The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 44,001-45,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
46615DORFOREBRAINGUINEA PIG3H-DADLE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46616DORFOREBRAINGUINEA PIG3H-DADLEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46617DORFOREBRAINGUINEA PIG3H-DADLE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46618DORFOREBRAINGUINEA PIG3H-DADLE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46619DORFOREBRAINGUINEA PIG3H-DADLE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46620DORFOREBRAINGUINEA PIG3H-DADLEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46621DORFOREBRAINGUINEA PIG3H-DADLE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46622DORFOREBRAINGUINEA PIG3H-DADLE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46623DORFOREBRAINGUINEA PIG3H-DADLEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46624DORFOREBRAINGUINEA PIG3H-DADLE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46625DORFOREBRAINGUINEA PIG3H-DADLE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46626DORFOREBRAINGUINEA PIG3H-DADLE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46627DORFOREBRAINGUINEA PIG3H-DADLE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46628DORFOREBRAINGUINEA PIG3H-DADLE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46629DORFOREBRAINGUINEA PIG3H-DADLE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46630DORFOREBRAINGUINEA PIG3H-DADLE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46631DORFOREBRAINGUINEA PIG3H-DADLE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46632DORFOREBRAINGUINEA PIG3H-DADLEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46633DORFOREBRAINGUINEA PIG3H-DADLE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46634DORFOREBRAINGUINEA PIG3H-DADLE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46635KORFOREBRAINRAT3H-MUSCIMOL(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46636KORFOREBRAINRAT3H-MUSCIMOL(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46637KORFOREBRAINRAT3H-MUSCIMOLPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46638KORFOREBRAINRAT3H-MUSCIMOL(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46639KORFOREBRAINRAT3H-MUSCIMOL(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46640KORFOREBRAINRAT3H-MUSCIMOLN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46641KORFOREBRAINRAT3H-MUSCIMOLPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46642KORFOREBRAINRAT3H-MUSCIMOLPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46643KORFOREBRAINRAT3H-MUSCIMOL(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46644KORFOREBRAINRAT3H-MUSCIMOL(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46645KORFOREBRAINRAT3H-MUSCIMOLPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46646KORFOREBRAINRAT3H-MUSCIMOL(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46647KORFOREBRAINRAT3H-MUSCIMOL(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46648KORFOREBRAINRAT3H-MUSCIMOL(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46649KORFOREBRAINRAT3H-MUSCIMOL(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46650KORFOREBRAINRAT3H-MUSCIMOL(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46651KORFOREBRAINRAT3H-MUSCIMOL(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46652KORFOREBRAINRAT3H-MUSCIMOL(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46653KORFOREBRAINRAT3H-MUSCIMOL(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46654KORFOREBRAINRAT3H-MUSCIMOL(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46655KORFOREBRAINRAT3H-MUSCIMOL(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46656KORFOREBRAINRAT3H-MUSCIMOL(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46657KORFOREBRAINRAT3H-MUSCIMOL(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46658KORFOREBRAINRAT3H-MUSCIMOL(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46659KORFOREBRAINRAT3H-MUSCIMOL(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46660KORFOREBRAINRAT3H-MUSCIMOL(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46661KORFOREBRAINRAT3H-MUSCIMOL(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46662KORFOREBRAINRAT3H-MUSCIMOL(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 27, 2025
46663H1CLONEDHUMAN3H-PYRILAMINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46664H1CLONEDHUMAN3H-PYRILAMINE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46665H1CLONEDHUMAN3H-PYRILAMINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46666H1CLONEDHUMAN3H-PYRILAMINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46667H1CLONEDHUMAN3H-PYRILAMINE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46668H1CLONEDHUMAN3H-PYRILAMINE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46669H1CLONEDHUMAN3H-PYRILAMINE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46670H1CLONEDHUMAN3H-PYRILAMINE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46671H1CLONEDHUMAN3H-PYRILAMINE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46672H1CLONEDHUMAN3H-PYRILAMINE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46673H1CLONEDHUMAN3H-PYRILAMINE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46674H1CLONEDHUMAN3H-PYRILAMINE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46675H1CLONEDHUMAN3H-PYRILAMINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46676H1CLONEDHUMAN3H-PYRILAMINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46677H1CLONEDHUMAN3H-PYRILAMINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46678H1CLONEDHUMAN3H-PYRILAMINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46679H1CLONEDHUMAN3H-PYRILAMINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46680H1CLONEDHUMAN3H-PYRILAMINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46681H1CLONEDHUMAN3H-PYRILAMINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46682H1CLONEDHUMAN3H-PYRILAMINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46683H1CLONEDHUMAN3H-PYRILAMINEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46684H1CLONEDHUMAN3H-PYRILAMINE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46685H1CLONEDHUMAN3H-PYRILAMINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46686H1CLONEDHUMAN3H-PYRILAMINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46687H1CLONEDHUMAN3H-PYRILAMINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46688H1CLONEDHUMAN3H-PYRILAMINEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46689H1CLONEDHUMAN3H-PYRILAMINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46690H1CLONEDHUMAN3H-PYRILAMINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46691H1CLONEDHUMAN3H-PYRILAMINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46692H1CLONEDHUMAN3H-PYRILAMINE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46693H2CLONEDHUMAN3H-TIOTIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46694H2CLONEDHUMAN3H-TIOTIDINE(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46695H2CLONEDHUMAN3H-TIOTIDINEPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46696H2CLONEDHUMAN3H-TIOTIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46697H2CLONEDHUMAN3H-TIOTIDINE(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46698H2CLONEDHUMAN3H-TIOTIDINE(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46699H2CLONEDHUMAN3H-TIOTIDINEPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46700H2CLONEDHUMAN3H-TIOTIDINEPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46701H2CLONEDHUMAN3H-TIOTIDINE(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46702H2CLONEDHUMAN3H-TIOTIDINE(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione2688Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46703H2CLONEDHUMAN3H-TIOTIDINE(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46704H2CLONEDHUMAN3H-TIOTIDINE(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46705H2CLONEDHUMAN3H-TIOTIDINEPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46706H2CLONEDHUMAN3H-TIOTIDINE(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46707H2CLONEDHUMAN3H-TIOTIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46708H2CLONEDHUMAN3H-TIOTIDINE(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46709H2CLONEDHUMAN3H-TIOTIDINE(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46710H2CLONEDHUMAN3H-TIOTIDINE(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46711H2CLONEDHUMAN3H-TIOTIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46712H2CLONEDHUMAN3H-TIOTIDINE(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46713H2CLONEDHUMAN3H-TIOTIDINE(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46714H2CLONEDHUMAN3H-TIOTIDINE(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione4877Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46715H2CLONEDHUMAN3H-TIOTIDINE(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46716H2CLONEDHUMAN3H-TIOTIDINEN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46717H2CLONEDHUMAN3H-TIOTIDINE(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46718H2CLONEDHUMAN3H-TIOTIDINE(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46719H2CLONEDHUMAN3H-TIOTIDINE(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46720H2CLONEDHUMAN3H-TIOTIDINE(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46721H2CLONEDHUMAN3H-TIOTIDINE(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46722H2CLONEDHUMAN3H-TIOTIDINE(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46723H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46724H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46725H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46726H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46727H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46728H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46729H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46730H3CLONEDGUINEA PIG3H-Alpha-Me-histamineN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46731H3CLONEDGUINEA PIG3H-Alpha-Me-histaminePL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46732H3CLONEDGUINEA PIG3H-Alpha-Me-histaminePL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46733H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46734H3CLONEDGUINEA PIG3H-Alpha-Me-histaminePL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46735H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46736H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46737H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46738H3CLONEDGUINEA PIG3H-Alpha-Me-histaminePL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46739H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46740H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46741H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46742H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46743H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46744H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46745H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46746H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46747H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46748H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46749H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46750H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione4750Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46751H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46752H3CLONEDGUINEA PIG3H-Alpha-Me-histamine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46753H4CLONEDHUMAN3H-HistaminePL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46754H4CLONEDHUMAN3H-Histamine(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46755H4CLONEDHUMAN3H-Histamine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46756H4CLONEDHUMAN3H-Histamine(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46757H4CLONEDHUMAN3H-HistaminePL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46758H4CLONEDHUMAN3H-Histamine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46759H4CLONEDHUMAN3H-Histamine(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46760H4CLONEDHUMAN3H-Histamine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46761H4CLONEDHUMAN3H-HistaminePL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46762H4CLONEDHUMAN3H-Histamine(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46763H4CLONEDHUMAN3H-Histamine(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46764H4CLONEDHUMAN3H-Histamine(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46765H4CLONEDHUMAN3H-Histamine(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46766H4CLONEDHUMAN3H-Histamine(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46767H4CLONEDHUMAN3H-HistaminePL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46768H4CLONEDHUMAN3H-Histamine(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46769H4CLONEDHUMAN3H-Histamine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3279Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46770H4CLONEDHUMAN3H-HistamineN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46771H4CLONEDHUMAN3H-Histamine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46772H4CLONEDHUMAN3H-Histamine(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46773H4CLONEDHUMAN3H-Histamine(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46774H4CLONEDHUMAN3H-Histamine(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46775H4CLONEDHUMAN3H-Histamine(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46776H4CLONEDHUMAN3H-Histamine(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46777H4CLONEDHUMAN3H-Histamine(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46778H4CLONEDHUMAN3H-Histamine(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46779H4CLONEDHUMAN3H-Histamine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46780H4CLONEDHUMAN3H-Histamine(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46781H4CLONEDHUMAN3H-Histamine(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46782KORCLONEDHUMAN3H-Bremazocine(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46783KORCLONEDHUMAN3H-Bremazocine(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46784KORCLONEDHUMAN3H-Bremazocine(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46785KORCLONEDHUMAN3H-Bremazocine(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46786KORCLONEDHUMAN3H-Bremazocine(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46787KORCLONEDHUMAN3H-Bremazocine(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46788KORCLONEDHUMAN3H-Bremazocine(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid2304Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46789KORCLONEDHUMAN3H-Bremazocine(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46790KORCLONEDHUMAN3H-Bremazocine(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46791KORCLONEDHUMAN3H-Bremazocine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46792KORCLONEDHUMAN3H-Bremazocine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione827.8Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46793KORCLONEDHUMAN3H-Bremazocine(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46794KORCLONEDHUMAN3H-Bremazocine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46795KORCLONEDHUMAN3H-Bremazocine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46796KORCLONEDHUMAN3H-Bremazocine(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46797KORCLONEDHUMAN3H-Bremazocine(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46798KORCLONEDHUMAN3H-BremazocinePL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46799KORCLONEDHUMAN3H-Bremazocine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46800KORCLONEDHUMAN3H-Bremazocine(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46801KORCLONEDHUMAN3H-BremazocineN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46802KORCLONEDHUMAN3H-Bremazocine(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone4060Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46803KORCLONEDHUMAN3H-Bremazocine(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46804KORCLONEDHUMAN3H-Bremazocine(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46805KORCLONEDHUMAN3H-Bremazocine(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46806KORCLONEDHUMAN3H-Bremazocine(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46807KORCLONEDHUMAN3H-Bremazocine(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46808KORCLONEDHUMAN3H-BremazocinePL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46809KORCLONEDHUMAN3H-Bremazocine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46810KORCLONEDHUMAN3H-BremazocinePL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46811KORCLONEDHUMAN3H-BremazocinePL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46812M2CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46813M2CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46814M2CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46815M2CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46816M2CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46817M2CLONEDHUMAN3H-QNB(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46818M2CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46819M2CLONEDHUMAN3H-QNB(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46820M2CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46821M2CLONEDHUMAN3H-QNB(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46822M2CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46823M2CLONEDHUMAN3H-QNB(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46824M2CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46825M2CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46826M2CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46827M2CLONEDHUMAN3H-QNB(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46828M2CLONEDHUMAN3H-QNB(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46829M2CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46830M2CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46831M2CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46832M2CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46833M2CLONEDHUMAN3H-QNBN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46834M2CLONEDHUMAN3H-QNBPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46835M2CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46836M2CLONEDHUMAN3H-QNBPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46837M2CLONEDHUMAN3H-QNB(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46838M2CLONEDHUMAN3H-QNB(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46839M2CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46840M2CLONEDHUMAN3H-QNBPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46841M2CLONEDHUMAN3H-QNBPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46842M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46843M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46844M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46845M5CLONEDHUMAN3H-QNB(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46846M5CLONEDHUMAN3H-QNB(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46847M5CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46848M5CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46849M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46850M5CLONEDHUMAN3H-QNB(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46851M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46852M5CLONEDHUMAN3H-QNB(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46853M5CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46854M5CLONEDHUMAN3H-QNBPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46855M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46856M5CLONEDHUMAN3H-QNB(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46857M5CLONEDHUMAN3H-QNB(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46858M5CLONEDHUMAN3H-QNBPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46859M5CLONEDHUMAN3H-QNB(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46860M5CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46861M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46862M5CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46863M5CLONEDHUMAN3H-QNBN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46864M5CLONEDHUMAN3H-QNBPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46865M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46866M5CLONEDHUMAN3H-QNB(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46867M5CLONEDHUMAN3H-QNB(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46868M5CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46869M5CLONEDHUMAN3H-QNB(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46870M5CLONEDHUMAN3H-QNBPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46871M5CLONEDHUMAN3H-QNB(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46872mGluR5CLONEDRATFunctional(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46873mGluR5CLONEDRATFunctional(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46874mGluR5CLONEDRATFunctional(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46875mGluR5CLONEDRATFunctional(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46876mGluR5CLONEDRATFunctional(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46877mGluR5CLONEDRATFunctional(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46878mGluR5CLONEDRATFunctional(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46879mGluR5CLONEDRATFunctional(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46880mGluR5CLONEDRATFunctional(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46881mGluR5CLONEDRATFunctional(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46882mGluR5CLONEDRATFunctional(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46883mGluR5CLONEDRATFunctional(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46884mGluR5CLONEDRATFunctional(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46885mGluR5CLONEDRATFunctional(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46886mGluR5CLONEDRATFunctionalN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46887mGluR5CLONEDRATFunctional(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46888mGluR5CLONEDRATFunctional(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46889mGluR5CLONEDRATFunctional(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46890mGluR5CLONEDRATFunctional(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46891mGluR5CLONEDRATFunctional(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46892mGluR5CLONEDRATFunctional(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46893mGluR5CLONEDRATFunctionalPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46894mGluR5CLONEDRATFunctionalPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46895mGluR5CLONEDRATFunctionalPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46896mGluR5CLONEDRATFunctional(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46897mGluR5CLONEDRATFunctional(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46898mGluR5CLONEDRATFunctional(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46899mGluR5CLONEDRATFunctional(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 28, 2025
46900MORCLONEDHUMAN3H-Diprenorphine(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46901MORCLONEDHUMAN3H-Diprenorphine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46902MORCLONEDHUMAN3H-Diprenorphine(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46903MORCLONEDHUMAN3H-DiprenorphinePL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46904MORCLONEDHUMAN3H-Diprenorphine(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46905MORCLONEDHUMAN3H-Diprenorphine(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46906MORCLONEDHUMAN3H-Diprenorphine(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46907MORCLONEDHUMAN3H-Diprenorphine(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46908MORCLONEDHUMAN3H-Diprenorphine(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46909MORCLONEDHUMAN3H-Diprenorphine(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46910MORCLONEDHUMAN3H-Diprenorphine(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46911MORCLONEDHUMAN3H-Diprenorphine(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46912MORCLONEDHUMAN3H-Diprenorphine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46913MORCLONEDHUMAN3H-DiprenorphinePL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46914MORCLONEDHUMAN3H-Diprenorphine(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46915MORCLONEDHUMAN3H-DiprenorphinePL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46916MORCLONEDHUMAN3H-Diprenorphine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46917MORCLONEDHUMAN3H-Diprenorphine(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46918MORCLONEDHUMAN3H-Diprenorphine(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46919MORCLONEDHUMAN3H-Diprenorphine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46920MORCLONEDHUMAN3H-Diprenorphine(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46921MORCLONEDHUMAN3H-DiprenorphineN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46922MORCLONEDHUMAN3H-Diprenorphine(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46923MORCLONEDHUMAN3H-Diprenorphine(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46924MORCLONEDHUMAN3H-Diprenorphine(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46925MORCLONEDHUMAN3H-DiprenorphinePL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46926MORCLONEDHUMAN3H-Diprenorphine(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46927MORCLONEDHUMAN3H-Diprenorphine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46928MORCLONEDHUMAN3H-Diprenorphine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46929MORCLONEDHUMAN3H-Diprenorphine(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46930NETCLONEDHUMAN3H-Nisoxetine(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46931NETCLONEDHUMAN3H-Nisoxetine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46932NETCLONEDHUMAN3H-Nisoxetine(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46933NETCLONEDHUMAN3H-Nisoxetine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46934NETCLONEDHUMAN3H-Nisoxetine(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46935NETCLONEDHUMAN3H-Nisoxetine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46936NETCLONEDHUMAN3H-Nisoxetine(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46937NETCLONEDHUMAN3H-NisoxetineN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46938NETCLONEDHUMAN3H-NisoxetinePL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46939NETCLONEDHUMAN3H-NisoxetinePL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46940NETCLONEDHUMAN3H-Nisoxetine(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46941NETCLONEDHUMAN3H-NisoxetinePL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46942NETCLONEDHUMAN3H-Nisoxetine(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46943NETCLONEDHUMAN3H-Nisoxetine(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46944NETCLONEDHUMAN3H-Nisoxetine(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46945NETCLONEDHUMAN3H-NisoxetinePL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46946NETCLONEDHUMAN3H-Nisoxetine(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46947NETCLONEDHUMAN3H-Nisoxetine(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46948NETCLONEDHUMAN3H-Nisoxetine(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46949NETCLONEDHUMAN3H-Nisoxetine(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46950NETCLONEDHUMAN3H-Nisoxetine(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46951NETCLONEDHUMAN3H-Nisoxetine(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46952NETCLONEDHUMAN3H-Nisoxetine(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46953NETCLONEDHUMAN3H-Nisoxetine(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46954NETCLONEDHUMAN3H-Nisoxetine(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46955NETCLONEDHUMAN3H-Nisoxetine(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46956NETCLONEDHUMAN3H-Nisoxetine(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46957NETCLONEDHUMAN3H-Nisoxetine(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46958NETCLONEDHUMAN3H-Nisoxetine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46959NETCLONEDHUMAN3H-Nisoxetine(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46960SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46961SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46962SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46963SLC6A4CLONEDHUMAN3H-CITALOPRAM(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46964SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46965SLC6A4CLONEDHUMAN3H-CITALOPRAM(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46966SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46967SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46968SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46969SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46970SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46971SLC6A4CLONEDHUMAN3H-CITALOPRAM(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46972SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46973SLC6A4CLONEDHUMAN3H-CITALOPRAM(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46974SLC6A4CLONEDHUMAN3H-CITALOPRAM(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46975SLC6A4CLONEDHUMAN3H-CITALOPRAMPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46976SLC6A4CLONEDHUMAN3H-CITALOPRAM(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46977SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46978SLC6A4CLONEDHUMAN3H-CITALOPRAM(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46979SLC6A4CLONEDHUMAN3H-CITALOPRAM(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46980SLC6A4CLONEDHUMAN3H-CITALOPRAMN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46981SLC6A4CLONEDHUMAN3H-CITALOPRAMPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46982SLC6A4CLONEDHUMAN3H-CITALOPRAMPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46983SLC6A4CLONEDHUMAN3H-CITALOPRAM(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46984SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46985SLC6A4CLONEDHUMAN3H-CITALOPRAM(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46986SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46987SLC6A4CLONEDHUMAN3H-CITALOPRAMPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46988SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46989SLC6A4CLONEDHUMAN3H-CITALOPRAM(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46990Sigma 1BRAINRAT3H-Pentazocine(+)(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46991Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46992Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46993Sigma 1BRAINRAT3H-Pentazocine(+)(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46994Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46995Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46996Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46997Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46998Sigma 1BRAINRAT3H-Pentazocine(+)(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
46999Sigma 1BRAINRAT3H-Pentazocine(+)(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47000Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47001Sigma 1BRAINRAT3H-Pentazocine(+)(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47002Sigma 1BRAINRAT3H-Pentazocine(+)(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione4343Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47003Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47004Sigma 1BRAINRAT3H-Pentazocine(+)(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3956Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47005Sigma 1BRAINRAT3H-Pentazocine(+)(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47006Sigma 1BRAINRAT3H-Pentazocine(+)(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47007Sigma 1BRAINRAT3H-Pentazocine(+)(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47008Sigma 1BRAINRAT3H-Pentazocine(+)PL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47009Sigma 1BRAINRAT3H-Pentazocine(+)(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione557.7Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47010Sigma 1BRAINRAT3H-Pentazocine(+)N,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47011Sigma 1BRAINRAT3H-Pentazocine(+)PL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47012Sigma 1BRAINRAT3H-Pentazocine(+)(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47013Sigma 1BRAINRAT3H-Pentazocine(+)(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47014Sigma 1BRAINRAT3H-Pentazocine(+)(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47015Sigma 1BRAINRAT3H-Pentazocine(+)(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47016Sigma 1BRAINRAT3H-Pentazocine(+)(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47017Sigma 1BRAINRAT3H-Pentazocine(+)PL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47018Sigma 1BRAINRAT3H-Pentazocine(+)PL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47019Sigma 1BRAINRAT3H-Pentazocine(+)(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47020Sigma 2PC12RAT3H-DTGPL-3-025>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47021Sigma 2PC12RAT3H-DTG(3S,4S,6aS,9S,10S,12aS)-4,10-bis(2-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3386Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47022Sigma 2PC12RAT3H-DTG(3S,4S,6aS,9S,10S,12aS)-4,10-bis(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione8594Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47023Sigma 2PC12RAT3H-DTG(3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-4,10-bis(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47024Sigma 2PC12RAT3H-DTG(2S,5S,6S)-6-(3-allylphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47025Sigma 2PC12RAT3H-DTG(1S,3S)-1-(3,4,5-trimethoxyphenyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47026Sigma 2PC12RAT3H-DTG(2S,5R,6R)-6-(4'-methoxybiphenyl-2-yl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47027Sigma 2PC12RAT3H-DTG(2S,5R,6R)-6-(4-(3-methoxyprop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47028Sigma 2PC12RAT3H-DTG(2S,5R,6R)-5-methyl-6-(3-morpholinophenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47029Sigma 2PC12RAT3H-DTG(2S,5R,6R)-6-(4-acetamidophenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47030Sigma 2PC12RAT3H-DTG(2S,5S,6S)-5-methyl-6-(3-(2-oxopyrrolidin-1-yl)phenyl)piperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47031Sigma 2PC12RAT3H-DTG(3R,4R,6aS,9R,10R,12aS)-4,10-bis(3-bromophenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47032Sigma 2PC12RAT3H-DTG(2S,5R,6R)-6-(4-(furan-2-yl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47033Sigma 2PC12RAT3H-DTGPL-3-017>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47034Sigma 2PC12RAT3H-DTG(2S,5S,6S)-6-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47035Sigma 2PC12RAT3H-DTG(3R,4R,6aS,9S,10S,12aS)-4-(4-(furan-2-yl)phenyl)-3,9-dimethyl-10-(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47036Sigma 2PC12RAT3H-DTG(2S,5S,6S)-6-(3-methoxyphenyl)-5-methylpiperidine-2-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47037Sigma 2PC12RAT3H-DTGPL-3-048-4>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47038Sigma 2PC12RAT3H-DTG(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(3-methoxyprop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47039Sigma 2PC12RAT3H-DTG(3S,6S,7S,9aS)-3-isopropyl-6-(3-methoxyphenyl)-2,7-dimethylhexahydro-1H-pyrido[1,2-a]pyrazine-1,4(6H)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47040Sigma 2PC12RAT3H-DTG(5aS,8R,9R,11aS)-9-(4-bromophenyl)-8-methylhexahydro-1H-pyrido[1,2-a]pyrrolo[1,2-d]pyrazine-5,11(5aH,11aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47041Sigma 2PC12RAT3H-DTG(3R,4R,6aS,9R,10R,12aS)-4-(3-bromophenyl)-3,9-dimethyl-10-(3-morpholinophenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47042Sigma 2PC12RAT3H-DTGPL-3-016>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47043Sigma 2PC12RAT3H-DTGN,N'-(4,4'-((3R,4R,6aS,9R,10R,12aS)-3,9-dimethyl-6,12-dioxododecahydrodipyrido[1,2-a:1',2'-d]pyrazine-4,10-diyl)bis(4,1-phenylene))diacetamide>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47044Sigma 2PC12RAT3H-DTG(3S,4S,6aS,9S,10S,12aS)-3,9-dimethyl-4,10-bis(3-(2-oxopyrrolidin-1-yl)phenyl)octahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47045Sigma 2PC12RAT3H-DTG(3R,4R,6aS,9R,10R,12aS)-4,10-bis(4-(furan-2-yl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47046Sigma 2PC12RAT3H-DTG(3S,4S,7S,8S,9aS,10aS)-4,8-Bis-(3-methoxy-phenyl)-3,7-dimethyl-octahydro-4a,8a-diaza-anthraquinone>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47047Sigma 2PC12RAT3H-DTG(3S,4S,6aS,9S,10S,12aS)-4,10-bis(3-allylphenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47048Sigma 2PC12RAT3H-DTG(1R,3S)-1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid>10000Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47049Sigma 2PC12RAT3H-DTG(3S,4S,6aS,9S,10S,12aS)-4-(2-bromophenyl)-10-(4-(3-(dimethylamino)prop-1-ynyl)phenyl)-3,9-dimethyloctahydrodipyrido[1,2-a:1',2'-d]pyrazine-6,12(6aH,12aH)-dione3093Dandapani S, et al., 2006Jan 15, 2025Jan 15, 2025
47050CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25S)-DLAM-1P2.74Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47051CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25S)-DLAM-2P8Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47052CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25R)-DLAM-2P 0.34Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47053CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25S)-DLAM-3P0.68Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47054CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25S)-DLAM-4P5.24Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47055CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25S)-DLAM-MPM2.2Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47056CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25S)-DLAM-03I1.52Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47057CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R,25R)-DLAM-1P0.25Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47058CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S,25R)-DLAM-1P0.18Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47059CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R,25S)-DLAM-1P0.25Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47060CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25R)-DLAM-2P0.51Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47061CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25R)-DLAM-3P0.19Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47062CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25S)-DLAM-2P0.19Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47063CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25R)-DLAM-3P0.09Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47064CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25S)-DLAM-3P0.03Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47065CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25R)-DLAM-4P0.3Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47066CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25R)-DLAM-4P0.09Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47067CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25S)-DLAM-4P0.1Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47068CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25R)-DLAM-MPM0.3Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47069CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25R)-DLAM-MPM0.09Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47070CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25S)-DLAM-MPM0.1Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47071CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25R)-DLAM-03I0.14Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47072CLONEDHUMAN26,27-methyl-3H-1,25-D3(23S, 25R)-DLAM-03I0.14Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47073CLONEDHUMAN26,27-methyl-3H-1,25-D3(23R, 25S)-DLAM-03I0.11Nakano Y, et al., 2006Jan 15, 2025Jan 15, 2025
47074H3CORTEXRAT125I-IPPIodophenpropit0.97Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47075H1CLONEDGUINEA PIG3H-MEPYRAMINEIodophenpropit1710Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47076H1CLONEDGUINEA PIG3H-MEPYRAMINEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47077H2CLONEDGUINEA PIG125I-aminopotentidineIodophenpropit2280Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47078H2CLONEDGUINEA PIG125I-aminopotentidineThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47079H3CORTEXRAT125I-IPPThioperamide4.3Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47080WHOLE BRAINRAT3H-PRAZOSINIodophenpropit1500Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47081WHOLE BRAINRAT3H-PRAZOSINThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47082WHOLE BRAIN MINUS CEREBELLUMRAT3H-CLONIDINEIodophenpropit120Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47083WHOLE BRAIN MINUS CEREBELLUMRAT3H-CLONIDINEThioperamide4000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47084Beta2CORTEXRAT3H-DHAIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47085Beta2CORTEXRAT3H-DHAThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47086LIVERRAT3H-IDAZOXANIodophenpropit530Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47087LIVERRAT3H-IDAZOXANThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47088D1CAUDATE NUCLEUSRAT3H-dopamineIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47089D1CAUDATE NUCLEUSRAT3H-dopamineThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47090D2Corpus StriatumRAT3H-SPIPERONEIodophenpropit4500Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47091D2Corpus StriatumRAT3H-SPIPERONEIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47092D3S. NigraRAT3H-SPIPERONEIodophenpropit1800Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47093D3S. NigraRAT3H-SPIPERONEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
470945-HT1AFR. CORTEXRAT3H-8-OH-DPATIodophenpropit2300Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
470955-HT1AFR. CORTEXRAT3H-8-OH-DPATThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
470965-HT1BFR. CORTEXRAT3H-5HTIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
470975-HT1BFR. CORTEXRAT3H-5HTThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
470985-HT1DCAUDATE NUCLEUSRAT3H-5HTIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
470995-HT1DCAUDATE NUCLEUSRAT3H-5HTThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471005-HT2AFR. CORTEXRAT3H-SPIPERONEIodophenpropit1900Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471015-HT2AFR. CORTEXRAT3H-SPIPERONEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471025-HT2CFR. CORTEXRAT3H-SPIPERONEIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471035-HT2CFR. CORTEXRAT3H-SPIPERONEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471045-HT3ILEUMGUINEA PIG3H-GR-65630Iodophenpropit11Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471055-HT3ILEUMGUINEA PIG3H-GR-65630Thioperamide120Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471065-HT4BRAINGUINEA PIG3H-GR-113808Iodophenpropit530Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
471075-HT4BRAINGUINEA PIG3H-GR-113808Thioperamide2800Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47108SLC6A4BRAINGUINEA PIG3H-PAROXETINEIodophenpropit1250Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47109SLC6A4BRAINGUINEA PIG3H-PAROXETINEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47110M1CORTEXRAT3H-PIRENZEPINEIodophenpropit1500Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47111M1CORTEXRAT3H-PIRENZEPINEThioperamide4600Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47112M2HEARTRAT3H-NMSIodophenpropit1980Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47113M2HEARTRAT3H-NMSThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47114M3CLONEDHUMAN3H-NMSIodophenpropit3700Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47115M3CLONEDHUMAN3H-NMSThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47116FR. CORTEXRAT3H-5HTIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47117FR. CORTEXRAT3H-5HTThioperamide6400Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47118DORWHOLE BRAIN MINUS CEREBELLUMRAT3H-DADLEIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47119DORWHOLE BRAIN MINUS CEREBELLUMRAT3H-DADLEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47120KORWHOLE BRAIN MINUS CEREBELLUMRAT3H-EKCIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47121KORWHOLE BRAIN MINUS CEREBELLUMRAT3H-EKCThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47122MORWHOLE BRAIN MINUS CEREBELLUMRAT3H-NALOXONEIodophenpropit8400Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47123MORWHOLE BRAIN MINUS CEREBELLUMRAT3H-NALOXONEThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47124WHOLE BRAINRAT3H-3-PPP,(+)Iodophenpropit170Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47125WHOLE BRAINRAT3H-3-PPP,(+)Thioperamide180Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47126GABAACEREBELLUMRAT3H-DIAZEPAMIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47127GABAACEREBELLUMRAT3H-DIAZEPAMThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47128CORTEXRAT3H-CCK8Iodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47129CORTEXRAT3H-CCK8Thioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47130PANCREASRAT3H-CCK8Iodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47131PANCREASRAT3H-CCK8Thioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47132CLONEDHUMAN3H-SUBSTANCE PIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47133CLONEDHUMAN3H-SUBSTANCE PThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47134BRAINChick125I-IodomelatoninIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47135BRAINChick125I-IodomelatoninThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47136NMDABRAINRAT3H-CGS-19755Iodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47137NMDABRAINRAT3H-CGS-19755Thioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47138KORCEREBELLUMRAT3H-MUSCIMOLIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47139KORCEREBELLUMRAT3H-MUSCIMOLThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47140GlyRmedulla, ponsRAT3H-StrychnineIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47141GlyRmedulla, ponsRAT3H-StrychnineThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47142GlyRBRAINRAT3H-5,7-DCKAIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47143GlyRBRAINRAT3H-5,7-DCKAThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47144Total CortexRAT3H-BatrachotoxinIodophenpropit1000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47145Total CortexRAT3H-BatrachotoxinThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47146BRAINRAT3H-NitrendipineIodophenpropit>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47147BRAINRAT3H-NitrendipineThioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 15, 2025
47148Calcium channelBRAINRAT3H-D-888Iodophenpropit400Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47149Calcium channelBRAINRAT3H-D-888Thioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47150Calcium channelHEARTRAT3H-D-888Iodophenpropit560Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47151Calcium channelHEARTRAT3H-D-888Thioperamide>10000Leurs R. et. al. 1995Jan 15, 2025Jan 27, 2025
47152H1CLONEDHUMAN3H-MEPYRAMINEHISTAMINE>10000Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47153H1CLONEDHUMAN3H-MEPYRAMINE5-APT3090Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47154H1CLONEDHUMAN3H-MEPYRAMINECF3-5-APT6270Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47155H1CLONEDHUMAN3H-MEPYRAMINEOCH3-5-APT3200Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47156H1CLONEDHUMAN3H-MEPYRAMINECL-5-APT2650Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47157H1CLONEDHUMAN3H-MEPYRAMINE6-APT9570Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47158H1CLONEDHUMAN3H-MEPYRAMINECF3-6-APT2740Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47159H1CLONEDHUMAN3H-MEPYRAMINEOCH3-6-APT1220Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47160H1CLONEDHUMAN3H-MEPYRAMINECL-6-APT1310Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47161H1CLONEDHUMAN3H-MEPYRAMINEBr-6-APT130Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471625-HT2ACLONEDHUMAN3H-KETANSERIN5-APT800Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471635-HT2CCLONEDHUMAN3H-MESULERGINE5-APT310Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471645-HT2ACLONEDHUMAN3H-KETANSERIN6-APT1200Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471655-HT2CCLONEDHUMAN3H-MESULERGINE6-APT1500Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471665-HT2ACLONEDHUMAN3H-KETANSERINCL-6-APT1200Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471675-HT2CCLONEDHUMAN3H-MESULERGINECL-6-APT4600Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471685-HT2ACLONEDHUMAN3H-KETANSERINBr-6-APT580Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
471695-HT2CCLONEDHUMAN3H-MESULERGINEBr-6-APT540Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47170H1CLONEDHUMAN3H-MEPYRAMINE2-(Dimethylamino)tetralin165Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47171H1CLONEDHUMAN3H-MEPYRAMINEDiphenhydramine9.57Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47172H1CLONEDHUMAN3H-MEPYRAMINEBUTACLAMOL,(+)147Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47173H1CLONEDHUMAN3H-MEPYRAMINE(R)-Chlopheniramine80Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47174H1CLONEDHUMAN3H-MEPYRAMINEl-Chlorpheniramine0.31Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47175H1CLONEDHUMAN3H-MEPYRAMINETriprolidine0.69Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47176H1CLONEDHUMAN3H-MEPYRAMINEATR1240Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47177H1CLONEDHUMAN3H-MEPYRAMINE(-)-NANM5000Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47178H1CLONEDHUMAN3H-MEPYRAMINEDOXEPIN0.16Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47179H1CLONEDHUMAN3H-MEPYRAMINEFLUPENTHIXOL, Alpha0.86Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47180H1CLONEDHUMAN3H-MEPYRAMINEFlupenthixol, Beta5.73Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47181H1CLONEDHUMAN3H-MEPYRAMINESCH 23390101Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47182H1CLONEDHUMAN3H-MEPYRAMINEMETHYSERGIDE3000Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47183H1CLONEDHUMAN3H-MEPYRAMINEMAZINDOL600Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47184H1CLONEDHUMAN3H-MEPYRAMINESKF 383932500Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47185H1CLONEDHUMAN3H-MEPYRAMINEAMITRIPTYLINE0.5Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47186H1CLONEDHUMAN3H-MEPYRAMINEDESIPRAMINE45.4Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47187H1CLONEDHUMAN3H-MEPYRAMINE7-OH-DPAT1500Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47188H1CLONEDHUMAN3H-MEPYRAMINEHALOPERIDOL215Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47189H1CLONEDHUMAN3H-MEPYRAMINELoperamide2000Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47190H1CLONEDHUMAN3H-MEPYRAMINEMIANSERIN0.3Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47191H1CLONEDHUMAN3H-MEPYRAMINERIMCAZOLE5000Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47192H1CLONEDHUMAN3H-MEPYRAMINESPIPERONE272Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47193H1CLONEDHUMAN3H-MEPYRAMINEKETANSERIN1.79Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47194H1CLONEDHUMAN3H-MEPYRAMINEPROMETHAZINE0.24Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47195H1CLONEDHUMAN3H-MEPYRAMINEMEPYRAMINE0.74Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47196H1CLONEDHUMAN3H-MEPYRAMINEGBR-129099.33Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47197H1CLONEDHUMAN3H-MEPYRAMINENORTRYPTYLINE15.1Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47198H1CLONEDHUMAN3H-MEPYRAMINE(+/-)-BMY-1402180Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47199H1CLONEDHUMAN3H-MEPYRAMINE3-Aminofluoranthene4800Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47200H1CLONEDHUMAN3H-MEPYRAMINE3-(Dimethylamino)fluoranthene4800Ghoneim OM, et al., 2006Jan 15, 2025Jan 15, 2025
47201CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-methylthiourea>10000Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47202CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-butylthiourea4650Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47203CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-tert-butylthiourea>10000Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47204CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-isopropylthiourea>10000Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47205CLONEDHUMANFunctional1-(Bicyclo[2.2.1]hept-5-en-2-yl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea3660Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47206CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-cyclohexylthiourea4700Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47207CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-benzylthiourea5670Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47208CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-phenylthiourea4480Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47209CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-naphthalen-1-ylthiourea2790Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47210CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methylphenyl)thiourea2140Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47211CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-ethylphenyl)thiourea2780Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47212CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-fluorophenyl)thiourea4730Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47213CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(dimethylamino)phenyl)thiourea2030Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47214CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-nitrophenyl)thiourea2680Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47215CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-acetylphenyl)thiourea1790Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47216CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)-propyl)-3-(4-methylsulfanyl-phenyl)-thiourea1660Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47217CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-(benzyloxy)phenyl)thiourea970Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47218CLONEDHUMANFunctional1-(4-Ethoxy-phenyl)-3-(3-(1H-imidazol-1-yl)-propyl)thiourea890Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47219CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(4-methoxyphenyl)thiourea700Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47220CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(benzo[d][1,3]dioxol-6-yl)thiourea5660Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47221CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3-methoxyphenyl)thiourea1860Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47222CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxybenzyl)thiourea1550Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47223CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,3-dihydrobenzo[b][1,4]dioxin-7-yl)thiourea1120Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47224CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,5-dimethoxyphenyl)thiourea750Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47225CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(2,4-dimethoxyphenyl)thiourea560Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47226CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)urea490Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47227CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4,5-trimethoxyphenyl)thiourea340Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47228CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)thiourea60Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47229CLONEDHUMANFunctional1-(2-(1H-Imidazol-1-yl)ethyl)-3-(3,4-dimethoxyphenyl)thiourea>10000Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47230CLONEDHUMANFunctional1-(4-(1H-Imidazol-1-yl)butyl)-3-(3,4-dimethoxyphenyl)thiourea550Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47231CLONEDHUMANFunctional1-((R)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea340Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47232CLONEDHUMANFunctional1-((S)-3-(1H-Imidazol-1-yl)-2-methylpropyl)-3-(3,4-dimethoxyphenyl)thiourea760Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47233CLONEDHUMANFunctional1-((1-((1H-Imidazol-1-yl)methyl)cyclopropyl)methyl)-3-(3,4-dimethoxyphenyl)thiourea2330Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47234CLONEDHUMANFunctional1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dimethoxyphenyl)-1-methylthiourea4830Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47235CLONEDHUMANFunctionalN-(3-(1H-imidazol-1-yl)propyl)benzo[d]thiazol-2-amine3730Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47236CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-6-chlorobenzo[d]thiazol-2-amine3350Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47237CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-6-methoxybenzo[d]thiazol-2-amine1570Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47238CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-5,6-dimethoxybenzo[d]thiazol-2-amine2000Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47239CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-2-(3,4-dimethoxyphenyl)ethanethioamide390Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47240CLONEDHUMANFunctional(R)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide7340Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47241CLONEDHUMANFunctional(S)-N-(3-(1H-Imidazol-1-yl)propyl)-2-phenylpropanethioamide3510Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47242CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-2,2-diphenylethanethioamide4480Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47243CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-1-(4-methoxyphenyl)cyclopropanecarbothioamide400Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47244CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-1-(4-chlorophenyl)cyclobutanecarbothioamide4880Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47245CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-1-(4-chlorophenyl)cyclopentanecarbothioamide7330Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47246CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-1-(4-methoxyphenyl)cyclohexanecarbothioamide2220Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47247CLONEDHUMANFunctionalN-(3-(1H-Imidazol-1-yl)propyl)-1-(3,4-dimethoxyphenyl)cyclopropanecarbothioamide90Buchholz M, et al., 2006Jan 15, 2025Jan 15, 2025
47248CLONEDHUMANFunctionalMotilin0.15Li JJ, et al., 2004Jan 15, 2025Jan 15, 2025
47249CLONEDHUMAN125I-MotilinMotilin3.1Li JJ, et al., 2004Jan 15, 2025Jan 15, 2025
47250CLONEDHUMANFunctionalABT-2294.2Li JJ, et al., 2004Jan 15, 2025Jan 15, 2025
47251CLONEDHUMAN125I-MotilinABT-2293.4Li JJ, et al., 2004Jan 15, 2025Jan 15, 2025
47252CLONEDHUMANFunctionalerythromycin-A400Li JJ, et al., 2004Jan 15, 2025Jan 15, 2025
47253CLONEDHUMAN125I-Motilinerythromycin-A>10000Li JJ, et al., 2004Jan 15, 2025Jan 15, 2025
47254duodenumRABBIT125I-MotilinSK-8963.5Tsukamoto K, et al., 2000Jan 15, 2025Jan 15, 2025
47255duodenumRABBIT125I-MotilinMotilin3.1Tsukamoto K, et al., 2000Jan 15, 2025Jan 15, 2025
47256duodenumHUMAN125I-Motilin[Leu13]motilin3.6Tsukamoto K, et al., 2000Jan 15, 2025Jan 15, 2025
47257duodenumRABBIT125I-Motilin[Leu13]motilin1.1Tsukamoto K, et al., 2000Jan 15, 2025Jan 15, 2025
47258duodenumRABBIT125I-MotilinSK-8963.4Tsukamoto K, et al., 2000Jan 15, 2025Jan 15, 2025
47259duodenumHUMAN125I-MotilinMotilin3.4Tsukamoto K, et al., 2000Jan 15, 2025Jan 15, 2025
47260Beta1CEREBRAL CORTEXRAT125I-ICYPArotinolol0.18197Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47261Beta1CEREBRAL CORTEXRAT125I-ICYPPINDOLOL,(+/-)0.660693Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47262Beta1CEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, l-0.691831Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47263Beta1CEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, dl2.81838Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47264Beta1CEREBRAL CORTEXRAT125I-ICYPALPRENOLOL4.16869Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47265Beta1CEREBRAL CORTEXRAT125I-ICYPYM-095384.36516Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47266Beta1CEREBRAL CORTEXRAT125I-ICYPOXPRENOLOL7.76247Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47267Beta1CEREBRAL CORTEXRAT125I-ICYPLABETALOL12.0226Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47268Beta1CEREBRAL CORTEXRAT125I-ICYPBETAXOLOL12.3027Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47269Beta1CEREBRAL CORTEXRAT125I-ICYPl-Metoprolol13.8038Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47270Beta1CEREBRAL CORTEXRAT125I-ICYPmetoprolol63.0957Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47271Beta1CEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, d81.2831Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47272Beta1CEREBRAL CORTEXRAT125I-ICYPATENOLOL97.7237Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47273Beta1CEREBRAL CORTEXRAT125I-ICYPacebutolol125.893Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47274Beta1CEREBRAL CORTEXRAT125I-ICYPICI 118,551194.984Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47275Beta1CEREBRAL CORTEXRAT125I-ICYPPRACTOLOL245.471Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47276Beta1CEREBRAL CORTEXRAT125I-ICYPSotalol2238.72Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47277Beta1CEREBRAL CORTEXRAT125I-ICYPButoxamine3715.35Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47278Beta1CEREBRAL CORTEXRAT125I-ICYPd-Metoprolol>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47279Beta2CEREBRAL CORTEXRAT125I-ICYPArotinolol0.549541Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47280Beta2CEREBRAL CORTEXRAT125I-ICYPPINDOLOL,(+/-)0.316228Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47281Beta2CEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, l-0.457088Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47282Beta2CEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, dl2.45471Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47283Beta2CEREBRAL CORTEXRAT125I-ICYPALPRENOLOL0.57544Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47284Beta2CEREBRAL CORTEXRAT125I-ICYPYM-0953813.1826Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47285Beta2CEREBRAL CORTEXRAT125I-ICYPLABETALOL67.6083Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47286Beta2CEREBRAL CORTEXRAT125I-ICYPBETAXOLOL2041.74Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47287Beta2CEREBRAL CORTEXRAT125I-ICYPl-Metoprolol2454.71Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47288Beta2CEREBRAL CORTEXRAT125I-ICYPmetoprolol1698.24Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47289Beta2CEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, d43.6516Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47290Beta2CEREBRAL CORTEXRAT125I-ICYPATENOLOL2818.38Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47291Beta2CEREBRAL CORTEXRAT125I-ICYPacebutolol7079.46Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47292Beta2CEREBRAL CORTEXRAT125I-ICYPICI 118,5511.77828Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47293Beta2CEREBRAL CORTEXRAT125I-ICYPPRACTOLOL>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47294Beta2CEREBRAL CORTEXRAT125I-ICYPSotalol338.844Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47295Beta2CEREBRAL CORTEXRAT125I-ICYPButoxamine467.735Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
47296Beta2CEREBRAL CORTEXRAT125I-ICYPd-Metoprolol>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
472975-HT1BCEREBRAL CORTEXRAT125I-ICYPArotinolol10.7152Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
472985-HT1BCEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, dl56.2341Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
472995-HT1BCEREBRAL CORTEXRAT125I-ICYPPINDOLOL,(+/-)58.8844Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473005-HT1BCEREBRAL CORTEXRAT125I-ICYPALPRENOLOL70.7946Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473015-HT1BCEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, l-77.6247Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473025-HT1BCEREBRAL CORTEXRAT125I-ICYPOXPRENOLOL173.78Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473035-HT1BCEREBRAL CORTEXRAT125I-ICYPYM-095381288.25Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473045-HT1BCEREBRAL CORTEXRAT125I-ICYPLABETALOL1995.26Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473055-HT1BCEREBRAL CORTEXRAT125I-ICYPICI 118,5513890.45Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473065-HT1BCEREBRAL CORTEXRAT125I-ICYPacebutolol4168.69Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473075-HT1BCEREBRAL CORTEXRAT125I-ICYPPROPRANOLOL, d7079.46Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473085-HT1BCEREBRAL CORTEXRAT125I-ICYPBETAXOLOL>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473095-HT1BCEREBRAL CORTEXRAT125I-ICYPmetoprolol>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473105-HT1BCEREBRAL CORTEXRAT125I-ICYPl-Metoprolol>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473115-HT1BCEREBRAL CORTEXRAT125I-ICYPPRACTOLOL>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473125-HT1BCEREBRAL CORTEXRAT125I-ICYPSotalol>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473135-HT1BCEREBRAL CORTEXRAT125I-ICYPButoxamine>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473145-HT1BCEREBRAL CORTEXRAT125I-ICYPd-Metoprolol>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
47315Beta2CEREBRAL CORTEXRAT125I-ICYPOXPRENOLOL9.77237Tsuchihashi H, et al., 1990Jan 15, 2025Jan 28, 2025
473165-HT1BCEREBRAL CORTEXRAT125I-ICYPATENOLOL>10000Tsuchihashi H, et al., 1990Jan 15, 2025Jan 15, 2025
473175-HT1ACLONEDHUMAN3H-8-OH-DPATWAY 100,6352.2Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473185-HT1BCLONEDHUMAN3H-GR-125743WAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473195-HT1DCLONEDHUMAN3H-GR-125743WAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473205-HT1ECLONEDHUMAN3H-5HTWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473215-HT2ACLONEDHUMAN3H-KETANSERINWAY 100,6356260Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473225-HT2CCLONEDRAT3H-MESULERGINEWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47323CB1CLONEDHUMAN3H-LSDWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 27, 2025
473245-HT6CLONEDHUMAN3H-LSDWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473255-HT7CLONEDHUMAN3H-LSDWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
473265-HT2BCLONEDHUMAN3H-LSDWAY 100,63524Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47327H1CLONEDHUMAN3H-PYRILAMINEWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47328H2CLONEDHUMAN3H-TIOTIDINEWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47329H3CLONEDGUINEA PIG3H-Alpha-Me-histamineWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47330H4CLONEDHUMAN3H-HistamineWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47331D1CLONEDHUMAN3H-SCH23390WAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47332D2CLONEDHUMAN3H-NMSPWAY 100,635940Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47333D3CLONEDRAT3H-NMSPWAY 100,635370Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47334D4CLONEDHUMAN3H-NMSPWAY 100,63516.4Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47335D5CLONEDHUMAN3H-SCH23390WAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47336Alpha1ACLONEDHUMAN3H-PRAZOSINWAY 100,63519.9Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47337Alpha1BCLONEDHUMAN3H-PRAZOSINWAY 100,635322Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47338Alpha2ACLONEDHUMAN3H-CLONIDINEWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47339Alpha2BCLONEDHUMAN3H-CLONIDINEWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47340Alpha2CCLONEDHUMAN3H-CLONIDINEWAY 100,6352573Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47341Beta1CLONEDRAT125I-PindololWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47342Beta2CLONEDRAT125I-PindololWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 28, 2025
47343MORCLONEDHUMAN3H-QNBWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47344M2CLONEDHUMAN3H-QNBWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47345DORCLONEDHUMAN3H-QNBWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47346KORCLONEDHUMAN3H-QNBWAY 100,635412Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47347M5CLONEDHUMAN3H-QNBWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 15, 2025
47348KORFOREBRAINRAT3H-MUSCIMOLWAY 100,635>10000Chemel BR, et.al., 2006Jan 15, 2025Jan 27, 2025
47349GRIA1CLONEDHUMAN3H-AMPALY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47350GRIA1CLONEDHUMAN3H-AMPALY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47351GRIA1CLONEDHUMAN3H-AMPALY 2935589200Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47352GRIA2CLONEDHUMAN3H-AMPALY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47353GRIA2CLONEDHUMAN3H-AMPALY 4576915500Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47354GRIA2CLONEDHUMAN3H-AMPALY 4585458300Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47355GRIA2CLONEDHUMAN3H-AMPALY 294486>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47356GRIA2CLONEDHUMAN3H-AMPALY 302679820Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47357GRIA2CLONEDHUMAN3H-AMPALY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47358GRIA2CLONEDHUMAN3H-AMPALY 2935583200Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47359GRIA2CLONEDHUMAN3H-AMPALY 467711>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47360GRIA2CLONEDHUMAN3H-AMPALY 525327>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47361CLONEDHUMAN3H-AMPALY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47362CLONEDHUMAN3H-AMPALY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47363CLONEDHUMAN3H-AMPALY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47364GRIA4CLONEDHUMAN3H-AMPALY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47365GRIA4CLONEDHUMAN3H-AMPALY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47366GRIA4CLONEDHUMAN3H-AMPALY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47367Kainate receptorCLONEDHUMAN3H-Kainic acidLY 466195>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
47368Kainate receptorCLONEDHUMAN3H-Kainic acidLY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
47369Kainate receptorCLONEDHUMAN3H-Kainic acidLY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 28, 2025
47370Grik5CLONEDHUMAN3H-Kainic acidLY 46619550Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47371Grik5CLONEDHUMAN3H-Kainic acidLY 4576911550Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47372Grik5CLONEDHUMAN3H-Kainic acidLY 4585451690Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47373Grik5CLONEDHUMAN3H-Kainic acidLY 2944863060Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47374Grik5CLONEDHUMAN3H-Kainic acidLY 3026793410Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47375Grik5CLONEDHUMAN3H-Kainic acidLY 3828844000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47376Grik5CLONEDHUMAN3H-Kainic acidLY 2935584200Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47377Grik5CLONEDHUMAN3H-Kainic acidLY 4677117400Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47378Grik5CLONEDHUMAN3H-Kainic acidLY 525327>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47379CLONEDHUMAN3H-Kainic acidLY 4661958900Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47380CLONEDHUMAN3H-Kainic acidLY 382884>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
47381CLONEDHUMAN3H-Kainic acidLY 293558>10000Weiss B, et. al., 2006Jan 15, 2025Jan 15, 2025
473825-HT2BCLONEDHUMAN3H-5HTZiprasidone27.23PDSP Certified DataJan 15, 2025Jan 15, 2025
47383D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-Benzylpiperidin-4-yl)-1-naphthamide162Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
473845-HT2ACLONEDRAT3H-KETANSERINN-(1-Benzylpiperidin-4-yl)-1-naphthamide1000Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47385D2CLONEDHUMAN3H-SPIPERONEN-(1-Benzylpiperidin-4-yl)-1-naphthamide1000Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47386D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-Benzylpiperidin-4-yl)-2-naphthamide11Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
473875-HT2ACLONEDRAT3H-KETANSERINN-(1-Benzylpiperidin-4-yl)-2-naphthamide44Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47388D2CLONEDHUMAN3H-SPIPERONEN-(1-Benzylpiperidin-4-yl)-2-naphthamide1000Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47389D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-Phenylethylpiperidin-4-yl)-2-naphthamide139Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
473905-HT2ACLONEDRAT3H-KETANSERINN-(1-Phenylethylpiperidin-4-yl)-2-naphthamide42Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47391D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide29Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
473925-HT2ACLONEDRAT3H-KETANSERINN-(1-(1-Phenylethyl)piperidin-4-yl)-2-naphthamide110Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47393D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Phenylpropyl)piperidin-4-yl)-2-naphthamide63Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
473945-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Phenylpropyl)piperidin-4-yl)-2-naphthamide50Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47395D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Phenylbutyl)piperidin-4-yl)-2-naphthamide281Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
473965-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Phenylbutyl)piperidin-4-yl)-2-naphthamide213Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47397D4CLONEDHUMAN3H-NEMONAPRIDE(4-(Benzylamino)piperidin-1-yl)-(naphthalen-2-yl)methadone167Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47398D4CLONEDHUMAN3H-NEMONAPRIDENaphthalen-2-yl(4-(Phenylamino)piperidin-1-yl)methadone210Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47399D4CLONEDHUMAN3H-NEMONAPRIDENaphthalen-2-yl(4-(3-Phenylpropylamino)piperidin-1-yl)methadone222Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
47400D4CLONEDHUMAN3H-NEMONAPRIDEN-(2-Phenylethylpiperidin-4-yl)-1-naphthamide230Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
474015-HT2ACLONEDRAT3H-KETANSERINN-(2-Phenylethylpiperidin-4-yl)-1-naphthamide543Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
474025-HT2ACLONEDRAT3H-KETANSERINN-(1-Phenylethylpiperidin-4-yl)-1-naphthamide248Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47403D4CLONEDHUMAN3H-NEMONAPRIDEN-(3-Phenylpropylpiperidin-4-yl)-1-naphthamide71Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
474045-HT2ACLONEDRAT3H-KETANSERINN-(3-Phenylpropylpiperidin-4-yl)-1-naphthamide228Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
474055-HT2ACLONEDRAT3H-KETANSERINN-((S)-3-(1-hydroxy-1-phenyl)propylpiperidin-4-yl)-1-naphthamide390Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47406D4CLONEDHUMAN3H-NEMONAPRIDEN-(4-Phenylbutylpiperidin-4-yl)-1-naphthamide362Carato P, et al., 2007Jan 15, 2025Jan 27, 2025
474075-HT2ACLONEDRAT3H-KETANSERINN-(4-Phenylbutylpiperidin-4-yl)-1-naphthamide487Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
474085-HT2ACLONEDRAT3H-KETANSERINN-(2-Phenylethylpiperidin-4-yl)-1-naphthamide211Carato P, et al., 2007Jan 15, 2025Jan 15, 2025
47409D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(2-Cl-benzyl)-piperidin-4-yl)-1-naphthamide329Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47410D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Cl-benzyl)-piperidin-4-yl)-1-naphthamide116Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47411D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-Cl-benzyl)-piperidin-4-yl)-1-naphthamide43Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47412D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Br-benzyl)-piperidin-4-yl)-1-naphthamide66Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474135-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Br-benzyl)-piperidin-4-yl)-1-naphthamide462Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47414D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-Br-benzyl)-piperidin-4-yl)-1-naphthamide44Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47415D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-CF3-benzyl)-piperidin-4-yl)-1-naphthamide119Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47416D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-CF3-benzyl)-piperidin-4-yl)-1-naphthamide96Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474175-HT2ACLONEDRAT3H-KETANSERINN-(1-(2,3,4,5,6-F-benzyl)-piperidin-4-yl)-1-naphthamide228Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47418D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-MeO-benzyl)-piperidin-4-yl)-1-naphthamide168Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47419D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-MeO-benzyl)-piperidin-4-yl)-1-naphthamide223Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47420D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(2-Me-benzyl)-piperidin-4-yl)-1-naphthamide155Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47421D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Me-benzyl)-piperidin-4-yl)-1-naphthamide77Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47422D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-Me-benzyl)-piperidin-4-yl)-1-naphthamide69Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474235-HT2ACLONEDRAT3H-KETANSERINN-(1-(2-Cl-benzyl)-piperidin-4-yl)-2-naphthamide133Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
474245-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Cl-benzyl)-piperidin-4-yl)-2-naphthamide133Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47425D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Cl-benzyl)-piperidin-4-yl)-2-naphthamide54Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47426D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-Cl-benzyl)-piperidin-4-yl)-2-naphthamide37Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474275-HT2ACLONEDRAT3H-KETANSERINN-(1-(4-Cl-benzyl)-piperidin-4-yl)-2-naphthamide242Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47428D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Br-benzyl)-piperidin-4-yl)-2-naphthamide36Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474295-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Br-benzyl)-piperidin-4-yl)-2-naphthamide53Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47430D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-Br-benzyl)-piperidin-4-yl)-2-naphthamide34Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474315-HT2ACLONEDRAT3H-KETANSERINN-(1-(4-Br-benzyl)-piperidin-4-yl)-2-naphthamide223Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47432D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-CF3-benzyl)-piperidin-4-yl)-2-naphthamide103Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47433D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-CF3-benzyl)-piperidin-4-yl)-2-naphthamide84Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
47434D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-NO2-benzyl)-piperidin-4-yl)-2-naphthamide181Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474355-HT2ACLONEDRAT3H-KETANSERINN-(1-(4-NO2-benzyl)-piperidin-4-yl)-2-naphthamide278Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47436D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-MeO-benzyl)-piperidin-4-yl)-2-naphthamide16Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474375-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-MeO-benzyl)-piperidin-4-yl)-2-naphthamide158Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47438D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-MeO-benzyl)-piperidin-4-yl)-2-naphthamide31Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474395-HT2ACLONEDRAT3H-KETANSERINN-(1-(4-MeO-benzyl)-piperidin-4-yl)-2-naphthamide151Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47440D4CLONEDHUMAN3H-NEMONAPRIDEN-(2-(2-Me-benzyl)-piperidin-4-yl)-2-naphthamide26Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474415-HT2ACLONEDRAT3H-KETANSERINN-(1-(2-Me-benzyl)-piperidin-4-yl)-2-naphthamide175Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47442D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Me-benzyl)-piperidin-4-yl)-2-naphthamide11Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474435-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Me-benzyl)-piperidin-4-yl)-2-naphthamide87Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47444D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(4-Me-benzyl)-piperidin-4-yl)-2-naphthamide21Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474455-HT2ACLONEDRAT3H-KETANSERINN-(1-(4-Me-benzyl)-piperidin-4-yl)-2-naphthamide222Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47446D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(2-Pyridyl)-piperidin-4-yl)-2-naphthamide299Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474475-HT2ACLONEDRAT3H-KETANSERINN-(1-(2-Pyridyl)-piperidin-4-yl)-2-naphthamide545Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47448D4CLONEDHUMAN3H-NEMONAPRIDEN-(1-(3-Pyridyl)-piperidin-4-yl)-2-naphthamide326Carato P, et al., 2007aJan 15, 2025Jan 27, 2025
474495-HT2ACLONEDRAT3H-KETANSERINN-(1-(3-Pyridyl)-piperidin-4-yl)-2-naphthamide524Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
474505-HT2ACLONEDRAT3H-KETANSERINN-(1-(4-Pyridyl)-piperidin-4-yl)-2-naphthamide695Carato P, et al., 2007aJan 15, 2025Jan 15, 2025
47451CLONEDHUMANFunctional5-(4-Aminophenyl)-6-methylthieno[2,3-d]pyrimidin-4-amine4600Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47452CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-3-methylbenzamide4600Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47453CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]benzenesulfonamide>10000Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47454CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-phenylurea36Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47455CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea6Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47456CLONEDHUMANFunctional4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)-N-phenylbenzamide>10000Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47457CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)thiourea2800Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47458CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N' '-cyano-N'-(3-methylphenyl)guanidine1100Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47459CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-1H-indole-2-carboxamide>10000Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47460CLONEDHUMANFunctional5-[4-(1,3-Benzoxazol-2-ylamino)phenyl]-6-methylthieno[2,3-d]pyrimidin-4-amine170Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47461CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-2-(3-methylphenyl)acetamide760Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47462CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N-methyl-N'-(3-methylphenyl)urea55Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47463CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-methyl-N'-(3-methylphenyl)urea1900Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47464CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-benzylurea330Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47465CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-cyclohexylmethylurea790Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47466CLONEDHUMANFunctionalN-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea26Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47467CLONEDHUMANFunctionalN-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-cyclohexylurea170Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47468CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea3Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47469CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-butylurea180Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47470CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-isobutylurea1700Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47471CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-methylphenyl)urea260Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47472CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-methylphenyl)urea53Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47473CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-methoxyphenyl)urea110Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47474CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methoxyphenyl)urea34Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47475CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-methoxyphenyl)urea69Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47476CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-fluorophenyl)urea110Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47477CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-fluorophenyl)urea54Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47478CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-fluorophenyl)urea52Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47479CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-chlorophenyl)urea340Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47480CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-chlorophenyl)urea35Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47481CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-chlorophenyl)urea96Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47482CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-bromophenyl)urea46Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47483CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(4-bromophenyl)urea120Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47484CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea52Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47485CLONEDHUMANFunctionalMethyl 3-[({[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]amino}carbonyl)amino]benzoate290Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47486CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3,5-dimethylphenyl)urea12Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47487CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3,5-dichlorophenyl)urea160Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47488CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[2-fluoro-5-(trifluoromethyl)phenyl]urea45Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47489CLONEDHUMANFunctional3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}propanamide17Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47490CLONEDHUMANFunctional3-{4-Amino-5-[4-({[(3-methylphenyl)amino]carbonyl}amino)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N-methylpropanamide330Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47491CLONEDHUMANFunctional3-{4-Amino-5-[4-(3-m-tolylureido)phenyl]thieno[2,3-d]pyrimidin-6-yl}-N,N-dimethylpropionamide210Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47492CLONEDHUMANFunctionalN-{4-[4-Amino-6-(morpholin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea210Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47493CLONEDHUMANFunctionalN-(4-{4-Amino-6-[(4-methylpiperazin-1-yl)methyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea590Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47494CLONEDHUMANFunctionalN-(4-{4-Amino-6-[(dimethylamino)methyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea180Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47495CLONEDHUMANFunctionalN-[4-(4-Amino-6-propylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea26Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47496CLONEDHUMANFunctionalN-[4-(4-Amino-6-isopropylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea130Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47497CLONEDHUMANFunctionalN-[4-(4-Amino-6-benzylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-methylphenyl)urea280Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47498CLONEDHUMANFunctionalN-{4-[4-Amino-6-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea34Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47499CLONEDHUMANFunctionalN-{4-[4-Amino-6-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea53Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47500CLONEDHUMANFunctionalN-{4-[4-Amino-6-(2-hydroxyethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea19Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47501CLONEDHUMANFunctionalN-{4-[4-Amino-6-(2-methoxyethyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea64Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47502CLONEDHUMANFunctionalN-{4-[4-Amino-6-(3-hydroxypropyl)thieno[2,3-d]pyrimidin-5-yl]phenyl}-N'-(3-methylphenyl)urea15Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47503CLONEDHUMANFunctionalN-(4-{4-Amino-6-[2-(dimethylamino)ethyl]thieno[2,3-d]pyrimidin-5-yl}phenyl)-N'-(3-methylphenyl)urea230Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47504CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-fluorophenyl]-N'-(3-methylphenyl)urea19Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47505CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-chlorophenyl]-N'-(3-methylphenyl)urea83Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47506CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)-2-methoxyphenyl]-N'-(3-methylphenyl)urea13Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47507CLONEDHUMANFunctionalN-(11-Amino-5,6-dihydro-7-thia-8,10-diazabenzo[c]fluoren-3-yl)-N'-(3-methylphenyl)urea150Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47508CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[4-(trifluoromethyl)phenyl]urea61Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47509CLONEDHUMANFunctionalN-[4-(4-Amino-6-methylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(2-fluoro-5-methylphenyl)urea34Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47510CLONEDHUMANFunctionalN-[4-(4-Amino-6-ethylthieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-[3-(trifluoromethyl)phenyl]urea50Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47511CLONEDHUMANFunctionalN-[4-(4-Aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-N'-(3-chlorophenyl)urea3Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47512CLONEDHUMANFunctionalSU1124818Dai Y, et al., 2005Jan 15, 2025Jan 15, 2025
47513Y1BRAINRAT125I-[Leu31,Pro34]PYYPYY,[leu31,Pro34], human0.05Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47514Y1BRAINRAT125I-[Leu31,Pro34]PYYPP, human0.08Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47515Y1BRAINRAT125I-[Leu31,Pro34]PYYPP, rat92Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47516Y1BRAINRAT125I-[Leu31,Pro34]PYYGR2311184.3Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47517Y1BRAINRAT125I-[Leu31,Pro34]PYYNPY [Ala31, Aib32], porcine2.5Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47518Y1BRAINRAT125I-[Leu31,Pro34]PYYNPY [hPP(1-17), Ala31,Aib32], human0.5Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47519Y1BRAINRAT125I-[Leu31,Pro34]PYYPP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human0.1Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47520Y1BRAINRAT125I-[Leu31,Pro34]PYYCGP71683A1.3Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47521Y1BRAINRAT125I-[Leu31,Pro34]PYYJCF1099.2Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47522Y1BRAINRAT125I-[Leu31,Pro34]PYYCP7329251.6Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47523Y1BRAINRAT125I-[Leu31,Pro34]PYYCP7605242.6Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47524Y1BRAINRAT125I-[Leu31,Pro34]PYYCP7812144.2Dumont Y, et al., 2005Jan 15, 2025Jan 15, 2025
47525EAAT2CLONEDHUMAN3H-GLUTAMATEWAY 21361385Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47526EAAT2CLONEDHUMAN3H-GLUTAMATEWAY 213394145Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47527EAAT2CLONEDHUMAN3H-GLUTAMATEWAY 212922157Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47528EAAT2CLONEDHUMAN3H-GLUTAMATEWAY 211686190Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47529EAAT1CLONEDHUMAN3H-GLUTAMATEWAY 2136135004Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47530EAAT1CLONEDHUMAN3H-GLUTAMATEWAY 2133941971Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47531EAAT1CLONEDHUMAN3H-GLUTAMATEWAY 2129223426Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47532EAAT1CLONEDHUMAN3H-GLUTAMATEWAY 2116861681Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47533EAAT3CLONEDHUMAN3H-GLUTAMATEWAY 2136133787Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47534EAAT3CLONEDHUMAN3H-GLUTAMATEWAY 2133946561Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47535EAAT3CLONEDHUMAN3H-GLUTAMATEWAY 2116861453Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47536EAAT3CLONEDHUMAN3H-GLUTAMATEWAY 2129221837Dunlop J, et al., 2005Jan 15, 2025Jan 15, 2025
47537L1210 cellsUNDEFINEDFunctional(anthracen-9-ylmethyl)-3,3-triamine1800Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47538L1210 cellsUNDEFINEDFunctional(anthracen-9-ylmethyl)-4,4-triamine300Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47539L1210 cellsUNDEFINEDFunctionalN1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt3000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47540L1210 cellsUNDEFINEDFunctionalN1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47541L1210 cellsUNDEFINEDFunctionalN-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47542L1210 cellsUNDEFINED14C-spermidine(anthracen-9-ylmethyl)-3,3-triamine>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47543L1210 cellsUNDEFINED14C-spermidine(anthracen-9-ylmethyl)-4,4-triamine1800Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47544L1210 cellsUNDEFINED14C-spermidineN1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt9900Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47545L1210 cellsUNDEFINED14C-spermidineN1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt6200Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47546L1210 cellsUNDEFINED14C-spermidineN-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47547CLONEDUNDEFINEDFunctional(anthracen-9-ylmethyl)-3,3-triamine1900Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47548CLONEDUNDEFINEDFunctional(anthracen-9-ylmethyl)-4,4-triamine450Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47549CLONEDUNDEFINEDFunctionalN1-[3-(Azacyclopentadec-1-yl)propyl]propane-1,3-diamine Hydrochloride Salt>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47550CLONEDUNDEFINEDFunctionalN1-[4-(Azacyclopentadec-1-yl)butyl]butane-1,4-diamine Hydrochloride Salt>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47551CLONEDUNDEFINEDFunctionalN-(4-Aminobutyl)-N'-anthracen-9-ylmethyl-N'-ethylbutane-1,4-diamine Hydrochloride Salt>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
47552BRAINRAT3H-3-PPP,(+)PHENTOLAMINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47553BRAINRAT3H-3-PPP,(+)IPRINDOLE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47554BRAINRAT3H-3-PPP,(+)Amphetamine,(+)>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47555BRAINRAT3H-3-PPP,(+)COCAINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47556BRAINRAT3H-3-PPP,(+)Levorphanol>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47557BRAINRAT3H-3-PPP,(+)Bradykinin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47558BRAINRAT3H-3-PPP,(+)CCK33>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47559BRAINRAT3H-3-PPP,(+)DOPAMINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47560BRAINRAT3H-3-PPP,(+)APOMORPHINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47561BRAINRAT3H-3-PPP,(+)LISURIDE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47562BRAINRAT3H-3-PPP,(+)NALOXONE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47563BRAINRAT3H-3-PPP,(+)DIHYDROMORPHINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47564BRAINRAT3H-3-PPP,(+)[D-Ala2-D-Leu5]enkephalin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47565BRAINRAT3H-3-PPP,(+)Alpha-Neoendorphin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47566BRAINRAT3H-3-PPP,(+)Beta-Neoendorphin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47567BRAINRAT3H-3-PPP,(+)HEXAMETHONIUM>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47568BRAINRAT3H-3-PPP,(+)Decamethonium>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47569BRAINRAT3H-3-PPP,(+)SCOPOLAMINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47570BRAINRAT3H-3-PPP,(+)RAUWOLSCINE>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47571BRAINRAT3H-3-PPP,(+)Picrotoxin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47572BRAINRAT3H-3-PPP,(+)Bicuculline>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47573BRAINRAT3H-3-PPP,(+)Gamma-Aminobutyric acid>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47574BRAINRAT3H-3-PPP,(+)amrinone>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47575BRAINRAT3H-3-PPP,(+)tetrodotoxin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47576BRAINRAT3H-3-PPP,(+)LYSERGIC ACID>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47577BRAINRAT3H-3-PPP,(+)Cannabinol>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47578BRAINRAT3H-3-PPP,(+)THC, delta 9>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47579BRAINRAT3H-3-PPP,(+)Angiotensin II>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47580BRAINRAT3H-3-PPP,(+)Neurotensin>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47581BRAINRAT3H-3-PPP,(+)CCK4>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47582BRAINRAT3H-3-PPP,(+)CCK8>10000Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
47583PKCαCLONEDHUMAN3H-PDBU(Z)-CH2OCOC(CH3)3 2.9Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47584PKCαCLONEDHUMAN3H-PDBU(E)-CH2OCOC(CH3)3 4.51Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47585PKCαCLONEDHUMAN3H-PDBUCH2OCOC(CH3)3 1.45Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47586PKCαCLONEDHUMAN3H-PDBU5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone3.78Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47587PKCαCLONEDHUMAN3H-PDBU5-Hexanoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone6.18Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47588PKCαCLONEDHUMAN3H-PDBU5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone4.97Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47589PKCαCLONEDHUMAN3H-PDBU5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-octanoyloxymethyltetrahydro-2-furanone6.04Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47590PKCαCLONEDHUMAN3H-PDBU5-Benzoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone6.66Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47591PKCαCLONEDHUMAN3H-PDBU5-Benzoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone16.1Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47592PKCαCLONEDHUMAN3H-PDBU5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone6.87Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47593PKCαCLONEDHUMAN3H-PDBU5-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-5-(3-isopropyl-4-methyl-pentanoyloxymethyl)tetrahydro-2-furanone4.46Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47594PKCαCLONEDHUMAN3H-PDBU5-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-5-(3-isobutyl-5-methyl-hexanoyloxymethyl)tetrahydro-2-furanone6.88Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47595PKCαCLONEDHUMAN3H-PDBU5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(Z)-3-isobutyl-5 -methylhexylidene]tetrahydro-2-furanone18Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47596PKCαCLONEDHUMAN3H-PDBU5-[(E)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone173Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47597PKCαCLONEDHUMAN3H-PDBU5-[(Z)-3-(tert-Butoxy)-3-oxo-1-propenyl]-5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]tetrahydro-2-furanone>10000Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47598PKCαCLONEDHUMAN3H-PDBU5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methyl-2-butenyl)dihydro-2(3H)-furanone2100Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47599PKCαCLONEDHUMAN3H-PDBU5-(Hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-methylbutyl)dihydro-2(3H)-furanone>10000Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47600PKCαCLONEDHUMAN3H-PDBU6-Hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone28Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47601PKCαCLONEDHUMAN3H-PDBU6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-pivaloyloxymethyl-tetrahydro-2-pyranone48Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47602PKCαCLONEDHUMAN3H-PDBU6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-hexanoyloxymethyl-tetrahydro-2-pyranone147Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47603PKCαCLONEDHUMAN3H-PDBU6-Hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylidene]-6-octanoyloxymethyl-tetrahydro-2-pyranone129Lee J, et al., 2006Jan 15, 2025Jan 15, 2025
47604ADKrecombinantHUMANFunctional4-N-Phenylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine100Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47605ADKrecombinantHUMANFunctional4-N-Benzylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine800Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47606ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine550Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47607ADKrecombinantHUMANFunctional4-N-(4-Methoxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine775Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47608ADKrecombinantHUMANFunctional4-N-(4-Hydroxyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine200Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47609ADKrecombinantHUMANFunctional4-N-Cyclohexylamino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine>10000Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47610ADKrecombinantHUMANFunctional4-N-(Cyanoyphenyl)amino-5-iodo-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine1200Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47611ADKrecombinantHUMANFunctional4-N-Phenylamino-5-iodo-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine120Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47612ADKrecombinantHUMANFunctional4-N-Phenylamino-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine1250Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47613ADKrecombinantHUMANFunctional4-Amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine320Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025
47614ADKrecombinantHUMANFunctional4-N-Phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine0.5Ugarkar BG, et al., 2000Jan 15, 2025Jan 15, 2025