45615 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE mirtazepine(+) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45616 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE mirtazepine(-) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45617 NET CLONED HUMAN 3H-Nisoxetine mirtazepine(-) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45618 SLC6A3 CLONED HUMAN 3H-WIN 35,428 mirtazepine(-) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45619 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Nefazodone 200 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45620 NET CLONED HUMAN 3H-Nisoxetine Nefazodone 360 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45621 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Nefazodone 360 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45622 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NOMIFENSINE 1010 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45623 NET CLONED HUMAN 3H-Nisoxetine NOMIFENSINE 15.6 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45624 SLC6A3 CLONED HUMAN 3H-WIN 35,428 NOMIFENSINE 56 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45625 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NORFLUOXETINE 1.47 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45626 NET CLONED HUMAN 3H-Nisoxetine NORFLUOXETINE 1426 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45627 SLC6A3 CLONED HUMAN 3H-WIN 35,428 NORFLUOXETINE 420 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45628 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NORTRYPTYLINE 18 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45629 NET CLONED HUMAN 3H-Nisoxetine NORTRYPTYLINE 4.37 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45630 SLC6A3 CLONED HUMAN 3H-WIN 35,428 NORTRYPTYLINE 1140 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45631 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Oxaprotiline 3900 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45632 NET CLONED HUMAN 3H-Nisoxetine Oxaprotiline 4.9 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45633 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Oxaprotiline 4340 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45634 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE PAROXETINE 0.13 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45635 NET CLONED HUMAN 3H-Nisoxetine PAROXETINE 40 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45636 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PAROXETINE 490 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45637 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Phenelzine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45638 NET CLONED HUMAN 3H-Nisoxetine Phenelzine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45639 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Phenelzine 8400 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45640 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Protriptyline 19.6 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45641 NET CLONED HUMAN 3H-Nisoxetine Protriptyline 1.41 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45642 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Protriptyline 2100 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45643 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE SERTRALINE 0.29 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45644 NET CLONED HUMAN 3H-Nisoxetine SERTRALINE 420 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45645 SLC6A3 CLONED HUMAN 3H-WIN 35,428 SERTRALINE 25 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45646 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Tomoxetine 8.9 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45647 NET CLONED HUMAN 3H-Nisoxetine Tomoxetine 2.03 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45648 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Tomoxetine 1080 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45649 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE TRANYLCYPROMINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45650 NET CLONED HUMAN 3H-Nisoxetine TRANYLCYPROMINE 5900 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45651 SLC6A3 CLONED HUMAN 3H-WIN 35,428 TRANYLCYPROMINE 5100 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45652 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE TRAZODONE 160 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45653 NET CLONED HUMAN 3H-Nisoxetine TRAZODONE 8500 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45654 SLC6A3 CLONED HUMAN 3H-WIN 35,428 TRAZODONE 7400 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45655 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Trimipramine 149 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45656 NET CLONED HUMAN 3H-Nisoxetine Trimipramine 2450 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45657 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Trimipramine 3780 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45658 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Venlafaxine 8.9 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45659 NET CLONED HUMAN 3H-Nisoxetine Venlafaxine 1060 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45660 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Venlafaxine 9300 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45661 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Viloxazine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45662 NET CLONED HUMAN 3H-Nisoxetine Viloxazine 155 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45663 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Viloxazine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45664 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE ZIMELIDINE 152 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45665 NET CLONED HUMAN 3H-Nisoxetine ZIMELIDINE 9400 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45666 SLC6A3 CLONED HUMAN 3H-WIN 35,428 ZIMELIDINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
45667 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45668 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45669 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PL-3-016 1760 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45670 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid 7308 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45671 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PL-3-025 2150 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45672 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PL-3-048-4 5000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45673 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45674 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione 7049 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45675 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid 2790 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45676 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45677 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45678 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45679 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide 2546 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45680 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 3275 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45681 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45682 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 4274 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45683 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45684 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45685 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45686 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45687 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45688 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 597.9 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45689 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45690 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45691 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 165.3 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45692 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45693 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45694 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45695 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid 1382 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45696 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45697 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45698 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 1774 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45699 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 63.46 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45700 5-HT1B CLONED HUMAN 3H-GR-125743 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45701 5-HT1B CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45702 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45703 5-HT1B CLONED HUMAN 3H-GR-125743 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45704 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45705 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45706 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45707 5-HT1B CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45708 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45709 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45710 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45711 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 8213 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45712 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45713 5-HT1B CLONED HUMAN 3H-GR-125743 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45714 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45715 5-HT1B CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45716 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45717 5-HT1B CLONED HUMAN 3H-GR-125743 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45718 5-HT1B CLONED HUMAN 3H-GR-125743 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45719 5-HT1B CLONED HUMAN 3H-GR-125743 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45720 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45721 5-HT1B CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45722 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45723 5-HT1B CLONED HUMAN 3H-GR-125743 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45724 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45725 5-HT1B CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45726 5-HT1B CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45727 5-HT1B CLONED HUMAN 3H-GR-125743 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45728 5-HT1B CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45729 5-HT1B CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45730 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45731 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45732 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45733 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45734 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45735 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45736 5-HT1D CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45737 5-HT1D CLONED HUMAN 3H-GR-125743 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45738 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45739 5-HT1D CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45740 5-HT1D CLONED HUMAN 3H-GR-125743 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45741 5-HT1D CLONED HUMAN 3H-GR-125743 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45742 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45743 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45744 5-HT1D CLONED HUMAN 3H-GR-125743 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45745 5-HT1D CLONED HUMAN 3H-GR-125743 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45746 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45747 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45748 5-HT1D CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45749 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45750 5-HT1D CLONED HUMAN 3H-GR-125743 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45751 5-HT1D CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45752 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45753 5-HT1D CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45754 5-HT1D CLONED HUMAN 3H-GR-125743 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45755 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45756 5-HT1D CLONED HUMAN 3H-GR-125743 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45757 5-HT1D CLONED HUMAN 3H-GR-125743 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45758 5-HT1D CLONED HUMAN 3H-GR-125743 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45759 5-HT1D CLONED HUMAN 3H-GR-125743 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45760 5-HT1E CLONED HUMAN 3H-5HT (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 5489 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45761 5-HT1E CLONED HUMAN 3H-5HT (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45762 5-HT1E CLONED HUMAN 3H-5HT (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45763 5-HT1E CLONED HUMAN 3H-5HT PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45764 5-HT1E CLONED HUMAN 3H-5HT N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45765 5-HT1E CLONED HUMAN 3H-5HT (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45766 5-HT1E CLONED HUMAN 3H-5HT (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45767 5-HT1E CLONED HUMAN 3H-5HT (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45768 5-HT1E CLONED HUMAN 3H-5HT PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45769 5-HT1E CLONED HUMAN 3H-5HT (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 5680 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45770 5-HT1E CLONED HUMAN 3H-5HT (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45771 5-HT1E CLONED HUMAN 3H-5HT PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45772 5-HT1E CLONED HUMAN 3H-5HT (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid 272.5 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45773 5-HT1E CLONED HUMAN 3H-5HT (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45774 5-HT1E CLONED HUMAN 3H-5HT (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45775 5-HT1E CLONED HUMAN 3H-5HT (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45776 5-HT1E CLONED HUMAN 3H-5HT (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45777 5-HT1E CLONED HUMAN 3H-5HT (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45778 5-HT1E CLONED HUMAN 3H-5HT (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45779 5-HT1E CLONED HUMAN 3H-5HT (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45780 5-HT1E CLONED HUMAN 3H-5HT (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45781 5-HT1E CLONED HUMAN 3H-5HT (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45782 5-HT1E CLONED HUMAN 3H-5HT (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45783 5-HT1E CLONED HUMAN 3H-5HT (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45784 5-HT1E CLONED HUMAN 3H-5HT (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45785 5-HT1E CLONED HUMAN 3H-5HT PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45786 5-HT1E CLONED HUMAN 3H-5HT (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45787 5-HT1E CLONED HUMAN 3H-5HT (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45788 5-HT1E CLONED HUMAN 3H-5HT (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45789 5-HT1E CLONED HUMAN 3H-5HT (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45790 5-HT2A CLONED HUMAN 3H-KETANSERIN PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45791 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45792 5-HT2A CLONED HUMAN 3H-KETANSERIN PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45793 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45794 5-HT2A CLONED HUMAN 3H-KETANSERIN (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45795 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45796 5-HT2A CLONED HUMAN 3H-KETANSERIN (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45797 5-HT2A CLONED HUMAN 3H-KETANSERIN PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45798 5-HT2A CLONED HUMAN 3H-KETANSERIN (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45799 5-HT2A CLONED HUMAN 3H-KETANSERIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45800 5-HT2A CLONED HUMAN 3H-KETANSERIN N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45801 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45802 5-HT2A CLONED HUMAN 3H-KETANSERIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45803 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45804 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45805 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45806 5-HT2A CLONED HUMAN 3H-KETANSERIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45807 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45808 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45809 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45810 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45811 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45812 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45813 5-HT2A CLONED HUMAN 3H-KETANSERIN (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45814 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45815 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45816 5-HT2A CLONED HUMAN 3H-KETANSERIN (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45817 5-HT2A CLONED HUMAN 3H-KETANSERIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45818 5-HT2A CLONED HUMAN 3H-KETANSERIN (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45819 5-HT2A CLONED HUMAN 3H-KETANSERIN PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45820 5-HT2B CLONED HUMAN 3H-LSD N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45821 5-HT2B CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45822 5-HT2B CLONED HUMAN 3H-LSD PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45823 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45824 5-HT2B CLONED HUMAN 3H-LSD (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45825 5-HT2B CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45826 5-HT2B CLONED HUMAN 3H-LSD (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45827 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45828 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45829 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45830 5-HT2B CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45831 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45832 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45833 5-HT2B CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45834 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45835 5-HT2B CLONED HUMAN 3H-LSD (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45836 5-HT2B CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45837 5-HT2B CLONED HUMAN 3H-LSD (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45838 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45839 5-HT2B CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45840 5-HT2B CLONED HUMAN 3H-LSD PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45841 5-HT2B CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45842 5-HT2B CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45843 5-HT2B CLONED HUMAN 3H-LSD (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45844 5-HT2B CLONED HUMAN 3H-LSD (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione 1460 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45845 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45846 5-HT2B CLONED HUMAN 3H-LSD PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45847 5-HT2B CLONED HUMAN 3H-LSD PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45848 5-HT2B CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45849 5-HT2B CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45850 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45851 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45852 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45853 5-HT2C CLONED RAT 3H-MESULERGINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45854 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45855 5-HT2C CLONED RAT 3H-MESULERGINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45856 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45857 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45858 5-HT2C CLONED RAT 3H-MESULERGINE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45859 5-HT2C CLONED RAT 3H-MESULERGINE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45860 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45861 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45862 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45863 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45864 5-HT2C CLONED RAT 3H-MESULERGINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45865 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45866 5-HT2C CLONED RAT 3H-MESULERGINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45867 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45868 5-HT2C CLONED RAT 3H-MESULERGINE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45869 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45870 5-HT2C CLONED RAT 3H-MESULERGINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45871 5-HT2C CLONED RAT 3H-MESULERGINE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45872 5-HT2C CLONED RAT 3H-MESULERGINE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45873 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45874 5-HT2C CLONED RAT 3H-MESULERGINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45875 5-HT2C CLONED RAT 3H-MESULERGINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45876 5-HT2C CLONED RAT 3H-MESULERGINE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45877 5-HT2C CLONED RAT 3H-MESULERGINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45878 5-HT2C CLONED RAT 3H-MESULERGINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45879 5-HT2C CLONED RAT 3H-MESULERGINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45880 5-HT2C CLONED RAT 3H-MESULERGINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45881 5-HT3 CLONED HUMAN 3H-ZACOPRIDE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45882 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45883 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45884 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45885 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45886 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45887 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45888 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45889 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45890 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45891 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45892 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45893 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45894 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45895 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45896 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45897 5-HT3 CLONED HUMAN 3H-ZACOPRIDE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45898 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45899 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45900 5-HT3 CLONED HUMAN 3H-ZACOPRIDE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45901 5-HT3 CLONED HUMAN 3H-ZACOPRIDE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45902 5-HT3 CLONED HUMAN 3H-ZACOPRIDE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45903 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45904 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45905 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45906 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45907 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45908 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45909 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45910 5-HT3 CLONED HUMAN 3H-ZACOPRIDE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45911 5-HT5A CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45912 5-HT5A CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45913 5-HT5A CLONED HUMAN 3H-LSD (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45914 5-HT5A CLONED HUMAN 3H-LSD (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45915 5-HT5A CLONED HUMAN 3H-LSD (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45916 5-HT5A CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45917 5-HT5A CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45918 5-HT5A CLONED HUMAN 3H-LSD (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45919 5-HT5A CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45920 5-HT5A CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45921 5-HT5A CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45922 5-HT5A CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45923 5-HT5A CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45924 5-HT5A CLONED HUMAN 3H-LSD (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45925 5-HT5A CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45926 5-HT5A CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45927 5-HT5A CLONED HUMAN 3H-LSD PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45928 5-HT5A CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45929 5-HT5A CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45930 5-HT5A CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45931 5-HT5A CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45932 5-HT5A CLONED HUMAN 3H-LSD PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45933 5-HT5A CLONED HUMAN 3H-LSD PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45934 5-HT5A CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45935 5-HT5A CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45936 5-HT5A CLONED HUMAN 3H-LSD (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45937 5-HT5A CLONED HUMAN 3H-LSD (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45938 5-HT5A CLONED HUMAN 3H-LSD PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45939 5-HT5A CLONED HUMAN 3H-LSD (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45940 5-HT5A CLONED HUMAN 3H-LSD N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45941 5-HT6 CLONED HUMAN 3H-LSD (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45942 5-HT6 CLONED HUMAN 3H-LSD (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45943 5-HT6 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45944 5-HT6 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45945 5-HT6 CLONED HUMAN 3H-LSD PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45946 5-HT6 CLONED HUMAN 3H-LSD PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45947 5-HT6 CLONED HUMAN 3H-LSD N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45948 5-HT6 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45949 5-HT6 CLONED HUMAN 3H-LSD PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45950 5-HT6 CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45951 5-HT6 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45952 5-HT6 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45953 5-HT6 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45954 5-HT6 CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45955 5-HT6 CLONED HUMAN 3H-LSD (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45956 5-HT6 CLONED HUMAN 3H-LSD (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45957 5-HT6 CLONED HUMAN 3H-LSD (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45958 5-HT6 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45959 5-HT6 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45960 5-HT6 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45961 5-HT6 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45962 5-HT6 CLONED HUMAN 3H-LSD (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45963 5-HT6 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45964 5-HT6 CLONED HUMAN 3H-LSD (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45965 5-HT6 CLONED HUMAN 3H-LSD PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45966 5-HT6 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45967 5-HT6 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45968 5-HT6 CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45969 5-HT6 CLONED HUMAN 3H-LSD (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45970 5-HT6 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45971 5-HT7 CLONED HUMAN 3H-LSD PL-3-017 3197 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45972 5-HT7 CLONED HUMAN 3H-LSD PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45973 5-HT7 CLONED HUMAN 3H-LSD N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide 775.2 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45974 5-HT7 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45975 5-HT7 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 793 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45976 5-HT7 CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45977 5-HT7 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45978 5-HT7 CLONED HUMAN 3H-LSD (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45979 5-HT7 CLONED HUMAN 3H-LSD PL-3-048-4 7290 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45980 5-HT7 CLONED HUMAN 3H-LSD (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione 2053 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45981 5-HT7 CLONED HUMAN 3H-LSD (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45982 5-HT7 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45983 5-HT7 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45984 5-HT7 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45985 5-HT7 CLONED HUMAN 3H-LSD (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45986 5-HT7 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 2005 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45987 5-HT7 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45988 5-HT7 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45989 5-HT7 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45990 5-HT7 CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45991 5-HT7 CLONED HUMAN 3H-LSD (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45992 5-HT7 CLONED HUMAN 3H-LSD (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45993 5-HT7 CLONED HUMAN 3H-LSD (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid 3761 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45994 5-HT7 CLONED HUMAN 3H-LSD (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45995 5-HT7 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45996 5-HT7 CLONED HUMAN 3H-LSD (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45997 5-HT7 CLONED HUMAN 3H-LSD (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45998 5-HT7 CLONED HUMAN 3H-LSD (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
45999 5-HT7 CLONED HUMAN 3H-LSD PL-3-025 2762 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46000 5-HT7 CLONED HUMAN 3H-LSD (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46001 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46002 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46003 Alpha1A CLONED HUMAN 3H-PRAZOSIN PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46004 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46005 Alpha1A CLONED HUMAN 3H-PRAZOSIN PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46006 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46007 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46008 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46009 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46010 Alpha1A CLONED HUMAN 3H-PRAZOSIN N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46011 Alpha1A CLONED HUMAN 3H-PRAZOSIN PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46012 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46013 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46014 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46015 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46016 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46017 Alpha1A CLONED HUMAN 3H-PRAZOSIN PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46018 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46019 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46020 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46021 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46022 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46023 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46024 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46025 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46026 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46027 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46028 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46029 Alpha1A CLONED HUMAN 3H-PRAZOSIN (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46030 Alpha1A CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46031 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46032 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46033 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46034 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46035 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46036 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46037 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46038 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46039 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46040 Alpha1B CLONED HUMAN 3H-PRAZOSIN PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46041 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46042 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46043 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46044 Alpha1B CLONED HUMAN 3H-PRAZOSIN (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46045 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46046 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46047 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46048 Alpha1B CLONED HUMAN 3H-PRAZOSIN PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46049 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46050 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46051 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46052 Alpha1B CLONED HUMAN 3H-PRAZOSIN PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46053 Alpha1B CLONED HUMAN 3H-PRAZOSIN PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46054 Alpha1B CLONED HUMAN 3H-PRAZOSIN N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46055 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46056 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46057 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46058 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46059 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46060 Alpha1B CLONED HUMAN 3H-PRAZOSIN (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46061 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46062 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46063 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46064 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46065 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46066 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46067 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46068 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46069 Alpha2A CLONED HUMAN 3H-CLONIDINE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46070 Alpha2A CLONED HUMAN 3H-CLONIDINE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46071 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46072 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46073 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46074 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46075 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46076 Alpha2A CLONED HUMAN 3H-CLONIDINE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46077 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46078 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46079 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46080 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46081 Alpha2A CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46082 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46083 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46084 Alpha2A CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46085 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46086 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46087 Alpha2A CLONED HUMAN 3H-CLONIDINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46088 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46089 Alpha2A CLONED HUMAN 3H-CLONIDINE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46090 Alpha2A CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46091 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46092 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46093 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46094 Alpha2B CLONED HUMAN 3H-CLONIDINE PL-3-048-4 325.9 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46095 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46096 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46097 Alpha2B CLONED HUMAN 3H-CLONIDINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46098 Alpha2B CLONED HUMAN 3H-CLONIDINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46099 Alpha2B CLONED HUMAN 3H-CLONIDINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46100 Alpha2B CLONED HUMAN 3H-CLONIDINE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46101 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46102 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 1498 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46103 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46104 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46105 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone 1205 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46106 Alpha2B CLONED HUMAN 3H-CLONIDINE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46107 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46108 Alpha2B CLONED HUMAN 3H-CLONIDINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46109 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone 23.36 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46110 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46111 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46112 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46113 Alpha2B CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46114 Alpha2B CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46115 Alpha2B CLONED HUMAN 3H-CLONIDINE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46116 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46117 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46118 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46119 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46120 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46121 Alpha2B CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46122 Alpha2C CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46123 Alpha2C CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46124 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46125 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46126 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46127 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46128 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46129 Alpha2C CLONED HUMAN 3H-CLONIDINE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46130 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 3998 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46131 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46132 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 27.03 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46133 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46134 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46135 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46136 Alpha2C CLONED HUMAN 3H-CLONIDINE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46137 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46138 Alpha2C CLONED HUMAN 3H-CLONIDINE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46139 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46140 Alpha2C CLONED HUMAN 3H-CLONIDINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46141 Alpha2C CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46142 Alpha2C CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46143 Alpha2C CLONED HUMAN 3H-CLONIDINE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46144 Alpha2C CLONED HUMAN 3H-CLONIDINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46145 Alpha2C CLONED HUMAN 3H-CLONIDINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46146 Alpha2C CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46147 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46148 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46149 Alpha2C CLONED HUMAN 3H-CLONIDINE PL-3-025 263.3 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46150 Alpha2C CLONED HUMAN 3H-CLONIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46151 Alpha2C CLONED HUMAN 3H-CLONIDINE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46152 Alpha2C CLONED HUMAN 3H-CLONIDINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone 205.3 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46153 Beta1 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46154 Beta1 CLONED RAT 125I-Pindolol (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46155 Beta1 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46156 Beta1 CLONED RAT 125I-Pindolol (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46157 Beta1 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46158 Beta1 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46159 Beta1 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46160 Beta1 CLONED RAT 125I-Pindolol (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46161 Beta1 CLONED RAT 125I-Pindolol (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46162 Beta1 CLONED RAT 125I-Pindolol (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46163 Beta1 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46164 Beta1 CLONED RAT 125I-Pindolol (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46165 Beta1 CLONED RAT 125I-Pindolol PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46166 Beta1 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46167 Beta1 CLONED RAT 125I-Pindolol (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46168 Beta1 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46169 Beta1 CLONED RAT 125I-Pindolol PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46170 Beta1 CLONED RAT 125I-Pindolol (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46171 Beta1 CLONED RAT 125I-Pindolol PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46172 Beta1 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46173 Beta1 CLONED RAT 125I-Pindolol PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46174 Beta1 CLONED RAT 125I-Pindolol N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46175 Beta1 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46176 Beta1 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46177 Beta1 CLONED RAT 125I-Pindolol (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46178 Beta1 CLONED RAT 125I-Pindolol (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46179 Beta1 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46180 Beta1 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46181 Beta1 CLONED RAT 125I-Pindolol (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46182 Beta1 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46183 Beta2 CLONED RAT 125I-Pindolol (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46184 Beta2 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46185 Beta2 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46186 Beta2 CLONED RAT 125I-Pindolol PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46187 Beta2 CLONED RAT 125I-Pindolol (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46188 Beta2 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46189 Beta2 CLONED RAT 125I-Pindolol (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46190 Beta2 CLONED RAT 125I-Pindolol PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46191 Beta2 CLONED RAT 125I-Pindolol (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46192 Beta2 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46193 Beta2 CLONED RAT 125I-Pindolol PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46194 Beta2 CLONED RAT 125I-Pindolol (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46195 Beta2 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46196 Beta2 CLONED RAT 125I-Pindolol (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46197 Beta2 CLONED RAT 125I-Pindolol (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46198 Beta2 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46199 Beta2 CLONED RAT 125I-Pindolol (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46200 Beta2 CLONED RAT 125I-Pindolol (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46201 Beta2 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46202 Beta2 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46203 Beta2 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46204 Beta2 CLONED RAT 125I-Pindolol (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46205 Beta2 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46206 Beta2 CLONED RAT 125I-Pindolol N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46207 Beta2 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46208 Beta2 CLONED RAT 125I-Pindolol PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46209 Beta2 CLONED RAT 125I-Pindolol (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46210 Beta2 CLONED RAT 125I-Pindolol (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46211 Beta2 CLONED RAT 125I-Pindolol (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46212 Beta2 CLONED RAT 125I-Pindolol (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46213 GABAA CLONED HUMAN FNZ (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46214 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46215 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46216 GABAA CLONED HUMAN FNZ PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46217 GABAA CLONED HUMAN FNZ PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46218 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46219 GABAA CLONED HUMAN FNZ PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46220 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46221 GABAA CLONED HUMAN FNZ N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46222 GABAA CLONED HUMAN FNZ (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46223 GABAA CLONED HUMAN FNZ (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46224 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46225 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46226 GABAA CLONED HUMAN FNZ (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46227 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46228 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46229 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46230 GABAA CLONED HUMAN FNZ (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46231 GABAA CLONED HUMAN FNZ (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46232 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46233 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46234 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46235 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46236 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46237 GABAA CLONED HUMAN FNZ PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46238 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46239 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46240 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46241 GABAA CLONED HUMAN FNZ (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46242 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46243 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46244 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46245 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46246 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46247 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46248 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46249 GABAA CLONED HUMAN FNZ (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46250 GABAA CLONED HUMAN FNZ (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46251 GABAA CLONED HUMAN FNZ (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46252 GABAA CLONED HUMAN FNZ (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46253 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46254 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46255 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46256 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46257 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46258 GABAA CLONED HUMAN FNZ N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46259 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46260 GABAA CLONED HUMAN FNZ (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46261 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46262 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46263 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46264 GABAA CLONED HUMAN FNZ PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46265 GABAA CLONED HUMAN FNZ PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46266 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46267 GABAA CLONED HUMAN FNZ PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46268 GABAA CLONED HUMAN FNZ (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46269 GABAA CLONED HUMAN FNZ PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46270 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46271 GABAA CLONED HUMAN FNZ (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46272 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46273 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46274 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46275 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46276 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46277 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46278 GABAA CLONED HUMAN FNZ (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46279 GABAA CLONED HUMAN FNZ (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46280 GABAA CLONED HUMAN FNZ (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46281 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46282 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46283 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46284 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46285 GABAA CLONED HUMAN FNZ PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46286 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46287 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46288 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46289 GABAA CLONED HUMAN FNZ PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46290 GABAA CLONED HUMAN FNZ (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46291 GABAA CLONED HUMAN FNZ (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46292 GABAA CLONED HUMAN FNZ (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46293 GABAA CLONED HUMAN FNZ PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46294 GABAA CLONED HUMAN FNZ PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46295 GABAA CLONED HUMAN FNZ N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46296 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46297 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46298 GABAA CLONED HUMAN FNZ (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46299 GABAA CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46300 GABAA CLONED HUMAN FNZ (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46301 GABAA CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46302 GABAA CLONED HUMAN FNZ (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46303 CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46304 CLONED HUMAN FNZ PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46305 CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46306 CLONED HUMAN FNZ (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46307 CLONED HUMAN FNZ (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46308 CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46309 CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46310 CLONED HUMAN FNZ PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46311 CLONED HUMAN FNZ N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46312 CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46313 CLONED HUMAN FNZ (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46314 CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46315 CLONED HUMAN FNZ PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46316 CLONED HUMAN FNZ (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46317 CLONED HUMAN FNZ (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46318 CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46319 CLONED HUMAN FNZ (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46320 CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46321 CLONED HUMAN FNZ (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46322 CLONED HUMAN FNZ (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46323 CLONED HUMAN FNZ (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46324 CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46325 CLONED HUMAN FNZ (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46326 CLONED HUMAN FNZ (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46327 CLONED HUMAN FNZ (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46328 CLONED HUMAN FNZ (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46329 CLONED HUMAN FNZ (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46330 CLONED HUMAN FNZ PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46331 CLONED HUMAN FNZ (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46332 CLONED HUMAN FNZ (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46333 HEART RAT 3H-Nitrendipine (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46334 HEART RAT 3H-Nitrendipine PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46335 HEART RAT 3H-Nitrendipine (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46336 HEART RAT 3H-Nitrendipine PL-3-025 411 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46337 HEART RAT 3H-Nitrendipine (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 643.1 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46338 HEART RAT 3H-Nitrendipine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46339 HEART RAT 3H-Nitrendipine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46340 HEART RAT 3H-Nitrendipine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46341 HEART RAT 3H-Nitrendipine (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46342 HEART RAT 3H-Nitrendipine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 2976 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46343 HEART RAT 3H-Nitrendipine (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 589.3 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46344 HEART RAT 3H-Nitrendipine (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46345 HEART RAT 3H-Nitrendipine PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46346 HEART RAT 3H-Nitrendipine PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46347 HEART RAT 3H-Nitrendipine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46348 HEART RAT 3H-Nitrendipine (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46349 HEART RAT 3H-Nitrendipine (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46350 HEART RAT 3H-Nitrendipine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46351 HEART RAT 3H-Nitrendipine (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46352 HEART RAT 3H-Nitrendipine (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46353 HEART RAT 3H-Nitrendipine (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46354 HEART RAT 3H-Nitrendipine (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46355 HEART RAT 3H-Nitrendipine (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46356 HEART RAT 3H-Nitrendipine (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46357 HEART RAT 3H-Nitrendipine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46358 HEART RAT 3H-Nitrendipine (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46359 HEART RAT 3H-Nitrendipine (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46360 HEART RAT 3H-Nitrendipine (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46361 HEART RAT 3H-Nitrendipine N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46362 CB1 BRAIN RAT 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46363 CB1 BRAIN RAT 3H-CP-55940 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46364 CB1 BRAIN RAT 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46365 CB1 BRAIN RAT 3H-CP-55940 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46366 CB1 BRAIN RAT 3H-CP-55940 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46367 CB1 BRAIN RAT 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 5610 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46368 CB1 BRAIN RAT 3H-CP-55940 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46369 CB1 BRAIN RAT 3H-CP-55940 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46370 CB1 BRAIN RAT 3H-CP-55940 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46371 CB1 BRAIN RAT 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46372 CB1 BRAIN RAT 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46373 CB1 BRAIN RAT 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46374 CB1 BRAIN RAT 3H-CP-55940 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46375 CB1 BRAIN RAT 3H-CP-55940 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46376 CB1 BRAIN RAT 3H-CP-55940 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46377 CB1 BRAIN RAT 3H-CP-55940 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46378 CB1 BRAIN RAT 3H-CP-55940 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46379 CB1 BRAIN RAT 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46380 CB1 BRAIN RAT 3H-CP-55940 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46381 CB1 BRAIN RAT 3H-CP-55940 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46382 CB1 BRAIN RAT 3H-CP-55940 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46383 CB1 BRAIN RAT 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46384 CB1 BRAIN RAT 3H-CP-55940 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46385 CB1 BRAIN RAT 3H-CP-55940 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46386 CB1 BRAIN RAT 3H-CP-55940 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46387 CB1 BRAIN RAT 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46388 CB1 BRAIN RAT 3H-CP-55940 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46389 CB1 BRAIN RAT 3H-CP-55940 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46390 CB1 BRAIN RAT 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46391 CB1 BRAIN RAT 3H-CP-55940 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46392 CB2 CLONED HUMAN 3H-CP-55940 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46393 CB2 CLONED HUMAN 3H-CP-55940 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46394 CB2 CLONED HUMAN 3H-CP-55940 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46395 CB2 CLONED HUMAN 3H-CP-55940 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46396 CB2 CLONED HUMAN 3H-CP-55940 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46397 CB2 CLONED HUMAN 3H-CP-55940 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46398 CB2 CLONED HUMAN 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46399 CB2 CLONED HUMAN 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46400 CB2 CLONED HUMAN 3H-CP-55940 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46401 CB2 CLONED HUMAN 3H-CP-55940 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46402 CB2 CLONED HUMAN 3H-CP-55940 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46403 CB2 CLONED HUMAN 3H-CP-55940 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46404 CB2 CLONED HUMAN 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46405 CB2 CLONED HUMAN 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46406 CB2 CLONED HUMAN 3H-CP-55940 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46407 CB2 CLONED HUMAN 3H-CP-55940 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46408 CB2 CLONED HUMAN 3H-CP-55940 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46409 CB2 CLONED HUMAN 3H-CP-55940 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46410 CB2 CLONED HUMAN 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46411 CB2 CLONED HUMAN 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46412 CB2 CLONED HUMAN 3H-CP-55940 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46413 CB2 CLONED HUMAN 3H-CP-55940 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 6129 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46414 CB2 CLONED HUMAN 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46415 CB2 CLONED HUMAN 3H-CP-55940 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46416 CB2 CLONED HUMAN 3H-CP-55940 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46417 CB2 CLONED HUMAN 3H-CP-55940 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46418 CB2 CLONED HUMAN 3H-CP-55940 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46419 CB2 CLONED HUMAN 3H-CP-55940 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46420 CB2 CLONED HUMAN 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46421 CB2 CLONED HUMAN 3H-CP-55940 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46422 D1 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46423 D1 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46424 D1 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46425 D1 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46426 D1 CLONED HUMAN 3H-SCH23390 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46427 D1 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46428 D1 CLONED HUMAN 3H-SCH23390 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46429 D1 CLONED HUMAN 3H-SCH23390 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46430 D1 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46431 D1 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46432 D1 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46433 D1 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46434 D1 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46435 D1 CLONED HUMAN 3H-SCH23390 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46436 D1 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46437 D1 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46438 D1 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 1676 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46439 D1 CLONED HUMAN 3H-SCH23390 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46440 D1 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46441 D1 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46442 D1 CLONED HUMAN 3H-SCH23390 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46443 D1 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46444 D1 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46445 D1 CLONED HUMAN 3H-SCH23390 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46446 D1 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46447 D1 CLONED HUMAN 3H-SCH23390 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46448 D1 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46449 D1 CLONED HUMAN 3H-SCH23390 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46450 D1 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46451 D1 CLONED HUMAN 3H-SCH23390 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46452 D2 CLONED HUMAN 3H-NMSP (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46453 D2 CLONED HUMAN 3H-NMSP (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46454 D2 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46455 D2 CLONED HUMAN 3H-NMSP (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46456 D2 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46457 D2 CLONED HUMAN 3H-NMSP (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46458 D2 CLONED HUMAN 3H-NMSP (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46459 D2 CLONED HUMAN 3H-NMSP (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46460 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46461 D2 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46462 D2 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46463 D2 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46464 D2 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46465 D2 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46466 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 443.5 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46467 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46468 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46469 D2 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46470 D2 CLONED HUMAN 3H-NMSP (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46471 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46472 D2 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46473 D2 CLONED HUMAN 3H-NMSP N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46474 D2 CLONED HUMAN 3H-NMSP (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46475 D2 CLONED HUMAN 3H-NMSP PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46476 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46477 D2 CLONED HUMAN 3H-NMSP PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46478 D2 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46479 D2 CLONED HUMAN 3H-NMSP PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46480 D2 CLONED HUMAN 3H-NMSP (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46481 D2 CLONED HUMAN 3H-NMSP (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46482 D2 CLONED HUMAN 3H-NMSP PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46483 D3 CLONED RAT 3H-NMSP (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46484 D3 CLONED RAT 3H-NMSP (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46485 D3 CLONED RAT 3H-NMSP (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46486 D3 CLONED RAT 3H-NMSP (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46487 D3 CLONED RAT 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46488 D3 CLONED RAT 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46489 D3 CLONED RAT 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46490 D3 CLONED RAT 3H-NMSP (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46491 D3 CLONED RAT 3H-NMSP (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46492 D3 CLONED RAT 3H-NMSP (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46493 D3 CLONED RAT 3H-NMSP (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46494 D3 CLONED RAT 3H-NMSP (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46495 D3 CLONED RAT 3H-NMSP (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46496 D3 CLONED RAT 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46497 D3 CLONED RAT 3H-NMSP (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46498 D3 CLONED RAT 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46499 D3 CLONED RAT 3H-NMSP (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46500 D3 CLONED RAT 3H-NMSP (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46501 D3 CLONED RAT 3H-NMSP (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46502 D3 CLONED RAT 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46503 D3 CLONED RAT 3H-NMSP N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46504 D3 CLONED RAT 3H-NMSP PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46505 D3 CLONED RAT 3H-NMSP PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46506 D3 CLONED RAT 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 9446 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46507 D3 CLONED RAT 3H-NMSP PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46508 D3 CLONED RAT 3H-NMSP (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46509 D3 CLONED RAT 3H-NMSP PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46510 D3 CLONED RAT 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46511 D3 CLONED RAT 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 7244 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46512 D3 CLONED RAT 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46513 D4 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46514 D4 CLONED HUMAN 3H-NMSP (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46515 D4 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46516 D4 CLONED HUMAN 3H-NMSP (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46517 D4 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46518 D4 CLONED HUMAN 3H-NMSP (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46519 D4 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 2988 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46520 D4 CLONED HUMAN 3H-NMSP (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46521 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46522 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46523 D4 CLONED HUMAN 3H-NMSP (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid 2457 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46524 D4 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46525 D4 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46526 D4 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46527 D4 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46528 D4 CLONED HUMAN 3H-NMSP (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46529 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46530 D4 CLONED HUMAN 3H-NMSP (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46531 D4 CLONED HUMAN 3H-NMSP PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46532 D4 CLONED HUMAN 3H-NMSP (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46533 D4 CLONED HUMAN 3H-NMSP (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46534 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46535 D4 CLONED HUMAN 3H-NMSP N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46536 D4 CLONED HUMAN 3H-NMSP PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46537 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46538 D4 CLONED HUMAN 3H-NMSP (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46539 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46540 D4 CLONED HUMAN 3H-NMSP PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46541 D4 CLONED HUMAN 3H-NMSP (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46542 D4 CLONED HUMAN 3H-NMSP PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46543 D4 CLONED HUMAN 3H-NMSP (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46544 D4 CLONED HUMAN 3H-NMSP (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46545 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46546 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46547 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46548 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid 1824 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46549 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46550 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46551 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46552 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46553 D5 CLONED HUMAN 3H-SCH23390 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46554 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46555 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46556 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46557 D5 CLONED HUMAN 3H-SCH23390 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46558 D5 CLONED HUMAN 3H-SCH23390 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46559 D5 CLONED HUMAN 3H-SCH23390 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46560 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46561 D5 CLONED HUMAN 3H-SCH23390 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46562 D5 CLONED HUMAN 3H-SCH23390 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46563 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46564 D5 CLONED HUMAN 3H-SCH23390 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46565 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46566 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46567 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46568 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46569 D5 CLONED HUMAN 3H-SCH23390 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46570 D5 CLONED HUMAN 3H-SCH23390 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46571 D5 CLONED HUMAN 3H-SCH23390 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46572 D5 CLONED HUMAN 3H-SCH23390 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46573 D5 CLONED HUMAN 3H-SCH23390 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46574 D5 CLONED HUMAN 3H-SCH23390 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46575 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46576 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46577 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46578 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46579 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46580 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46581 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46582 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46583 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46584 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46585 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46586 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46587 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46588 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46589 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46590 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46591 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46592 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46593 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46594 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46595 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid 6121 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46596 SLC6A3 CLONED HUMAN 3H-WIN 35,428 N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46597 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46598 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46599 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46600 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46601 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46602 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46603 SLC6A3 CLONED HUMAN 3H-WIN 35,428 (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46604 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46605 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46606 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46607 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46608 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46609 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46610 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46611 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46612 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46613 DOR FOREBRAIN GUINEA PIG 3H-DADLE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46614 DOR FOREBRAIN GUINEA PIG 3H-DADLE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025