73749 5-HT7 ?CLONED ? HUMAN 3H- LSD {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73750 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73751 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73752 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73753 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 1008 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73754 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73755 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73756 Beta 1 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73757 Beta3 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73758 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73759 D1 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73760 D5 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73761 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73762 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73763 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73764 SERT ?CLONED ? HUMAN 3H-CITALOPRAM {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 1550 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73765 NET ?CLONED ? HUMAN 3H-Nisoxetine {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73766 DAT ?CLONED ? HUMAN [3H] WIN35428 {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73767 H1 ?CLONED ? HUMAN 3H-PYRILAMINE {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73768 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73769 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73770 H4 ?CLONED ? HUMAN 3H-Histamine {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73771 M1 ?CLONED ? HUMAN 3H-QNB {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73772 M2 ?CLONED ? HUMAN 3H-QNB {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73773 M3 ?CLONED ? HUMAN 3H-QNB {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73774 M4 ?CLONED ? HUMAN 3H-QNB {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73775 M5 ?CLONED ? HUMAN 3H-QNB {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73776 MOR ?CLONED ? HUMAN 3H-DAMGO {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73777 DOR ?CLONED ? HUMAN 3H-DADLE {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73778 KOR ?CLONED ? HUMAN 3H-U69593 {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73779 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 1574 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73780 Sigma 2 ?CLONED RODENT 3H-DTG 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 410 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73781 PBR KIDNEY RODENT 3H-PK11195 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73782 BZP BRAIN RODENT FNZ 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
73783 5-HT1A ?CLONED ? HUMAN [3H] Way100635 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73784 5-HT1B ?CLONED ? HUMAN 3H-GR125743 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73785 5-HT1D ?CLONED ? HUMAN 3H-GR125743 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73786 5-HT1E ?CLONED ? HUMAN 3H-5-HT 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73787 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73788 5-HT2B ?CLONED ? HUMAN 3H- LSD 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 969 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73789 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73790 5-HT3 ?CLONED ? HUMAN 3H-LY278584 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate 671 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73791 5-HT5A ?CLONED ? HUMAN 3H-LSD 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73792 5-HT6 ?CLONED ? HUMAN 3H-LSD 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73793 5-HT7 ?CLONED ? HUMAN 3H-LSD 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73794 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73795 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73796 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73797 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73798 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73799 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73800 Beta 1 ?CLONED ? HUMAN 125I-Pindolol 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73801 Beta3 ?CLONED ? HUMAN 125I-Pindolol 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73802 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73803 D1 ?CLONED ? HUMAN 3H-SCH23390 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73804 D5 ?CLONED ? HUMAN 3H-SCH23390 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73805 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73806 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73807 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73808 SERT ?CLONED ? HUMAN 3H-CITALOPRAM 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73809 NET ?CLONED ? HUMAN 3H-Nisoxetine 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73810 DAT ?CLONED ? HUMAN 3H-WIN35428 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73811 H1 ?CLONED ? HUMAN 3H-PYRILAMINE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73812 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73813 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73814 H4 ?CLONED ? HUMAN 3H-Histamine 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73815 M1 ?CLONED ? HUMAN 3H-QNB 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73816 M2 ?CLONED ? HUMAN 3H-QNB 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73817 M3 ?CLONED ? HUMAN 3H-QNB 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73818 M4 ?CLONED ? HUMAN 3H-QNB 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73819 M5 ?CLONED ? HUMAN 3H-QNB 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73820 MOR ?CLONED ? HUMAN 3H-DAMGO 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73821 KOR ?CLONED ? HUMAN 3H-U69593 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73822 DOR ?CLONED ? HUMAN 3H-DADLE 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73823 Sigma 2 ?CLONED RODENT 3H-DTG {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 40 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73824 5-HT1A ?CLONED ? HUMAN [3H] Way100635 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73825 5-HT1B ?CLONED ? HUMAN 3H-GR125743 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73826 5-HT1D ?CLONED ? HUMAN 3H-GR125743 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73827 5-HT1E ?CLONED ? HUMAN 3H-5HT {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73828 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73829 5-HT2B ?CLONED ? HUMAN 3H- LSD {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 68 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73830 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 820 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73831 5-HT3 ?CLONED ? HUMAN 3H-LY278584 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73832 5-HT5A ?CLONED ? HUMAN 3H-LSD {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73833 5-HT6 ?CLONED ? HUMAN 3H-LSD {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73834 5-HT7 ?CLONED ? HUMAN 3H- LSD {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 697 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73835 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73836 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73837 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73838 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 834 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73839 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 510 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73840 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 1379 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73841 Beta 1 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73842 Beta3 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73843 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73844 D1 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73845 D5 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73846 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73847 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73848 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73849 SERT ?CLONED ? HUMAN 3H-CITALOPRAM {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 1213 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73850 NET ?CLONED ? HUMAN 3H-Nisoxetine {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73851 DAT ?CLONED ? HUMAN 3H-WIN35428 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73852 H1 ?CLONED ? HUMAN 3H-PYRILAMINE {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73853 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 1769 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73854 H4 ?CLONED ? HUMAN 3H-Histamine {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73855 M1 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73856 M2 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73857 M3 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73858 M4 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73859 M5 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73860 MOR ?CLONED ? HUMAN 3H-DAMGO {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73861 KOR ?CLONED ? HUMAN 3H-U69593 {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73862 DOR ?CLONED ? HUMAN 3H-DADLE {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73863 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate 0.5 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73864 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 0.8 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73865 Sigma 2 ?CLONED RODENT 3H-DTG {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 47 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73866 5-HT1A ?CLONED ? HUMAN [3H] Way100635 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73867 5-HT1B ?CLONED ? HUMAN 3H-GR125743 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73868 5-HT1D ?CLONED ? HUMAN 3H-GR125743 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73869 5-HT1E ?CLONED ? HUMAN 3H-5-HT {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73870 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73871 5-HT2B ?CLONED ? HUMAN 3H-LSD {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 86 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73872 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 764 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73873 5-HT3 ?CLONED ? HUMAN 3H-LY278584 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73874 5-HT5A ?CLONED ? HUMAN 3H-LSD {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73875 5-HT6 ?CLONED ? HUMAN 3H-LSD {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73876 5-HT7 ?CLONED ? HUMAN 3H-LSD {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73877 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73878 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73879 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73880 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73881 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73882 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73883 Beta 1 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73884 Beta3 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73885 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73886 D1 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73887 D5 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73888 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73889 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73890 D4 ?CLONED ? HUMAN 3H-N-Methylspiporone {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73891 SERT ?CLONED ? HUMAN 3H-CITALOPRAM {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73892 NET ?CLONED ? HUMAN 3H-Nisoxetine {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73893 DAT ?CLONED ? HUMAN [3H] WIN35428 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73894 H1 ?CLONED ? HUMAN 3H-PYRILAMINE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73895 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate 542 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73896 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73897 M1 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73898 M2 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73899 M3 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73900 M4 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73901 M5 ?CLONED ? HUMAN 3H-QNB {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73902 MOR ?CLONED ? HUMAN 3H-DAMGO {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73903 KOR ?CLONED ? HUMAN 3H-U69593 {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73904 DOR ?CLONED ? HUMAN 3H-DADLE {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73905 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73906 Sigma 2 ?CLONED RODENT 3H-DTG {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 17 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73907 5-HT1A ?CLONED ? HUMAN [3H] Way100635 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73908 5-HT1B ?CLONED ? HUMAN 3H-GR125743 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73909 5-HT1D ?CLONED ? HUMAN 3H-GR125743 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73910 5-HT1E ?CLONED ? HUMAN 3H-5-HT {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73911 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1663 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73912 5-HT2B ?CLONED ? HUMAN 3H- LSD {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 90 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73913 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 916 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73914 5-HT3 ?CLONED ? HUMAN 3H-LY278584 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73915 5-HT5A ?CLONED ? HUMAN 3H- LSD {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73916 5-HT6 ?CLONED ? HUMAN 3H- LSD {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73917 5-HT7 ?CLONED ? HUMAN 3H- LSD {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 255 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73918 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73919 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73920 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73921 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1077 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73922 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1390 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73923 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1560 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73924 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73925 Beta 1 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73926 Beta3 ?CLONED ? HUMAN 125I-Pindolol {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73927 D1 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73928 D5 ?CLONED ? HUMAN 3H-SCH23390 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73929 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73930 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73931 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 2591 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73932 SERT ?CLONED ? HUMAN 3H-CITALOPRAM {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 764 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73933 NET ?CLONED ? HUMAN 3H-Nisoxetine {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 3094 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73934 DAT ?CLONED ? HUMAN [3H] WIN35428 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73935 H1 ?CLONED ? HUMAN 3H-PYRILAMINE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73936 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 729 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73937 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1174 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73938 H4 ?CLONED ? HUMAN 3H-Histamine {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate 1702 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73939 M1 ?CLONED ? HUMAN 3H-QNB {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73940 M2 ?CLONED ? HUMAN 3H-QNB {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73941 M3 ?CLONED ? HUMAN 3H-QNB {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73942 M4 ?CLONED ? HUMAN 3H-QNB {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73943 MOR ?CLONED ? HUMAN 3H-DAMGO {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73944 DOR ?CLONED ? HUMAN 3H-DADLE {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73945 KOR ?CLONED ? HUMAN 3H-U69593 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73946 PBR KIDNEY RODENT 3H-PK11195 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73947 BZP BRAIN RODENT 3H-PK11195 {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
73948 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 67 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73949 Sigma 2 ?CLONED RODENT 3H-DTG 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 136 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73950 PBR KIDNEY RODENT 3H-PK11195 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73951 BZP BRAIN RODENT FNZ 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
73952 5-HT1A ?CLONED ? HUMAN [3H] Way100635 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73953 5-HT1B ?CLONED ? HUMAN 3H-GR125743 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73954 5-HT1D ?CLONED ? HUMAN 3H-GR125743 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73955 5-HT1E ?CLONED ? HUMAN 3H-5-HT 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73956 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73957 5-HT2B ?CLONED ? HUMAN 3H- LSD 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 416 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73958 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73959 5-HT3 ?CLONED ? HUMAN 3H-LY278584 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73960 5-HT5A ?CLONED ? HUMAN 3H- LSD 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73961 5-HT6 ?CLONED ? HUMAN 3H- LSD 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73962 5-HT7 ?CLONED ? HUMAN 3H- LSD 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73963 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 1695 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73964 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 2196 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73965 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73966 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73967 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73968 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 1073 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73969 Beta 1 ?CLONED ? HUMAN 125I-Pindolol 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73970 Beta3 ?CLONED ? HUMAN 125I-Pindolol 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73971 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73972 D1 ?CLONED ? HUMAN 3H-SCH23390 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73973 D5 ?CLONED ? HUMAN 3H-SCH23390 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73974 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73975 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 3372 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73976 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 416 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73977 SERT ?CLONED ? HUMAN 3H-CITALOPRAM 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73978 NET ?CLONED ? HUMAN 3H-Nisoxetine 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73979 DAT ?CLONED ? HUMAN [3H] WIN35428 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73980 H1 ?CLONED ? HUMAN 3H-PYRILAMINE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride 644 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73981 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73982 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73983 H4 ?CLONED ? HUMAN 3H-Histamine 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73984 M1 ?CLONED ? HUMAN 3H-QNB 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73985 M2 ?CLONED ? HUMAN 3H-QNB 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73986 M3 ?CLONED ? HUMAN 3H-QNB 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73987 M4 ?CLONED ? HUMAN 3H-QNB 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73988 M5 ?CLONED ? HUMAN 3H-QNB 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73989 MOR ?CLONED ? HUMAN 3H-DAMGO 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73990 DOR ?CLONED ? HUMAN 3H-DADLE 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73991 KOR ?CLONED ? HUMAN 3H-U69593 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73992 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 171 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73993 Sigma 2 ?CLONED RODENT 3H-DTG 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 19 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
73994 PBR KIDNEY RODENT 3H-PK11195 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73995 BZP BRAIN RODENT FNZ 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
73996 5-HT1A ?CLONED ? HUMAN [3H] Way100635 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 348 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73997 5-HT1B ?CLONED ? HUMAN 3H-GR125743 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73998 5-HT1D ?CLONED ? HUMAN 3H-GR125743 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 2307 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
73999 5-HT1E ?CLONED ? HUMAN 3H-5-HT 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74000 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 814 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74001 5-HT2B ?CLONED ? HUMAN 3H- LSD 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 412 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74002 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 113 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74003 5-HT3 ?CLONED ? HUMAN 3H-LY278584 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 241 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74004 5-HT5A ?CLONED ? HUMAN 3H- LSD 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74005 5-HT6 ?CLONED ? HUMAN 3H- LSD 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74006 5-HT7 ?CLONED ? HUMAN 3H- LSD 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 161 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74007 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 60 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74008 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 707.5 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74009 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 41 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74010 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 792 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74011 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 387 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74012 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 868 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74013 Beta 1 ?CLONED ? HUMAN 125I-Pindolol 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 957 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74014 Beta3 ?CLONED ? HUMAN 125I-Pindolol 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 1014 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74015 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 752 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74016 D1 ?CLONED ? HUMAN 3H-SCH23390 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74017 D5 ?CLONED ? HUMAN 3H-SCH23390 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74018 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 1359 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74019 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 1157 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74020 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 94 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74021 SERT ?CLONED ? HUMAN 3H-CITALOPRAM 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 1181 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74022 NET ?CLONED ? HUMAN 3H-Nisoxetine 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 2359 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74023 DAT ?CLONED ? HUMAN [3H] WIN35428 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74024 H1 ?CLONED ? HUMAN 3H-PYRILAMINE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 145 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74025 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 5058 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74026 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74027 H4 ?CLONED ? HUMAN 3H-Histamine 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74028 M1 ?CLONED ? HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74029 M2 ?CLONED ? HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74030 M3 ?CLONED ? HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74031 M4 ?CLONED ? HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74032 M5 ?CLONED ? HUMAN 3H-QNB 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74033 MOR ?CLONED ? HUMAN 3H-DAMGO 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride 2351.5 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74034 KOR ?CLONED ? HUMAN 3H-U69593 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74035 DOR ?CLONED ? HUMAN 3H-DADLE 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74036 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 34 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74037 Sigma 2 ?CLONED RODENT 3H-DTG 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 119 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74038 PBR KIDNEY RODENT 3H-PK11195 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74039 BZP BRAIN RODENT FNZ 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74040 5-HT1A ?CLONED ? HUMAN [3H] Way100635 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 58 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74041 5-HT1B ?CLONED ? HUMAN 3H-GR125743 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74042 5-HT1D ?CLONED ? HUMAN 3H-GR125743 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 4549 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74043 5-HT1E ?CLONED ? HUMAN 3H-5-HT 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74044 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 135 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74045 5-HT2B ?CLONED ? HUMAN 3H- LSD 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74046 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 490 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74047 5-HT3 ?CLONED ? HUMAN 3H-LY278584 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74048 5-HT5A ?CLONED ? HUMAN 3H- LSD 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74049 5-HT6 ?CLONED ? HUMAN 3H- LSD 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74050 5-HT7 ?CLONED ? HUMAN 3H-LSD 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 82 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74051 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 336 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74052 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 501 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74053 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 1022 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74054 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 2902 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74055 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 409 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74056 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 467 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74057 Beta 1 ?CLONED ? HUMAN 125I-Pindolol 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74058 Beta3 ?CLONED ? HUMAN 125I-Pindolol 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74059 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74060 D1 ?CLONED ? HUMAN 3H-SCH23390 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74061 D5 ?CLONED ? HUMAN 3H-SCH23390 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74062 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74063 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 425 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74064 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 222 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74065 SERT ?CLONED ? HUMAN 3H-CITALOPRAM 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 2112 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74066 NET ?CLONED ? HUMAN 3H-Nisoxetine 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 1249 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74067 DAT ?CLONED ? HUMAN [3H] WIN35428 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 1762.5 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74068 H1 ?CLONED ? HUMAN 3H-PYRILAMINE 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride 304 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74069 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74070 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74071 H4 ?CLONED ? HUMAN 3H-Histamine 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74072 M1 ?CLONED ? HUMAN 3H-QNB 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74073 M2 ?CLONED ? HUMAN 3H-QNB 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74074 M3 ?CLONED ? HUMAN 3H-QNB 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74075 M4 ?CLONED ? HUMAN 3H-QNB 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74076 M5 ?CLONED ? HUMAN 3H-QNB 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74077 MOR ?CLONED ? HUMAN 3H-DAMGO 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74078 DOR ?CLONED ? HUMAN 3H-DADLE 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74079 KOR ?CLONED ? HUMAN 3H-U69593 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74080 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 620 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74081 Sigma 2 ?CLONED RODENT 3H-DTG 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 235 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74082 PBR KIDNEY RODENT 3H-PK11195 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74083 BZP BRAIN RODENT FNZ 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74084 5-HT1A ?CLONED ? HUMAN [3H] Way100635 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 4.7 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74085 5-HT1B ?CLONED ? HUMAN 3H-GR125743 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74086 5-HT1D ?CLONED ? HUMAN 3H-GR125743 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74087 5-HT1E ?CLONED ? HUMAN 3H-5-HT 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74088 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74089 5-HT2B ?CLONED ? HUMAN 3H- LSD 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 248 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74090 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74091 5-HT3 ?CLONED ? HUMAN 3H-LY278584 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74092 5-HT5A ?CLONED ? HUMAN 3H- LSD 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74093 5-HT6 ?CLONED ? HUMAN 3H- LSD 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74094 5-HT7 ?CLONED ? HUMAN 3H- LSD 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 32 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74095 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 53 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74096 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 50 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74097 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74098 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 597 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74099 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 1255 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74100 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 426 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74101 Beta 1 ?CLONED ? HUMAN 125I-Pindolol 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74102 Beta3 ?CLONED ? HUMAN 125I-Pindolol 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74103 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74104 D1 ?CLONED ? HUMAN 3H-SCH23390 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74105 D5 ?CLONED ? HUMAN 3H-SCH23390 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74106 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 216 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74107 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 145 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74108 D4 ?CLONED ? HUMAN 3H-N-Methylspiporone 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 7.1 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74109 SERT ?CLONED ? HUMAN 3H-CITALOPRAM 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74110 NET ?CLONED ? HUMAN 3H-Nisoxetine 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74111 DAT ?CLONED ? HUMAN [3H] WIN35428 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74112 H1 ?CLONED ? HUMAN 3H-PYRILAMINE 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride 114 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74113 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74114 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74115 H4 ?CLONED ? HUMAN 3H-Histamine 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74116 M1 ?CLONED ? HUMAN 3H-QNB 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74117 M2 ?CLONED ? HUMAN 3H-QNB 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74118 M3 ?CLONED ? HUMAN 3H-QNB 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74119 M4 ?CLONED ? HUMAN 3H-QNB 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74120 M5 ?CLONED ? HUMAN 3H-QNB 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74121 MOR ?CLONED ? HUMAN 3H-DAMGO 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74122 DOR ?CLONED ? HUMAN 3H-DADLE 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74123 KOR ?CLONED ? HUMAN 3H-U69593 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74124 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) naftopidil 150 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74125 Sigma 2 ?CLONED RODENT 3H-DTG naftopidil 37 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74126 PBR KIDNEY RODENT 3H-PK11195 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74127 BZP BRAIN RODENT FNZ naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74128 5-HT1A ?CLONED ? HUMAN [3H] Way100635 naftopidil 18 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74129 5-HT1B ?CLONED ? HUMAN 3H-GR125743 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74130 5-HT1D ?CLONED ? HUMAN 3H-GR125743 naftopidil 986 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74131 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin naftopidil 422 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74132 5-HT1E ?CLONED ? HUMAN 3H-5-HT naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74133 5-HT2B ?CLONED ? HUMAN 3H- LSD naftopidil 24 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74134 5-HT3 ?CLONED ? HUMAN 3H-LY278584 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74135 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74136 5-HT5A ?CLONED ? HUMAN 3H- LSD naftopidil 989 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74137 5-HT6 ?CLONED ? HUMAN 3H- LSD naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74138 5-HT7 ?CLONED ? HUMAN 3H- LSD naftopidil 44 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74139 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN naftopidil 33 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74140 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN naftopidil 117.5 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74141 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN naftopidil 14 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74142 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE naftopidil 135 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74143 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE naftopidil 97 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74144 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE naftopidil 90 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74145 Beta 1 ?CLONED ? HUMAN 125I-Pindolol naftopidil 223 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74146 Beta3 ?CLONED ? HUMAN 125I-Pindolol naftopidil 250 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74147 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 naftopidil 250 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74148 D1 ?CLONED ? HUMAN 3H-SCH23390 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74149 D5 ?CLONED ? HUMAN 3H-SCH23390 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74150 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone naftopidil 448 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74151 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone naftopidil 184 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74152 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone naftopidil 5.2 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74153 SERT ?CLONED ? HUMAN 3H-CITALOPRAM naftopidil 185 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74154 NET ?CLONED ? HUMAN 3H-Nisoxetine naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74155 DAT ?CLONED ? HUMAN [3H] WIN35428 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74156 H1 ?CLONED ? HUMAN 3H-PYRILAMINE naftopidil 89 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74157 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine naftopidil 577 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74158 MOR ?CLONED ? HUMAN 3H-DAMGO naftopidil 1080 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74159 DOR ?CLONED ? HUMAN 3H-DADLE naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74160 KOR ?CLONED ? HUMAN 3H-U69593 naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74161 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74162 H4 ?CLONED ? HUMAN 3H-Histamine naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74163 M1 ?CLONED ? HUMAN 3H-QNB naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74164 M2 ?CLONED ? HUMAN 3H-QNB naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74165 M3 ?CLONED ? HUMAN 3H-QNB naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74166 M4 ?CLONED ? HUMAN 3H-QNB naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74167 M5 ?CLONED ? HUMAN 3H-QNB naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74168 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 4.2 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74169 Sigma 2 ?CLONED RODENT 3H-DTG N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 140 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74170 PBR KIDNEY RODENT 3H-PK11195 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74171 BZP BRAIN RODENT FNZ N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74172 5-HT1A ?CLONED ? HUMAN [3H] Way100635 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74173 5-HT1B ?CLONED ? HUMAN 3H-GR125743 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74174 5-HT1D ?CLONED ? HUMAN 3H-GR125743 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 2148 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74175 5-HT1E ?CLONED ? HUMAN 3H-5-HT N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74176 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 533 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74177 5-HT2B ?CLONED ? HUMAN 3H- LSD N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 130 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74178 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 2664 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74179 5-HT3 ?CLONED ? HUMAN 3H-LY278584 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74180 5-HT5A ?CLONED ? HUMAN 3H- LSD N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74181 5-HT6 ?CLONED ? HUMAN 3H- LSD N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74182 5-HT7 ?CLONED ? HUMAN 3H- LSD N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 2897 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74183 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74184 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 1446 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74185 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74186 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 63 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74187 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 8.3 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74188 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 8.5 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74189 Beta 1 ?CLONED ? HUMAN 125I-Pindolol N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 3389 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74190 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74191 Beta3 ?CLONED ? HUMAN 125I-Pindolol N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74192 D1 ?CLONED ? HUMAN 3H-SCH23390 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74193 D5 ?CLONED ? HUMAN 3H-SCH23390 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74194 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74195 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74196 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 1201 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74197 SERT ?CLONED ? HUMAN 3H-CITALOPRAM N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 238 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74198 NET ?CLONED ? HUMAN 3H-Nisoxetine N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 145 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74199 DAT ?CLONED ? HUMAN [3H] WIN35428 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 443 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74200 H1 ?CLONED ? HUMAN 3H-PYRILAMINE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 230 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74201 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 744 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74202 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74203 H4 ?CLONED ? HUMAN 3H-Histamine N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74204 M1 ?CLONED ? HUMAN 3H-QNB N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74205 M3 ?CLONED ? HUMAN 3H-QNB N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74206 M4 ?CLONED ? HUMAN 3H-QNB N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74207 M5 ?CLONED ? HUMAN 3H-QNB N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74208 M2 ?CLONED ? HUMAN 3H-QNB N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 3114 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74209 MOR ?CLONED ? HUMAN 3H-DAMGO N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74210 KOR ?CLONED ? HUMAN 3H-U69593 N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74211 DOR ?CLONED ? HUMAN 3H-DADLE N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74212 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 46 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74213 Sigma 2 ?CLONED RODENT 3H-DTG N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 426 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74214 PBR KIDNEY RODENT 3H-PK11195 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74215 BZP BRAIN RODENT FNZ N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74216 5-HT1A ?CLONED ? HUMAN [3H] Way100635 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74217 5-HT1B ?CLONED ? HUMAN 3H-GR125743 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74218 5-HT1D ?CLONED ? HUMAN 3H-GR125743 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74219 5-HT1E ?CLONED ? HUMAN 3H-5-HT N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74220 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 1572 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74221 5-HT2B ?CLONED ? HUMAN 3H- LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 913 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74222 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74223 5-HT3 ?CLONED ? HUMAN 3H-LY278584 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74224 5-HT5A ?CLONED ? HUMAN 3H- LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74225 5-HT6 ?CLONED ? HUMAN 3H- LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74226 5-HT7 ?CLONED ? HUMAN 3H- LSD N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74227 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74228 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74229 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74230 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 127 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74231 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 27 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74232 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 90 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74233 Beta 1 ?CLONED ? HUMAN 125I-Pindolol N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74234 Beta3 ?CLONED ? HUMAN 125I-Pindolol N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74235 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74236 D1 ?CLONED ? HUMAN 3H-SCH23390 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74237 D5 ?CLONED ? HUMAN 3H-SCH23390 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74238 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74239 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 1854 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74240 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 1760 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74241 DAT ?CLONED ? HUMAN [3H] WIN35428 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 3592 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74242 H1 ?CLONED ? HUMAN 3H-PYRILAMINE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide 409 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74243 SERT ?CLONED ? HUMAN 3H-CITALOPRAM N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74244 NET ?CLONED ? HUMAN 3H-Nisoxetine N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74245 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74246 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74247 H4 ?CLONED ? HUMAN 3H-Histamine N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74248 M1 ?CLONED ? HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74249 M2 ?CLONED ? HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74250 M3 ?CLONED ? HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74251 M4 ?CLONED ? HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74252 M5 ?CLONED ? HUMAN 3H-QNB N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74253 MOR ?CLONED ? HUMAN 3H-DAMGO N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74254 KOR ?CLONED ? HUMAN 3H-U69593 N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74255 DOR ?CLONED ? HUMAN 3H-DADLE N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74256 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 241 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74257 Sigma 2 ?CLONED RODENT 3H-DTG N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 678 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74258 PBR KIDNEY RODENT 3H-PK11195 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74259 BZP BRAIN RODENT FNZ N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74260 5-HT1A ?CLONED ? HUMAN [3H] Way100635 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 52 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74261 5-HT1B ?CLONED ? HUMAN 3H-GR125743 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74262 5-HT1D ?CLONED ? HUMAN 3H-GR125743 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74263 5-HT1E ?CLONED ? HUMAN 3H-5HT N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74264 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 2396 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74265 5-HT2B ?CLONED ? HUMAN 3H-LSD N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 485 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74266 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74267 5-HT3 ?CLONED ? HUMAN 3H-LY278584 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74268 5-HT5A ?CLONED ? HUMAN 3H-LSD N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74269 5-HT6 ?CLONED ? HUMAN 3H-LSD N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74270 5-HT7 ?CLONED ? HUMAN 3H- LSD N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 268 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74271 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 144 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74272 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74273 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 160 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74274 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 241 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74275 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 974 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74276 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 548 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74277 Beta 1 ?CLONED ? HUMAN 125I-Pindolol N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74278 Beta3 ?CLONED ? HUMAN 125I-Pindolol N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74279 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74280 D1 ?CLONED ? HUMAN 3H-SCH23390 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74281 D5 ?CLONED ? HUMAN 3H-SCH23390 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74282 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 521 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74283 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 347 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74284 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 67 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74285 SERT ?CLONED ? HUMAN 3H-CITALOPRAM N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 4836 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74286 NET ?CLONED ? HUMAN 3H-Nisoxetine N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 2365 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74287 DAT ?CLONED ? HUMAN [3H] WIN35428 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 3617 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74288 H1 ?CLONED ? HUMAN 3H-PYRILAMINE N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide 106 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74289 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74290 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74291 H4 ?CLONED ? HUMAN 3H-Histamine N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74292 M1 ?CLONED ? HUMAN 3H-QNB N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74293 M2 ?CLONED ? HUMAN 3H-QNB N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74294 M3 ?CLONED ? HUMAN 3H-QNB N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74295 M4 ?CLONED ? HUMAN 3H-QNB N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74296 M5 ?CLONED ? HUMAN 3H-QNB N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74297 MOR ?CLONED ? HUMAN 3H-DAMGO N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74298 KOR ?CLONED ? HUMAN 3H-U69593 N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74299 DOR ?CLONED ? HUMAN 3H-DADLE N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74300 Sigma 1 ?CLONED RODENT 3H-Pentazocine(+) N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 9.3 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74301 Sigma 2 ?CLONED RODENT 3H-DTG N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 51 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74302 PBR KIDNEY RODENT 3H-PK11195 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74303 BZP BRAIN RODENT FNZ N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 29, 2025
74304 5-HT1A ?CLONED ? HUMAN [3H] Way100635 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74305 5-HT1B ?CLONED ? HUMAN 3H-GR125743 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74306 5-HT1D ?CLONED ? HUMAN 3H-GR125743 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74307 5-HT1E ?CLONED ? HUMAN 3H-5-HT N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74308 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74309 5-HT2B ?CLONED ? HUMAN 3H- LSD N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 223 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74310 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74311 5-HT3 ?CLONED ? HUMAN 3H-LY278584 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74312 5-HT5A ?CLONED ? HUMAN 3H- LSD N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74313 5-HT6 ?CLONED ? HUMAN 3H- LSD N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74314 5-HT7 ?CLONED ? HUMAN 3H- LSD N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74315 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74316 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74317 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74318 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 353 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74319 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 329 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74320 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 398 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74321 Beta 1 ?CLONED ? HUMAN 125I-Pindolol N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74322 Beta3 ?CLONED ? HUMAN 125I-Pindolol N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74323 Beta 2 ?CLONED ? HUMAN 3H-CGP12177 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74324 D1 ?CLONED ? HUMAN 3H-SCH23390 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74325 D5 ?CLONED ? HUMAN 3H-SCH23390 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74326 D2 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74327 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74328 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 793 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74329 SERT ?CLONED ? HUMAN 3H-CITALOPRAM N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 2242 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74330 NET ?CLONED ? HUMAN 3H-Nisoxetine N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 125 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74331 DAT ?CLONED ? HUMAN [3H] WIN35428 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 3820 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74332 H1 ?CLONED ? HUMAN 3H-PYRILAMINE N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 6285 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74333 5-HT1D ?CLONED ? HUMAN 125I-iodoaminopotentidine N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide 610 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74334 H3 ?CLONED ? HUMAN 3H-Alpha-methylhistamine N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74335 H4 ?CLONED ? HUMAN 3H-Histamine N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74336 M1 ?CLONED ? HUMAN 3H-QNB N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74337 M2 ?CLONED ? HUMAN 3H-QNB N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74338 M3 ?CLONED ? HUMAN 3H-QNB N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74339 M4 ?CLONED ? HUMAN 3H-QNB N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74340 M5 ?CLONED ? HUMAN 3H-QNB N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74341 MOR ?CLONED ? HUMAN 3H-DAMGO N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74342 KOR ?CLONED ? HUMAN 3H-U69593 N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74343 DOR ?CLONED ? HUMAN 3H-DADLE N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 28, 2025
74344 M5 ?CLONED ? HUMAN 3H-QNB {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 15, 2025
74345 KOR BRAIN RODENT 3H-MUSCIMOL N-(3-methylphenyl)-2-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]acetamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74346 KOR BRAIN RODENT 3H-MUSCIMOL N-(3,4-dimethylphenyl)-3-(4-phenyl-1-piperazinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74347 KOR BRAIN RODENT 3H-MUSCIMOL 3-(piperazin-1-yl)-N-(m-tolyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74348 KOR BRAIN RODENT 3H-MUSCIMOL N-(2-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74349 KOR BRAIN RODENT 3H-MUSCIMOL N-(3-chlorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74350 KOR BRAIN RODENT 3H-MUSCIMOL naftopidil >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74351 KOR BRAIN RODENT 3H-MUSCIMOL 1-(3-methoxyphenoxy)-3-[4-(2-methoxyphenyl)-1-piperazinyl]-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74352 KOR BRAIN RODENT 3H-MUSCIMOL 1-(2,3-dihydro-1,4-benzodioxin-2-ylmethoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74353 KOR BRAIN RODENT 3H-MUSCIMOL 1-[4-(5-chloro-2-methylphenyl)-1-piperazinyl]-3-(2,5-dimethylphenoxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74354 KOR BRAIN RODENT 3H-MUSCIMOL 1-[4-(4-methoxyphenyl)-1-piperazinyl]-3-(2-naphthyloxy)-2-propanol dihydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74355 KOR BRAIN RODENT 3H-MUSCIMOL {2-[2-(3,4-dichlorophenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74356 KOR BRAIN RODENT 3H-MUSCIMOL {2-[2-(4-tert-butyl-2-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74357 KOR BRAIN RODENT 3H-MUSCIMOL {2-[2-(4-chloro-3-ethylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74358 KOR BRAIN RODENT 3H-MUSCIMOL 1-{2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}-1H-imidazole oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74359 KOR BRAIN RODENT 3H-MUSCIMOL {2-[2-(3-isopropyl-5-methylphenoxy)ethoxy]ethyl}dimethylamine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74360 KOR BRAIN RODENT 3H-MUSCIMOL [2-(3-isopropyl-5-methylphenoxy)ethyl](2-methoxyethyl)amine oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74361 KOR BRAIN RODENT 3H-MUSCIMOL N-(3,4-dimethylphenyl)-3-[4-(2-methoxyphenyl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74362 KOR BRAIN RODENT 3H-MUSCIMOL ethyl 1-{3-[(2-fluorophenyl)amino]-3-oxopropyl}-4-piperidinecarboxylate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74363 KOR BRAIN RODENT 3H-MUSCIMOL 3-(1-azepanyl)-N-(3,4-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74364 KOR BRAIN RODENT 3H-MUSCIMOL N-(4-bromo-3-methylphenyl)-3-(1-piperidinyl)propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74365 KOR BRAIN RODENT 3H-MUSCIMOL 3-(1-azepanyl)-N-(3,5-dimethylphenyl)propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74366 KOR BRAIN RODENT 3H-MUSCIMOL N-(2-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide oxalate >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74367 KOR BRAIN RODENT 3H-MUSCIMOL N-(2,3-dihydro-1H-inden-5-yl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74368 KOR BRAIN RODENT 3H-MUSCIMOL N-phenyl-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74369 KOR BRAIN RODENT 3H-MUSCIMOL N-(4-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74370 KOR BRAIN RODENT 3H-MUSCIMOL N-(3-fluorophenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74371 KOR BRAIN RODENT 3H-MUSCIMOL N-(3-methylphenyl)-3-[4-(3-phenyl-2-propen-1-yl)-1-piperazinyl]propanamide hydrochloride >10000 Rennekamp AJ et al 2016 Jan 15, 2025 Jan 27, 2025
74372 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74373 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74374 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74375 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74376 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74377 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74378 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74379 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74380 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74381 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74382 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74383 CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74384 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74385 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74386 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74387 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74388 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74389 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74390 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74391 Beta 2 CLONED HUMAN 3H-CGP-12177 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74392 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74393 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74394 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74395 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74396 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74397 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74398 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74399 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74400 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74401 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74402 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74403 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74404 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74405 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 2480 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74406 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74407 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74408 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74409 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74410 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74411 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74412 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 340 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74413 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74414 5-HT1B CLONED HUMAN 3H-5CT (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74415 5-HT1D CLONED HUMAN 3H-5CT (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74416 5-HT1E CLONED HUMAN 3H-5HT (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74417 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74418 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74419 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74420 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74421 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74422 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74423 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74424 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74425 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74426 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74427 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74428 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74429 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74430 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74431 Beta 2 CLONED HUMAN 3H-CGP-12177 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74432 BZP CORTICAL MEMBRANES RAT 3H-CGP-12177 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74433 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74434 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74435 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74436 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74437 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74438 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74439 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74440 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74441 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74442 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74443 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74444 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74445 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74446 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74447 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74448 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74449 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74450 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74451 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74452 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[2-chloro-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74453 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74454 5-HT1B CLONED HUMAN 5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74455 5-HT1D CLONED HUMAN 5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74456 5-HT1E CLONED HUMAN 5-HT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74457 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74458 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74459 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74460 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74461 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74462 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74463 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74464 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74465 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74466 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74467 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74468 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74469 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74470 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74471 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74472 Beta 2 CLONED HUMAN 3H-CGP-12177 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74473 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74474 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74475 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74476 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74477 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74478 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74479 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74480 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74481 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74482 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74483 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74484 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74485 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74486 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74487 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74488 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74489 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74490 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74491 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74492 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74493 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74494 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 2650 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74495 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74496 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74497 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74498 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74499 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74500 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74501 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74502 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74503 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74504 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74505 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74506 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74507 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74508 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74509 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74510 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74511 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74512 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74513 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74514 Beta 2 CLONED HUMAN 3H-CGP-12177 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74515 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74516 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74517 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74518 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74519 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74520 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74521 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 6620 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74522 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74523 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74524 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74525 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74526 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74527 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74528 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74529 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74530 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74531 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74532 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74533 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74534 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74535 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74536 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(4-fluorophenyl)ethynyl]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 253 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74537 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74538 5-HT1B CLONED HUMAN 3H-5CT (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74539 5-HT1D CLONED HUMAN 3H-5CT (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74540 5-HT1E CLONED HUMAN 3H-5HT (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74541 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74542 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74543 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74544 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74545 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74546 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74547 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74548 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74549 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74550 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74551 Alpha2A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74552 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74553 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74554 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74555 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74556 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74557 Beta 2 CLONED HUMAN 3H-CGP12177 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74558 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74559 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74560 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74561 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74562 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74563 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74564 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74565 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74566 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74567 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74568 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74569 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74570 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74571 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74572 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74573 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74574 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74575 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74576 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74577 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74578 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74579 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-[(3-chlorophenyl)methylamino]purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 344 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74580 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74581 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74582 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74583 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74584 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74585 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74586 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74587 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74588 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74589 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74590 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74591 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74592 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74593 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74594 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74595 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74596 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74597 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74598 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74599 Beta 2 CLONED HUMAN 3H-CGP12177 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74600 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74601 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74602 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74603 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74604 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74605 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74606 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 5870 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74607 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74608 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74609 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74610 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74611 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74612 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74613 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74614 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74615 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74616 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74617 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74618 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74619 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74620 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74621 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[2-[2-(3-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide 1770 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74622 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74623 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74624 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74625 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74626 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74627 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74628 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74629 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74630 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74631 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74632 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74633 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74634 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74635 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74636 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74637 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74638 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74639 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74640 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74641 Beta 2 CLONED HUMAN 3H-CGP-12177 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74642 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74643 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74644 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74645 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74646 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74647 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74648 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74649 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74650 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74651 KOR CLONED HUMAN 3H-MUSCIMOL (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74652 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74653 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74654 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74655 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74656 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74657 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74658 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74659 DAT CLONED HUMAN 3H-WIN 35,428 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide 2310 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74660 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74661 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74662 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74663 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-[(2-phenylcyclopropyl)amino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74664 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74665 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74666 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74667 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74668 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74669 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74670 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74671 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74672 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74673 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74674 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74675 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74676 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74677 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74678 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74679 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74680 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74681 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74682 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74683 Beta 2 CLONED HUMAN 3H-CGP-12177 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74684 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74685 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74686 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74687 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74688 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74689 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74690 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74691 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74692 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74693 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 27, 2025
74694 M1 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74695 M2 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74696 M3 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74697 M4 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74698 M5 CLONED HUMAN 3H-QNB (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74699 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74700 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74701 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74702 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74703 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74704 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-4-[2-[2-(3,4-difluorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74705 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74706 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74707 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74708 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74709 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74710 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74711 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74712 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74713 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74714 5-HT6 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74715 5-HT7 CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74716 Alpha1A CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74717 Alpha1B CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74718 Alpha1D CLONED HUMAN 3H-PRAZOSIN (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74719 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74720 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74721 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74722 Beta 1 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74723 Beta3 CLONED HUMAN 125I-Pindolol (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74724 Beta 2 CLONED HUMAN 3H-CGP12177 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74725 BZP CORTICAL MEMBRANES RAT FNZ (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74726 D1 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74727 D5 CLONED HUMAN 3H-SCH23390 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74728 D2 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74729 D3 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74730 D4 CLONED HUMAN 3H-N-Methylspiperone (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74731 DOR CLONED HUMAN 3H-DADLE (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74732 KOR CLONED HUMAN 3H-U69593 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74733 MOR CLONED HUMAN 3H-DAMGO (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74734 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74735 Sigma 2 CLONED HUMAN 3H-DTG (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74736 SERT CLONED HUMAN 3H-CITALOPRAM (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 28, 2025
74737 NET CLONED HUMAN 3H-Nisoxetine (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74738 NOP CLONED HUMAN 3H-Nociceptin (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 29, 2025
74739 PBR Kidney membranes RAT 3H-PK11195 (1S,2R,3S,4R,5S)-2,3-dihydroxy-N-methyl-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74740 5-HT1A CLONED HUMAN 3H-WAY100635 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74741 5-HT1B CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74742 5-HT1D CLONED HUMAN 3H-5-CT (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74743 5-HT1E CLONED HUMAN 3H-5-HT (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74744 5-HT2A CLONED HUMAN 3H-KETANSERIN (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74745 5-HT2B CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74746 5-HT2C CLONED HUMAN 3H-MESULERGINE (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74747 5-HT3 CLONED HUMAN 3H-GR-65630 (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025
74748 5-HT5A CLONED HUMAN 3H-LSD (1S,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide >10000 Tosh DK et al 2018 Jan 15, 2025 Jan 15, 2025