92749 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13:15,16-diepoxylabdane-6b,15a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92750 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13:15,16-diepoxylabdane-6b,16b-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92751 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13:15,16-diepoxylabdane-6b,16a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92752 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13-epoxylabd-5-en-7-on-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92753 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92754 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13-epoxy-15,16-dihydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92755 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13-epoxylabd-5-ene-7 b,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92756 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) (8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92757 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92758 Sigma 1 CLONED HUMAN M3 3H-Pentazocine(+) 9,13-epoxy-6-hydroxylabdan-15,16-olide 2900 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92759 Sigma 2 CLONED HUMAN M3 3H-DTG (5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92760 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13:15,16-diepoxylabdane-6b,15a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92761 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13:15,16-diepoxylabdane-6b,16b-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92762 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13:15,16-diepoxylabdane-6b,16a-diol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92763 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13-epoxylabd-5-en-7-on-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92764 Sigma 2 CLONED HUMAN M3 3H-DTG 15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92765 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13-epoxy-15,16-dihydroxylabd-5-en-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92766 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13-epoxylabd-5-ene-7 b,15,16-triol >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92767 Sigma 2 CLONED HUMAN M3 3H-DTG (8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92768 Sigma 2 CLONED HUMAN M3 3H-DTG 15,16-epoxylabda-5,8,13(16),14-tetraen-7-one >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92769 Sigma 2 CLONED HUMAN M3 3H-DTG 9,13-epoxy-6-hydroxylabdan-15,16-olide >10000 Wu H et al 2013 Jan 15, 2025 Jan 28, 2025
92770 A1 CLONED HUMAN 3H-PIA 2-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine 1620 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92771 A1 CLONED HUMAN 3H-PIA thio-Cl-IB-MECA 20.2 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92772 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 3310 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92773 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 570 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92774 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 220 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92775 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide 480 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92776 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide 1880 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92777 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1090 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92778 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide 440 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92779 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carboxamide 420 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92780 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 83.5 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92781 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 37.5 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92782 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 25.2 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92783 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide 2060 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92784 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92785 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 232 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92786 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 156 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92787 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 311 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92788 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide 186 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92789 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 61.7 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92790 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide 59.4 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92791 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92792 A1 CLONED HUMAN 3H-PIA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92793 A2A CLONED HUMAN 3H-CGS-21680 2-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine 2910 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92794 A2A CLONED HUMAN 3H-CGS-21680 thio-Cl-IB-MECA 475 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92795 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1350 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92796 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 555 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92797 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 560 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92798 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide 1080 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92799 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide 1260 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92800 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1160 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92801 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide 195 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92802 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carboxamide 2480 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92803 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92804 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1080 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92805 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1090 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92806 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92807 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92808 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 238 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92809 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 1230 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92810 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 1200 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92811 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92812 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 899 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92813 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide 1120 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92814 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92815 A2A CLONED HUMAN 3H-CGS-21680 (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide >10000 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92816 A3 CLONED HUMAN 125I-AB-MECA thio-Cl-IB-MECA 0.25 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92817 A3 CLONED HUMAN 125I-AB-MECA 2-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine 1.8 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92818 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 2.3 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92819 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 3.45 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92820 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 0.9 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92821 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide 0.57 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92822 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide 3.75 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92823 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 4.41 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92824 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide 1.76 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92825 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carboxamide 3.93 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92826 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 2.49 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92827 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1.39 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92828 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 7.07 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92829 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide 1.49 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92830 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 3.35 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92831 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 1.96 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92832 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 1.99 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92833 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 4.2 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92834 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide 1.9 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92835 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide 1 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92836 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide 3.56 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92837 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide 4180 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92838 A3 CLONED HUMAN 125I-AB-MECA (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide 7360 Yu J et al 2017 Jan 15, 2025 Jan 15, 2025
92839 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92840 A1 CLONED HUMAN 3H-DPCPX 2-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92841 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92842 A1 CLONED HUMAN 3H-DPCPX 2-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92843 A1 CLONED HUMAN 3H-DPCPX 2-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92844 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92845 A1 CLONED HUMAN 3H-DPCPX 2-(4-Hydroxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92846 A1 CLONED HUMAN 3H-DPCPX 4-(5-Methyl-7-oxo-6,7-dihydro-thiazolo[5,4-d]pyrimidin-2- yl)-benzoic acid 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92847 A1 CLONED HUMAN 3H-DPCPX 2-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92848 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92849 A1 CLONED HUMAN 3H-DPCPX 2-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92850 A1 CLONED HUMAN 3H-DPCPX 2-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92851 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92852 A1 CLONED HUMAN 3H-DPCPX 2-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92853 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92854 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92855 A1 CLONED HUMAN 3H-DPCPX 2-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92856 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92857 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92858 A1 CLONED HUMAN 3H-DPCPX 2-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92859 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92860 A1 CLONED HUMAN 3H-DPCPX 2-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92861 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92862 A1 CLONED HUMAN 3H-DPCPX 2-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92863 A1 CLONED HUMAN 3H-DPCPX 2-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92864 A1 CLONED HUMAN 3H-DPCPX 5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92865 A1 CLONED HUMAN 3H-DPCPX 2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92866 A1 CLONED HUMAN 3H-DPCPX 2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92867 A1 CLONED HUMAN 3H-DPCPX 7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92868 A1 CLONED HUMAN 3H-DPCPX 7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92869 A1 CLONED HUMAN 3H-DPCPX 2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92870 A1 CLONED HUMAN 3H-DPCPX 7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92871 A1 CLONED HUMAN 3H-DPCPX 7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92872 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92873 A2A CLONED HUMAN 3H-ZM241385 2-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92874 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92875 A2A CLONED HUMAN 3H-ZM241385 2-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92876 A2A CLONED HUMAN 3H-ZM241385 2-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92877 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92878 A2A CLONED HUMAN 3H-ZM241385 2-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92879 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92880 A2A CLONED HUMAN 3H-ZM241385 2-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92881 A2A CLONED HUMAN 3H-ZM241385 2-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92882 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92883 A2A CLONED HUMAN 3H-ZM241385 2-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92884 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92885 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92886 A2A CLONED HUMAN 3H-ZM241385 2-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92887 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92888 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92889 A2A CLONED HUMAN 3H-ZM241385 2-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92890 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92891 A2A CLONED HUMAN 3H-ZM241385 2-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92892 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-on 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92893 A2A CLONED HUMAN 3H-ZM241385 2-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92894 A2A CLONED HUMAN 3H-ZM241385 2-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92895 A2A CLONED HUMAN 3H-ZM241385 5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92896 A2A CLONED HUMAN 3H-ZM241385 2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92897 A2A CLONED HUMAN 3H-ZM241385 2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92898 A2A CLONED HUMAN 3H-ZM241385 7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92899 A2A CLONED HUMAN 3H-ZM241385 7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92900 A2A CLONED HUMAN 3H-ZM241385 2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92901 A2A CLONED HUMAN 3H-ZM241385 7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92902 A2A CLONED HUMAN 3H-ZM241385 7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92903 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one 85 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92904 A3 CLONED HUMAN 125I-AB-MECA 2-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 38 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92905 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 33 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92906 A3 CLONED HUMAN 125I-AB-MECA 2-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 18 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92907 A3 CLONED HUMAN 125I-AB-MECA 2-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 107 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92908 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92909 A3 CLONED HUMAN 125I-AB-MECA 2-(4-Hydroxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92910 A3 CLONED HUMAN 125I-AB-MECA 4-(5-Methyl-7-oxo-6,7-dihydro-thiazolo[5,4-d]pyrimidin-2- yl)-benzoic acid 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92911 A3 CLONED HUMAN 125I-AB-MECA 2-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92912 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one 384 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92913 A3 CLONED HUMAN 125I-AB-MECA 2-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one 826 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92914 A3 CLONED HUMAN 125I-AB-MECA 2-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 109 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92915 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92916 A3 CLONED HUMAN 125I-AB-MECA 2-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 427 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92917 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92918 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92919 A3 CLONED HUMAN 125I-AB-MECA 2-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92920 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one 248 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92921 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one 227 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92922 A3 CLONED HUMAN 125I-AB-MECA 2-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92923 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92924 A3 CLONED HUMAN 125I-AB-MECA 2-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92925 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92926 A3 CLONED HUMAN 125I-AB-MECA 2-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92927 A3 CLONED HUMAN 125I-AB-MECA 2-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 113 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92928 A3 CLONED HUMAN 125I-AB-MECA 5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one 450 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92929 A3 CLONED HUMAN 125I-AB-MECA 2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92930 A3 CLONED HUMAN 125I-AB-MECA 2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92931 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92932 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92933 A3 CLONED HUMAN 125I-AB-MECA 2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92934 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine 1000 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92935 A3 CLONED HUMAN 125I-AB-MECA 7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine 110 Varano F et al 2015 Jan 15, 2025 Jan 15, 2025
92936 5-HT6 CLONED HUMAN 3H-LSD WA-13 23 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92937 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine 21 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92938 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 16 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92939 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 6 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92940 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 23 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92941 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 73 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92942 5-HT6 CLONED HUMAN 3H-LSD 4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 274 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92943 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 13 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92944 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 6 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92945 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 12 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92946 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 17 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92947 5-HT6 CLONED HUMAN 3H-LSD 4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 470 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92948 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride 95 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92949 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 86 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92950 5-HT6 CLONED HUMAN 3H-LSD 4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 1061 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92951 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 27 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92952 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 11 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92953 5-HT6 CLONED HUMAN 3H-LSD (RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 26 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92954 5-HT6 CLONED HUMAN 3H-LSD (RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 51 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92955 5-HT6 CLONED HUMAN 3H-LSD 4-[3-(2,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 999 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92956 5-HT6 CLONED HUMAN 3H-LSD OLANZAPINE 7 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92957 5-HT2A CLONED HUMAN 3H-KETANSERIN WA-13 1830 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92958 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine 5047 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92959 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 268 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92960 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 209 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92961 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 310 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92962 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 470 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92963 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 649 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92964 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 355 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92965 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 484 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92966 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 382 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92967 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 431 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92968 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 1457 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92969 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride 576 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92970 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 696 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92971 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 906 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92972 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 412 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92973 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 463 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92974 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 488 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92975 5-HT2A CLONED HUMAN 3H-KETANSERIN (RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 839 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92976 5-HT7 CLONED HUMAN 3H-5-CT WA-13 >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92977 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92978 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92979 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 5202 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92980 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92981 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 5265 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92982 5-HT7 CLONED HUMAN 3H-5-CT 4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 8592 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92983 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92984 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 5706 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92985 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92986 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 6263 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92987 5-HT7 CLONED HUMAN 3H-5-CT 4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 7924 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92988 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride 5928 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92989 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 5098 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92990 5-HT7 CLONED HUMAN 3H-5-CT 4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 4879 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92991 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 9398 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92992 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 9483 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92993 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92994 5-HT7 CLONED HUMAN 3H-5-CT (RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine >10000 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92995 5-HT7 CLONED HUMAN 3H-5-CT 4-[3-(2,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 1904 Sudol S et al 2020 Jan 15, 2025 Jan 15, 2025
92996 D2 CLONED HUMAN 3H-RACLOPRIDE WA-13 1001 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
92997 D2 CLONED HUMAN 3H-RACLOPRIDE RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine (2) 1506 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
92998 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 432 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
92999 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 421 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93000 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 495 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93001 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 506 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93002 D2 CLONED HUMAN 3H-RACLOPRIDE 4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine 206 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93003 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine 375 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93004 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 320 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93005 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 229 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93006 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 103 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93007 D2 CLONED HUMAN 3H-RACLOPRIDE 4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 413 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93008 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride 754 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93009 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 580 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93010 D2 CLONED HUMAN 3H-RACLOPRIDE 4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine 356 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93011 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine 157 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93012 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 368 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93013 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 377 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93014 D2 CLONED HUMAN 3H-RACLOPRIDE (RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine 270 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93015 D2 CLONED HUMAN 3H-RACLOPRIDE OLANZAPINE 9 Sudol S et al 2020 Jan 15, 2025 Jan 28, 2025
93016 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 67 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93017 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93018 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93019 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 481 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93020 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 25 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93021 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 11.5 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93022 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines 785 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93023 A1 CLONED HUMAN 3H-DPCPX 7-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93024 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93025 A1 CLONED HUMAN 3H-DPCPX 7-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93026 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 153 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93027 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93028 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 415 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93029 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 71 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93030 A1 CLONED HUMAN 3H-DPCPX 7-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 647 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93031 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 162 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93032 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 518 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93033 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 204 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93034 A1 CLONED HUMAN 3H-DPCPX 7-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine 193 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93035 A1 CLONED HUMAN 3H-DPCPX 7-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine 580 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93036 A1 CLONED HUMAN 3H-DPCPX Tert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate 615 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93037 A1 CLONED HUMAN 3H-DPCPX 2-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine 92 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93038 A1 CLONED HUMAN 3H-DPCPX 7-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93039 A1 CLONED HUMAN 3H-DPCPX 7-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine 429 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93040 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 412 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93041 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93042 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93043 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93044 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-benzylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 123 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93045 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93046 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93047 A2A CLONED HUMAN 3H-ZM241385 7-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93048 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93049 A2A CLONED HUMAN 3H-ZM241385 7-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93050 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93051 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 150 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93052 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 189 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93053 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 238 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93054 A2A CLONED HUMAN 3H-ZM241385 7-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93055 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93056 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93057 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93058 A2A CLONED HUMAN 3H-ZM241385 7-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93059 A2A CLONED HUMAN 3H-ZM241385 7-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93060 A2A CLONED HUMAN 3H-ZM241385 Tert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93061 A2A CLONED HUMAN 3H-ZM241385 2-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93062 A2A CLONED HUMAN 3H-ZM241385 7-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93063 A2A CLONED HUMAN 3H-ZM241385 7-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93064 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 13 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93065 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 27 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93066 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 61 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93067 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93068 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-benzylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 28 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93069 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93070 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93071 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93072 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93073 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93074 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93075 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93076 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93077 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93078 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93079 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93080 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93081 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93082 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93083 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93084 A3 CLONED HUMAN 125I-AB-MECA Tert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93085 A3 CLONED HUMAN 125I-AB-MECA 2-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93086 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93087 A3 CLONED HUMAN 125I-AB-MECA 7-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine 1000 Squarcialupi L et al 2017 Jan 15, 2025 Jan 15, 2025
93088 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93089 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-(6-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93090 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93091 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93092 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93093 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93094 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93095 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93096 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93097 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine 1400 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93098 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93099 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93100 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-(6-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93101 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93102 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93103 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93104 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine 2500 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93105 Sigma 2 liver membranes RAT 3H-DTG (±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine 5800 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93106 Sigma 2 liver membranes RAT 3H-DTG (±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93107 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93108 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93109 Sigma 2 liver membranes RAT 3H-DTG (±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93110 Sigma 2 liver membranes RAT 3H-DTG (±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93111 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93112 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93113 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93114 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine 893 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93115 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine 413 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93116 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine 712 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93117 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93118 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93119 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93120 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 ((±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93121 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93122 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (S)-(+)-ketamine 419 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93123 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 PCP 28 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93124 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 Dexoxadrol 19 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93125 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 Etoxadrol 22 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93126 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93127 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93128 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93129 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93130 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93131 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93132 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93133 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93134 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93135 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93136 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93137 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93138 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93139 NMDA CORTICAL MEMBRANES PIG 3H-MK-801 (±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 15, 2025
93140 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine 155 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93141 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine 542 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93142 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine 543 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93143 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine 607 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93144 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine 1500 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93145 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine 2700 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93146 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine 4900 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93147 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine 502 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93148 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine 192 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93149 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine 37 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93150 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine 7.37 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93151 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine 297 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93152 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine 314 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93153 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) (±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine 3000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93154 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) PENTAZOCINE (+) 6.03 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93155 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93156 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine 4300 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93157 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93158 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93159 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine 4900 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93160 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93161 Sigma 2 liver membranes RAT 3H-DTG (±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine 1600 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93162 Sigma 2 liver membranes RAT 3H-DTG (±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93163 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine 698 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93164 Sigma 2 liver membranes RAT 3H-DTG (±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine >10000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93165 Sigma 2 liver membranes RAT 3H-DTG (±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine 1000 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93166 Sigma 2 liver membranes RAT 3H-DTG (±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine 841 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93167 Sigma 2 liver membranes RAT 3H-DTG (±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine 174 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93168 Sigma 2 liver membranes RAT 3H-DTG (±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine 111 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93169 Sigma 2 liver membranes RAT 3H-DTG DTG 64 Bonifazi A et al 2015 Jan 15, 2025 Jan 28, 2025
93170 D1 CHO cells PORCINE 3H-SPIPERONE 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 6400 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93171 D2 CHO cells HUMAN 3H-SPIPERONE 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 95 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93172 D2 CHO cells HUMAN 3H-SPIPERONE 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 76 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93173 D3 CHO cells HUMAN 3H-SPIPERONE 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 370 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93174 D4 CHO cells HUMAN 3H-SPIPERONE 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 9.5 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93175 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 680 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93176 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 2100 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93177 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine 230 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93178 D1 CHO cells PORCINE 3H-SPIPERONE 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1300 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93179 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 65 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93180 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 67 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93181 D3 CHO cells HUMAN 3H-SPIPERONE 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 210 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93182 D4 CHO cells HUMAN 3H-SPIPERONE 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 16 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93183 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 770 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93184 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1000 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93185 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 370 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93186 D1 CHO cells PORCINE 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1400 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93187 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 76 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93188 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 60 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93189 D3 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 370 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93190 D4 CHO cells HUMAN 3H-SPIPERONE 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 19 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93191 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 410 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93192 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1300 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93193 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 210 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93194 D1 CHO cells PORCINE 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 860 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93195 D2 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 150 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93196 D2 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 68 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93197 D3 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 580 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93198 D4 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 0.71 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93199 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 120 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93200 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 990 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93201 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 57 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93202 CEREBRAL CORTEX PORCINE 3H-RX821002 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 44 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93203 H1 Sf9 HUMAN 3H-MEPYRAMINE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol 1400 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93204 5-HT1D Sf9 HUMAN 3H-UR-DE257 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93205 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93206 H4 Sf9 HUMAN 3H-UR-PI294 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93207 D1 CHO cells PORCINE 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 410 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93208 D2 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 8.3 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93209 D2 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 39 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93210 D3 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 530 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93211 D4 CHO cells HUMAN 3H-SPIPERONE 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 2.4 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93212 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 110 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93213 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 380 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93214 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril 31 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93215 D1 CHO cells PORCINE 3H-SPIPERONE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 4500 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93216 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 210 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93217 D2 CHO cells HUMAN 3H-SPIPERONE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 140 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93218 D3 CHO cells HUMAN 3H-SPIPERONE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 390 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93219 D4 CHO cells HUMAN 3H-SPIPERONE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1.5 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93220 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 110 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93221 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 1800 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93222 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 33 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93223 CEREBRAL CORTEX PORCINE 3H-RX821002 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 23 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93224 H1 Sf9 HUMAN 3H-MEPYRAMINE 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 2600 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93225 5-HT1D Sf9 HUMAN 3H-UR-DE247 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine 3200 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93226 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93227 H4 Sf9 HUMAN 3H-UR-PI294 1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93228 D1 CHO cells PORCINE 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 4100 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93229 D2 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 51 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93230 D2 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 37 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93231 D3 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 160 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93232 D4 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 1.9 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93233 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 65 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93234 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 1300 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93235 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 32 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93236 CEREBRAL CORTEX PORCINE 3H-RX821002 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 140 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93237 H1 Sf9 HUMAN 3H-MEPYRAMINE 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 5500 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93238 5-HT1D Sf9 HUMAN 3H-UR-DE257 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine 4200 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93239 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93240 H4 Sf9 HUMAN 3H-UR-PI294 1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93241 D1 CHO cells PORCINE 3H-SPIPERONE 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 5000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93242 D2 CHO cells HUMAN 3H-SPIPERONE 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 130 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93243 D2 CHO cells HUMAN 3H-SPIPERONE 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 92 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93244 D3 CHO cells HUMAN 3H-SPIPERONE 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 350 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93245 D4 CHO cells HUMAN 3H-SPIPERONE 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 4.6 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93246 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 99 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93247 CEREBRAL CORTEX PORCINE 3H-KETANSERIN 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 1000 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93248 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 57 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93249 CEREBRAL CORTEX PORCINE 3H-RX821002 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 220 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93250 H1 Sf9 HUMAN 3H-MEPYRAMINE 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 6500 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93251 5-HT1D Sf9 HUMAN 3H-UR-DE257 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine 6100 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93252 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93253 H4 Sf9 HUMAN 3H-UR-PI294 4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93254 D1 CHO cells PORCINE 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 6400 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93255 D2 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 60 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93256 D2 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 57 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93257 D3 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 460 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93258 D4 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 3.8 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93259 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 91 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93260 CEREBRAL CORTEX PORCINE 3H-WAY100635 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 2100 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93261 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 66 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93262 CEREBRAL CORTEX PORCINE 3H-RX821002 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 170 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93263 H1 Sf9 HUMAN 3H-MEPYRAMINE 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93264 5-HT1D Sf9 HUMAN 3H-UR-DE257 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 5500 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93265 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine 5500 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93266 H4 Sf9 HUMAN 3H-UR-PI294 1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93267 D1 CHO cells PORCINE 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 740 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93268 D2 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 17 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93269 D2 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 34 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93270 D3 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 33 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93271 D4 CHO cells HUMAN 3H-SPIPERONE 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 0.79 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93272 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 100 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93273 CEREBRAL CORTEX PORCINE 3H- Ketanserin 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 560 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93274 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 8.3 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93275 CEREBRAL CORTEX PORCINE 3H-RX821002 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 120 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93276 H1 Sf9 HUMAN 3H-MEPYRAMINE 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93277 5-HT1D Sf9 HUMAN 3H-UR-DE257 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 530 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93278 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93279 H4 Sf9 HUMAN 3H-UR-PI294 1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93280 D1 CHO cells PORCINE 3H-SPIPERONE 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1100 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93281 D2 CHO cells HUMAN 3H-SPIPERONE 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 95 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93282 D2 CHO cells HUMAN 3H-SPIPERONE 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 160 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93283 D3 CHO cells HUMAN 3H-SPIPERONE 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 85 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93284 D4 CHO cells HUMAN 3H-SPIPERONE 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 6 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93285 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 760 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93286 CEREBRAL CORTEX PORCINE 3H- Ketanserin 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1600 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93287 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 27 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93288 CEREBRAL CORTEX PORCINE 3H-RX821002 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1200 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93289 H1 Sf9 HUMAN 3H-MEPYRAMINE 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 490 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93290 5-HT1D Sf9 HUMAN 3H-DE257 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 460 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93291 H3 Sf9 HUMAN 3H-N-alpha-methylhistamine 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine >10000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93292 H4 Sf9 HUMAN 3H-UR-PI294 1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine 1000 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93293 D1 CHO cells PORCINE 3H-SPIPERONE FAUC 3019 500 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93294 D2 CHO cells HUMAN 3H-SPIPERONE FAUC 3019 33 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93295 D2 CHO cells HUMAN 3H-SPIPERONE FAUC 3019 24 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93296 D3 CHO cells HUMAN 3H-SPIPERONE FAUC 3019 83 Lober S et al 2012 Jan 15, 2025 Jan 28, 2025
93297 D4 CHO cells HUMAN 3H-SPIPERONE FAUC 3019 0.4 Lober S et al 2012 Jan 15, 2025 Jan 29, 2025
93298 5-HT1A CEREBRAL CORTEX PORCINE 3H-WAY100635 FAUC 3019 54 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93299 CEREBRAL CORTEX PORCINE 3H- Ketanserin FAUC 3019 92 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93300 CEREBRAL CORTEX PORCINE 3H-PRAZOSIN FAUC 3019 20 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93301 CEREBRAL CORTEX PORCINE 3H-RX821002 FAUC 3019 39 Lober S et al 2012 Jan 15, 2025 Jan 15, 2025
93302 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 1,3,7-Trimethyl-8-[3-(4-phenyl-1-piperazinyl)- propylamino]-purine-2,6-dione hydrochloride 385 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93303 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT 1,3-Dimethyl-7-n-butyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione hydrochloride 100 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93304 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT Ethyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-acetic acid hydrochloride 592 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93305 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT Ethyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-butyric acid 457 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93306 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT N-[(4-Phenyl-1-piperazinyl)-propyl]-3-phenylpyrrolidine-2,5-dione dihydrochloride 1069 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93307 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT N-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride 177 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93308 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT N-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-chlorophenyl)-pyrrolidine-2,5-dione dihydrochloride 258 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93309 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT N-[(4-Phenyl-1-piperazinyl)-propyl]-3-(4-fluorophenyl)-pyrrolidine-2,5-dione dihydrochloride 223 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93310 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT N-[(4-Phenyl-1-piperazinyl)-propyl-3-(4-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride 510 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93311 5-HT1A HIPPOCAMPUS RAT 3H-8-OH-DPAT N-[(4-Phenyl-1-piperazinyl)-propyl]-3,3- diphenyl-pyrrolidine-2,5-dione dihydrochloride 444 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93312 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN N-[(4-Phenyl-1-piperazinyl)-propyl]-3,3- diphenyl-pyrrolidine-2,5-dione dihydrochloride 842 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93313 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN N-[(4-Phenyl-1-piperazinyl)-propyl-3-(4-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride 436 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93314 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN N-[(4-Phenyl-1-piperazinyl)-propyl]-3-(4-fluorophenyl)-pyrrolidine-2,5-dione dihydrochloride 436 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93315 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN N-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-chlorophenyl)-pyrrolidine-2,5-dione dihydrochloride 388 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93316 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN N-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride 329 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93317 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN N-[(4-Phenyl-1-piperazinyl)-propyl]-3-phenylpyrrolidine-2,5-dione dihydrochloride 268 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93318 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN Ethyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-butyric acid 1010 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93319 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN Ethyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-acetic acid hydrochloride 179 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93320 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN 1,3-Dimethyl-7-n-butyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione hydrochloride 614 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93321 5-HT2A BRAIN CORTEX RAT 3H-KETANSERIN 1,3,7-Trimethyl-8-[3-(4-phenyl-1-piperazinyl)- propylamino]-purine-2,6-dione hydrochloride 197 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93322 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 39 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93323 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 68 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93324 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 20 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93325 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 4.3 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93326 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 4.5 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93327 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 4.5 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93328 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 25 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93329 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 66 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93330 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 18 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93331 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride 204 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93332 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 146 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93333 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride 488 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93334 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 354 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93335 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 56 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93336 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 104 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93337 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 70 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93338 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 15 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93339 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 20 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93340 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 133 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93341 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride 899 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93342 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 230 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93343 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride 7.6 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93344 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 64 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93345 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 48 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93346 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 477 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93347 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 151 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93348 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 631 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93349 5-HT1A CORTICAL MEMBRANES RAT 3H-8-OH-DPAT 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 34 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93350 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 259 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93351 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 298 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93352 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 116 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93353 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 162 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93354 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 400 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93355 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 179 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93356 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 68 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93357 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 115 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93358 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 114 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93359 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride 428 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93360 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 3517 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93361 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride 1789 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93362 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 574 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93363 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 2335 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93364 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 269 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93365 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 302 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93366 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 1411 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93367 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 475 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93368 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 72 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93369 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride 902 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93370 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93371 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride 348 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93372 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 154 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93373 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 480 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93374 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 388 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93375 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 398 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93376 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 80 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93377 5-HT2A HIPPOCAMPUS RAT 3H-KETANSERIN 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 210 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93378 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93379 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93380 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 958 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93381 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93382 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93383 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93384 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93385 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 911 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93386 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 98 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93387 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93388 5-HT6 CLONED HUMAN 3H-5-CT 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93389 5-HT6 CLONED HUMAN 3H-5-CT 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93390 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93391 5-HT6 CLONED HUMAN 3H-5-CT 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93392 5-HT6 CLONED HUMAN 3H-5-CT 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93393 5-HT6 CLONED HUMAN 3H-5-CT 7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 5706 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93394 5-HT6 CLONED HUMAN 3H-5-CT 7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93395 5-HT6 CLONED HUMAN 3H-5-CT 7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93396 5-HT6 CLONED HUMAN 3H-5-CT 7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93397 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93398 5-HT6 CLONED HUMAN 3H-5-CT 8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93399 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93400 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93401 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93402 5-HT6 CLONED HUMAN 3H-5-CT 7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93403 5-HT6 CLONED HUMAN 3H-5-CT 1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93404 5-HT6 CLONED HUMAN 3H-5-CT 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 1000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93405 5-HT6 CLONED HUMAN 3H-5-CT 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 717 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93406 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 90 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93407 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 25 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93408 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 36 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93409 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 40 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93410 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 10 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93411 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 20 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93412 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 65 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93413 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 113 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93414 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 85 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93415 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride 454 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93416 5-HT7 CLONED HUMAN 3H-LSD 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 3590 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93417 5-HT7 CLONED HUMAN 3H-LSD 8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride >10000 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93418 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride 302 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93419 5-HT7 CLONED HUMAN 3H-LSD 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride 99 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93420 5-HT7 CLONED HUMAN 3H-LSD 8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 239 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93421 5-HT7 CLONED HUMAN 3H-LSD 7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride 476 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93422 5-HT7 CLONED HUMAN 3H-LSD 7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 274 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93423 5-HT7 CLONED HUMAN 3H-LSD 7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 622 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93424 5-HT7 CLONED HUMAN 3H-LSD 7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride 269 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93425 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride 1200 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93426 5-HT7 CLONED HUMAN 3H-LSD 8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 740 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93427 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride 89 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93428 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 165 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93429 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 75 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93430 5-HT7 CLONED HUMAN 3H-LSD 7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 295 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93431 5-HT7 CLONED HUMAN 3H-LSD 1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride 936 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93432 5-HT7 CLONED HUMAN 3H-LSD 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride 105 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93433 5-HT7 CLONED HUMAN 3H-LSD 8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride 63 Chlon-Rzepa G et al 2013 Jan 15, 2025 Jan 15, 2025
93434 A1 C.H.O. ? HUMAN 3H-CCPA 6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93435 A1 C.H.O. ? HUMAN 3H-CCPA 6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 8200 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93436 A1 C.H.O. ? HUMAN 3H-CCPA 6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93437 A1 C.H.O. ? HUMAN 3H-CCPA 6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93438 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate 8800 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93439 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate 900 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93440 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate 4000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93441 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate 3500 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93442 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93443 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93444 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93445 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93446 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate 4300 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93447 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 2800 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93448 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93449 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 700 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93450 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 2700 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93451 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate 5100 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93452 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate 5000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93453 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate 2500 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93454 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93455 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate 2600 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93456 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93457 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93458 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93459 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93460 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93461 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93462 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate 5900 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93463 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 600 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93464 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 2700 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93465 A1 C.H.O. ? HUMAN 3H-CCPA Ethyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 600 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93466 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 2400 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93467 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93468 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93469 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 5700 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93470 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 8800 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93471 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93472 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93473 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate 7300 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93474 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93475 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93476 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93477 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93478 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93479 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93480 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93481 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93482 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93483 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93484 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93485 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93486 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate 4200 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93487 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93488 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93489 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate 6000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93490 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate 7500 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93491 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93492 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93493 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate 6100 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93494 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate 3700 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93495 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93496 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93497 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 5700 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93498 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 2300 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93499 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93500 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93501 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93502 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93503 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate 2800 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93504 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate 3300 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93505 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93506 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93507 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93508 A2A CHO cells ? HUMAN 3H-NECA Ethyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93509 A2B CHO cells ? HUMAN 3H-NECA Ethyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93510 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93511 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93512 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93513 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93514 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate 4800 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93515 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93516 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93517 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate 5000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93518 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate 2600 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93519 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93520 A2B CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93521 A2A CHO cells ? HUMAN 3H-NECA Ethyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate 2000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93522 A2A CHO cells ? HUMAN 3H-NECA 6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93523 A2B CHO cells ? HUMAN 3H-NECA 6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93524 A2B CHO cells ? HUMAN 3H-NECA 6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93525 A2A CHO cells ? HUMAN 3H-NECA 6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93526 A2A CHO cells ? HUMAN 3H-NECA 6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 9200 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93527 A2B CHO cells ? HUMAN 3H-NECA 6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93528 A2B CHO cells ? HUMAN 3H-NECA 6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93529 A2A CHO cells ? HUMAN 3H-NECA 6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide 3000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93530 A3 CHO cells ? HUMAN 3H-HEMADO 6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93531 A3 CHO cells ? HUMAN 3H-HEMADO 6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93532 A3 CHO cells ? HUMAN 3H-HEMADO 6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93533 A3 CHO cells ? HUMAN 3H-HEMADO 6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93534 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate 900 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93535 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93536 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93537 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93538 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93539 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93540 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93541 A3 CHO cells ? HUMAN 3H-HEMADO Ethyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate >10000 Venkatesan G et al 2015 Jan 15, 2025 Jan 15, 2025
93542 A1 CLONED HUMAN 3H-CCPA N2 -benzyl-9-propyl-9H-purine-2,6-diamine 7600 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93543 A2A CLONED HUMAN 3H-NECA N2 -benzyl-9-propyl-9H-purine-2,6-diamine 1400 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93544 A3 CLONED HUMAN 3H-HEMADO N2 -benzyl-9-propyl-9H-purine-2,6-diamine 5840 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93545 A3 CLONED HUMAN 3H-HEMADO N2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine 650 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93546 A2A CLONED HUMAN 3H-NECA N2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine 36 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93547 A1 CLONED HUMAN 3H-CCPA N2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine 358 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93548 A1 CLONED HUMAN 3H-CCPA N2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine 138 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93549 A2A CLONED HUMAN 3H-NECA N2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine 6.6 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93550 A3 CLONED HUMAN 3H-HEMADO N2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine 29 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93551 A3 CLONED HUMAN 3H-HEMADO N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 5880 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93552 A2A CLONED HUMAN 3H-NECA N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 738 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93553 A1 CLONED HUMAN 3H-CCPA N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 2330 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93554 A1 CLONED HUMAN 3H-CCPA 8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 373 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93555 A2A CLONED HUMAN 3H-NECA 8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 27 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93556 A3 CLONED HUMAN 3H-HEMADO 8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 1160 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93557 A3 CLONED HUMAN 3H-HEMADO 8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 56 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93558 A2A CLONED HUMAN 3H-NECA 8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 14 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93559 A1 CLONED HUMAN 3H-CCPA 8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine 80.3 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93560 A1 CLONED HUMAN 3H-CCPA N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 3640 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93561 A2A CLONED HUMAN 3H-NECA N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 9110 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93562 A3 CLONED HUMAN 3H-HEMADO N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93563 A3 CLONED HUMAN 3H-HEMADO 8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 1950 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93564 A2A CLONED HUMAN 3H-NECA 8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 284 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93565 A1 CLONED HUMAN 3H-CCPA 8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 583 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93566 A1 CLONED HUMAN 3H-CCPA 8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 230 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93567 CLONED HUMAN 3H-NECA 8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 113 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93568 A3 CLONED HUMAN 3H-HEMADO 8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine 266 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93569 A3 CLONED HUMAN 3H-HEMADO N-benzyl-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93570 A2A CLONED HUMAN 3H-NECA N-benzyl-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93571 A1 CLONED HUMAN 3H-CCPA N-benzyl-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93572 A1 CLONED HUMAN 3H-CCPA N-benzyl-8-bromo-9-propyl-9H-purin-6-amine 5620 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93573 A2A CLONED HUMAN 3H-NECA N-benzyl-8-bromo-9-propyl-9H-purin-6-amine 1180 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93574 A3 CLONED HUMAN 3H-HEMADO N-benzyl-8-bromo-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93575 A3 CLONED HUMAN 3H-HEMADO N-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine 402 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93576 A2A CLONED HUMAN 3H-NECA N-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine 80 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93577 A1 CLONED HUMAN 3H-CCPA N-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine 546 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93578 A1 CLONED HUMAN 3H-CCPA N-phenethyl-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93579 A2A CLONED HUMAN 3H-NECA N-phenethyl-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93580 A3 CLONED HUMAN 3H-HEMADO N-phenethyl-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93581 A3 CLONED HUMAN 3H-HEMADO 8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine 2520 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93582 A2A CLONED HUMAN 3H-NECA 8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine 503 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93583 A1 CLONED HUMAN 3H-CCPA 8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine 1940 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93584 A1 CLONED HUMAN 3H-CCPA 8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine 2440 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93585 A2A CLONED HUMAN 3H-NECA 8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine 547 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93586 A3 CLONED HUMAN 3H-HEMADO 8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine 811 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93587 A3 CLONED HUMAN 3H-HEMADO N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93588 A2A CLONED HUMAN 3H-NECA N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93589 A1 CLONED HUMAN 3H-CCPA N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93590 A1 CLONED HUMAN 3H-CCPA 8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 2670 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93591 A2A CLONED HUMAN 3H-NECA 8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 1020 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93592 A3 CLONED HUMAN 3H-HEMADO 8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine >10000 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93593 A3 CLONED HUMAN 3H-HEMADO 8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 959 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93594 A2A CLONED HUMAN 3H-NECA 8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 181 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93595 A1 CLONED HUMAN 3H-CCPA 8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine 378 Lambertucci C et al 2015 Jan 15, 2025 Jan 15, 2025
93596 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 2604 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93597 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 1536 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93598 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 1311 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93599 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 417 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93600 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 8269 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93601 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate >10000 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93602 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 433 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93603 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 1029 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93604 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 879 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93605 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 145 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93606 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 309 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93607 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 574 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93608 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 1352 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93609 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 158 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93610 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate >10000 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93611 Sigma 2 LIVER RAT 3H-DTG 7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate >10000 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93612 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate 3087 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93613 D4 CLONED HUMAN 125I-IABN 7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate 865 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93614 D3 CLONED HUMAN 125I-IABN 7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate 427 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93615 D2 CLONED HUMAN 125I-IABN 7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate 611 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93616 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 0.22 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93617 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 13.1 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93618 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 212 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93619 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 1176 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93620 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 598 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93621 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 4988 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93622 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate >10000 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93623 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 185 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93624 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 13.5 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93625 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate 0.26 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93626 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 102 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93627 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 930 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93628 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 359 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93629 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 170 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93630 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 665 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93631 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 3340 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93632 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 620 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93633 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 286 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93634 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 785 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93635 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 25.3 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93636 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 4.6 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93637 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 251 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93638 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 27.2 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93639 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 377 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93640 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate 6393 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93641 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 1309 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93642 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 2631 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93643 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 30.1 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93644 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 5.4 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93645 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 0.14 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93646 D2 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 0.07 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93647 D3 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 2.7 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93648 D4 CLONED HUMAN 125I-IABN 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 31.9 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93649 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate >10000 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93650 Sigma 2 LIVER RAT 3H-DTG 7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate 4952 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93651 Sigma 2 LIVER RAT 3H-DTG 7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 1907 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93652 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 759 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93653 D4 CLONED HUMAN 125I-IABN 7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 38.5 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93654 D3 CLONED HUMAN 125I-IABN 7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 7.4 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93655 D2 CLONED HUMAN 125I-IABN 7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate 4.8 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93656 D2 CLONED HUMAN 125I-IABN 7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate 2.6 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93657 D3 CLONED HUMAN 125I-IABN 7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate 5.7 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93658 D4 CLONED HUMAN 125I-IABN 7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate 52.7 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93659 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate 2600 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93660 Sigma 2 LIVER RAT 3H-DTG 7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate 2838 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93661 Sigma 2 LIVER RAT 3H-DTG 7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate 231 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93662 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate 1349 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93663 D4 CLONED HUMAN 125I-IABN 7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate 234 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93664 D3 CLONED HUMAN 125I-IABN 7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate 7 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93665 D2 CLONED HUMAN 125I-IABN 7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate 7.3 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93666 D2 CLONED HUMAN 125I-IABN 7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate 7.4 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93667 D3 CLONED HUMAN 125I-IABN 7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate 3.8 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93668 D4 CLONED HUMAN 125I-IABN 7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate 201 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93669 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate 1614 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93670 Sigma 2 LIVER RAT 3H-DTG 7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate 608 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93671 D4 CLONED HUMAN 125I-IABN ARIPIPRAZOLE 168 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93672 D3 CLONED HUMAN 125I-IABN ARIPIPRAZOLE 6.8 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93673 D2 CLONED HUMAN 125I-IABN ARIPIPRAZOLE 3.1 Vangveravong S et al 2011 Jan 15, 2025 Jan 28, 2025
93674 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester 744 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93675 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester 86.5 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93676 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester 2.75 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93677 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester 7.21 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93678 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester 114 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93679 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester 277 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93680 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester 48.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93681 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester 197 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93682 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester 1.99 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93683 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester 30.6 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93684 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester 37.2 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93685 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester 93.9 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93686 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester 79.7 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93687 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester 21 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93688 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester 10.8 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93689 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester 3.72 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93690 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester 62.2 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93691 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester 190 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93692 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester 55.2 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93693 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester 13.2 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93694 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester 1.71 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93695 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester 7.42 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93696 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester 14.9 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93697 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester 34.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93698 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 102 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93699 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 194 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93700 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester 5.62 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93701 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 6.05 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93702 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 32 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93703 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester 348 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93704 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 26.4 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93705 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 15.7 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93706 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester 6.73 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93707 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester 4.88 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93708 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester 71.9 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93709 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester 216 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93710 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester 313 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93711 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester 24.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93712 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester 14.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93713 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester 3.37 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93714 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester 32.5 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93715 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester 130 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93716 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester 556 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93717 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester 71.5 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93718 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester 5.21 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93719 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester 1.21 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93720 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester 21 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93721 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester 119 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93722 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester 51 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93723 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester 11 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93724 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester 3.19 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93725 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 3.73 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93726 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 18.6 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93727 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide 23.4 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93728 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide 28.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93729 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide 61.6 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93730 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide 5.08 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93731 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide 5.02 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93732 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide 100 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93733 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide 46.6 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93734 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide 41 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93735 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide 81.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93736 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide 12.5 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93737 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide 15.3 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93738 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide 2950 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93739 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide 3850 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93740 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide 137 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93741 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide 59.4 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93742 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide 10 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93743 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide 7.23 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93744 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide 47.6 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93745 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide 250 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93746 A1 CLONED HUMAN 3H-CCPA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide >10000 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93747 A2A CLONED HUMAN 3H-NECA 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide 9390 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025
93748 A3 CLONED HUMAN 3H-HEMADO 2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide 521 Federico S et al 2018 Jan 15, 2025 Jan 15, 2025