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Kᵢ ID60146
ReceptorsA2A
SourcesCLONED
SpeciesHUMAN
Hot Ligands[3 H]2-[p-(2- carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamido-adenosine
Test Ligands(1S,2S,3R,4R,5S)-2,3-Dihydroxy-N-methyl-4-(6-(methylamino)-2- ((3-(trifluoromethyl)phenyl)ethynyl)-9H-purin-9-yl)bicyclo[3.1.0]- hexane-1-carboxamide
Kᵢ Value>10000
Submitted AtJan 15, 2025 2:29 pm
Updated AtJan 15, 2025 2:29 pm

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