The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

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Showing 90,001-91,000 of 98,686 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
92749Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13:15,16-diepoxylabdane-6b,15a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92750Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13:15,16-diepoxylabdane-6b,16b-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92751Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13:15,16-diepoxylabdane-6b,16a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92752Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13-epoxylabd-5-en-7-on-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92753Sigma 1CLONEDHUMAN M33H-Pentazocine(+)15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92754Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13-epoxy-15,16-dihydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92755Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13-epoxylabd-5-ene-7 b,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92756Sigma 1CLONEDHUMAN M33H-Pentazocine(+)(8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92757Sigma 1CLONEDHUMAN M33H-Pentazocine(+)15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92758Sigma 1CLONEDHUMAN M33H-Pentazocine(+)9,13-epoxy-6-hydroxylabdan-15,16-olide2900Wu H et al 2013Jan 15, 2025Jan 28, 2025
92759Sigma 2CLONEDHUMAN M33H-DTG(5S,6R,8R,9R,10S,13S)-9,13-epoxylabdane-6,15,16- triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92760Sigma 2CLONEDHUMAN M33H-DTG9,13:15,16-diepoxylabdane-6b,15a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92761Sigma 2CLONEDHUMAN M33H-DTG9,13:15,16-diepoxylabdane-6b,16b-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92762Sigma 2CLONEDHUMAN M33H-DTG9,13:15,16-diepoxylabdane-6b,16a-diol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92763Sigma 2CLONEDHUMAN M33H-DTG9,13-epoxylabd-5-en-7-on-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92764Sigma 2CLONEDHUMAN M33H-DTG15-acetoxy-9,13-epoxy-16-hydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92765Sigma 2CLONEDHUMAN M33H-DTG9,13-epoxy-15,16-dihydroxylabd-5-en-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92766Sigma 2CLONEDHUMAN M33H-DTG9,13-epoxylabd-5-ene-7 b,15,16-triol>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92767Sigma 2CLONEDHUMAN M33H-DTG(8S,9R,10S)-15,16-epoxy-9a-hydroxylabda-5,13(16), 14-trien-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92768Sigma 2CLONEDHUMAN M33H-DTG15,16-epoxylabda-5,8,13(16),14-tetraen-7-one>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92769Sigma 2CLONEDHUMAN M33H-DTG9,13-epoxy-6-hydroxylabdan-15,16-olide>10000Wu H et al 2013Jan 15, 2025Jan 28, 2025
92770A1CLONEDHUMAN3H-PIA2-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine1620Yu J et al 2017Jan 15, 2025Jan 15, 2025
92771A1CLONEDHUMAN3H-PIAthio-Cl-IB-MECA20.2Yu J et al 2017Jan 15, 2025Jan 15, 2025
92772A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide3310Yu J et al 2017Jan 15, 2025Jan 15, 2025
92773A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide570Yu J et al 2017Jan 15, 2025Jan 15, 2025
92774A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide220Yu J et al 2017Jan 15, 2025Jan 15, 2025
92775A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide480Yu J et al 2017Jan 15, 2025Jan 15, 2025
92776A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide1880Yu J et al 2017Jan 15, 2025Jan 15, 2025
92777A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1090Yu J et al 2017Jan 15, 2025Jan 15, 2025
92778A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide440Yu J et al 2017Jan 15, 2025Jan 15, 2025
92779A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carboxamide420Yu J et al 2017Jan 15, 2025Jan 15, 2025
92780A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide83.5Yu J et al 2017Jan 15, 2025Jan 15, 2025
92781A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide37.5Yu J et al 2017Jan 15, 2025Jan 15, 2025
92782A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide25.2Yu J et al 2017Jan 15, 2025Jan 15, 2025
92783A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide2060Yu J et al 2017Jan 15, 2025Jan 15, 2025
92784A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92785A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide232Yu J et al 2017Jan 15, 2025Jan 15, 2025
92786A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide156Yu J et al 2017Jan 15, 2025Jan 15, 2025
92787A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide311Yu J et al 2017Jan 15, 2025Jan 15, 2025
92788A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide186Yu J et al 2017Jan 15, 2025Jan 15, 2025
92789A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide61.7Yu J et al 2017Jan 15, 2025Jan 15, 2025
92790A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide59.4Yu J et al 2017Jan 15, 2025Jan 15, 2025
92791A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92792A1CLONEDHUMAN3H-PIA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92793A2ACLONEDHUMAN3H-CGS-216802-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine2910Yu J et al 2017Jan 15, 2025Jan 15, 2025
92794A2ACLONEDHUMAN3H-CGS-21680thio-Cl-IB-MECA475Yu J et al 2017Jan 15, 2025Jan 15, 2025
92795A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1350Yu J et al 2017Jan 15, 2025Jan 15, 2025
92796A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide555Yu J et al 2017Jan 15, 2025Jan 15, 2025
92797A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide560Yu J et al 2017Jan 15, 2025Jan 15, 2025
92798A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide1080Yu J et al 2017Jan 15, 2025Jan 15, 2025
92799A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide1260Yu J et al 2017Jan 15, 2025Jan 15, 2025
92800A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1160Yu J et al 2017Jan 15, 2025Jan 15, 2025
92801A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide195Yu J et al 2017Jan 15, 2025Jan 15, 2025
92802A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carboxamide2480Yu J et al 2017Jan 15, 2025Jan 15, 2025
92803A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92804A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1080Yu J et al 2017Jan 15, 2025Jan 15, 2025
92805A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1090Yu J et al 2017Jan 15, 2025Jan 15, 2025
92806A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92807A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92808A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide238Yu J et al 2017Jan 15, 2025Jan 15, 2025
92809A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide1230Yu J et al 2017Jan 15, 2025Jan 15, 2025
92810A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide1200Yu J et al 2017Jan 15, 2025Jan 15, 2025
92811A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92812A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide899Yu J et al 2017Jan 15, 2025Jan 15, 2025
92813A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide1120Yu J et al 2017Jan 15, 2025Jan 15, 2025
92814A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92815A2ACLONEDHUMAN3H-CGS-21680(2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide>10000Yu J et al 2017Jan 15, 2025Jan 15, 2025
92816A3CLONEDHUMAN125I-AB-MECAthio-Cl-IB-MECA0.25Yu J et al 2017Jan 15, 2025Jan 15, 2025
92817A3CLONEDHUMAN125I-AB-MECA2-chloro-N6 -(3- iodobenzyl)-5′-N-methylcarbamoyladenosine1.8Yu J et al 2017Jan 15, 2025Jan 15, 2025
92818A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-((3-Fluorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide2.3Yu J et al 2017Jan 15, 2025Jan 15, 2025
92819A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-((3-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide3.45Yu J et al 2017Jan 15, 2025Jan 15, 2025
92820A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide0.9Yu J et al 2017Jan 15, 2025Jan 15, 2025
92821A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide0.57Yu J et al 2017Jan 15, 2025Jan 15, 2025
92822A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((2-methoxybenzyl)amino)-9H-purin-9-yl)-Nmethyltetrahydroselenophene-2-carboxamide3.75Yu J et al 2017Jan 15, 2025Jan 15, 2025
92823A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-((2-Chlorobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide4.41Yu J et al 2017Jan 15, 2025Jan 15, 2025
92824A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-((naphthalen-1- ylmethyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2-carboxamide1.76Yu J et al 2017Jan 15, 2025Jan 15, 2025
92825A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(((1R,2R)-2- phenylcyclopropyl)amino)-9H-purin-9-yl)tetrahydroselenophene-2- carboxamide3.93Yu J et al 2017Jan 15, 2025Jan 15, 2025
92826A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-(Cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide2.49Yu J et al 2017Jan 15, 2025Jan 15, 2025
92827A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-(Cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1.39Yu J et al 2017Jan 15, 2025Jan 15, 2025
92828A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-(Cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide7.07Yu J et al 2017Jan 15, 2025Jan 15, 2025
92829A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-3,4-Dihydroxy-N-methyl-5-(6-(methylamino)-9H-purin-9- yl)tetrahydroselenophene-2-carboxamide1.49Yu J et al 2017Jan 15, 2025Jan 15, 2025
92830A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-fluorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide3.35Yu J et al 2017Jan 15, 2025Jan 15, 2025
92831A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-chlorobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide1.96Yu J et al 2017Jan 15, 2025Jan 15, 2025
92832A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(6-((3-Bromobenzyl)amino)-2-chloro-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide1.99Yu J et al 2017Jan 15, 2025Jan 15, 2025
92833A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide4.2Yu J et al 2017Jan 15, 2025Jan 15, 2025
92834A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopropylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide1.9Yu J et al 2017Jan 15, 2025Jan 15, 2025
92835A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclobutylamino)-9H-purin-9-yl)-3,4-dihydroxy-Nmethyltetrahydroselenophene-2-carboxamide1Yu J et al 2017Jan 15, 2025Jan 15, 2025
92836A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxyN-methyltetrahydroselenophene-2-carboxamide3.56Yu J et al 2017Jan 15, 2025Jan 15, 2025
92837A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-3,4-Dihydroxy-5-(6-((3-iodobenzyl)amino)-7H-purin-7-yl)-Nmethyl tetrahydroselenophene-2-carboxamide4180Yu J et al 2017Jan 15, 2025Jan 15, 2025
92838A3CLONEDHUMAN125I-AB-MECA(2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-7H-purin-7-yl)-3,4- dihydroxy-N-methyltetrahydroselenophene-2-carboxamide7360Yu J et al 2017Jan 15, 2025Jan 15, 2025
92839A1CLONEDHUMAN3H-DPCPX5-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92840A1CLONEDHUMAN3H-DPCPX2-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92841A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92842A1CLONEDHUMAN3H-DPCPX2-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92843A1CLONEDHUMAN3H-DPCPX2-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92844A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92845A1CLONEDHUMAN3H-DPCPX2-(4-Hydroxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92846A1CLONEDHUMAN3H-DPCPX4-(5-Methyl-7-oxo-6,7-dihydro-thiazolo[5,4-d]pyrimidin-2- yl)-benzoic acid1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92847A1CLONEDHUMAN3H-DPCPX2-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92848A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92849A1CLONEDHUMAN3H-DPCPX2-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92850A1CLONEDHUMAN3H-DPCPX2-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92851A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92852A1CLONEDHUMAN3H-DPCPX2-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92853A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92854A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92855A1CLONEDHUMAN3H-DPCPX2-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92856A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92857A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92858A1CLONEDHUMAN3H-DPCPX2-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92859A1CLONEDHUMAN3H-DPCPX5-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92860A1CLONEDHUMAN3H-DPCPX2-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92861A1CLONEDHUMAN3H-DPCPX5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92862A1CLONEDHUMAN3H-DPCPX2-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92863A1CLONEDHUMAN3H-DPCPX2-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92864A1CLONEDHUMAN3H-DPCPX5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92865A1CLONEDHUMAN3H-DPCPX2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92866A1CLONEDHUMAN3H-DPCPX2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92867A1CLONEDHUMAN3H-DPCPX7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92868A1CLONEDHUMAN3H-DPCPX7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92869A1CLONEDHUMAN3H-DPCPX2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92870A1CLONEDHUMAN3H-DPCPX7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92871A1CLONEDHUMAN3H-DPCPX7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92872A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92873A2ACLONEDHUMAN3H-ZM2413852-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92874A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92875A2ACLONEDHUMAN3H-ZM2413852-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92876A2ACLONEDHUMAN3H-ZM2413852-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92877A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92878A2ACLONEDHUMAN3H-ZM2413852-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92879A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92880A2ACLONEDHUMAN3H-ZM2413852-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92881A2ACLONEDHUMAN3H-ZM2413852-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92882A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92883A2ACLONEDHUMAN3H-ZM2413852-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92884A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92885A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92886A2ACLONEDHUMAN3H-ZM2413852-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92887A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92888A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92889A2ACLONEDHUMAN3H-ZM2413852-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92890A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92891A2ACLONEDHUMAN3H-ZM2413852-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92892A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-on1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92893A2ACLONEDHUMAN3H-ZM2413852-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92894A2ACLONEDHUMAN3H-ZM2413852-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92895A2ACLONEDHUMAN3H-ZM2413855-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92896A2ACLONEDHUMAN3H-ZM2413852-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92897A2ACLONEDHUMAN3H-ZM2413852-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92898A2ACLONEDHUMAN3H-ZM2413857-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92899A2ACLONEDHUMAN3H-ZM2413857-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92900A2ACLONEDHUMAN3H-ZM2413852-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92901A2ACLONEDHUMAN3H-ZM2413857-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92902A2ACLONEDHUMAN3H-ZM2413857-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92903A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-phenyl-thiazolo[5,4-d]pyrimidin-7-one85Varano F et al 2015Jan 15, 2025Jan 15, 2025
92904A3CLONEDHUMAN125I-AB-MECA2-(4-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one38Varano F et al 2015Jan 15, 2025Jan 15, 2025
92905A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one33Varano F et al 2015Jan 15, 2025Jan 15, 2025
92906A3CLONEDHUMAN125I-AB-MECA2-(4-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one18Varano F et al 2015Jan 15, 2025Jan 15, 2025
92907A3CLONEDHUMAN125I-AB-MECA2-(4-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one107Varano F et al 2015Jan 15, 2025Jan 15, 2025
92908A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(4-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92909A3CLONEDHUMAN125I-AB-MECA2-(4-Hydroxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92910A3CLONEDHUMAN125I-AB-MECA4-(5-Methyl-7-oxo-6,7-dihydro-thiazolo[5,4-d]pyrimidin-2- yl)-benzoic acid1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92911A3CLONEDHUMAN125I-AB-MECA2-(3-Methoxyphenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92912A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(3-methylphenyl)-thiazolo[5,4-d]pyrimidin-7- one384Varano F et al 2015Jan 15, 2025Jan 15, 2025
92913A3CLONEDHUMAN125I-AB-MECA2-(3-Chlorophenyl)-5-methyl-thiazolo[5,4-d]pirimidin-7-one826Varano F et al 2015Jan 15, 2025Jan 15, 2025
92914A3CLONEDHUMAN125I-AB-MECA2-(3-Fluorophenyl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one109Varano F et al 2015Jan 15, 2025Jan 15, 2025
92915A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(3-trifluoromethyl-phenyl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92916A3CLONEDHUMAN125I-AB-MECA2-Benzyl-5-methyl-thiazolo[5,4-d]pyrimidin-7-one427Varano F et al 2015Jan 15, 2025Jan 15, 2025
92917A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(pyridin-3-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92918A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(pyridin-4-yl)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92919A3CLONEDHUMAN125I-AB-MECA2-(Furan-2-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92920A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(thiophen-2-yl)-thiazolo[5,4-d]pyrimidin-7-one248Varano F et al 2015Jan 15, 2025Jan 15, 2025
92921A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(1H-pyrrol-1-yl)-thiazolo[5,4-d]pyrimidin-7-one227Varano F et al 2015Jan 15, 2025Jan 15, 2025
92922A3CLONEDHUMAN125I-AB-MECA2-(1H-Imidazol-1-yl)-5-methyl-thiazolo[5,4-d]pyrimidin-7- one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92923A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-(phenylamino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92924A3CLONEDHUMAN125I-AB-MECA2-((4-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92925A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-((4-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92926A3CLONEDHUMAN125I-AB-MECA2-((4-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92927A3CLONEDHUMAN125I-AB-MECA2-((3-Methoxyphenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one113Varano F et al 2015Jan 15, 2025Jan 15, 2025
92928A3CLONEDHUMAN125I-AB-MECA5-Methyl-2-((3-methylphenyl)amino)-thiazolo[5,4-d]pyrimidin-7-one450Varano F et al 2015Jan 15, 2025Jan 15, 2025
92929A3CLONEDHUMAN125I-AB-MECA2-((3-Chlorophenyl)amino)-5-methyl-thiazolo[5,4-d]pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92930A3CLONEDHUMAN125I-AB-MECA2-((3,4-Dichlorophenyl)amino)-5-methyl-thiazolo[5,4-d] pyrimidin-7-one1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92931A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-5-methyl-2-phenyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92932A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-5-methyl-2-(4-methylphenyl)-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92933A3CLONEDHUMAN125I-AB-MECA2-(4-Chlorophenyl)-7-ethoxy-5-methyl-thiazolo[5,4-d]pyrimidine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92934A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-5-methyl-N-phenyl-thiazolo[5,4-d]pyrimidin-2- amine1000Varano F et al 2015Jan 15, 2025Jan 15, 2025
92935A3CLONEDHUMAN125I-AB-MECA7-Ethoxy-N-(3-methoxyphenyl)-5-methyl-thiazolo[5,4-d] pyrimidin-2-amine110Varano F et al 2015Jan 15, 2025Jan 15, 2025
929365-HT6CLONEDHUMAN3H-LSDWA-1323Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929375-HT6CLONEDHUMAN3H-LSD(RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine21Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929385-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine16Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929395-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine6Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929405-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine23Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929415-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine73Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929425-HT6CLONEDHUMAN3H-LSD4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine274Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929435-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine13Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929445-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine6Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929455-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine12Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929465-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine17Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929475-HT6CLONEDHUMAN3H-LSD4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine470Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929485-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride95Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929495-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine86Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929505-HT6CLONEDHUMAN3H-LSD4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine1061Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929515-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine27Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929525-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine11Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929535-HT6CLONEDHUMAN3H-LSD(RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine26Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929545-HT6CLONEDHUMAN3H-LSD(RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine51Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929555-HT6CLONEDHUMAN3H-LSD4-[3-(2,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine999Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929565-HT6CLONEDHUMAN3H-LSDOLANZAPINE7Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929575-HT2ACLONEDHUMAN3H-KETANSERINWA-131830Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929585-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine5047Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929595-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine268Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929605-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine209Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929615-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine310Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929625-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine470Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929635-HT2ACLONEDHUMAN3H-KETANSERIN4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine649Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929645-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine355Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929655-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine484Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929665-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine382Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929675-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine431Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929685-HT2ACLONEDHUMAN3H-KETANSERIN4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine1457Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929695-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride576Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929705-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine696Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929715-HT2ACLONEDHUMAN3H-KETANSERIN4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine906Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929725-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine412Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929735-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine463Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929745-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine488Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929755-HT2ACLONEDHUMAN3H-KETANSERIN(RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine839Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929765-HT7CLONEDHUMAN3H-5-CTWA-13>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929775-HT7CLONEDHUMAN3H-5-CT(RS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929785-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929795-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine5202Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929805-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929815-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine5265Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929825-HT7CLONEDHUMAN3H-5-CT4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine8592Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929835-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929845-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine5706Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929855-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929865-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine6263Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929875-HT7CLONEDHUMAN3H-5-CT4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine7924Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929885-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride5928Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929895-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine5098Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929905-HT7CLONEDHUMAN3H-5-CT4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine4879Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929915-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine9398Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929925-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine9483Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929935-HT7CLONEDHUMAN3H-5-CT(RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929945-HT7CLONEDHUMAN3H-5-CT(RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine>10000Sudol S et al 2020Jan 15, 2025Jan 15, 2025
929955-HT7CLONEDHUMAN3H-5-CT4-[3-(2,4-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine1904Sudol S et al 2020Jan 15, 2025Jan 15, 2025
92996D2CLONEDHUMAN3H-RACLOPRIDEWA-131001Sudol S et al 2020Jan 15, 2025Jan 28, 2025
92997D2CLONEDHUMAN3H-RACLOPRIDERS)-4-(4-methylpiperazin-1-yl)-6-(1-phenoxypropyl)-1,3,5- triazin-2-amine (2)1506Sudol S et al 2020Jan 15, 2025Jan 28, 2025
92998D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,3-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine432Sudol S et al 2020Jan 15, 2025Jan 28, 2025
92999D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,3-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine421Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93000D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,3-dic hlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine495Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93001D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,3-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine506Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93002D2CLONEDHUMAN3H-RACLOPRIDE4-[3-(2,3-dichlorophenoxy)propyl]-6-(4-methylpiperazin-1- yl)-1,3,5-triazin-2-amine206Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93003D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,5-dichlorophenoxy)ethyl]-6-(4-methylpiperazin1-yl)-1,3,5-triazin-2-amine375Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93004D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine320Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93005D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine229Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93006D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(2,5-dichlorophenoxy)penthyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine103Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93007D2CLONEDHUMAN3H-RACLOPRIDE4-[3-(2,5-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine413Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93008D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(3,4-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine hydrochloride754Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93009D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(3,4-dichlorophenoxy)propyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine580Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93010D2CLONEDHUMAN3H-RACLOPRIDE4-[3-(3,4-dichlorophenoxy)propyl]-6-(4-methylopiperazin1-yl)-1,3,5-triazin-2-amine356Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93011D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(3,5-dichlorophenoxy)ethyl]-6-(4- methylopiperazin-1-yl)-1,3,5-triazin-2-amine157Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93012D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(3,5-dichlorophenoxy)propyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine368Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93013D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4- [1-(3,5-dichlorophenoxy)butyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine377Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93014D2CLONEDHUMAN3H-RACLOPRIDE(RS)-4-[1-(3,5-dichlorophenoxy)pentyl]-6-(4- methylpiperazin-1-yl)-1,3,5-triazin-2-amine270Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93015D2CLONEDHUMAN3H-RACLOPRIDEOLANZAPINE9Sudol S et al 2020Jan 15, 2025Jan 28, 2025
93016A1CLONEDHUMAN3H-DPCPX7-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine67Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93017A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93018A1CLONEDHUMAN3H-DPCPX7-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93019A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine481Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93020A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine25Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93021A1CLONEDHUMAN3H-DPCPX7-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine11.5Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93022A1CLONEDHUMAN3H-DPCPX7-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines785Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93023A1CLONEDHUMAN3H-DPCPX7-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93024A1CLONEDHUMAN3H-DPCPX7-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93025A1CLONEDHUMAN3H-DPCPX7-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93026A1CLONEDHUMAN3H-DPCPX7-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine153Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93027A1CLONEDHUMAN3H-DPCPX7-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93028A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine415Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93029A1CLONEDHUMAN3H-DPCPX7-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine71Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93030A1CLONEDHUMAN3H-DPCPX7-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine647Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93031A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine162Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93032A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine518Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93033A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine204Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93034A1CLONEDHUMAN3H-DPCPX7-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine193Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93035A1CLONEDHUMAN3H-DPCPX7-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine580Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93036A1CLONEDHUMAN3H-DPCPXTert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate615Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93037A1CLONEDHUMAN3H-DPCPX2-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine92Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93038A1CLONEDHUMAN3H-DPCPX7-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93039A1CLONEDHUMAN3H-DPCPX7-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine429Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93040A2ACLONEDHUMAN3H-ZM2413857-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine412Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93041A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93042A2ACLONEDHUMAN3H-ZM2413857-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93043A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93044A2ACLONEDHUMAN3H-ZM2413857-Amino-5-benzylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine123Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93045A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93046A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93047A2ACLONEDHUMAN3H-ZM2413857-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93048A2ACLONEDHUMAN3H-ZM2413857-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93049A2ACLONEDHUMAN3H-ZM2413857-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93050A2ACLONEDHUMAN3H-ZM2413857-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93051A2ACLONEDHUMAN3H-ZM2413857-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine150Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93052A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine189Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93053A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine238Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93054A2ACLONEDHUMAN3H-ZM2413857-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93055A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93056A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93057A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93058A2ACLONEDHUMAN3H-ZM2413857-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93059A2ACLONEDHUMAN3H-ZM2413857-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93060A2ACLONEDHUMAN3H-ZM241385Tert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93061A2ACLONEDHUMAN3H-ZM2413852-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93062A2ACLONEDHUMAN3H-ZM2413857-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93063A2ACLONEDHUMAN3H-ZM2413857-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93064A3CLONEDHUMAN125I-AB-MECA7-Amino-5-phenylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine13Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93065A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-methoxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine27Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93066A3CLONEDHUMAN125I-AB-MECA7-Amino-5–(2,4-dichlorophenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine61Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93067A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-hydroxyphenyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93068A3CLONEDHUMAN125I-AB-MECA7-Amino-5-benzylamino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine28Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93069A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(2-phenylethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93070A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(3-phenylpropyl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidines1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93071A3CLONEDHUMAN125I-AB-MECA7-Amino-2-methyl-5-phenylamino-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93072A3CLONEDHUMAN125I-AB-MECA7-Amino-5-benzylamino-2-methyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93073A3CLONEDHUMAN125I-AB-MECA7-Amino-2-benzyl-5-benzylamino-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93074A3CLONEDHUMAN125I-AB-MECA7-Amino-5-[2–(4-methoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93075A3CLONEDHUMAN125I-AB-MECA7-Amino-5-[2-(3,4-dimethoxyphenyl)ethyl]amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93076A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-hydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93077A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(3,4-dihydroxyphenethyl)amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93078A3CLONEDHUMAN125I-AB-MECA7-Amino-2-phenyl-5-(4-phenylpiperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93079A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93080A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-phenylethylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93081A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-(2,4,6-trifluoro)benzylpiperazin-1-yl)-2-phenyl-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93082A3CLONEDHUMAN125I-AB-MECA7-Amino-5-(4-(2-chloro-4-fluoro)benzylpiperazin-1-yl)-2-phenyl-2Hpyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93083A3CLONEDHUMAN125I-AB-MECA7-Amino-2-phenyl-5-[(4-(2-furoyl)piperazin-1-yl]-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93084A3CLONEDHUMAN125I-AB-MECATert-butyl 4-(7-amino-2-phenyl-2H-pyrazolo[4,3-d]pyrimidin-5-yl)piperazine 1-carboxylate1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93085A3CLONEDHUMAN125I-AB-MECA2-phenyl-5-(4-(methyl-2-furyl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93086A3CLONEDHUMAN125I-AB-MECA7-Amino-2-phenyl-5-(4-(3,3-dimethylbutiryl)piperazin-1-yl)-2H-pyrazolo[4,3-d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93087A3CLONEDHUMAN125I-AB-MECA7-Amino-2-phenyl-5-(4-phenylacetylpiperazin-1-yl)-2H-pyrazolo[4,3- d]pyrimidine1000Squarcialupi L et al 2017Jan 15, 2025Jan 15, 2025
93088Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93089Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93090Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93091Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93092Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93093Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93094Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93095Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93096Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93097Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine1400Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93098Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93099Sigma 2liver membranesRAT3H-DTG(±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93100Sigma 2liver membranesRAT3H-DTG(±)-trans-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93101Sigma 2liver membranesRAT3H-DTG(±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93102Sigma 2liver membranesRAT3H-DTG(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93103Sigma 2liver membranesRAT3H-DTG(±)-cis-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93104Sigma 2liver membranesRAT3H-DTG(±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine2500Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93105Sigma 2liver membranesRAT3H-DTG(±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine5800Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93106Sigma 2liver membranesRAT3H-DTG(±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93107Sigma 2liver membranesRAT3H-DTG(±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93108Sigma 2liver membranesRAT3H-DTG(±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93109Sigma 2liver membranesRAT3H-DTG(±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93110Sigma 2liver membranesRAT3H-DTG(±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93111NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-(6-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93112NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93113NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93114NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(6-Ethyl-6-phenyl-1,4-dioxan-2-yl)methanamine893Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93115NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methanamine413Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93116NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-(6,6-Diphenyl-1,4-dioxan-2-yl)methanamine712Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93117NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-2-(6,6-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93118NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93119NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-(5-Phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93120NMDACORTICAL MEMBRANESPIG3H-MK-801((±)-(5,5-Diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93121NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-2-(5,5-Diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93122NMDACORTICAL MEMBRANESPIG3H-MK-801(S)-(+)-ketamine419Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93123NMDACORTICAL MEMBRANESPIG3H-MK-801PCP28Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93124NMDACORTICAL MEMBRANESPIG3H-MK-801Dexoxadrol19Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93125NMDACORTICAL MEMBRANESPIG3H-MK-801Etoxadrol22Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93126NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93127NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93128NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93129NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93130NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93131NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93132NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93133NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93134NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93135NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93136NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93137NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93138NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93139NMDACORTICAL MEMBRANESPIG3H-MK-801(±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 15, 2025
93140Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine155Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93141Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine542Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93142Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine543Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93143Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine607Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93144Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine1500Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93145Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine2700Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93146Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine4900Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93147Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine502Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93148Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine192Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93149Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine37Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93150Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine7.37Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93151Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine297Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93152Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine314Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93153Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)(±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine3000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93154Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)PENTAZOCINE (+)6.03Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93155Sigma 2liver membranesRAT3H-DTG(±)-cis-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93156Sigma 2liver membranesRAT3H-DTG(±)-trans-N-Benzyl-1-(6-phenyl-1,4-dioxan-2-yl)methanamine4300Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93157Sigma 2liver membranesRAT3H-DTG(±)-cis-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93158Sigma 2liver membranesRAT3H-DTG(±)-trans-N-Benzyl-1-(6-ethyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93159Sigma 2liver membranesRAT3H-DTG(±)-cis-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine4900Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93160Sigma 2liver membranesRAT3H-DTG(±)-trans-N-Benzyl-1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)- methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93161Sigma 2liver membranesRAT3H-DTG(±)-N-Benzyl-1-(6,6-diphenyl-1,4-dioxan-2-yl)methanamine1600Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93162Sigma 2liver membranesRAT3H-DTG(±)-N-Benzyl-2-(6,6-diphenyl-1,4-dioxan-2-yl)ethanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93163Sigma 2liver membranesRAT3H-DTG(±)-cis-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine698Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93164Sigma 2liver membranesRAT3H-DTG(±)-trans-N-Benzyl-1-(5-phenyl-1,4-dioxan-2-yl)methanamine>10000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93165Sigma 2liver membranesRAT3H-DTG(±)-N-Benzyl-1-(5,5-diphenyl-1,4-dioxan-2-yl)methanamine1000Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93166Sigma 2liver membranesRAT3H-DTG(±)-N-Benzyl-2-(5,5-diphenyl-1,4-dioxan-2-yl)ethanamine841Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93167Sigma 2liver membranesRAT3H-DTG(±)-cis-N-Benzyl-1-(2-phenyl-1,3-dioxan-4-yl)methanamine174Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93168Sigma 2liver membranesRAT3H-DTG(±)-N-Benzyl-1-(2,2-diphenyl-1,3-dioxan-4-yl)methanamine111Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93169Sigma 2liver membranesRAT3H-DTGDTG64Bonifazi A et al 2015Jan 15, 2025Jan 28, 2025
93170D1CHO cellsPORCINE3H-SPIPERONE1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine6400Lober S et al 2012Jan 15, 2025Jan 28, 2025
93171D2CHO cellsHUMAN3H-SPIPERONE1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine95Lober S et al 2012Jan 15, 2025Jan 28, 2025
93172D2CHO cellsHUMAN3H-SPIPERONE1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine76Lober S et al 2012Jan 15, 2025Jan 29, 2025
93173D3CHO cellsHUMAN3H-SPIPERONE1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine370Lober S et al 2012Jan 15, 2025Jan 28, 2025
93174D4CHO cellsHUMAN3H-SPIPERONE1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine9.5Lober S et al 2012Jan 15, 2025Jan 29, 2025
931755-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine680Lober S et al 2012Jan 15, 2025Jan 15, 2025
93176CEREBRAL CORTEXPORCINE3H-KETANSERIN1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine2100Lober S et al 2012Jan 15, 2025Jan 15, 2025
93177CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-(3-Ethynylazulen-1-ylmethyl)-4-(2-methoxyphenyl)piperazine230Lober S et al 2012Jan 15, 2025Jan 15, 2025
93178D1CHO cellsPORCINE3H-SPIPERONE1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine1300Lober S et al 2012Jan 15, 2025Jan 28, 2025
93179D2CHO cellsHUMAN3H-SPIPERONE1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine65Lober S et al 2012Jan 15, 2025Jan 28, 2025
93180D2CHO cellsHUMAN3H-SPIPERONE1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine67Lober S et al 2012Jan 15, 2025Jan 29, 2025
93181D3CHO cellsHUMAN3H-SPIPERONE1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine210Lober S et al 2012Jan 15, 2025Jan 28, 2025
93182D4CHO cellsHUMAN3H-SPIPERONE1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine16Lober S et al 2012Jan 15, 2025Jan 29, 2025
931835-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine770Lober S et al 2012Jan 15, 2025Jan 15, 2025
93184CEREBRAL CORTEXPORCINE3H-KETANSERIN1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine1000Lober S et al 2012Jan 15, 2025Jan 15, 2025
93185CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-[3-(Phenylethynyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine370Lober S et al 2012Jan 15, 2025Jan 15, 2025
93186D1CHO cellsPORCINE3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine1400Lober S et al 2012Jan 15, 2025Jan 28, 2025
93187D2CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine76Lober S et al 2012Jan 15, 2025Jan 28, 2025
93188D2CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine60Lober S et al 2012Jan 15, 2025Jan 29, 2025
93189D3CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine370Lober S et al 2012Jan 15, 2025Jan 28, 2025
93190D4CHO cellsHUMAN3H-SPIPERONE1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine19Lober S et al 2012Jan 15, 2025Jan 29, 2025
931915-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine410Lober S et al 2012Jan 15, 2025Jan 15, 2025
93192CEREBRAL CORTEXPORCINE3H-KETANSERIN1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine1300Lober S et al 2012Jan 15, 2025Jan 15, 2025
93193CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-[3-(1-Pentyn-1-yl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine210Lober S et al 2012Jan 15, 2025Jan 15, 2025
93194D1CHO cellsPORCINE3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol860Lober S et al 2012Jan 15, 2025Jan 28, 2025
93195D2CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol150Lober S et al 2012Jan 15, 2025Jan 28, 2025
93196D2CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol68Lober S et al 2012Jan 15, 2025Jan 29, 2025
93197D3CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol580Lober S et al 2012Jan 15, 2025Jan 28, 2025
93198D4CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol0.71Lober S et al 2012Jan 15, 2025Jan 29, 2025
931995-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006353-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol120Lober S et al 2012Jan 15, 2025Jan 15, 2025
93200CEREBRAL CORTEXPORCINE3H-KETANSERIN3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol990Lober S et al 2012Jan 15, 2025Jan 15, 2025
93201CEREBRAL CORTEXPORCINE3H-PRAZOSIN3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol57Lober S et al 2012Jan 15, 2025Jan 15, 2025
93202CEREBRAL CORTEXPORCINE3H-RX8210023-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol44Lober S et al 2012Jan 15, 2025Jan 15, 2025
93203H1Sf9HUMAN3H-MEPYRAMINE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol1400Lober S et al 2012Jan 15, 2025Jan 28, 2025
932045-HT1DSf9HUMAN3H-UR-DE2573-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93205H3Sf9HUMAN3H-N-alpha-methylhistamine3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93206H4Sf9HUMAN3H-UR-PI2943-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulen-1-ylmethanol>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93207D1CHO cellsPORCINE3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril410Lober S et al 2012Jan 15, 2025Jan 28, 2025
93208D2CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril8.3Lober S et al 2012Jan 15, 2025Jan 28, 2025
93209D2CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril39Lober S et al 2012Jan 15, 2025Jan 29, 2025
93210D3CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril530Lober S et al 2012Jan 15, 2025Jan 28, 2025
93211D4CHO cellsHUMAN3H-SPIPERONE3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril2.4Lober S et al 2012Jan 15, 2025Jan 29, 2025
932125-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006353-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril110Lober S et al 2012Jan 15, 2025Jan 15, 2025
93213CEREBRAL CORTEXPORCINE3H-KETANSERIN3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril380Lober S et al 2012Jan 15, 2025Jan 15, 2025
93214CEREBRAL CORTEXPORCINE3H-PRAZOSIN3-[4-(2-Methoxyphenyl)piperazin-1-ylmethyl]azulene-1-carbonitril31Lober S et al 2012Jan 15, 2025Jan 15, 2025
93215D1CHO cellsPORCINE3H-SPIPERONE1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine4500Lober S et al 2012Jan 15, 2025Jan 28, 2025
93216D2CHO cellsHUMAN3H-SPIPERONE1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine210Lober S et al 2012Jan 15, 2025Jan 28, 2025
93217D2CHO cellsHUMAN3H-SPIPERONE1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine140Lober S et al 2012Jan 15, 2025Jan 29, 2025
93218D3CHO cellsHUMAN3H-SPIPERONE1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine390Lober S et al 2012Jan 15, 2025Jan 28, 2025
93219D4CHO cellsHUMAN3H-SPIPERONE1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine1.5Lober S et al 2012Jan 15, 2025Jan 29, 2025
932205-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine110Lober S et al 2012Jan 15, 2025Jan 15, 2025
93221CEREBRAL CORTEXPORCINE3H-KETANSERIN1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine1800Lober S et al 2012Jan 15, 2025Jan 15, 2025
93222CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine33Lober S et al 2012Jan 15, 2025Jan 15, 2025
93223CEREBRAL CORTEXPORCINE3H-RX8210021-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine23Lober S et al 2012Jan 15, 2025Jan 15, 2025
93224H1Sf9HUMAN3H-MEPYRAMINE1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine2600Lober S et al 2012Jan 15, 2025Jan 28, 2025
932255-HT1DSf9HUMAN3H-UR-DE2471-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine3200Lober S et al 2012Jan 15, 2025Jan 28, 2025
93226H3Sf9HUMAN3H-N-alpha-methylhistamine1-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93227H4Sf9HUMAN3H-UR-PI2941-[3-(N,N-Dimethylaminomethyl)azulen-1-ylmethyl]-4-(2-methoxyphenyl)piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93228D1CHO cellsPORCINE3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine4100Lober S et al 2012Jan 15, 2025Jan 28, 2025
93229D2CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine51Lober S et al 2012Jan 15, 2025Jan 28, 2025
93230D2CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine37Lober S et al 2012Jan 15, 2025Jan 29, 2025
93231D3CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine160Lober S et al 2012Jan 15, 2025Jan 28, 2025
93232D4CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine1.9Lober S et al 2012Jan 15, 2025Jan 29, 2025
932335-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine65Lober S et al 2012Jan 15, 2025Jan 15, 2025
93234CEREBRAL CORTEXPORCINE3H-KETANSERIN1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine1300Lober S et al 2012Jan 15, 2025Jan 15, 2025
93235CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine32Lober S et al 2012Jan 15, 2025Jan 15, 2025
93236CEREBRAL CORTEXPORCINE3H-RX8210021-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine140Lober S et al 2012Jan 15, 2025Jan 15, 2025
93237H1Sf9HUMAN3H-MEPYRAMINE1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine5500Lober S et al 2012Jan 15, 2025Jan 28, 2025
932385-HT1DSf9HUMAN3H-UR-DE2571-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine4200Lober S et al 2012Jan 15, 2025Jan 28, 2025
93239H3Sf9HUMAN3H-N-alpha-methylhistamine1-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93240H4Sf9HUMAN3H-UR-PI2941-(2-Methoxyphenyl)-4-[[3-(1-piperidylmethyl)azulen-1-yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93241D1CHO cellsPORCINE3H-SPIPERONE4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine5000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93242D2CHO cellsHUMAN3H-SPIPERONE4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine130Lober S et al 2012Jan 15, 2025Jan 28, 2025
93243D2CHO cellsHUMAN3H-SPIPERONE4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine92Lober S et al 2012Jan 15, 2025Jan 29, 2025
93244D3CHO cellsHUMAN3H-SPIPERONE4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine350Lober S et al 2012Jan 15, 2025Jan 28, 2025
93245D4CHO cellsHUMAN3H-SPIPERONE4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine4.6Lober S et al 2012Jan 15, 2025Jan 29, 2025
932465-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006354-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine99Lober S et al 2012Jan 15, 2025Jan 15, 2025
93247CEREBRAL CORTEXPORCINE3H-KETANSERIN4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine1000Lober S et al 2012Jan 15, 2025Jan 15, 2025
93248CEREBRAL CORTEXPORCINE3H-PRAZOSIN4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine57Lober S et al 2012Jan 15, 2025Jan 15, 2025
93249CEREBRAL CORTEXPORCINE3H-RX8210024-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine220Lober S et al 2012Jan 15, 2025Jan 15, 2025
93250H1Sf9HUMAN3H-MEPYRAMINE4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine6500Lober S et al 2012Jan 15, 2025Jan 28, 2025
932515-HT1DSf9HUMAN3H-UR-DE2574-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine6100Lober S et al 2012Jan 15, 2025Jan 28, 2025
93252H3Sf9HUMAN3H-N-alpha-methylhistamine4-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93253H4Sf9HUMAN3H-UR-PI2944-[[3-[[4-(2-Methoxyphenyl)piperazin-1-yl]methyl]azulen-1-yl]methyl]morpholine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93254D1CHO cellsPORCINE3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine6400Lober S et al 2012Jan 15, 2025Jan 28, 2025
93255D2CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine60Lober S et al 2012Jan 15, 2025Jan 28, 2025
93256D2CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine57Lober S et al 2012Jan 15, 2025Jan 29, 2025
93257D3CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine460Lober S et al 2012Jan 15, 2025Jan 28, 2025
93258D4CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine3.8Lober S et al 2012Jan 15, 2025Jan 29, 2025
932595-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine91Lober S et al 2012Jan 15, 2025Jan 15, 2025
93260CEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine2100Lober S et al 2012Jan 15, 2025Jan 15, 2025
93261CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine66Lober S et al 2012Jan 15, 2025Jan 15, 2025
93262CEREBRAL CORTEXPORCINE3H-RX8210021-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine170Lober S et al 2012Jan 15, 2025Jan 15, 2025
93263H1Sf9HUMAN3H-MEPYRAMINE1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
932645-HT1DSf9HUMAN3H-UR-DE2571-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine5500Lober S et al 2012Jan 15, 2025Jan 28, 2025
93265H3Sf9HUMAN3H-N-alpha-methylhistamine1-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine5500Lober S et al 2012Jan 15, 2025Jan 28, 2025
93266H4Sf9HUMAN3H-UR-PI2941-(2-Methoxyphenyl)-4-[[3-[(4-methylpiperazin-1-yl)methyl]azulen-1-yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93267D1CHO cellsPORCINE3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine740Lober S et al 2012Jan 15, 2025Jan 28, 2025
93268D2CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine17Lober S et al 2012Jan 15, 2025Jan 28, 2025
93269D2CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine34Lober S et al 2012Jan 15, 2025Jan 29, 2025
93270D3CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine33Lober S et al 2012Jan 15, 2025Jan 28, 2025
93271D4CHO cellsHUMAN3H-SPIPERONE1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine0.79Lober S et al 2012Jan 15, 2025Jan 29, 2025
932725-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine100Lober S et al 2012Jan 15, 2025Jan 15, 2025
93273CEREBRAL CORTEXPORCINE3H- Ketanserin1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine560Lober S et al 2012Jan 15, 2025Jan 15, 2025
93274CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine8.3Lober S et al 2012Jan 15, 2025Jan 15, 2025
93275CEREBRAL CORTEXPORCINE3H-RX8210021-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine120Lober S et al 2012Jan 15, 2025Jan 15, 2025
93276H1Sf9HUMAN3H-MEPYRAMINE1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine1000Lober S et al 2012Jan 15, 2025Jan 28, 2025
932775-HT1DSf9HUMAN3H-UR-DE2571-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine530Lober S et al 2012Jan 15, 2025Jan 28, 2025
93278H3Sf9HUMAN3H-N-alpha-methylhistamine1-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93279H4Sf9HUMAN3H-UR-PI2941-(2-Methoxyphenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93280D1CHO cellsPORCINE3H-SPIPERONE1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine1100Lober S et al 2012Jan 15, 2025Jan 28, 2025
93281D2CHO cellsHUMAN3H-SPIPERONE1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine95Lober S et al 2012Jan 15, 2025Jan 28, 2025
93282D2CHO cellsHUMAN3H-SPIPERONE1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine160Lober S et al 2012Jan 15, 2025Jan 29, 2025
93283D3CHO cellsHUMAN3H-SPIPERONE1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine85Lober S et al 2012Jan 15, 2025Jan 28, 2025
93284D4CHO cellsHUMAN3H-SPIPERONE1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine6Lober S et al 2012Jan 15, 2025Jan 29, 2025
932855-HT1ACEREBRAL CORTEXPORCINE3H-WAY1006351-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine760Lober S et al 2012Jan 15, 2025Jan 15, 2025
93286CEREBRAL CORTEXPORCINE3H- Ketanserin1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine1600Lober S et al 2012Jan 15, 2025Jan 15, 2025
93287CEREBRAL CORTEXPORCINE3H-PRAZOSIN1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine27Lober S et al 2012Jan 15, 2025Jan 15, 2025
93288CEREBRAL CORTEXPORCINE3H-RX8210021-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine1200Lober S et al 2012Jan 15, 2025Jan 15, 2025
93289H1Sf9HUMAN3H-MEPYRAMINE1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine490Lober S et al 2012Jan 15, 2025Jan 28, 2025
932905-HT1DSf9HUMAN3H-DE2571-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine460Lober S et al 2012Jan 15, 2025Jan 28, 2025
93291H3Sf9HUMAN3H-N-alpha-methylhistamine1-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine>10000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93292H4Sf9HUMAN3H-UR-PI2941-(4-Chlorophenyl)-4-[[3-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]azulen-1- yl]methyl]piperazine1000Lober S et al 2012Jan 15, 2025Jan 28, 2025
93293D1CHO cellsPORCINE3H-SPIPERONEFAUC 3019500Lober S et al 2012Jan 15, 2025Jan 28, 2025
93294D2CHO cellsHUMAN3H-SPIPERONEFAUC 301933Lober S et al 2012Jan 15, 2025Jan 28, 2025
93295D2CHO cellsHUMAN3H-SPIPERONEFAUC 301924Lober S et al 2012Jan 15, 2025Jan 29, 2025
93296D3CHO cellsHUMAN3H-SPIPERONEFAUC 301983Lober S et al 2012Jan 15, 2025Jan 28, 2025
93297D4CHO cellsHUMAN3H-SPIPERONEFAUC 30190.4Lober S et al 2012Jan 15, 2025Jan 29, 2025
932985-HT1ACEREBRAL CORTEXPORCINE3H-WAY100635FAUC 301954Lober S et al 2012Jan 15, 2025Jan 15, 2025
93299CEREBRAL CORTEXPORCINE3H- KetanserinFAUC 301992Lober S et al 2012Jan 15, 2025Jan 15, 2025
93300CEREBRAL CORTEXPORCINE3H-PRAZOSINFAUC 301920Lober S et al 2012Jan 15, 2025Jan 15, 2025
93301CEREBRAL CORTEXPORCINE3H-RX821002FAUC 301939Lober S et al 2012Jan 15, 2025Jan 15, 2025
933025-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT1,3,7-Trimethyl-8-[3-(4-phenyl-1-piperazinyl)- propylamino]-purine-2,6-dione hydrochloride385Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933035-HT1AHIPPOCAMPUSRAT3H-8-OH-DPAT1,3-Dimethyl-7-n-butyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione hydrochloride100Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933045-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATEthyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-acetic acid hydrochloride592Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933055-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATEthyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-butyric acid457Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933065-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-Phenyl-1-piperazinyl)-propyl]-3-phenylpyrrolidine-2,5-dione dihydrochloride1069Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933075-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride177Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933085-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-chlorophenyl)-pyrrolidine-2,5-dione dihydrochloride258Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933095-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-Phenyl-1-piperazinyl)-propyl]-3-(4-fluorophenyl)-pyrrolidine-2,5-dione dihydrochloride223Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933105-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-Phenyl-1-piperazinyl)-propyl-3-(4-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride510Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933115-HT1AHIPPOCAMPUSRAT3H-8-OH-DPATN-[(4-Phenyl-1-piperazinyl)-propyl]-3,3- diphenyl-pyrrolidine-2,5-dione dihydrochloride444Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933125-HT2ABRAIN CORTEXRAT3H-KETANSERINN-[(4-Phenyl-1-piperazinyl)-propyl]-3,3- diphenyl-pyrrolidine-2,5-dione dihydrochloride842Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933135-HT2ABRAIN CORTEXRAT3H-KETANSERINN-[(4-Phenyl-1-piperazinyl)-propyl-3-(4-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride436Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933145-HT2ABRAIN CORTEXRAT3H-KETANSERINN-[(4-Phenyl-1-piperazinyl)-propyl]-3-(4-fluorophenyl)-pyrrolidine-2,5-dione dihydrochloride436Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933155-HT2ABRAIN CORTEXRAT3H-KETANSERINN-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-chlorophenyl)-pyrrolidine-2,5-dione dihydrochloride388Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933165-HT2ABRAIN CORTEXRAT3H-KETANSERINN-[(4-phenyl-1-piperazinyl)-propyl]-3-(3-bromophenyl)-pyrrolidine-2,5-dione dihydrochloride329Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933175-HT2ABRAIN CORTEXRAT3H-KETANSERINN-[(4-Phenyl-1-piperazinyl)-propyl]-3-phenylpyrrolidine-2,5-dione dihydrochloride268Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933185-HT2ABRAIN CORTEXRAT3H-KETANSERINEthyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-butyric acid1010Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933195-HT2ABRAIN CORTEXRAT3H-KETANSERINEthyl ester of 1,3-dimethyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione-7-acetic acid hydrochloride179Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933205-HT2ABRAIN CORTEXRAT3H-KETANSERIN1,3-Dimethyl-7-n-butyl-8-[3-(4-phenyl-1- piperazinyl)-propylamino]-purine-2,6-dione hydrochloride614Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933215-HT2ABRAIN CORTEXRAT3H-KETANSERIN1,3,7-Trimethyl-8-[3-(4-phenyl-1-piperazinyl)- propylamino]-purine-2,6-dione hydrochloride197Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933225-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride39Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933235-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride68Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933245-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride20Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933255-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride4.3Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933265-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride4.5Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933275-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride4.5Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933285-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride25Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933295-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride66Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933305-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride18Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933315-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride204Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933325-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride146Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933335-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride488Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933345-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride354Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933355-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride56Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933365-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride104Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933375-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride70Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933385-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride15Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933395-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride20Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933405-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride133Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933415-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride899Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933425-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride230Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933435-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride7.6Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933445-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride64Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933455-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride48Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933465-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride477Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933475-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride151Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933485-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride631Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933495-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPAT8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride34Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933505-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride259Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933515-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride298Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933525-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride116Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933535-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride162Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933545-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride400Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933555-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride179Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933565-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride68Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933575-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride115Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933585-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride114Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933595-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride428Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933605-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride3517Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933615-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride1789Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933625-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride574Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933635-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride2335Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933645-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride269Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933655-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride302Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933665-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride1411Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933675-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride475Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933685-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride72Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933695-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride902Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933705-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933715-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride348Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933725-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride154Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933735-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride480Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933745-HT2AHIPPOCAMPUSRAT3H-KETANSERIN7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride388Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933755-HT2AHIPPOCAMPUSRAT3H-KETANSERIN1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride398Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933765-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride80Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933775-HT2AHIPPOCAMPUSRAT3H-KETANSERIN8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride210Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933785-HT6CLONEDHUMAN3H-5-CT7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933795-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933805-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride958Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933815-HT6CLONEDHUMAN3H-5-CT7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933825-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933835-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933845-HT6CLONEDHUMAN3H-5-CT7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933855-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride911Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933865-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride98Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933875-HT6CLONEDHUMAN3H-5-CT7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933885-HT6CLONEDHUMAN3H-5-CT8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933895-HT6CLONEDHUMAN3H-5-CT8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933905-HT6CLONEDHUMAN3H-5-CT7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933915-HT6CLONEDHUMAN3H-5-CT8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933925-HT6CLONEDHUMAN3H-5-CT8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933935-HT6CLONEDHUMAN3H-5-CT7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride5706Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933945-HT6CLONEDHUMAN3H-5-CT7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933955-HT6CLONEDHUMAN3H-5-CT7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933965-HT6CLONEDHUMAN3H-5-CT7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933975-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933985-HT6CLONEDHUMAN3H-5-CT8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
933995-HT6CLONEDHUMAN3H-5-CT7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934005-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934015-HT6CLONEDHUMAN3H-5-CT7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934025-HT6CLONEDHUMAN3H-5-CT7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934035-HT6CLONEDHUMAN3H-5-CT1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934045-HT6CLONEDHUMAN3H-5-CT8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride1000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934055-HT6CLONEDHUMAN3H-5-CT8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride717Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934065-HT7CLONEDHUMAN3H-LSD7-Benzyl-1,3-dimethyl-8-((4-(4-phenylpiperazin1-yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride90Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934075-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-7-phenethyl-8-((4-(4-phenylpiperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride25Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934085-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-8-((4-(4-phenylpiperazin-1-yl) butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride36Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934095-HT7CLONEDHUMAN3H-LSD7-Benzyl-8-((4-(4-(2-methoxyphenyl)piperazin1-yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride40Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934105-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-7-phenethyl-8-((4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride10Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934115-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride20Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934125-HT7CLONEDHUMAN3H-LSD7-Benzyl-8-((4-(4-(3-chlorophenyl)piperazin-1- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride65Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934135-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-7-phenethyl-8-((4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride113Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934145-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-8-((4-(4-(3-chlorophenyl)piperazin1-yl)butyl)amino)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride85Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934155-HT7CLONEDHUMAN3H-LSD7-Benzyl-8-((3-(3,4-dihydroisoquinolin2(1H)-yl)propyl)amino)-1,3-dimethyl-1Hpurine-2,6(3H,7H)-dione hydrochloride454Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934165-HT7CLONEDHUMAN3H-LSD8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride3590Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934175-HT7CLONEDHUMAN3H-LSD8-((3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)-1Hpurine-2,6(3H,7H)-dione hydrochloride>10000Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934185-HT7CLONEDHUMAN3H-LSD7-Benzyl-8-((4-(3,4-dihydroisoquinolin- 2(1H)- yl)butyl)amino)-1,3-dimethyl-1H-purine2,6(3H,7H)-dione hydrochloride302Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934195-HT7CLONEDHUMAN3H-LSD8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl) amino)-1,3-dimethyl-7-phenethyl-1H-purine2,6(3H,7H)-dione hydrochloride99Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934205-HT7CLONEDHUMAN3H-LSD8-((4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)- amino)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride239Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934215-HT7CLONEDHUMAN3H-LSD7-Allyl-1,3-dimethyl-8-((4-(4-phenylpiperazin-1- yl)butyl)amino)-1H-purine-2,6(3H,7H)-dione hydrochloride476Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934225-HT7CLONEDHUMAN3H-LSD7-Allyl-1,3-dimethyl-8-((3-(4-(2-methoxyphenyl)- piperazin-1-yl)propyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride274Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934235-HT7CLONEDHUMAN3H-LSD7-Allyl-1,3-dimethyl-8-((4-(4-(2-methoxyphenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride622Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934245-HT7CLONEDHUMAN3H-LSD7-Allyl-1,3-dimethyl-8-((4-(4-(4-fluorophenyl)- piperazin-1-yl)butyl)amino)-1H-purine2,6(3H,7H)-dione hydrochloride269Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934255-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-8-((3-(4-phenylpiperazin-1-yl)propyl)amino)-7-(prop-1-yn-1-yl)-1H-purine2,6(3H,7H)-dione hydrochloride1200Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934265-HT7CLONEDHUMAN3H-LSD8-((3-(4-(2-Methoxyphenyl)piperazin-1-yl)propyl)amino)-1,3-dimethyl-7-(prop-1-yn-1-yl)- 1H-purine-2,6(3H,7H)-dione hydrochloride740Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934275-HT7CLONEDHUMAN3H-LSD7-Benzyl-1,3-dimethyl-8-(3-(4-phenylpiperazin1-yl)propoxy)-1H-purine-2,6(3H,7H)-dione hydrochloride89Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934285-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-8-(3-(4-phenylpiperazin-1- yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride165Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934295-HT7CLONEDHUMAN3H-LSD7-Benzyl-8-(3-(4-(2-methoxyphenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride75Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934305-HT7CLONEDHUMAN3H-LSD7-Benzyl-8-(3-(4-(3-chlorophenyl)piperazin-1- yl)propoxy)-1,3-dimethyl-1H-purine-2,6(3H,7H)- dione hydrochloride295Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934315-HT7CLONEDHUMAN3H-LSD1,3-Dimethyl-8-(3-(4-(3-chlorophenyl)piperazin1-yl)propoxy)-7-(3-phenylpropyl)-1H-purine2,6(3H,7H)-dione hydrochloride936Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934325-HT7CLONEDHUMAN3H-LSD8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)- 1,3-dimethyl-7-phenethyl-1H-purine-2,6(3H,7H)- dione hydrochloride105Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
934335-HT7CLONEDHUMAN3H-LSD8-(3-(4-(4-Fluorophenyl)piperazin-1-yl)propoxy)-1,3-dimethyl-7-(3-phenylpropyl)- 1H-purine-2,6(3H,7H)-dione hydrochloride63Chlon-Rzepa G et al 2013Jan 15, 2025Jan 15, 2025
93434A1C.H.O.? HUMAN3H-CCPA6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93435A1C.H.O.? HUMAN3H-CCPA6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide8200Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93436A1C.H.O.? HUMAN3H-CCPA6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93437A1C.H.O.? HUMAN3H-CCPA6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93438A1C.H.O.? HUMAN3H-CCPAEthyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate8800Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93439A1C.H.O.? HUMAN3H-CCPAEthyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate900Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93440A1C.H.O.? HUMAN3H-CCPAEthyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate4000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93441A1C.H.O.? HUMAN3H-CCPAEthyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate3500Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93442A1C.H.O.? HUMAN3H-CCPAEthyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93443A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93444A1C.H.O.? HUMAN3H-CCPAEthyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93445A1C.H.O.? HUMAN3H-CCPAEthyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93446A1C.H.O.? HUMAN3H-CCPAEthyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate4300Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93447A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate2800Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93448A1C.H.O.? HUMAN3H-CCPAEthyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93449A1C.H.O.? HUMAN3H-CCPAEthyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate700Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93450A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate2700Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93451A1C.H.O.? HUMAN3H-CCPAEthyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate5100Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93452A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate5000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93453A1C.H.O.? HUMAN3H-CCPAEthyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate2500Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93454A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93455A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate2600Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93456A1C.H.O.? HUMAN3H-CCPAEthyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93457A1C.H.O.? HUMAN3H-CCPAEthyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93458A1C.H.O.? HUMAN3H-CCPAEthyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93459A1C.H.O.? HUMAN3H-CCPAEthyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93460A1C.H.O.? HUMAN3H-CCPAEthyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93461A1C.H.O.? HUMAN3H-CCPAEthyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93462A1C.H.O.? HUMAN3H-CCPAEthyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate5900Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93463A1C.H.O.? HUMAN3H-CCPAEthyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate600Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93464A1C.H.O.? HUMAN3H-CCPAEthyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate2700Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93465A1C.H.O.? HUMAN3H-CCPAEthyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate600Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93466A2ACHO cells? HUMAN3H-NECAEthyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate2400Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93467A2BCHO cells? HUMAN3H-NECAEthyl-2-phenethyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93468A2BCHO cells? HUMAN3H-NECAEthyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93469A2ACHO cells? HUMAN3H-NECAEthyl-2-neopentyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate5700Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93470A2ACHO cells? HUMAN3H-NECAEthyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate8800Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93471A2BCHO cells? HUMAN3H-NECAEthyl-2-isopropyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93472A2BCHO cells? HUMAN3H-NECAEthyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93473A2ACHO cells? HUMAN3H-NECAEthyl-2-methyl-6-(2-phenylacetamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate7300Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93474A2ACHO cells? HUMAN3H-NECAEthyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93475A2BCHO cells? HUMAN3H-NECAEthyl-6-(N-benzoylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93476A2BCHO cells? HUMAN3H-NECAEthyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93477A2ACHO cells? HUMAN3H-NECAEthyl-6-(N-benzoylbenzamido)-2-isopropyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93478A2ACHO cells? HUMAN3H-NECAEthyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93479A2BCHO cells? HUMAN3H-NECAEthyl-6-(N-(3,4-difluorobenzoyl)-3,4-difluorobenzamido)- 2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93480A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93481A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-bromo-N-(4-bromobenzoyl)benzamido)-2- methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93482A2ACHO cells? HUMAN3H-NECAEthyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93483A2BCHO cells? HUMAN3H-NECAEthyl-6-(N-benzoylbenzamido)-2-methyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93484A2BCHO cells? HUMAN3H-NECAEthyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93485A2ACHO cells? HUMAN3H-NECAEthyl-6-(3,4-dichlorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93486A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate4200Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93487A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-bromobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93488A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93489A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-methylbenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate6000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93490A2ACHO cells? HUMAN3H-NECAEthyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate7500Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93491A2BCHO cells? HUMAN3H-NECAEthyl-2-phenethyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93492A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93493A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-phenethyl-2H-pyrazolo [3,4-d]pyrimidine-4-carboxylate6100Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93494A2ACHO cells? HUMAN3H-NECAEthyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate3700Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93495A2BCHO cells? HUMAN3H-NECAEthyl-6-benzamido-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93496A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93497A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-neopentyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate5700Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93498A2ACHO cells? HUMAN3H-NECAEthyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate2300Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93499A2BCHO cells? HUMAN3H-NECAEthyl-2-isopropyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93500A2ACHO cells? HUMAN3H-NECAEthyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93501A2BCHO cells? HUMAN3H-NECAEthyl-2-isopropyl-6-(4-(trifluoromethyl)benzamido)-2Hpyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93502A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93503A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-isopropyl-2H-pyrazolo[3,4- d]pyrimidine-4-carboxylate2800Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93504A2ACHO cells? HUMAN3H-NECAEthyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate3300Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93505A2BCHO cells? HUMAN3H-NECAEthyl-6-benzamido-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93506A2BCHO cells? HUMAN3H-NECAEthyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93507A2ACHO cells? HUMAN3H-NECAEthyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93508A2ACHO cells? HUMAN3H-NECAEthyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93509A2BCHO cells? HUMAN3H-NECAEthyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93510A2BCHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93511A2ACHO cells? HUMAN3H-NECAEthyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93512A2BCHO cells? HUMAN3H-NECAEthyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93513A2ACHO cells? HUMAN3H-NECAEthyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93514A2ACHO cells? HUMAN3H-NECAEthyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate4800Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93515A2BCHO cells? HUMAN3H-NECAEthyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93516A2BCHO cells? HUMAN3H-NECAEthyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93517A2ACHO cells? HUMAN3H-NECAEthyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate5000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93518A2ACHO cells? HUMAN3H-NECAEthyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate2600Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93519A2BCHO cells? HUMAN3H-NECAEthyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93520A2BCHO cells? HUMAN3H-NECAEthyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93521A2ACHO cells? HUMAN3H-NECAEthyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate2000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93522A2ACHO cells? HUMAN3H-NECA6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93523A2BCHO cells? HUMAN3H-NECA6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93524A2BCHO cells? HUMAN3H-NECA6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93525A2ACHO cells? HUMAN3H-NECA6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93526A2ACHO cells? HUMAN3H-NECA6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide9200Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93527A2BCHO cells? HUMAN3H-NECA6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93528A2BCHO cells? HUMAN3H-NECA6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93529A2ACHO cells? HUMAN3H-NECA6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide3000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93530A3CHO cells? HUMAN3H-HEMADO6-Amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93531A3CHO cells? HUMAN3H-HEMADO6-Amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93532A3CHO cells? HUMAN3H-HEMADO6-Amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93533A3CHO cells? HUMAN3H-HEMADO6-Amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxamide>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93534A3CHO cells? HUMAN3H-HEMADOEthyl-6-amino-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4- carboxylate900Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93535A3CHO cells? HUMAN3H-HEMADOEthyl-6-amino-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93536A3CHO cells? HUMAN3H-HEMADOEthyl-6-amino-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93537A3CHO cells? HUMAN3H-HEMADOEthyl-6-amino-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidine4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93538A3CHO cells? HUMAN3H-HEMADOEthyl-6-benzamido-2-methyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93539A3CHO cells? HUMAN3H-HEMADOEthyl-6-(4-fluorobenzamido)-2-methyl-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93540A3CHO cells? HUMAN3H-HEMADOEthyl-2-methyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93541A3CHO cells? HUMAN3H-HEMADOEthyl-2-methyl-6-(4-methylbenzamido)-2H-pyrazolo[3,4-d] pyrimidine-4-carboxylate>10000Venkatesan G et al 2015Jan 15, 2025Jan 15, 2025
93542A1CLONEDHUMAN3H-CCPAN2 -benzyl-9-propyl-9H-purine-2,6-diamine7600Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93543A2ACLONEDHUMAN3H-NECAN2 -benzyl-9-propyl-9H-purine-2,6-diamine1400Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93544A3CLONEDHUMAN3H-HEMADON2 -benzyl-9-propyl-9H-purine-2,6-diamine5840Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93545A3CLONEDHUMAN3H-HEMADON2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine650Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93546A2ACLONEDHUMAN3H-NECAN2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine36Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93547A1CLONEDHUMAN3H-CCPAN2 -Benzyl-8-bromo-9-propyl-9H-purine-2,6-diamine358Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93548A1CLONEDHUMAN3H-CCPAN2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine138Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93549A2ACLONEDHUMAN3H-NECAN2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine6.6Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93550A3CLONEDHUMAN3H-HEMADON2 -benzyl-8-(furan-2-yl)-9-propyl-9H-purine-2,6-diamine29Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93551A3CLONEDHUMAN3H-HEMADON2 -phenethyl-9-propyl-9H-purine-2,6-diamine5880Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93552A2ACLONEDHUMAN3H-NECAN2 -phenethyl-9-propyl-9H-purine-2,6-diamine738Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93553A1CLONEDHUMAN3H-CCPAN2 -phenethyl-9-propyl-9H-purine-2,6-diamine2330Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93554A1CLONEDHUMAN3H-CCPA8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine373Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93555A2ACLONEDHUMAN3H-NECA8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine27Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93556A3CLONEDHUMAN3H-HEMADO8-Bromo-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine1160Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93557A3CLONEDHUMAN3H-HEMADO8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine56Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93558A2ACLONEDHUMAN3H-NECA8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine14Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93559A1CLONEDHUMAN3H-CCPA8-(Furan-2-yl)-N2 -phenethyl-9-propyl-9H-purine-2,6-diamine80.3Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93560A1CLONEDHUMAN3H-CCPAN2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine3640Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93561A2ACLONEDHUMAN3H-NECAN2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine9110Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93562A3CLONEDHUMAN3H-HEMADON2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93563A3CLONEDHUMAN3H-HEMADO8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine1950Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93564A2ACLONEDHUMAN3H-NECA8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine284Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93565A1CLONEDHUMAN3H-CCPA8-Bromo-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine583Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93566A1CLONEDHUMAN3H-CCPA8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine230Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93567CLONEDHUMAN3H-NECA8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine113Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93568A3CLONEDHUMAN3H-HEMADO8-(Furan-2-yl)-N2 -(3-phenylpropyl)-9-propyl-9H-purine-2,6-diamine266Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93569A3CLONEDHUMAN3H-HEMADON-benzyl-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93570A2ACLONEDHUMAN3H-NECAN-benzyl-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93571A1CLONEDHUMAN3H-CCPAN-benzyl-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93572A1CLONEDHUMAN3H-CCPAN-benzyl-8-bromo-9-propyl-9H-purin-6-amine5620Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93573A2ACLONEDHUMAN3H-NECAN-benzyl-8-bromo-9-propyl-9H-purin-6-amine1180Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93574A3CLONEDHUMAN3H-HEMADON-benzyl-8-bromo-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93575A3CLONEDHUMAN3H-HEMADON-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine402Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93576A2ACLONEDHUMAN3H-NECAN-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine80Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93577A1CLONEDHUMAN3H-CCPAN-benzyl-8-(furan-2-yl)-9-propyl-9H-purin-6-amine546Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93578A1CLONEDHUMAN3H-CCPAN-phenethyl-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93579A2ACLONEDHUMAN3H-NECAN-phenethyl-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93580A3CLONEDHUMAN3H-HEMADON-phenethyl-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93581A3CLONEDHUMAN3H-HEMADO8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine2520Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93582A2ACLONEDHUMAN3H-NECA8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine503Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93583A1CLONEDHUMAN3H-CCPA8-Bromo-N-phenethyl-9-propyl-9H-purin-6-amine1940Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93584A1CLONEDHUMAN3H-CCPA8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine2440Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93585A2ACLONEDHUMAN3H-NECA8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine547Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93586A3CLONEDHUMAN3H-HEMADO8-(Furan-2-yl)-N-phenethyl-9-propyl-9H-purin-6-amine811Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93587A3CLONEDHUMAN3H-HEMADON-(3-phenylpropyl)-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93588A2ACLONEDHUMAN3H-NECAN-(3-phenylpropyl)-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93589A1CLONEDHUMAN3H-CCPAN-(3-phenylpropyl)-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93590A1CLONEDHUMAN3H-CCPA8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine2670Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93591A2ACLONEDHUMAN3H-NECA8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine1020Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93592A3CLONEDHUMAN3H-HEMADO8-Bromo-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine>10000Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93593A3CLONEDHUMAN3H-HEMADO8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine959Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93594A2ACLONEDHUMAN3H-NECA8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine181Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93595A1CLONEDHUMAN3H-CCPA8-(Furan-2-yl)-N-(3-phenylpropyl)-9-propyl-9H-purin-6-amine378Lambertucci C et al 2015Jan 15, 2025Jan 15, 2025
93596D2CLONEDHUMAN125I-IABN7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate2604Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93597D3CLONEDHUMAN125I-IABN7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate1536Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93598D4CLONEDHUMAN125I-IABN7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate1311Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93599Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate417Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93600Sigma 2LIVERRAT3H-DTG7-(4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate8269Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93601Sigma 2LIVERRAT3H-DTG7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate>10000Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93602Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate433Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93603D4CLONEDHUMAN125I-IABN7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate1029Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93604D3CLONEDHUMAN125I-IABN7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate879Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93605D2CLONEDHUMAN125I-IABN7-(4-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)- piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate145Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93606D2CLONEDHUMAN125I-IABN7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate309Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93607D3CLONEDHUMAN125I-IABN7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate574Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93608D4CLONEDHUMAN125I-IABN7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate1352Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93609Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate158Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93610Sigma 2LIVERRAT3H-DTG7-(4-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol1-yl)piperidin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate>10000Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93611Sigma 2LIVERRAT3H-DTG7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate>10000Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93612Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate3087Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93613D4CLONEDHUMAN125I-IABN7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate865Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93614D3CLONEDHUMAN125I-IABN7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate427Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93615D2CLONEDHUMAN125I-IABN7-(4-(3Methyl-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan8-yl)butoxy)-3,4-dihydro-quinolin-2(1H)-one oxalate611Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93616D2CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate0.22Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93617D3CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate13.1Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93618D4CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate212Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93619Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate1176Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93620Sigma 2LIVERRAT3H-DTG7-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate598Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93621Sigma 2LIVERRAT3H-DTG7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate4988Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93622Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate>10000Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93623D4CLONEDHUMAN125I-IABN7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate185Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93624D3CLONEDHUMAN125I-IABN7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate13.5Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93625D2CLONEDHUMAN125I-IABN7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1-yl)butoxy)- 3,4-dihydroquinolin-2(1H)-one oxalate0.26Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93626D2CLONEDHUMAN125I-IABN7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate102Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93627D3CLONEDHUMAN125I-IABN7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate930Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93628D4CLONEDHUMAN125I-IABN7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate359Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93629Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate170Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93630Sigma 2LIVERRAT3H-DTG7-(4-(4-(4-Methoxyphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate665Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93631Sigma 2LIVERRAT3H-DTG7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate3340Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93632Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate620Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93633D4CLONEDHUMAN125I-IABN7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate286Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93634D3CLONEDHUMAN125I-IABN7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate785Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93635D2CLONEDHUMAN125I-IABN7-(4-(4-(2,4-Dimethoxyphenyl)piperazin-1-yl)butoxy)-3,4- dihydroquinolin-2(1H)-one oxalate25.3Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93636D2CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate4.6Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93637D3CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate251Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93638D4CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate27.2Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93639Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate377Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93640Sigma 2LIVERRAT3H-DTG7-(4-(4-(2-Methoxy-4-methylphenyl)piperazin-1-yl)butoxy)-3,4-dihydroquinolin-2(1H)-one oxalate6393Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93641Sigma 2LIVERRAT3H-DTG7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate1309Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93642Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate2631Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93643D4CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate30.1Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93644D3CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate5.4Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93645D2CLONEDHUMAN125I-IABN7-(4-(4-(2-Methoxyphenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate0.14Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93646D2CLONEDHUMAN125I-IABN7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate0.07Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93647D3CLONEDHUMAN125I-IABN7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate2.7Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93648D4CLONEDHUMAN125I-IABN7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate31.9Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93649Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate>10000Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93650Sigma 2LIVERRAT3H-DTG7-(4-(4-(2-(2-Fluoroethoxy)phenyl)piperazin-1- yl)butoxy)quinolin-2(1H)-one oxalate4952Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93651Sigma 2LIVERRAT3H-DTG7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate1907Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93652Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate759Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93653D4CLONEDHUMAN125I-IABN7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate38.5Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93654D3CLONEDHUMAN125I-IABN7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate7.4Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93655D2CLONEDHUMAN125I-IABN7-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propoxy)-3,4- dihydroquinolin-2(1H)-one oxalate4.8Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93656D2CLONEDHUMAN125I-IABN7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate2.6Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93657D3CLONEDHUMAN125I-IABN7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate5.7Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93658D4CLONEDHUMAN125I-IABN7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate52.7Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93659Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate2600Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93660Sigma 2LIVERRAT3H-DTG7-(3-(4-(2-Methoxyphenyl)piperazin-1- yl)propoxy)quinolin-2(1H)-one oxalate2838Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93661Sigma 2LIVERRAT3H-DTG7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate231Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93662Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate1349Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93663D4CLONEDHUMAN125I-IABN7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate234Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93664D3CLONEDHUMAN125I-IABN7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate7Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93665D2CLONEDHUMAN125I-IABN7-(5-(4-(2-Methoxyphenyl)piperazin-1-yl)pentyloxy)-3,4- dihydroquinolin-2(1H)-one oxalate7.3Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93666D2CLONEDHUMAN125I-IABN7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate7.4Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93667D3CLONEDHUMAN125I-IABN7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate3.8Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93668D4CLONEDHUMAN125I-IABN7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate201Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93669Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate1614Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93670Sigma 2LIVERRAT3H-DTG7-(5-(4-(2-Methoxyphenyl)piperazin-1- yl)pentyloxy)quinolin-2(1H)-one oxalate608Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93671D4CLONEDHUMAN125I-IABNARIPIPRAZOLE168Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93672D3CLONEDHUMAN125I-IABNARIPIPRAZOLE6.8Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93673D2CLONEDHUMAN125I-IABNARIPIPRAZOLE3.1Vangveravong S et al 2011Jan 15, 2025Jan 28, 2025
93674A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester744Federico S et al 2018Jan 15, 2025Jan 15, 2025
93675A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester86.5Federico S et al 2018Jan 15, 2025Jan 15, 2025
93676A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid isopropyl ester2.75Federico S et al 2018Jan 15, 2025Jan 15, 2025
93677A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester7.21Federico S et al 2018Jan 15, 2025Jan 15, 2025
93678A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester114Federico S et al 2018Jan 15, 2025Jan 15, 2025
93679A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzyl ester277Federico S et al 2018Jan 15, 2025Jan 15, 2025
93680A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester48.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93681A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester197Federico S et al 2018Jan 15, 2025Jan 15, 2025
93682A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl ester1.99Federico S et al 2018Jan 15, 2025Jan 15, 2025
93683A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester30.6Federico S et al 2018Jan 15, 2025Jan 15, 2025
93684A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester37.2Federico S et al 2018Jan 15, 2025Jan 15, 2025
93685A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methyl-benzyl ester93.9Federico S et al 2018Jan 15, 2025Jan 15, 2025
93686A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester79.7Federico S et al 2018Jan 15, 2025Jan 15, 2025
93687A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester21Federico S et al 2018Jan 15, 2025Jan 15, 2025
93688A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methyl-benzyl ester10.8Federico S et al 2018Jan 15, 2025Jan 15, 2025
93689A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester3.72Federico S et al 2018Jan 15, 2025Jan 15, 2025
93690A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester62.2Federico S et al 2018Jan 15, 2025Jan 15, 2025
93691A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzyl ester190Federico S et al 2018Jan 15, 2025Jan 15, 2025
93692A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester55.2Federico S et al 2018Jan 15, 2025Jan 15, 2025
93693A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester13.2Federico S et al 2018Jan 15, 2025Jan 15, 2025
93694A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-methoxy-benzyl ester1.71Federico S et al 2018Jan 15, 2025Jan 15, 2025
93695A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester7.42Federico S et al 2018Jan 15, 2025Jan 15, 2025
93696A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester14.9Federico S et al 2018Jan 15, 2025Jan 15, 2025
93697A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-methoxy-benzyl ester34.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93698A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester102Federico S et al 2018Jan 15, 2025Jan 15, 2025
93699A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester194Federico S et al 2018Jan 15, 2025Jan 15, 2025
93700A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzyl ester5.62Federico S et al 2018Jan 15, 2025Jan 15, 2025
93701A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester6.05Federico S et al 2018Jan 15, 2025Jan 15, 2025
93702A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester32Federico S et al 2018Jan 15, 2025Jan 15, 2025
93703A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-chloro-benzyl ester348Federico S et al 2018Jan 15, 2025Jan 15, 2025
93704A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester26.4Federico S et al 2018Jan 15, 2025Jan 15, 2025
93705A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester15.7Federico S et al 2018Jan 15, 2025Jan 15, 2025
93706A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-chloro-benzyl ester6.73Federico S et al 2018Jan 15, 2025Jan 15, 2025
93707A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester4.88Federico S et al 2018Jan 15, 2025Jan 15, 2025
93708A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester71.9Federico S et al 2018Jan 15, 2025Jan 15, 2025
93709A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzyl ester216Federico S et al 2018Jan 15, 2025Jan 15, 2025
93710A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester313Federico S et al 2018Jan 15, 2025Jan 15, 2025
93711A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester24.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93712A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 2-bromo-benzyl ester14.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93713A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester3.37Federico S et al 2018Jan 15, 2025Jan 15, 2025
93714A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester32.5Federico S et al 2018Jan 15, 2025Jan 15, 2025
93715A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3-fluoro-benzyl ester130Federico S et al 2018Jan 15, 2025Jan 15, 2025
93716A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester556Federico S et al 2018Jan 15, 2025Jan 15, 2025
93717A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester71.5Federico S et al 2018Jan 15, 2025Jan 15, 2025
93718A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzyl ester5.21Federico S et al 2018Jan 15, 2025Jan 15, 2025
93719A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester1.21Federico S et al 2018Jan 15, 2025Jan 15, 2025
93720A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester21Federico S et al 2018Jan 15, 2025Jan 15, 2025
93721A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-ethyl-benzyl ester119Federico S et al 2018Jan 15, 2025Jan 15, 2025
93722A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester51Federico S et al 2018Jan 15, 2025Jan 15, 2025
93723A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester11Federico S et al 2018Jan 15, 2025Jan 15, 2025
93724A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 1-methyl-2-phenyl-ethyl ester3.19Federico S et al 2018Jan 15, 2025Jan 15, 2025
93725A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide3.73Federico S et al 2018Jan 15, 2025Jan 15, 2025
93726A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide18.6Federico S et al 2018Jan 15, 2025Jan 15, 2025
93727A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzylamide23.4Federico S et al 2018Jan 15, 2025Jan 15, 2025
93728A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide28.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93729A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide61.6Federico S et al 2018Jan 15, 2025Jan 15, 2025
93730A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid benzhydryl-amide5.08Federico S et al 2018Jan 15, 2025Jan 15, 2025
93731A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide5.02Federico S et al 2018Jan 15, 2025Jan 15, 2025
93732A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide100Federico S et al 2018Jan 15, 2025Jan 15, 2025
93733A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methyl-benzylamide46.6Federico S et al 2018Jan 15, 2025Jan 15, 2025
93734A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide41Federico S et al 2018Jan 15, 2025Jan 15, 2025
93735A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide81.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93736A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-methoxy-benzylamide12.5Federico S et al 2018Jan 15, 2025Jan 15, 2025
93737A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide15.3Federico S et al 2018Jan 15, 2025Jan 15, 2025
93738A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide2950Federico S et al 2018Jan 15, 2025Jan 15, 2025
93739A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-trifluoromethyl-benzylamide3850Federico S et al 2018Jan 15, 2025Jan 15, 2025
93740A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide137Federico S et al 2018Jan 15, 2025Jan 15, 2025
93741A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide59.4Federico S et al 2018Jan 15, 2025Jan 15, 2025
93742A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-chloro-benzylamide10Federico S et al 2018Jan 15, 2025Jan 15, 2025
93743A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide7.23Federico S et al 2018Jan 15, 2025Jan 15, 2025
93744A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide47.6Federico S et al 2018Jan 15, 2025Jan 15, 2025
93745A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 4-fluoro-benzylamide250Federico S et al 2018Jan 15, 2025Jan 15, 2025
93746A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93747A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide9390Federico S et al 2018Jan 15, 2025Jan 15, 2025
93748A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (biphenyl-4-ylmethyl)-amide521Federico S et al 2018Jan 15, 2025Jan 15, 2025