46615 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46616 DOR FOREBRAIN GUINEA PIG 3H-DADLE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46617 DOR FOREBRAIN GUINEA PIG 3H-DADLE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46618 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46619 DOR FOREBRAIN GUINEA PIG 3H-DADLE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46620 DOR FOREBRAIN GUINEA PIG 3H-DADLE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46621 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46622 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46623 DOR FOREBRAIN GUINEA PIG 3H-DADLE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46624 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46625 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46626 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46627 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46628 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46629 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46630 DOR FOREBRAIN GUINEA PIG 3H-DADLE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46631 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46632 DOR FOREBRAIN GUINEA PIG 3H-DADLE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46633 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46634 DOR FOREBRAIN GUINEA PIG 3H-DADLE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46635 KOR FOREBRAIN RAT 3H-MUSCIMOL (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46636 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46637 KOR FOREBRAIN RAT 3H-MUSCIMOL PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46638 KOR FOREBRAIN RAT 3H-MUSCIMOL (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46639 KOR FOREBRAIN RAT 3H-MUSCIMOL (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46640 KOR FOREBRAIN RAT 3H-MUSCIMOL N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46641 KOR FOREBRAIN RAT 3H-MUSCIMOL PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46642 KOR FOREBRAIN RAT 3H-MUSCIMOL PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46643 KOR FOREBRAIN RAT 3H-MUSCIMOL (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46644 KOR FOREBRAIN RAT 3H-MUSCIMOL (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46645 KOR FOREBRAIN RAT 3H-MUSCIMOL PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46646 KOR FOREBRAIN RAT 3H-MUSCIMOL (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46647 KOR FOREBRAIN RAT 3H-MUSCIMOL (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46648 KOR FOREBRAIN RAT 3H-MUSCIMOL (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46649 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46650 KOR FOREBRAIN RAT 3H-MUSCIMOL (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46651 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46652 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46653 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46654 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46655 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46656 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46657 KOR FOREBRAIN RAT 3H-MUSCIMOL (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46658 KOR FOREBRAIN RAT 3H-MUSCIMOL (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46659 KOR FOREBRAIN RAT 3H-MUSCIMOL (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46660 KOR FOREBRAIN RAT 3H-MUSCIMOL (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46661 KOR FOREBRAIN RAT 3H-MUSCIMOL (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46662 KOR FOREBRAIN RAT 3H-MUSCIMOL (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 27, 2025
46663 H1 CLONED HUMAN 3H-PYRILAMINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46664 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46665 H1 CLONED HUMAN 3H-PYRILAMINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46666 H1 CLONED HUMAN 3H-PYRILAMINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46667 H1 CLONED HUMAN 3H-PYRILAMINE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46668 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46669 H1 CLONED HUMAN 3H-PYRILAMINE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46670 H1 CLONED HUMAN 3H-PYRILAMINE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46671 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46672 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46673 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46674 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46675 H1 CLONED HUMAN 3H-PYRILAMINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46676 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46677 H1 CLONED HUMAN 3H-PYRILAMINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46678 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46679 H1 CLONED HUMAN 3H-PYRILAMINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46680 H1 CLONED HUMAN 3H-PYRILAMINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46681 H1 CLONED HUMAN 3H-PYRILAMINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46682 H1 CLONED HUMAN 3H-PYRILAMINE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46683 H1 CLONED HUMAN 3H-PYRILAMINE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46684 H1 CLONED HUMAN 3H-PYRILAMINE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46685 H1 CLONED HUMAN 3H-PYRILAMINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46686 H1 CLONED HUMAN 3H-PYRILAMINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46687 H1 CLONED HUMAN 3H-PYRILAMINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46688 H1 CLONED HUMAN 3H-PYRILAMINE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46689 H1 CLONED HUMAN 3H-PYRILAMINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46690 H1 CLONED HUMAN 3H-PYRILAMINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46691 H1 CLONED HUMAN 3H-PYRILAMINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46692 H1 CLONED HUMAN 3H-PYRILAMINE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46693 H2 CLONED HUMAN 3H-TIOTIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46694 H2 CLONED HUMAN 3H-TIOTIDINE (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46695 H2 CLONED HUMAN 3H-TIOTIDINE PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46696 H2 CLONED HUMAN 3H-TIOTIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46697 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46698 H2 CLONED HUMAN 3H-TIOTIDINE (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46699 H2 CLONED HUMAN 3H-TIOTIDINE PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46700 H2 CLONED HUMAN 3H-TIOTIDINE PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46701 H2 CLONED HUMAN 3H-TIOTIDINE (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46702 H2 CLONED HUMAN 3H-TIOTIDINE (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 2688 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46703 H2 CLONED HUMAN 3H-TIOTIDINE (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46704 H2 CLONED HUMAN 3H-TIOTIDINE (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46705 H2 CLONED HUMAN 3H-TIOTIDINE PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46706 H2 CLONED HUMAN 3H-TIOTIDINE (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46707 H2 CLONED HUMAN 3H-TIOTIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46708 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46709 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46710 H2 CLONED HUMAN 3H-TIOTIDINE (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46711 H2 CLONED HUMAN 3H-TIOTIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46712 H2 CLONED HUMAN 3H-TIOTIDINE (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46713 H2 CLONED HUMAN 3H-TIOTIDINE (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46714 H2 CLONED HUMAN 3H-TIOTIDINE (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 4877 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46715 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46716 H2 CLONED HUMAN 3H-TIOTIDINE N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46717 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46718 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46719 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46720 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46721 H2 CLONED HUMAN 3H-TIOTIDINE (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46722 H2 CLONED HUMAN 3H-TIOTIDINE (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46723 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46724 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46725 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46726 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46727 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46728 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46729 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46730 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46731 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46732 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46733 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46734 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46735 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46736 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46737 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46738 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46739 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46740 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46741 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46742 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46743 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46744 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46745 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46746 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46747 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46748 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46749 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46750 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 4750 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46751 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46752 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46753 H4 CLONED HUMAN 3H-Histamine PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46754 H4 CLONED HUMAN 3H-Histamine (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46755 H4 CLONED HUMAN 3H-Histamine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46756 H4 CLONED HUMAN 3H-Histamine (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46757 H4 CLONED HUMAN 3H-Histamine PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46758 H4 CLONED HUMAN 3H-Histamine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46759 H4 CLONED HUMAN 3H-Histamine (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46760 H4 CLONED HUMAN 3H-Histamine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46761 H4 CLONED HUMAN 3H-Histamine PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46762 H4 CLONED HUMAN 3H-Histamine (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46763 H4 CLONED HUMAN 3H-Histamine (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46764 H4 CLONED HUMAN 3H-Histamine (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46765 H4 CLONED HUMAN 3H-Histamine (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46766 H4 CLONED HUMAN 3H-Histamine (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46767 H4 CLONED HUMAN 3H-Histamine PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46768 H4 CLONED HUMAN 3H-Histamine (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46769 H4 CLONED HUMAN 3H-Histamine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 3279 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46770 H4 CLONED HUMAN 3H-Histamine N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46771 H4 CLONED HUMAN 3H-Histamine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46772 H4 CLONED HUMAN 3H-Histamine (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46773 H4 CLONED HUMAN 3H-Histamine (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46774 H4 CLONED HUMAN 3H-Histamine (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46775 H4 CLONED HUMAN 3H-Histamine (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46776 H4 CLONED HUMAN 3H-Histamine (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46777 H4 CLONED HUMAN 3H-Histamine (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46778 H4 CLONED HUMAN 3H-Histamine (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46779 H4 CLONED HUMAN 3H-Histamine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46780 H4 CLONED HUMAN 3H-Histamine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46781 H4 CLONED HUMAN 3H-Histamine (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46782 KOR CLONED HUMAN 3H-Bremazocine (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46783 KOR CLONED HUMAN 3H-Bremazocine (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46784 KOR CLONED HUMAN 3H-Bremazocine (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46785 KOR CLONED HUMAN 3H-Bremazocine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46786 KOR CLONED HUMAN 3H-Bremazocine (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46787 KOR CLONED HUMAN 3H-Bremazocine (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46788 KOR CLONED HUMAN 3H-Bremazocine (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid 2304 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46789 KOR CLONED HUMAN 3H-Bremazocine (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46790 KOR CLONED HUMAN 3H-Bremazocine (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46791 KOR CLONED HUMAN 3H-Bremazocine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46792 KOR CLONED HUMAN 3H-Bremazocine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 827.8 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46793 KOR CLONED HUMAN 3H-Bremazocine (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46794 KOR CLONED HUMAN 3H-Bremazocine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46795 KOR CLONED HUMAN 3H-Bremazocine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46796 KOR CLONED HUMAN 3H-Bremazocine (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46797 KOR CLONED HUMAN 3H-Bremazocine (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46798 KOR CLONED HUMAN 3H-Bremazocine PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46799 KOR CLONED HUMAN 3H-Bremazocine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46800 KOR CLONED HUMAN 3H-Bremazocine (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46801 KOR CLONED HUMAN 3H-Bremazocine N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46802 KOR CLONED HUMAN 3H-Bremazocine (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone 4060 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46803 KOR CLONED HUMAN 3H-Bremazocine (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46804 KOR CLONED HUMAN 3H-Bremazocine (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46805 KOR CLONED HUMAN 3H-Bremazocine (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46806 KOR CLONED HUMAN 3H-Bremazocine (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46807 KOR CLONED HUMAN 3H-Bremazocine (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46808 KOR CLONED HUMAN 3H-Bremazocine PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46809 KOR CLONED HUMAN 3H-Bremazocine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46810 KOR CLONED HUMAN 3H-Bremazocine PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46811 KOR CLONED HUMAN 3H-Bremazocine PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46812 M2 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46813 M2 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46814 M2 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46815 M2 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46816 M2 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46817 M2 CLONED HUMAN 3H-QNB (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46818 M2 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46819 M2 CLONED HUMAN 3H-QNB (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46820 M2 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46821 M2 CLONED HUMAN 3H-QNB (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46822 M2 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46823 M2 CLONED HUMAN 3H-QNB (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46824 M2 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46825 M2 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46826 M2 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46827 M2 CLONED HUMAN 3H-QNB (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46828 M2 CLONED HUMAN 3H-QNB (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46829 M2 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46830 M2 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46831 M2 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46832 M2 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46833 M2 CLONED HUMAN 3H-QNB N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46834 M2 CLONED HUMAN 3H-QNB PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46835 M2 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46836 M2 CLONED HUMAN 3H-QNB PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46837 M2 CLONED HUMAN 3H-QNB (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46838 M2 CLONED HUMAN 3H-QNB (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46839 M2 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46840 M2 CLONED HUMAN 3H-QNB PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46841 M2 CLONED HUMAN 3H-QNB PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46842 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46843 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46844 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46845 M5 CLONED HUMAN 3H-QNB (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46846 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46847 M5 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46848 M5 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46849 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46850 M5 CLONED HUMAN 3H-QNB (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46851 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46852 M5 CLONED HUMAN 3H-QNB (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46853 M5 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46854 M5 CLONED HUMAN 3H-QNB PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46855 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46856 M5 CLONED HUMAN 3H-QNB (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46857 M5 CLONED HUMAN 3H-QNB (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46858 M5 CLONED HUMAN 3H-QNB PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46859 M5 CLONED HUMAN 3H-QNB (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46860 M5 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46861 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46862 M5 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46863 M5 CLONED HUMAN 3H-QNB N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46864 M5 CLONED HUMAN 3H-QNB PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46865 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46866 M5 CLONED HUMAN 3H-QNB (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46867 M5 CLONED HUMAN 3H-QNB (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46868 M5 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46869 M5 CLONED HUMAN 3H-QNB (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46870 M5 CLONED HUMAN 3H-QNB PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46871 M5 CLONED HUMAN 3H-QNB (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46872 mGluR5 CLONED RAT Functional (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46873 mGluR5 CLONED RAT Functional (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46874 mGluR5 CLONED RAT Functional (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46875 mGluR5 CLONED RAT Functional (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46876 mGluR5 CLONED RAT Functional (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46877 mGluR5 CLONED RAT Functional (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46878 mGluR5 CLONED RAT Functional (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46879 mGluR5 CLONED RAT Functional (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46880 mGluR5 CLONED RAT Functional (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46881 mGluR5 CLONED RAT Functional (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46882 mGluR5 CLONED RAT Functional (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46883 mGluR5 CLONED RAT Functional (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46884 mGluR5 CLONED RAT Functional (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46885 mGluR5 CLONED RAT Functional (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46886 mGluR5 CLONED RAT Functional N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46887 mGluR5 CLONED RAT Functional (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46888 mGluR5 CLONED RAT Functional (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46889 mGluR5 CLONED RAT Functional (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46890 mGluR5 CLONED RAT Functional (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46891 mGluR5 CLONED RAT Functional (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46892 mGluR5 CLONED RAT Functional (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46893 mGluR5 CLONED RAT Functional PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46894 mGluR5 CLONED RAT Functional PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46895 mGluR5 CLONED RAT Functional PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46896 mGluR5 CLONED RAT Functional (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46897 mGluR5 CLONED RAT Functional (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46898 mGluR5 CLONED RAT Functional (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46899 mGluR5 CLONED RAT Functional (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 28, 2025
46900 MOR CLONED HUMAN 3H-Diprenorphine (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46901 MOR CLONED HUMAN 3H-Diprenorphine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46902 MOR CLONED HUMAN 3H-Diprenorphine (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46903 MOR CLONED HUMAN 3H-Diprenorphine PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46904 MOR CLONED HUMAN 3H-Diprenorphine (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46905 MOR CLONED HUMAN 3H-Diprenorphine (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46906 MOR CLONED HUMAN 3H-Diprenorphine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46907 MOR CLONED HUMAN 3H-Diprenorphine (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46908 MOR CLONED HUMAN 3H-Diprenorphine (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46909 MOR CLONED HUMAN 3H-Diprenorphine (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46910 MOR CLONED HUMAN 3H-Diprenorphine (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46911 MOR CLONED HUMAN 3H-Diprenorphine (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46912 MOR CLONED HUMAN 3H-Diprenorphine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46913 MOR CLONED HUMAN 3H-Diprenorphine PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46914 MOR CLONED HUMAN 3H-Diprenorphine (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46915 MOR CLONED HUMAN 3H-Diprenorphine PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46916 MOR CLONED HUMAN 3H-Diprenorphine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46917 MOR CLONED HUMAN 3H-Diprenorphine (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46918 MOR CLONED HUMAN 3H-Diprenorphine (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46919 MOR CLONED HUMAN 3H-Diprenorphine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46920 MOR CLONED HUMAN 3H-Diprenorphine (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46921 MOR CLONED HUMAN 3H-Diprenorphine N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46922 MOR CLONED HUMAN 3H-Diprenorphine (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46923 MOR CLONED HUMAN 3H-Diprenorphine (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46924 MOR CLONED HUMAN 3H-Diprenorphine (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46925 MOR CLONED HUMAN 3H-Diprenorphine PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46926 MOR CLONED HUMAN 3H-Diprenorphine (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46927 MOR CLONED HUMAN 3H-Diprenorphine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46928 MOR CLONED HUMAN 3H-Diprenorphine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46929 MOR CLONED HUMAN 3H-Diprenorphine (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46930 NET CLONED HUMAN 3H-Nisoxetine (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46931 NET CLONED HUMAN 3H-Nisoxetine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46932 NET CLONED HUMAN 3H-Nisoxetine (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46933 NET CLONED HUMAN 3H-Nisoxetine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46934 NET CLONED HUMAN 3H-Nisoxetine (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46935 NET CLONED HUMAN 3H-Nisoxetine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46936 NET CLONED HUMAN 3H-Nisoxetine (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46937 NET CLONED HUMAN 3H-Nisoxetine N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46938 NET CLONED HUMAN 3H-Nisoxetine PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46939 NET CLONED HUMAN 3H-Nisoxetine PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46940 NET CLONED HUMAN 3H-Nisoxetine (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46941 NET CLONED HUMAN 3H-Nisoxetine PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46942 NET CLONED HUMAN 3H-Nisoxetine (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46943 NET CLONED HUMAN 3H-Nisoxetine (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46944 NET CLONED HUMAN 3H-Nisoxetine (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46945 NET CLONED HUMAN 3H-Nisoxetine PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46946 NET CLONED HUMAN 3H-Nisoxetine (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46947 NET CLONED HUMAN 3H-Nisoxetine (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46948 NET CLONED HUMAN 3H-Nisoxetine (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46949 NET CLONED HUMAN 3H-Nisoxetine (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46950 NET CLONED HUMAN 3H-Nisoxetine (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46951 NET CLONED HUMAN 3H-Nisoxetine (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46952 NET CLONED HUMAN 3H-Nisoxetine (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46953 NET CLONED HUMAN 3H-Nisoxetine (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46954 NET CLONED HUMAN 3H-Nisoxetine (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46955 NET CLONED HUMAN 3H-Nisoxetine (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46956 NET CLONED HUMAN 3H-Nisoxetine (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46957 NET CLONED HUMAN 3H-Nisoxetine (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46958 NET CLONED HUMAN 3H-Nisoxetine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46959 NET CLONED HUMAN 3H-Nisoxetine (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46960 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46961 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46962 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46963 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46964 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46965 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46966 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46967 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46968 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46969 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46970 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46971 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46972 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46973 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46974 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46975 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46976 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46977 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46978 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46979 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46980 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46981 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46982 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46983 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46984 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46985 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46986 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46987 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46988 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46989 SLC6A4 CLONED HUMAN 3H-CITALOPRAM (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46990 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46991 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46992 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46993 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46994 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46995 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46996 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46997 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46998 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
46999 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47000 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47001 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47002 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 4343 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47003 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47004 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 3956 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47005 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47006 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47007 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47008 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47009 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 557.7 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47010 Sigma 1 BRAIN RAT 3H-Pentazocine(+) N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47011 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47012 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47013 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47014 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47015 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47016 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47017 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47018 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47019 Sigma 1 BRAIN RAT 3H-Pentazocine(+) (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47020 Sigma 2 PC12 RAT 3H-DTG PL-3-025 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47021 Sigma 2 PC12 RAT 3H-DTG (3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 3386 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47022 Sigma 2 PC12 RAT 3H-DTG (3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 8594 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47023 Sigma 2 PC12 RAT 3H-DTG (3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47024 Sigma 2 PC12 RAT 3H-DTG (2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47025 Sigma 2 PC12 RAT 3H-DTG (1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47026 Sigma 2 PC12 RAT 3H-DTG (2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47027 Sigma 2 PC12 RAT 3H-DTG (2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47028 Sigma 2 PC12 RAT 3H-DTG (2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47029 Sigma 2 PC12 RAT 3H-DTG (2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47030 Sigma 2 PC12 RAT 3H-DTG (2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47031 Sigma 2 PC12 RAT 3H-DTG (3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47032 Sigma 2 PC12 RAT 3H-DTG (2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47033 Sigma 2 PC12 RAT 3H-DTG PL-3-017 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47034 Sigma 2 PC12 RAT 3H-DTG (2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47035 Sigma 2 PC12 RAT 3H-DTG (3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47036 Sigma 2 PC12 RAT 3H-DTG (2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47037 Sigma 2 PC12 RAT 3H-DTG PL-3-048-4 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47038 Sigma 2 PC12 RAT 3H-DTG (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47039 Sigma 2 PC12 RAT 3H-DTG (3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47040 Sigma 2 PC12 RAT 3H-DTG (5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47041 Sigma 2 PC12 RAT 3H-DTG (3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47042 Sigma 2 PC12 RAT 3H-DTG PL-3-016 >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47043 Sigma 2 PC12 RAT 3H-DTG N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47044 Sigma 2 PC12 RAT 3H-DTG (3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47045 Sigma 2 PC12 RAT 3H-DTG (3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47046 Sigma 2 PC12 RAT 3H-DTG (3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47047 Sigma 2 PC12 RAT 3H-DTG (3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47048 Sigma 2 PC12 RAT 3H-DTG (1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid >10000 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47049 Sigma 2 PC12 RAT 3H-DTG (3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione 3093 Dandapani S, et al., 2006 Jan 15, 2025 Jan 15, 2025
47050 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-1P 2.74 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47051 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-2P 8 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47052 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-2P 0.34 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47053 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-3P 0.68 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47054 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-4P 5.24 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47055 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-MPM 2.2 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47056 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25S)-DLAM-03I 1.52 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47057 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R,25R)-DLAM-1P 0.25 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47058 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S,25R)-DLAM-1P 0.18 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47059 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R,25S)-DLAM-1P 0.25 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47060 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-2P 0.51 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47061 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-3P 0.19 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47062 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-2P 0.19 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47063 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-3P 0.09 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47064 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-3P 0.03 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47065 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-4P 0.3 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47066 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-4P 0.09 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47067 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-4P 0.1 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47068 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-MPM 0.3 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47069 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-MPM 0.09 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47070 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-MPM 0.1 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47071 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25R)-DLAM-03I 0.14 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47072 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23S, 25R)-DLAM-03I 0.14 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47073 CLONED HUMAN 26,27-methyl-3H-1,25-D3 (23R, 25S)-DLAM-03I 0.11 Nakano Y, et al., 2006 Jan 15, 2025 Jan 15, 2025
47074 H3 CORTEX RAT 125I-IPP Iodophenpropit 0.97 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47075 H1 CLONED GUINEA PIG 3H-MEPYRAMINE Iodophenpropit 1710 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47076 H1 CLONED GUINEA PIG 3H-MEPYRAMINE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47077 H2 CLONED GUINEA PIG 125I-aminopotentidine Iodophenpropit 2280 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47078 H2 CLONED GUINEA PIG 125I-aminopotentidine Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47079 H3 CORTEX RAT 125I-IPP Thioperamide 4.3 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47080 WHOLE BRAIN RAT 3H-PRAZOSIN Iodophenpropit 1500 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47081 WHOLE BRAIN RAT 3H-PRAZOSIN Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47082 WHOLE BRAIN MINUS CEREBELLUM RAT 3H-CLONIDINE Iodophenpropit 120 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47083 WHOLE BRAIN MINUS CEREBELLUM RAT 3H-CLONIDINE Thioperamide 4000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47084 Beta2 CORTEX RAT 3H-DHA Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47085 Beta2 CORTEX RAT 3H-DHA Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47086 LIVER RAT 3H-IDAZOXAN Iodophenpropit 530 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47087 LIVER RAT 3H-IDAZOXAN Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47088 D1 CAUDATE NUCLEUS RAT 3H-dopamine Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47089 D1 CAUDATE NUCLEUS RAT 3H-dopamine Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47090 D2 Corpus Striatum RAT 3H-SPIPERONE Iodophenpropit 4500 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47091 D2 Corpus Striatum RAT 3H-SPIPERONE Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47092 D3 S. Nigra RAT 3H-SPIPERONE Iodophenpropit 1800 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47093 D3 S. Nigra RAT 3H-SPIPERONE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47094 5-HT1A FR. CORTEX RAT 3H-8-OH-DPAT Iodophenpropit 2300 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47095 5-HT1A FR. CORTEX RAT 3H-8-OH-DPAT Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47096 5-HT1B FR. CORTEX RAT 3H-5HT Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47097 5-HT1B FR. CORTEX RAT 3H-5HT Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47098 5-HT1D CAUDATE NUCLEUS RAT 3H-5HT Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47099 5-HT1D CAUDATE NUCLEUS RAT 3H-5HT Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47100 5-HT2A FR. CORTEX RAT 3H-SPIPERONE Iodophenpropit 1900 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47101 5-HT2A FR. CORTEX RAT 3H-SPIPERONE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47102 5-HT2C FR. CORTEX RAT 3H-SPIPERONE Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47103 5-HT2C FR. CORTEX RAT 3H-SPIPERONE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47104 5-HT3 ILEUM GUINEA PIG 3H-GR-65630 Iodophenpropit 11 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47105 5-HT3 ILEUM GUINEA PIG 3H-GR-65630 Thioperamide 120 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47106 5-HT4 BRAIN GUINEA PIG 3H-GR-113808 Iodophenpropit 530 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47107 5-HT4 BRAIN GUINEA PIG 3H-GR-113808 Thioperamide 2800 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47108 SLC6A4 BRAIN GUINEA PIG 3H-PAROXETINE Iodophenpropit 1250 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47109 SLC6A4 BRAIN GUINEA PIG 3H-PAROXETINE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47110 M1 CORTEX RAT 3H-PIRENZEPINE Iodophenpropit 1500 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47111 M1 CORTEX RAT 3H-PIRENZEPINE Thioperamide 4600 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47112 M2 HEART RAT 3H-NMS Iodophenpropit 1980 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47113 M2 HEART RAT 3H-NMS Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47114 M3 CLONED HUMAN 3H-NMS Iodophenpropit 3700 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47115 M3 CLONED HUMAN 3H-NMS Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47116 FR. CORTEX RAT 3H-5HT Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47117 FR. CORTEX RAT 3H-5HT Thioperamide 6400 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47118 DOR WHOLE BRAIN MINUS CEREBELLUM RAT 3H-DADLE Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47119 DOR WHOLE BRAIN MINUS CEREBELLUM RAT 3H-DADLE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47120 KOR WHOLE BRAIN MINUS CEREBELLUM RAT 3H-EKC Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47121 KOR WHOLE BRAIN MINUS CEREBELLUM RAT 3H-EKC Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47122 MOR WHOLE BRAIN MINUS CEREBELLUM RAT 3H-NALOXONE Iodophenpropit 8400 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47123 MOR WHOLE BRAIN MINUS CEREBELLUM RAT 3H-NALOXONE Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47124 WHOLE BRAIN RAT 3H-3-PPP,(+) Iodophenpropit 170 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47125 WHOLE BRAIN RAT 3H-3-PPP,(+) Thioperamide 180 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47126 GABAA CEREBELLUM RAT 3H-DIAZEPAM Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47127 GABAA CEREBELLUM RAT 3H-DIAZEPAM Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47128 CORTEX RAT 3H-CCK8 Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47129 CORTEX RAT 3H-CCK8 Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47130 PANCREAS RAT 3H-CCK8 Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47131 PANCREAS RAT 3H-CCK8 Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47132 CLONED HUMAN 3H-SUBSTANCE P Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47133 CLONED HUMAN 3H-SUBSTANCE P Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47134 BRAIN Chick 125I-Iodomelatonin Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47135 BRAIN Chick 125I-Iodomelatonin Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47136 NMDA BRAIN RAT 3H-CGS-19755 Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47137 NMDA BRAIN RAT 3H-CGS-19755 Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47138 KOR CEREBELLUM RAT 3H-MUSCIMOL Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47139 KOR CEREBELLUM RAT 3H-MUSCIMOL Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47140 GlyR medulla, pons RAT 3H-Strychnine Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47141 GlyR medulla, pons RAT 3H-Strychnine Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47142 GlyR BRAIN RAT 3H-5,7-DCKA Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47143 GlyR BRAIN RAT 3H-5,7-DCKA Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47144 Total Cortex RAT 3H-Batrachotoxin Iodophenpropit 1000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47145 Total Cortex RAT 3H-Batrachotoxin Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47146 BRAIN RAT 3H-Nitrendipine Iodophenpropit >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47147 BRAIN RAT 3H-Nitrendipine Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 15, 2025
47148 Calcium channel BRAIN RAT 3H-D-888 Iodophenpropit 400 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47149 Calcium channel BRAIN RAT 3H-D-888 Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47150 Calcium channel HEART RAT 3H-D-888 Iodophenpropit 560 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47151 Calcium channel HEART RAT 3H-D-888 Thioperamide >10000 Leurs R. et. al. 1995 Jan 15, 2025 Jan 27, 2025
47152 H1 CLONED HUMAN 3H-MEPYRAMINE HISTAMINE >10000 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47153 H1 CLONED HUMAN 3H-MEPYRAMINE 5-APT 3090 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47154 H1 CLONED HUMAN 3H-MEPYRAMINE CF3-5-APT 6270 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47155 H1 CLONED HUMAN 3H-MEPYRAMINE OCH3-5-APT 3200 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47156 H1 CLONED HUMAN 3H-MEPYRAMINE CL-5-APT 2650 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47157 H1 CLONED HUMAN 3H-MEPYRAMINE 6-APT 9570 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47158 H1 CLONED HUMAN 3H-MEPYRAMINE CF3-6-APT 2740 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47159 H1 CLONED HUMAN 3H-MEPYRAMINE OCH3-6-APT 1220 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47160 H1 CLONED HUMAN 3H-MEPYRAMINE CL-6-APT 1310 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47161 H1 CLONED HUMAN 3H-MEPYRAMINE Br-6-APT 130 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47162 5-HT2A CLONED HUMAN 3H-KETANSERIN 5-APT 800 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47163 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-APT 310 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47164 5-HT2A CLONED HUMAN 3H-KETANSERIN 6-APT 1200 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47165 5-HT2C CLONED HUMAN 3H-MESULERGINE 6-APT 1500 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47166 5-HT2A CLONED HUMAN 3H-KETANSERIN CL-6-APT 1200 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47167 5-HT2C CLONED HUMAN 3H-MESULERGINE CL-6-APT 4600 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47168 5-HT2A CLONED HUMAN 3H-KETANSERIN Br-6-APT 580 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47169 5-HT2C CLONED HUMAN 3H-MESULERGINE Br-6-APT 540 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47170 H1 CLONED HUMAN 3H-MEPYRAMINE 2-(Dimethylamino)tetralin 165 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47171 H1 CLONED HUMAN 3H-MEPYRAMINE Diphenhydramine 9.57 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47172 H1 CLONED HUMAN 3H-MEPYRAMINE BUTACLAMOL,(+) 147 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47173 H1 CLONED HUMAN 3H-MEPYRAMINE (R)-Chlopheniramine 80 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47174 H1 CLONED HUMAN 3H-MEPYRAMINE l-Chlorpheniramine 0.31 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47175 H1 CLONED HUMAN 3H-MEPYRAMINE Triprolidine 0.69 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47176 H1 CLONED HUMAN 3H-MEPYRAMINE ATR 1240 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47177 H1 CLONED HUMAN 3H-MEPYRAMINE (-)-NANM 5000 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47178 H1 CLONED HUMAN 3H-MEPYRAMINE DOXEPIN 0.16 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47179 H1 CLONED HUMAN 3H-MEPYRAMINE FLUPENTHIXOL, Alpha 0.86 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47180 H1 CLONED HUMAN 3H-MEPYRAMINE Flupenthixol, Beta 5.73 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47181 H1 CLONED HUMAN 3H-MEPYRAMINE SCH 23390 101 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47182 H1 CLONED HUMAN 3H-MEPYRAMINE METHYSERGIDE 3000 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47183 H1 CLONED HUMAN 3H-MEPYRAMINE MAZINDOL 600 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47184 H1 CLONED HUMAN 3H-MEPYRAMINE SKF 38393 2500 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47185 H1 CLONED HUMAN 3H-MEPYRAMINE AMITRIPTYLINE 0.5 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47186 H1 CLONED HUMAN 3H-MEPYRAMINE DESIPRAMINE 45.4 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47187 H1 CLONED HUMAN 3H-MEPYRAMINE 7-OH-DPAT 1500 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47188 H1 CLONED HUMAN 3H-MEPYRAMINE HALOPERIDOL 215 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47189 H1 CLONED HUMAN 3H-MEPYRAMINE Loperamide 2000 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47190 H1 CLONED HUMAN 3H-MEPYRAMINE MIANSERIN 0.3 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47191 H1 CLONED HUMAN 3H-MEPYRAMINE RIMCAZOLE 5000 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47192 H1 CLONED HUMAN 3H-MEPYRAMINE SPIPERONE 272 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47193 H1 CLONED HUMAN 3H-MEPYRAMINE KETANSERIN 1.79 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47194 H1 CLONED HUMAN 3H-MEPYRAMINE PROMETHAZINE 0.24 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47195 H1 CLONED HUMAN 3H-MEPYRAMINE MEPYRAMINE 0.74 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47196 H1 CLONED HUMAN 3H-MEPYRAMINE GBR-12909 9.33 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47197 H1 CLONED HUMAN 3H-MEPYRAMINE NORTRYPTYLINE 15.1 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47198 H1 CLONED HUMAN 3H-MEPYRAMINE (+/-)-BMY-1402 180 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47199 H1 CLONED HUMAN 3H-MEPYRAMINE 3-Aminofluoranthene 4800 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47200 H1 CLONED HUMAN 3H-MEPYRAMINE 3-(Dimethylamino)fluoranthene 4800 Ghoneim OM, et al., 2006 Jan 15, 2025 Jan 15, 2025
47201 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-methylthiourea >10000 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47202 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-butylthiourea 4650 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47203 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-tert-butylthiourea >10000 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47204 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-isopropylthiourea >10000 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47205 CLONED HUMAN Functional 1-(Bicyclo[2.2.1]hept-5-en-2-yl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea 3660 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47206 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-cyclohexylthiourea 4700 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47207 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-benzylthiourea 5670 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47208 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-phenylthiourea 4480 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47209 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-naphthalen-1-ylthiourea 2790 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47210 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methylphenyl)thiourea 2140 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47211 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-ethylphenyl)thiourea 2780 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47212 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-fluorophenyl)thiourea 4730 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47213 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(dimethylamino)phenyl)thiourea 2030 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47214 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-nitrophenyl)thiourea 2680 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47215 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-acetylphenyl)thiourea 1790 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47216 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)-propyl)-3-(4-methylsulfanyl-phenyl)-thiourea 1660 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47217 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(benzyloxy)phenyl)thiourea 970 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47218 CLONED HUMAN Functional 1-(4-Ethoxy-phenyl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea 890 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47219 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methoxyphenyl)thiourea 700 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47220 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(benzo[d][1,3]dioxol-6-yl)thiourea 5660 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47221 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3-methoxyphenyl)thiourea 1860 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47222 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxybenzyl)thiourea 1550 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47223 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,3-dihydrobenzo[b][1,4]dioxin-7-yl)thiourea 1120 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47224 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,5-dimethoxyphenyl)thiourea 750 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47225 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,4-dimethoxyphenyl)thiourea 560 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47226 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)urea 490 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47227 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4,5-trimethoxyphenyl)thiourea 340 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47228 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)thiourea 60 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47229 CLONED HUMAN Functional 1-(2-(1H-Imidazol-1-yl)ethyl)-3-(3,4-dimethoxyphenyl)thiourea >10000 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47230 CLONED HUMAN Functional 1-(4-(1H-Imidazol-1-yl)butyl)-3-(3,4-dimethoxyphenyl)thiourea 550 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47231 CLONED HUMAN Functional 1-((R)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea 340 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47232 CLONED HUMAN Functional 1-((S)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea 760 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47233 CLONED HUMAN Functional 1-((1-((1H-Imidazol-1-yl)methyl)cyclopropyl)methyl)-3-(3,4-dimethoxyphenyl)thiourea 2330 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47234 CLONED HUMAN Functional 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)-1-methylthiourea 4830 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47235 CLONED HUMAN Functional N-(3-(1H-imidazol-1-yl)propyl)benzo[d]thiazol-2-amine 3730 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47236 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-6-chlorobenzo[d]thiazol-2-amine 3350 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47237 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-6-methoxybenzo[d]thiazol-2-amine 1570 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47238 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-5,6-dimethoxybenzo[d]thiazol-2-amine 2000 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47239 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-2-(3,4-dimethoxyphenyl)ethanethioamide 390 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47240 CLONED HUMAN Functional (R)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide 7340 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47241 CLONED HUMAN Functional (S)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide 3510 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47242 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-2,2-diphenylethanethioamide 4480 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47243 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-methoxyphenyl)cyclopropanecarbothioamide 400 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47244 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-chlorophenyl)cyclobutanecarbothioamide 4880 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47245 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-chlorophenyl)cyclopentanecarbothioamide 7330 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47246 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-1-(4-methoxyphenyl)cyclohexanecarbothioamide 2220 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47247 CLONED HUMAN Functional N-(3-(1H-Imidazol-1-yl)propyl)-1-(3,4-dimethoxyphenyl)cyclopropanecarbothioamide 90 Buchholz M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47248 CLONED HUMAN Functional Motilin 0.15 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
47249 CLONED HUMAN 125I-Motilin Motilin 3.1 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
47250 CLONED HUMAN Functional ABT-229 4.2 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
47251 CLONED HUMAN 125I-Motilin ABT-229 3.4 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
47252 CLONED HUMAN Functional erythromycin-A 400 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
47253 CLONED HUMAN 125I-Motilin erythromycin-A >10000 Li JJ, et al., 2004 Jan 15, 2025 Jan 15, 2025
47254 duodenum RABBIT 125I-Motilin SK-896 3.5 Tsukamoto K, et al., 2000 Jan 15, 2025 Jan 15, 2025
47255 duodenum RABBIT 125I-Motilin Motilin 3.1 Tsukamoto K, et al., 2000 Jan 15, 2025 Jan 15, 2025
47256 duodenum HUMAN 125I-Motilin [Leu13]motilin 3.6 Tsukamoto K, et al., 2000 Jan 15, 2025 Jan 15, 2025
47257 duodenum RABBIT 125I-Motilin [Leu13]motilin 1.1 Tsukamoto K, et al., 2000 Jan 15, 2025 Jan 15, 2025
47258 duodenum RABBIT 125I-Motilin SK-896 3.4 Tsukamoto K, et al., 2000 Jan 15, 2025 Jan 15, 2025
47259 duodenum HUMAN 125I-Motilin Motilin 3.4 Tsukamoto K, et al., 2000 Jan 15, 2025 Jan 15, 2025
47260 Beta1 CEREBRAL CORTEX RAT 125I-ICYP Arotinolol 0.18197 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47261 Beta1 CEREBRAL CORTEX RAT 125I-ICYP PINDOLOL,(+/-) 0.660693 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47262 Beta1 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, l- 0.691831 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47263 Beta1 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, dl 2.81838 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47264 Beta1 CEREBRAL CORTEX RAT 125I-ICYP ALPRENOLOL 4.16869 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47265 Beta1 CEREBRAL CORTEX RAT 125I-ICYP YM-09538 4.36516 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47266 Beta1 CEREBRAL CORTEX RAT 125I-ICYP OXPRENOLOL 7.76247 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47267 Beta1 CEREBRAL CORTEX RAT 125I-ICYP LABETALOL 12.0226 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47268 Beta1 CEREBRAL CORTEX RAT 125I-ICYP BETAXOLOL 12.3027 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47269 Beta1 CEREBRAL CORTEX RAT 125I-ICYP l-Metoprolol 13.8038 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47270 Beta1 CEREBRAL CORTEX RAT 125I-ICYP metoprolol 63.0957 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47271 Beta1 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, d 81.2831 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47272 Beta1 CEREBRAL CORTEX RAT 125I-ICYP ATENOLOL 97.7237 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47273 Beta1 CEREBRAL CORTEX RAT 125I-ICYP acebutolol 125.893 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47274 Beta1 CEREBRAL CORTEX RAT 125I-ICYP ICI 118,551 194.984 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47275 Beta1 CEREBRAL CORTEX RAT 125I-ICYP PRACTOLOL 245.471 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47276 Beta1 CEREBRAL CORTEX RAT 125I-ICYP Sotalol 2238.72 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47277 Beta1 CEREBRAL CORTEX RAT 125I-ICYP Butoxamine 3715.35 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47278 Beta1 CEREBRAL CORTEX RAT 125I-ICYP d-Metoprolol >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47279 Beta2 CEREBRAL CORTEX RAT 125I-ICYP Arotinolol 0.549541 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47280 Beta2 CEREBRAL CORTEX RAT 125I-ICYP PINDOLOL,(+/-) 0.316228 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47281 Beta2 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, l- 0.457088 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47282 Beta2 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, dl 2.45471 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47283 Beta2 CEREBRAL CORTEX RAT 125I-ICYP ALPRENOLOL 0.57544 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47284 Beta2 CEREBRAL CORTEX RAT 125I-ICYP YM-09538 13.1826 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47285 Beta2 CEREBRAL CORTEX RAT 125I-ICYP LABETALOL 67.6083 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47286 Beta2 CEREBRAL CORTEX RAT 125I-ICYP BETAXOLOL 2041.74 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47287 Beta2 CEREBRAL CORTEX RAT 125I-ICYP l-Metoprolol 2454.71 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47288 Beta2 CEREBRAL CORTEX RAT 125I-ICYP metoprolol 1698.24 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47289 Beta2 CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, d 43.6516 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47290 Beta2 CEREBRAL CORTEX RAT 125I-ICYP ATENOLOL 2818.38 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47291 Beta2 CEREBRAL CORTEX RAT 125I-ICYP acebutolol 7079.46 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47292 Beta2 CEREBRAL CORTEX RAT 125I-ICYP ICI 118,551 1.77828 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47293 Beta2 CEREBRAL CORTEX RAT 125I-ICYP PRACTOLOL >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47294 Beta2 CEREBRAL CORTEX RAT 125I-ICYP Sotalol 338.844 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47295 Beta2 CEREBRAL CORTEX RAT 125I-ICYP Butoxamine 467.735 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47296 Beta2 CEREBRAL CORTEX RAT 125I-ICYP d-Metoprolol >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47297 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP Arotinolol 10.7152 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47298 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, dl 56.2341 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47299 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP PINDOLOL,(+/-) 58.8844 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47300 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP ALPRENOLOL 70.7946 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47301 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, l- 77.6247 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47302 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP OXPRENOLOL 173.78 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47303 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP YM-09538 1288.25 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47304 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP LABETALOL 1995.26 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47305 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP ICI 118,551 3890.45 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47306 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP acebutolol 4168.69 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47307 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP PROPRANOLOL, d 7079.46 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47308 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP BETAXOLOL >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47309 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP metoprolol >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47310 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP l-Metoprolol >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47311 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP PRACTOLOL >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47312 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP Sotalol >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47313 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP Butoxamine >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47314 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP d-Metoprolol >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47315 Beta2 CEREBRAL CORTEX RAT 125I-ICYP OXPRENOLOL 9.77237 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 28, 2025
47316 5-HT1B CEREBRAL CORTEX RAT 125I-ICYP ATENOLOL >10000 Tsuchihashi H, et al., 1990 Jan 15, 2025 Jan 15, 2025
47317 5-HT1A CLONED HUMAN 3H-8-OH-DPAT WAY 100,635 2.2 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47318 5-HT1B CLONED HUMAN 3H-GR-125743 WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47319 5-HT1D CLONED HUMAN 3H-GR-125743 WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47320 5-HT1E CLONED HUMAN 3H-5HT WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47321 5-HT2A CLONED HUMAN 3H-KETANSERIN WAY 100,635 6260 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47322 5-HT2C CLONED RAT 3H-MESULERGINE WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47323 CB1 CLONED HUMAN 3H-LSD WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 27, 2025
47324 5-HT6 CLONED HUMAN 3H-LSD WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47325 5-HT7 CLONED HUMAN 3H-LSD WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47326 5-HT2B CLONED HUMAN 3H-LSD WAY 100,635 24 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47327 H1 CLONED HUMAN 3H-PYRILAMINE WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47328 H2 CLONED HUMAN 3H-TIOTIDINE WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47329 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47330 H4 CLONED HUMAN 3H-Histamine WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47331 D1 CLONED HUMAN 3H-SCH23390 WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47332 D2 CLONED HUMAN 3H-NMSP WAY 100,635 940 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47333 D3 CLONED RAT 3H-NMSP WAY 100,635 370 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47334 D4 CLONED HUMAN 3H-NMSP WAY 100,635 16.4 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47335 D5 CLONED HUMAN 3H-SCH23390 WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47336 Alpha1A CLONED HUMAN 3H-PRAZOSIN WAY 100,635 19.9 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47337 Alpha1B CLONED HUMAN 3H-PRAZOSIN WAY 100,635 322 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47338 Alpha2A CLONED HUMAN 3H-CLONIDINE WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47339 Alpha2B CLONED HUMAN 3H-CLONIDINE WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47340 Alpha2C CLONED HUMAN 3H-CLONIDINE WAY 100,635 2573 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47341 Beta1 CLONED RAT 125I-Pindolol WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47342 Beta2 CLONED RAT 125I-Pindolol WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 28, 2025
47343 MOR CLONED HUMAN 3H-QNB WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47344 M2 CLONED HUMAN 3H-QNB WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47345 DOR CLONED HUMAN 3H-QNB WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47346 KOR CLONED HUMAN 3H-QNB WAY 100,635 412 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47347 M5 CLONED HUMAN 3H-QNB WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 15, 2025
47348 KOR FOREBRAIN RAT 3H-MUSCIMOL WAY 100,635 >10000 Chemel BR, et.al., 2006 Jan 15, 2025 Jan 27, 2025
47349 GRIA1 CLONED HUMAN 3H-AMPA LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47350 GRIA1 CLONED HUMAN 3H-AMPA LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47351 GRIA1 CLONED HUMAN 3H-AMPA LY 293558 9200 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47352 GRIA2 CLONED HUMAN 3H-AMPA LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47353 GRIA2 CLONED HUMAN 3H-AMPA LY 457691 5500 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47354 GRIA2 CLONED HUMAN 3H-AMPA LY 458545 8300 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47355 GRIA2 CLONED HUMAN 3H-AMPA LY 294486 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47356 GRIA2 CLONED HUMAN 3H-AMPA LY 302679 820 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47357 GRIA2 CLONED HUMAN 3H-AMPA LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47358 GRIA2 CLONED HUMAN 3H-AMPA LY 293558 3200 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47359 GRIA2 CLONED HUMAN 3H-AMPA LY 467711 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47360 GRIA2 CLONED HUMAN 3H-AMPA LY 525327 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47361 CLONED HUMAN 3H-AMPA LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47362 CLONED HUMAN 3H-AMPA LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47363 CLONED HUMAN 3H-AMPA LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47364 GRIA4 CLONED HUMAN 3H-AMPA LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47365 GRIA4 CLONED HUMAN 3H-AMPA LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47366 GRIA4 CLONED HUMAN 3H-AMPA LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47367 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 466195 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
47368 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
47369 Kainate receptor CLONED HUMAN 3H-Kainic acid LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 28, 2025
47370 Grik5 CLONED HUMAN 3H-Kainic acid LY 466195 50 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47371 Grik5 CLONED HUMAN 3H-Kainic acid LY 457691 1550 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47372 Grik5 CLONED HUMAN 3H-Kainic acid LY 458545 1690 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47373 Grik5 CLONED HUMAN 3H-Kainic acid LY 294486 3060 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47374 Grik5 CLONED HUMAN 3H-Kainic acid LY 302679 3410 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47375 Grik5 CLONED HUMAN 3H-Kainic acid LY 382884 4000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47376 Grik5 CLONED HUMAN 3H-Kainic acid LY 293558 4200 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47377 Grik5 CLONED HUMAN 3H-Kainic acid LY 467711 7400 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47378 Grik5 CLONED HUMAN 3H-Kainic acid LY 525327 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47379 CLONED HUMAN 3H-Kainic acid LY 466195 8900 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47380 CLONED HUMAN 3H-Kainic acid LY 382884 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47381 CLONED HUMAN 3H-Kainic acid LY 293558 >10000 Weiss B, et. al., 2006 Jan 15, 2025 Jan 15, 2025
47382 5-HT2B CLONED HUMAN 3H-5HT Ziprasidone 27.23 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
47383 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-Benzylpiperidin-4-yl)-1-naphthamide 162 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47384 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-Benzylpiperidin-4-yl)-1-naphthamide 1000 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47385 D2 CLONED HUMAN 3H-SPIPERONE N-(1-Benzylpiperidin-4-yl)-1-naphthamide 1000 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47386 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-Benzylpiperidin-4-yl)-2-naphthamide 11 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47387 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-Benzylpiperidin-4-yl)-2-naphthamide 44 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47388 D2 CLONED HUMAN 3H-SPIPERONE N-(1-Benzylpiperidin-4-yl)-2-naphthamide 1000 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47389 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-Phenylethylpiperidin-4-yl)-2-naphthamide 139 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47390 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-Phenylethylpiperidin-4-yl)-2-naphthamide 42 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47391 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide 29 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47392 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide 110 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47393 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Phenylpropyl)piperidin-4-yl)-2-naphthamide 63 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47394 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Phenylpropyl)piperidin-4-yl)-2-naphthamide 50 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47395 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Phenylbutyl)piperidin-4-yl)-2-naphthamide 281 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47396 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Phenylbutyl)piperidin-4-yl)-2-naphthamide 213 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47397 D4 CLONED HUMAN 3H-NEMONAPRIDE (4-(Benzylamino)piperidin-1-yl)-(naphthalen-2-yl)methadone 167 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47398 D4 CLONED HUMAN 3H-NEMONAPRIDE Naphthalen-2-yl(4-(Phenylamino)piperidin-1-yl)methadone 210 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47399 D4 CLONED HUMAN 3H-NEMONAPRIDE Naphthalen-2-yl(4-(3-Phenylpropylamino)piperidin-1-yl)methadone 222 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47400 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(2-Phenylethylpiperidin-4-yl)-1-naphthamide 230 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47401 5-HT2A CLONED RAT 3H-KETANSERIN N-(2-Phenylethylpiperidin-4-yl)-1-naphthamide 543 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47402 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-Phenylethylpiperidin-4-yl)-1-naphthamide 248 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47403 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(3-Phenylpropylpiperidin-4-yl)-1-naphthamide 71 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47404 5-HT2A CLONED RAT 3H-KETANSERIN N-(3-Phenylpropylpiperidin-4-yl)-1-naphthamide 228 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47405 5-HT2A CLONED RAT 3H-KETANSERIN N-((S)-3-(1-hydroxy-1-phenyl)propylpiperidin-4-yl)-1-naphthamide 390 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47406 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(4-Phenylbutylpiperidin-4-yl)-1-naphthamide 362 Carato P, et al., 2007 Jan 15, 2025 Jan 27, 2025
47407 5-HT2A CLONED RAT 3H-KETANSERIN N-(4-Phenylbutylpiperidin-4-yl)-1-naphthamide 487 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47408 5-HT2A CLONED RAT 3H-KETANSERIN N-(2-Phenylethylpiperidin-4-yl)-1-naphthamide 211 Carato P, et al., 2007 Jan 15, 2025 Jan 15, 2025
47409 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(2-Cl-benzyl)-piperidin-4-yl)-1-naphthamide 329 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47410 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Cl-benzyl)-piperidin-4-yl)-1-naphthamide 116 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47411 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-Cl-benzyl)-piperidin-4-yl)-1-naphthamide 43 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47412 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Br-benzyl)-piperidin-4-yl)-1-naphthamide 66 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47413 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Br-benzyl)-piperidin-4-yl)-1-naphthamide 462 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47414 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-Br-benzyl)-piperidin-4-yl)-1-naphthamide 44 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47415 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-CF3-benzyl)-piperidin-4-yl)-1-naphthamide 119 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47416 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-CF3-benzyl)-piperidin-4-yl)-1-naphthamide 96 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47417 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(2,3,4,5,6-F-benzyl)-piperidin-4-yl)-1-naphthamide 228 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47418 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-MeO-benzyl)-piperidin-4-yl)-1-naphthamide 168 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47419 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-MeO-benzyl)-piperidin-4-yl)-1-naphthamide 223 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47420 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(2-Me-benzyl)-piperidin-4-yl)-1-naphthamide 155 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47421 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Me-benzyl)-piperidin-4-yl)-1-naphthamide 77 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47422 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-Me-benzyl)-piperidin-4-yl)-1-naphthamide 69 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47423 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(2-Cl-benzyl)-piperidin-4-yl)-2-naphthamide 133 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47424 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Cl-benzyl)-piperidin-4-yl)-2-naphthamide 133 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47425 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Cl-benzyl)-piperidin-4-yl)-2-naphthamide 54 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47426 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-Cl-benzyl)-piperidin-4-yl)-2-naphthamide 37 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47427 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(4-Cl-benzyl)-piperidin-4-yl)-2-naphthamide 242 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47428 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Br-benzyl)-piperidin-4-yl)-2-naphthamide 36 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47429 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Br-benzyl)-piperidin-4-yl)-2-naphthamide 53 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47430 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-Br-benzyl)-piperidin-4-yl)-2-naphthamide 34 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47431 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(4-Br-benzyl)-piperidin-4-yl)-2-naphthamide 223 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47432 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-CF3-benzyl)-piperidin-4-yl)-2-naphthamide 103 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47433 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-CF3-benzyl)-piperidin-4-yl)-2-naphthamide 84 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47434 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-NO2-benzyl)-piperidin-4-yl)-2-naphthamide 181 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47435 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(4-NO2-benzyl)-piperidin-4-yl)-2-naphthamide 278 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47436 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-MeO-benzyl)-piperidin-4-yl)-2-naphthamide 16 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47437 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-MeO-benzyl)-piperidin-4-yl)-2-naphthamide 158 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47438 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-MeO-benzyl)-piperidin-4-yl)-2-naphthamide 31 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47439 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(4-MeO-benzyl)-piperidin-4-yl)-2-naphthamide 151 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47440 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(2-(2-Me-benzyl)-piperidin-4-yl)-2-naphthamide 26 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47441 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(2-Me-benzyl)-piperidin-4-yl)-2-naphthamide 175 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47442 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Me-benzyl)-piperidin-4-yl)-2-naphthamide 11 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47443 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Me-benzyl)-piperidin-4-yl)-2-naphthamide 87 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47444 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(4-Me-benzyl)-piperidin-4-yl)-2-naphthamide 21 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47445 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(4-Me-benzyl)-piperidin-4-yl)-2-naphthamide 222 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47446 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(2-Pyridyl)-piperidin-4-yl)-2-naphthamide 299 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47447 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(2-Pyridyl)-piperidin-4-yl)-2-naphthamide 545 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47448 D4 CLONED HUMAN 3H-NEMONAPRIDE N-(1-(3-Pyridyl)-piperidin-4-yl)-2-naphthamide 326 Carato P, et al., 2007a Jan 15, 2025 Jan 27, 2025
47449 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(3-Pyridyl)-piperidin-4-yl)-2-naphthamide 524 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47450 5-HT2A CLONED RAT 3H-KETANSERIN N-(1-(4-Pyridyl)-piperidin-4-yl)-2-naphthamide 695 Carato P, et al., 2007a Jan 15, 2025 Jan 15, 2025
47451 CLONED HUMAN Functional 5-(4-Aminophenyl)-6-methylthieno[2,3-d]pyrimidin-4-amine 4600 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47452 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-3-methylbenzamide 4600 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47453 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]benzenesulfonamide >10000 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47454 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-phenylurea 36 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47455 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea 6 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47456 CLONED HUMAN Functional 4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-N-phenylbenzamide >10000 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47457 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)thiourea 2800 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47458 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N' '-cyano-N'-(3-methylphenyl)guanidine 1100 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47459 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-1H-indole-2-carboxamide >10000 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47460 CLONED HUMAN Functional 5-[4-(1,3-Benzoxazol-2-ylamino)phenyl]-6-methylthieno[2,3-d]pyrimidin-4-amine 170 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47461 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-2-(3-methylphenyl)acetamide 760 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47462 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N-methyl-N'-(3-methylphenyl)urea 55 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47463 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-methyl-N'-(3-methylphenyl)urea 1900 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47464 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-benzylurea 330 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47465 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-cyclohexylmethylurea 790 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47466 CLONED HUMAN Functional N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea 26 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47467 CLONED HUMAN Functional N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-cyclohexylurea 170 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47468 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea 3 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47469 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-butylurea 180 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47470 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-isobutylurea 1700 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47471 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-methylphenyl)urea 260 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47472 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-methylphenyl)urea 53 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47473 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-methoxyphenyl)urea 110 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47474 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methoxyphenyl)urea 34 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47475 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-methoxyphenyl)urea 69 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47476 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-fluorophenyl)urea 110 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47477 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-fluorophenyl)urea 54 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47478 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-fluorophenyl)urea 52 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47479 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-chlorophenyl)urea 340 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47480 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-chlorophenyl)urea 35 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47481 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-chlorophenyl)urea 96 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47482 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-bromophenyl)urea 46 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47483 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-bromophenyl)urea 120 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47484 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea 52 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47485 CLONED HUMAN Functional Methyl 3-[({[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]amino}carbonyl)amino]benzoate 290 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47486 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3,5-dimethylphenyl)urea 12 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47487 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3,5-dichlorophenyl)urea 160 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47488 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[2-fluoro-5-(trifluoromethyl)phenyl]urea 45 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47489 CLONED HUMAN Functional 3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}propanamide 17 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47490 CLONED HUMAN Functional 3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N-methylpropanamide 330 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47491 CLONED HUMAN Functional 3-{4-Amino-5-[4-(3-m-tolylureido)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N,N-dimethylpropionamide 210 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47492 CLONED HUMAN Functional N-{4-[4-Amino-6-(morpholin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea 210 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47493 CLONED HUMAN Functional N-(4-{4-Amino-6-[(4-methylpiperazin-1-yl)methyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea 590 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47494 CLONED HUMAN Functional N-(4-{4-Amino-6-[(dimethylamino)methyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea 180 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47495 CLONED HUMAN Functional N-[4-(4-Amino-6-propylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea 26 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47496 CLONED HUMAN Functional N-[4-(4-Amino-6-isopropylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea 130 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47497 CLONED HUMAN Functional N-[4-(4-Amino-6-benzylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea 280 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47498 CLONED HUMAN Functional N-{4-[4-Amino-6-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea 34 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47499 CLONED HUMAN Functional N-{4-[4-Amino-6-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea 53 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47500 CLONED HUMAN Functional N-{4-[4-Amino-6-(2-hydroxyethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea 19 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47501 CLONED HUMAN Functional N-{4-[4-Amino-6-(2-methoxyethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea 64 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47502 CLONED HUMAN Functional N-{4-[4-Amino-6-(3-hydroxypropyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea 15 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47503 CLONED HUMAN Functional N-(4-{4-Amino-6-[2-(dimethylamino)ethyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea 230 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47504 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-fluorophenyl]-N'-(3-methylphenyl)urea 19 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47505 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-chlorophenyl]-N'-(3-methylphenyl)urea 83 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47506 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-methoxyphenyl]-N'-(3-methylphenyl)urea 13 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47507 CLONED HUMAN Functional N-(11-Amino-5,6-dihydro-7-thia-8,10-diazabenzo[c]fluoren-3-yl)-N'-(3-methylphenyl)urea 150 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47508 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[4-(trifluoromethyl)phenyl]urea 61 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47509 CLONED HUMAN Functional N-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-fluoro-5-methylphenyl)urea 34 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47510 CLONED HUMAN Functional N-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea 50 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47511 CLONED HUMAN Functional N-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-chlorophenyl)urea 3 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47512 CLONED HUMAN Functional SU11248 18 Dai Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47513 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PYY,[leu31,Pro34], human 0.05 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47514 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PP, human 0.08 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47515 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PP, rat 92 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47516 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY GR231118 4.3 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47517 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY NPY [Ala31, Aib32], porcine 2.5 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47518 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY NPY [hPP(1-17), Ala31,Aib32], human 0.5 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47519 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 0.1 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47520 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY CGP71683A 1.3 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47521 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY JCF109 9.2 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47522 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY CP732925 1.6 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47523 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY CP760524 2.6 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47524 Y1 BRAIN RAT 125I-[Leu31,Pro34]PYY CP781214 4.2 Dumont Y, et al., 2005 Jan 15, 2025 Jan 15, 2025
47525 EAAT2 CLONED HUMAN 3H-GLUTAMATE WAY 213613 85 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47526 EAAT2 CLONED HUMAN 3H-GLUTAMATE WAY 213394 145 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47527 EAAT2 CLONED HUMAN 3H-GLUTAMATE WAY 212922 157 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47528 EAAT2 CLONED HUMAN 3H-GLUTAMATE WAY 211686 190 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47529 EAAT1 CLONED HUMAN 3H-GLUTAMATE WAY 213613 5004 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47530 EAAT1 CLONED HUMAN 3H-GLUTAMATE WAY 213394 1971 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47531 EAAT1 CLONED HUMAN 3H-GLUTAMATE WAY 212922 3426 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47532 EAAT1 CLONED HUMAN 3H-GLUTAMATE WAY 211686 1681 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47533 EAAT3 CLONED HUMAN 3H-GLUTAMATE WAY 213613 3787 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47534 EAAT3 CLONED HUMAN 3H-GLUTAMATE WAY 213394 6561 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47535 EAAT3 CLONED HUMAN 3H-GLUTAMATE WAY 211686 1453 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47536 EAAT3 CLONED HUMAN 3H-GLUTAMATE WAY 212922 1837 Dunlop J, et al., 2005 Jan 15, 2025 Jan 15, 2025
47537 L1210 cells UNDEFINED Functional (anthracen-9-ylmethyl)-3,3-triamine 1800 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47538 L1210 cells UNDEFINED Functional (anthracen-9-ylmethyl)-4,4-triamine 300 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47539 L1210 cells UNDEFINED Functional N1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt 3000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47540 L1210 cells UNDEFINED Functional N1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47541 L1210 cells UNDEFINED Functional N-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47542 L1210 cells UNDEFINED 14C-spermidine (anthracen-9-ylmethyl)-3,3-triamine >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47543 L1210 cells UNDEFINED 14C-spermidine (anthracen-9-ylmethyl)-4,4-triamine 1800 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47544 L1210 cells UNDEFINED 14C-spermidine N1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt 9900 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47545 L1210 cells UNDEFINED 14C-spermidine N1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt 6200 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47546 L1210 cells UNDEFINED 14C-spermidine N-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47547 CLONED UNDEFINED Functional (anthracen-9-ylmethyl)-3,3-triamine 1900 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47548 CLONED UNDEFINED Functional (anthracen-9-ylmethyl)-4,4-triamine 450 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47549 CLONED UNDEFINED Functional N1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47550 CLONED UNDEFINED Functional N1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47551 CLONED UNDEFINED Functional N-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt >10000 Kaur N, et al., 2005 Jan 15, 2025 Jan 15, 2025
47552 BRAIN RAT 3H-3-PPP,(+) PHENTOLAMINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47553 BRAIN RAT 3H-3-PPP,(+) IPRINDOLE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47554 BRAIN RAT 3H-3-PPP,(+) Amphetamine,(+) >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47555 BRAIN RAT 3H-3-PPP,(+) COCAINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47556 BRAIN RAT 3H-3-PPP,(+) Levorphanol >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47557 BRAIN RAT 3H-3-PPP,(+) Bradykinin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47558 BRAIN RAT 3H-3-PPP,(+) CCK33 >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47559 BRAIN RAT 3H-3-PPP,(+) DOPAMINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47560 BRAIN RAT 3H-3-PPP,(+) APOMORPHINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47561 BRAIN RAT 3H-3-PPP,(+) LISURIDE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47562 BRAIN RAT 3H-3-PPP,(+) NALOXONE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47563 BRAIN RAT 3H-3-PPP,(+) DIHYDROMORPHINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47564 BRAIN RAT 3H-3-PPP,(+) [D-Ala2-D-Leu5]enkephalin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47565 BRAIN RAT 3H-3-PPP,(+) Alpha-Neoendorphin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47566 BRAIN RAT 3H-3-PPP,(+) Beta-Neoendorphin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47567 BRAIN RAT 3H-3-PPP,(+) HEXAMETHONIUM >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47568 BRAIN RAT 3H-3-PPP,(+) Decamethonium >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47569 BRAIN RAT 3H-3-PPP,(+) SCOPOLAMINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47570 BRAIN RAT 3H-3-PPP,(+) RAUWOLSCINE >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47571 BRAIN RAT 3H-3-PPP,(+) Picrotoxin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47572 BRAIN RAT 3H-3-PPP,(+) Bicuculline >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47573 BRAIN RAT 3H-3-PPP,(+) Gamma-Aminobutyric acid >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47574 BRAIN RAT 3H-3-PPP,(+) amrinone >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47575 BRAIN RAT 3H-3-PPP,(+) tetrodotoxin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47576 BRAIN RAT 3H-3-PPP,(+) LYSERGIC ACID >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47577 BRAIN RAT 3H-3-PPP,(+) Cannabinol >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47578 BRAIN RAT 3H-3-PPP,(+) THC, delta 9 >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47579 BRAIN RAT 3H-3-PPP,(+) Angiotensin II >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47580 BRAIN RAT 3H-3-PPP,(+) Neurotensin >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47581 BRAIN RAT 3H-3-PPP,(+) CCK4 >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47582 BRAIN RAT 3H-3-PPP,(+) CCK8 >10000 Largent BL, et al., 1984 Jan 15, 2025 Jan 15, 2025
47583 PKCα CLONED HUMAN 3H-PDBU (Z)-CH2OCOC(CH3)3 2.9 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47584 PKCα CLONED HUMAN 3H-PDBU (E)-CH2OCOC(CH3)3 4.51 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47585 PKCα CLONED HUMAN 3H-PDBU CH2OCOC(CH3)3 1.45 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47586 PKCα CLONED HUMAN 3H-PDBU 5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 3.78 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47587 PKCα CLONED HUMAN 3H-PDBU 5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 6.18 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47588 PKCα CLONED HUMAN 3H-PDBU 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 4.97 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47589 PKCα CLONED HUMAN 3H-PDBU 5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone 6.04 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47590 PKCα CLONED HUMAN 3H-PDBU 5-Benzoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 6.66 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47591 PKCα CLONED HUMAN 3H-PDBU 5-Benzoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 16.1 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47592 PKCα CLONED HUMAN 3H-PDBU 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 6.87 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47593 PKCα CLONED HUMAN 3H-PDBU 5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone 4.46 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47594 PKCα CLONED HUMAN 3H-PDBU 5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isobutyl-5-methyl-hexanoyloxymethyl)tetrahydro-2-furanone 6.88 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47595 PKCα CLONED HUMAN 3H-PDBU 5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(Z)-3-isobutyl-5 -methylhexylidene]tetrahydro-2-furanone 18 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47596 PKCα CLONED HUMAN 3H-PDBU 5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone 173 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47597 PKCα CLONED HUMAN 3H-PDBU 5-[(Z)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone >10000 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47598 PKCα CLONED HUMAN 3H-PDBU 5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methyl-2-butenyl)dihydro-2(3H)-furanone 2100 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47599 PKCα CLONED HUMAN 3H-PDBU 5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methylbutyl)dihydro-2(3H)-furanone >10000 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47600 PKCα CLONED HUMAN 3H-PDBU 6-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone 28 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47601 PKCα CLONED HUMAN 3H-PDBU 6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone 48 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47602 PKCα CLONED HUMAN 3H-PDBU 6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-hexanoyloxymethyl-tetrahydro-2-pyranone 147 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47603 PKCα CLONED HUMAN 3H-PDBU 6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-octanoyloxymethyl-tetrahydro-2-pyranone 129 Lee J, et al., 2006 Jan 15, 2025 Jan 15, 2025
47604 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 100 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47605 ADK recombinant HUMAN Functional 4-N-Benzylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 800 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47606 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 550 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47607 ADK recombinant HUMAN Functional 4-N-(4-Methoxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 775 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47608 ADK recombinant HUMAN Functional 4-N-(4-Hydroxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 200 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47609 ADK recombinant HUMAN Functional 4-N-Cyclohexylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine >10000 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47610 ADK recombinant HUMAN Functional 4-N-(Cyanoyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1200 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47611 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-iodo-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 120 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47612 ADK recombinant HUMAN Functional 4-N-Phenylamino-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 1250 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47613 ADK recombinant HUMAN Functional 4-Amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 320 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47614 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 0.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025