The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 85,001-86,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
87749D2CLONEDHUMAN3H-RACLOPRIDEN‐[3‐(dimethylamino)propyl]‐N‐(2‐phenylethyl)aniline55Staron J et al 2016Jan 15, 2025Jan 28, 2025
877505-HT7CLONEDHUMAN3H-5-CTN‐[3‐(dimethylamino)propyl]‐N‐(2‐phenylethyl)aniline623Staron J et al 2016Jan 15, 2025Jan 15, 2025
877515-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[3‐(dimethylamino)propyl]‐N‐(2‐phenylethyl)aniline4486Staron J et al 2016Jan 15, 2025Jan 15, 2025
877525-HT2ACLONEDHUMAN3H-KETANSERINN‐[3‐(dimethylamino)propyl]‐N‐(2‐phenylethyl)aniline228Staron J et al 2016Jan 15, 2025Jan 15, 2025
877535-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline58Staron J et al 2016Jan 15, 2025Jan 15, 2025
877545-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(dimethylamino)ethyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline5707Staron J et al 2016Jan 15, 2025Jan 15, 2025
877555-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline31Staron J et al 2016Jan 15, 2025Jan 15, 2025
87756D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline37Staron J et al 2016Jan 15, 2025Jan 28, 2025
877575-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline23Staron J et al 2016Jan 15, 2025Jan 15, 2025
877585-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline25Staron J et al 2016Jan 15, 2025Jan 15, 2025
87759D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline33Staron J et al 2016Jan 15, 2025Jan 28, 2025
877605-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline10Staron J et al 2016Jan 15, 2025Jan 15, 2025
877615-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(dimethylamino)ethyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline482Staron J et al 2016Jan 15, 2025Jan 15, 2025
877625-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline70Staron J et al 2016Jan 15, 2025Jan 15, 2025
877635-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)‐4‐(trifluoromethyl)aniline809Staron J et al 2016Jan 15, 2025Jan 15, 2025
877645-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)‐4‐(trifluoromethyl)aniline5341Staron J et al 2016Jan 15, 2025Jan 15, 2025
877655-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)‐4‐(trifluoromethyl)aniline30Staron J et al 2016Jan 15, 2025Jan 15, 2025
87766D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)‐4‐(trifluoromethyl)aniline274Staron J et al 2016Jan 15, 2025Jan 28, 2025
877675-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)‐4‐(trifluoromethyl)aniline61Staron J et al 2016Jan 15, 2025Jan 15, 2025
877685-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐4‐methoxy‐N‐(2‐phenylethyl)aniline234Staron J et al 2016Jan 15, 2025Jan 15, 2025
87769D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐4‐methoxy‐N‐(2‐phenylethyl)aniline1147Staron J et al 2016Jan 15, 2025Jan 28, 2025
877705-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐4‐methoxy‐N‐(2‐phenylethyl)aniline141Staron J et al 2016Jan 15, 2025Jan 15, 2025
877715-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐4‐methoxy‐N‐(2‐phenylethyl)aniline863Staron J et al 2016Jan 15, 2025Jan 15, 2025
877725-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐3‐methyl‐N‐(2‐phenylethyl)aniline777Staron J et al 2016Jan 15, 2025Jan 15, 2025
877735-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(dimethylamino)ethyl]‐3‐methyl‐N‐(2‐phenylethyl)aniline605Staron J et al 2016Jan 15, 2025Jan 15, 2025
877745-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐3‐methyl‐N‐(2‐phenylethyl)aniline2253Staron J et al 2016Jan 15, 2025Jan 15, 2025
877755-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐3‐methyl‐N‐(2‐phenylethyl)aniline264Staron J et al 2016Jan 15, 2025Jan 15, 2025
877765-HT6CLONEDHUMAN3H-LSDN‐[3‐(dimethylamino)propyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline38Staron J et al 2016Jan 15, 2025Jan 15, 2025
87777D2CLONEDHUMAN3H-RACLOPRIDEN‐[3‐(dimethylamino)propyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline80Staron J et al 2016Jan 15, 2025Jan 28, 2025
877785-HT7CLONEDHUMAN3H-5-CTN‐[3‐(dimethylamino)propyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline38Staron J et al 2016Jan 15, 2025Jan 15, 2025
877795-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[3‐(dimethylamino)propyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline8969Staron J et al 2016Jan 15, 2025Jan 15, 2025
877805-HT2ACLONEDHUMAN3H-KETANSERINN‐[3‐(dimethylamino)propyl]‐4‐fluoro‐N‐(2‐phenylethyl)aniline27Staron J et al 2016Jan 15, 2025Jan 15, 2025
877815-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐3‐fluoro‐N‐(2‐phenylethyl)aniline312Staron J et al 2016Jan 15, 2025Jan 15, 2025
877825-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐3‐fluoro‐N‐(2‐phenylethyl)aniline748Staron J et al 2016Jan 15, 2025Jan 15, 2025
87783D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐3‐fluoro‐N‐(2‐phenylethyl)aniline594Staron J et al 2016Jan 15, 2025Jan 28, 2025
877845-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐3‐fluoro‐N‐(2‐phenylethyl)aniline64Staron J et al 2016Jan 15, 2025Jan 15, 2025
877855-HT6CLONEDHUMAN3H-LSD2,4‐dichloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline597Staron J et al 2016Jan 15, 2025Jan 15, 2025
87786D2CLONEDHUMAN3H-RACLOPRIDE2,4‐dichloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline1167Staron J et al 2016Jan 15, 2025Jan 28, 2025
877875-HT7CLONEDHUMAN3H-5-CT2,4‐dichloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline387Staron J et al 2016Jan 15, 2025Jan 15, 2025
877885-HT2ACLONEDHUMAN3H-KETANSERIN2,4‐dichloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline472Staron J et al 2016Jan 15, 2025Jan 15, 2025
877895-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐3‐methoxy‐N‐(2‐phenylethyl)aniline721Staron J et al 2016Jan 15, 2025Jan 15, 2025
877905-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐3‐methoxy‐N‐(2‐phenylethyl)aniline4512Staron J et al 2016Jan 15, 2025Jan 15, 2025
87791D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐3‐methoxy‐N‐(2‐phenylethyl)aniline1738Staron J et al 2016Jan 15, 2025Jan 28, 2025
877925-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐3‐methoxy‐N‐(2‐phenylethyl)aniline355Staron J et al 2016Jan 15, 2025Jan 15, 2025
877935-HT6CLONEDHUMAN3H-LSDN‐[3‐(dimethylamino)propyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline83Staron J et al 2016Jan 15, 2025Jan 15, 2025
87794D2CLONEDHUMAN3H-RACLOPRIDEN‐[3‐(dimethylamino)propyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline108Staron J et al 2016Jan 15, 2025Jan 28, 2025
877955-HT7CLONEDHUMAN3H-5-CTN‐[3‐(dimethylamino)propyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline24Staron J et al 2016Jan 15, 2025Jan 15, 2025
877965-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[3‐(dimethylamino)propyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline2140Staron J et al 2016Jan 15, 2025Jan 15, 2025
877975-HT2ACLONEDHUMAN3H-KETANSERINN‐[3‐(dimethylamino)propyl]‐4‐methyl‐N‐(2‐phenylethyl)aniline204Staron J et al 2016Jan 15, 2025Jan 15, 2025
877985-HT2ACLONEDHUMAN3H-KETANSERIN4‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline212Staron J et al 2016Jan 15, 2025Jan 15, 2025
877995-HT1ACLONEDHUMAN3H-8-OH-DPAT4‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline5960Staron J et al 2016Jan 15, 2025Jan 15, 2025
878005-HT7CLONEDHUMAN3H-5-CT4‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline4Staron J et al 2016Jan 15, 2025Jan 15, 2025
87801D2CLONEDHUMAN3H-RACLOPRIDE4‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline153Staron J et al 2016Jan 15, 2025Jan 28, 2025
878025-HT6CLONEDHUMAN3H-LSD4‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline24Staron J et al 2016Jan 15, 2025Jan 15, 2025
878035-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐2‐methyl‐N‐(2‐phenylethyl)aniline380Staron J et al 2016Jan 15, 2025Jan 15, 2025
878045-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐2‐methyl‐N‐(2‐phenylethyl)aniline1040Staron J et al 2016Jan 15, 2025Jan 15, 2025
878055-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐2‐methyl‐N‐(2‐phenylethyl)aniline348Staron J et al 2016Jan 15, 2025Jan 15, 2025
878065-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine621Staron J et al 2016Jan 15, 2025Jan 15, 2025
878075-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine4749Staron J et al 2016Jan 15, 2025Jan 15, 2025
878085-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine2037Staron J et al 2016Jan 15, 2025Jan 15, 2025
87809D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine423Staron J et al 2016Jan 15, 2025Jan 28, 2025
878105-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)naphthalen‐1‐amine137Staron J et al 2016Jan 15, 2025Jan 15, 2025
878115-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline21Staron J et al 2016Jan 15, 2025Jan 15, 2025
878125-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline114Staron J et al 2016Jan 15, 2025Jan 15, 2025
878135-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐3,4‐difluoro‐N‐(2‐phenylethyl)aniline79Staron J et al 2016Jan 15, 2025Jan 15, 2025
878145-HT2ACLONEDHUMAN3H-KETANSERIN4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline295Staron J et al 2016Jan 15, 2025Jan 15, 2025
878155-HT7CLONEDHUMAN3H-5-CT4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline19Staron J et al 2016Jan 15, 2025Jan 15, 2025
87816D2CLONEDHUMAN3H-RACLOPRIDE4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline505Staron J et al 2016Jan 15, 2025Jan 28, 2025
878175-HT6CLONEDHUMAN3H-LSD4‐bromo‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline90Staron J et al 2016Jan 15, 2025Jan 15, 2025
878185-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline79Staron J et al 2016Jan 15, 2025Jan 15, 2025
87819D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline691Staron J et al 2016Jan 15, 2025Jan 28, 2025
878205-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline10Staron J et al 2016Jan 15, 2025Jan 15, 2025
878215-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐4‐iodo‐N‐(2‐phenylethyl)aniline372Staron J et al 2016Jan 15, 2025Jan 15, 2025
878225-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline518Staron J et al 2016Jan 15, 2025Jan 15, 2025
878235-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline597Staron J et al 2016Jan 15, 2025Jan 15, 2025
87824D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline1751Staron J et al 2016Jan 15, 2025Jan 28, 2025
878255-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐2,4‐dimethyl‐N‐(2‐phenylethyl)aniline347Staron J et al 2016Jan 15, 2025Jan 15, 2025
878265-HT6CLONEDHUMAN3H-LSD3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline150Staron J et al 2016Jan 15, 2025Jan 15, 2025
87827D2CLONEDHUMAN3H-RACLOPRIDE3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline675Staron J et al 2016Jan 15, 2025Jan 28, 2025
878285-HT7CLONEDHUMAN3H-5-CT3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline353Staron J et al 2016Jan 15, 2025Jan 15, 2025
878295-HT2ACLONEDHUMAN3H-KETANSERIN3‐chloro‐N‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline311Staron J et al 2016Jan 15, 2025Jan 15, 2025
87830A2B?CLONEDHUMAN3H-PSB-6038- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1.91Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87831A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione4.31Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87832A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione322Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87833A2A?CLONEDHUMAN3H-MSX-28- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87834A1?CLONEDHUMAN3H-CCPA8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87835A1?CLONEDHUMAN3H-CCPA8-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87836A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-ethyl1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87837A3?CLONEDHUMAN3H-PSB-118- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87838A2B?CLONEDMOUSE3H-PSB-6038- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione8.34Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87839A1?CLONEDMOUSE3H-CCPA8- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1520Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87840A3?CLONEDMOUSE3H-PSB-118- (4-((4-(4-Chlorophenyl)piperazin-1-yl)sulfonyl)phenyl)-3-methyl-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87841A3?CLONEDMOUSE3H-PSB-118-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87842A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87843A1?CLONEDHUMAN3H-CCPA8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione928Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87844A1?CLONEDMOUSE3H-CCPA8-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione107Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87845A2B?CLONEDMOUSE3H-PSB-6038-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.901Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87846A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.148Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87847A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione92.4Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87848A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione77.8Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87849A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.153Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87850A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87851A1?CLONEDHUMAN3H-CCPA8-(4-((4-(4-Bromobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87852A1?CLONEDHUMAN3H-CCPA8-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione205Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87853A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1.28Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87854A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.397Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87855A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.244Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87856A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione96.7Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87857A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione12.2Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87858A2B?CLONEDHUMAN3H-PSB-6038-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione7.02Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87859A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.894Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87860A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione0.629Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87861A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione1.02Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87862A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione0.473Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87863A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.643Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87864A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.644Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87865A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.632Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87866A2B?CLONEDMOUSE3H-PSB-6038-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.926Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87867A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione6.08Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87868A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione4.3Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87869A2B?CLONEDHUMAN3H-PSB-6031-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.432Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87870A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.706Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87871A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione0.616Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87872A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione0.159Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87873A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.137Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87874A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.234Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87875A2B?CLONEDMOUSE3H-PSB-6038-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.131Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87876A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.0835Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87877A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione0.403Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87878A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.342Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87879A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione3.22Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87880A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87881A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione131Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87882A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione189Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87883A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione208Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87884A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1160Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87885A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione241Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87886A2A?CLONEDHUMAN3H-MSX-28-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione314Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87887A2A?CLONEDHUMAN3H-MSX-28-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione122Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87888A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione108Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87889A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87890A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87891A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione204Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87892A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87893A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87894A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione89.5Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87895A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione2990Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87896A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione197Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87897A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87898A2A?CLONEDHUMAN3H-MSX-21-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione140Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87899A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione96.7Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87900A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione168Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87901A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87902A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione40.7Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87903A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione93.8Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87904A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione35.3Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87905A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87906A2A?CLONEDHUMAN3H-MSX-28-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87907A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione403Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87908A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione160Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87909A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione135Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87910A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione245Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87911A2A?CLONEDHUMAN3H-MSX-28-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione140Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87912A2A?CLONEDHUMAN3H-MSX-24-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide52.7Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87913A2A?CLONEDHUMAN3H-MSX-24-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide357Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87914A2A?CLONEDHUMAN3H-MSX-28-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione293Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87915A2A?CLONEDHUMAN3H-MSX-28-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione143Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87916A2A?CLONEDHUMAN3H-MSX-28-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87917A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione8.34Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87918A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione5.69Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87919A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione7.15Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87920A2B?CLONEDHUMAN3H-PSB-6038-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1.91Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87921A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.421Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87922A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione3.55Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87923A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.215Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87924A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione0.352Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87925A2B?CLONEDHUMAN3H-PSB-6038-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1.24Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87926A1?CLONEDHUMAN3H-CCPA8-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87927A1?CLONEDHUMAN3H-CCPA8-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87928A1?CLONEDHUMAN3H-CCPA8-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione535Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87929A1?CLONEDHUMAN3H-CCPA8-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87930A1?CLONEDHUMAN3H-CCPA8-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione113Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87931A1?CLONEDHUMAN3H-CCPA8-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87932A1?CLONEDHUMAN3H-CCPA4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide190Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87933A1?CLONEDHUMAN3H-CCPA4-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide1036Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87934A1?CLONEDHUMAN3H-CCPA8-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione334Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87935A1?CLONEDHUMAN3H-CCPA8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione364Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87936A1?CLONEDHUMAN3H-CCPA8-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87937A1?CLONEDHUMAN3H-CCPA8-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87938A1?CLONEDHUMAN3H-CCPA8-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87939A1?CLONED? HUMAN3H-CCPA8-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione795Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87940A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione492Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87941A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87942A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione560Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87943A1?CLONED? HUMAN3H-CCPA8-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione1010Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87944A1?CLONED? HUMAN3H-CCPA8-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione364Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87945A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87946A1?CLONED? HUMAN3H-CCPA8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87947A1?CLONED? HUMAN3H-CCPA8-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87948A1?CLONED? HUMAN3H-CCPA8-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87949A1?CLONED? HUMAN3H-CCPA8-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87950A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87951A1?CLONEDMOUSE3H-CCPA8-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87952A1?CLONED? HUMAN3H-CCPA8-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87953A1?CLONED? HUMAN3H-CCPA8-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87954A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87955A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87956A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87957A1?CLONED? HUMAN3H-CCPA1-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione419Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87958A1?CLONED? HUMAN3H-CCPA8-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione356Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87959A1?CLONEDMOUSE3H-CCPA8-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione300Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87960A1?CLONEDHUMAN3H-CCPA8-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87961A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-(2-Hydroxyethoxy)phenyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87962A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Chloro-2-fluorophenyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87963A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(4-Chloro-3-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87964A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(3-Chloro-4-hydroxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87965A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(4-Chloro-3-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87966A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(3-Chloro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87967A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(3-Fluoro-4-methoxyphenyl)piperazin-1-yl]sulfonyl}- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87968A3?CLONEDHUMAN3H-PSB-118-(4-((4-Methylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87969A3?CLONEDHUMAN3H-PSB-114-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N,N-dimethylbenzenesulfonamide1220Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87970A3?CLONEDHUMAN3H-PSB-114-(2,6-Dioxo-1-propyl-2,3,6,7-tetrahydro-purin-8-yl)-N-methylN-phenethylbenzenesulfonamide1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87971A3?CLONEDHUMAN3H-PSB-118-(4-((4-Methyl-3-phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87972A3?CLONEDHUMAN3H-PSB-118-(4-((4-(1-Phenylethyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87973A3?CLONEDHUMAN3H-PSB-118-(4-((4-Benzoylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87974A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Hydroxyphenyl)piperazine-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87975A3?CLONEDHUMAN3H-PSB-111-Propyl-8-(4-((4-(o-tolyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87976A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Methylphenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87977A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Methoxyphenyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87978A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Iodophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87979A3?CLONEDHUMAN3H-PSB-118-(4-((4-(2-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87980A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87981A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87982A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(2-Chlorophenyl)piperazin-1-yl]sulfonyl} phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87983A3?CLONEDHUMAN3H-PSB-118-(4-{[4-(3-Chlorophenyl)piperazin-1-yl]sulfonyl}phenyl)-1-propyl-3,7-dihydropurine-2,6-dione53.5Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87984A3?CLONEDMOUSE3H-PSB-118-(4-((4-(4-Bromophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87985A3?CLONEDMOUSE3H-PSB-118-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87986A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87987A3?CLONEDHUMAN3H-PSB-118-(4-((4-(2-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87988A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Fluorophenyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87989A3?CLONEDHUMAN3H-PSB-118-(4-((4-Phenylpiperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87990A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87991A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87992A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87993A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87994A3?CLONEDHUMAN3H-PSB-118-(4-(4-((p-(2-(2-Methoxyethoxy)ethoxy)-phenyl)methyl)-1- piperazinylthio)phenyl)-1-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87995A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-(2-Hydroxyethoxy)benzyl)piperazine-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87996A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Carboxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87997A3?CLONEDHUMAN3H-PSB-118-(4-((4-(4-Azidobenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87998A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Methylbenzyl)piperazin-1-yl)sulfonyl)phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
87999A3?CLONEDHUMAN3H-PSB-118-(4-((4-(3-Methoxybenzyl)piperazin-1-yl)sulfonyl)phenyl)-1- propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
88000A1?CLONEDHUMAN3H-CCPA8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
88001A1?CLONEDHUMAN3H-CCPA8-(4-((4-(3-Fluoro-4-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydropurine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
88002A1?CLONEDHUMAN3H-CCPA8-(4-((4-(4-Fluoro-3-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
88003A1?CLONEDHUMAN3H-CCPA8-(4-((4-(3-Fluoro-5-methoxybenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione1000Jiang J et al 2019Jan 15, 2025Jan 15, 2025
88004A1?CLONEDHUMAN3H-CCPA8-(4-((4-(4-Bromo-3-fluorobenzyl)piperazin-1-yl)sulfonyl)- phenyl)-1-propyl-3,7-dihydro-purine-2,6-dione326Jiang J et al 2019Jan 15, 2025Jan 15, 2025
88005A1CORTEXRAT3H-CCPAH2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88006A1CORTEXRAT3H-CCPA1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88007A1CORTEXRAT3H-CCPA9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88008A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3870Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88009A1CORTEXRAT3H-CCPA9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4320Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88010A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3160Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88011A1CORTEXRAT3H-CCPA9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2870Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88012A1CORTEXRAT3H-CCPA9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88013A1CORTEXRAT3H-CCPA9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2690Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88014A1CORTEXRAT3H-CCPA9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88015A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88016A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88017A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88018A1CORTEXRAT3H-CCPA9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88019A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione7690Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88020A1CORTEXRAT3H-CCPA9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88021A1CORTEXRAT3H-CCPA9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4400Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88022A1CORTEXRAT3H-CCPA1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88023A1CORTEXRAT3H-CCPAcompound 25>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88024A1CORTEXRAT3H-CCPA10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione2240Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88025A1CORTEXRAT3H-CCPA1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1240Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88026A1CORTEXRAT3H-CCPA10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1530Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88027A1CORTEXRAT3H-CCPA10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione)>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88028A1CORTEXRAT3H-CCPA1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88029A1CORTEXRAT3H-CCPA1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1330Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88030A1CORTEXRAT3H-CCPA10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1880Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88031A1CORTEXRAT3H-CCPAcompound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88032A1CORTEXRAT3H-CCPA8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione1120Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88033A1CORTEXRAT3H-CCPA9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione280Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88034A1CORTEXRAT3H-CCPAcaffeine>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88035A1CORTEXRAT3H-CCPAPreladenant (SCH420814)68.7Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88036A1CORTEXRAT3H-CCPAPSB-360.368Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88037A2ACORTEXRAT3H-MSX-2H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH25220Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88038A2ACORTEXRAT3H-MSX-21,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4300Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88039A2ACORTEXRAT3H-MSX-29-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2650Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88040A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1290Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88041A2ACORTEXRAT3H-MSX-29-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1750Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88042A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3060Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88043A2ACORTEXRAT3H-MSX-29-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione820Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88044A2ACORTEXRAT3H-MSX-29-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4950Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88045A2ACORTEXRAT3H-MSX-29-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione870Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88046A2ACORTEXRAT3H-MSX-29-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4640Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88047A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione8870Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88048A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione5370Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88049A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88050A2ACORTEXRAT3H-MSX-29-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2380Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88051A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2030Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88052A2ACORTEXRAT3H-MSX-29-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88053A2ACORTEXRAT3H-MSX-29-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2620Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88054A2ACORTEXRAT3H-MSX-21,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione7400Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88055A2ACORTEXRAT3H-MSX-2compound 25>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88056A2ACORTEXRAT3H-MSX-210-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1730Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88057A2ACORTEXRAT3H-MSX-21,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione850Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88058A2ACORTEXRAT3H-MSX-210-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione280Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88059A2ACORTEXRAT3H-MSX-210-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione)3820Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88060A2ACORTEXRAT3H-MSX-21,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione3510Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88061A2ACORTEXRAT3H-MSX-21,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione2270Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88062A2ACORTEXRAT3H-MSX-210-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione2260Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88063A2ACORTEXRAT3H-MSX-2compound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88064A2ACORTEXRAT3H-MSX-28-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione3800Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88065A2ACORTEXRAT3H-MSX-29-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione300Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88066A2ACORTEXRAT3H-MSX-2caffeine>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88067A2ACORTEXRAT3H-MSX-2Preladenant (SCH420814)0.661Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88068A2ACORTEXRAT3H-MSX-2PSB-36371Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88069A1CLONEDHUMAN3H-CCPAH2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88070A1CLONEDHUMAN3H-CCPA1,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88071A1CLONEDHUMAN3H-CCPA9-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88072A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88073A1CLONEDHUMAN3H-CCPA9-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88074A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88075A1CLONEDHUMAN3H-CCPA9-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3800Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88076A1CLONEDHUMAN3H-CCPA9-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88077A1CLONEDHUMAN3H-CCPA9-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1910Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88078A1CLONEDHUMAN3H-CCPA9-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88079A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88080A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88081A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88082A1CLONEDHUMAN3H-CCPA9-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88083A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88084A1CLONEDHUMAN3H-CCPA9-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88085A1CLONEDHUMAN3H-CCPA9-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88086A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88087A1CLONEDHUMAN3H-CCPAcompound 25>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88088A1CLONEDHUMAN3H-CCPA10-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88089A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione2470Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88090A1CLONEDHUMAN3H-CCPA10-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione4130Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88091A1CLONEDHUMAN3H-CCPA10-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione)>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88092A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88093A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88094A1CLONEDHUMAN3H-CCPA10-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88095A1CLONEDHUMAN3H-CCPAcompound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88096A1CLONEDHUMAN3H-CCPA8-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88097A1CLONEDHUMAN3H-CCPA9-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione600Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88098A1CLONEDHUMAN3H-CCPAPreladenant (SCH420814)295Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88099A1CLONEDHUMAN3H-CCPAPSB-363.97Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88100A2ACLONEDHUMAN3H-MSX-2H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88101A2ACLONEDHUMAN3H-MSX-21,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88102A2ACLONEDHUMAN3H-MSX-29-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88103A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88104A2ACLONEDHUMAN3H-MSX-29-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88105A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88106A2ACLONEDHUMAN3H-MSX-29-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2070Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88107A2ACLONEDHUMAN3H-MSX-29-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88108A2ACLONEDHUMAN3H-MSX-29-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione930Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88109A2ACLONEDHUMAN3H-MSX-29-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88110A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88111A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88112A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88113A2ACLONEDHUMAN3H-MSX-29-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88114A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88115A2ACLONEDHUMAN3H-MSX-29-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88116A2ACLONEDHUMAN3H-MSX-29-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88117A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88118A2ACLONEDHUMAN3H-MSX-2compound 25>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88119A2ACLONEDHUMAN3H-MSX-210-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88120A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1690Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88121A2ACLONEDHUMAN3H-MSX-210-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione1100Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88122A2ACLONEDHUMAN3H-MSX-210-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione)>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88123A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88124A2ACLONEDHUMAN3H-MSX-21,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88125A2ACLONEDHUMAN3H-MSX-210-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88126A2ACLONEDHUMAN3H-MSX-2compound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88127A2ACLONEDHUMAN3H-MSX-28-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88128A2ACLONEDHUMAN3H-MSX-29-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1390Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88129A2ACLONEDHUMAN3H-MSX-2Preladenant (SCH420814)0.884Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88130A2ACLONEDHUMAN3H-MSX-2PSB-36332Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88131A2BCLONEDHUMAN3H-PSB-603H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88132A2BCLONEDHUMAN3H-PSB-6031,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88133A2BCLONEDHUMAN3H-PSB-6039-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88134A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88135A2BCLONEDHUMAN3H-PSB-6039-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88136A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88137A2BCLONEDHUMAN3H-PSB-6039-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88138A2BCLONEDHUMAN3H-PSB-6039-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88139A2BCLONEDHUMAN3H-PSB-6039-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88140A2BCLONEDHUMAN3H-PSB-6039-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88141A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88142A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88143A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88144A2BCLONEDHUMAN3H-PSB-6039-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88145A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88146A2BCLONEDHUMAN3H-PSB-6039-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88147A2BCLONEDHUMAN3H-PSB-6039-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88148A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88149A2BCLONEDHUMAN3H-PSB-603compound 25>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88150A2BCLONEDHUMAN3H-PSB-60310-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88151A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88152A2BCLONEDHUMAN3H-PSB-60310-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88153A2BCLONEDHUMAN3H-PSB-60310-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione)>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88154A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88155A2BCLONEDHUMAN3H-PSB-6031,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88156A2BCLONEDHUMAN3H-PSB-60310-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88157A2BCLONEDHUMAN3H-PSB-603compound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88158A2BCLONEDHUMAN3H-PSB-6038-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88159A3CLONEDHUMAN3H-PSB-6039-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1320Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88160A2BCLONEDHUMAN3H-PSB-603Preladenant (SCH420814)1000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88161A2BCLONEDHUMAN3H-PSB-603PSB-3648.6Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88162A3CLONEDHUMAN3H-PSB-11H2N-4-NO2-D-Phe-c[D-Cys-Tyr-D-Trp-Lys-Val-Cys]-Tyr-NH2>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88163A3CLONEDHUMAN3H-PSB-111,3,9-Trimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88164A3CLONEDHUMAN3H-PSB-119-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88165A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-propyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88166A3CLONEDHUMAN3H-PSB-119-Butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88167A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-pentyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88168A3CLONEDHUMAN3H-PSB-119-Hexyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88169A3CLONEDHUMAN3H-PSB-119-Isopropyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88170A3CLONEDHUMAN3H-PSB-119-Isobutyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88171A3CLONEDHUMAN3H-PSB-119-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88172A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-(pentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione 1,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88173A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-(4-methylpentan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88174A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-(2-methylhexyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88175A3CLONEDHUMAN3H-PSB-119-(Heptan-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88176A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-(6-methylheptan-2-yl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2570Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88177A3CLONEDHUMAN3H-PSB-119-ethenyl 1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88178A3CLONEDHUMAN3H-PSB-119-Allyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88179A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-9-(prop-2-ynyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88180A3CLONEDHUMAN3H-PSB-11compound 25>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88181A3CLONEDHUMAN3H-PSB-1110-Ethyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88182A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-10-propyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88183A3CLONEDHUMAN3H-PSB-1110-Butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88184A3CLONEDHUMAN3H-PSB-1110-Sec-butyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione)>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88185A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-10-(4-methylpentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88186A3CLONEDHUMAN3H-PSB-111,3-Dimethyl-10-(pentan-2-yl)-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88187A3CLONEDHUMAN3H-PSB-1110-Allyl-1,3-dimethyl-6,7,8,9-tetrahydrodiazepino[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88188A3CLONEDHUMAN3H-PSB-11compound 33>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88189A3CLONEDHUMAN3H-PSB-118-Isopropyl-1,3-dimethyl-6,7-dihydro-1H-imidazo[2,1-f]purine-2,4(1H,3H)-dione>10000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88190A3CLONEDHUMAN3H-PSB-119-Butyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione660Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88191A3CLONEDHUMAN3H-PSB-11Preladenant (SCH420814)1000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88192A3CLONEDHUMAN3H-PSB-11PSB-361000Drabczynska A et al 2013Jan 15, 2025Jan 15, 2025
88193A1?CLONED? HUMAN3H-CCPA8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione396Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88194A1?CLONED? HUMAN3H-CCPA8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88195A1?CLONED? HUMAN3H-CCPA8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88196A1?CLONED? HUMAN3H-CCPA8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88197A1?CLONED? HUMAN3H-CCPA8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88198A1?CLONED? HUMAN3H-CCPA8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88199A1BRAIN CORTEXRAT3H-CCPA9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1780Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88200A1BRAIN CORTEXRAT3H-CCPA9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88201A1BRAIN CORTEXRAT3H-CCPA1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88202A1BRAIN CORTEXRAT3H-CCPA9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88203A1BRAIN CORTEXRAT3H-CCPA9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4360Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88204A1BRAIN CORTEXRAT3H-CCPA1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88205A1BRAIN CORTEXRAT3H-CCPA1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2650Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88206A1BRAIN CORTEXRAT3H-CCPA9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione486Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88207A1BRAIN CORTEXRAT3H-CCPA1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88208A1BRAIN CORTEXRAT3H-CCPA9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88209A1BRAIN CORTEXRAT3H-CCPA9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4900Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88210A1BRAIN CORTEXRAT3H-CCPA9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione4130Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88211A1BRAIN CORTEXRAT3H-CCPA9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione965Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88212A1BRAIN CORTEXRAT3H-CCPA9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88213A1BRAIN CORTEXRAT3H-CCPA9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2320Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88214A1BRAIN CORTEXRAT3H-CCPA9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione927Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88215A1BRAIN CORTEXRAT3H-CCPA9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione931Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88216A1BRAIN CORTEXRAT3H-CCPA9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88217A1BRAIN CORTEXRAT3H-CCPA1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1410Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88218A1BRAIN CORTEXRAT3H-CCPA1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1910Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88219A1BRAIN CORTEXRAT3H-CCPA9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1550Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88220A1BRAIN CORTEXRAT3H-CCPA9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3020Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88221A1?CLONED? HUMAN3H-CCPA10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88222A1?CLONED? HUMAN3H-CCPA10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88223A1?CLONED? HUMAN3H-CCPA10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione651Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88224A1?CLONED? HUMAN3H-CCPA10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88225A1?CLONED? HUMAN3H-CCPA10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88226A1?CLONED? HUMAN3H-CCPA10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88227A1?CLONED? HUMAN3H-CCPA10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88228A1?CLONED? HUMAN3H-CCPA10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88229A1?CLONED? HUMAN3H-CCPA10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88230A2A?CLONED? HUMAN3H-MSX-210-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88231A2A?CLONED? HUMAN3H-MSX-210-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1580Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88232A2A?CLONED? HUMAN3H-MSX-210-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione959Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88233A2A?CLONED? HUMAN3H-MSX-210-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88234A2A?CLONED? HUMAN3H-MSX-210-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione767Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88235A2A?CLONED? HUMAN3H-MSX-210-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88236A2A?CLONED? HUMAN3H-MSX-210-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88237A2A?CLONED? HUMAN3H-MSX-210-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1080Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88238A2A?CLONED? HUMAN3H-MSX-210-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione881Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88239A2A?CLONED? HUMAN3H-MSX-29-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88240A2A?CLONED? HUMAN3H-MSX-29-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione189Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88241A2A?CLONED? HUMAN3H-MSX-21,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88242A2A?CLONED? HUMAN3H-MSX-21,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1020Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88243A2A?CLONED? HUMAN3H-MSX-29-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88244A2A?CLONED? HUMAN3H-MSX-29-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88245A2A?CLONED? HUMAN3H-MSX-29-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione627Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88246A2A?CLONED? HUMAN3H-MSX-29-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88247A2A?CLONED? HUMAN3H-MSX-29-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1610Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88248A2A?CLONED? HUMAN3H-MSX-29-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1700Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88249A2A?CLONED? HUMAN3H-MSX-29-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88250A2A?CLONED? HUMAN3H-MSX-29-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione8910Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88251A2A?CLONED? HUMAN3H-MSX-29-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione8000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88252A2A?CLONED? HUMAN3H-MSX-21,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88253A2A?CLONED? HUMAN3H-MSX-29-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88254A2A?CLONED? HUMAN3H-MSX-21,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione2020Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88255A2A?CLONED? HUMAN3H-MSX-21,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88256A2A?CLONED? HUMAN3H-MSX-29-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88257A2A?CLONED? HUMAN3H-MSX-29-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione8270Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88258A2A?CLONED? HUMAN3H-MSX-21,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione3040Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88259A2A?CLONED? HUMAN3H-MSX-29-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88260A2A?CLONED? HUMAN3H-MSX-29-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1210Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88261A2A?CLONED? HUMAN3H-MSX-28-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione784Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88262A2A?CLONED? HUMAN3H-MSX-28-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88263A2A?CLONED? HUMAN3H-MSX-28-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88264A2A?CLONED? HUMAN3H-MSX-28-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione (887Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88265A2A?CLONED? HUMAN3H-MSX-28-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione369Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88266A2A?CLONED? HUMAN3H-MSX-28-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88267A2A?CLONED? HUMAN3H-MSX-2caffeine>10000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88268A2B?CLONED? HUMAN[ 3 H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)caffeine>10000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88269A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)8-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88270A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)8-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88271A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)8-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88272A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88273A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)8-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88274A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)8-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88275A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88276A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88277A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)1,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88278A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88279A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88280A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)1,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88281A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)1,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88282A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88283A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)1,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88284A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88285A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88286A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(4-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88287A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88288A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88289A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88290A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88291A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88292A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88293A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)1,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88294A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)1,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88295A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88296A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)9-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88297A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88298A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88299A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88300A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88301A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88302A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88303A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88304A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88305A2B?CLONED? HUMAN[ 3H]8-(4-(4-(4-chlorophenyl)piperazine-1-sulfonyl)phenyl)-1-propylxanthine ([3H]PSB-603)10-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88306A3?CLONED? HUMAN3H-PSB-1110-(4-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88307A3?CLONED? HUMAN3H-PSB-1110-(2,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88308A3?CLONED? HUMAN3H-PSB-1110-(2-methoxybenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88309A3?CLONED? HUMAN3H-PSB-1110-(3-bromo-4-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro1H-[1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88310A3?CLONED? HUMAN3H-PSB-1110-(2-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88311A3?CLONED? HUMAN3H-PSB-1110-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H- [1,3]diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88312A3?CLONED? HUMAN3H-PSB-1110-(3-Bromobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88313A3?CLONED? HUMAN3H-PSB-1110-(2-fluorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88314A3?CLONED? HUMAN3H-PSB-1110-(2-chlorobenzyl)-1,3-dimethyl-7,8,9,10-tetrahydro-1H-[1,3] diazepino[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88315A3?CLONED? HUMAN3H-PSB-119-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88316A3?CLONED? HUMAN3H-PSB-119-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88317A3?CLONED? HUMAN3H-PSB-111,3-Dimethyl-9-(3-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88318A3?CLONED? HUMAN3H-PSB-111,3-Dimethyl-9-(2-methylbenzyl)-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88319A3?CLONED? HUMAN3H-PSB-119-(4-(tert-Butyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88320A3?CLONED? HUMAN3H-PSB-119-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88321A3?CLONED? HUMAN3H-PSB-119-(6-Chloro-2-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88322A3?CLONED? HUMAN3H-PSB-119-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88323A3?CLONED? HUMAN3H-PSB-119-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88324A3?CLONED? HUMAN3H-PSB-119-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido [2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88325A3?CLONED? HUMAN3H-PSB-119-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88326A3?CLONED? HUMAN3H-PSB-119-(3-Chloro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88327A3?CLONED? HUMAN3H-PSB-111,3-Dimethyl-9-(2-(pyridin-4-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88328A3?CLONED? HUMAN3H-PSB-119-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88329A3?CLONED? HUMAN3H-PSB-111,3-Dimethyl-9-(thiophen-2-ylmethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88330A3?CLONED? HUMAN3H-PSB-111,3-Dimethyl-9-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88331A3?CLONED? HUMAN3H-PSB-119-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88332A3?CLONED? HUMAN3H-PSB-119-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88333A3?CLONED? HUMAN3H-PSB-111,3-Dimethyl-9-(2-(pyridin-3-yl)ethyl)-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88334A3?CLONED? HUMAN3H-PSB-119-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9- tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88335A3?CLONED? HUMAN3H-PSB-119-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[2,1-f]purine-2,4(1H,3H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88336A3?CLONED? HUMAN3H-PSB-118-(2-Methoxybenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1- f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88337A3?CLONED? HUMAN3H-PSB-118-(4-Chlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88338A3?CLONED? HUMAN3H-PSB-118-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-7,8-dihydro-1Himidazo[2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88339A3?CLONED? HUMAN3H-PSB-118-(3,4-dichlorobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo [2,1-f]purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88340A3?CLONED? HUMAN3H-PSB-118-(2-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88341A3?CLONED? HUMAN3H-PSB-118-(3-Bromobenzyl)-1,3-dimethyl-7,8-dihydro-1H-imidazo[2,1-f] purine-2,4(3H,6H)-dione1000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88342A3?CLONED? HUMAN3H-PSB-11caffeine>10000Zaluski M et al 2019Jan 15, 2025Jan 15, 2025
88343Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(2-((6-Methyl2-phenylpyrimidin-4-yl)oxy)ethyl)morpholine2000Lan Y et al 2014Jan 15, 2025Jan 15, 2025
88344Sigma 2BRAINGUINEA PIG3H-DTG4-(2-((6-Methyl2-phenylpyrimidin-4-yl)oxy)ethyl)morpholine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88345Sigma 2BRAINGUINEA PIG3H-DTG4-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)morpholine949Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88346Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)morpholine36.3Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88347Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)butyl)morpholine95.2Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88348Sigma 2BRAINGUINEA PIG3H-DTG4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)butyl)morpholine1072Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88349Sigma 2BRAINGUINEA PIG3H-DTG4-(5-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)pentyl)morpholine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88350Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(5-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)pentyl)morpholine389Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88351Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(6-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)hexyl)morpholine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88352Sigma 2BRAINGUINEA PIG3H-DTG4-(6-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)hexyl)morpholine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88353Sigma 2BRAINGUINEA PIG3H-DTG(E)-4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)but-2-en-1-yl)- morpholine1451Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88354Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(E)-4-(4-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)but-2-en-1-yl)- morpholine116Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88355Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(2-(2-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)ethoxy)ethyl)- morpholine422Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88356Sigma 2BRAINGUINEA PIG3H-DTG4-(2-(2-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)ethoxy)ethyl)- morpholine1924Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88357Sigma 2BRAINGUINEA PIG3H-DTG1-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-3-morpholinopropan2-ol1644Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88358Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)1-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-3-morpholinopropan2-ol486Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88359Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine1051Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88360Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine11.8Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88361Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-6-(3-(4-methylpiperidin-1-yl)propoxy)-2-phenylpyrimidine16.7Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88362Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-6-(3-(4-methylpiperidin-1-yl)propoxy)-2-phenylpyrimidine1416Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88363Sigma 2BRAINGUINEA PIG3H-DTG4-(3-(3,5-Dimethylpiperidin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine1662Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88364Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(3-(3,5-Dimethylpiperidin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine30.2Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88365Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-2-phenyl-6-(3-(2,2,6,6-tetramethylpiperidin-1-yl)- propoxy)pyrimidine377Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88366Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-2-phenyl-6-(3-(2,2,6,6-tetramethylpiperidin-1-yl)- propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88367Sigma 2BRAINGUINEA PIG3H-DTG1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4-ol1763Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88368Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4-ol462Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88369Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4- one319Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88370Sigma 2BRAINGUINEA PIG3H-DTG1-(3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)propyl)piperidin-4- one1492Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88371Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-2-phenyl-6-(3-(piperazin-1-yl)propoxy)pyrimidine1212Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88372Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-2-phenyl-6-(3-(piperazin-1-yl)propoxy)pyrimidine151Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88373Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-6-(3-(4-methylpiperazin-1-yl)propoxy)-2-phenylpyrimidine22.7Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88374Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-6-(3-(4-methylpiperazin-1-yl)propoxy)-2-phenylpyrimidine1325Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88375Sigma 2BRAINGUINEA PIG3H-DTG4-(3-(4-Ethylpiperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine1179Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88376Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(3-(4-Ethylpiperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine30.6Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88377Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)1-Methyl-4-(3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propyl)-1,4- diazepane18.7Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88378Sigma 2BRAINGUINEA PIG3H-DTG1-Methyl-4-(3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propyl)-1,4- diazepane1295Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88379Sigma 2BRAINGUINEA PIG3H-DTG4-(3-(4-Boc-piperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88380Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-(3-(4-Boc-piperazin-1-yl)propoxy)-6-methyl-2-phenylpyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88381Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-2-phenyl-6-(3-(4-phenylpiperazin-1-yl)propoxy)- pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88382Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-2-phenyl-6-(3-(4-phenylpiperazin-1-yl)propoxy)- pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88383Sigma 2BRAINGUINEA PIG3H-DTG4-Methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine1253Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88384Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine13.6Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88385Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N,N-Dimethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan1-amine82.3Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88386Sigma 2BRAINGUINEA PIG3H-DTGN,N-Dimethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan1-amine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88387Sigma 2BRAINGUINEA PIG3H-DTGN,N-Diethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan-1- amine1317Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88388Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N,N-Diethyl-3-((6-methyl-2-phenylpyrimidin-4-yl)oxy)propan-1- amine47.1Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88389Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-N,N-dipropylpropan-1- amine38.8Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88390Sigma 2BRAINGUINEA PIG3H-DTG3-((6-Methyl-2-phenylpyrimidin-4-yl)oxy)-N,N-dipropylpropan-1- amine1069Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88391Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Ethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine20.5Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88392Sigma 2BRAINGUINEA PIG3H-DTG4-Ethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine1141Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88393Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-propylpyrimidine1456Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88394Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-propylpyrimidine34.9Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88395Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Isopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine188Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88396Sigma 2BRAINGUINEA PIG3H-DTG4-Isopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine1836Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88397Sigma 2BRAINGUINEA PIG3H-DTG4-Methoxy-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine892Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88398Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methoxy-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine19.3Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88399Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-(trifluoromethyl)- pyrimidine27.6Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88400Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6-(trifluoromethyl)- pyrimidine1327Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88401Sigma 2BRAINGUINEA PIG3H-DTG4-Cyclopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88402Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Cyclopropyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine253Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88403Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2,4-Diphenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine966Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88404Sigma 2BRAINGUINEA PIG3H-DTG2,4-Diphenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88405Sigma 2BRAINGUINEA PIG3H-DTG4,5-Dimethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine1221Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88406Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4,5-Dimethyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine9.51Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88407Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Fluoro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine3.75Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88408Sigma 2BRAINGUINEA PIG3H-DTG5-Fluoro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine1361Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88409Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine1649Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88410Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-4-methyl-2-phenyl-6-(3-(piperidin-1-yl)propoxy)- pyrimidine2.33Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88411Sigma 2BRAINGUINEA PIG3H-DTG4-Ethyl-2-phenyl6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine1429Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88412Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Ethyl-2-phenyl6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine22.4Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88413Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-propylpyrimidine38.9Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88414Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-propylpyrimidine1396Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88415Sigma 2BRAINGUINEA PIG3H-DTG4-Isopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine1092Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88416Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Isopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine218Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88417Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Methoxy-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine19.3Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88418Sigma 2BRAINGUINEA PIG3H-DTG4-Methoxy-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine892Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88419Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-(trifluoromethyl)-pyrimidine1327Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88420Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6-(trifluoromethyl)-pyrimidine27.6Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88421Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-Cyclopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine278Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88422Sigma 2BRAINGUINEA PIG3H-DTG4-Cyclopropyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88423Sigma 2BRAINGUINEA PIG3H-DTG2,4-Diphenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88424Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2,4-Diphenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine735Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88425Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4,5-Dimethyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine11.4Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88426Sigma 2BRAINGUINEA PIG3H-DTG4,5-Dimethyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)pyrimidine1279Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88427Sigma 2BRAINGUINEA PIG3H-DTG5-Fluoro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine1194Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88428Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Fluoro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine3.51Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88429Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine4.02Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88430Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-4-methyl-2-phenyl-6-(3-(pyrrolidin-1-yl)propoxy)-pyrimidine1684Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88431Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine1626Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88432Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine44.2Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88433Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine58.9Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88434Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-6,7-dihydro-5Hcyclopenta[d]pyrimidine1896Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88435Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88436Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(piperidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline138.5Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88437Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline111.8Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88438Sigma 2BRAINGUINEA PIG3H-DTG2-Phenyl-4-(3-(pyrrolidin-1-yl)propoxy)-5,6,7,8-tetrahydroquinazoline1916Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88439Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(p-tolyl)-pyrimidine1554Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88440Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(p-tolyl)-pyrimidine1.96Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88441Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2-(4-methoxyphenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine3.88Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88442Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2-(4-methoxyphenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine1288Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88443Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(4- (trifluoromethyl)phenyl)pyrimidine1776Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88444Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)-2-(4- (trifluoromethyl)phenyl)pyrimidine4.42Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88445Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2-(4-fluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine1.14Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88446Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2-(4-fluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine1329Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88447Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2-(3,4-difluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine943Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88448Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2-(3,4-difluorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine0.97Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88449Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2-(4-chlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine1.06Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88450Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2-(4-chlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)-propoxy)pyrimidine1425Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88451Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2-(3,4-dichlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88452Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2-(3,4-dichlorophenyl)-4-methyl-6-(3-(piperidin-1-yl)- propoxy)pyrimidine89.8Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88453Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-4-methyl-2-(naphthalen-2-yl)-6-(3-(piperidin-1-yl)-propoxy)pyrimidine102Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88454Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-4-methyl-2-(naphthalen-2-yl)-6-(3-(piperidin-1-yl)-propoxy)pyrimidine2000Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88455Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine1104Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88456Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-4-methyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine187Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88457Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2,4-dimethyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine58.8Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88458Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2,4-dimethyl-6-(3-(piperidin-1-yl)propoxy)pyrimidine1081Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88459Sigma 2BRAINGUINEA PIG3H-DTG5-Chloro-2-cyclopropyl-4-methyl-6-(3-(piperidin-1-yl)propoxy)-pyrimidine1328Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88460Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Chloro-2-cyclopropyl-4-methyl-6-(3-(piperidin-1-yl)propoxy)-pyrimidine39.5Lan Y et al 2014Jan 15, 2025Jan 28, 2025
88461D2CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol24Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88462D3CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol666Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88463D4CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol1.5Peprah K et al 2012Jan 15, 2025Jan 28, 2025
884645-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol658Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884655-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol302Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884665-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88467D2CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol8.8Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88468D3CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol49Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88469D4CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol247.8Peprah K et al 2012Jan 15, 2025Jan 28, 2025
884705-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol317Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884715-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol72Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884725-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88473D2CLONEDHUMAN3H-N-Methylspiperone4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol5.3Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88474D3CLONEDHUMAN3H-N-Methylspiperone4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol182Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88475D4CLONEDHUMAN3H-N-Methylspiperone4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol2.4Peprah K et al 2012Jan 15, 2025Jan 28, 2025
884765-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol74Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884775-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol93Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884785-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-Chloro-phenyl)-1-[3-(4-fluoro-phenoxy)-propyl]-pi peridin-4-ol>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88479D2CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride185Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88480D3CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride130Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88481D4CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride39Peprah K et al 2012Jan 15, 2025Jan 28, 2025
884825-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride454Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884835-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride112Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884845-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)pi peridine hydrochloride>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88485D2CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine41Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88486D3CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine696Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88487D4CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine9.5Peprah K et al 2012Jan 15, 2025Jan 28, 2025
884885-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine169Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884895-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine121Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884905-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-Chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperi dine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88491D2CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl998Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88492D3CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl243Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88493D4CLONEDHUMAN3H-N-Methylspiperone4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl35Peprah K et al 2012Jan 15, 2025Jan 28, 2025
884945-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl613Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884955-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl222Peprah K et al 2012Jan 15, 2025Jan 15, 2025
884965-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-Chlorophenyl)-1-(3-((4-fluorophenyl)sulfinyl)propyl) piperidine HCl>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88497D2CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine284Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88498D3CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine261Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88499D4CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine7.8Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885005-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine112Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885015-HT2ACLONEDHUMAN3H-KETANSERIN1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine81Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885025-HT2CCLONEDHUMAN3H-MESULERGINE1-(4-Chlorophenyl)-4-(4-(4-fluorophenyl)butyl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88503D2CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine211Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88504D3CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine422Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88505D4CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine8.7Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885065-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine166Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885075-HT2ACLONEDHUMAN3H-KETANSERIN1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine53Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885085-HT2CCLONEDHUMAN3H-MESULERGINE1-(4-Chlorophenyl)-4-(3-((4-fluorophenyl)thio)propyl)pi perazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88509D2CLONEDHUMAN3H-N-Methylspiperone1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl4753Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88510D3CLONEDHUMAN3H-N-Methylspiperone1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl544Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88511D4CLONEDHUMAN3H-N-Methylspiperone1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl89Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885125-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl1080Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885135-HT2ACLONEDHUMAN3H-KETANSERIN1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl1129Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885145-HT2CCLONEDHUMAN3H-MESULERGINE1-(3-((4-Fluorophenyl)thio)propyl)-4-(4-(trifluoromethyl) phenyl)piperazine HCl>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88515D2CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine390Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88516D3CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine885Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88517D4CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine6.9Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885185-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine80Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885195-HT2ACLONEDHUMAN3H-KETANSERIN1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine60Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885205-HT2CCLONEDHUMAN3H-MESULERGINE1-(4-Chlorophenyl)-4-(3-(4-fluorophenoxy)propyl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88521D2CLONEDHUMAN3H-N-Methylspiperone1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine37Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88522D3CLONEDHUMAN3H-N-Methylspiperone1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine207Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88523D4CLONEDHUMAN3H-N-Methylspiperone1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine7.4Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885245-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine24Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885255-HT2ACLONEDHUMAN3H-KETANSERIN1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine57.6Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885265-HT2CCLONEDHUMAN3H-MESULERGINE1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88527D2CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl447Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88528D3CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl726Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88529D4CLONEDHUMAN3H-N-Methylspiperone1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl5.6Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885305-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl154Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885315-HT2ACLONEDHUMAN3H-KETANSERIN1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl19.8Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885325-HT2CCLONEDHUMAN3H-MESULERGINE1-(4-Chlorophenyl)-4-(3-phenoxypropyl)piperazine HCl>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88533D2CLONEDHUMAN3H-N-Methylspiperone1-(3-Phenoxypropyl)-4-phenylpiperazine119Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88534D3CLONEDHUMAN3H-N-Methylspiperone1-(3-Phenoxypropyl)-4-phenylpiperazine79.3Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88535D4CLONEDHUMAN3H-N-Methylspiperone1-(3-Phenoxypropyl)-4-phenylpiperazine4.5Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885365-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(3-Phenoxypropyl)-4-phenylpiperazine25Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885375-HT2ACLONEDHUMAN3H-KETANSERIN1-(3-Phenoxypropyl)-4-phenylpiperazine46Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885385-HT2CCLONEDHUMAN3H-MESULERGINE1-(3-Phenoxypropyl)-4-phenylpiperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88539D2CLONEDHUMAN3H-N-Methylspiperone(4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine269Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88540D3CLONEDHUMAN3H-N-Methylspiperone(4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine262Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88541D4CLONEDHUMAN3H-N-Methylspiperone(4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine6.2Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885425-HT1ACLONEDHUMAN3H-8-OH-DPAT(4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine8.6Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885435-HT2ACLONEDHUMAN3H-KETANSERIN(4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine41Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885445-HT2CCLONEDHUMAN3H-MESULERGINE(4-(4-(4-Fluorophenyl)butyl)piperazin-1-yl)pyrimidine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88545D2CLONEDHUMAN3H-N-Methylspiperone2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine424Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88546D3CLONEDHUMAN3H-N-Methylspiperone2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine68Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88547D4CLONEDHUMAN3H-N-Methylspiperone2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine21Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885485-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine93.1Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885495-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine27Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885505-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-(3-((4-Fluorophenyl)thio)propyl)piperazin-1- yl)pyrimidine8829Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88551D2CLONEDHUMAN3H-N-Methylspiperone2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine636Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88552D3CLONEDHUMAN3H-N-Methylspiperone2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine778Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88553D4CLONEDHUMAN3H-N-Methylspiperone2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine4.2Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885545-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine23Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885555-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine23Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885565-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-(3-(4-Fluorophenoxy)propyl)piperazin-1- yl)pyrimidine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88557D2CLONEDHUMAN3H-N-Methylspiperone1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine124Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88558D3CLONEDHUMAN3H-N-Methylspiperone1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine86Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88559D4CLONEDHUMAN3H-N-Methylspiperone1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine3.5Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885605-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine1.1Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885615-HT2ACLONEDHUMAN3H-KETANSERIN1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine50Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885625-HT2CCLONEDHUMAN3H-MESULERGINE1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88563D2CLONEDHUMAN3H-N-Methylspiperone1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine183Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88564D3CLONEDHUMAN3H-N-Methylspiperone1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine160Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88565D4CLONEDHUMAN3H-N-Methylspiperone1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine5.7Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885665-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine6.2Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885675-HT2ACLONEDHUMAN3H-KETANSERIN1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine26Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885685-HT2CCLONEDHUMAN3H-MESULERGINE1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine8097Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88569D2CLONEDHUMAN3H-N-Methylspiperone1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine186Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88570D3CLONEDHUMAN3H-N-Methylspiperone1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine229Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88571D4CLONEDHUMAN3H-N-Methylspiperone1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine1.8Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885725-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine3.6Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885735-HT2ACLONEDHUMAN3H-KETANSERIN1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine18Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885745-HT2CCLONEDHUMAN3H-MESULERGINE1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine8277Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88575H1CLONEDHUMAN3H-PYRILAMINE1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine62.9Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88576M1CLONEDHUMAN3H-QNB1-(3-(4-Fluorophenoxy)propyl)-4-phenylpiperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88577M1CLONEDHUMAN3H-QNB1-(3-Phenoxypropyl)-4-phenylpiperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88578H1CLONEDHUMAN3H-PYRILAMINE1-(3-Phenoxypropyl)-4-phenylpiperazine67.9Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88579H1CLONEDHUMAN3H-PYRILAMINE1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine167Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88580M1CLONEDHUMAN3H-QNB1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885815-HT7CLONEDHUMAN3H-LSD1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine90Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88582Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(4-(4-Fluorophenyl)butyl)-4-(pyridin-2-yl)piperazine308.2Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885835-HT7CLONEDHUMAN3H-LSD1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine291Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88584H1CLONEDHUMAN3H-PYRILAMINE1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine212Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88585M1CLONEDHUMAN3H-QNB1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88586Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(3-((4-Fluorophenyl)thio)propyl)-4-(pyridin-2-yl)piperazine45.1Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88587Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine194.5Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885885-HT7CLONEDHUMAN3H-LSD1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine208Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88589H1CLONEDHUMAN3H-PYRILAMINE1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine262Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88590M1CLONEDHUMAN3H-QNB1-(3-(4-Fluorophenoxy)propyl)-4-(pyridin-2-yl)piperazine>10000Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88591D2CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE130Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88592D4CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE54Peprah K et al 2012Jan 15, 2025Jan 28, 2025
885935-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE140Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885945-HT2ACLONEDHUMAN3H-KETANSERINCLOZAPINE8.9Peprah K et al 2012Jan 15, 2025Jan 15, 2025
885955-HT2CCLONEDHUMAN3H-MESULERGINECLOZAPINE17Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88596H1CLONEDHUMAN3H-PYRILAMINECLOZAPINE1.8Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88597M1CLONEDHUMAN3H-QNBCLOZAPINE1.8Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88598D2CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL0.89Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88599D4CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL10Peprah K et al 2012Jan 15, 2025Jan 28, 2025
886005-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL3600Peprah K et al 2012Jan 15, 2025Jan 15, 2025
886015-HT2ACLONEDHUMAN3H-KETANSERINHALOPERIDOL120Peprah K et al 2012Jan 15, 2025Jan 15, 2025
886025-HT2CCLONEDHUMAN3H-MESULERGINEHALOPERIDOL4700Peprah K et al 2012Jan 15, 2025Jan 15, 2025
88603H1CLONEDHUMAN3H-PYRILAMINEHALOPERIDOL440Peprah K et al 2012Jan 15, 2025Jan 28, 2025
88604M1CLONEDHUMAN3H-QNBHALOPERIDOL1600Peprah K et al 2012Jan 15, 2025Jan 15, 2025
886055-HT1ACLONEDHUMAN3H-8-OH-DPATHALOPERIDOL3600Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886065-HT2ACLONEDHUMAN3H-KETANSERINHALOPERIDOL120Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88607D1CLONEDHUMAN3H-SCH23390HALOPERIDOL120Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88608D2CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL0.89Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88609D3CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL2.5Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88610D4CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL10Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886115-HT2CCLONEDHUMAN3H-MESULERGINEHALOPERIDOL4700Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88612H1CLONEDHUMAN3H-PYRILAMINEHALOPERIDOL440Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88613NETCLONEDHUMAN3H-NisoxetineHALOPERIDOL5500Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88614SERTCLONEDHUMAN3H-CITALOPRAMHALOPERIDOL1800Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886155-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol658Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886165-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol302Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886175-HT7CLONEDHUMAN3H-LSD4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol1042Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88618D1CLONEDHUMAN3H-SCH233904-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol130Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88619D5CLONEDHUMAN3H-SCH233904-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol414Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88620D2CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol24Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88621D3CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol668Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88622D4CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol1.5Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886235-HT2BCLONEDHUMAN3H-LSD4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol723Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886245-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88625H1CLONEDHUMAN3H-PYRILAMINE4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol128.5Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88626M1CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88627M2CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88628M3CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88629DATCLONEDHUMAN3H-WIN354284-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88630NETCLONEDHUMAN3H-Nisoxetine4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol1225Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88631SERTCLONEDHUMAN3H-CITALOPRAM4-(4-chlorophenyl)-1-(4-(4-fluorophenyl)butyl)piperidin-4-ol1867Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886325-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol317Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886335-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol72Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886345-HT7CLONEDHUMAN3H-LSD4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol656Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88635D1CLONEDHUMAN3H-SCH233904-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol22Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88636D5CLONEDHUMAN3H-SCH233904-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol103Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88637D2CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol8.8Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88638D3CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol49Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88639D4CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol4.3Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886405-HT2BCLONEDHUMAN3H-LSD4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol1622Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886415-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88642H1CLONEDHUMAN3H-PYRILAMINE4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol699Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88643M1CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88644M2CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88645M3CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88646DATCLONEDHUMAN3H-WIN 35,4284-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88647NETCLONEDHUMAN3H-Nisoxetine4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol3959Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88648SERTCLONEDHUMAN3H-CITALOPRAM4-(4-chlorophenyl)-1-(3-(4-fluorophenoxy)propyl)piperidin-4-ol2228Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886495-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol74Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886505-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol93Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886515-HT7CLONEDHUMAN3H-LSD4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol1044Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88652D1CLONEDHUMAN3H-SCH233904-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol27Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88653D5CLONEDHUMAN3H-SCH233904-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol113Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88654D2CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol5.3Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88655D3CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol182Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88656D4CLONEDHUMAN3H-N-Methylspiperone4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol2.4Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886575-HT2BCLONEDHUMAN3H-LSD4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol790Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886585-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88659H1CLONEDHUMAN3H-PYRILAMINE4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol115Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88660M1CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88661M2CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88662M3CLONEDHUMAN3H-QNB4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88663DATCLONEDHUMAN3H-WIN 35,4284-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol497Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88664NETCLONEDHUMAN3H-Nisoxetine4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol2249Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88665SERTCLONEDHUMAN3H-CITALOPRAM4-(4-chlorophenyl)-1-(3-((4-fluorophenyl)thio)propyl)piperidin-4-ol160Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88666D2CLONEDHUMAN3H-N-Methylspiperone4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one0.31Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88667D3CLONEDHUMAN3H-N-Methylspiperone4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one0.71Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88668D4CLONEDHUMAN3H-N-Methylspiperone4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one12Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886695-HT2CCLONEDHUMAN3H-MESULERGINE4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one872Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88670H1CLONEDHUMAN3H-PYRILAMINE4-(3-(4-chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one8780Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886715-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol102Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886725-HT2ACLONEDHUMAN3H-KETANSERIN3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol317Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886735-HT7CLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol472Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88674D1CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88675D5CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88676D2CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol33Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88677D3CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol9.7Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88678D4CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol9.4Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886795-HT2BCLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol1381Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886805-HT2CCLONEDHUMAN3H-MESULERGINE3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol2434Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88681H1CLONEDHUMAN3H-PYRILAMINE3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol1719Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88682M1CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88683M2CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88684M3CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88685DATCLONEDHUMAN3H-WIN 35,4283-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol778Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88686NETCLONEDHUMAN3H-Nisoxetine3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88687SERTCLONEDHUMAN3H-CITALOPRAM3-(4-chlorophenyl)-8-(4-(4-fluorophenyl)butyl)-8-azabicyclo[3.2.1]octan-3-ol414Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886885-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol123Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886895-HT2ACLONEDHUMAN3H-KETANSERIN3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol236Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886905-HT7CLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol420Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88691D1CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88692D5CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88693D2CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol22Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88694D3CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol4.1Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88695D4CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol49Sampson D et al 2014Jan 15, 2025Jan 28, 2025
886965-HT2BCLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol898Sampson D et al 2014Jan 15, 2025Jan 15, 2025
886975-HT2CCLONEDHUMAN3H-MESULERGINE3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88698H1CLONEDHUMAN3H-PYRILAMINE3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol4149Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88699M1CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88700M2CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88701M3CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88702DATCLONEDHUMAN3H-WIN 35,4283-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol620Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88703NETCLONEDHUMAN3H-Nisoxetine3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol1791Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88704SERTCLONEDHUMAN3H-CITALOPRAM3-(4-chlorophenyl)-8-(3-(4-fluorophenoxy)propyl)-8-azabicyclo[3.2.1]octan-3-ol255Sampson D et al 2014Jan 15, 2025Jan 28, 2025
887055-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol20Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887065-HT2ACLONEDHUMAN3H-KETANSERIN3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol89Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887075-HT7CLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol97Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88708D1CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol347Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88709D5CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88710D2CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol2.9Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88711D3CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol0.7Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88712D4CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol8.9Sampson D et al 2014Jan 15, 2025Jan 28, 2025
887135-HT2BCLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1057Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887145-HT2CCLONEDHUMAN3H-MESULERGINE3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1498Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88715H1CLONEDHUMAN3H-PYRILAMINE3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol977Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88716M1CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88717M2CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88718M3CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88719DATCLONEDHUMAN3H-WIN 35,4283-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1081Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88720NETCLONEDHUMAN3H-Nisoxetine3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1409Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88721SERTCLONEDHUMAN3H-CITALOPRAM3-(4-chlorophenyl)-8-(3-((4-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol316Sampson D et al 2014Jan 15, 2025Jan 28, 2025
887225-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol13Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887235-HT2ACLONEDHUMAN3H-KETANSERIN3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol509Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887245-HT7CLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol917Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88725D1CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88726D5CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88727D2CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol27Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88728D3CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol11Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88729D4CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol28Sampson D et al 2014Jan 15, 2025Jan 28, 2025
887305-HT2BCLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol270Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887315-HT2CCLONEDHUMAN3H-MESULERGINE3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1861Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88732H1CLONEDHUMAN3H-PYRILAMINE3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1207Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88733M1CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88734M2CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88735M3CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88736DATCLONEDHUMAN3H-WIN 35,4283-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol285Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88737NETCLONEDHUMAN3H-Nisoxetine3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol510Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88738SERTCLONEDHUMAN3H-CITALOPRAM3-(4-chlorophenyl)-8-(3-((3-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol227Sampson D et al 2014Jan 15, 2025Jan 28, 2025
887395-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol8.2Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887405-HT2ACLONEDHUMAN3H-KETANSERIN3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol115Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887415-HT7CLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol882Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88742D1CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol4093Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88743D5CLONEDHUMAN3H-SCH233903-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88744D2CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol4.8Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88745D3CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1.3Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88746D4CLONEDHUMAN3H-N-Methylspiperone3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol27Sampson D et al 2014Jan 15, 2025Jan 28, 2025
887475-HT2BCLONEDHUMAN3H-LSD3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol520Sampson D et al 2014Jan 15, 2025Jan 15, 2025
887485-HT2CCLONEDHUMAN3H-MESULERGINE3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1122Sampson D et al 2014Jan 15, 2025Jan 15, 2025