The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 53,001-54,000 of 98,685 items.

Kᵢ Database

Reset Grid
Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
557495-HT1DUNDEFINEDHUMANUNDEFINEDN1,N14-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tetradecanediamide1.7Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557505-HT1DUNDEFINEDHUMANUNDEFINEDN1,N13-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tridecanediamide1.4Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557515-HT1DUNDEFINEDHUMANUNDEFINEDN1,N11-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)undecanediamide0.9Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557525-HT1DUNDEFINEDHUMANUNDEFINEDN1,N10-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)decanediamide0.95Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557535-HT1DUNDEFINEDHUMANUNDEFINEDN1,N8-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)octanediamide0.9Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557545-HT1DUNDEFINEDHUMANUNDEFINEDN1,N5-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)glutaramide0.95Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557555-HT1DUNDEFINEDHUMANUNDEFINED2-(5-{2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethoxy}-1H-indol-3-yl)-ethylamine0.4Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557565-HT1DUNDEFINEDHUMANUNDEFINEDC-[3-(2-Dimethylamino-ethyl)-1H-indol-5-yl]-N-[4-({[3-(2-dimethylamino-ethyl)-1H-indol-5-ylmethanesulfonyl]-methyl-amino}-methyl)-benzyl]-N-methyl-methanesulfonamide0.89Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557575-HT1DUNDEFINEDHUMANUNDEFINED2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine0.11Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557585-HT1AUNDEFINEDUNDEFINEDUNDEFINED2-(5-{2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethoxy}-1H-indol-3-yl)-ethylamine0.96Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557595-HT1AUNDEFINEDUNDEFINEDUNDEFINEDC-[3-(2-Dimethylamino-ethyl)-1H-indol-5-yl]-N-[4-({[3-(2-dimethylamino-ethyl)-1H-indol-5-ylmethanesulfonyl]-methyl-amino}-methyl)-benzyl]-N-methyl-methanesulfonamide17.7Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557605-HT1AUNDEFINEDUNDEFINEDUNDEFINED2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine1.6Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557615-HT1FUNDEFINEDHUMANUNDEFINED4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-benzamide1.6Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
55762CB1UNDEFINEDHUMANUNDEFINED1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1Hpyrazole-3-carboxamide34.2Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55763CB1UNDEFINEDHUMANUNDEFINEDRimonabant6.18Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55764CB1UNDEFINEDHUMANUNDEFINED9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4,5,6,7-tetrahydro-1H-benzo[7,8]cycloocta[1,2-c]pyrazole-3-carboxamide40.9Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55765CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide194Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55766CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide251Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55767CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide16.1Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55768CB1UNDEFINEDHUMANUNDEFINED5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide261Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55769CB1UNDEFINEDHUMANUNDEFINED8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide18.4Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55770CB1UNDEFINEDHUMANUNDEFINED1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1Hpyrazole-3-carboxamide17.9Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55771CB1UNDEFINEDHUMANUNDEFINEDRimonabant1.18Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55772CB1UNDEFINEDHUMANUNDEFINED9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4,5,6,7-tetrahydro-1H-benzo[7,8]cycloocta[1,2-c]pyrazole-3-carboxamide14.7Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55773CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide116Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55774CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide152Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55775CB1UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide5.83Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55776CB1UNDEFINEDHUMANUNDEFINED5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide148Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55777CB1UNDEFINEDHUMANUNDEFINED8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide5.55Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55778CB2UNDEFINEDHUMANUNDEFINED1,5-bis(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1Hpyrazole-3-carboxamide1044Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55779CB2UNDEFINEDHUMANUNDEFINEDRimonabant313Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55780CB2UNDEFINEDHUMANUNDEFINED9-Chloro-1-(2,4-dichlorophenyl)-N-piperidin-1-yl-4,5,6,7-tetrahydro-1H-benzo[7,8]cycloocta[1,2-c]pyrazole-3-carboxamide492Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55781CB2UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2,6-dimethylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide758Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55782CB2UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2-methylphenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide1781Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55783CB2UNDEFINEDHUMANUNDEFINED5-(4-Chloro-2-methylphenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-yl-1H-pyrazole-3-carboxamide1124Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55784CB2UNDEFINEDHUMANUNDEFINED5-(2,4-Dichlorophenyl)-4-methyl-N-piperidin-1-yl-1-(2,4,6-trichlorophenyl)-1H-pyrazole-3-carboxamide1109Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55785CB1UNDEFINEDUNDEFINEDUNDEFINED7-chloro-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide15Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55786CB1UNDEFINEDUNDEFINEDUNDEFINED8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide0.00035Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55787CB2UNDEFINEDUNDEFINEDUNDEFINED7-chloro-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide230Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55788CB2UNDEFINEDUNDEFINEDUNDEFINED8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide20Zhang Y et al., 2008Jan 15, 2025Jan 15, 2025
55789AChEUNDEFINEDHUMANUNDEFINEDIrinotecan50.5Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55790AChEUNDEFINEDHUMANUNDEFINEDBW284C5110Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55791AChEUNDEFINEDHUMANUNDEFINED2-(2,6-bis(2-(diethylamino)ethoxy)phenoxy)-N,N-diethylethanamine>10000Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55792AChEUNDEFINEDHUMANUNDEFINEDN-{4-[(1,2,3, 4-Tetrahydroacridin-9-yl)amino]butyl}-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)sulfanyl]propyl}acetamide27.95Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55793SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline4.11Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55794SLC6A4UNDEFINEDHUMANUNDEFINEDMDMA0.73Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55795SLC6A4UNDEFINEDHUMANUNDEFINEDCITALOPRAM4.38Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55796SLC6A4UNDEFINEDHUMANUNDEFINEDPAROXETINE0.42Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55797SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline213Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55798SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline374Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55799SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline1910Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55800SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline11.4Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55801SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline6.46Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55802SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline25.3Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55803SLC6A4UNDEFINEDHUMANUNDEFINEDMDMA2.03Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55804SLC6A4UNDEFINEDHUMANUNDEFINEDCITALOPRAM32.8Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55805SLC6A4UNDEFINEDHUMANUNDEFINEDPAROXETINE0.38Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55806SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline2660Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55807SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline1110Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55808SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline2980Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55809SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline13.3Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55810SLC6A4UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline44.7Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
558115-HT1AUNDEFINEDRATUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline54Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
558125-HT1AUNDEFINEDRATUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline1120Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
558135-HT1AUNDEFINEDRATUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline685Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
558145-HT1AUNDEFINEDRATUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline1990Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
558155-HT1AUNDEFINEDRATUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline50Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
558165-HT1AUNDEFINEDRATUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline164Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55817SLC6A2UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline1680Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55818SLC6A2UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline1810Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55819SLC6A2UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline712Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55820SLC6A2UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline6600Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55821SLC6A2UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline2770Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55822SLC6A2UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline2880Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55823SLC6A3UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline2490Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55824SLC6A3UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline1155Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55825SLC6A3UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Iodo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro isoquinoline3650Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55826SLC6A3UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline3490Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55827SLC6A3UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Bromo-1H-indol-3-yl)-propyl]-6-methoxy-1,2,3,4-tetrahydro-isoquinoline1030Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55828SLC6A3UNDEFINEDHUMANUNDEFINED[C11]-2-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-5-methoxy-1,2,3,4-tetrahydro-isoquinoline1485Ben-Daniel R et al., 2008Jan 15, 2025Jan 15, 2025
55829D1UNDEFINEDRATUNDEFINEDRISPERIDONE50Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55830D1UNDEFINEDRATUNDEFINEDOPC-145971960Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55831D1UNDEFINEDRATUNDEFINEDOLANZAPINE25Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55832D1UNDEFINEDRATUNDEFINEDCLOZAPINE353Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55833D1UNDEFINEDRATUNDEFINEDHALOPERIDOL318Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55834D1UNDEFINEDRATUNDEFINED3,4-Dihydro-2-[4-(3,4-dihydro-6-methoxypyrazino[1,2-a]indol-2(1H)-yl)butyl]pyrazino[1,2-a]indol-1(2H)-one>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55835D1UNDEFINEDRATUNDEFINED3-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyloxy]isoquinoline7124Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55836D1UNDEFINEDRATUNDEFINEDN-(4-(4-(m-Tolyl)piperazin-1-yl)butyl)benzo[b]furan-2-carboxamide3290Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55837D1UNDEFINEDRATUNDEFINEDN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one4370Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55838D1UNDEFINEDRATUNDEFINEDN-[4-[4-(2,4-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one4315Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55839D1UNDEFINEDRATUNDEFINEDN-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55840D1UNDEFINEDRATUNDEFINEDN-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55841D1UNDEFINEDRATUNDEFINEDN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide4600Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55842D1UNDEFINEDRATUNDEFINEDN-[4-[4-(3-Chlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide5500Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55843D1UNDEFINEDRATUNDEFINEDN-[4-(3,4-Dihydro-6-methoxypyrazino[1,2-a]1ndol-2(1H)-yl)-butyl]isoquinoline-3-carboxamide>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55844D1UNDEFINEDRATUNDEFINEDN-[4-(1,2,3,4-Tetrahydro-5-methoxy--carbolin-2-yl)butyl]isoquinoline-3-carboxamide>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55845D3UNDEFINEDUNDEFINEDUNDEFINED1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide0.18Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55846D3UNDEFINEDUNDEFINEDUNDEFINED5-Chloro-1H-indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide0.38Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55847D3UNDEFINEDUNDEFINEDUNDEFINEDRISPERIDONE6.7Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55848D3UNDEFINEDUNDEFINEDUNDEFINEDOPC-145973.3Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55849D3UNDEFINEDUNDEFINEDUNDEFINEDOLANZAPINE39Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55850D3UNDEFINEDUNDEFINEDUNDEFINEDCLOZAPINE319Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55851D3UNDEFINEDUNDEFINEDUNDEFINEDHALOPERIDOL0.9Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55852D3UNDEFINEDUNDEFINEDUNDEFINED3,4-Dihydro-2-[4-(3,4-dihydro-6-methoxypyrazino[1,2-a]indol-2(1H)-yl)butyl]pyrazino[1,2-a]indol-1(2H)-one8.6Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55853D3UNDEFINEDUNDEFINEDUNDEFINED3-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyloxy]isoquinoline0.14Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55854D3UNDEFINEDUNDEFINEDUNDEFINED3-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butoxy]isoquinoline32.92Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55855D3UNDEFINEDUNDEFINEDUNDEFINED7-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyloxy]quinoline8.2Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55856D3UNDEFINEDUNDEFINEDUNDEFINEDN-(4-(4-(m-Tolyl)piperazin-1-yl)butyl)benzo[b]furan-2-carboxamide4.5Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55857D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one0.105Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55858D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-[4-(2,4-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one3.2Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55859D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one3.7Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55860D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide0.54Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55861D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide0.099Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55862D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-[4-(3-Chlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide0.27Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55863D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-(3,4-Dihydro-6-methoxypyrazino[1,2-a]1ndol-2(1H)-yl)-butyl]isoquinoline-3-carboxamide33.5Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55864D3UNDEFINEDUNDEFINEDUNDEFINEDN-[4-(1,2,3,4-Tetrahydro-5-methoxy--carbolin-2-yl)butyl]isoquinoline-3-carboxamide6Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558655-HT1AUNDEFINEDRATUNDEFINED1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558665-HT1AUNDEFINEDRATUNDEFINED5-Chloro-1H-indole-2-carboxylic acid {4-[4-(2,4-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide>10000Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558675-HT1AUNDEFINEDRATUNDEFINEDRISPERIDONE190Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558685-HT1AUNDEFINEDRATUNDEFINEDOPC-145975.6Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558695-HT1AUNDEFINEDRATUNDEFINEDOLANZAPINE610Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558705-HT1AUNDEFINEDRATUNDEFINEDCLOZAPINE160Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558715-HT1AUNDEFINEDRATUNDEFINEDHALOPERIDOL1800Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558725-HT1AUNDEFINEDRATUNDEFINED3,4-Dihydro-2-[4-(3,4-dihydro-6-methoxypyrazino[1,2-a]indol-2(1H)-yl)butyl]pyrazino[1,2-a]indol-1(2H)-one33Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558735-HT1AUNDEFINEDRATUNDEFINED3-[5-[4-(2,3-Dichlorophenyl)piperazin-1-yl]pentyloxy]isoquinoline18Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558745-HT1AUNDEFINEDRATUNDEFINED3-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butoxy]isoquinoline24.2Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558755-HT1AUNDEFINEDRATUNDEFINED7-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyloxy]quinoline4Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558765-HT1AUNDEFINEDRATUNDEFINEDN-(4-(4-(m-Tolyl)piperazin-1-yl)butyl)benzo[b]furan-2-carboxamide11.9Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558775-HT1AUNDEFINEDRATUNDEFINEDN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]3,4-dihydropyrazino[1,2-a]indol-1(2H)-one9.3Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558785-HT1AUNDEFINEDRATUNDEFINEDN-[4-[4-(3-Cyanophenyl)piperazin-1-yl]butyl]benzo[b]furan-2-carboxamide876Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558795-HT1AUNDEFINEDRATUNDEFINEDN-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide5Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558805-HT1AUNDEFINEDRATUNDEFINEDN-[4-[4-(3-Chlorophenyl)piperazin-1-yl]butyl]isoquinoline-3-carboxamide14.7Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558815-HT1AUNDEFINEDRATUNDEFINEDN-[4-(3,4-Dihydro-6-methoxypyrazino[1,2-a]1ndol-2(1H)-yl)-butyl]isoquinoline-3-carboxamide28Butini S et al., 2009Jan 15, 2025Jan 15, 2025
558825-HT1AUNDEFINEDRATUNDEFINEDN-[4-(1,2,3,4-Tetrahydro-5-methoxy--carbolin-2-yl)butyl]isoquinoline-3-carboxamide118Butini S et al., 2009Jan 15, 2025Jan 15, 2025
55883MORUNDEFINEDHUMANUNDEFINEDTramadol(+-)1600Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55884MORUNDEFINEDHUMANUNDEFINEDrel-3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)benzamide9.5Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55885MORUNDEFINEDHUMANUNDEFINED3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol8.6Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55886MORUNDEFINEDHUMANUNDEFINED(1S,2S,7S,8R,12S,20R,24R,32R)-9,33-bis(cyclopropylmethyl)-2,7-dihydroxy-19,25-dioxa-9,22,33-triazaundecacyclo[24.9.1.1^{8,14}.0^{1,24}.0^{2,32}.0^{4,23}.0^{5,21}.0^{7,12}.0^{12,20}.0^{13,18}.0^{30,36}]heptatriaconta-13(18),14,16,26(36),27,29-hexaene-17,27400Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55887MORUNDEFINEDHUMANUNDEFINEDnorbinaltorphimine2.7Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55888MORUNDEFINEDHUMANUNDEFINED(1S,2R,6S,14R,15S,16R)-3-(cyclopropylmethyl)-16-[(2R)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.1^{2,8}.0^{1,6}.0^{6,14}.0^{7,12}]icosa-7(12),8,10-triene-11-carboxamide0.77Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55889MORUNDEFINEDHUMANUNDEFINEDBUPRENORPHINE0.21Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55890MORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,14S,17R)-14-hydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18),15-tetraene-10-carboxamide18Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55891MORUNDEFINEDHUMANUNDEFINEDNalorphine0.19Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55892MORUNDEFINEDHUMANUNDEFINEDCyclazocine0.16Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55893MORUNDEFINEDHUMANUNDEFINED3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide0.31Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55894MORUNDEFINEDHUMANUNDEFINEDNaltrexone0.11Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55895MORUNDEFINEDHUMANUNDEFINED3-desoxy-3-carboxamidonaltrexone0.71Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55896MORUNDEFINEDHUMANUNDEFINEDPENTAZOCINE (-)6.9Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55897MORUNDEFINEDHUMANUNDEFINEDrel-(2R,6R,11R)-6,11-Dimethyl-3-(3-methyl-but-2-enyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide5.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55898MORUNDEFINEDHUMANUNDEFINEDMetazocine3.8Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55899MORUNDEFINEDHUMANUNDEFINED3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide1.6Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55900MORUNDEFINEDHUMANUNDEFINEDPhenazocine0.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55901MORUNDEFINEDHUMANUNDEFINED6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide0.015Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55902MORUNDEFINEDHUMANUNDEFINEDButorphanol0.12Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55903MORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclobutylmethyl)-10-hydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-triene-4-carboxamide0.15Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55904MORUNDEFINEDHUMANUNDEFINEDNaloxone(-)0.66Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55905MORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17S)-17-hydroxy-14-oxo-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide4.5Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55906MORUNDEFINEDHUMANUNDEFINEDNaltrexone-6-beta-ol0.19Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55907MORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide2.5Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55908MORUNDEFINEDHUMANUNDEFINEDNaltrexone-6-alpha-ol0.21Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55909MORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14S,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide7.1Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55910MORUNDEFINEDHUMANUNDEFINEDnalmefene0.44Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55911MORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide2.6Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55912DORUNDEFINEDHUMANUNDEFINEDTramadol(+-)9.4Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55913DORUNDEFINEDHUMANUNDEFINEDrel-3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)benzamide2400Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55914DORUNDEFINEDHUMANUNDEFINED3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol2900Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55915DORUNDEFINEDHUMANUNDEFINED(1S,2S,7S,8R,12S,20R,24R,32R)-9,33-bis(cyclopropylmethyl)-2,7-dihydroxy-19,25-dioxa-9,22,33-triazaundecacyclo[24.9.1.1^{8,14}.0^{1,24}.0^{2,32}.0^{4,23}.0^{5,21}.0^{7,12}.0^{12,20}.0^{13,18}.0^{30,36}]heptatriaconta-13(18),14,16,26(36),27,29-hexaene-17,271000Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55916DORUNDEFINEDHUMANUNDEFINEDnorbinaltorphimine24Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55917DORUNDEFINEDHUMANUNDEFINED(1S,2R,6S,14R,15S,16R)-3-(cyclopropylmethyl)-16-[(2R)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.1^{2,8}.0^{1,6}.0^{6,14}.0^{7,12}]icosa-7(12),8,10-triene-11-carboxamide54Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55918DORUNDEFINEDHUMANUNDEFINEDBUPRENORPHINE2.9Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55919DORUNDEFINEDHUMANUNDEFINEDNalorphine120Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55920DORUNDEFINEDHUMANUNDEFINEDCyclazocine2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55921DORUNDEFINEDHUMANUNDEFINED3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide5.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55922DORUNDEFINEDHUMANUNDEFINEDNaltrexone60Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55923DORUNDEFINEDHUMANUNDEFINED3-desoxy-3-carboxamidonaltrexone550Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55924DORUNDEFINEDHUMANUNDEFINEDPENTAZOCINE (-)180Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55925DORUNDEFINEDHUMANUNDEFINEDrel-(2R,6R,11R)-6,11-Dimethyl-3-(3-methyl-but-2-enyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide220Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55926DORUNDEFINEDHUMANUNDEFINEDMetazocine140Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55927DORUNDEFINEDHUMANUNDEFINED3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide320Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55928DORUNDEFINEDHUMANUNDEFINEDPhenazocine5Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55929DORUNDEFINEDHUMANUNDEFINED6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide1.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55930DORUNDEFINEDHUMANUNDEFINEDButorphanol12Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55931DORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclobutylmethyl)-10-hydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-triene-4-carboxamide14Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55932DORUNDEFINEDHUMANUNDEFINEDNaloxone(-)120Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55933DORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17S)-17-hydroxy-14-oxo-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide1000Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55934DORUNDEFINEDHUMANUNDEFINEDNaltrexone-6-beta-ol53Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55935DORUNDEFINEDHUMANUNDEFINEDNaltrexone-6-alpha-ol56Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55936DORUNDEFINEDHUMANUNDEFINEDnalmefene9.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55937DORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide67Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55938DORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,14S,17R)-14-hydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18),15-tetraene-10-carboxamide>10000Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55939DORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide>10000Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55940DORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14S,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide>10000Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55941KORUNDEFINEDHUMANUNDEFINEDTramadol(+-)14Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55942KORUNDEFINEDHUMANUNDEFINEDrel-3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)benzamide350Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55943KORUNDEFINEDHUMANUNDEFINED3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol450Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55944KORUNDEFINEDHUMANUNDEFINED(1S,2S,7S,8R,12S,20R,24R,32R)-9,33-bis(cyclopropylmethyl)-2,7-dihydroxy-19,25-dioxa-9,22,33-triazaundecacyclo[24.9.1.1^{8,14}.0^{1,24}.0^{2,32}.0^{4,23}.0^{5,21}.0^{7,12}.0^{12,20}.0^{13,18}.0^{30,36}]heptatriaconta-13(18),14,16,26(36),27,29-hexaene-17,2721Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55945KORUNDEFINEDHUMANUNDEFINEDnorbinaltorphimine0.027Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55946KORUNDEFINEDHUMANUNDEFINED(1S,2R,6S,14R,15S,16R)-3-(cyclopropylmethyl)-16-[(2R)-2-hydroxy-3,3-dimethylbutan-2-yl]-15-methoxy-13-oxa-3-azahexacyclo[13.2.2.1^{2,8}.0^{1,6}.0^{6,14}.0^{7,12}]icosa-7(12),8,10-triene-11-carboxamide2.1Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55947KORUNDEFINEDHUMANUNDEFINEDBUPRENORPHINE0.62Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55948KORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,14S,17R)-14-hydroxy-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18),15-tetraene-10-carboxamide100Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55949KORUNDEFINEDHUMANUNDEFINEDNalorphine0.38Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55950KORUNDEFINEDHUMANUNDEFINEDCyclazocine0.07Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55951KORUNDEFINEDHUMANUNDEFINED3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide0.06Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55952KORUNDEFINEDHUMANUNDEFINEDNaltrexone0.19Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55953KORUNDEFINEDHUMANUNDEFINED3-desoxy-3-carboxamidonaltrexone0.36Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55954KORUNDEFINEDHUMANUNDEFINEDPENTAZOCINE (-)3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55955KORUNDEFINEDHUMANUNDEFINEDrel-(2R,6R,11R)-6,11-Dimethyl-3-(3-methyl-but-2-enyl)-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide5.6Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55956KORUNDEFINEDHUMANUNDEFINEDMetazocine9.9Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55957KORUNDEFINEDHUMANUNDEFINED3,6,11-Trimethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide19Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55958KORUNDEFINEDHUMANUNDEFINEDPhenazocine2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55959KORUNDEFINEDHUMANUNDEFINED6,11-Dimethyl-3-phenethyl-1,2,3,4,5,6-hexahydro-2,6-methano-benzo[d]azocine-8-carboxylic acid amide0.55Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55960KORUNDEFINEDHUMANUNDEFINEDButorphanol0.22Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55961KORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclobutylmethyl)-10-hydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2,4,6-triene-4-carboxamide0.39Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55962KORUNDEFINEDHUMANUNDEFINEDNaloxone(-)1.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55963KORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17S)-17-hydroxy-14-oxo-4-(prop-2-en-1-yl)-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide46Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55964KORUNDEFINEDHUMANUNDEFINEDNaltrexone-6-beta-ol0.48Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55965KORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14R,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide30Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55966KORUNDEFINEDHUMANUNDEFINEDNaltrexone-6-alpha-ol0.56Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55967KORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14S,17S)-4-(cyclopropylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide100Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55968KORUNDEFINEDHUMANUNDEFINEDnalmefene0.12Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55969KORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-14-methylidene-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7,9,11(18)-triene-10-carboxamide2.1Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
55970SLC6A4UNDEFINEDRATUNDEFINEDFLUOXETINE48Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55971SLC6A4UNDEFINEDRATUNDEFINEDNisoxetine277Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55972SLC6A4UNDEFINEDRATUNDEFINEDTomoxetine1500Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55973SLC6A4UNDEFINEDRATUNDEFINEDDuloxetine4.6Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55974SLC6A4UNDEFINEDRATUNDEFINEDDuloxetine8.8Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55975SLC6A4UNDEFINEDRATUNDEFINED(R)-N-methyl-3-(naphthalen-1-yl)-3-(thiophen-2-yl)propan-1-amine hydrochloride12.1Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55976SLC6A4UNDEFINEDRATUNDEFINED(S)-N-methyl-3-(naphthalen-1-yl)-3-(thiophen-2-yl)propan-1-amine hydrochloride30.2Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55977SLC6A4UNDEFINEDRATUNDEFINED(R)-N-methyl-4-(naphthalen-1-yl)-4-(thiophen-2-yl)butan-1-amine hydrochloride9.5Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55978SLC6A4UNDEFINEDRATUNDEFINED(S)-N-methyl-4-(naphthalen-1-yl)-4-(thiophen-2-yl)butan-1-amine hydrochloride39.7Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55979SLC6A4UNDEFINEDRATUNDEFINED(R)-3-(1H-indol-4-yl)-N-methyl-3-(thiophen-2-yl)propan-1-amine hydrochloride166Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55980SLC6A4UNDEFINEDRATUNDEFINED(S)-3-(1H-indol-4-yl)-N-methyl-3-(thiophen-2-yl)propan-1-amine hydrochloride31.9Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55981SLC6A4UNDEFINEDRATUNDEFINED(R)-4-(1H-indol-4-yl)-N-methyl-4-(thiophen-2-yl)butan-1-amine hydrochloride271Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55982SLC6A4UNDEFINEDRATUNDEFINED(S)-4-(1H-indol-4-yl)-N-methyl-4-(thiophen-2-yl)butan-1-amine hydrochloride72.9Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55983SLC6A4UNDEFINEDRATUNDEFINED(S)-3-(3,4-dichlorophenyl)-N-methyl-3-(naphthalen-1-yl)propan-1-amine hydrochloride86Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55984SLC6A4UNDEFINEDRATUNDEFINED(R)-3-(3,4-dichlorophenyl)-N-methyl-3-(naphthalen-1-yl)propan-1-amine hydrochloride5.3Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55985SLC6A4UNDEFINEDRATUNDEFINED(S)-4-(3,4-dichlorophenyl)-N-methyl-4-(naphthalen-1-yl)butan-1-amine hydrochloride49.9Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55986SLC6A4UNDEFINEDRATUNDEFINED(R)-4-(3,4-dichlorophenyl)-N-methyl-4-(naphthalen-1-yl)butan-1-amine hydrochloride4.1Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55987SLC6A4UNDEFINEDRATUNDEFINED(S)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride3.63Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55988SLC6A4UNDEFINEDRATUNDEFINED(R)-3-(3,4-dichlorophenyl)-3-(1H-indol-4-yl)-N-methylpropan-1-amine hydrochloride1.68Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55989SLC6A4UNDEFINEDRATUNDEFINED(S)-4-(1-(3,4-dimethylphenyl)hexyl)-1H-indene hydrochloride2.72Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55990SLC6A4UNDEFINEDRATUNDEFINED(R)-4-(3,4-dichlorophenyl)-4-(1H-indol-4-yl)-N-methylbutan-1-amine hydrochloride0.82Manning JR et al., 2009Jan 15, 2025Jan 15, 2025
55991CB1UNDEFINEDHUMANUNDEFINEDRimonabant0.9Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55992CB1UNDEFINEDHUMANUNDEFINED1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride0.7Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55993CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-9H-purin-6-amine7.4Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55994CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophenyl)-9H-purin-6-amine7.1Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55995CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(piperidin-1-yl)-9H-purine6.1Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55996CB1UNDEFINEDHUMANUNDEFINED8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(piperidin-1-yl)-9H-purine2.3Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55997CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine5.2Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55998CB1UNDEFINEDHUMANUNDEFINED8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine2.8Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
55999CB1UNDEFINEDHUMANUNDEFINEDRimonabant0.19Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56000CB1UNDEFINEDHUMANUNDEFINED1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic Acid Amide Hydrochloride0.12Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56001CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-9H-purin-6-amine1.7Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56002CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-N-cyclohexyl-8-(2,4-dichlorophenyl)-9H-purin-6-amine1.5Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56003CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(piperidin-1-yl)-9H-purine1.7Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56004CB1UNDEFINEDHUMANUNDEFINED8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(piperidin-1-yl)-9H-purine1.1Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56005CB1UNDEFINEDHUMANUNDEFINED9-(4-chlorophenyl)-8-(2,4-dichlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine1.5Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56006CB1UNDEFINEDHUMANUNDEFINED8-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)-9H-purine1.6Griffith DA et al., 2009Jan 15, 2025Jan 15, 2025
56007D1UNDEFINEDRATUNDEFINEDAcetic acid (R)-2-methoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester526Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56008D1UNDEFINEDRATUNDEFINED11-Hydroxy-N-propylnoraporphine699Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56009D1UNDEFINEDRATUNDEFINED(R)-2-Methoxyaporphin-11-yl pentanoate1480Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56010D1UNDEFINEDRATUNDEFINEDacetic acid (R)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester>10000Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56011D1UNDEFINEDRATUNDEFINEDR(-)-2-methoxy-11-acetyloxy-N-n-propylnoraporphine>10000Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56012D1UNDEFINEDRATUNDEFINEDPentanoic acid (R)-2-methoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl ester>10000Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56013D1UNDEFINEDRATUNDEFINED11-valeryloxynoraporphine>10000Si YG et al., 2009Jan 15, 2025Jan 15, 2025
56014SLC6A3UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester371Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56015SLC6A3UNDEFINEDHUMANUNDEFINEDFLUOXETINE6670Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56016SLC6A3UNDEFINEDHUMANUNDEFINEDNORFLUOXETINE4544Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56017SLC6A3UNDEFINEDHUMANUNDEFINEDNORFLUOXETINE3661Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56018SLC6A3UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56019SLC6A3UNDEFINEDHUMANUNDEFINED2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8atetrahydro-2H-phthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56020SLC6A3UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxyphenyl)-2-(5-((S)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one2716Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56021SLC6A3UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxyphenyl)-2-(5-((R)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one4492Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56022SLC6A4UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester276Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56023SLC6A4UNDEFINEDHUMANUNDEFINEDFLUOXETINE1.1Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56024SLC6A4UNDEFINEDHUMANUNDEFINEDNORFLUOXETINE50Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56025SLC6A4UNDEFINEDHUMANUNDEFINEDNORFLUOXETINE26Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56026SLC6A4UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56027SLC6A4UNDEFINEDHUMANUNDEFINED2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8atetrahydro-2H-phthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56028SLC6A4UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxyphenyl)-2-(5-((S)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one300Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56029SLC6A4UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxyphenyl)-2-(5-((R)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one65Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56030SLC6A2UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester1115Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56031SLC6A2UNDEFINEDHUMANUNDEFINEDFLUOXETINE1560Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56032SLC6A2UNDEFINEDHUMANUNDEFINEDNORFLUOXETINE6186Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56033SLC6A2UNDEFINEDHUMANUNDEFINEDNORFLUOXETINE7490Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56034SLC6A2UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56035SLC6A2UNDEFINEDHUMANUNDEFINED2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8atetrahydro-2H-phthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56036SLC6A2UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxyphenyl)-2-(5-((S)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one4600Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56037SLC6A2UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxyphenyl)-2-(5-((R)-3-phenyl-3-(4-(trifluoromethyl)phenoxy)propylamino)pentyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one6567Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
56038MORUNDEFINEDUNDEFINEDUNDEFINEDNaltrexone0.26Li G et al., 2009Jan 15, 2025Jan 15, 2025
56039MORUNDEFINEDUNDEFINEDUNDEFINEDbeta-funaltrexamine0.41Li G et al., 2009Jan 15, 2025Jan 15, 2025
56040MORUNDEFINEDUNDEFINEDUNDEFINEDD-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr2.02Li G et al., 2009Jan 15, 2025Jan 15, 2025
56041MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-2-carboxylate0.14Li G et al., 2009Jan 15, 2025Jan 15, 2025
56042MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-3-carboxylate1.59Li G et al., 2009Jan 15, 2025Jan 15, 2025
56043MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-4-carboxylate5.58Li G et al., 2009Jan 15, 2025Jan 15, 2025
56044MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl benzoate123.23Li G et al., 2009Jan 15, 2025Jan 15, 2025
56045MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl isoquinoline-3-carboxylate68.4Li G et al., 2009Jan 15, 2025Jan 15, 2025
56046MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-2-carboxylate1.44Li G et al., 2009Jan 15, 2025Jan 15, 2025
56047MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-3-carboxylate2.69Li G et al., 2009Jan 15, 2025Jan 15, 2025
56048MORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl naphthalene-2-carboxylate225.27Li G et al., 2009Jan 15, 2025Jan 15, 2025
56049DORUNDEFINEDUNDEFINEDUNDEFINEDNaltrexone117Li G et al., 2009Jan 15, 2025Jan 15, 2025
56050DORUNDEFINEDUNDEFINEDUNDEFINEDbeta-funaltrexamine27.78Li G et al., 2009Jan 15, 2025Jan 15, 2025
56051DORUNDEFINEDUNDEFINEDUNDEFINEDD-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr1441Li G et al., 2009Jan 15, 2025Jan 15, 2025
56052DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-2-carboxylate117.38Li G et al., 2009Jan 15, 2025Jan 15, 2025
56053DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-3-carboxylate170.3Li G et al., 2009Jan 15, 2025Jan 15, 2025
56054DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-4-carboxylate405.32Li G et al., 2009Jan 15, 2025Jan 15, 2025
56055DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl benzoate>10000Li G et al., 2009Jan 15, 2025Jan 15, 2025
56056DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl isoquinoline-3-carboxylate>10000Li G et al., 2009Jan 15, 2025Jan 15, 2025
56057DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-2-carboxylate22.81Li G et al., 2009Jan 15, 2025Jan 15, 2025
56058DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-3-carboxylate818.43Li G et al., 2009Jan 15, 2025Jan 15, 2025
56059DORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl naphthalene-2-carboxylate907.18Li G et al., 2009Jan 15, 2025Jan 15, 2025
56060KORUNDEFINEDUNDEFINEDUNDEFINEDNaltrexone5.15Li G et al., 2009Jan 15, 2025Jan 15, 2025
56061KORUNDEFINEDUNDEFINEDUNDEFINEDbeta-funaltrexamine0.94Li G et al., 2009Jan 15, 2025Jan 15, 2025
56062KORUNDEFINEDUNDEFINEDUNDEFINEDD-Phe-Cys-Tyr-D-Trp-Arg-Thr-Pen-Thr1012.7Li G et al., 2009Jan 15, 2025Jan 15, 2025
56063KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-2-carboxylate25.5Li G et al., 2009Jan 15, 2025Jan 15, 2025
56064KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-3-carboxylate47.81Li G et al., 2009Jan 15, 2025Jan 15, 2025
56065KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl pyridine-4-carboxylate49.21Li G et al., 2009Jan 15, 2025Jan 15, 2025
56066KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl benzoate586.42Li G et al., 2009Jan 15, 2025Jan 15, 2025
56067KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl isoquinoline-3-carboxylate>10000Li G et al., 2009Jan 15, 2025Jan 15, 2025
56068KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-2-carboxylate67.15Li G et al., 2009Jan 15, 2025Jan 15, 2025
56069KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl quinoline-3-carboxylate148.23Li G et al., 2009Jan 15, 2025Jan 15, 2025
56070KORUNDEFINEDUNDEFINEDUNDEFINED(1S,5R,13R,17S)-4-(cyclopropylmethyl)-10-hydroxy-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-17-yl naphthalene-2-carboxylate46.57Li G et al., 2009Jan 15, 2025Jan 15, 2025
56071CB1UNDEFINEDHUMANUNDEFINEDHU-2101.5Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56072CB1UNDEFINEDHUMANUNDEFINED1-(2,4-Dichlorophenyl)-4-cyano-5-(4-(fluoromethoxy)phenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide10.3Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56073CB1UNDEFINEDHUMANUNDEFINED4-cyano-1-(2,4-dichlorophenyl)-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide11Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56074CB1UNDEFINEDHUMANUNDEFINEDRimonabant40Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56075CB1UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-morpholino-1H-pyrazole-3-carboxamide422Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56076CB1UNDEFINEDHUMANUNDEFINED1-(2-bromophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide4.7Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56077CB1UNDEFINEDHUMANUNDEFINED1-(2-Chloro-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide13Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56078CB1UNDEFINEDHUMANUNDEFINED1-(2-Bromo-4-fluorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide32Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56079CB1UNDEFINEDHUMANUNDEFINED1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide33Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56080CB1UNDEFINEDHUMANUNDEFINED1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide14Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56081CB1UNDEFINEDHUMANUNDEFINED1-(2-Bromophenyl)-5-(4-methoxyphenyl)-N3-(piperidin-1-yl)-1H-pyrazole-3,4-dicarboxamide>10000Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56082CB1UNDEFINEDHUMANUNDEFINED1-(2,4-Dichlorophenyl)-4-cyano-5-(4-iodophenyl)-N-morpholino-1H-pyrazole-3-carboxamide131Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56083CB1UNDEFINEDHUMANUNDEFINED1-(2,4-Dichlorophenyl)-4-cyano-5-(4-bromophenyl)-N-morpholino-1H-pyrazole-3-carboxamide1000Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56084CB1UNDEFINEDHUMANUNDEFINED1-(2,4-Dichlorophenyl)-4-cyano-5-(4-methoxyphenyl)-N-(pyrrolidin-1-yl)-1H-pyrazole-3-carboxamide2Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56085CB1UNDEFINEDHUMANUNDEFINED5-(4-chlorophenyl)-4-cyano-1-(2,4-dichlorophenyl)-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide24Fan H et al., 2009Jan 15, 2025Jan 15, 2025
56086MORUNDEFINEDHUMANUNDEFINEDNaltrexone0.11Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56087MORUNDEFINEDHUMANUNDEFINEDNALTRINDOLE5.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56088MORUNDEFINEDHUMANUNDEFINED(1S,2S,13R,21R)-22-(cyclopropylmethyl)-2-hydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaene-16-carboxamide46Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56089MORUNDEFINEDHUMANUNDEFINED(1R,13S,14R)-24-(cyclopropylmethyl)-13,20-dihydroxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene-19-carboxamide0.51Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56090MORUNDEFINEDHUMANUNDEFINEDhydromorphone0.28Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56091MORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17R)-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide1.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56092MORUNDEFINEDHUMANUNDEFINED(1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56093MORUNDEFINEDHUMANUNDEFINED6-desoxonaltrexone0.24Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56094MORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide2.5Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56095MORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.16Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56096MORUNDEFINEDHUMANUNDEFINEDNaltrexone methiodide2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56097MORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17S)-10-carbamoyl-4-(cyclopropylmethyl)-17-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-4-ium iodide37Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56098MORUNDEFINEDHUMANUNDEFINED(1R,9R,10S)-4-carbamoyl-17-(cyclopropylmethyl)-3,10-dihydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-trien-17-ium iodide1.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56099MORUNDEFINEDHUMANUNDEFINED(1R,9R,10S,13R)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.072Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56100MORUNDEFINEDHUMANUNDEFINEDNalbuphine1.6Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56101MORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14S,17S)-4-(cyclobutylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide3.8Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56102MORUNDEFINEDHUMANUNDEFINED(1R,9R,10S,13S)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.52Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56103MORUNDEFINEDHUMANUNDEFINED3-desoxy-3-carboxamidonaltrexone0.71Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56104MORUNDEFINEDHUMANUNDEFINEDCCDC 710249, HCl salt0.052Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56105DORUNDEFINEDHUMANUNDEFINEDNaltrexone60Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56106DORUNDEFINEDHUMANUNDEFINEDNALTRINDOLE0.14Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56107DORUNDEFINEDHUMANUNDEFINED(1S,2S,13R,21R)-22-(cyclopropylmethyl)-2-hydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaene-16-carboxamide0.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56108DORUNDEFINEDHUMANUNDEFINED(1R,13S,14R)-24-(cyclopropylmethyl)-13,20-dihydroxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene-19-carboxamide0.025Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56109DORUNDEFINEDHUMANUNDEFINEDhydromorphone38Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56110DORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17R)-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide260Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56111DORUNDEFINEDHUMANUNDEFINED(1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide8.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56112DORUNDEFINEDHUMANUNDEFINED6-desoxonaltrexone79Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56113DORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide630Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56114DORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide4.2Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56115DORUNDEFINEDHUMANUNDEFINEDNaltrexone methiodide900Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56116DORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17S)-10-carbamoyl-4-(cyclopropylmethyl)-17-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-4-ium iodide>10000Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56117DORUNDEFINEDHUMANUNDEFINED(1R,9R,10S)-4-carbamoyl-17-(cyclopropylmethyl)-3,10-dihydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-trien-17-ium iodide280Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56118DORUNDEFINEDHUMANUNDEFINED(1R,9R,10S,13R)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide3.9Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56119DORUNDEFINEDHUMANUNDEFINEDNalbuphine580Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56120DORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14S,17S)-4-(cyclobutylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide150Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56121DORUNDEFINEDHUMANUNDEFINED(1R,9R,10S,13S)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide78Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56122DORUNDEFINEDHUMANUNDEFINED3-desoxy-3-carboxamidonaltrexone550Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56123DORUNDEFINEDHUMANUNDEFINEDCCDC 710249, HCl salt2.6Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56124KORUNDEFINEDHUMANUNDEFINEDhydromorphone2.8Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56125KORUNDEFINEDHUMANUNDEFINEDNaltrexone0.19Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56126KORUNDEFINEDHUMANUNDEFINEDNALTRINDOLE2.9Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56127KORUNDEFINEDHUMANUNDEFINED(1S,2S,13R,21R)-22-(cyclopropylmethyl)-2-hydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5(10),6,8,15,17,19(25)-heptaene-16-carboxamide47Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56128KORUNDEFINEDHUMANUNDEFINED(1R,13S,14R)-24-(cyclopropylmethyl)-13,20-dihydroxy-4,24-diazahexacyclo[12.7.3.0^{1,13}.0^{3,11}.0^{5,10}.0^{16,21}]tetracosa-3(11),5(10),6,8,16(21),17,19-heptaene-19-carboxamide0.81Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56129KORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17R)-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide19Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56130KORUNDEFINEDHUMANUNDEFINED(1S,9R,10R)-3-hydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide2.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56131KORUNDEFINEDHUMANUNDEFINED6-desoxonaltrexone0.24Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56132KORUNDEFINEDHUMANUNDEFINED(1S,5R,13S,17S)-4-(cyclopropylmethyl)-17-hydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide16Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56133KORUNDEFINEDHUMANUNDEFINED(1S,9R,10S)-17-(cyclopropylmethyl)-3,10-dihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.29Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56134KORUNDEFINEDHUMANUNDEFINEDNaltrexone methiodide6.3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56135KORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,17S)-10-carbamoyl-4-(cyclopropylmethyl)-17-hydroxy-4-methyl-14-oxo-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-trien-4-ium iodide210Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56136KORUNDEFINEDHUMANUNDEFINED(1R,9R,10S)-4-carbamoyl-17-(cyclopropylmethyl)-3,10-dihydroxy-17-methyl-13-oxo-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-trien-17-ium iodide7.7Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56137KORUNDEFINEDHUMANUNDEFINED(1R,9R,10S,13R)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide0.34Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56138KORUNDEFINEDHUMANUNDEFINEDNalbuphine3Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56139KORUNDEFINEDHUMANUNDEFINED(1S,5R,13R,14S,17S)-4-(cyclobutylmethyl)-14,17-dihydroxy-12-oxa-4-azapentacyclo[9.6.1.0^{1,13}.0^{5,17}.0^{7,18}]octadeca-7(18),8,10-triene-10-carboxamide0.46Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56140KORUNDEFINEDHUMANUNDEFINED(1R,9R,10S,13S)-17-(cyclobutylmethyl)-3,10,13-trihydroxy-17-azatetracyclo[7.5.3.0^{1,10}.0^{2,7}]heptadeca-2(7),3,5-triene-4-carboxamide9Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56141KORUNDEFINEDHUMANUNDEFINED3-desoxy-3-carboxamidonaltrexone11Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
56142KORUNDEFINEDHUMANUNDEFINEDCCDC 710249, HCl salt0.23Wentland MP et al., 2009Jan 15, 2025Jan 15, 2025
561435-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide3775Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561445-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)benzamide>10000Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561455-HT1AUNDEFINEDRATUNDEFINEDN-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide7586Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561465-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide7440Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561475-HT1AUNDEFINEDRATUNDEFINED2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2,5-dioxopyrrolidin-3-yl)acetamide497Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561485-HT1AUNDEFINEDRATUNDEFINEDAdamantane-1-carboxylic acid ((S)-1-{2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-2,5-dioxo-pyrrolidin-3-yl)-amide579Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561495-HT1AUNDEFINEDRATUNDEFINED(S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide8518Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561505-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide1001Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561515-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-5-oxopyrrolidine-2-carboxamide1507Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561525-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide1950Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561535-HT1AUNDEFINEDRATUNDEFINED(S)-1-acetyl-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide6600Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561545-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)pyrrolidine-2-carboxamide3553Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561555-HT1AUNDEFINEDRATUNDEFINED(S)-1-(Adamantane-1-carbonyl)-pyrrolidine-2-carboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-amide350Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561565-HT1AUNDEFINEDRATUNDEFINED(S)-N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-1-(cyclopentanecarbonyl)pyrrolidine-2-carboxamide2013Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561575-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide360Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561585-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide480Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561595-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide230Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561605-HT1AUNDEFINEDRATUNDEFINED2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2,5-dioxopyrrolidin-3-yl)acetamide40Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561615-HT1AUNDEFINEDRATUNDEFINEDN-[(3S)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide63Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561625-HT1AUNDEFINEDRATUNDEFINED(S)-N-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide1730Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561635-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-5-oxopyrrolidine-2-carboxamide390Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561645-HT1AUNDEFINEDRATUNDEFINED(S)-1-acetyl-N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)pyrrolidine-2-carboxamide580Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561655-HT1AUNDEFINEDRATUNDEFINEDN-((S)-1-{4-[4-(3-chlorophenyl)piperazin-1-yl]butyl}pyrrolidin-2,5-dion-3-yl)cyclohexanecarboxamide26Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561665-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)benzamide41Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561675-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide69Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561685-HT1AUNDEFINEDRATUNDEFINED(S)-N-(1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)cyclohexanecarboxamide19Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561695-HT1AUNDEFINEDRATUNDEFINED2-(bicyclo[2.2.1]heptan-2-yl)-N-((S)-1-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2,5-dioxopyrrolidin-3-yl)acetamide9Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561705-HT1AUNDEFINEDRATUNDEFINEDN-[(3S)-1-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}-2,5-dioxopyrrolidin-3-yl]adamantane-1-carboxamide4Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561715-HT1AUNDEFINEDRATUNDEFINED(S)-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-1-(cyclohexanecarbonyl)-5-oxopyrrolidine-2-carboxamide111Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561725-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-5-oxopyrrolidine-2-carboxamide17Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561735-HT1AUNDEFINEDRATUNDEFINED(S)-1-benzoyl-N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide78Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561745-HT1AUNDEFINEDRATUNDEFINED(S)-1-(cyclohexanecarbonyl)-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)pyrrolidine-2-carboxamide19Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561755-HT1AUNDEFINEDRATUNDEFINED(2S)-1-[(adamantan-1-yl)carbonyl]-N-{4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}pyrrolidine-2-carboxamide3Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561765-HT1AUNDEFINEDRATUNDEFINEDBUSPIRONE36Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561775-HT1AUNDEFINEDRATUNDEFINEDN-[2-{4-(2-Methoxyphenyl)-piperazin-1-yl}-ethyl]-pyrrolidine-2,5-dione2087Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561785-HT1AUNDEFINEDRATUNDEFINEDN-[2-{4-(3-Chlorophenyl)-piperazin-1-yl}-ethyl]-pyrrolidine-2,5-dione3675Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561795-HT1AUNDEFINEDRATUNDEFINEDN-[2-{4-(2-Methoxyphenyl)-piperazin-1-yl}-ethyl]-3-cyclohexyl-pyrrolidine-2,5-dione24Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561805-HT1AUNDEFINEDRATUNDEFINEDN-[2-{4-(3-Chlorophenyl)-piperazin-1-yl}-ethyl]-3-cyclohexyl-pyrrolidine-2,5-dione227Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561815-HT1AUNDEFINEDRATUNDEFINED2-{2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-2-aza-spiro[4.5]decane-1,3-dione5.7Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
561825-HT1AUNDEFINEDRATUNDEFINED2-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)-2-azaspiro[4.5]decane-1,3-dione4.3Zajdel P et al., 2009Jan 15, 2025Jan 15, 2025
56183CHRNA4UNDEFINEDRATUNDEFINEDNicotine0.94Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56184CHRNA4UNDEFINEDRATUNDEFINEDEpibatidine0.047Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56185CHRNA4UNDEFINEDRATUNDEFINEDABT-5940.048Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56186CHRNA4UNDEFINEDRATUNDEFINED(1S,4S)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]heptane0.15Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56187CHRNA4UNDEFINEDRATUNDEFINED3-(pyridin-3-yl)-3,6-diazabicyclo[3.2.0]heptane1.2Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56188CHRNA4UNDEFINEDRATUNDEFINED6-(6-chloropyridin-3-yl)-1,6-diazaspiro[3.4]octane21Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56189CHRNA4UNDEFINEDRATUNDEFINED6-(pyridin-3-yl)-1,6-diazaspiro[3.4]octane11Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56190CHRNA4UNDEFINEDRATUNDEFINED7-(6-chloropyridin-3-yl)-1,7-diazaspiro[4.4]nonane48Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56191CHRNA4UNDEFINEDRATUNDEFINED7-(pyridin-3-yl)-1,7-diazaspiro[4.4]nonane33Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56192CHRNA4UNDEFINEDRATUNDEFINED2-(6-chloropyridin-3-yl)-2,7-diazaspiro[4.4]nonane240Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56193CHRNA4UNDEFINEDRATUNDEFINED2-(pyridin-3-yl)-2,7-diazaspiro[4.4]nonane74Sippy KB et al., 2009Jan 15, 2025Jan 15, 2025
56194Sigmar1UNDEFINEDUNDEFINEDUNDEFINED6-allyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-one1600Holl R et al., 2009Jan 15, 2025Jan 15, 2025
56195Sigmar1UNDEFINEDUNDEFINEDUNDEFINED6-benzyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-one53Holl R et al., 2009Jan 15, 2025Jan 15, 2025
56196Sigmar1UNDEFINEDUNDEFINEDUNDEFINED(2S)-6-allyl-8-(4-methoxybenzyl)-6,8-diazabicyclo[3.2.2]nonan-2-ol2240Holl R et al., 2009Jan 15, 2025Jan 15, 2025
56197Sigmar1UNDEFINEDUNDEFINEDUNDEFINED1-benzyl-4-(4-methoxybenzyl)piperazine0.47Holl R et al., 2009Jan 15, 2025Jan 15, 2025
56198Sigmar1UNDEFINEDUNDEFINEDUNDEFINED(R)-(1-benzyl-4-(4-methoxybenzyl)piperazin-2-yl)methanol12Holl R et al., 2009Jan 15, 2025Jan 15, 2025
56199SLC6A3UNDEFINEDHUMANUNDEFINEDBUPROPION441Lapinsky DJ et al., 2009Jan 15, 2025Jan 15, 2025
56200SLC6A3UNDEFINEDHUMANUNDEFINED1-(4-amino-3-iodophenyl)-2-pyrrolidin-1-yl-pentan-1-one28Lapinsky DJ et al., 2009Jan 15, 2025Jan 15, 2025
56201SLC6A3UNDEFINEDHUMANUNDEFINED1-(4-aminophenyl)-2-pyrrolidin-1-yl-pentan-1-one5Lapinsky DJ et al., 2009Jan 15, 2025Jan 15, 2025
56202SLC6A3UNDEFINEDHUMANUNDEFINED1-(4-azio-3-iodophenyl)-2-pyrroldin-1-yl-pentan-1-one78Lapinsky DJ et al., 2009Jan 15, 2025Jan 15, 2025
56203SLC6A3UNDEFINEDHUMANUNDEFINEDpyrovalerone8Lapinsky DJ et al., 2009Jan 15, 2025Jan 15, 2025
56204SLC6A4UNDEFINEDRATUNDEFINEDFLUOXETINE2.7Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56205SLC6A4UNDEFINEDRATUNDEFINED(2S)-2-{[4-(6-Fluoroquinolin-2-yl)-1,4-diazepan-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline3.9Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56206SLC6A4UNDEFINEDRATUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}-1,4-diazepan-1-yl)-quinoline-6-carbonitrile1.1Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56207SLC6A4UNDEFINEDRATUNDEFINED(2S)-8-Methyl-2-[(4-quinolin-2-yl-1,4-diazepan-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]-quinoline7.4Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56208SLC6A4UNDEFINEDRATUNDEFINED2-((3R)-3-Methyl-4-{[(2S)-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}pipera-zin-1-yl)quinoline-6-carbonitrile89.6Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56209SLC6A4UNDEFINEDRATUNDEFINED(2S)-8-Methyl-2-{[(2R)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline32.8Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56210SLC6A4UNDEFINEDRATUNDEFINED(2S)-8-Methyl-2-{[(2S)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline10.3Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56211SLC6A4UNDEFINEDRATUNDEFINED(2S)-8-Methyl-2-[(4-quinolin-2-ylpiperazin-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]quinoline75Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56212SLC6A4UNDEFINEDRATUNDEFINED(2S)-8-Methyl-2-({4-[6-(trifluoromethoxy)quinolin-2-yl]piperazin-1-yl}methyl)-2,3-dihydro-[1,4]dioxino[2,3-f]quinoline148.5Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56213SLC6A4UNDEFINEDRATUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)quino-line-6-carboxamide17Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56214SLC6A4UNDEFINEDRATUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile13.8Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56215SLC6A4UNDEFINEDRATUNDEFINED(2S)-2-{[4-(6-Bromoquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline12.7Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56216SLC6A4UNDEFINEDRATUNDEFINED(2S)-2-{[4-(6-Chloroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline0.88Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56217SLC6A4UNDEFINEDRATUNDEFINED(2S)-2-{[4-(6-Fluoroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline66Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56218SLC6A4UNDEFINEDRATUNDEFINED(2S)-8-Methyl-2-{[4-(6-nitroquinolin-2-yl)piperazin-1-yl]-methyl}-2,3-dihydro[1,4]dioxino[2,3-f]quinoline0.25Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56219SLC6A4UNDEFINEDRATUNDEFINED(S)-2-((4-(1H-Indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)-methyl)-8-methyl-2,3-dihydro-[1,4]dioxino-[2,3-f]quinoline2.34Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562205-HT1AUNDEFINEDHUMANUNDEFINEDCyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide0.9Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562215-HT1AUNDEFINEDHUMANUNDEFINED(2S)-2-{[4-(6-Fluoroquinolin-2-yl)-1,4-diazepan-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline1.5Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562225-HT1AUNDEFINEDHUMANUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}-1,4-diazepan-1-yl)-quinoline-6-carbonitrile2Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562235-HT1AUNDEFINEDHUMANUNDEFINED(2S)-8-Methyl-2-[(4-quinolin-2-yl-1,4-diazepan-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]-quinoline6.8Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562245-HT1AUNDEFINEDHUMANUNDEFINED2-((3R)-3-Methyl-4-{[(2S)-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}pipera-zin-1-yl)quinoline-6-carbonitrile2.8Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562255-HT1AUNDEFINEDHUMANUNDEFINED(2S)-8-Methyl-2-{[(2R)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline5.5Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562265-HT1AUNDEFINEDHUMANUNDEFINED(2S)-8-Methyl-2-{[(2S)-2-methyl-4-quinolin-2-ylpiperazin-1-yl]methyl}-2,3-dihydro[1,4]dioxino-[2,3-f]quinoline167Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562275-HT1AUNDEFINEDHUMANUNDEFINED(2S)-8-Methyl-2-[(4-quinolin-2-ylpiperazin-1-yl)methyl]-2,3-dihydro[1,4]dioxino[2,3-f]quinoline47.3Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562285-HT1AUNDEFINEDHUMANUNDEFINED(2S)-8-Methyl-2-({4-[6-(trifluoromethoxy)quinolin-2-yl]piperazin-1-yl}methyl)-2,3-dihydro-[1,4]dioxino[2,3-f]quinoline172Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562295-HT1AUNDEFINEDHUMANUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)quino-line-6-carboxamide7.2Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562305-HT1AUNDEFINEDHUMANUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile3.7Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562315-HT1AUNDEFINEDHUMANUNDEFINED(2S)-2-{[4-(6-Bromoquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline17.2Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562325-HT1AUNDEFINEDHUMANUNDEFINED(2S)-2-{[4-(6-Chloroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline214.1Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562335-HT1AUNDEFINEDHUMANUNDEFINED(2S)-2-{[4-(6-Fluoroquinolin-2-yl)piperazin-1-yl]methyl}-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline32.9Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562345-HT1AUNDEFINEDHUMANUNDEFINED(2S)-8-Methyl-2-{[4-(6-nitroquinolin-2-yl)piperazin-1-yl]-methyl}-2,3-dihydro[1,4]dioxino[2,3-f]quinoline20Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
562355-HT1AUNDEFINEDHUMANUNDEFINED(S)-2-((4-(1H-Indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)-methyl)-8-methyl-2,3-dihydro-[1,4]dioxino-[2,3-f]quinoline3.02Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56236D2UNDEFINEDHUMANUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile1306Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56237D3UNDEFINEDHUMANUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile1316Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56238D4UNDEFINEDHUMANUNDEFINED2-(4-{[(2S)-8-Methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}piperazin-1-yl)-quinoline-6-carbonitrile1418Zhou D et al., 2009Jan 15, 2025Jan 15, 2025
56239H3UNDEFINEDHUMANUNDEFINED3-methyl-2-(4-(3-(pyrrolidin-1-yl)propoxy)phenyl)quinazolin-4(3H)-one4.2Mitobe Y et al., 2009Jan 15, 2025Jan 15, 2025
56240D1UNDEFINEDUNDEFINEDUNDEFINEDDOPAMINE124Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56241D1UNDEFINEDUNDEFINEDUNDEFINEDAPOMORPHINE72Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56242D1UNDEFINEDUNDEFINEDUNDEFINED(R)-6-Methyl-2-phenyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol88Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56243D1UNDEFINEDUNDEFINEDUNDEFINED(R)-2-(4-Hydroxy-phenyl)-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol755Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56244D1UNDEFINEDUNDEFINEDUNDEFINEDN-Ethyl-2-methylnorapomorphine hydrochloride1340Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56245D1UNDEFINEDUNDEFINEDUNDEFINEDN-Ethyl-2-phenylnorapomorphine hydrochloride31Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56246D1UNDEFINEDUNDEFINEDUNDEFINEDN-Ethyl-2-(4-hydroxyphenyl)-norapomorphine hydrochloride124Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56247D1UNDEFINEDUNDEFINEDUNDEFINEDN-Propyl-2-methylnorapomorphine hydrochloride278Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56248D1UNDEFINEDUNDEFINEDUNDEFINEDN-Propyl-2-phenylnorapomorphine hydrochloride669Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56249D1UNDEFINEDUNDEFINEDUNDEFINEDN-Propyl-2-(4-hydroxyphenyl)-norapomorphine hydrochloride94Herm L et al., 2009Jan 15, 2025Jan 15, 2025
56250D2UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine2300Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56251D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}2,5,7-rimethylimidazo[1,2-c]pyrimidine260Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56252D2UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56253D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine9100Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56254D2UNDEFINEDHUMANUNDEFINED2-(dimethylamino)-6-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-3H-pyrrolo[2,3-d]pyrimidin-4(7H)-one130Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56255D2UNDEFINEDHUMANUNDEFINED7-Chloro-3-[(4-phenylpiperazin-1-yl)methyl]-1Hpyrrolo[2,3-c]pyridine2600Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56256D2UNDEFINEDHUMANUNDEFINED2,5,7-Trimethyl-3-[4-(phenylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine8600Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56257D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Chlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56258D2UNDEFINEDHUMANUNDEFINED3-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine3300Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56259D2UNDEFINEDHUMANUNDEFINED2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56260D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine4700Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56261D2UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-5,7-dimethylimidazo[1,2-c]pyrimidine1300Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56262D2UNDEFINEDHUMANUNDEFINED3-Methyl-7-[(4-phenylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one390Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56263D2UNDEFINEDHUMANUNDEFINED7-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one570Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56264D2UNDEFINEDHUMANUNDEFINED3-Methyl-7-[(4-pyridin-2-ylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one270Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56265D2UNDEFINEDHUMANUNDEFINED7-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one840Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56266D2UNDEFINEDHUMANUNDEFINED3-Methyl-2-morpholin-4-yl-7-[(4-phenylpiperazin-1-yl)methyl]-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one1100Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56267D2UNDEFINEDHUMANUNDEFINEDCLOZAPINE41Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56268D2UNDEFINEDHUMANUNDEFINEDL-745870>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56269D2UNDEFINEDHUMANUNDEFINED5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-N,N,6-trimethyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine2600Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56270D2UNDEFINEDHUMANUNDEFINED5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-N,N,6-trimethyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine2900Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56271D2UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine2900Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56272D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}2,5,7-rimethylimidazo[1,2-c]pyrimidine160Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56273D2UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56274D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56275D2UNDEFINEDHUMANUNDEFINED2-(dimethylamino)-6-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-3H-pyrrolo[2,3-d]pyrimidin-4(7H)-one170Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56276D2UNDEFINEDHUMANUNDEFINED7-Chloro-3-[(4-phenylpiperazin-1-yl)methyl]-1Hpyrrolo[2,3-c]pyridine2900Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56277D2UNDEFINEDHUMANUNDEFINED2,5,7-Trimethyl-3-[4-(phenylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56278D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Chlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56279D2UNDEFINEDHUMANUNDEFINED3-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine5500Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56280D2UNDEFINEDHUMANUNDEFINED2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56281D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine3500Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56282D2UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-5,7-dimethylimidazo[1,2-c]pyrimidine570Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56283D2UNDEFINEDHUMANUNDEFINED3-Methyl-7-[(4-phenylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one180Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56284D2UNDEFINEDHUMANUNDEFINED7-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one380Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56285D2UNDEFINEDHUMANUNDEFINED3-Methyl-7-[(4-pyridin-2-ylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one150Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56286D2UNDEFINEDHUMANUNDEFINED7-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one400Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56287D2UNDEFINEDHUMANUNDEFINED3-Methyl-2-morpholin-4-yl-7-[(4-phenylpiperazin-1-yl)methyl]-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one730Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56288D2UNDEFINEDHUMANUNDEFINEDCLOZAPINE28Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56289D2UNDEFINEDHUMANUNDEFINEDL-745870>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56290D3UNDEFINEDHUMANUNDEFINED5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-N,N,6-trimethyl-7H-pyrrolo[2,3-d]pyrimidin-2-amine6100Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56291D3UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine3400Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56292D3UNDEFINEDHUMANUNDEFINED3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}2,5,7-rimethylimidazo[1,2-c]pyrimidine8.5Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56293D3UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56294D3UNDEFINEDHUMANUNDEFINED3-{[4-(4-Methoxyphenyl)piperazin-1-yl]methyl}-2,7-dimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56295D3UNDEFINEDHUMANUNDEFINED2-(dimethylamino)-6-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-3H-pyrrolo[2,3-d]pyrimidin-4(7H)-one960Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56296D3UNDEFINEDHUMANUNDEFINED7-Chloro-3-[(4-phenylpiperazin-1-yl)methyl]-1Hpyrrolo[2,3-c]pyridine6100Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56297D3UNDEFINEDHUMANUNDEFINED2,5,7-Trimethyl-3-[4-(phenylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine4200Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56298D3UNDEFINEDHUMANUNDEFINED3-{[4-(4-Chlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine3100Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56299D3UNDEFINEDHUMANUNDEFINED3-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine1300Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56300D3UNDEFINEDHUMANUNDEFINED2,5,7-Trimethyl-3-[4-(2-pyridin-2-ylpiperazin-1-yl)methyl]imidazo[1,2-c]pyrimidine640Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56301D3UNDEFINEDHUMANUNDEFINED3-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-2,5,7-trimethylimidazo[1,2-c]pyrimidine>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56302D3UNDEFINEDHUMANUNDEFINED3-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-5,7-dimethylimidazo[1,2-c]pyrimidine1500Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56303D3UNDEFINEDHUMANUNDEFINED3-Methyl-7-[(4-phenylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one330Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56304D3UNDEFINEDHUMANUNDEFINED7-{[4-(3,4-Dichlorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one480Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56305D3UNDEFINEDHUMANUNDEFINED3-Methyl-7-[(4-pyridin-2-ylpiperazin-1-yl)methyl]-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one310Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56306D3UNDEFINEDHUMANUNDEFINED7-{[4-(4-Fluorophenyl)piperazin-1-yl]methyl}-3-methyl-2-pyrrolidin-1-yl-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one630Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56307D3UNDEFINEDHUMANUNDEFINED3-Methyl-2-morpholin-4-yl-7-[(4-phenylpiperazin-1-yl)methyl]-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one2700Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56308D3UNDEFINEDHUMANUNDEFINEDCLOZAPINE960Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56309D3UNDEFINEDHUMANUNDEFINEDL-745870>10000Linz S et al., 2009Jan 15, 2025Jan 15, 2025
56310A2AUNDEFINEDHUMANUNDEFINEDCGS 2168046.2Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56311A2AUNDEFINEDHUMANUNDEFINEDCaffeine (1,3,7-trimethylxanthine)>10000Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56312A2AUNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione1470Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56313A2AUNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione164Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56314A2AUNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione3630Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56315A2AUNDEFINEDHUMANUNDEFINED2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione570Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56316A2AUNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione893Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56317A2AUNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione>10000Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56318A1UNDEFINEDHUMANUNDEFINEDXAC9Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56319A1UNDEFINEDHUMANUNDEFINEDCaffeine (1,3,7-trimethylxanthine)>10000Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56320A1UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione921Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56321A1UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione346Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56322A1UNDEFINEDHUMANUNDEFINED2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione132Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56323A1UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione1410Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56324A1UNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione379Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56325A1UNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione>10000Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56326A3UNDEFINEDHUMANUNDEFINEDNECA20Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56327A3UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione209Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56328A3UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione3.82Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56329A3UNDEFINEDHUMANUNDEFINED2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione16.8Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56330A3UNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione13.9Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56331A3UNDEFINEDHUMANUNDEFINED2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione290Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56332A3UNDEFINEDHUMANUNDEFINED2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione526Ishiyama H et al., 2009Jan 15, 2025Jan 15, 2025
56333Chrna3UNDEFINEDRATUNDEFINEDNicotine47Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56334Chrna3UNDEFINEDRATUNDEFINEDEpibatidine0.035Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56335Chrna3UNDEFINEDRATUNDEFINED3-((S)-1-Azetidin-2-ylmethoxy)-2-fluoro-pyridine3Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56336Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine0.25Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56337Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine0.33Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56338Chrna3UNDEFINEDRATUNDEFINED5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine0.041Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56339Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine0.26Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56340Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(R)-pyrrolidinyl)methoxy)pyridine0.85Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56341Chrna3UNDEFINEDRATUNDEFINED(S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine0.71Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56342Chrna3UNDEFINEDRATUNDEFINEDNicotine440Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56343Chrna3UNDEFINEDRATUNDEFINEDEpibatidine0.57Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56344Chrna3UNDEFINEDRATUNDEFINED3-((S)-1-Azetidin-2-ylmethoxy)-2-fluoro-pyridine3700Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56345Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine43Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56346Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine90Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56347Chrna3UNDEFINEDRATUNDEFINED5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine79Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56348Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine320Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56349Chrna3UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(R)-pyrrolidinyl)methoxy)pyridine350Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56350Chrna3UNDEFINEDRATUNDEFINED(S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine590Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56351CHRNA4UNDEFINEDRATUNDEFINEDNicotine10Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56352CHRNA4UNDEFINEDRATUNDEFINEDEpibatidine0.061Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56353CHRNA4UNDEFINEDRATUNDEFINED3-((S)-1-Azetidin-2-ylmethoxy)-2-fluoro-pyridine1.3Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56354CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine0.13Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56355CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine0.062Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56356CHRNA4UNDEFINEDRATUNDEFINED5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine0.028Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56357CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine0.055Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56358CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(R)-pyrrolidinyl)methoxy)pyridine1.1Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56359CHRNA4UNDEFINEDRATUNDEFINED(S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine0.062Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56360CHRNA4UNDEFINEDRATUNDEFINEDNicotine40Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56361CHRNA4UNDEFINEDRATUNDEFINEDEpibatidine0.16Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56362CHRNA4UNDEFINEDRATUNDEFINED3-((S)-1-Azetidin-2-ylmethoxy)-2-fluoro-pyridine190Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56363CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-(2-(S)-pyrrolidinyl)methoxy)-pyridine1.1Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56364CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-fluoro-4-(pyridinyl)methoxy)-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)pyridine1.6Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56365CHRNA4UNDEFINEDRATUNDEFINED5-(((S)-Pyrrolidin-2-yl)methoxy)-3-((6-chloropyridin-3-yl)methoxy)-2-chloropyridine0.49Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56366CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(S)-pyrrolidinyl)methoxy)pyridine6.6Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56367CHRNA4UNDEFINEDRATUNDEFINED2-Chloro-3-(2-chloro-5-(pyridinyl)methoxy)-5-((1-methyl)-2-(R)-pyrrolidinyl)methoxy)pyridine7.6Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56368CHRNA4UNDEFINEDRATUNDEFINED(S)-2-chloro-2'-fluoro-5-((1-methylpyrrolidin-2-yl)methoxy)-3,4'-bipyridine16Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56369CHRNA4UNDEFINEDRATUNDEFINED(S)-2-chloro-5-((1-methylpyrrolidin-2-yl)methoxy)-3-(2-(pyridin-4-yl)vinyl)pyridine0.028Gao Y et al., 2009Jan 15, 2025Jan 15, 2025
56370CB1UNDEFINEDHUMANUNDEFINEDRimonabant1.9Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56371CB1UNDEFINEDHUMANUNDEFINEDibipinabant7.8Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56372CB1UNDEFINEDHUMANUNDEFINEDTaranabant0.3Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56373CB1UNDEFINEDHUMANUNDEFINED2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one2.2Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56374CB1UNDEFINEDHUMANUNDEFINED1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone227Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56375CB1UNDEFINEDHUMANUNDEFINED4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzamide256Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56376CB1UNDEFINEDHUMANUNDEFINED2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,3-d]pyrimidin-4-ylthio)-N-(2-methoxyphenyl)propanamide264Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56377CB1UNDEFINEDHUMANUNDEFINEDethyl 2-(6-bromo-2-(4-fluorophenyl)-4-phenyl-1,2-dihydroquinazolin-3(4H)-yl)acetate273Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56378CB1UNDEFINEDHUMANUNDEFINEDethyl 4-(3-(2-chlorophenyl)-1-(2,4-dimethylphenyl)-1H-pyrazole-5-carbonyl)piperazine-1-carboxylate287Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56379CB1UNDEFINEDHUMANUNDEFINED3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)urea308Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56380CB1UNDEFINEDHUMANUNDEFINED2-[2-(2,4,6-Trimethyl-phenoxy)-acetylamino]-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid (1,1-dioxo-tetrahydro-1lambda*6*-thiophen-3-yl)-amide325Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56381CB1UNDEFINEDHUMANUNDEFINEDN-cyclopropyl-N-(2-oxo-2-(4-p-tolylpyrrolo[1,2-a]quinoxalin-5(4H)-yl)ethyl)cyclopentanecarboxamide520Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56382CB1UNDEFINEDHUMANUNDEFINED2-(1-(4-(4-chlorophenyl)-2,2,4-trimethyl-3,4-dihydroquinolin-1(2H)-yl)-1-oxopropan-2-yl)hexahydro-1H-isoindole-1,3(2H)-dione520Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56383CB1UNDEFINEDHUMANUNDEFINEDN-benzhydryl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-2-fluorobenzamide611Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56384CB1UNDEFINEDHUMANUNDEFINEDN-(2-(4-(4-fluorophenyl)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-2-oxoethyl)-N-isobutylfuran-2-carboxamide875Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56385CB1UNDEFINEDHUMANUNDEFINEDN-(2-(4-(4-fluorophenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)-N-isopropyl-3,3-dimethylbutanamide1030Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56386CB1UNDEFINEDHUMANUNDEFINEDN-phenyl-N-(1-(phenylcarbamoyl)cyclohexyl)-4-(1H-tetrazol-1-yl)benzamide1049Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56387CB1UNDEFINEDHUMANUNDEFINEDethyl 6'-amino-1-benzyl-5',5',7'-tricyano-2-oxo-5',8a'-dihydro-1'H-spiro[indoline-3,8'-isoquinoline]-2'(3'H)-carboxylate1086Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56388CB1UNDEFINEDHUMANUNDEFINEDN-benzhydryl-6-(2,6-dimethylmorpholino)-5-nitropyrimidin-4-amine1177Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56389CB1UNDEFINEDHUMANUNDEFINED3-(benzo[d][1,3]dioxol-5-yl)-N-(2-(2,3-dihydrobenzo[b][1,4]dioxin-6-ylamino)-2-oxo-1-p-tolylethyl)-N-methylacrylamide1473Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56390CB1UNDEFINEDHUMANUNDEFINEDmethyl 4-(4-(9H-fluoren-9-yl)piperazin-1-ylsulfonyl)-2,5-dimethylfuran-3-carboxylate1606Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56391CB1UNDEFINEDHUMANUNDEFINEDN-(2,6-diisopropylphenyl)-4-(3-(4-methylbenzyl)-1,2,4-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide1764Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56392CB1UNDEFINEDHUMANUNDEFINED1-(4-(3-(2,4-dimethoxyphenyl)-1-m-tolyl-1H-pyrazole-5-carbonyl)piperazin-1-yl)ethanone1943Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56393CB1UNDEFINEDHUMANUNDEFINED2-(5-benzyl-5H-[1,2,4]triazino[5,6-b]indol-3-ylthio)-N-isopropylpropanamide2269Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56394CB1UNDEFINEDHUMANUNDEFINED(3-((2-(4,6-dimorpholino-1,3,5-triazin-2-yl)hydrazono)methyl)-1H-indol-1-yl)(p-tolyl)methanone2299Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56395CB1UNDEFINEDHUMANUNDEFINED1-(4-(2-methoxyphenyl)piperazin-1-yl)-2-(4-phenyl-6-(trifluoromethyl)pyrimidin-2-ylthio)propan-1-one2314Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56396CB1UNDEFINEDHUMANUNDEFINED2-cyclohexyl-3-(4-methoxyphenyl)-N-(6-methylpyridin-2-yl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-4-carboxamide2396Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56397CB1UNDEFINEDHUMANUNDEFINEDN-isopropyl-N-(2-(4-(4-methoxyphenyl)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-2-oxoethyl)cyclohexanecarboxamide2593Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56398CB1UNDEFINEDHUMANUNDEFINED1-benzyl-4-methyl-6-phenyl-3-(phenylsulfonyl)pyridin-2(1H)-one2716Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56399CB1UNDEFINEDHUMANUNDEFINED2-chloro-N-(2,6-dimethylphenyl)-N-(2-morpholino-2-(4-nitrophenyl)acetyl)benzamide2785Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56400CB1UNDEFINEDHUMANUNDEFINED4-(8-benzyl-5-cyano-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridin-6-yl)-N-propylpiperazine-1-carboxamide3949Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56401CB1UNDEFINEDHUMANUNDEFINED3-(4-tert-butylbenzoyl)-2-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)thiazolidine-4-carboxamide7490Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56402CB1UNDEFINEDHUMANUNDEFINEDmethyl N-4-(5-(thiophen-2-yl)-3-(trifluoromethyl)-1H-pyrazol-1-yl)phenylsulfonylpyrrolidine-1-carbimidothioate1000Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56403CB2UNDEFINEDHUMANUNDEFINEDRimonabant1000Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56404CB2UNDEFINEDHUMANUNDEFINEDibipinabant7943Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56405CB2UNDEFINEDHUMANUNDEFINEDTaranabant290Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56406CB2UNDEFINEDHUMANUNDEFINED2-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-methyl-5-(piperidin-1-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-one1300Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56407CB2UNDEFINEDHUMANUNDEFINED1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-morpholinophenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethanone3919Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56408CB2UNDEFINEDHUMANUNDEFINED4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzamide>10000Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56409CB2UNDEFINEDHUMANUNDEFINED2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,3-d]pyrimidin-4-ylthio)-N-(2-methoxyphenyl)propanamide>10000Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56410CB2UNDEFINEDHUMANUNDEFINEDethyl 4-(3-(2-chlorophenyl)-1-(2,4-dimethylphenyl)-1H-pyrazole-5-carbonyl)piperazine-1-carboxylate1069Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56411CB2UNDEFINEDHUMANUNDEFINED3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)pyrrolo[1,2-a]quinoxalin-5(4H)-yl)-2-oxoethyl)urea4953Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56412CB2UNDEFINEDHUMANUNDEFINED2-[2-(2,4,6-Trimethyl-phenoxy)-acetylamino]-4,5,6,7-tetrahydro-benzo[b]thiophene-3-carboxylic acid (1,1-dioxo-tetrahydro-1lambda*6*-thiophen-3-yl)-amide58Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56413CB2UNDEFINEDHUMANUNDEFINEDN-cyclopropyl-N-(2-oxo-2-(4-p-tolylpyrrolo[1,2-a]quinoxalin-5(4H)-yl)ethyl)cyclopentanecarboxamide>10000Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56414CB2UNDEFINEDHUMANUNDEFINEDN-benzhydryl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-2-fluorobenzamide>10000Foloppe N et al., 2009Jan 15, 2025Jan 15, 2025
56415SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride7.47White JD et al., 2009Jan 15, 2025Jan 15, 2025
56416SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1S,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride33.2White JD et al., 2009Jan 15, 2025Jan 15, 2025
56417SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride17.6White JD et al., 2009Jan 15, 2025Jan 15, 2025
56418SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride2.01White JD et al., 2009Jan 15, 2025Jan 15, 2025
56419SLC6A4UNDEFINEDUNDEFINEDUNDEFINED(Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride2.1White JD et al., 2009Jan 15, 2025Jan 15, 2025
56420SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride30.4White JD et al., 2009Jan 15, 2025Jan 15, 2025
56421SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDIMIPRAMINE7.57White JD et al., 2009Jan 15, 2025Jan 15, 2025
56422SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride75.7White JD et al., 2009Jan 15, 2025Jan 15, 2025
56423SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1S,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride153White JD et al., 2009Jan 15, 2025Jan 15, 2025
56424SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride330White JD et al., 2009Jan 15, 2025Jan 15, 2025
56425SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride4.16White JD et al., 2009Jan 15, 2025Jan 15, 2025
56426SLC6A2UNDEFINEDUNDEFINEDUNDEFINED(Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride1.19White JD et al., 2009Jan 15, 2025Jan 15, 2025
56427SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride27.8White JD et al., 2009Jan 15, 2025Jan 15, 2025
56428SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDDESIPRAMINE5.11White JD et al., 2009Jan 15, 2025Jan 15, 2025
56429SLC6A3UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride586White JD et al., 2009Jan 15, 2025Jan 15, 2025
56430SLC6A3UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1S,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride913White JD et al., 2009Jan 15, 2025Jan 15, 2025
56431SLC6A3UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2S)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride790White JD et al., 2009Jan 15, 2025Jan 15, 2025
56432SLC6A3UNDEFINEDUNDEFINEDUNDEFINED(Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride283White JD et al., 2009Jan 15, 2025Jan 15, 2025
56433SLC6A3UNDEFINEDUNDEFINEDUNDEFINED(Z)-N-Methyl-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine Hydrochloride223White JD et al., 2009Jan 15, 2025Jan 15, 2025
56434SLC6A3UNDEFINEDUNDEFINEDUNDEFINEDN-methyl-1-((1R,2R)-2-(naphthalen-1-yloxy)-2-(thiophen-2-yl)cyclopropyl)methanamine hydrochloride1910White JD et al., 2009Jan 15, 2025Jan 15, 2025
56435SLC6A3UNDEFINEDUNDEFINEDUNDEFINED1-{2-[Bis-(4-fluoro-phenyl)-methoxy]-ethyl}-4-(3-phenyl-propyl)-piperazine5.07White JD et al., 2009Jan 15, 2025Jan 15, 2025
56436SLC6A2UNDEFINEDHUMANUNDEFINEDDESIPRAMINE2.1Zhang P et al., 2009Jan 15, 2025Jan 15, 2025
56437SLC6A3UNDEFINEDHUMANUNDEFINEDMAZINDOL22.1Zhang P et al., 2009Jan 15, 2025Jan 15, 2025
56438CB1UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide56Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56439CB1UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-sifluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide840Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56440CB1UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide41Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56441CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide99Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56442CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide54Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56443CB1UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide50Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56444CB1UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide165Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56445CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide56Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56446CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide560Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56447CB1UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide560Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56448CB1UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide2400Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56449CB1UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide380Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56450CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide948Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56451CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide310Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56452CB1UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide80Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56453CB1UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide345Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56454CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide340Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56455CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2100Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56456CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzhydryl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide2820Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56457CB1UNDEFINEDHUMANUNDEFINEDN-[1-(1-Phenyl)ethyl]1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide80Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56458CB1UNDEFINEDHUMANUNDEFINEDN-(Adamant-1-yl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide5.6Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56459CB1UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide12Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56460CB1UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide36Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56461CB1UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide390Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56462CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide100Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56463CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide2820Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56464CB1UNDEFINEDHUMANUNDEFINED(S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3.4Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56465CB1UNDEFINEDHUMANUNDEFINED(R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide14Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56466CB1UNDEFINEDHUMANUNDEFINEDN-(Adamant-1-yl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide31Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56467CB1UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide5.6Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56468CB1UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide50Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56469CB1UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide240Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56470CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide70Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56471CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1300Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56472CB1UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide56Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56473CB1UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide150Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56474CB1UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide156Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56475CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide112Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56476CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide117Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56477CB1UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide30Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56478CB1UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide144Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56479CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide90Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56480CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide96Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56481CB1UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide20Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56482CB1UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide84Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56483CB1UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide218Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56484CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide368Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56485CB1UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide157Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56486CB1UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide70Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56487CB1UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide227Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56488CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide140Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56489CB1UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide120Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56490CB1UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide5.6Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56491CB1UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide28Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56492CB1UNDEFINEDHUMANUNDEFINEDSR 1445282820Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56493CB1UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide2.3Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56494CB1UNDEFINEDHUMANUNDEFINEDRimonabant12Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56495CB2UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide110Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56496CB2UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-sifluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide900Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56497CB2UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide721Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56498CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56499CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56500CB2UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56501CB2UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide373Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56502CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56503CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-difluorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56504CB2UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide200Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56505CB2UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-difluorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide1100Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56506CB2UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide667Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56507CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1945Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56508CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1291Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56509CB2UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56510CB2UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide739Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56511CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3400Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56512CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-difluorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56513CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzhydryl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56514CB2UNDEFINEDHUMANUNDEFINEDN-[1-(1-Phenyl)ethyl]1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide5.7Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56515CB2UNDEFINEDHUMANUNDEFINEDN-(Adamant-1-yl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide12Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56516CB2UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide4.2Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56517CB2UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide12Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56518CB2UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56519CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide790Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56520CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56521CB2UNDEFINEDHUMANUNDEFINED(S)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2.4Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56522CB2UNDEFINEDHUMANUNDEFINED(R)-N-[1-(1-Cyclohexyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1.6Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56523CB2UNDEFINEDHUMANUNDEFINEDN-(Adamant-1-yl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide20Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56524CB2UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide1.3Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56525CB2UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide12Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56526CB2UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1200Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56527CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide100Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56528CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide790Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56529CB2UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide80Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56530CB2UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide310Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56531CB2UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56532CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3483Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56533CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56534CB2UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56535CB2UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide553Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56536CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56537CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56538CB2UNDEFINEDHUMANUNDEFINEDN-Cycloheptyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide20Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56539CB2UNDEFINEDHUMANUNDEFINEDN-Cyclopentyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1Hpyrrol-1-yl)-1H-pyrazole-3-carboxamide170Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56540CB2UNDEFINEDHUMANUNDEFINEDN-[2-(2,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56541CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3-Chloro-4-methoxyphenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide2887Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56542CB2UNDEFINEDHUMANUNDEFINEDN-[2-(3,4-Dichlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56543CB2UNDEFINEDHUMANUNDEFINEDN-[2-(4-Chlorophenyl)ethyl]1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56544CB2UNDEFINEDHUMANUNDEFINEDN-(2-Bromo-3,4,5-trimethoxybenzyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide609Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56545CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorobenzyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56546CB2UNDEFINEDHUMANUNDEFINEDN-(4-Chlorophenyl)1-(2,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide80Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56547CB2UNDEFINEDHUMANUNDEFINEDN-cyclohexyl 1-(3,4-dichlorophenyl)-4-methyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide1.7Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56548CB2UNDEFINEDHUMANUNDEFINEDN-3,4-dichlorobenzyl 1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-1H-pyrazole-3-carboxamide3940Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56549CB2UNDEFINEDHUMANUNDEFINEDSR 1445285.4Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56550CB2UNDEFINEDHUMANUNDEFINED1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide112Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56551CB2UNDEFINEDHUMANUNDEFINEDRimonabant790Silvestri R et al., 2009Jan 15, 2025Jan 15, 2025
56552A1UNDEFINEDUNDEFINEDUNDEFINED(2S,3S,4R,5S)-5-(6-(cyclopentylamino)-9H-purin-8-yl)-3,4-dihydroxy-N-(1-(4-(N-(1-phenethylpiperidin-4-yl)propionamido)phenyl)ethyl)tetrahydrofuran-2-carboxamide800Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56553A1UNDEFINEDUNDEFINEDUNDEFINEDDPCPX12.9Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56554A1UNDEFINEDUNDEFINEDUNDEFINEDNaloxone(-)>10000Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56555A1UNDEFINEDUNDEFINEDUNDEFINEDDAMGO>10000Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56556A2AUNDEFINEDUNDEFINEDUNDEFINED(2S,3S,4R,5S)-5-(6-(cyclopentylamino)-9H-purin-8-yl)-3,4-dihydroxy-N-(1-(4-(N-(1-phenethylpiperidin-4-yl)propionamido)phenyl)ethyl)tetrahydrofuran-2-carboxamide>10000Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56557MORUNDEFINEDUNDEFINEDUNDEFINED(2S,3S,4R,5S)-5-(6-(cyclopentylamino)-9H-purin-8-yl)-3,4-dihydroxy-N-(1-(4-(N-(1-phenethylpiperidin-4-yl)propionamido)phenyl)ethyl)tetrahydrofuran-2-carboxamide728Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56558MORUNDEFINEDUNDEFINEDUNDEFINEDDPCPX>10000Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56559MORUNDEFINEDUNDEFINEDUNDEFINEDNaloxone(-)1.5Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56560MORUNDEFINEDUNDEFINEDUNDEFINEDDAMGO3.8Mathew SC et al., 2009Jan 15, 2025Jan 15, 2025
56561MORUNDEFINEDUNDEFINEDUNDEFINED1'-benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4'-piperidine]201Maestrup EG et al., 2009Jan 15, 2025Jan 15, 2025
56562DORUNDEFINEDUNDEFINEDUNDEFINED1'-benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4'-piperidine]308Maestrup EG et al., 2009Jan 15, 2025Jan 15, 2025
56563KORUNDEFINEDUNDEFINEDUNDEFINED1'-benzyl-3-(3-fluoropropyl)-3H-spiro[[2]benzofuran-1,4'-piperidine]344Maestrup EG et al., 2009Jan 15, 2025Jan 15, 2025
56564MORUNDEFINEDHUMANUNDEFINEDMorphine2.55Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56565MORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol1330Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56566MORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol600Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56567MORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol200Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56568MORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol1330Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56569MORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro-[2,3-c]pyridin-6-ol3500Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56570MORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol80Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56571MORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol9.3Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56572MORUNDEFINEDHUMANUNDEFINED4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol0.7Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56573MORUNDEFINEDHUMANUNDEFINED(4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol15.9Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56574MORUNDEFINEDHUMANUNDEFINED4aS,9aR-(-)-cis-4a-Ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro-[2,3-c]pyridin-6-ol48Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56575DORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol3100Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56576DORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol2490Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56577DORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol2690Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56578DORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol4270Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56579DORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol807Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56580DORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol443Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56581DORUNDEFINEDHUMANUNDEFINED4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol75Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56582DORUNDEFINEDHUMANUNDEFINED(4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol1350Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56583KORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'R-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol9500Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56584KORUNDEFINEDHUMANUNDEFINED4aR,9aS,2'S-(+)-cis-2-(2'-Hydroxy-2'-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol5870Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56585KORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-phenylethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol2325Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56586KORUNDEFINEDHUMANUNDEFINED4aR,9aS-(+)-cis-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol1000Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56587KORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'R-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol1090Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56588KORUNDEFINEDHUMANUNDEFINED4aS,9aR,2'S-(-)-cis-2-(2'-Hydroxy-2-phenylethyl)-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol413Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56589KORUNDEFINEDHUMANUNDEFINED4aS,9aR-(-)-cis-4a-Ethyl-2-(2-phenylethyl)-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ol88Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
56590KORUNDEFINEDHUMANUNDEFINED(4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridin-6-ol450Zhang Y et al., 2009Jan 15, 2025Jan 15, 2025
565915-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-((benzo[d][1,3]dioxol-5-yl)methyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565925-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565935-HT1AUNDEFINEDRATUNDEFINEDethyl 5-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565945-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(2-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565955-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(2-cyanophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565965-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-o-tolylpiperazin-1-yl)propoxy)-1H-indole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565975-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate35.8Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565985-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(4-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate14Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
565995-HT1AUNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(3-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate39Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
566005-HT1AUNDEFINEDRATUNDEFINED8-OH-DPAT0.8Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
56601D1UNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-(3-chlorophenyl)piperazin-1-yl)propoxy)-1Hindole-2-carboxylate1070Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
56602D1UNDEFINEDRATUNDEFINEDEthyl 5-(3-(4-((benzo[d][1,3]dioxol-5-yl)methyl)piperazin-1-yl)propoxy)-1H-indole-2-carboxylate>10000Frecentese F et al., 2010Jan 15, 2025Jan 15, 2025
56603NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol134Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56604NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol1150Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56605NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol7Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56606NR3C1UNDEFINEDHUMANUNDEFINEDBenzo[b]thiophen-3-yl(1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol36Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56607NR3C1UNDEFINEDHUMANUNDEFINED(4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol25Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56608NR3C1UNDEFINEDHUMANUNDEFINED(4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol21Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56609NR3C1UNDEFINEDHUMANUNDEFINED1-(1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo-[1,5-b]isoquinolin-6-yl)but-3-en-1-ol8Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56610NR3C1UNDEFINEDHUMANUNDEFINED1-(1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo-[1,5-b]isoquinolin-6-yl)but-3-en-1-ol9Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56611NR3C1UNDEFINEDHUMANUNDEFINED(1R)-benzo[b]thiophen-3-yl((4aR)-1-(4-fluorophenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl)methanol1.8Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56612NR3C1UNDEFINEDHUMANUNDEFINED(1S)-1-((4aR)-1-(4-fluorophenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl)but-3-en-1-ol3.9Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56613NR3C1UNDEFINEDHUMANUNDEFINEDdexamethasone1.2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56614NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-2-yl)ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56615NR3C1UNDEFINEDHUMANUNDEFINED(5aR,6S)-1-(4-Fluorophenyl)-6-((S)-1-methoxy-1-(thiophen-2-yl)-ethyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinoline33Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56616NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-(4-Fluorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]-isoquinolin-6-yl)ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56617NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-phenylethanol1Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56618NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-o-tolylethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56619NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-m-tolylethanol2.5Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56620NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-(4-Chlorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56621NR3C1UNDEFINEDHUMANUNDEFINED3-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonitrile1Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56622NR3C1UNDEFINEDHUMANUNDEFINED4-((S)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-hydroxyethyl)benzonitrile2.5Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56623NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-2-yl)ethanol31Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56624NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-3-yl)ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56625NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(pyridin-4-yl)ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56626NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(3-methylthiophen-2-yl)-ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56627NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(5-methylthiophen-2-yl)-ethanol1.5Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56628NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-(5-Chlorothiophen-2-yl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-ethanol4Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56629NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-3-yl)ethanol1Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56630NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[,5-b]isoquinolin-6-yl)-1-(thiazol-2-yl)ethanol3Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56631NR3C1UNDEFINEDHUMANUNDEFINED(R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)pent-4-en-2-ol4.3Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56632NR3C1UNDEFINEDHUMANUNDEFINED(R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)hexan-2-ol7.9Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56633NR3C1UNDEFINEDHUMANUNDEFINED(R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-4-phenylbutan-2-ol47Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56634NR3C1UNDEFINEDHUMANUNDEFINED(R)-1-(4-Fluorophenyl)-2-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)propan-2-ol11Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56635NR3C1UNDEFINEDHUMANUNDEFINED(R)-1-Cyclopropyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol2.6Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56636NR3C1UNDEFINEDHUMANUNDEFINED(R)-1-Cyclohexyl-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol3.1Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56637NR3C1UNDEFINEDHUMANUNDEFINED(R)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(tetrahydro-2H-pyran-4-yl)-ethanol2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56638NR3C1UNDEFINEDHUMANUNDEFINED(S)-1,1,1-Trifluoro-2-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)propan-2-ol5.2Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56639NR3C1UNDEFINEDHUMANUNDEFINED(R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-4-methylpentan-2-ol9Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56640NR3C1UNDEFINEDHUMANUNDEFINED1-((S)-4-Fluoro-phenyl)-1-[(4aR,5S)-1-(4-fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-ethanol2.5Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56641NR3C1UNDEFINEDHUMANUNDEFINED(S)-1-[(4aR,5S)-1-(4-Fluoro-phenyl)-4a-methyl-4,4a,5,6,7,8-hexahydro-1H-benzo[f]indazol-5-yl]-1-thiophen-3-yl-ethanol0.8Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56642PGRUNDEFINEDUNDEFINEDUNDEFINED(S)-1-(4-Chlorophenyl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)ethanol238Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56643PGRUNDEFINEDUNDEFINEDUNDEFINED(R)-2-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)pent-4-en-2-ol1810Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56644PGRUNDEFINEDUNDEFINEDUNDEFINED(S)-1-(5-Chlorothiophen-2-yl)-1-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-ethanol409Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56645PGRUNDEFINEDUNDEFINEDUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(3-methylthiophen-2-yl)-ethanol132Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56646PGRUNDEFINEDUNDEFINEDUNDEFINED(S)-1-((5aR,6S)-1-(4-Fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)-1-(thiophen-2-yl)ethanol230Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56647PGRUNDEFINEDUNDEFINEDUNDEFINED(4-fluorophenyl)-((5aR,6S)-1-(4-fluorophenyl)-5a-methyl-5,5a,6,7,8,9-hexahydroimidazo[1,5-b]isoquinolin-6-yl)methanol451Xiao HY et al., 2010Jan 15, 2025Jan 15, 2025
56648CB1UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[3-(dimethylamino)propyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine HCl3.1Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56649CB1UNDEFINEDHUMANUNDEFINED[3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-{[2-(dimethylamino)ethylpiperazin-4-yl]methylene}-4-chlorobenzenesulfonamide9.6Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56650CB1UNDEFINEDHUMANUNDEFINED1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide14Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56651CB1UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(methyl)-piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine19Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56652CB1UNDEFINEDHUMANUNDEFINED3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide25Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56653CB1UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(pyrrolidin-1-yl)butyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine27Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56654CB1UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-(2-hydroxy-2-methylpropyl)-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine43Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56655CB1UNDEFINEDHUMANUNDEFINED4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl][4-(1,2,3,4-tetrahydroacridin-9-ylamino)butylamino]methylene}benzenesulfonamide42Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56656CB1UNDEFINEDHUMANUNDEFINED4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl]-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptylamino]-methylene}benzenesulfonamide54Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56657CB1UNDEFINEDHUMANUNDEFINEDSR 141716A25Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56658CB1UNDEFINEDHUMANUNDEFINED[3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-[4-(1,1-dioxothiomorpholinyl)methylene]-4-chlorobenzenesulfonamide31Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56659CB1UNDEFINEDHUMANUNDEFINEDN-[4-(1,2,3,4-Tetrahydroacridin-9-ylamino)butyl]-2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-1H-imidazole-4-carboxamide48Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56660CB1UNDEFINEDHUMANUNDEFINEDN-[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl]-2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-1H-imidazole-4-carboxamide88Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56661CB1UNDEFINEDHUMANUNDEFINEDTacrine1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56662CB2UNDEFINEDHUMANUNDEFINEDSR 141716A1580Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56663CB2UNDEFINEDHUMANUNDEFINED[3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-[4-(1,1-dioxothiomorpholinyl)methylene]-4-chlorobenzenesulfonamide571Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56664CB2UNDEFINEDHUMANUNDEFINEDTacrine1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56665CB2UNDEFINEDHUMANUNDEFINED3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)-N-methyl-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56666CB2UNDEFINEDHUMANUNDEFINED1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(piperidin-1-yl)-1H-imidazole-4-carboxamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56667CB2UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-(2-hydroxy-2-methylpropyl)-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56668CB2UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[3-(dimethylamino)propyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine HCl1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56669CB2UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(methyl)-piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56670CB2UNDEFINEDHUMANUNDEFINED[3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazol-1-yl]-{[2-(dimethylamino)ethylpiperazin-4-yl]methylene}-4-chlorobenzenesulfonamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56671CB2UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N-[4-(pyrrolidin-1-yl)butyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamidine1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56672CB2UNDEFINEDHUMANUNDEFINED4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl][4-(1,2,3,4-tetrahydroacridin-9-ylamino)butylamino]methylene}benzenesulfonamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56673CB2UNDEFINEDHUMANUNDEFINED4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazolyl]-[7-(1,2,3,4-tetrahydroacridin-9-ylamino)heptylamino]-methylene}benzenesulfonamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56674CB2UNDEFINEDHUMANUNDEFINEDN-[4-(1,2,3,4-Tetrahydroacridin-9-ylamino)butyl]-2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-1H-imidazole-4-carboxamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56675CB2UNDEFINEDHUMANUNDEFINEDN-[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl]-2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-1H-imidazole-4-carboxamide1000Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56676MORUNDEFINEDUNDEFINEDUNDEFINED5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(7-(N-(1-phenethylpiperidin-4-yl)propionamido)heptyl)-1H-pyrazole-3-carboxamide6543Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56677CB1UNDEFINEDUNDEFINEDUNDEFINED5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(7-(N-(1-phenethylpiperidin-4-yl)propionamido)heptyl)-1H-pyrazole-3-carboxamide701Lange JH et al., 2010Jan 15, 2025Jan 15, 2025
56678KORUNDEFINEDHUMANUNDEFINEDNaloxone(-)3Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56679KORUNDEFINEDHUMANUNDEFINED(4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol0.1Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56680KORUNDEFINEDHUMANUNDEFINEDPENTAZOCINE (-)2.2Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56681KORUNDEFINEDHUMANUNDEFINED(-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol15Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56682KORUNDEFINEDHUMANUNDEFINED(+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol14Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56683KORUNDEFINEDHUMANUNDEFINED(-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline41Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56684KORUNDEFINEDHUMANUNDEFINED(4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol699Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56685KORUNDEFINEDHUMANUNDEFINED(-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol565Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56686KORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline1140Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56687KORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline1850Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56688KORUNDEFINEDHUMANUNDEFINED(-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol1240Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56689KORUNDEFINEDHUMANUNDEFINED(-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol1850Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56690KORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline3470Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56691KORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline7230Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56692KORUNDEFINEDHUMANUNDEFINED(+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol6900Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56693KORUNDEFINEDHUMANUNDEFINED(-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56694KORUNDEFINEDHUMANUNDEFINED(-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56695KORUNDEFINEDHUMANUNDEFINED(-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56696MORUNDEFINEDHUMANUNDEFINED(-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol0.3Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56697MORUNDEFINEDHUMANUNDEFINED(4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol0.08Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56698MORUNDEFINEDHUMANUNDEFINEDNaloxone(-)0.98Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56699MORUNDEFINEDHUMANUNDEFINED(+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol0.65Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56700MORUNDEFINEDHUMANUNDEFINEDPENTAZOCINE (-)3.9Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56701MORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline24Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56702MORUNDEFINEDHUMANUNDEFINED(-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol27Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56703MORUNDEFINEDHUMANUNDEFINED(-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline30Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56704MORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline145Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56705MORUNDEFINEDHUMANUNDEFINED(-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol275Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56706MORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline236Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56707MORUNDEFINEDHUMANUNDEFINED(4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol1330Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56708MORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline7610Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56709MORUNDEFINEDHUMANUNDEFINED(-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline8840Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56710MORUNDEFINEDHUMANUNDEFINED(+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol8000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56711MORUNDEFINEDHUMANUNDEFINED(-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56712MORUNDEFINEDHUMANUNDEFINED(-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56713MORUNDEFINEDHUMANUNDEFINED(-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56714DORUNDEFINEDHUMANUNDEFINED(4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol2Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56715DORUNDEFINEDHUMANUNDEFINED(-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol6Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56716DORUNDEFINEDHUMANUNDEFINED(+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol44Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56717DORUNDEFINEDHUMANUNDEFINEDNaloxone(-)51Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56718DORUNDEFINEDHUMANUNDEFINEDPENTAZOCINE (-)49Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56719DORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline490Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56720DORUNDEFINEDHUMANUNDEFINED(-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline544Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56721DORUNDEFINEDHUMANUNDEFINED(-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol1050Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56722DORUNDEFINEDHUMANUNDEFINED(-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1Hbenzo[4,5]furo[3,2-e]isoquinolin-9-ol5000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56723DORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline8390Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56724DORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline9750Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56725DORUNDEFINEDHUMANUNDEFINED(-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56726DORUNDEFINEDHUMANUNDEFINED(-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56727DORUNDEFINEDHUMANUNDEFINED(-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56728DORUNDEFINEDHUMANUNDEFINED(-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinoline>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56729DORUNDEFINEDHUMANUNDEFINED(+)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo-[4,5]furo[3,2-e]isoquinolin-9-ol>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56730DORUNDEFINEDHUMANUNDEFINED(4aR,7aS,12bS)-3-Cyclopropylmethyl-2,3,4,4a,5,6,7,7a-octahydro-1H-8-oxa-3-aza-benzo[d]fluoren-9-ol>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56731DORUNDEFINEDHUMANUNDEFINED(-)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octahydro-1H-benzo[4,5]furo[3,2-e]isoquinolin-9-ol>10000Hsin LW et al., 2010Jan 15, 2025Jan 15, 2025
56732SLC6A3UNDEFINEDHUMANUNDEFINED2-(N,N-Diethylamino)-3'-chloropropiophenone2214Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56733SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-Cyclopentylamino)-3'-chloropropiophenone2200Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56734SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-4'-chloropropiophenone2195Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56735SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-4'-bromopropiophenone1918Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56736SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-4'-bromo-5'-methylpropiophenone1740Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56737SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chlorophenyl-4-cyclohexylbutanophenone1700Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56738SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-Cyclopropylamino)-3-chloropropiophenone1150Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56739SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chloro-4'-methylpropiophenone1150Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56740SLC6A3UNDEFINEDHUMANUNDEFINED2-Piperidino-3'-chloropropiophenone1148Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56741SLC6A3UNDEFINEDHUMANUNDEFINEDBUPROPION871Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56742SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chloroheptanophenone709Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56743SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chlorooctanophenone510Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56744SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3',4'-dichloropropiophenone472Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56745SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chlorobutyrophenone459Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56746SLC6A3UNDEFINEDHUMANUNDEFINED2-(N-tert-Butylamino)-3'-chlorohexanophenone350Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56747SLC6A3UNDEFINEDHUMANUNDEFINED2-(tert-Butylamino)-3',4'-dichlorobutyrophenone278Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025
56748SLC6A3UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester272Carroll FI et al., 2009Jan 15, 2025Jan 15, 2025