The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

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Showing 43,001-44,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
45615SLC6A4CLONEDHUMAN3H-IMIPRAMINEmirtazepine(+)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45616SLC6A4CLONEDHUMAN3H-IMIPRAMINEmirtazepine(-)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45617NETCLONEDHUMAN3H-Nisoxetinemirtazepine(-)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45618SLC6A3CLONEDHUMAN3H-WIN 35,428mirtazepine(-)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45619SLC6A4CLONEDHUMAN3H-IMIPRAMINENefazodone200Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45620NETCLONEDHUMAN3H-NisoxetineNefazodone360Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45621SLC6A3CLONEDHUMAN3H-WIN 35,428Nefazodone360Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45622SLC6A4CLONEDHUMAN3H-IMIPRAMINENOMIFENSINE1010Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45623NETCLONEDHUMAN3H-NisoxetineNOMIFENSINE15.6Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45624SLC6A3CLONEDHUMAN3H-WIN 35,428NOMIFENSINE56Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45625SLC6A4CLONEDHUMAN3H-IMIPRAMINENORFLUOXETINE1.47Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45626NETCLONEDHUMAN3H-NisoxetineNORFLUOXETINE1426Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45627SLC6A3CLONEDHUMAN3H-WIN 35,428NORFLUOXETINE420Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45628SLC6A4CLONEDHUMAN3H-IMIPRAMINENORTRYPTYLINE18Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45629NETCLONEDHUMAN3H-NisoxetineNORTRYPTYLINE4.37Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45630SLC6A3CLONEDHUMAN3H-WIN 35,428NORTRYPTYLINE1140Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45631SLC6A4CLONEDHUMAN3H-IMIPRAMINEOxaprotiline3900Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45632NETCLONEDHUMAN3H-NisoxetineOxaprotiline4.9Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45633SLC6A3CLONEDHUMAN3H-WIN 35,428Oxaprotiline4340Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45634SLC6A4CLONEDHUMAN3H-IMIPRAMINEPAROXETINE0.13Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45635NETCLONEDHUMAN3H-NisoxetinePAROXETINE40Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45636SLC6A3CLONEDHUMAN3H-WIN 35,428PAROXETINE490Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45637SLC6A4CLONEDHUMAN3H-IMIPRAMINEPhenelzine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45638NETCLONEDHUMAN3H-NisoxetinePhenelzine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45639SLC6A3CLONEDHUMAN3H-WIN 35,428Phenelzine8400Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45640SLC6A4CLONEDHUMAN3H-IMIPRAMINEProtriptyline19.6Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45641NETCLONEDHUMAN3H-NisoxetineProtriptyline1.41Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45642SLC6A3CLONEDHUMAN3H-WIN 35,428Protriptyline2100Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45643SLC6A4CLONEDHUMAN3H-IMIPRAMINESERTRALINE0.29Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45644NETCLONEDHUMAN3H-NisoxetineSERTRALINE420Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45645SLC6A3CLONEDHUMAN3H-WIN 35,428SERTRALINE25Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45646SLC6A4CLONEDHUMAN3H-IMIPRAMINETomoxetine8.9Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45647NETCLONEDHUMAN3H-NisoxetineTomoxetine2.03Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45648SLC6A3CLONEDHUMAN3H-WIN 35,428Tomoxetine1080Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45649SLC6A4CLONEDHUMAN3H-IMIPRAMINETRANYLCYPROMINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45650NETCLONEDHUMAN3H-NisoxetineTRANYLCYPROMINE5900Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45651SLC6A3CLONEDHUMAN3H-WIN 35,428TRANYLCYPROMINE5100Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45652SLC6A4CLONEDHUMAN3H-IMIPRAMINETRAZODONE160Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45653NETCLONEDHUMAN3H-NisoxetineTRAZODONE8500Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45654SLC6A3CLONEDHUMAN3H-WIN 35,428TRAZODONE7400Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45655SLC6A4CLONEDHUMAN3H-IMIPRAMINETrimipramine149Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45656NETCLONEDHUMAN3H-NisoxetineTrimipramine2450Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45657SLC6A3CLONEDHUMAN3H-WIN 35,428Trimipramine3780Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45658SLC6A4CLONEDHUMAN3H-IMIPRAMINEVenlafaxine8.9Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45659NETCLONEDHUMAN3H-NisoxetineVenlafaxine1060Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45660SLC6A3CLONEDHUMAN3H-WIN 35,428Venlafaxine9300Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45661SLC6A4CLONEDHUMAN3H-IMIPRAMINEViloxazine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45662NETCLONEDHUMAN3H-NisoxetineViloxazine155Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45663SLC6A3CLONEDHUMAN3H-WIN 35,428Viloxazine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45664SLC6A4CLONEDHUMAN3H-IMIPRAMINEZIMELIDINE152Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45665NETCLONEDHUMAN3H-NisoxetineZIMELIDINE9400Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
45666SLC6A3CLONEDHUMAN3H-WIN 35,428ZIMELIDINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
456675-HT1ACLONEDHUMAN3H-8-OH-DPAT(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456685-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456695-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-0161760Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456705-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid7308Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456715-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-0252150Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456725-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-048-45000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456735-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456745-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione7049Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456755-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid2790Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456765-HT1ACLONEDHUMAN3H-8-OH-DPATPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456775-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456785-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456795-HT1ACLONEDHUMAN3H-8-OH-DPATN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide2546Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456805-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3275Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456815-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456825-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione4274Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456835-HT1ACLONEDHUMAN3H-8-OH-DPAT(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456845-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456855-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456865-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456875-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456885-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione597.9Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456895-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456905-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456915-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione165.3Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456925-HT1ACLONEDHUMAN3H-8-OH-DPAT(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456935-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456945-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456955-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid1382Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456965-HT1ACLONEDHUMAN3H-8-OH-DPAT(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456975-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456985-HT1ACLONEDHUMAN3H-8-OH-DPAT(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione1774Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
456995-HT1ACLONEDHUMAN3H-8-OH-DPAT(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione63.46Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457005-HT1BCLONEDHUMAN3H-GR-125743PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457015-HT1BCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457025-HT1BCLONEDHUMAN3H-GR-125743(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457035-HT1BCLONEDHUMAN3H-GR-125743(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457045-HT1BCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457055-HT1BCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457065-HT1BCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457075-HT1BCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457085-HT1BCLONEDHUMAN3H-GR-125743(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457095-HT1BCLONEDHUMAN3H-GR-125743(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457105-HT1BCLONEDHUMAN3H-GR-125743(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457115-HT1BCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione8213Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457125-HT1BCLONEDHUMAN3H-GR-125743(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457135-HT1BCLONEDHUMAN3H-GR-125743(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457145-HT1BCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457155-HT1BCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457165-HT1BCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457175-HT1BCLONEDHUMAN3H-GR-125743PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457185-HT1BCLONEDHUMAN3H-GR-125743PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457195-HT1BCLONEDHUMAN3H-GR-125743N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457205-HT1BCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457215-HT1BCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457225-HT1BCLONEDHUMAN3H-GR-125743(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457235-HT1BCLONEDHUMAN3H-GR-125743PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457245-HT1BCLONEDHUMAN3H-GR-125743(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457255-HT1BCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457265-HT1BCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457275-HT1BCLONEDHUMAN3H-GR-125743(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457285-HT1BCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457295-HT1BCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457305-HT1DCLONEDHUMAN3H-GR-125743(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457315-HT1DCLONEDHUMAN3H-GR-125743(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457325-HT1DCLONEDHUMAN3H-GR-125743(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457335-HT1DCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457345-HT1DCLONEDHUMAN3H-GR-125743(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457355-HT1DCLONEDHUMAN3H-GR-125743(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457365-HT1DCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457375-HT1DCLONEDHUMAN3H-GR-125743(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457385-HT1DCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457395-HT1DCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457405-HT1DCLONEDHUMAN3H-GR-125743(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457415-HT1DCLONEDHUMAN3H-GR-125743PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457425-HT1DCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457435-HT1DCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457445-HT1DCLONEDHUMAN3H-GR-125743N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457455-HT1DCLONEDHUMAN3H-GR-125743PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457465-HT1DCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457475-HT1DCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457485-HT1DCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457495-HT1DCLONEDHUMAN3H-GR-125743(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457505-HT1DCLONEDHUMAN3H-GR-125743PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457515-HT1DCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457525-HT1DCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457535-HT1DCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457545-HT1DCLONEDHUMAN3H-GR-125743PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457555-HT1DCLONEDHUMAN3H-GR-125743(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457565-HT1DCLONEDHUMAN3H-GR-125743(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457575-HT1DCLONEDHUMAN3H-GR-125743(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457585-HT1DCLONEDHUMAN3H-GR-125743(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457595-HT1DCLONEDHUMAN3H-GR-125743(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457605-HT1ECLONEDHUMAN3H-5HT(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione5489Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457615-HT1ECLONEDHUMAN3H-5HT(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457625-HT1ECLONEDHUMAN3H-5HT(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457635-HT1ECLONEDHUMAN3H-5HTPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457645-HT1ECLONEDHUMAN3H-5HTN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457655-HT1ECLONEDHUMAN3H-5HT(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457665-HT1ECLONEDHUMAN3H-5HT(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457675-HT1ECLONEDHUMAN3H-5HT(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457685-HT1ECLONEDHUMAN3H-5HTPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457695-HT1ECLONEDHUMAN3H-5HT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione5680Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457705-HT1ECLONEDHUMAN3H-5HT(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457715-HT1ECLONEDHUMAN3H-5HTPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457725-HT1ECLONEDHUMAN3H-5HT(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid272.5Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457735-HT1ECLONEDHUMAN3H-5HT(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457745-HT1ECLONEDHUMAN3H-5HT(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457755-HT1ECLONEDHUMAN3H-5HT(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457765-HT1ECLONEDHUMAN3H-5HT(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457775-HT1ECLONEDHUMAN3H-5HT(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457785-HT1ECLONEDHUMAN3H-5HT(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457795-HT1ECLONEDHUMAN3H-5HT(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457805-HT1ECLONEDHUMAN3H-5HT(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457815-HT1ECLONEDHUMAN3H-5HT(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457825-HT1ECLONEDHUMAN3H-5HT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457835-HT1ECLONEDHUMAN3H-5HT(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457845-HT1ECLONEDHUMAN3H-5HT(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457855-HT1ECLONEDHUMAN3H-5HTPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457865-HT1ECLONEDHUMAN3H-5HT(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457875-HT1ECLONEDHUMAN3H-5HT(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457885-HT1ECLONEDHUMAN3H-5HT(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457895-HT1ECLONEDHUMAN3H-5HT(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457905-HT2ACLONEDHUMAN3H-KETANSERINPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457915-HT2ACLONEDHUMAN3H-KETANSERIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457925-HT2ACLONEDHUMAN3H-KETANSERINPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457935-HT2ACLONEDHUMAN3H-KETANSERIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457945-HT2ACLONEDHUMAN3H-KETANSERIN(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457955-HT2ACLONEDHUMAN3H-KETANSERIN(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457965-HT2ACLONEDHUMAN3H-KETANSERIN(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457975-HT2ACLONEDHUMAN3H-KETANSERINPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457985-HT2ACLONEDHUMAN3H-KETANSERIN(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
457995-HT2ACLONEDHUMAN3H-KETANSERIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458005-HT2ACLONEDHUMAN3H-KETANSERINN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458015-HT2ACLONEDHUMAN3H-KETANSERIN(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458025-HT2ACLONEDHUMAN3H-KETANSERIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458035-HT2ACLONEDHUMAN3H-KETANSERIN(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458045-HT2ACLONEDHUMAN3H-KETANSERIN(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458055-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458065-HT2ACLONEDHUMAN3H-KETANSERIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458075-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458085-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458095-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458105-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458115-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458125-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458135-HT2ACLONEDHUMAN3H-KETANSERIN(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458145-HT2ACLONEDHUMAN3H-KETANSERIN(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458155-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458165-HT2ACLONEDHUMAN3H-KETANSERIN(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458175-HT2ACLONEDHUMAN3H-KETANSERIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458185-HT2ACLONEDHUMAN3H-KETANSERIN(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458195-HT2ACLONEDHUMAN3H-KETANSERINPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458205-HT2BCLONEDHUMAN3H-LSDN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458215-HT2BCLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458225-HT2BCLONEDHUMAN3H-LSDPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458235-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458245-HT2BCLONEDHUMAN3H-LSD(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458255-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458265-HT2BCLONEDHUMAN3H-LSD(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458275-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458285-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458295-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458305-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458315-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458325-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458335-HT2BCLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458345-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458355-HT2BCLONEDHUMAN3H-LSD(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458365-HT2BCLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458375-HT2BCLONEDHUMAN3H-LSD(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458385-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458395-HT2BCLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458405-HT2BCLONEDHUMAN3H-LSDPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458415-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458425-HT2BCLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458435-HT2BCLONEDHUMAN3H-LSD(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458445-HT2BCLONEDHUMAN3H-LSD(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione1460Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458455-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458465-HT2BCLONEDHUMAN3H-LSDPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458475-HT2BCLONEDHUMAN3H-LSDPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458485-HT2BCLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458495-HT2BCLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458505-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458515-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458525-HT2CCLONEDRAT3H-MESULERGINE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458535-HT2CCLONEDRAT3H-MESULERGINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458545-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458555-HT2CCLONEDRAT3H-MESULERGINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458565-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458575-HT2CCLONEDRAT3H-MESULERGINE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458585-HT2CCLONEDRAT3H-MESULERGINE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458595-HT2CCLONEDRAT3H-MESULERGINE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458605-HT2CCLONEDRAT3H-MESULERGINE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458615-HT2CCLONEDRAT3H-MESULERGINE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458625-HT2CCLONEDRAT3H-MESULERGINE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458635-HT2CCLONEDRAT3H-MESULERGINE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458645-HT2CCLONEDRAT3H-MESULERGINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458655-HT2CCLONEDRAT3H-MESULERGINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458665-HT2CCLONEDRAT3H-MESULERGINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458675-HT2CCLONEDRAT3H-MESULERGINE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458685-HT2CCLONEDRAT3H-MESULERGINEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458695-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458705-HT2CCLONEDRAT3H-MESULERGINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458715-HT2CCLONEDRAT3H-MESULERGINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458725-HT2CCLONEDRAT3H-MESULERGINE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458735-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458745-HT2CCLONEDRAT3H-MESULERGINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458755-HT2CCLONEDRAT3H-MESULERGINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458765-HT2CCLONEDRAT3H-MESULERGINEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458775-HT2CCLONEDRAT3H-MESULERGINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458785-HT2CCLONEDRAT3H-MESULERGINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458795-HT2CCLONEDRAT3H-MESULERGINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458805-HT2CCLONEDRAT3H-MESULERGINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458815-HT3CLONEDHUMAN3H-ZACOPRIDEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458825-HT3CLONEDHUMAN3H-ZACOPRIDE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458835-HT3CLONEDHUMAN3H-ZACOPRIDE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458845-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458855-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458865-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458875-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458885-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458895-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458905-HT3CLONEDHUMAN3H-ZACOPRIDE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458915-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458925-HT3CLONEDHUMAN3H-ZACOPRIDE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458935-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458945-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458955-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458965-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458975-HT3CLONEDHUMAN3H-ZACOPRIDEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458985-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
458995-HT3CLONEDHUMAN3H-ZACOPRIDE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459005-HT3CLONEDHUMAN3H-ZACOPRIDEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459015-HT3CLONEDHUMAN3H-ZACOPRIDEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459025-HT3CLONEDHUMAN3H-ZACOPRIDEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459035-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459045-HT3CLONEDHUMAN3H-ZACOPRIDE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459055-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459065-HT3CLONEDHUMAN3H-ZACOPRIDE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459075-HT3CLONEDHUMAN3H-ZACOPRIDE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459085-HT3CLONEDHUMAN3H-ZACOPRIDE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459095-HT3CLONEDHUMAN3H-ZACOPRIDE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459105-HT3CLONEDHUMAN3H-ZACOPRIDE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459115-HT5ACLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459125-HT5ACLONEDHUMAN3H-LSD(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459135-HT5ACLONEDHUMAN3H-LSD(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459145-HT5ACLONEDHUMAN3H-LSD(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459155-HT5ACLONEDHUMAN3H-LSD(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459165-HT5ACLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459175-HT5ACLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459185-HT5ACLONEDHUMAN3H-LSD(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459195-HT5ACLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459205-HT5ACLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459215-HT5ACLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459225-HT5ACLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459235-HT5ACLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459245-HT5ACLONEDHUMAN3H-LSD(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459255-HT5ACLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459265-HT5ACLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459275-HT5ACLONEDHUMAN3H-LSDPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459285-HT5ACLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459295-HT5ACLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459305-HT5ACLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459315-HT5ACLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459325-HT5ACLONEDHUMAN3H-LSDPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459335-HT5ACLONEDHUMAN3H-LSDPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459345-HT5ACLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459355-HT5ACLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459365-HT5ACLONEDHUMAN3H-LSD(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459375-HT5ACLONEDHUMAN3H-LSD(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459385-HT5ACLONEDHUMAN3H-LSDPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459395-HT5ACLONEDHUMAN3H-LSD(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459405-HT5ACLONEDHUMAN3H-LSDN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459415-HT6CLONEDHUMAN3H-LSD(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459425-HT6CLONEDHUMAN3H-LSD(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459435-HT6CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459445-HT6CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459455-HT6CLONEDHUMAN3H-LSDPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459465-HT6CLONEDHUMAN3H-LSDPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459475-HT6CLONEDHUMAN3H-LSDN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459485-HT6CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459495-HT6CLONEDHUMAN3H-LSDPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459505-HT6CLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459515-HT6CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459525-HT6CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459535-HT6CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459545-HT6CLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459555-HT6CLONEDHUMAN3H-LSD(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459565-HT6CLONEDHUMAN3H-LSD(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459575-HT6CLONEDHUMAN3H-LSD(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459585-HT6CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459595-HT6CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459605-HT6CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459615-HT6CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459625-HT6CLONEDHUMAN3H-LSD(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459635-HT6CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459645-HT6CLONEDHUMAN3H-LSD(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459655-HT6CLONEDHUMAN3H-LSDPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459665-HT6CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459675-HT6CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459685-HT6CLONEDHUMAN3H-LSD(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459695-HT6CLONEDHUMAN3H-LSD(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459705-HT6CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459715-HT7CLONEDHUMAN3H-LSDPL-3-0173197Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459725-HT7CLONEDHUMAN3H-LSDPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459735-HT7CLONEDHUMAN3H-LSDN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide775.2Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459745-HT7CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459755-HT7CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione793Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459765-HT7CLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459775-HT7CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459785-HT7CLONEDHUMAN3H-LSD(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459795-HT7CLONEDHUMAN3H-LSDPL-3-048-47290Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459805-HT7CLONEDHUMAN3H-LSD(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione2053Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459815-HT7CLONEDHUMAN3H-LSD(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459825-HT7CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459835-HT7CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459845-HT7CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459855-HT7CLONEDHUMAN3H-LSD(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459865-HT7CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione2005Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459875-HT7CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459885-HT7CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459895-HT7CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459905-HT7CLONEDHUMAN3H-LSD(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459915-HT7CLONEDHUMAN3H-LSD(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459925-HT7CLONEDHUMAN3H-LSD(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459935-HT7CLONEDHUMAN3H-LSD(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid3761Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459945-HT7CLONEDHUMAN3H-LSD(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459955-HT7CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459965-HT7CLONEDHUMAN3H-LSD(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459975-HT7CLONEDHUMAN3H-LSD(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459985-HT7CLONEDHUMAN3H-LSD(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
459995-HT7CLONEDHUMAN3H-LSDPL-3-0252762Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
460005-HT7CLONEDHUMAN3H-LSD(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46001Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46002Alpha1ACLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46003Alpha1ACLONEDHUMAN3H-PRAZOSINPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46004Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46005Alpha1ACLONEDHUMAN3H-PRAZOSINPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46006Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46007Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46008Alpha1ACLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46009Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46010Alpha1ACLONEDHUMAN3H-PRAZOSINN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46011Alpha1ACLONEDHUMAN3H-PRAZOSINPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46012Alpha1ACLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46013Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46014Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46015Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46016Alpha1ACLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46017Alpha1ACLONEDHUMAN3H-PRAZOSINPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46018Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46019Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46020Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46021Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46022Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46023Alpha1ACLONEDHUMAN3H-PRAZOSIN(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46024Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46025Alpha1ACLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46026Alpha1ACLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46027Alpha1ACLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46028Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46029Alpha1ACLONEDHUMAN3H-PRAZOSIN(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46030Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46031Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46032Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46033Alpha1BCLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46034Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46035Alpha1BCLONEDHUMAN3H-PRAZOSIN(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46036Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46037Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46038Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46039Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46040Alpha1BCLONEDHUMAN3H-PRAZOSINPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46041Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46042Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46043Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46044Alpha1BCLONEDHUMAN3H-PRAZOSIN(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46045Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46046Alpha1BCLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46047Alpha1BCLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46048Alpha1BCLONEDHUMAN3H-PRAZOSINPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46049Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46050Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46051Alpha1BCLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46052Alpha1BCLONEDHUMAN3H-PRAZOSINPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46053Alpha1BCLONEDHUMAN3H-PRAZOSINPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46054Alpha1BCLONEDHUMAN3H-PRAZOSINN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46055Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46056Alpha1BCLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46057Alpha1BCLONEDHUMAN3H-PRAZOSIN(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46058Alpha1BCLONEDHUMAN3H-PRAZOSIN(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46059Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46060Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46061Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46062Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46063Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46064Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46065Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46066Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46067Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46068Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46069Alpha2ACLONEDHUMAN3H-CLONIDINE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46070Alpha2ACLONEDHUMAN3H-CLONIDINE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46071Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46072Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46073Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46074Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46075Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46076Alpha2ACLONEDHUMAN3H-CLONIDINEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46077Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46078Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46079Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46080Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46081Alpha2ACLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46082Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46083Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46084Alpha2ACLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46085Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46086Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46087Alpha2ACLONEDHUMAN3H-CLONIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46088Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46089Alpha2ACLONEDHUMAN3H-CLONIDINEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46090Alpha2ACLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46091Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46092Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46093Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46094Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-048-4325.9Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46095Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46096Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46097Alpha2BCLONEDHUMAN3H-CLONIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46098Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46099Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46100Alpha2BCLONEDHUMAN3H-CLONIDINEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46101Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46102Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione1498Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46103Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46104Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46105Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone1205Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46106Alpha2BCLONEDHUMAN3H-CLONIDINE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46107Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46108Alpha2BCLONEDHUMAN3H-CLONIDINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46109Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone23.36Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46110Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46111Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46112Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46113Alpha2BCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46114Alpha2BCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46115Alpha2BCLONEDHUMAN3H-CLONIDINE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46116Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46117Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46118Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46119Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46120Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46121Alpha2BCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46122Alpha2CCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46123Alpha2CCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46124Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46125Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46126Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46127Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46128Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46129Alpha2CCLONEDHUMAN3H-CLONIDINE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46130Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3998Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46131Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46132Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione27.03Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46133Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46134Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46135Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46136Alpha2CCLONEDHUMAN3H-CLONIDINE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46137Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46138Alpha2CCLONEDHUMAN3H-CLONIDINE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46139Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46140Alpha2CCLONEDHUMAN3H-CLONIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46141Alpha2CCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46142Alpha2CCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46143Alpha2CCLONEDHUMAN3H-CLONIDINEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46144Alpha2CCLONEDHUMAN3H-CLONIDINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46145Alpha2CCLONEDHUMAN3H-CLONIDINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46146Alpha2CCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46147Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46148Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46149Alpha2CCLONEDHUMAN3H-CLONIDINEPL-3-025263.3Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46150Alpha2CCLONEDHUMAN3H-CLONIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46151Alpha2CCLONEDHUMAN3H-CLONIDINEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46152Alpha2CCLONEDHUMAN3H-CLONIDINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone205.3Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46153Beta1CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46154Beta1CLONEDRAT125I-Pindolol(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46155Beta1CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46156Beta1CLONEDRAT125I-Pindolol(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46157Beta1CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46158Beta1CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46159Beta1CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46160Beta1CLONEDRAT125I-Pindolol(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46161Beta1CLONEDRAT125I-Pindolol(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46162Beta1CLONEDRAT125I-Pindolol(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46163Beta1CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46164Beta1CLONEDRAT125I-Pindolol(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46165Beta1CLONEDRAT125I-PindololPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46166Beta1CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46167Beta1CLONEDRAT125I-Pindolol(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46168Beta1CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46169Beta1CLONEDRAT125I-PindololPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46170Beta1CLONEDRAT125I-Pindolol(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46171Beta1CLONEDRAT125I-PindololPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46172Beta1CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46173Beta1CLONEDRAT125I-PindololPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46174Beta1CLONEDRAT125I-PindololN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46175Beta1CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46176Beta1CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46177Beta1CLONEDRAT125I-Pindolol(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46178Beta1CLONEDRAT125I-Pindolol(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46179Beta1CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46180Beta1CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46181Beta1CLONEDRAT125I-Pindolol(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46182Beta1CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46183Beta2CLONEDRAT125I-Pindolol(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46184Beta2CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46185Beta2CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46186Beta2CLONEDRAT125I-PindololPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46187Beta2CLONEDRAT125I-Pindolol(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46188Beta2CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46189Beta2CLONEDRAT125I-Pindolol(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46190Beta2CLONEDRAT125I-PindololPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46191Beta2CLONEDRAT125I-Pindolol(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46192Beta2CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46193Beta2CLONEDRAT125I-PindololPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46194Beta2CLONEDRAT125I-Pindolol(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46195Beta2CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46196Beta2CLONEDRAT125I-Pindolol(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46197Beta2CLONEDRAT125I-Pindolol(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46198Beta2CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46199Beta2CLONEDRAT125I-Pindolol(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46200Beta2CLONEDRAT125I-Pindolol(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46201Beta2CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46202Beta2CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46203Beta2CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46204Beta2CLONEDRAT125I-Pindolol(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46205Beta2CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46206Beta2CLONEDRAT125I-PindololN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46207Beta2CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46208Beta2CLONEDRAT125I-PindololPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46209Beta2CLONEDRAT125I-Pindolol(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46210Beta2CLONEDRAT125I-Pindolol(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46211Beta2CLONEDRAT125I-Pindolol(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46212Beta2CLONEDRAT125I-Pindolol(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46213GABAACLONEDHUMANFNZ(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46214GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46215GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46216GABAACLONEDHUMANFNZPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46217GABAACLONEDHUMANFNZPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46218GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46219GABAACLONEDHUMANFNZPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46220GABAACLONEDHUMANFNZ(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46221GABAACLONEDHUMANFNZN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46222GABAACLONEDHUMANFNZ(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46223GABAACLONEDHUMANFNZ(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46224GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46225GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46226GABAACLONEDHUMANFNZ(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46227GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46228GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46229GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46230GABAACLONEDHUMANFNZ(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46231GABAACLONEDHUMANFNZ(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46232GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46233GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46234GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46235GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46236GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46237GABAACLONEDHUMANFNZPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46238GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46239GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46240GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46241GABAACLONEDHUMANFNZ(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46242GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46243GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46244GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46245GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46246GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46247GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46248GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46249GABAACLONEDHUMANFNZ(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46250GABAACLONEDHUMANFNZ(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46251GABAACLONEDHUMANFNZ(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46252GABAACLONEDHUMANFNZ(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46253GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46254GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46255GABAACLONEDHUMANFNZ(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46256GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46257GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46258GABAACLONEDHUMANFNZN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46259GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46260GABAACLONEDHUMANFNZ(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46261GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46262GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46263GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46264GABAACLONEDHUMANFNZPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46265GABAACLONEDHUMANFNZPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46266GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46267GABAACLONEDHUMANFNZPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46268GABAACLONEDHUMANFNZ(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46269GABAACLONEDHUMANFNZPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46270GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46271GABAACLONEDHUMANFNZ(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46272GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46273GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46274GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46275GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46276GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46277GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46278GABAACLONEDHUMANFNZ(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46279GABAACLONEDHUMANFNZ(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46280GABAACLONEDHUMANFNZ(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46281GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46282GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46283GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46284GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46285GABAACLONEDHUMANFNZPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46286GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46287GABAACLONEDHUMANFNZ(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46288GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46289GABAACLONEDHUMANFNZPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46290GABAACLONEDHUMANFNZ(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46291GABAACLONEDHUMANFNZ(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46292GABAACLONEDHUMANFNZ(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46293GABAACLONEDHUMANFNZPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46294GABAACLONEDHUMANFNZPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46295GABAACLONEDHUMANFNZN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46296GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46297GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46298GABAACLONEDHUMANFNZ(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46299GABAACLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46300GABAACLONEDHUMANFNZ(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46301GABAACLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46302GABAACLONEDHUMANFNZ(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46303CLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46304CLONEDHUMANFNZPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46305CLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46306CLONEDHUMANFNZ(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46307CLONEDHUMANFNZ(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46308CLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46309CLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46310CLONEDHUMANFNZPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46311CLONEDHUMANFNZN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46312CLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46313CLONEDHUMANFNZ(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46314CLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46315CLONEDHUMANFNZPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46316CLONEDHUMANFNZ(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46317CLONEDHUMANFNZ(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46318CLONEDHUMANFNZ(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46319CLONEDHUMANFNZ(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46320CLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46321CLONEDHUMANFNZ(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46322CLONEDHUMANFNZ(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46323CLONEDHUMANFNZ(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46324CLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46325CLONEDHUMANFNZ(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46326CLONEDHUMANFNZ(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46327CLONEDHUMANFNZ(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46328CLONEDHUMANFNZ(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46329CLONEDHUMANFNZ(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46330CLONEDHUMANFNZPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46331CLONEDHUMANFNZ(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46332CLONEDHUMANFNZ(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46333HEARTRAT3H-Nitrendipine(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46334HEARTRAT3H-NitrendipinePL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46335HEARTRAT3H-Nitrendipine(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46336HEARTRAT3H-NitrendipinePL-3-025411Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46337HEARTRAT3H-Nitrendipine(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione643.1Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46338HEARTRAT3H-Nitrendipine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46339HEARTRAT3H-Nitrendipine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46340HEARTRAT3H-Nitrendipine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46341HEARTRAT3H-Nitrendipine(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46342HEARTRAT3H-Nitrendipine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione2976Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46343HEARTRAT3H-Nitrendipine(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione589.3Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46344HEARTRAT3H-Nitrendipine(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46345HEARTRAT3H-NitrendipinePL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46346HEARTRAT3H-NitrendipinePL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46347HEARTRAT3H-Nitrendipine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46348HEARTRAT3H-Nitrendipine(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46349HEARTRAT3H-Nitrendipine(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46350HEARTRAT3H-Nitrendipine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46351HEARTRAT3H-Nitrendipine(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46352HEARTRAT3H-Nitrendipine(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46353HEARTRAT3H-Nitrendipine(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46354HEARTRAT3H-Nitrendipine(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46355HEARTRAT3H-Nitrendipine(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46356HEARTRAT3H-Nitrendipine(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46357HEARTRAT3H-Nitrendipine(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46358HEARTRAT3H-Nitrendipine(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46359HEARTRAT3H-Nitrendipine(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46360HEARTRAT3H-Nitrendipine(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46361HEARTRAT3H-NitrendipineN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46362CB1BRAINRAT3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46363CB1BRAINRAT3H-CP-55940(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46364CB1BRAINRAT3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46365CB1BRAINRAT3H-CP-55940PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46366CB1BRAINRAT3H-CP-55940(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46367CB1BRAINRAT3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione5610Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46368CB1BRAINRAT3H-CP-55940(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46369CB1BRAINRAT3H-CP-55940(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46370CB1BRAINRAT3H-CP-55940N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46371CB1BRAINRAT3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46372CB1BRAINRAT3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46373CB1BRAINRAT3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46374CB1BRAINRAT3H-CP-55940(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46375CB1BRAINRAT3H-CP-55940PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46376CB1BRAINRAT3H-CP-55940(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46377CB1BRAINRAT3H-CP-55940(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46378CB1BRAINRAT3H-CP-55940PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46379CB1BRAINRAT3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46380CB1BRAINRAT3H-CP-55940(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46381CB1BRAINRAT3H-CP-55940PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46382CB1BRAINRAT3H-CP-55940(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46383CB1BRAINRAT3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46384CB1BRAINRAT3H-CP-55940(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46385CB1BRAINRAT3H-CP-55940(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46386CB1BRAINRAT3H-CP-55940(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46387CB1BRAINRAT3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46388CB1BRAINRAT3H-CP-55940(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46389CB1BRAINRAT3H-CP-55940(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46390CB1BRAINRAT3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46391CB1BRAINRAT3H-CP-55940(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46392CB2CLONEDHUMAN3H-CP-55940N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46393CB2CLONEDHUMAN3H-CP-55940(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46394CB2CLONEDHUMAN3H-CP-55940(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46395CB2CLONEDHUMAN3H-CP-55940PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46396CB2CLONEDHUMAN3H-CP-55940PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46397CB2CLONEDHUMAN3H-CP-55940(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46398CB2CLONEDHUMAN3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46399CB2CLONEDHUMAN3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46400CB2CLONEDHUMAN3H-CP-55940(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46401CB2CLONEDHUMAN3H-CP-55940PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46402CB2CLONEDHUMAN3H-CP-55940(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46403CB2CLONEDHUMAN3H-CP-55940(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46404CB2CLONEDHUMAN3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46405CB2CLONEDHUMAN3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46406CB2CLONEDHUMAN3H-CP-55940(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46407CB2CLONEDHUMAN3H-CP-55940(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46408CB2CLONEDHUMAN3H-CP-55940(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46409CB2CLONEDHUMAN3H-CP-55940PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46410CB2CLONEDHUMAN3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46411CB2CLONEDHUMAN3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46412CB2CLONEDHUMAN3H-CP-55940(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46413CB2CLONEDHUMAN3H-CP-55940(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione6129Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46414CB2CLONEDHUMAN3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46415CB2CLONEDHUMAN3H-CP-55940(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46416CB2CLONEDHUMAN3H-CP-55940(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46417CB2CLONEDHUMAN3H-CP-55940(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46418CB2CLONEDHUMAN3H-CP-55940(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46419CB2CLONEDHUMAN3H-CP-55940(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46420CB2CLONEDHUMAN3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46421CB2CLONEDHUMAN3H-CP-55940(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46422D1CLONEDHUMAN3H-SCH23390(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46423D1CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46424D1CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46425D1CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46426D1CLONEDHUMAN3H-SCH23390(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46427D1CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46428D1CLONEDHUMAN3H-SCH23390PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46429D1CLONEDHUMAN3H-SCH23390N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46430D1CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46431D1CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46432D1CLONEDHUMAN3H-SCH23390(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46433D1CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46434D1CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46435D1CLONEDHUMAN3H-SCH23390(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46436D1CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46437D1CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46438D1CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione1676Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46439D1CLONEDHUMAN3H-SCH23390PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46440D1CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46441D1CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46442D1CLONEDHUMAN3H-SCH23390(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46443D1CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46444D1CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46445D1CLONEDHUMAN3H-SCH23390(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46446D1CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46447D1CLONEDHUMAN3H-SCH23390PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46448D1CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46449D1CLONEDHUMAN3H-SCH23390(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46450D1CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46451D1CLONEDHUMAN3H-SCH23390PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46452D2CLONEDHUMAN3H-NMSP(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46453D2CLONEDHUMAN3H-NMSP(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46454D2CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46455D2CLONEDHUMAN3H-NMSP(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46456D2CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46457D2CLONEDHUMAN3H-NMSP(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46458D2CLONEDHUMAN3H-NMSP(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46459D2CLONEDHUMAN3H-NMSP(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46460D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46461D2CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46462D2CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46463D2CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46464D2CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46465D2CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46466D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione443.5Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46467D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46468D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46469D2CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46470D2CLONEDHUMAN3H-NMSP(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46471D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46472D2CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46473D2CLONEDHUMAN3H-NMSPN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46474D2CLONEDHUMAN3H-NMSP(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46475D2CLONEDHUMAN3H-NMSPPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46476D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46477D2CLONEDHUMAN3H-NMSPPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46478D2CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46479D2CLONEDHUMAN3H-NMSPPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46480D2CLONEDHUMAN3H-NMSP(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46481D2CLONEDHUMAN3H-NMSP(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46482D2CLONEDHUMAN3H-NMSPPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46483D3CLONEDRAT3H-NMSP(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46484D3CLONEDRAT3H-NMSP(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46485D3CLONEDRAT3H-NMSP(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46486D3CLONEDRAT3H-NMSP(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46487D3CLONEDRAT3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46488D3CLONEDRAT3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46489D3CLONEDRAT3H-NMSP(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46490D3CLONEDRAT3H-NMSP(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46491D3CLONEDRAT3H-NMSP(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46492D3CLONEDRAT3H-NMSP(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46493D3CLONEDRAT3H-NMSP(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46494D3CLONEDRAT3H-NMSP(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46495D3CLONEDRAT3H-NMSP(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46496D3CLONEDRAT3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46497D3CLONEDRAT3H-NMSP(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46498D3CLONEDRAT3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46499D3CLONEDRAT3H-NMSP(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46500D3CLONEDRAT3H-NMSP(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46501D3CLONEDRAT3H-NMSP(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46502D3CLONEDRAT3H-NMSP(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46503D3CLONEDRAT3H-NMSPN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46504D3CLONEDRAT3H-NMSPPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46505D3CLONEDRAT3H-NMSPPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46506D3CLONEDRAT3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione9446Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46507D3CLONEDRAT3H-NMSPPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46508D3CLONEDRAT3H-NMSP(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46509D3CLONEDRAT3H-NMSPPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46510D3CLONEDRAT3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46511D3CLONEDRAT3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione7244Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46512D3CLONEDRAT3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46513D4CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46514D4CLONEDHUMAN3H-NMSP(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46515D4CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46516D4CLONEDHUMAN3H-NMSP(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46517D4CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46518D4CLONEDHUMAN3H-NMSP(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46519D4CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione2988Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46520D4CLONEDHUMAN3H-NMSP(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46521D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46522D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46523D4CLONEDHUMAN3H-NMSP(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid2457Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46524D4CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46525D4CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46526D4CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46527D4CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46528D4CLONEDHUMAN3H-NMSP(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46529D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46530D4CLONEDHUMAN3H-NMSP(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46531D4CLONEDHUMAN3H-NMSPPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46532D4CLONEDHUMAN3H-NMSP(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46533D4CLONEDHUMAN3H-NMSP(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46534D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46535D4CLONEDHUMAN3H-NMSPN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46536D4CLONEDHUMAN3H-NMSPPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46537D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46538D4CLONEDHUMAN3H-NMSP(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46539D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46540D4CLONEDHUMAN3H-NMSPPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46541D4CLONEDHUMAN3H-NMSP(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46542D4CLONEDHUMAN3H-NMSPPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46543D4CLONEDHUMAN3H-NMSP(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46544D4CLONEDHUMAN3H-NMSP(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46545D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46546D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46547D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46548D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid1824Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46549D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46550D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46551D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46552D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46553D5CLONEDHUMAN3H-SCH23390(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46554D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46555D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46556D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46557D5CLONEDHUMAN3H-SCH23390(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46558D5CLONEDHUMAN3H-SCH23390(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46559D5CLONEDHUMAN3H-SCH23390(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46560D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46561D5CLONEDHUMAN3H-SCH23390(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46562D5CLONEDHUMAN3H-SCH23390N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46563D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46564D5CLONEDHUMAN3H-SCH23390PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46565D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46566D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46567D5CLONEDHUMAN3H-SCH23390(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46568D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46569D5CLONEDHUMAN3H-SCH23390(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46570D5CLONEDHUMAN3H-SCH23390(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46571D5CLONEDHUMAN3H-SCH23390PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46572D5CLONEDHUMAN3H-SCH23390(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46573D5CLONEDHUMAN3H-SCH23390PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46574D5CLONEDHUMAN3H-SCH23390PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46575SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46576SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46577SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46578SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46579SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46580SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46581SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46582SLC6A3CLONEDHUMAN3H-WIN 35,428(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46583SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46584SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46585SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46586SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46587SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46588SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46589SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46590SLC6A3CLONEDHUMAN3H-WIN 35,428PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46591SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46592SLC6A3CLONEDHUMAN3H-WIN 35,428(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46593SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46594SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46595SLC6A3CLONEDHUMAN3H-WIN 35,428(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid6121Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46596SLC6A3CLONEDHUMAN3H-WIN 35,428N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46597SLC6A3CLONEDHUMAN3H-WIN 35,428(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46598SLC6A3CLONEDHUMAN3H-WIN 35,428PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46599SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46600SLC6A3CLONEDHUMAN3H-WIN 35,428PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46601SLC6A3CLONEDHUMAN3H-WIN 35,428(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46602SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46603SLC6A3CLONEDHUMAN3H-WIN 35,428(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46604SLC6A3CLONEDHUMAN3H-WIN 35,428PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46605DORFOREBRAINGUINEA PIG3H-DADLE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46606DORFOREBRAINGUINEA PIG3H-DADLE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46607DORFOREBRAINGUINEA PIG3H-DADLE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46608DORFOREBRAINGUINEA PIG3H-DADLE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46609DORFOREBRAINGUINEA PIG3H-DADLE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46610DORFOREBRAINGUINEA PIG3H-DADLE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46611DORFOREBRAINGUINEA PIG3H-DADLE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46612DORFOREBRAINGUINEA PIG3H-DADLE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46613DORFOREBRAINGUINEA PIG3H-DADLE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46614DORFOREBRAINGUINEA PIG3H-DADLEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025