1-yl-piperazin-1-yl)-cyclohexyl]-1H-indole42.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535975-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-trans)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile9.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535985-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-cis)-4-(4-Quinoxalin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile156.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
535995-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-trans)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile2.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536005-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-cis)-4-(4-Quinolin-8-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile43.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536015-HT1AUNDEFINEDHUMANUNDEFINED8-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline6.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536025-HT1AUNDEFINEDHUMANUNDEFINED8-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline69.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536035-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-trans)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile6.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536045-HT1AUNDEFINEDHUMANUNDEFINED3-[(1,4-cis)-4-(4-Quinolin-5-yl-piperazin-1-yl)-cyclohexyl]-1H-indole-5-carbonitrile58.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536055-HT1AUNDEFINEDHUMANUNDEFINED5-{4-[(1,4-trans)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline8.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536065-HT1AUNDEFINEDHUMANUNDEFINED5-{4-[(1,4-cis)-4-(5-Fluoro-1H-indol-3-yl)-cyclohexyl]-piperazin-1-yl}-quinoline97.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536075-HT1AUNDEFINEDHUMANUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole3.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536085-HT1AUNDEFINEDHUMANUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-(trifluoromethyl)-1H-benzimidazole16.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536095-HT1AUNDEFINEDHUMANUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]piperazin-1-yl}-2-methyl-1H-benzimidazole3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536105-HT1AUNDEFINEDHUMANUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-2-methyl-1H-benzimidazole10.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536115-HT1AUNDEFINEDHUMANUNDEFINED4-{trans-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole1.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536125-HT1AUNDEFINEDHUMANUNDEFINED4-{cis-4-[4-(1H-Indol-3-yl)cyclohexyl]-piperazin-1-yl}-1H-benzimidazole7.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536135-HT1AUNDEFINEDHUMANUNDEFINED3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-2-methyl-1H-indole13Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536145-HT1AUNDEFINEDHUMANUNDEFINED3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclohexyl]-2-methyl-1H-indole87.1Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536155-HT1AUNDEFINEDHUMANUNDEFINED5-Chloro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole58.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536165-HT1AUNDEFINEDHUMANUNDEFINED5-Chloro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole325.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536175-HT1AUNDEFINEDHUMANUNDEFINED5-Methoxy-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole2.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536185-HT1AUNDEFINEDHUMANUNDEFINED5-Methoxy-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole60.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536195-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-isopropyl-1H-indole-5-carbonitrile694.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536205-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-propyl-1H-indole-5-carbonitrile819.8Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536215-HT1AUNDEFINEDHUMANUNDEFINED1-Ethyl-3-{(1,4-trans)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile827.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536225-HT1AUNDEFINEDHUMANUNDEFINED1-Ethyl-3-{(1,4-cis)-4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile563.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536235-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-trans)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile53.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536245-HT1AUNDEFINEDHUMANUNDEFINED3-{(1,4-cis)-4-[4-(1H-Indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1-methyl-1H-indole-5-carbonitrile232.9Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536255-HT1AUNDEFINEDHUMANUNDEFINED3-{4-[(1,4-trans)-4-(1H-indol-4-yl)-pipera-zinyl-1-yl]cyclohexyl}-1H-indole-5-carbonitrile3.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536265-HT1AUNDEFINEDHUMANUNDEFINED3-{4-[(1,4-cis)-4-(1H-Indol-4-yl)-pipera-zinyl-1-yl]-cyclohexyl}-1H-indole-5-carbonitrile69.6Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536275-HT1AUNDEFINEDHUMANUNDEFINED4-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole22.2Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536285-HT1AUNDEFINEDHUMANUNDEFINED4-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl]-1H-indole117.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536295-HT1AUNDEFINEDHUMANUNDEFINED6-Fluoro-3-[trans-4-[4-(1H-indol-4-yl)-1-pipera-zinyl]cyclohexyl]-1H-indole5.4Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536305-HT1AUNDEFINEDHUMANUNDEFINED5-Fluoro-3-{trans-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole90Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536315-HT1AUNDEFINEDHUMANUNDEFINED5-Fluoro-3-{cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]-cyclohexyl}-1-methyl-1H-indole124Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536325-HT1AUNDEFINEDHUMANUNDEFINED3-[trans-4-[4-(1H-Indol-4-yl)-1-pipera-zinyl]-cyclohexyl]-1H-indole5.3Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536335-HT1AUNDEFINEDHUMANUNDEFINED3-[cis-4-[4-(1H-Indol-4-yl)-1-piperazinyl]-cyclo-hexyl]-1H-indole32Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536345-HT1AUNDEFINEDHUMANUNDEFINED5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole4.62Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536355-HT1AUNDEFINEDHUMANUNDEFINED5-Fluoro-3-{4-[4-(1H-indol-4-yl)-piperazin-1-yl]-cyclohexyl}-1H-indole36.7Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
536365-HT1AUNDEFINEDHUMANUNDEFINED6-Fluoro-3-[cis-4-[4-(1H-indol-4-yl)-1-piperazinyl]cyclohexyl]-1H-indole33.5Zhou D et al., 2008Jan 15, 2025Jan 15, 2025
53637CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-chloro-2,2-diphenylacetamide280Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53638CB1UNDEFINEDHUMANUNDEFINEDSR 1445285600Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53639CB1UNDEFINEDHUMANUNDEFINEDRimonabant8Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53640CB1UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide2.3Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53641CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-(4-bromophenyl) acetamide800Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53642CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-(4-chlorophenyl)acetamide1600Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53643CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-phenylacetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53644CB1UNDEFINEDHUMANUNDEFINEDN-(3-Phenyl)propyl-2-(4-bromophenylacetamide)1900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53645CB1UNDEFINEDHUMANUNDEFINEDN-(3-Phenyl)propyl-2-(4-chlorophenyl)-2-phenylacetamide2200Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53646CB1UNDEFINEDHUMANUNDEFINEDN-(3-Phenyl)propyl-2,2-diphenylacetamide3400Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53647CB1UNDEFINEDHUMANUNDEFINED2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53648CB1UNDEFINEDHUMANUNDEFINED2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53649CB1UNDEFINEDHUMANUNDEFINED2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53650CB1UNDEFINEDHUMANUNDEFINED2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53651CB1UNDEFINEDHUMANUNDEFINED2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53652CB1UNDEFINEDHUMANUNDEFINED2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide220Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53653CB1UNDEFINEDHUMANUNDEFINED2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53654CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-hydroxy-2,2-diphenylacetamide2200Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53655CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-methyl-2,2-diphenylacetamide560Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53656CB1UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2,2-diphenylacetamide58Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53657CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-chloro-2,2-diphenylacetamide1400Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53658CB2UNDEFINEDHUMANUNDEFINEDSR 1445285.4Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53659CB2UNDEFINEDHUMANUNDEFINEDRimonabant790Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53660CB2UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide110Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53661CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-(4-bromophenyl) acetamide1300Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53662CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-(4-chlorophenyl)acetamide2400Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53663CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-phenylacetamide7900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53664CB2UNDEFINEDHUMANUNDEFINEDN-(3-Phenyl)propyl-2-(4-bromophenylacetamide)1800Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53665CB2UNDEFINEDHUMANUNDEFINEDN-(3-Phenyl)propyl-2-(4-chlorophenyl)-2-phenylacetamide2400Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53666CB2UNDEFINEDHUMANUNDEFINEDN-(3-Phenyl)propyl-2,2-diphenylacetamide7900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53667CB2UNDEFINEDHUMANUNDEFINED2-(4-Aminophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide1200Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53668CB2UNDEFINEDHUMANUNDEFINED2-(4-Hydroxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide1100Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53669CB2UNDEFINEDHUMANUNDEFINED2-(4-Nitrophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide790Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53670CB2UNDEFINEDHUMANUNDEFINED2-(4-Methylphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide650Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53671CB2UNDEFINEDHUMANUNDEFINED2-(4-Methoxyphenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide790Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53672CB2UNDEFINEDHUMANUNDEFINED2-(4-Bromophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide7900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53673CB2UNDEFINEDHUMANUNDEFINED2-(4-Chlorophenyl)-2-phenyl-N-(3,3-diphenylpropyl)-acetamide7900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53674CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-hydroxy-2,2-diphenylacetamide2300Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53675CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2-methyl-2,2-diphenylacetamide290Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
53676CB2UNDEFINEDHUMANUNDEFINEDN-(3,3-Diphenyl)propyl-2,2-diphenylacetamide7900Urbani P et al., 2008Jan 15, 2025Jan 15, 2025
536775-HT6UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one295.9Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536785-HT6UNDEFINEDHUMANUNDEFINEDHALOPERIDOL6000Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536795-HT6UNDEFINEDHUMANUNDEFINEDQuetiapine1400Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536805-HT6UNDEFINEDHUMANUNDEFINEDOLANZAPINE10Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536815-HT6UNDEFINEDHUMANUNDEFINEDZiprasidone76Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536825-HT6UNDEFINEDHUMANUNDEFINEDRISPERIDONE2000Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536835-HT6UNDEFINEDHUMANUNDEFINEDCLOZAPINE11Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53684M1UNDEFINEDHUMANUNDEFINEDCLOZAPINE1.8Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53685M1UNDEFINEDHUMANUNDEFINEDHALOPERIDOL1600Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53686M1UNDEFINEDHUMANUNDEFINEDQuetiapine100Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53687M1UNDEFINEDHUMANUNDEFINEDOLANZAPINE4.7Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53688M1UNDEFINEDHUMANUNDEFINEDZiprasidone5100Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53689M1UNDEFINEDHUMANUNDEFINEDRISPERIDONE2800Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53690M1UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one871.6Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53691D1UNDEFINEDHUMANUNDEFINEDHALOPERIDOL120Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53692D1UNDEFINEDHUMANUNDEFINEDQuetiapine1300Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53693D1UNDEFINEDHUMANUNDEFINEDOLANZAPINE52Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53694D1UNDEFINEDHUMANUNDEFINEDZiprasidone130Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53695D1UNDEFINEDHUMANUNDEFINEDRISPERIDONE580Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53696D1UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one162.7Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53697D1UNDEFINEDHUMANUNDEFINEDCLOZAPINE290Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
536985-HT2BUNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one495.2Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53699D2UNDEFINEDHUMANUNDEFINEDCLOZAPINE130Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53700D2UNDEFINEDHUMANUNDEFINEDHALOPERIDOL1.4Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53701D2UNDEFINEDHUMANUNDEFINEDQuetiapine180Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53702D2UNDEFINEDHUMANUNDEFINEDOLANZAPINE20Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53703D2UNDEFINEDHUMANUNDEFINEDZiprasidone3.1Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53704D2UNDEFINEDHUMANUNDEFINEDRISPERIDONE2.2Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53705D2UNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one178.4Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53706D2UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one43.3Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53707D2UNDEFINEDHUMANUNDEFINED1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one98Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53708D2UNDEFINEDHUMANUNDEFINED4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one170Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53709D2UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(8-phenyl-3,8-diaza-bicyclo[3.2.1]octan-3-yl)butan-1-one155Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53710D2UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one489.4Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53711D2UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one51.1Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53712D2UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one124.4Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53713D2UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one2.3Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53714D2UNDEFINEDHUMANUNDEFINED4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one1.6Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53715D2UNDEFINEDHUMANUNDEFINED4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one253.5Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53716D3UNDEFINEDHUMANUNDEFINEDHALOPERIDOL2.5Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53717D3UNDEFINEDHUMANUNDEFINEDQuetiapine320Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53718D3UNDEFINEDHUMANUNDEFINEDOLANZAPINE45Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53719D3UNDEFINEDHUMANUNDEFINEDZiprasidone7.2Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53720D3UNDEFINEDHUMANUNDEFINEDRISPERIDONE9.6Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53721D3UNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one548.1Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53722D3UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one158.8Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53723D3UNDEFINEDHUMANUNDEFINED1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one244.1Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53724D3UNDEFINEDHUMANUNDEFINED4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one220Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53725D3UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(8-phenyl-3,8-diaza-bicyclo[3.2.1]octan-3-yl)butan-1-one600Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53726D3UNDEFINEDHUMANUNDEFINEDCLOZAPINE240Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53727D4UNDEFINEDHUMANUNDEFINEDCLOZAPINE54Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53728D4UNDEFINEDHUMANUNDEFINEDHALOPERIDOL3.3Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53729D4UNDEFINEDHUMANUNDEFINEDQuetiapine2200Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53730D4UNDEFINEDHUMANUNDEFINEDOLANZAPINE50Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53731D4UNDEFINEDHUMANUNDEFINEDZiprasidone32Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53732D4UNDEFINEDHUMANUNDEFINEDRISPERIDONE8.5Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53733D4UNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one41.8Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53734D4UNDEFINEDHUMANUNDEFINED4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one6.6Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53735D4UNDEFINEDHUMANUNDEFINED1-(4-Fluoro-phenyl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one6.53Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53736D4UNDEFINEDHUMANUNDEFINED4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one520Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53737D4UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(8-phenyl-3,8-diaza-bicyclo[3.2.1]octan-3-yl)butan-1-one2100Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53738D4UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one245.5Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53739D4UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one3.6Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53740D4UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one176.8Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53741D4UNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one19.2Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53742D4UNDEFINEDHUMANUNDEFINED4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one5.3Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
53743D4UNDEFINEDHUMANUNDEFINED4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one17.5Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
537445-HT2CUNDEFINEDHUMANUNDEFINED1-(4-fluorophenyl)-4-(3-hydroxy-3-phenyl-8-aza-bicyclo[3.2.1]octan-8-yl)butan-1-one>10000Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
537455-HT2CUNDEFINEDHUMANUNDEFINED4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one872.1Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
537465-HT2CUNDEFINEDHUMANUNDEFINED4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one3552Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
537475-HT2CUNDEFINEDHUMANUNDEFINEDCLOZAPINE17Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025
537485-HT2CUNDEFINEDHUMANUNDEFINEDHALOPERIDOL4700Ablordeppey SY et al., 2008Jan 15, 2025Jan 15, 2025