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Kᵢ ID99864
ReceptorsSigma 1
SourcesCLONED
SpeciesHUMAN
Hot Ligands[3H] pentazocine
Test Ligands(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide
Kᵢ Value1900
Submitted AtJan 15, 2025 2:29 pm
Updated AtJan 15, 2025 2:29 pm

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