87749 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[3â€(dimethylamino)propyl]â€Nâ€(2â€phenylethyl)aniline 55 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87750 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[3â€(dimethylamino)propyl]â€Nâ€(2â€phenylethyl)aniline 623 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87751 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[3â€(dimethylamino)propyl]â€Nâ€(2â€phenylethyl)aniline 4486 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87752 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[3â€(dimethylamino)propyl]â€Nâ€(2â€phenylethyl)aniline 228 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87753 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 58 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87754 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[2â€(dimethylamino)ethyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 5707 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87755 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 31 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87756 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 37 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87757 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 23 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87758 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 25 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87759 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 33 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87760 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 10 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87761 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[2â€(dimethylamino)ethyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 482 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87762 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 70 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87763 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)â€4â€(trifluoromethyl)aniline 809 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87764 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)â€4â€(trifluoromethyl)aniline 5341 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87765 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)â€4â€(trifluoromethyl)aniline 30 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87766 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)â€4â€(trifluoromethyl)aniline 274 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87767 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)â€4â€(trifluoromethyl)aniline 61 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87768 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€4â€methoxyâ€Nâ€(2â€phenylethyl)aniline 234 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87769 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€4â€methoxyâ€Nâ€(2â€phenylethyl)aniline 1147 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87770 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€4â€methoxyâ€Nâ€(2â€phenylethyl)aniline 141 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87771 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€4â€methoxyâ€Nâ€(2â€phenylethyl)aniline 863 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87772 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€3â€methylâ€Nâ€(2â€phenylethyl)aniline 777 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87773 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[2â€(dimethylamino)ethyl]â€3â€methylâ€Nâ€(2â€phenylethyl)aniline 605 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87774 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€3â€methylâ€Nâ€(2â€phenylethyl)aniline 2253 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87775 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€3â€methylâ€Nâ€(2â€phenylethyl)aniline 264 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87776 5-HT6 CLONED HUMAN 3H-LSD Nâ€[3â€(dimethylamino)propyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 38 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87777 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[3â€(dimethylamino)propyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 80 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87778 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[3â€(dimethylamino)propyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 38 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87779 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[3â€(dimethylamino)propyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 8969 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87780 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[3â€(dimethylamino)propyl]â€4â€fluoroâ€Nâ€(2â€phenylethyl)aniline 27 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87781 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€3â€fluoroâ€Nâ€(2â€phenylethyl)aniline 312 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87782 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€3â€fluoroâ€Nâ€(2â€phenylethyl)aniline 748 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87783 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€3â€fluoroâ€Nâ€(2â€phenylethyl)aniline 594 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87784 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€3â€fluoroâ€Nâ€(2â€phenylethyl)aniline 64 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87785 5-HT6 CLONED HUMAN 3H-LSD 2,4â€dichloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 597 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87786 D2 CLONED HUMAN 3H-RACLOPRIDE 2,4â€dichloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 1167 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87787 5-HT7 CLONED HUMAN 3H-5-CT 2,4â€dichloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 387 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87788 5-HT2A CLONED HUMAN 3H-KETANSERIN 2,4â€dichloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 472 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87789 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€3â€methoxyâ€Nâ€(2â€phenylethyl)aniline 721 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87790 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€3â€methoxyâ€Nâ€(2â€phenylethyl)aniline 4512 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87791 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€3â€methoxyâ€Nâ€(2â€phenylethyl)aniline 1738 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87792 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€3â€methoxyâ€Nâ€(2â€phenylethyl)aniline 355 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87793 5-HT6 CLONED HUMAN 3H-LSD Nâ€[3â€(dimethylamino)propyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 83 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87794 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[3â€(dimethylamino)propyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 108 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87795 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[3â€(dimethylamino)propyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 24 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87796 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[3â€(dimethylamino)propyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 2140 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87797 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[3â€(dimethylamino)propyl]â€4â€methylâ€Nâ€(2â€phenylethyl)aniline 204 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87798 5-HT2A CLONED HUMAN 3H-KETANSERIN 4â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 212 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87799 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 5960 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87800 5-HT7 CLONED HUMAN 3H-5-CT 4â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 4 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87801 D2 CLONED HUMAN 3H-RACLOPRIDE 4â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 153 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87802 5-HT6 CLONED HUMAN 3H-LSD 4â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 24 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87803 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€2â€methylâ€Nâ€(2â€phenylethyl)aniline 380 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87804 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€2â€methylâ€Nâ€(2â€phenylethyl)aniline 1040 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87805 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€2â€methylâ€Nâ€(2â€phenylethyl)aniline 348 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87806 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 621 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87807 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 4749 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87808 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 2037 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87809 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 423 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87810 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)naphthalenâ€1â€amine 137 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87811 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€3,4â€difluoroâ€Nâ€(2â€phenylethyl)aniline 21 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87812 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€3,4â€difluoroâ€Nâ€(2â€phenylethyl)aniline 114 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87813 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€3,4â€difluoroâ€Nâ€(2â€phenylethyl)aniline 79 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87814 5-HT2A CLONED HUMAN 3H-KETANSERIN 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 295 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87815 5-HT7 CLONED HUMAN 3H-5-CT 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 19 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87816 D2 CLONED HUMAN 3H-RACLOPRIDE 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 505 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87817 5-HT6 CLONED HUMAN 3H-LSD 4â€bromoâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 90 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87818 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€4â€iodoâ€Nâ€(2â€phenylethyl)aniline 79 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87819 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€4â€iodoâ€Nâ€(2â€phenylethyl)aniline 691 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87820 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€4â€iodoâ€Nâ€(2â€phenylethyl)aniline 10 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87821 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€4â€iodoâ€Nâ€(2â€phenylethyl)aniline 372 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87822 5-HT2A CLONED HUMAN 3H-KETANSERIN Nâ€[2â€(dimethylamino)ethyl]â€2,4â€dimethylâ€Nâ€(2â€phenylethyl)aniline 518 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87823 5-HT7 CLONED HUMAN 3H-5-CT Nâ€[2â€(dimethylamino)ethyl]â€2,4â€dimethylâ€Nâ€(2â€phenylethyl)aniline 597 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87824 D2 CLONED HUMAN 3H-RACLOPRIDE Nâ€[2â€(dimethylamino)ethyl]â€2,4â€dimethylâ€Nâ€(2â€phenylethyl)aniline 1751 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87825 5-HT6 CLONED HUMAN 3H-LSD Nâ€[2â€(dimethylamino)ethyl]â€2,4â€dimethylâ€Nâ€(2â€phenylethyl)aniline 347 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87826 5-HT6 CLONED HUMAN 3H-LSD 3â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 150 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87827 D2 CLONED HUMAN 3H-RACLOPRIDE 3â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 675 Staron J et al 2016 Jan 15, 2025 Jan 28, 2025
87828 5-HT7 CLONED HUMAN 3H-5-CT 3â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 353 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87829 5-HT2A CLONED HUMAN 3H-KETANSERIN 3â€chloroâ€Nâ€[2â€(dimethylamino)ethyl]â€Nâ€(2â€phenylethyl)aniline 311 Staron J et al 2016 Jan 15, 2025 Jan 15, 2025
87830 A2B ?CLONED HUMAN 3H-PSB-603 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1.91 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87831 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione 4.31 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87832 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione 322 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87833 A2A ?CLONED HUMAN 3H-MSX-2 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87834 A1 ?CLONED HUMAN 3H-CCPA 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87835 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87836 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87837 A3 ?CLONED HUMAN 3H-PSB-11 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87838 A2B ?CLONED MOUSE 3H-PSB-603 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 8.34 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87839 A1 ?CLONED MOUSE 3H-CCPA 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1520 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87840 A3 ?CLONED MOUSE 3H-PSB-11 8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87841 A3 ?CLONED MOUSE 3H-PSB-11 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87842 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87843 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 928 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87844 A1 ?CLONED MOUSE 3H-CCPA 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 107 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87845 A2B ?CLONED MOUSE 3H-PSB-603 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.901 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87846 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.148 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87847 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 92.4 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87848 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 77.8 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87849 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.153 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87850 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87851 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87852 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 205 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87853 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1.28 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87854 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.397 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87855 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.244 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87856 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 96.7 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87857 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 12.2 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87858 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione 7.02 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87859 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.894 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87860 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 0.629 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87861 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1.02 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87862 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 0.473 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87863 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.643 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87864 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.644 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87865 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.632 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87866 A2B ?CLONED MOUSE 3H-PSB-603 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.926 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87867 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 6.08 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87868 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 4.3 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87869 A2B ?CLONED HUMAN 3H-PSB-603 1-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.432 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87870 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.706 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87871 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 0.616 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87872 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 0.159 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87873 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.137 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87874 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.234 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87875 A2B ?CLONED MOUSE 3H-PSB-603 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.131 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87876 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.0835 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87877 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 0.403 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87878 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.342 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87879 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 3.22 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87880 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87881 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 131 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87882 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 189 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87883 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 208 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87884 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1160 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87885 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 241 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87886 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione 314 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87887 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 122 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87888 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 108 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87889 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87890 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87891 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 204 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87892 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87893 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87894 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 89.5 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87895 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 2990 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87896 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 197 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87897 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87898 A2A ?CLONED HUMAN 3H-MSX-2 1-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 140 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87899 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 96.7 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87900 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 168 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87901 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87902 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 40.7 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87903 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 93.8 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87904 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 35.3 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87905 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87906 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87907 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 403 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87908 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 160 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87909 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 135 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87910 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 245 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87911 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 140 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87912 A2A ?CLONED HUMAN 3H-MSX-2 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide 52.7 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87913 A2A ?CLONED HUMAN 3H-MSX-2 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide 357 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87914 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 293 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87915 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 143 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87916 A2A ?CLONED HUMAN 3H-MSX-2 8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87917 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 8.34 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87918 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 5.69 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87919 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 7.15 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87920 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1.91 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87921 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.421 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87922 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 3.55 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87923 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.215 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87924 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 0.352 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87925 A2B ?CLONED HUMAN 3H-PSB-603 8-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1.24 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87926 A1 ?CLONED HUMAN 3H-CCPA 8-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87927 A1 ?CLONED HUMAN 3H-CCPA 8-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87928 A1 ?CLONED HUMAN 3H-CCPA 8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 535 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87929 A1 ?CLONED HUMAN 3H-CCPA 8-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87930 A1 ?CLONED HUMAN 3H-CCPA 8-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 113 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87931 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87932 A1 ?CLONED HUMAN 3H-CCPA 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide 190 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87933 A1 ?CLONED HUMAN 3H-CCPA 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide 1036 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87934 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 334 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87935 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 364 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87936 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87937 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87938 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87939 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 795 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87940 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 492 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87941 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87942 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 560 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87943 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione 1010 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87944 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 364 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87945 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87946 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87947 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87948 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87949 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87950 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87951 A1 ?CLONED MOUSE 3H-CCPA 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87952 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87953 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87954 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87955 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87956 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87957 A1 ?CLONED ? HUMAN 3H-CCPA 1-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 419 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87958 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 356 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87959 A1 ?CLONED MOUSE 3H-CCPA 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 300 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87960 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87961 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87962 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87963 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87964 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87965 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87966 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87967 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87968 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87969 A3 ?CLONED HUMAN 3H-PSB-11 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide 1220 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87970 A3 ?CLONED HUMAN 3H-PSB-11 4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87971 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87972 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87973 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87974 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87975 A3 ?CLONED HUMAN 3H-PSB-11 1-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87976 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87977 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87978 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87979 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87980 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87981 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87982 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87983 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 53.5 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87984 A3 ?CLONED MOUSE 3H-PSB-11 8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87985 A3 ?CLONED MOUSE 3H-PSB-11 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87986 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87987 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87988 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87989 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87990 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87991 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87992 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87993 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87994 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87995 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87996 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87997 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87998 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
87999 A3 ?CLONED HUMAN 3H-PSB-11 8-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
88000 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
88001 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
88002 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
88003 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 1000 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
88004 A1 ?CLONED HUMAN 3H-CCPA 8-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione 326 Jiang J et al 2019 Jan 15, 2025 Jan 15, 2025
88005 A1 CORTEX RAT 3H-CCPA H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88006 A1 CORTEX RAT 3H-CCPA 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88007 A1 CORTEX RAT 3H-CCPA 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88008 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3870 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88009 A1 CORTEX RAT 3H-CCPA 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4320 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88010 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3160 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88011 A1 CORTEX RAT 3H-CCPA 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2870 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88012 A1 CORTEX RAT 3H-CCPA 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88013 A1 CORTEX RAT 3H-CCPA 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2690 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88014 A1 CORTEX RAT 3H-CCPA 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88015 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88016 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88017 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88018 A1 CORTEX RAT 3H-CCPA 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88019 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 7690 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88020 A1 CORTEX RAT 3H-CCPA 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88021 A1 CORTEX RAT 3H-CCPA 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4400 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88022 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88023 A1 CORTEX RAT 3H-CCPA compound 25 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88024 A1 CORTEX RAT 3H-CCPA 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 2240 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88025 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1240 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88026 A1 CORTEX RAT 3H-CCPA 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1530 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88027 A1 CORTEX RAT 3H-CCPA 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88028 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88029 A1 CORTEX RAT 3H-CCPA 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1330 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88030 A1 CORTEX RAT 3H-CCPA 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1880 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88031 A1 CORTEX RAT 3H-CCPA compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88032 A1 CORTEX RAT 3H-CCPA 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione 1120 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88033 A1 CORTEX RAT 3H-CCPA 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 280 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88034 A1 CORTEX RAT 3H-CCPA caffeine >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88035 A1 CORTEX RAT 3H-CCPA Preladenant (SCH420814) 68.7 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88036 A1 CORTEX RAT 3H-CCPA PSB-36 0.368 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88037 A2A CORTEX RAT 3H-MSX-2 H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 5220 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88038 A2A CORTEX RAT 3H-MSX-2 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4300 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88039 A2A CORTEX RAT 3H-MSX-2 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2650 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88040 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1290 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88041 A2A CORTEX RAT 3H-MSX-2 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1750 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88042 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3060 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88043 A2A CORTEX RAT 3H-MSX-2 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 820 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88044 A2A CORTEX RAT 3H-MSX-2 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4950 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88045 A2A CORTEX RAT 3H-MSX-2 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 870 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88046 A2A CORTEX RAT 3H-MSX-2 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4640 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88047 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 8870 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88048 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 5370 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88049 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88050 A2A CORTEX RAT 3H-MSX-2 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2380 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88051 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2030 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88052 A2A CORTEX RAT 3H-MSX-2 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88053 A2A CORTEX RAT 3H-MSX-2 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2620 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88054 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 7400 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88055 A2A CORTEX RAT 3H-MSX-2 compound 25 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88056 A2A CORTEX RAT 3H-MSX-2 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1730 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88057 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 850 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88058 A2A CORTEX RAT 3H-MSX-2 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 280 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88059 A2A CORTEX RAT 3H-MSX-2 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) 3820 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88060 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 3510 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88061 A2A CORTEX RAT 3H-MSX-2 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 2270 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88062 A2A CORTEX RAT 3H-MSX-2 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 2260 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88063 A2A CORTEX RAT 3H-MSX-2 compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88064 A2A CORTEX RAT 3H-MSX-2 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione 3800 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88065 A2A CORTEX RAT 3H-MSX-2 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 300 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88066 A2A CORTEX RAT 3H-MSX-2 caffeine >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88067 A2A CORTEX RAT 3H-MSX-2 Preladenant (SCH420814) 0.661 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88068 A2A CORTEX RAT 3H-MSX-2 PSB-36 371 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88069 A1 CLONED HUMAN 3H-CCPA H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88070 A1 CLONED HUMAN 3H-CCPA 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88071 A1 CLONED HUMAN 3H-CCPA 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88072 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88073 A1 CLONED HUMAN 3H-CCPA 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88074 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88075 A1 CLONED HUMAN 3H-CCPA 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3800 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88076 A1 CLONED HUMAN 3H-CCPA 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88077 A1 CLONED HUMAN 3H-CCPA 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1910 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88078 A1 CLONED HUMAN 3H-CCPA 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88079 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88080 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88081 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88082 A1 CLONED HUMAN 3H-CCPA 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88083 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88084 A1 CLONED HUMAN 3H-CCPA 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88085 A1 CLONED HUMAN 3H-CCPA 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88086 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88087 A1 CLONED HUMAN 3H-CCPA compound 25 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88088 A1 CLONED HUMAN 3H-CCPA 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88089 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 2470 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88090 A1 CLONED HUMAN 3H-CCPA 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 4130 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88091 A1 CLONED HUMAN 3H-CCPA 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88092 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88093 A1 CLONED HUMAN 3H-CCPA 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88094 A1 CLONED HUMAN 3H-CCPA 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88095 A1 CLONED HUMAN 3H-CCPA compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88096 A1 CLONED HUMAN 3H-CCPA 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88097 A1 CLONED HUMAN 3H-CCPA 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 600 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88098 A1 CLONED HUMAN 3H-CCPA Preladenant (SCH420814) 295 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88099 A1 CLONED HUMAN 3H-CCPA PSB-36 3.97 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88100 A2A CLONED HUMAN 3H-MSX-2 H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88101 A2A CLONED HUMAN 3H-MSX-2 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88102 A2A CLONED HUMAN 3H-MSX-2 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88103 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88104 A2A CLONED HUMAN 3H-MSX-2 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88105 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88106 A2A CLONED HUMAN 3H-MSX-2 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2070 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88107 A2A CLONED HUMAN 3H-MSX-2 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88108 A2A CLONED HUMAN 3H-MSX-2 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 930 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88109 A2A CLONED HUMAN 3H-MSX-2 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88110 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88111 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88112 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88113 A2A CLONED HUMAN 3H-MSX-2 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88114 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88115 A2A CLONED HUMAN 3H-MSX-2 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88116 A2A CLONED HUMAN 3H-MSX-2 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88117 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88118 A2A CLONED HUMAN 3H-MSX-2 compound 25 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88119 A2A CLONED HUMAN 3H-MSX-2 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88120 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1690 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88121 A2A CLONED HUMAN 3H-MSX-2 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione 1100 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88122 A2A CLONED HUMAN 3H-MSX-2 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88123 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88124 A2A CLONED HUMAN 3H-MSX-2 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88125 A2A CLONED HUMAN 3H-MSX-2 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88126 A2A CLONED HUMAN 3H-MSX-2 compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88127 A2A CLONED HUMAN 3H-MSX-2 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88128 A2A CLONED HUMAN 3H-MSX-2 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1390 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88129 A2A CLONED HUMAN 3H-MSX-2 Preladenant (SCH420814) 0.884 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88130 A2A CLONED HUMAN 3H-MSX-2 PSB-36 332 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88131 A2B CLONED HUMAN 3H-PSB-603 H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88132 A2B CLONED HUMAN 3H-PSB-603 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88133 A2B CLONED HUMAN 3H-PSB-603 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88134 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88135 A2B CLONED HUMAN 3H-PSB-603 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88136 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88137 A2B CLONED HUMAN 3H-PSB-603 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88138 A2B CLONED HUMAN 3H-PSB-603 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88139 A2B CLONED HUMAN 3H-PSB-603 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88140 A2B CLONED HUMAN 3H-PSB-603 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88141 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88142 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88143 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88144 A2B CLONED HUMAN 3H-PSB-603 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88145 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88146 A2B CLONED HUMAN 3H-PSB-603 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88147 A2B CLONED HUMAN 3H-PSB-603 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88148 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88149 A2B CLONED HUMAN 3H-PSB-603 compound 25 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88150 A2B CLONED HUMAN 3H-PSB-603 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88151 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88152 A2B CLONED HUMAN 3H-PSB-603 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88153 A2B CLONED HUMAN 3H-PSB-603 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88154 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88155 A2B CLONED HUMAN 3H-PSB-603 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88156 A2B CLONED HUMAN 3H-PSB-603 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88157 A2B CLONED HUMAN 3H-PSB-603 compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88158 A2B CLONED HUMAN 3H-PSB-603 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88159 A3 CLONED HUMAN 3H-PSB-603 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1320 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88160 A2B CLONED HUMAN 3H-PSB-603 Preladenant (SCH420814) 1000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88161 A2B CLONED HUMAN 3H-PSB-603 PSB-36 48.6 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88162 A3 CLONED HUMAN 3H-PSB-11 H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88163 A3 CLONED HUMAN 3H-PSB-11 1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88164 A3 CLONED HUMAN 3H-PSB-11 9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88165 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88166 A3 CLONED HUMAN 3H-PSB-11 9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88167 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88168 A3 CLONED HUMAN 3H-PSB-11 9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88169 A3 CLONED HUMAN 3H-PSB-11 9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88170 A3 CLONED HUMAN 3H-PSB-11 9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88171 A3 CLONED HUMAN 3H-PSB-11 9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88172 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88173 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88174 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88175 A3 CLONED HUMAN 3H-PSB-11 9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88176 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2570 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88177 A3 CLONED HUMAN 3H-PSB-11 9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88178 A3 CLONED HUMAN 3H-PSB-11 9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88179 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88180 A3 CLONED HUMAN 3H-PSB-11 compound 25 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88181 A3 CLONED HUMAN 3H-PSB-11 10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88182 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88183 A3 CLONED HUMAN 3H-PSB-11 10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88184 A3 CLONED HUMAN 3H-PSB-11 10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione) >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88185 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88186 A3 CLONED HUMAN 3H-PSB-11 1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88187 A3 CLONED HUMAN 3H-PSB-11 10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88188 A3 CLONED HUMAN 3H-PSB-11 compound 33 >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88189 A3 CLONED HUMAN 3H-PSB-11 8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione >10000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88190 A3 CLONED HUMAN 3H-PSB-11 9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 660 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88191 A3 CLONED HUMAN 3H-PSB-11 Preladenant (SCH420814) 1000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88192 A3 CLONED HUMAN 3H-PSB-11 PSB-36 1000 Drabczynska A et al 2013 Jan 15, 2025 Jan 15, 2025
88193 A1 ?CLONED ? HUMAN 3H-CCPA 8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 396 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88194 A1 ?CLONED ? HUMAN 3H-CCPA 8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88195 A1 ?CLONED ? HUMAN 3H-CCPA 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88196 A1 ?CLONED ? HUMAN 3H-CCPA 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88197 A1 ?CLONED ? HUMAN 3H-CCPA 8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88198 A1 ?CLONED ? HUMAN 3H-CCPA 8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88199 A1 BRAIN CORTEX RAT 3H-CCPA 9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1780 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88200 A1 BRAIN CORTEX RAT 3H-CCPA 9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88201 A1 BRAIN CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88202 A1 BRAIN CORTEX RAT 3H-CCPA 9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88203 A1 BRAIN CORTEX RAT 3H-CCPA 9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4360 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88204 A1 BRAIN CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88205 A1 BRAIN CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2650 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88206 A1 BRAIN CORTEX RAT 3H-CCPA 9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 486 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88207 A1 BRAIN CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88208 A1 BRAIN CORTEX RAT 3H-CCPA 9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88209 A1 BRAIN CORTEX RAT 3H-CCPA 9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4900 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88210 A1 BRAIN CORTEX RAT 3H-CCPA 9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 4130 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88211 A1 BRAIN CORTEX RAT 3H-CCPA 9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 965 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88212 A1 BRAIN CORTEX RAT 3H-CCPA 9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88213 A1 BRAIN CORTEX RAT 3H-CCPA 9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2320 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88214 A1 BRAIN CORTEX RAT 3H-CCPA 9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 927 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88215 A1 BRAIN CORTEX RAT 3H-CCPA 9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 931 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88216 A1 BRAIN CORTEX RAT 3H-CCPA 9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88217 A1 BRAIN CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1410 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88218 A1 BRAIN CORTEX RAT 3H-CCPA 1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1910 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88219 A1 BRAIN CORTEX RAT 3H-CCPA 9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1550 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88220 A1 BRAIN CORTEX RAT 3H-CCPA 9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3020 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88221 A1 ?CLONED ? HUMAN 3H-CCPA 10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88222 A1 ?CLONED ? HUMAN 3H-CCPA 10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88223 A1 ?CLONED ? HUMAN 3H-CCPA 10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 651 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88224 A1 ?CLONED ? HUMAN 3H-CCPA 10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88225 A1 ?CLONED ? HUMAN 3H-CCPA 10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88226 A1 ?CLONED ? HUMAN 3H-CCPA 10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88227 A1 ?CLONED ? HUMAN 3H-CCPA 10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88228 A1 ?CLONED ? HUMAN 3H-CCPA 10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88229 A1 ?CLONED ? HUMAN 3H-CCPA 10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88230 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88231 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1580 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88232 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 959 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88233 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88234 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 767 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88235 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88236 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88237 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1080 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88238 A2A ?CLONED ? HUMAN 3H-MSX-2 10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 881 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88239 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88240 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 189 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88241 A2A ?CLONED ? HUMAN 3H-MSX-2 1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88242 A2A ?CLONED ? HUMAN 3H-MSX-2 1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1020 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88243 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88244 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88245 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 627 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88246 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88247 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1610 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88248 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1700 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88249 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88250 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 8910 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88251 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 8000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88252 A2A ?CLONED ? HUMAN 3H-MSX-2 1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88253 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88254 A2A ?CLONED ? HUMAN 3H-MSX-2 1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 2020 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88255 A2A ?CLONED ? HUMAN 3H-MSX-2 1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88256 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88257 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 8270 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88258 A2A ?CLONED ? HUMAN 3H-MSX-2 1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 3040 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88259 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88260 A2A ?CLONED ? HUMAN 3H-MSX-2 9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1210 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88261 A2A ?CLONED ? HUMAN 3H-MSX-2 8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione 784 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88262 A2A ?CLONED ? HUMAN 3H-MSX-2 8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88263 A2A ?CLONED ? HUMAN 3H-MSX-2 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88264 A2A ?CLONED ? HUMAN 3H-MSX-2 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione ( 887 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88265 A2A ?CLONED ? HUMAN 3H-MSX-2 8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 369 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88266 A2A ?CLONED ? HUMAN 3H-MSX-2 8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88267 A2A ?CLONED ? HUMAN 3H-MSX-2 caffeine >10000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88268 A2B ?CLONED ? HUMAN [ 3 H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) caffeine >10000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88269 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88270 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88271 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88272 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88273 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88274 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88275 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88276 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88277 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88278 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88279 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88280 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88281 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88282 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88283 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88284 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88285 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88286 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88287 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88288 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88289 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88290 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88291 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88292 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88293 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88294 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88295 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88296 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88297 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88298 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88299 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88300 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88301 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88302 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88303 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88304 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88305 A2B ?CLONED ? HUMAN [ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603) 10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88306 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88307 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88308 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88309 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88310 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88311 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88312 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88313 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88314 A3 ?CLONED ? HUMAN 3H-PSB-11 10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88315 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88316 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88317 A3 ?CLONED ? HUMAN 3H-PSB-11 1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88318 A3 ?CLONED ? HUMAN 3H-PSB-11 1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88319 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88320 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88321 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88322 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88323 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88324 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88325 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88326 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88327 A3 ?CLONED ? HUMAN 3H-PSB-11 1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88328 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88329 A3 ?CLONED ? HUMAN 3H-PSB-11 1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88330 A3 ?CLONED ? HUMAN 3H-PSB-11 1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88331 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88332 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88333 A3 ?CLONED ? HUMAN 3H-PSB-11 1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88334 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88335 A3 ?CLONED ? HUMAN 3H-PSB-11 9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88336 A3 ?CLONED ? HUMAN 3H-PSB-11 8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88337 A3 ?CLONED ? HUMAN 3H-PSB-11 8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88338 A3 ?CLONED ? HUMAN 3H-PSB-11 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88339 A3 ?CLONED ? HUMAN 3H-PSB-11 8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88340 A3 ?CLONED ? HUMAN 3H-PSB-11 8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88341 A3 ?CLONED ? HUMAN 3H-PSB-11 8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione 1000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88342 A3 ?CLONED ? HUMAN 3H-PSB-11 caffeine >10000 Zaluski M et al 2019 Jan 15, 2025 Jan 15, 2025
88343 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(2-((6-Methyl2-phenylpyrimidin-4-yl)oxy)ethyl)morpholine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 15, 2025
88344 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(2-((6-Methyl2-phenylpyrimidin-4-yl)oxy)ethyl)morpholine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88345 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)morpholine 949 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88346 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)morpholine 36.3 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88347 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)butyl)morpholine 95.2 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88348 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)butyl)morpholine 1072 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88349 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(5-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)pentyl)morpholine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88350 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(5-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)pentyl)morpholine 389 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88351 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(6-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)hexyl)morpholine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88352 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(6-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)hexyl)morpholine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88353 Sigma 2 BRAIN GUINEA PIG 3H-DTG (E)-4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)but-2-en-1-yl)- morpholine 1451 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88354 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (E)-4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)but-2-en-1-yl)- morpholine 116 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88355 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(2-(2-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)ethoxy)ethyl)- morpholine 422 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88356 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(2-(2-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)ethoxy)ethyl)- morpholine 1924 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88357 Sigma 2 BRAIN GUINEA PIG 3H-DTG 1-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-3-morpholinopropan2-ol 1644 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88358 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 1-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-3-morpholinopropan2-ol 486 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88359 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 1051 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88360 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 11.8 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88361 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-6-(3-(4-methylpiperidin-1-yl)propoxy)-2-phenylpyrimidine 16.7 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88362 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-6-(3-(4-methylpiperidin-1-yl)propoxy)-2-phenylpyrimidine 1416 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88363 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(3-(3,5-Dimethylpiperidin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 1662 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88364 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(3-(3,5-Dimethylpiperidin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 30.2 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88365 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-2-phenyl-6-(3-(2,2,6,6-tetramethylpiperidin-1-yl)- propoxy)pyrimidine 377 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88366 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-2-phenyl-6-(3-(2,2,6,6-tetramethylpiperidin-1-yl)- propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88367 Sigma 2 BRAIN GUINEA PIG 3H-DTG 1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4-ol 1763 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88368 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4-ol 462 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88369 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4- one 319 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88370 Sigma 2 BRAIN GUINEA PIG 3H-DTG 1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4- one 1492 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88371 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-2-phenyl-6-(3-(piperazin-1-yl)propoxy)pyrimidine 1212 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88372 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-2-phenyl-6-(3-(piperazin-1-yl)propoxy)pyrimidine 151 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88373 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-6-(3-(4-methylpiperazin-1-yl)propoxy)-2-phenylpyrimidine 22.7 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88374 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-6-(3-(4-methylpiperazin-1-yl)propoxy)-2-phenylpyrimidine 1325 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88375 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(3-(4-Ethylpiperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 1179 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88376 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(3-(4-Ethylpiperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 30.6 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88377 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 1-Methyl-4-(3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propyl)-1,4- diazepane 18.7 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88378 Sigma 2 BRAIN GUINEA PIG 3H-DTG 1-Methyl-4-(3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propyl)-1,4- diazepane 1295 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88379 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-(3-(4-Boc-piperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88380 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-(3-(4-Boc-piperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88381 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-2-phenyl-6-(3-(4-phenylpiperazin-1-yl)propoxy)- pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88382 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-2-phenyl-6-(3-(4-phenylpiperazin-1-yl)propoxy)- pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88383 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 1253 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88384 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 13.6 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88385 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N,N-Dimethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan1-amine 82.3 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88386 Sigma 2 BRAIN GUINEA PIG 3H-DTG N,N-Dimethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan1-amine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88387 Sigma 2 BRAIN GUINEA PIG 3H-DTG N,N-Diethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan-1- amine 1317 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88388 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N,N-Diethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan-1- amine 47.1 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88389 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-N,N-dipropylpropan-1- amine 38.8 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88390 Sigma 2 BRAIN GUINEA PIG 3H-DTG 3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-N,N-dipropylpropan-1- amine 1069 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88391 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Ethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 20.5 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88392 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Ethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 1141 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88393 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-propylpyrimidine 1456 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88394 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-propylpyrimidine 34.9 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88395 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Isopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 188 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88396 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Isopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 1836 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88397 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methoxy-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 892 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88398 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methoxy-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 19.3 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88399 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-(trifluoromethyl)- pyrimidine 27.6 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88400 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-(trifluoromethyl)- pyrimidine 1327 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88401 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Cyclopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88402 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Cyclopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 253 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88403 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2,4-Diphenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 966 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88404 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2,4-Diphenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88405 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4,5-Dimethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 1221 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88406 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4,5-Dimethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 9.51 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88407 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Fluoro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 3.75 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88408 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Fluoro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 1361 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88409 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 1649 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88410 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine 2.33 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88411 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Ethyl-2-phenyl6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 1429 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88412 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Ethyl-2-phenyl6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 22.4 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88413 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-propylpyrimidine 38.9 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88414 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-propylpyrimidine 1396 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88415 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Isopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 1092 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88416 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Isopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 218 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88417 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Methoxy-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 19.3 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88418 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Methoxy-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 892 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88419 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-(trifluoromethyl)-pyrimidine 1327 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88420 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-(trifluoromethyl)-pyrimidine 27.6 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88421 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-Cyclopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 278 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88422 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4-Cyclopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88423 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2,4-Diphenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88424 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2,4-Diphenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 735 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88425 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4,5-Dimethyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 11.4 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88426 Sigma 2 BRAIN GUINEA PIG 3H-DTG 4,5-Dimethyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine 1279 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88427 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Fluoro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine 1194 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88428 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Fluoro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine 3.51 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88429 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine 4.02 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88430 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine 1684 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88431 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine 1626 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88432 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine 44.2 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88433 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine 58.9 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88434 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine 1896 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88435 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88436 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline 138.5 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88437 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline 111.8 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88438 Sigma 2 BRAIN GUINEA PIG 3H-DTG 2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline 1916 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88439 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(p-tolyl)-pyrimidine 1554 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88440 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(p-tolyl)-pyrimidine 1.96 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88441 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2-(4-methoxyphenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine 3.88 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88442 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2-(4-methoxyphenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine 1288 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88443 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(4- (trifluoromethyl)phenyl)pyrimidine 1776 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88444 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(4- (trifluoromethyl)phenyl)pyrimidine 4.42 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88445 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2-(4-fluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 1.14 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88446 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2-(4-fluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 1329 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88447 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2-(3,4-difluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 943 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88448 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2-(3,4-difluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 0.97 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88449 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2-(4-chlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 1.06 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88450 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2-(4-chlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 1425 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88451 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2-(3,4-dichlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88452 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2-(3,4-dichlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine 89.8 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88453 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-2-(naphthalen-2-yl)-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 102 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88454 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-4-methyl-2-(naphthalen-2-yl)-6-(3-(piperidin-1-yl)-propoxy)pyrimidine 2000 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88455 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 1104 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88456 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 187 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88457 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2,4-dimethyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 58.8 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88458 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2,4-dimethyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine 1081 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88459 Sigma 2 BRAIN GUINEA PIG 3H-DTG 5-Chloro-2-cyclopropyl-4-methyl-6-(3-(piperidin-1-yl)propoxy)-pyrimidine 1328 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88460 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Chloro-2-cyclopropyl-4-methyl-6-(3-(piperidin-1-yl)propoxy)-pyrimidine 39.5 Lan Y et al 2014 Jan 15, 2025 Jan 28, 2025
88461 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 24 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88462 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 666 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88463 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88464 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 658 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88465 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 302 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88466 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88467 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 8.8 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88468 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 49 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88469 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 247.8 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88470 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 317 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88471 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 72 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88472 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88473 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 5.3 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88474 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 182 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88475 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 2.4 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88476 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 74 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88477 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol 93 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88478 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88479 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride 185 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88480 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride 130 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88481 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride 39 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88482 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride 454 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88483 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride 112 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88484 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88485 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine 41 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88486 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine 696 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88487 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine 9.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88488 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine 169 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88489 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine 121 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88490 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88491 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl 998 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88492 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl 243 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88493 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl 35 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88494 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl 613 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88495 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl 222 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88496 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88497 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine 284 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88498 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine 261 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88499 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine 7.8 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88500 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine 112 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88501 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine 81 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88502 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88503 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine 211 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88504 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine 422 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88505 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine 8.7 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88506 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine 166 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88507 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine 53 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88508 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88509 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl 4753 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88510 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl 544 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88511 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl 89 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88512 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl 1080 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88513 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl 1129 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88514 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88515 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine 390 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88516 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine 885 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88517 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine 6.9 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88518 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine 80 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88519 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine 60 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88520 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88521 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 37 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88522 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 207 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88523 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 7.4 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88524 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 24 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88525 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 57.6 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88526 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88527 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl 447 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88528 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl 726 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88529 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl 5.6 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88530 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl 154 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88531 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl 19.8 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88532 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88533 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(3-Phenoxypropyl)-4-phenylpiperazine 119 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88534 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(3-Phenoxypropyl)-4-phenylpiperazine 79.3 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88535 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(3-Phenoxypropyl)-4-phenylpiperazine 4.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88536 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(3-Phenoxypropyl)-4-phenylpiperazine 25 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88537 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(3-Phenoxypropyl)-4-phenylpiperazine 46 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88538 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-Phenoxypropyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88539 D2 CLONED HUMAN 3H-N-Methylspiperone (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine 269 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88540 D3 CLONED HUMAN 3H-N-Methylspiperone (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine 262 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88541 D4 CLONED HUMAN 3H-N-Methylspiperone (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine 6.2 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88542 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine 8.6 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88543 5-HT2A CLONED HUMAN 3H-KETANSERIN (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine 41 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88544 5-HT2C CLONED HUMAN 3H-MESULERGINE (4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88545 D2 CLONED HUMAN 3H-N-Methylspiperone 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 424 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88546 D3 CLONED HUMAN 3H-N-Methylspiperone 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 68 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88547 D4 CLONED HUMAN 3H-N-Methylspiperone 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 21 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88548 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 93.1 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88549 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 27 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88550 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine 8829 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88551 D2 CLONED HUMAN 3H-N-Methylspiperone 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine 636 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88552 D3 CLONED HUMAN 3H-N-Methylspiperone 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine 778 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88553 D4 CLONED HUMAN 3H-N-Methylspiperone 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine 4.2 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88554 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine 23 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88555 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine 23 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88556 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88557 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 124 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88558 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 86 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88559 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 3.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88560 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 1.1 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88561 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 50 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88562 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88563 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 183 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88564 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 160 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88565 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 5.7 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88566 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 6.2 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88567 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 26 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88568 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 8097 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88569 D2 CLONED HUMAN 3H-N-Methylspiperone 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 186 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88570 D3 CLONED HUMAN 3H-N-Methylspiperone 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 229 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88571 D4 CLONED HUMAN 3H-N-Methylspiperone 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 1.8 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88572 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 3.6 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88573 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 18 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88574 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 8277 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88575 H1 CLONED HUMAN 3H-PYRILAMINE 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine 62.9 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88576 M1 CLONED HUMAN 3H-QNB 1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88577 M1 CLONED HUMAN 3H-QNB 1-(3-Phenoxypropyl)-4-phenylpiperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88578 H1 CLONED HUMAN 3H-PYRILAMINE 1-(3-Phenoxypropyl)-4-phenylpiperazine 67.9 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88579 H1 CLONED HUMAN 3H-PYRILAMINE 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 167 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88580 M1 CLONED HUMAN 3H-QNB 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88581 5-HT7 CLONED HUMAN 3H-LSD 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 90 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88582 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine 308.2 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88583 5-HT7 CLONED HUMAN 3H-LSD 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 291 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88584 H1 CLONED HUMAN 3H-PYRILAMINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 212 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88585 M1 CLONED HUMAN 3H-QNB 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88586 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine 45.1 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88587 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 194.5 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88588 5-HT7 CLONED HUMAN 3H-LSD 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 208 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88589 H1 CLONED HUMAN 3H-PYRILAMINE 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine 262 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88590 M1 CLONED HUMAN 3H-QNB 1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine >10000 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88591 D2 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 130 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88592 D4 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 54 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88593 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 140 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88594 5-HT2A CLONED HUMAN 3H-KETANSERIN CLOZAPINE 8.9 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88595 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 17 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88596 H1 CLONED HUMAN 3H-PYRILAMINE CLOZAPINE 1.8 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88597 M1 CLONED HUMAN 3H-QNB CLOZAPINE 1.8 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88598 D2 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 0.89 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88599 D4 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 10 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88600 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88601 5-HT2A CLONED HUMAN 3H-KETANSERIN HALOPERIDOL 120 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88602 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL 4700 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88603 H1 CLONED HUMAN 3H-PYRILAMINE HALOPERIDOL 440 Peprah K et al 2012 Jan 15, 2025 Jan 28, 2025
88604 M1 CLONED HUMAN 3H-QNB HALOPERIDOL 1600 Peprah K et al 2012 Jan 15, 2025 Jan 15, 2025
88605 5-HT1A CLONED HUMAN 3H-8-OH-DPAT HALOPERIDOL 3600 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88606 5-HT2A CLONED HUMAN 3H-KETANSERIN HALOPERIDOL 120 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88607 D1 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 120 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88608 D2 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 0.89 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88609 D3 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 2.5 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88610 D4 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 10 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88611 5-HT2C CLONED HUMAN 3H-MESULERGINE HALOPERIDOL 4700 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88612 H1 CLONED HUMAN 3H-PYRILAMINE HALOPERIDOL 440 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88613 NET CLONED HUMAN 3H-Nisoxetine HALOPERIDOL 5500 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88614 SERT CLONED HUMAN 3H-CITALOPRAM HALOPERIDOL 1800 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88615 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 658 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88616 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 302 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88617 5-HT7 CLONED HUMAN 3H-LSD 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1042 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88618 D1 CLONED HUMAN 3H-SCH23390 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 130 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88619 D5 CLONED HUMAN 3H-SCH23390 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 414 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88620 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 24 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88621 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 668 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88622 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1.5 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88623 5-HT2B CLONED HUMAN 3H-LSD 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 723 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88624 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88625 H1 CLONED HUMAN 3H-PYRILAMINE 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 128.5 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88626 M1 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88627 M2 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88628 M3 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88629 DAT CLONED HUMAN 3H-WIN35428 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88630 NET CLONED HUMAN 3H-Nisoxetine 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1225 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88631 SERT CLONED HUMAN 3H-CITALOPRAM 4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol 1867 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88632 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 317 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88633 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 72 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88634 5-HT7 CLONED HUMAN 3H-LSD 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 656 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88635 D1 CLONED HUMAN 3H-SCH23390 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 22 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88636 D5 CLONED HUMAN 3H-SCH23390 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 103 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88637 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 8.8 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88638 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 49 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88639 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 4.3 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88640 5-HT2B CLONED HUMAN 3H-LSD 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 1622 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88641 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88642 H1 CLONED HUMAN 3H-PYRILAMINE 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 699 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88643 M1 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88644 M2 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88645 M3 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88646 DAT CLONED HUMAN 3H-WIN 35,428 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88647 NET CLONED HUMAN 3H-Nisoxetine 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 3959 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88648 SERT CLONED HUMAN 3H-CITALOPRAM 4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol 2228 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88649 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 74 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88650 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 93 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88651 5-HT7 CLONED HUMAN 3H-LSD 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 1044 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88652 D1 CLONED HUMAN 3H-SCH23390 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 27 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88653 D5 CLONED HUMAN 3H-SCH23390 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 113 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88654 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 5.3 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88655 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 182 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88656 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 2.4 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88657 5-HT2B CLONED HUMAN 3H-LSD 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 790 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88658 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88659 H1 CLONED HUMAN 3H-PYRILAMINE 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 115 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88660 M1 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88661 M2 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88662 M3 CLONED HUMAN 3H-QNB 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88663 DAT CLONED HUMAN 3H-WIN 35,428 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 497 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88664 NET CLONED HUMAN 3H-Nisoxetine 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 2249 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88665 SERT CLONED HUMAN 3H-CITALOPRAM 4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol 160 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88666 D2 CLONED HUMAN 3H-N-Methylspiperone 4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 0.31 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88667 D3 CLONED HUMAN 3H-N-Methylspiperone 4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 0.71 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88668 D4 CLONED HUMAN 3H-N-Methylspiperone 4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 12 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88669 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 872 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88670 H1 CLONED HUMAN 3H-PYRILAMINE 4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one 8780 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88671 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 102 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88672 5-HT2A CLONED HUMAN 3H-KETANSERIN 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 317 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88673 5-HT7 CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 472 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88674 D1 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88675 D5 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88676 D2 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 33 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88677 D3 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 9.7 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88678 D4 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 9.4 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88679 5-HT2B CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 1381 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88680 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 2434 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88681 H1 CLONED HUMAN 3H-PYRILAMINE 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 1719 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88682 M1 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88683 M2 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88684 M3 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88685 DAT CLONED HUMAN 3H-WIN 35,428 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 778 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88686 NET CLONED HUMAN 3H-Nisoxetine 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88687 SERT CLONED HUMAN 3H-CITALOPRAM 3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol 414 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88688 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 123 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88689 5-HT2A CLONED HUMAN 3H-KETANSERIN 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 236 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88690 5-HT7 CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 420 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88691 D1 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88692 D5 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88693 D2 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 22 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88694 D3 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 4.1 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88695 D4 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 49 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88696 5-HT2B CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 898 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88697 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88698 H1 CLONED HUMAN 3H-PYRILAMINE 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 4149 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88699 M1 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88700 M2 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88701 M3 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88702 DAT CLONED HUMAN 3H-WIN 35,428 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 620 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88703 NET CLONED HUMAN 3H-Nisoxetine 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1791 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88704 SERT CLONED HUMAN 3H-CITALOPRAM 3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol 255 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88705 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 20 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88706 5-HT2A CLONED HUMAN 3H-KETANSERIN 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 89 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88707 5-HT7 CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 97 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88708 D1 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 347 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88709 D5 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88710 D2 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 2.9 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88711 D3 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 0.7 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88712 D4 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 8.9 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88713 5-HT2B CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1057 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88714 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1498 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88715 H1 CLONED HUMAN 3H-PYRILAMINE 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 977 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88716 M1 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88717 M2 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88718 M3 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88719 DAT CLONED HUMAN 3H-WIN 35,428 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1081 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88720 NET CLONED HUMAN 3H-Nisoxetine 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1409 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88721 SERT CLONED HUMAN 3H-CITALOPRAM 3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 316 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88722 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 13 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88723 5-HT2A CLONED HUMAN 3H-KETANSERIN 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 509 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88724 5-HT7 CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 917 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88725 D1 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88726 D5 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88727 D2 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 27 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88728 D3 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 11 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88729 D4 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 28 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88730 5-HT2B CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 270 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88731 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1861 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88732 H1 CLONED HUMAN 3H-PYRILAMINE 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1207 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88733 M1 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88734 M2 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88735 M3 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88736 DAT CLONED HUMAN 3H-WIN 35,428 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 285 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88737 NET CLONED HUMAN 3H-Nisoxetine 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 510 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88738 SERT CLONED HUMAN 3H-CITALOPRAM 3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 227 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88739 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 8.2 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88740 5-HT2A CLONED HUMAN 3H-KETANSERIN 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 115 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88741 5-HT7 CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 882 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88742 D1 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 4093 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88743 D5 CLONED HUMAN 3H-SCH23390 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88744 D2 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 4.8 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88745 D3 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1.3 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88746 D4 CLONED HUMAN 3H-N-Methylspiperone 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 27 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88747 5-HT2B CLONED HUMAN 3H-LSD 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 520 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88748 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1122 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025