The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 98,001-98,685 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
100753PDE3aCLONEDHUMANFunctionalRoflumilast>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100754PDE3bCLONEDHUMANFunctionalRoflumilast>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100755PDE4aCLONEDHUMANFunctionalRoflumilast0.2Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100756PDE4bCLONEDHUMANFunctionalRoflumilast0.1Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100757PDE4cCLONEDHUMANFunctionalRoflumilast0.6Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100758PDE4dCLONEDHUMANFunctionalRoflumilast0.1Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100759PDE7aCLONEDHUMANFunctionalRoflumilast>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100760PDE8bCLONEDHUMANFunctionalRoflumilast>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100761PDE1CLONEDHUMANFunctionalL-826,141>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100762PDE3aCLONEDHUMANFunctionalL-826,1412100Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100763PDE3bCLONEDHUMANFunctionalL-826,1411100Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100764PDE4aCLONEDHUMANFunctionalL-826,1411.3Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100765PDE4bCLONEDHUMANFunctionalL-826,1410.4Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100766PDE4cCLONEDHUMANFunctionalL-826,1412.4Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100767PDE4dCLONEDHUMANFunctionalL-826,1410.3Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100768PDE7aCLONEDHUMANFunctionalL-826,141>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100769PDE8bCLONEDHUMANFunctionalL-826,1417200Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100770PDE1CLONEDHUMANFunctionalTrequinsin7800Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100771PDE3aCLONEDHUMANFunctionalTrequinsin0.04Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100772PDE3bCLONEDHUMANFunctionalTrequinsin0.05Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100773PDE4aCLONEDHUMANFunctionalTrequinsin360Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100774PDE4bCLONEDHUMANFunctionalTrequinsin437Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100775PDE4cCLONEDHUMANFunctionalTrequinsin790Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100776PDE4dCLONEDHUMANFunctionalTrequinsin230Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100777PDE7aCLONEDHUMANFunctionalTrequinsin9000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100778PDE8bCLONEDHUMANFunctionalTrequinsin2100Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100779PDE1CLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide4200Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100780PDE3aCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100781PDE3bCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100782PDE4aCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide315Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100783PDE4bCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide200Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100784PDE4cCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide970Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100785PDE4dCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide1.4Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100786PDE7aCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100787PDE8bCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1S)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100788PDE1CLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide5300Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100789PDE3aCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100790PDE3bCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100791PDE4aCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide156Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100792PDE4bCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide76Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100793PDE4cCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide1160Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100794PDE4dCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide39Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100795PDE7aCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100796PDE8bCLONEDHUMANFunctional2-(4-fluorophenoxy)-N-[(1R)-1-(4-methoxyphenyl)ethyl]nicotinamide>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025
100797mGluR5CLONEDHUMANFunctionalGlutamate27Kinney GG, et al., 2005Jan 15, 2025Jan 28, 2025
100798mGluR5CLONEDHUMANFunctional3,5-DHPG29.4Kinney GG, et al., 2005Jan 15, 2025Jan 28, 2025
100799mGluR5CLONEDHUMANFunctionalQuisqualate47.6Kinney GG, et al., 2005Jan 15, 2025Jan 28, 2025
100800mGluR5CLONEDRATFunctionalGlutamate113Kinney GG, et al., 2005Jan 15, 2025Jan 28, 2025
100801mGluR5CLONEDRATFunctional3,5-DHPG95.3Kinney GG, et al., 2005Jan 15, 2025Jan 28, 2025
100802mGluR5CLONEDRATFunctionalQuisqualate153Kinney GG, et al., 2005Jan 15, 2025Jan 28, 2025
100803CLONEDHUMANFunctional1,3-bis(2-chloroethyl)-1-nitrosourea14.5Kuo CC, et al., 2006Jan 15, 2025Jan 15, 2025
100804CLONEDHUMANFunctionalcamptothecin40.5Kuo CC, et al., 2006Jan 15, 2025Jan 15, 2025
100805CLONEDHUMANFunctional7-ethyl-10-hydrocamptothecin31Kuo CC, et al., 2006Jan 15, 2025Jan 15, 2025
100806CLONEDHUMANFunctionalTopotecan90Kuo CC, et al., 2006Jan 15, 2025Jan 15, 2025
100807nAChRCLONEDHUMAN3H-EpibatidineEpibatidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100808nAChRCLONEDHUMAN3H-EpibatidineCytisine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100809nAChRCLONEDHUMAN3H-EpibatidineLobeline>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100810nAChRCLONEDHUMAN3H-EpibatidineNicotine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100811nAChRCLONEDHUMAN3H-EpibatidineSuberyldicholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100812nAChRCLONEDHUMAN3H-EpibatidineAcetylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100813nAChRCLONEDHUMAN3H-Epibatidinedimethyl-phenyl-piperazinium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100814nAChRCLONEDHUMAN3H-EpibatidineDihydro-Beta-erythroidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100815nAChRCLONEDHUMAN3H-EpibatidineCarbamylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100816nAChRCLONEDHUMAN3H-EpibatidineDecamethonium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100817nAChRCLONEDHUMAN3H-EpibatidineMethyllycaconitine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100818nAChRCLONEDHUMAN3H-Epibatidined-Tubocurarine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100819nAChRCLONEDHUMAN3H-EpibatidineHEXAMETHONIUM>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100820nAChRCLONEDHUMAN3H-EpibatidinePancuronium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100821nAChRCLONEDHUMAN3H-EpibatidineMecamylamine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100822nAChRCLONEDHUMAN3H-EpibatidineEpibatidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100823nAChRCLONEDHUMAN3H-EpibatidineCytisine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100824nAChRCLONEDHUMAN3H-EpibatidineLobeline>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100825nAChRCLONEDHUMAN3H-EpibatidineNicotine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100826nAChRCLONEDHUMAN3H-EpibatidineSuberyldicholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100827nAChRCLONEDHUMAN3H-EpibatidineAcetylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100828nAChRCLONEDHUMAN3H-Epibatidinedimethyl-phenyl-piperazinium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100829nAChRCLONEDHUMAN3H-EpibatidineDihydro-alpha-ergocryptine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100830nAChRCLONEDHUMAN3H-EpibatidineCarbamylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100831nAChRCLONEDHUMAN3H-EpibatidineDecamethonium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100832nAChRCLONEDHUMAN3H-EpibatidineMethyllycaconitine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100833nAChRCLONEDHUMAN3H-Epibatidined-Tubocurarine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100834nAChRCLONEDHUMAN3H-EpibatidineTrimethaphan>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100835nAChRCLONEDHUMAN3H-EpibatidineHEXAMETHONIUM>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100836nAChRCLONEDHUMAN3H-EpibatidinePancuronium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100837nAChRCLONEDHUMAN3H-EpibatidineMecamylamine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100838nAChRCLONEDHUMANFunctionalEpibatidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100839nAChRCLONEDHUMANFunctionalNicotine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100840nAChRCLONEDHUMANFunctionalAcetylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100841nAChRCLONEDHUMANFunctionalCytisine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100842nAChRCLONEDHUMANFunctionaldimethyl-phenyl-piperazinium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100843nAChRCLONEDHUMANFunctionalCarbamylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100844nAChRCLONEDHUMANFunctionalEpibatidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100845nAChRCLONEDHUMANFunctionalNicotine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100846nAChRCLONEDHUMANFunctionalAcetylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100847nAChRCLONEDHUMANFunctionalCytisine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100848nAChRCLONEDHUMANFunctionaldimethyl-phenyl-piperazinium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100849nAChRCLONEDHUMANFunctionalCarbamylcholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100850nAChRCLONEDHUMANFunctionalMecamylamine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100851nAChRCLONEDHUMANFunctionalDihydro-Beta-erythroidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100852nAChRCLONEDHUMANFunctionalMethyllycaconitine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100853nAChRCLONEDHUMANFunctionalLobeline>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100854nAChRCLONEDHUMANFunctionalTrimethaphan>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100855nAChRCLONEDHUMANFunctionalHEXAMETHONIUM>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100856nAChRCLONEDHUMANFunctionald-Tubocurarine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100857nAChRCLONEDHUMANFunctionalSuberyldicholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100858nAChRCLONEDHUMANFunctionalDecamethonium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100859nAChRCLONEDHUMANFunctionalPancuronium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 15, 2025
100860nAChRCLONEDHUMANFunctionalMecamylamine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100861nAChRCLONEDHUMANFunctionalDihydro-Beta-erythroidine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100862nAChRCLONEDHUMANFunctionalMethyllycaconitine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100863nAChRCLONEDHUMANFunctionalLobeline>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100864nAChRCLONEDHUMANFunctionalTrimethaphan>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100865nAChRCLONEDHUMANFunctionalHEXAMETHONIUM>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100866nAChRCLONEDHUMANFunctionald-Tubocurarine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100867nAChRCLONEDHUMANFunctionalSuberyldicholine>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100868nAChRCLONEDHUMANFunctionalDecamethonium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
100869nAChRCLONEDHUMANFunctionalPancuronium>10000Kuo YP, et al., 2005Jan 15, 2025Jan 29, 2025
1008705-HT1ACLONEDHUMAN3H-WAY1006351-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1)85.7Stephenson, K. et. al., 2008Jan 15, 2025Jan 15, 2025
100871Beta2CLONEDHUMAN3H-CGP-121771-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)2Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
100872Beta2CLONEDHUMAN3H-CGP-121771-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1)2Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
100873Beta1CLONEDHUMAN125I-Pindolol1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2R,2S)-1)6Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
100874Beta1CLONEDHUMAN125I-Pindolol1-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)7Stephenson, K. et. al., 2008Jan 15, 2025Jan 28, 2025
1008755-HT1ACLONEDHUMAN3H-WAY1006351-1(1-Fluoropropan-2-ylamino)-3-(20cyclohexlpheonxy)propan-2-ol ((2S)-1)24.6Stephenson, K. et. al., 2008Jan 15, 2025Jan 15, 2025
100876AChEBRAINHUMANFunctionalTacrine167Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100877AChEBRAINHUMANFunctional3-(1H-Indol-3-yl)-N-[5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]propionamide70Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100878BchEserumHUMANFunctionalTacrine24Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100879BchEserumHUMANFunctional3-(1H-Indol-3-yl)-N-[5-(1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]propionamide1Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100880AChEBRAINHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-3-(1H-indol-3-yl)propionamide4Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100881BchEserumHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-3-(1H-indol-3-yl)propionamide16Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100882AChEBRAINHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)propionamide0.02Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100883BchEserumHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)propionamide2.9Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100884BchEserumHUMANFunctionalN-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide0.1Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100885AChEBRAINHUMANFunctionalN-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide0.06Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100886AChEBRAINHUMANFunctionalN-[8-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)octyl]-3-(1H-indol-3-yl)propionamide0.5Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100887BchEserumHUMANFunctionalN-[8-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)octyl]-3-(1H-indol-3-yl)propionamide5.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100888AChEBRAINHUMANFunctionalN-[9-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)nonyl]-3-(1H-indol-3-yl)propionamide4.4Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100889BchEserumHUMANFunctionalN-[9-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)nonyl]-3-(1H-indol-3-yl)propionamide9.6Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100890BchEserumHUMANFunctionalN-[10-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)decyl]-3-(1H-indol-3-yl)propionamide54Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100891AChEBRAINHUMANFunctionalN-(3-{[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-methylamino}propyl)-3-(1H-indol-3-yl)propionamide147Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100892BchEserumHUMANFunctionalN-(3-{[3-(1,2,3,4-tetrahydroacridin-9-ylamino)propyl]-methylamino}propyl)-3-(1H-indol-3-yl)propionamide0.03Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100893AChEBRAINHUMANFunctionalN-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide2.9Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100894BchEserumHUMANFunctionalN-(3-{[3-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)propyl]methylamino}propyl)-3-(1H-indol-3-yl)propionamide21.4Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100895AChEBRAINHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(5-cyano-1H-indol-3-yl)propionamide0.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100896BchEserumHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(5-cyano-1H-indol-3-yl)propionamide11.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100897AChEBRAINHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)acrylamide18Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100898BchEserumHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)acrylamide77Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100899AChEBRAINHUMANFunctional1H-Indole-3-carboxylic acid [5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]amide180Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100900BchEserumHUMANFunctional1H-Indole-3-carboxylic acid [5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]amide9.5Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100901AChEBRAINHUMANFunctional1H-indole-3-carboxylic acid [6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]amide33Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100902BchEserumHUMANFunctional1H-indole-3-carboxylic acid [6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]amide1.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100903AChEBRAINHUMANFunctional1H-indole-3-carboxylic acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide36Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100904BchEserumHUMANFunctional1H-indole-3-carboxylic acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide19Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100905AChEBRAINHUMANFunctional1H-indole-3-carboxylic acid [8-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)octyl]amide46Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100906BchEserumHUMANFunctional1H-indole-3-carboxylic acid [8-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)octyl]amide22.4Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100907AChEBRAINHUMANFunctionalN-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-2-(1H-indol-3-yl)acetamide0.2Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100908BchEserumHUMANFunctionalN-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-2-(1H-indol-3-yl)acetamide11.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100909AChEBRAINHUMANFunctional2-(5-Bromo-1H-indol-3-yl)-N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]acetamide0.6Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100910BchEserumHUMANFunctional2-(5-Bromo-1H-indol-3-yl)-N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]acetamide1.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100911AChEBRAINHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-4-(1H-indol-3-yl)butyramide0.3Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100912BchEserumHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-4-(1H-indol-3-yl)butyramide3.2Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100913AChEBRAINHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-4-(1H-indol-3-yl)butyramide0.5Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100914BchEserumHUMANFunctionalN-[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-4-(1H-indol-3-yl)butyramide5.6Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100915AChEBRAINHUMANFunctional1H-Methylindole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide10.9Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100916BchEserumHUMANFunctional1H-Methylindole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide206Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100917AChEBRAINHUMANFunctional1H-indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide95Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100918BchEserumHUMANFunctional1H-indazole-3-carboxylic Acid [7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]amide79Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100919AChEBRAINHUMANFunctional[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]carbamic acid 2-(1H-indol-3-yl)ethyl Ester1.5Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100920BchEserumHUMANFunctional[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]carbamic acid 2-(1H-indol-3-yl)ethyl Ester136Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100921AChEBRAINHUMANFunctional[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]carbamic acid 2-(1H-indol-3-yl)ethyl ester0.7Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100922BchEserumHUMANFunctional[6-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]carbamic acid 2-(1H-indol-3-yl)ethyl ester60Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100923AChEBRAINHUMANFunctional[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]carbamic acid 2-(1H-indol-3-yl)ethyl ester3Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100924BchEserumHUMANFunctional[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]carbamic acid 2-(1H-indol-3-yl)ethyl ester59Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 15, 2025
100925AChEBRAINHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-3-(1H-indol-3-yl)propionamide0.014Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100926AChEBRAINHUMANFunctionalN-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-3-(1H-indol-3-yl)propionamide0.009Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100927AChEBRAINHUMANFunctionalN-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]-2-(1H-indol-3-yl)acetamide0.015Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100928AChEBRAINHUMANFunctional2-(5-Bromo-1H-indol-3-yl)-N-[7-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)heptyl]acetamide0.02Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100929AChEBRAINHUMANFunctionalN-[5-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)pentyl]-4-(1H-indol-3-yl)butyramide0.0017Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100930Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)Pentazocine,(+/-)3.09Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100931Sigma 2LIVERRAT3H-DTGDTG25.7Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100932AChEserumHUMANFunctionalN-[10-(6-Chloro-1,2,3,4-tetrahydroacridin-9-ylamino)decyl]-3-(1H-indol-3-yl)propionamide21.9Munoz-Ruiz P, et al., 2005Jan 15, 2025Jan 29, 2025
100933NETCELLSHEK293FunctionalCOCAINE272Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100934NETCELLSHEK293FunctionalCFT80Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100935NETCELLSHEK293FunctionalCIT2.63Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100936NETCELLSHEK293FunctionalBENZTROPINE390Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100937NETCELLSHEK293FunctionalGBR-12909261Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100938NETCELLSHEK293FunctionalNisoxetine8.96Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100939NETCELLSHEK293FunctionalDESIPRAMINE2.26Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100940NETCELLSHEK293FunctionalMAZINDOL2.84Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100941NETCELLSHEK2933H-NisoxetineCOCAINE3960Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100942NETCELLSHEK2933H-NisoxetineCFT1161Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100943NETCELLSHEK2933H-NisoxetineCIT47.6Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100944NETCELLSHEK2933H-NisoxetineBENZTROPINE3823Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100945NETCELLSHEK2933H-NisoxetineGBR-129091889Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100946NETCELLSHEK2933H-NisoxetineNisoxetine12Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100947NETCELLSHEK2933H-NisoxetineDESIPRAMINE3.54Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100948NETCELLSHEK2933H-NisoxetineMAZINDOL2.17Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100949NETCELLSHEK2933H-CITCOCAINE727Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100950NETCELLSHEK2933H-CITCFT264Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100951NETCELLSHEK2933H-CITCIT7.17Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100952NETCELLSHEK2933H-CITBENZTROPINE406Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100953NETCELLSHEK2933H-CITGBR-12909737Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100954NETCELLSHEK2933H-CITNisoxetine1.73Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100955NETCELLSHEK2933H-CITDESIPRAMINE2.21Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
100956NETCELLSHEK2933H-CITMAZINDOL0.738Reith ME, et al., 2005Jan 15, 2025Jan 15, 2025
1009575-HT2ACLONEDHUMAN3H-KETANSERINLumateperone0.5Snyder et al., 2015Jan 15, 2025Jan 15, 2025
100958D2CLONEDHUMAN3H-N-MethylspiperoneLumateperone32Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100959D1CLONEDHUMAN3H-SCH23390Lumateperone52Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100960SERTCLONEDHUMAN3H-CITALOPRAMLumateperone62Snyder et al., 2015Jan 15, 2025Jan 28, 2025
1009615-HT2ACLONEDHUMAN3H-KETANSERINRISPERIDONE0.5Snyder et al., 2015Jan 15, 2025Jan 15, 2025
100962D2CLONEDHUMAN3H-N-MethylspiperoneRISPERIDONE5.9Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100963D1CLONEDHUMAN3H-SCH23390RISPERIDONE564Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100964SERTCLONEDHUMAN3H-CITALOPRAMRISPERIDONE1000Snyder et al., 2015Jan 15, 2025Jan 28, 2025
1009655-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE2.5Snyder et al., 2015Jan 15, 2025Jan 15, 2025
100966D2CLONEDHUMAN3H-N-MethylspiperoneOLANZAPINE31Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100967D1CLONEDHUMAN3H-SCH23390OLANZAPINE128Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100968SERTCLONEDHUMAN3H-CITALOPRAMOLANZAPINE1000Snyder et al., 2015Jan 15, 2025Jan 28, 2025
1009695-HT2ACLONEDHUMAN3H-KETANSERINARIPIPRAZOLE9Snyder et al., 2015Jan 15, 2025Jan 15, 2025
100970D2CLONEDHUMAN3H-MethylspiperoneARIPIPRAZOLE1.6Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100971D1CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE1170Snyder et al., 2015Jan 15, 2025Jan 28, 2025
1009725-HT2ACLONEDHUMAN3H-KETANSERINFLUOXETINE141Snyder et al., 2015Jan 15, 2025Jan 15, 2025
100973D2CLONEDHUMAN3H-N-MethylspiperoneFLUOXETINE>10000Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100974D1CLONEDHUMAN3H-SCH23390FLUOXETINE>10000Snyder et al., 2015Jan 15, 2025Jan 28, 2025
100975OT1CLONEDHUMAN125I-Orexin-A(E)-N-((3R,3aR,3a1S,9aS)-9-(N-(cyclopropylmethyl)phenylsulfonamido)-9a-hydroxy-5-methoxy-1,2,3,3a,3a1,8,9,9a-octahydrophenanthro[4,5-bcd]furan-3-yl)-3-(furan-3-yl)-N-methylacrylamide101Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100976OT1CLONEDHUMAN125I-Orexin-A(E)-N-((3R,3aR,3a1S,9aR)-9-(N-(cyclopropylmethyl)phenylsulfonamido)-5-methoxy-1,2,3,3a,3a1,8,9,9a-octahydrophenanthro[4,5-bcd]furan-3-yl)-3-(furan-3-yl)-N-methylacrylamide20.9Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100977OT1CLONEDHUMAN125I-Orexin-A(E)-N-((3R,4aR,10R,10aS)-10-(N-(cyclopropylmethyl)phenylsulfonamido)-10a-hydroxy-6-methoxy-1,2,3,4,4a,9,10,10a-octahydrophenanthren-3-yl)-3-(furan-3-yl)-N-methylacrylamide842Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100978OT1CLONEDHUMAN125I-Orexin-AYNT-7078.14Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100979OT1CLONEDHUMAN125I-Orexin-AYNT-1369849Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100980OT1CLONEDHUMAN125I-Orexin-AYNT-81611.2Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100981OT2CLONEDHUMAN125I-Orexin-AYNT-816294Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100982OT1CLONEDHUMAN125I-Orexin-AYNT-81731.6Saitoh T et al., 2019Jan 15, 2025Jan 15, 2025
100983SERTCLONEDHUMAN125I-RTI-551, (S)-citalopram1.77Yarravarapu N, et. al., 2018Jan 15, 2025Jan 28, 2025
100984SERTCLONEDHUMAN125I-RTI-55(S)-1-(4-Fluorophenyl)-1-(3-(methyl(4-(4-(prop-2-yn-1-yloxy)benzoyl)benzyl)amino)propyl)-1,3-dihydroisobenzofuran-5-carbonitrile487Yarravarapu N, et. al., 2018Jan 15, 2025Jan 28, 2025
100985SERTCLONEDHUMAN125I-RTI-55(S)-N-((1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-yl)methyl)-4-(4-(prop-2-yn-1-yloxy)benzoyl)benzamide0.16Yarravarapu N, et. al., 2018Jan 15, 2025Jan 28, 2025
100986SERTCLONEDHUMAN125I-RTI-55(S)-3-Azido-5-(azidomethyl)-N-((1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-5-yl)methyl)benzamide10.7Yarravarapu N, et. al., 2018Jan 15, 2025Jan 28, 2025
1009875-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-fluorophenyl)-N-(3,4- dimethoxyphenethyl)propan-1-amine185Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009885-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-fluorophenyl)-N-(3,4- dimethoxyphenethyl)propan-1-amine14Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009895-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-fluorophenyl)-N-(3,4- dimethoxyphenethyl)propan-1-amine126Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009905-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine365Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009915-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine54Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009925-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine235Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009935-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine221Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009945-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine45Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009955-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine219Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009965-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine288Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009975-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine51Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009985-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(4-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine224Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1009995-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine185Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010005-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine18Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010015-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine167Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010025-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine125Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010035-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine17Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010045-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine206Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010055-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine103Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010065-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine14Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010075-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine143Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010085-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine169Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010095-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine18Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010105-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(3-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine154Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010115-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine65Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010125-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine1.7Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010135-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-fluorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine79Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010145-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine43Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010155-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine3.1Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010165-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-chlorophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine92Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010175-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine54Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010185-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine3.4Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010195-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-bromophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine124Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010205-HT2ACLONEDHUMAN3H- KetanserinN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine75Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010215-HT2BCLONEDHUMAN3H- LSDN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine13Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010225-HT2CCLONEDHUMAN3H-MESULERGINEN-(2-(benzo[d][1,3]dioxol-5-yl)ethyl)-3-(2-iodophenyl)-N-(3,4-dimethoxyphenethyl)propan-1-amine68Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010235-HT2ACLONEDHUMAN3H- KetanserinCLOZAPINE15Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010245-HT2BCLONEDHUMAN3H- LSDSB 20655321Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010255-HT2CCLONEDHUMAN3H-MESULERGINERITANSERIN1.8Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010265-HT2ACLONEDHUMAN3H- Ketanserin1,2-dimethoxy-4-propylbenzene; 2-(2H-1,3-benzodioxol-5-yl)ethan-1-amine; butylbenzene165Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010275-HT2BCLONEDHUMAN3H- LSD1,2-dimethoxy-4-propylbenzene; 2-(2H-1,3-benzodioxol-5-yl)ethan-1-amine; butylbenzene26Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
1010285-HT2CCLONEDHUMAN3H-MESULERGINE1,2-dimethoxy-4-propylbenzene; 2-(2H-1,3-benzodioxol-5-yl)ethan-1-amine; butylbenzene399Kapadia N et al 2016Jan 15, 2025Jan 15, 2025
101029A1CLONEDHUMAN3H-DPCPX5-Ethyl-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one782Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101030A2ACLONEDHUMAN3H-ZM2413855-Ethyl-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one2869Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101031A1CLONEDHUMAN3H-DPCPX5-Isopropyl-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one912Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101032A1CLONEDHUMAN3H-DPCPX5-Ethyl-7-(thiophen-2-yl)thieno[2,3-d]pyridazin-4(5H)-one724Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101033A1CLONEDHUMAN3H-DPCPX5-Ethyl-7-phenylthieno[2,3-d]pyridazin-4(5H)-one2665Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101034A3CLONEDHUMAN125I-AB-MECA5-Ethyl-7-phenylthieno[2,3-d]pyridazin-4(5H)-one2590Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101035A1CLONEDHUMAN3H-DPCPX5-Ethyl-7-(thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one113Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101036A2ACLONEDHUMAN3H-ZM2413855-Ethyl-7-(thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one2487Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101037A3CLONEDHUMAN125I-AB-MECA5-Ethyl-7-(thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one2928Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101038A1CLONEDHUMAN3H-DPCPX7-(Thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one1153Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101039A2ACLONEDHUMAN3H-ZM2413857-(Thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one3392Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101040A1CLONEDHUMAN3H-DPCPX5-Amino-7-(pyridin-2-yl)thieno[2,3-d]pyridazin-4(5H)-one3721Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101041A1CLONEDHUMAN3H-DPCPX5-Amino-7-(thiophen-2-yl)thieno[2,3-d]pyridazin-4(5H)-one3535Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101042A1CLONEDHUMAN3H-DPCPX5-Amino-7-(thiazol-2-yl)thieno[2,3-d]pyridazin-4(5H)-one2874Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101043A2ACLONEDHUMAN3H-ZM2413855,7-diethyl-2-phenylthieno[2,3-d]pyridazin-4(5H)-one3141Catarzi D, et al., 2018Jan 15, 2025Jan 15, 2025
101044Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-benzylpiperidin-4-yl)methyl)-N-propylacetamide36.8Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101045Sigma 2LIVERRAT3H-DTGN-((1-benzylpiperidin-4-yl)methyl)-N-butylacetamide1257Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101046Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-benzylpiperidin-4-yl)methyl)-N-butylacetamide67Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101047Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-benzylpiperidin-4-yl)methyl)-N-pentylacetamide17Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101048Sigma 2LIVERRAT3H-DTGN-((1-benzylpiperidin-4-yl)methyl)-N-pentylacetamide1117Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101049Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-benzylpiperidin-4-yl)methyl)-N-(cyclohexylmethy)acetamide58.5Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101050Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-ethylacetamide228Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101051Sigma 2LIVERRAT3H-DTGN-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-propylacetamide987Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101052Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-propylacetamide77.4Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101053Sigma 1LIVERRAT3H-Pentazocine(+)N-butyl-N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)acetamide 34.4Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101054Sigma 2LIVERRAT3H-DTGN-butyl-N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)acetamide 1377Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101055Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-pentylacetamide31.8Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101056Sigma 2LIVERRAT3H-DTGN-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-pentylacetamide825Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101057Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-(cyclohexylmethyl)acetamide95.3Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101058Sigma 2LIVERRAT3H-DTGN-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)-N-(cyclohexylmethyl)acetamide2425Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101059Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-ethylacetamide285Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101060Sigma 2LIVERRAT3H-DTGN-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-ethylacetamide19.6Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101061Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-propylacetamide143Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101062Sigma 2LIVERRAT3H-DTGN-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-propylacetamide2583Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101063Sigma 1LIVERRAT3H-Pentazocine(+)N-butyl-N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)acetamide75.9Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101064Sigma 2LIVERRAT3H-DTGN-butyl-N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)acetamide1837Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101065Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-pentylacetamide187Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101066Sigma 2LIVERRAT3H-DTGN-((1-(2,4-dichlorobenzyl)piperidin-4-yl)methyl)-N-pentylacetamide3204Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101067Sigma 1LIVERRAT3H-Pentazocine(+)N-(cyclohexylmethyl)-N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)acetamide51.9Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101068Sigma 2LIVERRAT3H-DTGN-(cyclohexylmethyl)-N-((1-(4-chlorobenzyl)piperidin-4-yl)methyl)acetamide2343Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101069Sigma 1LIVERRAT3H-Pentazocine(+)N-((1-benzylpiperidin-4-yl)methyl)-N-ethylacetamide97.2Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
101070Sigma 2LIVERRAT3H-DTGN-((1-benzylpiperidin-4-yl)methyl)-N-ethylacetamide422Zampieri D, et al., 2018Jan 15, 2025Jan 28, 2025
1010715-HT6CLONEDHUMAN3H-LSD1-methyl-4-[1-(2-methylpropanesulfonyl)-4-phenyl-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate16Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101072D2CLONEDHUMAN3H-N-Methylspiperone1-methyl-4-[1-(2-methylpropanesulfonyl)-4-phenyl-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate547Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010735-HT6CLONEDHUMAN3H-LSD1-[4-(4-ethylphenyl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Fumarate11Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101074D2CLONEDHUMAN3H-N-Methylspiperone1-[4-(4-ethylphenyl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Fumarate614Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010755-HT6CLONEDHUMAN3H-LSD1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate4Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101076D2CLONEDHUMAN3H-N-Methylspiperone1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[4-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate367Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010775-HT6CLONEDHUMAN3H-LSD1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[3-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate48Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101078D2CLONEDHUMAN3H-N-Methylspiperone1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[3-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate630Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010795-HT6CLONEDHUMAN3H-LSD1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[2-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate24Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101080D2CLONEDHUMAN3H-N-Methylspiperone1-methyl-4-[1-(2-methylpropanesulfonyl)-4-[2-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate113Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010815-HT6CLONEDHUMAN3H-LSD1-[4-(4-methoxyphenyl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Fumarate2Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101082D2CLONEDHUMAN3H-N-Methylspiperone1-[4-(4-methoxyphenyl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Fumarate22Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010835-HT6CLONEDHUMAN3H-LSD1-{4-[4-(benzyloxy)phenyl]-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-methylpiperazine Fumarate290Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101084D2CLONEDHUMAN3H-N-Methylspiperone1-{4-[4-(benzyloxy)phenyl]-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-methylpiperazine Fumarate86Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010855-HT6CLONEDHUMAN3H-LSD4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenol Fumarate22Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101086D2CLONEDHUMAN3H-N-Methylspiperone4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenol Fumarate108Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010875-HT6CLONEDHUMAN3H-LSD4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzonitrile Hydrobromide7Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101088D2CLONEDHUMAN3H-N-Methylspiperone4-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzonitrile Hydrobromide205Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010895-HT6CLONEDHUMAN3H- LSD5-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-indole Hydrochloride5Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101090D2CLONEDHUMAN3H-N-Methylspiperone5-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-indole Hydrochloride382Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010915-HT6CLONEDHUMAN3H-LSD1-methyl-4-[1-(2-methylpropanesulfonyl)-4-(pyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate36Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
1010925-HT6CLONEDHUMAN3H-LSD5-[6-(4-methylpiperazin-1-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2-dihydropyridin-2-one Hydrobromide231Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
1010935-HT6CLONEDHUMAN3H-LSD1-methyl-4-[4-(1-methyl-1H-pyrazol-4-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperazine Fumarate87Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
1010945-HT6CLONEDHUMAN3H-LSD1-[4-(2,5-dimethylthiophen-3-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Hydrobromide12Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101095D2CLONEDHUMAN3H-N-Methylspiperone1-[4-(2,5-dimethylthiophen-3-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Hydrobromide640Fabritius C, et al., 2016Jan 15, 2025Jan 28, 2025
1010965-HT6CLONEDHUMAN3H-LSD1-[4-(dimethyl-1,2-oxazol-4-yl)-1-(2-methylpropanesulfonyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]-4-methylpiperazine Hydrobromide129Fabritius C, et al., 2016Jan 15, 2025Jan 15, 2025
101097Sigma 1LIVERRAT3H-Pentazocine(+)1-Benzoyl-9-benzyl-4-cyclohexyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione7.2Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101098Sigma 2BRAINGUINEA PIG3H-DTG1-Benzoyl-9-benzyl-4-cyclohexyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione248Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101099Sigma 1LIVERRAT3H-Pentazocine(+)9-Benzyl-4-cyclohexyl-1-(4-methylbenzoyl)-1,4,9-triazaspiro[5.5]undecane-3,5-dione11.1Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101100Sigma 2BRAINGUINEA PIG3H-DTG9-Benzyl-4-cyclohexyl-1-(4-methylbenzoyl)-1,4,9-triazaspiro[5.5]undecane-3,5-dione134Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101101Sigma 1LIVERRAT3H-Pentazocine(+)9-Benzyl-4-cyclohexyl-1-(4-methoxybenzoyl)-1,4,9-triazaspiro[5.5]undecane-3,5-dione5.9Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101102Sigma 2BRAINGUINEA PIG3H-DTG9-Benzyl-4-cyclohexyl-1-(4-methoxybenzoyl)-1,4,9-triazaspiro[5.5]undecane-3,5-dione563Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101103Sigma 1LIVERRAT3H-Pentazocine(+)6-Benzoyl-9-cyclohexyl-6,9-diazaspiro[4.5]decane-8,10-dione79.8Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101104Sigma 2BRAINGUINEA PIG3H-DTG6-Benzoyl-9-cyclohexyl-6,9-diazaspiro[4.5]decane-8,10-dione118Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101105Sigma 1LIVERRAT3H-Pentazocine(+)9-Cyclohexyl-6-(4-methylbenzoyl)-6,9-diazaspiro[4.5]decane-8,10-dione189Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101106Sigma 2BRAINGUINEA PIG3H-DTG9-Cyclohexyl-6-(4-methylbenzoyl)-6,9-diazaspiro[4.5]decane-8,10-dione134Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101107Sigma 1LIVERRAT3H-Pentazocine(+)9-Cyclohexyl-6-(4-methoxybenzoyl)-6,9-diazaspiro[4.5]decane-8,10-dione429Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101108Sigma 2BRAINGUINEA PIG3H-DTG9-Cyclohexyl-6-(4-methoxybenzoyl)-6,9-diazaspiro[4.5]decane-8,10-dione98Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101109Sigma 1LIVERRAT3H-Pentazocine(+)1-Benzoyl-4-cyclohexyl-1,4-diazaspiro[5.5]undecane-3,5-dione227Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101110Sigma 2BRAINGUINEA PIG3H-DTG1-Benzoyl-4-cyclohexyl-1,4-diazaspiro[5.5]undecane-3,5-dione138Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101111Sigma 1LIVERRAT3H-Pentazocine(+)4-Cyclohexyl-1-(4-methylbenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione399Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101112Sigma 2BRAINGUINEA PIG3H-DTG4-Cyclohexyl-1-(4-methylbenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione2189Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101113Sigma 1LIVERRAT3H-Pentazocine(+)4-Cyclohexyl-1-(4-methoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione1370Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101114Sigma 2BRAINGUINEA PIG3H-DTG4-Cyclohexyl-1-(4-methoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione5381Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101115Sigma 1LIVERRAT3H-Pentazocine(+)4-Cyclohexyl-1-(2,4-dimethoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione968Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101116Sigma 2BRAINGUINEA PIG3H-DTG4-Cyclohexyl-1-(2,4-dimethoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione3174Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101117Sigma 1LIVERRAT3H-Pentazocine(+)1-Benzoyl-9-tert-butyl-4-cyclohexyl-1,4-diazaspiro[5.5]undecane-3,5-dione7896Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101118Sigma 1LIVERRAT3H-Pentazocine(+)9-tert-Butyl-4-cyclohexyl-1-(4-methoxybenzoyl)-1,4-diazaspiro[5.5]undecane-3,5-dione9365Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101119Sigma 1LIVERRAT3H-Pentazocine(+)HALOPERIDOL3.6Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101120Sigma 2BRAINGUINEA PIG3H-DTGHALOPERIDOL54.5Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101121Sigma 1LIVERRAT3H-Pentazocine(+)PENTAZOCINE (+)5Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101122Sigma 2BRAINGUINEA PIG3H-DTGPENTAZOCINE (+)1824Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101123Sigma 1LIVERRAT3H-Pentazocine(+)DTG36.7Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101124Sigma 2BRAINGUINEA PIG3H-DTGDTG59.1Ghandi M, et al., 2016Jan 15, 2025Jan 28, 2025
101125A1brain membranesRAT3H-DPCPX8-(4-Methoxyphenoxymethyl)caffeine4670Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101126A2AStriatal MembranesRAT3H-NECA8-(4-Methoxyphenoxymethyl)caffeine2400Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101127A2AStriatal MembranesRAT3H-NECA8-(4-Methylphenoxymethyl)caffeine3640Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101128A1brain membranesRAT3H-DPCPX8-(4-Methylphenoxymethyl)caffeine6760Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101129A1brain membranesRAT3H-DPCPX8-(4-Fluorophenoxymethyl)caffeine9190Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101130A2AStriatal MembranesRAT3H-NECA8-(4-Fluorophenoxymethyl)caffeine2570Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101131A1brain membranesRAT3H-DPCPX8-(4-Chlorophenoxymethyl)caffeine5560Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101132A2AStriatal MembranesRAT3H-NECA8-(4-Chlorophenoxymethyl)caffeine940Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101133A2AStriatal MembranesRAT3H-NECA8-(4-Bromophenoxymethyl)caffeine1730Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101134A1brain membranesRAT3H-DPCPX8-(4-Bromophenoxymethyl)caffeine3690Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101135A1brain membranesRAT3H-DPCPX8-(3-Phenylpropyl)-1,3,7-triethylxanthine5610Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101136A2AStriatal MembranesRAT3H-NECA8-(3-Phenylpropyl)-1,3,7-triethylxanthine2690Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101137A2AStriatal MembranesRAT3H-NECA1,3-Diethyl-7-methyl-8-(4-methoxyphenoxymethyl)xanthine237Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101138A1brain membranesRAT3H-DPCPX1,3-Diethyl-7-methyl-8-(4-methoxyphenoxymethyl)xanthine1220Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101139A1brain membranesRAT3H-DPCPX1,3-Diethyl-7-methyl-8-(4-methylphenoxymethyl)xanthine1420Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101140A2AStriatal MembranesRAT3H-NECA1,3-Diethyl-7-methyl-8-(4-methylphenoxymethyl)xanthine1300Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101141A2AStriatal MembranesRAT3H-NECA1,3-Diethyl-7-methyl-8-(4-fluorophenoxymethyl)xanthine841Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101142A1brain membranesRAT3H-DPCPX1,3-Diethyl-7-methyl-8-(4-fluorophenoxymethyl)xanthine1230Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101143A1brain membranesRAT3H-DPCPX1,3-Diethyl-7-methyl-8-(4-chlorophenoxymethyl)xanthine974Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101144A2AStriatal MembranesRAT3H-NECA1,3-Diethyl-7-methyl-8-(4-chlorophenoxymethyl)xanthine1040Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101145A2AStriatal MembranesRAT3H-NECA1,3-Diethyl-7-methyl-8-(4-bromophenoxymethyl)xanthine1360Harmse R et al 2016Jan 15, 2025Jan 15, 2025
101146A1brain membranesRAT3H-DPCPX1,3-Diethyl-7-methyl-8-(4-bromophenoxymethyl)xanthine264Harmse R et al 2016Jan 15, 2025Jan 15, 2025
1011475-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone26.2Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011485-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-(4-phenyl-1-piperazinyl)-1-propanone272Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011495-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone350Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011505-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-5-(4-phenyl-1-piperazinyl)-1-pentanone197Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011515-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone52Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011525-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(phenylmethy)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011535-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone33.5Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011545-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone32.7Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011555-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone462Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011565-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone1684Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011575-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(4-Phenyl-1-piperazinyl)-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone81.8Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011585-HT7CLONEDHUMAN3H-5-HT1-(4-Phenyl-1-piperazinyl)-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone80.3Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011595-HT7CLONEDHUMAN3H-5-HT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-(4-phenyl-1-piperazinyl)-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011605-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-(4-phenyl-1-piperazinyl)-1-propanone1074Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011615-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone101Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011625-HT7CLONEDHUMAN3H-5-HT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone54.7Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011635-HT7CLONEDHUMAN3H-5-HT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone2761Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011645-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(3-chlorophenyl)-1-piperazinyl]-1-propanone142Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011655-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone302Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011665-HT7CLONEDHUMAN3H-5-HT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(4-chlorophenyl)-1-piperazinyl]-1-propanone2366Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011675-HT7CLONEDHUMAN3H-5-HT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone119Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011685-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(3-Chlorophenyl)-1-piperazinyl]-3-[4-(2-ethoxyphenyl)-1-piperazinyl]-1-propanone15.2Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011695-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(4-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011705-HT7CLONEDHUMAN3H-5-HT1-[4-(4-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone36.6Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011715-HT7CLONEDHUMAN3H-5-HT1-[4-(2-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone50.2Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011725-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(2-Chlorophenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011735-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(4-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011745-HT7CLONEDHUMAN3H-5-HT1-[4-(4-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011755-HT7CLONEDHUMAN3H-5-HT1-[4-(2-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone24.2Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011765-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(2-Methoxyphenyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011775-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(2-Pyridyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011785-HT7CLONEDHUMAN3H-5-HT1-[4-(2-Pyrimidyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone23.5Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011795-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[4-(2-Pyrimidyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011805-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(Phenylmethyl)-1-(4-phenyl-1-piperazinyl)propan-1-one938Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011815-HT7CLONEDHUMAN3H-5-HT3-(Phenylmethyl)-1-(4-phenyl-1-piperazinyl)propan-1-one>10000Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011825-HT7CLONEDHUMAN3H-5-HTN-Phenylmethyl-3-[4-(phenylmethyl)-1-piperazinyl]propanamide4.34Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011835-HT1ACLONEDHUMAN3H-8-OH-DPATN-Phenylmethyl-3-[4-(phenylmethyl)-1-piperazinyl]propanamide0.34Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011845-HT1ACLONEDHUMAN3H-8-OH-DPATN-phenylmethyl-3-[(phenylmethyl)amino]propanamide 3750Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011855-HT7CLONEDHUMAN3H-5-HTN-phenylmethyl-3-[(phenylmethyl)amino]propanamide 176Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011865-HT7CLONEDHUMAN3H-5-HTSB-2699700.71Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011875-HT1ACLONEDHUMAN3H-8-OH-DPATSB-2699709024Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011885-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT2.65Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011895-HT7CLONEDHUMAN3H-5-HT8-OH-DPAT388Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011905-HT7CLONEDHUMAN3H-5-HT5-Hydroxy Tryptamine2.12Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011915-HT1ACLONEDHUMAN3H-8-OH-DPAT5-Hydroxy Tryptamine0.91Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
1011925-HT7CLONEDHUMAN3H-5-HT1-[4-(2-Pyridyl)-1-piperazinyl]-3-[4-(phenylmethyl)-1-piperazinyl]-1-propanone29.5Intagliata S et al 2016Jan 15, 2025Jan 15, 2025
101193MORCLONEDHUMAN3H-Diprenorphine(S)-1-((3-((3,4-Dihydroisoquinolin-2(1H)-yl)methyl)benzyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate0.23Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101194DORCLONEDHUMAN3H-Diprenorphine(S)-1-((3-((3,4-Dihydroisoquinolin-2(1H)-yl)methyl)benzyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate4.8Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101195KORCLONEDHUMAN3H-Diprenorphine(S)-1-((3-((3,4-Dihydroisoquinolin-2(1H)-yl)methyl)benzyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate46.3Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101196MORCLONEDHUMAN3H-Diprenorphine(S)-1-((5-(3,4-Dihydroisoquinolin-2(1H)-yl)pentyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate1.5Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101197DORCLONEDHUMAN3H-Diprenorphine(S)-1-((5-(3,4-Dihydroisoquinolin-2(1H)-yl)pentyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate142Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101198KORCLONEDHUMAN3H-Diprenorphine(S)-1-((5-(3,4-Dihydroisoquinolin-2(1H)-yl)pentyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate44.2Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101199MORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethoxy)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate0.64Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101200DORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethoxy)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate113Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101201KORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethoxy)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate45Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101202MORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)-2-oxoethoxy)-ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate1.28Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101203DORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)-2-oxoethoxy)-ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate17.5Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101204KORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)-2-oxoethoxy)-ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate12.5Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101205MORCLONEDHUMAN3H-Diprenorphine(S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperidin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate1.64Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101206DORCLONEDHUMAN3H-Diprenorphine(S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperidin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate130Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101207KORCLONEDHUMAN3H-Diprenorphine(S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperidin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate21Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101208MORCLONEDHUMAN3H-Diprenorphine(S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperazin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate3.59Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101209DORCLONEDHUMAN3H-Diprenorphine(S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperazin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate16.6Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101210KORCLONEDHUMAN3H-Diprenorphine(S)-1-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)piperazin-1-yl)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate173Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101211MORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopro-pan-2-aminium Trifluoroacetate1.7Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101212DORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopro-pan-2-aminium Trifluoroacetate77Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101213KORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)ethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopro-pan-2-aminium Trifluoroacetate8.5Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101214MORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate24Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101215DORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate24.7Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101216KORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)(methyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate780Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101217MORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate1.32Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101218DORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate7.3Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
101219KORCLONEDHUMAN3H-Diprenorphine(S)-1-((2-((2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)amino)-2-oxoethyl)amino)-3-(4-hydroxy-2,6-dimethylphenyl)-1-oxopropan-2-aminium Trifluoroacetate107Henry S,et al., 2021Jan 15, 2025Jan 28, 2025
1012205-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(4-(3,4-dichlorophenethyl)piperazin-1-yl)benzo[d]isothiazole hydrochloride0.84Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012215-HT7CLONEDHUMAN3H-LSD3-(4-(3,4-dichlorophenethyl)piperazin-1-yl)benzo[d]isothiazole hydrochloride12Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012225-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-([1,1'-biphenyl]-2-yl)piperazin-1-yl)-1-(3,4-dichlorophenyl)ethanol hydrochloride 2.4Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012235-HT7CLONEDHUMAN3H-LSD2-(4-([1,1'-biphenyl]-2-yl)piperazin-1-yl)-1-(3,4-dichlorophenyl)ethanol hydrochloride 3.2Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012245-HT1ACLONEDHUMAN3H-8-OH-DPAT1-([1,1'-biphenyl]-2-yl)-4-(3,4-dichlorophenethyl)piperazine hydrochloride 6.3Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012255-HT7CLONEDHUMAN3H-LSD1-([1,1'-biphenyl]-2-yl)-4-(3,4-dichlorophenethyl)piperazine hydrochloride 0.75Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012265-HT1ACLONEDHUMAN3H-8-OH-DPATVortioxetine9.5Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012275-HT7CLONEDHUMAN3H-LSDVortioxetine26Gu, Zheng-Song, et al., 2017Jan 15, 2025Jan 15, 2025
1012285-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one3755Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012295-HT2ACLONEDHUMAN3H-KETANSERIN1'-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one68Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012305-HT6CLONEDHUMAN3H-LSD1'-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one4737Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012315-HT7CLONEDHUMAN3H-5-CT1'-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one29Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012325-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 2891Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012335-HT2ACLONEDHUMAN3H-KETANSERIN1'-{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 715Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012345-HT6CLONEDHUMAN3H-LSD1'-{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 5559Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012355-HT7CLONEDHUMAN3H-5-CT1'-{3-[4-(4-chlorophenyl)piperazin-1-yl]propyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 67Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012365-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-[2-(4-phenylpiperazin-1-yl)ethyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 6005Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012375-HT2ACLONEDHUMAN3H-KETANSERIN1'-[2-(4-phenylpiperazin-1-yl)ethyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 496Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012385-HT6CLONEDHUMAN3H-LSD1'-[2-(4-phenylpiperazin-1-yl)ethyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 6556Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012395-HT7CLONEDHUMAN3H-5-CT1'-[2-(4-phenylpiperazin-1-yl)ethyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 100Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012405-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 2687Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012415-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 351Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012425-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 2005Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012435-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 55Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012445-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1096Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012455-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 452Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012465-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 2843Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012475-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 245Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012485-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 4054Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012495-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 270Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012505-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1131Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012515-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 38Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012525-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(4-chlorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one >10000Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012535-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(4-chlorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 404Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012545-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(4-chlorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 4577Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012555-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(4-chlorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 284Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012565-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(4-fluorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one >10000Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012575-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(4-fluorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 259Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012585-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(4-fluorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 5285Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012595-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(4-fluorophenyl)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 275Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012605-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-(2-(4-(4-fluorophenyl)-5,6-dihydropyridin-1(2H)-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one 3949Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012615-HT2ACLONEDHUMAN3H-KETANSERIN1'-(2-(4-(4-fluorophenyl)-5,6-dihydropyridin-1(2H)-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one 75Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012625-HT6CLONEDHUMAN3H-LSD1'-(2-(4-(4-fluorophenyl)-5,6-dihydropyridin-1(2H)-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one 6267Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012635-HT7CLONEDHUMAN3H-5-CT1'-(2-(4-(4-fluorophenyl)-5,6-dihydropyridin-1(2H)-yl)ethyl)spiro[indoline-3,3'-pyrrolidin]-2-one 43Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012645-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one >10000Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012655-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 59Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012665-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 4744Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012675-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(4-fluorophenyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 21Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012685-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(4-chlorophenoxy)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one >10000Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012695-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(4-chlorophenoxy)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 343Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012705-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(4-chlorophenoxy)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 1693Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012715-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(4-chlorophenoxy)piperidin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 121Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012725-HT1ACLONEDHUMAN3H-8-OH-DPAT1'-{2-[4-(4-chlorobenzoyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one >10000Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012735-HT2ACLONEDHUMAN3H-KETANSERIN1'-{2-[4-(4-chlorobenzoyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one >10000Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012745-HT6CLONEDHUMAN3H-LSD1'-{2-[4-(4-chlorobenzoyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 7746Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
1012755-HT7CLONEDHUMAN3H-5-CT1'-{2-[4-(4-chlorobenzoyl)piperazin-1-yl]ethyl}-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-2-one 529Kelemen A, et al., 2018Jan 15, 2025Jan 15, 2025
101276H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one23Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101277H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE2-Methyl-7-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one189Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101278H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(4-methylpiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one32Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101279H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE2-Methyl-7-(3-(4-methylpiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one279Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101280H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one6.5Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101281H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE2-Methyl-7-(3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one1027Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101282H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(2-methylpyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one26Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101283H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE2-Methyl-7-(3-(2-methylpyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one68Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101284H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(pyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one39Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101285H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE2-Methyl-7-(3-(pyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one169Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101286H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(4-ethylpiperazin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one1098Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101287H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(4-methylpiperazin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one706Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101288H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(diethylamino)propoxy)- 3,4-dihydroisoquinolin-1(2H)-one542Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101289H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(4-oxopiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one176Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101290H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(2-methylpiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one165Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101291H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(3-hydroxypyrrolidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one112Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101292H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(3-(4-hydroxypiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one35Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101293H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE2-Methyl-7-(3-(4-hydroxypiperidin-1-yl)propoxy)-3,4-dihydroisoquinolin-1(2H)-one908Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101294H1CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(2-morpholinoethoxy)-3,4-dihydroisoquinolin-1(2H)-one 1208Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101295H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(4-morpholinobutoxy)-3,4-dihydroisoquinolin-1(2H)-one856Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101296H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Methyl-7-(2-hydroxy-3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one2000Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101297H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamine2-Ethyl-7-(3-morpholinopropoxy)-3,4-dihydroisoquinolin-1(2H)-one252Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101298H3CEREBRAL CORTEXRAT3H-N-alpha-methylhistamineS380933.6Dou F, et al., 2019Jan 15, 2025Jan 28, 2025
101299CORTEXRAT3H-PRAZOSIN1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride11Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101300D2CLONEDHUMAN3H-Methylspiperone1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride97Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013015-HT7CLONEDHUMAN3H-LSD1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride15Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013025-HT2ACLONEDHUMAN3H-KETANSERIN1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride527Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013035-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[3-(2,4-Dimethylphenoxy)propyl]-4-(2-methoxyphenyl)piperazine hydrochloride2Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013045-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2-{4-[2-(Mesityloxy)ethyl]piperazin-1-yl}ethoxy)ethanol dihydrochloride3168Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101305CORTEXRAT3H-PRAZOSIN1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride 2117Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101306D2CLONEDHUMAN3H-Methylspiperone1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride 4963Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013075-HT7CLONEDHUMAN3H-LSD1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride 3027Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013085-HT2ACLONEDHUMAN3H-KETANSERIN1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride 772Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013095-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[3-(Mesityloxy)propyl]-4-(4-methoxyphenyl)piperazine dihydrochloride 146Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101310CORTEXRAT3H-PRAZOSIN1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 93Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013115-HT7CLONEDHUMAN3H-LSD 1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 90Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013125-HT2ACLONEDHUMAN3H-KETANSERIN1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 76Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013135-HT1ACLONEDHUMAN3H-8-OH-DPAT1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 20Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101314CORTEXRAT3H-PRAZOSIN1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride36Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101315D2CLONEDHUMAN3H-Methylspiperone1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride1206Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013165-HT7CLONEDHUMAN3H-LSD1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride388Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013175-HT6CLONEDHUMAN3H-LSD1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride200Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013185-HT2ACLONEDHUMAN3H-KETANSERIN1-{2-[2-(2,3-Dimethylphenoxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride220Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013195-HT7CLONEDHUMAN3H-LSD2-(4-{2-[2-(2,3,5-Trimethylphenoxy)ethoxy]ethyl}piperazin-1-yl)ethanol dihydrochloride3142Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101320CORTEXRAT3H-PRAZOSIN1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride14Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101321D2CLONEDHUMAN3H-Methylspiperone1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride162Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013225-HT7CLONEDHUMAN3H-LSD1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride89Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013235-HT6CLONEDHUMAN3H-LSD1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride1540Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013245-HT2ACLONEDHUMAN3H-KETANSERIN1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride159Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013255-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2-Methoxyphenyl)-4-{2-[2-(2,3,5-trimethylphenoxy)ethoxy]ethyl}piperazine dihydrochloride32Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101326CORTEXRAT3H-PRAZOSIN1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride15Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101327D2CLONEDHUMAN3H-Methylspiperone1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride189Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013285-HT7CLONEDHUMAN3H-LSD1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride70Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013295-HT6CLONEDHUMAN3H-LSD1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride2427Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013305-HT2ACLONEDHUMAN3H-KETANSERIN1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride245Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013315-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-(2-methoxyphenyl)piperazine dihydrochloride5Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013325-HT7CLONEDHUMAN3H-LSD1-Benzyl-4-{2-[2-(mesityloxy)ethoxy]ethyl}piperazine dihydrochloride3160Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013335-HT2ACLONEDHUMAN3H-KETANSERIN1-Benzyl-4-{2-[2-(mesityloxy)ethoxy]ethyl}piperazine dihydrochloride498Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101334CORTEXRAT3H-PRAZOSIN1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride772Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013355-HT7CLONEDHUMAN3H-LSD1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride1050Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013365-HT6CLONEDHUMAN3H-LSD1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride2155Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013375-HT2ACLONEDHUMAN3H-KETANSERIN1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride2805Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013385-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[2-(Mesityloxy)ethoxy]ethyl}-4-phenethylpiperazine dihydrochloride552Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101339D2CLONEDHUMAN3H-Methylspiperone1-[3-(4-Chloro-3-methylphenoxy)propyl]-4-phenylpiperazine dihydrochloride 299Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013405-HT7CLONEDHUMAN3H-LSDMETHIOTHEPIN1.7Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013415-HT6CLONEDHUMAN3H-LSDMETHIOTHEPIN0.9Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
1013425-HT1ACLONEDHUMAN3H-8-OH-DPATMETHIOTHEPIN4Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101343CORTEXRAT3H-PRAZOSINPHENTOLAMINE12Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101344D2CLONEDHUMAN3H-MethylspiperoneHALOPERIDOL5.9Panczyk K, et al., 2018Jan 15, 2025Jan 28, 2025
1013455-HT2ACLONEDHUMAN3H-KETANSERINMIANSERIN3.2Panczyk K, et al., 2018Jan 15, 2025Jan 15, 2025
101346D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one114Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013475-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one47Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013485-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one652Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013495-HT6CLONEDHUMAN3H-LSD1-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one1699Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013505-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one366Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101351D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one180Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013525-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one291Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013535-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one1927Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013545-HT6CLONEDHUMAN3H-LSD1-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one3666Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013555-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one3743Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101356D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one11Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013575-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one22Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013585-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one717Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013595-HT6CLONEDHUMAN3H-LSD1-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one1916Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013605-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one84Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101361D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 867Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013625-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 32Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013635-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 892Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013645-HT6CLONEDHUMAN3H-LSD1-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 1461Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013655-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one 184Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101366D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(2-pyrimidinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one188Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013675-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(2-pyrimidinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one94Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013685-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(2-pyrimidinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one43Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013695-HT6CLONEDHUMAN3H-LSD1-{6-[4-(2-pyrimidinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one5253Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013705-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(2-pyrimidinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one475Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101371D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one431Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013725-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one9473Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013735-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one3983Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013745-HT6CLONEDHUMAN3H-LSD1-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one952Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013755-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one696Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101376D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one82Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013775-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one22Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013785-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one222Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013795-HT6CLONEDHUMAN3H-LSD1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one999Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013805-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(8-quinolinyl)piperazin-1-yl]hexyl}benzo[cd]indol-2(1H)-one119Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101381D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione30Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013825-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione48Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013835-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione578Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013845-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione476Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013855-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione34Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101386D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione118Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013875-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione35Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013885-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione443Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013895-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione182Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013905-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione344Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101391D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione264Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013925-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione482Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013935-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione533Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013945-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione494Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013955-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-(2H)naphtho[1,8-cd][1,2]thiazole-1,1(2H)-dione822Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101396D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione10Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1013975-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione20Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013985-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione337Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1013995-HT6CLONEDHUMAN3H- LSD2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione671Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014005-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione266Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101401D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione271Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1014025-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione47Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014035-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione334Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014045-HT6CLONEDHUMAN3H-LSD2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione347Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014055-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(3-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione371Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101406D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione27Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1014075-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione28Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014085-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione461Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014095-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione246Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014105-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-ethoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione73Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101411D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione>10000Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1014125-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione3569Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014135-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione>10000Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014145-HT6CLONEDHUMAN3H-LSD2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione5765Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014155-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(4-methoxyphenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione>10000Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101416D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione1302Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1014175-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione172Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014185-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione563Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014195-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione1966Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014205-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-pyridinyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione1200Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101421D2CLONEDHUMAN3H-RACLOPRIDE2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione141Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1014225-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione373Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014235-HT2ACLONEDHUMAN3H-KETANSERIN2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione1918Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014245-HT6CLONEDHUMAN3H-LSD2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione1410Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014255-HT7CLONEDHUMAN3H-5-CT2-{6-[4-(2-nitrophenyl)piperazin-1-yl]hexyl}-1H-benzo[de]isoquinoline-1,3(2H)-dione710Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101426D2CLONEDHUMAN3H-RACLOPRIDE1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one2Zareba P, et al., 2019Jan 15, 2025Jan 28, 2025
1014275-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one19Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014285-HT2ACLONEDHUMAN3H-KETANSERIN1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one456Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014295-HT6CLONEDHUMAN3H-LSD1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one3270Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
1014305-HT7CLONEDHUMAN3H-5-CT1-{6-[4-(2-methoxyphenyl)piperazin-1-yl]hexyl}-5,6-dihydro-4H-imidazo[4,5,1-ij]quinolin-2(1H)-one291Zareba P, et al., 2019Jan 15, 2025Jan 15, 2025
101431KORCLONEDHUMAN3H-U69,5933-[2-[Diphenethylamino]ethyl]phenol211Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025
101432KORCLONEDHUMAN3H-U69,5934-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 36.3Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025
101433MORCLONEDHUMAN3H-DAMGO4-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 731Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025
101434DORCLONEDHUMAN3H-DPDPE4-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 2129Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025
101435KORCLONEDHUMAN3H-U69,5934-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride218Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025
101436MORCLONEDHUMAN3H-DAMGO4-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride1750Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025
101437DORCLONEDHUMAN3H-DPDPE4-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride2187Guerriera E, et al., 2016Jan 15, 2025Jan 29, 2025