Kᵢ ID75350
ReceptorsSigma 1
SourcesCLONED
SpeciesHUMAN
Hot Ligands3H-Pentazocine(+)
Test Ligandsethyl (1S,2R,3S,4R,5S)-4-[6-[2-(5-chlorothiophen-2-yl)ethynyl]-4-(methylamino)imidazo[4,5-c]pyridin-1-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate
Kᵢ Value>10000
Submitted AtJan 15, 2025 2:29 pm
Updated AtJan 28, 2025 12:03 pm