Kᵢ ID99118
ReceptorsH3
SourcesCLONED
SpeciesHUMAN
Hot Ligands3H-Alpha-methylhistamine
Test Ligands(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide
Kᵢ Value>10000
Submitted AtJan 15, 2025 2:29 pm
Updated AtJan 28, 2025 12:29 pm