The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 73,001-74,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
75749D5CLONEDHUMAN3H-SCH233903-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75750D2CLONEDHUMAN3H-N-Methylspiperone3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75751D3CLONEDHUMAN3H-N-Methylspiperone3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75752D4CLONEDHUMAN3H-N-Methylspiperone3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75753DORCLONEDHUMAN3H-DADLE3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75754KORCLONEDHUMAN3H-U695933-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate8920Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75755MORCLONEDHUMAN3H-DAMGO3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75756KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75757M1CLONEDHUMAN3H-QNB3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75758M2CLONEDHUMAN3H-QNB3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75759M3CLONEDHUMAN3H-QNB3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75760M4CLONEDHUMAN3H-QNB3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75761M5CLONEDHUMAN3H-QNB3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75762Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75763Sigma 2CLONEDHUMAN3H-DTG3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75764SERTCLONEDHUMAN3H-CITALOPRAM3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75765NETCLONEDHUMAN3H-Nisoxetine3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75766NOPCLONEDHUMAN3H-Nociceptin3-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75767PBRKidney membranesRAT3H-PK111953-phenylpropyl (1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate1090Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757685-HT1ACLONEDHUMAN3H-WAY1006351S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757695-HT1BCLONEDHUMAN3H-5-CT1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757705-HT1DCLONEDHUMAN3H-5-CT1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757715-HT1ECLONEDHUMAN3H-5-HT1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757725-HT2ACLONEDHUMAN3H-KETANSERIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757735-HT2BCLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757745-HT2CCLONEDHUMAN3H-MESULERGINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757755-HT3CLONEDHUMAN3H-GR-656301S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757765-HT5ACLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757775-HT6CLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
757785-HT7CLONEDHUMAN3H-LSD1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75779Alpha1ACLONEDHUMAN3H-PRAZOSIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75780Alpha1BCLONEDHUMAN3H-PRAZOSIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75781Alpha1DCLONEDHUMAN3H-PRAZOSIN1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75782Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75783Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75784Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75785Beta 1CLONEDHUMAN125I-Pindolol1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75786Beta3CLONEDHUMAN125I-Pindolol1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75787Beta 2CLONEDHUMAN3H-CGP121771S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75788BZPCORTICAL MEMBRANESRATFNZ1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75789D1CLONEDHUMAN3H-SCH233901S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75790D5CLONEDHUMAN3H-SCH233901S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75791D2CLONEDHUMAN3H-N-Methylspiperone1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75792D3CLONEDHUMAN3H-N-Methylspiperone1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75793D4CLONEDHUMAN3H-N-Methylspiperone1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75794DORCLONEDHUMAN3H-DADLE1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75795KORCLONEDHUMAN3H-U695931S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75796MORCLONEDHUMAN3H-DAMGO1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75797KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75798M1CLONEDHUMAN3H-QNB1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75799M2CLONEDHUMAN3H-QNB1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75800M3CLONEDHUMAN3H-QNB1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75801M4CLONEDHUMAN3H-QNB1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75802M5CLONEDHUMAN3H-QNB1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75803Sigma 1CLONEDHUMAN3H-Pentazocine(+)1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75804Sigma 2CLONEDHUMAN3H-DTG1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75805SERTCLONEDHUMAN3H-CITALOPRAM1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75806NETCLONEDHUMAN3H-Nisoxetine1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75807NOPCLONEDHUMAN3H-Nociceptin1S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75808PBRKidney membranesRAT3H-PK111951S,2R,3S,4R,5S)-4-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylic acid>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758095-HT1ACLONEDHUMAN3H-WAY100635Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758105-HT1BCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758115-HT1DCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758125-HT1ECLONEDHUMAN3H-5-HTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758135-HT2ACLONEDHUMAN3H-KETANSERINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758145-HT2BCLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758155-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758165-HT3CLONEDHUMAN3H-GR-65630Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758175-HT5ACLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758185-HT6CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758195-HT7CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75820Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75821Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75822Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75823Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75824Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75825Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75826Beta 1CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75827Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75828Beta 2CLONEDHUMAN3H-CGP12177Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75829BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75830D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75831D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75832D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75833D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75834D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75835DORCLONEDHUMAN3H-DADLEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate1590Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75836KORCLONEDHUMAN3H-U69593Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate104Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75837MORCLONEDHUMAN3H-DAMGOEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75838KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75839M1CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75840M2CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75841M3CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75842M4CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75843M5CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75844Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75845Sigma 2CLONEDHUMAN3H-DTGEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75846SERTCLONEDHUMAN3H-CITALOPRAMEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75847NETCLONEDHUMAN3H-NisoxetineEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75848NOPCLONEDHUMAN3H-NociceptinEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75849PBRKidney membranesRAT3H-PK11195Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(2-iodo-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]- hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758505-HT1ACLONEDHUMAN3H-WAY100635Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758515-HT1BCLONEDHUMAN3H-5-CTEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758525-HT1DCLONEDHUMAN3H-5-CTEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758535-HT1ECLONEDHUMAN3H-5-HTEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758545-HT2ACLONEDHUMAN3H-KETANSERINEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758555-HT2BCLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758565-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758575-HT3CLONEDHUMAN3H-GR-65630Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758585-HT5ACLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758595-HT6CLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758605-HT7CLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75861Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75862Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75863Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75864Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75865Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75866Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75867Beta 1CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75868Beta3CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75869Beta 2CLONEDHUMAN3H-CGP-12177Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75870BZPCORTICAL MEMBRANESRATFNZEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75871D1CLONEDHUMAN3H-SCH23390Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75872D5CLONEDHUMAN3H-SCH23390Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75873D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75874D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75875D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75876DORCLONEDHUMAN3H-DADLEEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75877KORCLONEDHUMAN3H-U69593Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate276Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75878MORCLONEDHUMAN3H-DAMGOEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate7600Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75879KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75880M1CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75881M2CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75882M3CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75883M4CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75884M5CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75885Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75886Sigma 2CLONEDHUMAN3H-DTGEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75887SERTCLONEDHUMAN3H-CITALOPRAMEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75888NETCLONEDHUMAN3H-NisoxetineEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75889NOPCLONEDHUMAN3H-NociceptinEthyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75890PBRKidney membranesRAT3H-PK11195Ethyl(3aR,3bS,4aS,5R,5aS)-5-(2-iodo-4-(methylamino)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,2- dimethyltetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]- dioxole-3b(3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758915-HT1ACLONEDHUMAN3H-WAY100635Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758925-HT1BCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758935-HT1DCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758945-HT1ECLONEDHUMAN3H-5-HTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758955-HT2ACLONEDHUMAN3H-KETANSERINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758965-HT2BCLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758975-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758985-HT3CLONEDHUMAN3H-GR-65630Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
758995-HT5ACLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759005-HT6CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759015-HT7CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75902Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75903Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75904Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75905Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75906Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75907Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75908Beta 1CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75909Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75910Beta 2CLONEDHUMAN3H-CGP12177Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75911BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75912D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75913D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75914D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75915D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75916D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75917DORCLONEDHUMAN3H-DADLEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate1780Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75918KORCLONEDHUMAN3H-U69593Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate91.5Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75919MORCLONEDHUMAN3H-DAMGOEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate1480Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75920KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75921M1CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75922M2CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75923M3CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75924M4CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75925M5CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75926Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75927Sigma 2CLONEDHUMAN3H-DTGEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75928SERTCLONEDHUMAN3H-CITALOPRAMEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75929NETCLONEDHUMAN3H-NisoxetineEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75930NOPCLONEDHUMAN3H-NociceptinEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75931PBRKidney membranesRAT3H-PK11195Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(methylamino)- 2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759325-HT1ACLONEDHUMAN3H-WAY100635Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759335-HT1BCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759345-HT1DCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759355-HT1ECLONEDHUMAN3H-5-HTEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759365-HT2ACLONEDHUMAN3H-KETANSERINEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759375-HT2BCLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759385-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759395-HT3CLONEDHUMAN3H-GR-65630Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759405-HT5ACLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759415-HT6CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759425-HT7CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75943Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75944Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75945Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75946Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75947Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75948Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75949Beta 1CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75950Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75951Beta 2CLONEDHUMAN3H-CGP12177Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75952BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75953D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75954D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75955D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75956D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75957D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75958DORCLONEDHUMAN3H-DADLEEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate2400Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75959KORCLONEDHUMAN3H-U69593Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate852Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75960MORCLONEDHUMAN3H-DAMGOEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate2110Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75961KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
75962M1CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75963M2CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75964M3CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75965M4CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75966M5CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75967Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75968Sigma 2CLONEDHUMAN3H-DTGEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75969SERTCLONEDHUMAN3H-CITALOPRAMEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75970NETCLONEDHUMAN3H-NisoxetineEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75971NOPCLONEDHUMAN3H-NociceptinEthyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75972PBRKidney membranesRAT3H-PK11195Ethyl(1S,2R,3S,4R,5S)-4-(4-(cyclopropylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759735-HT1ACLONEDHUMAN3H-WAY100635Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759745-HT1BCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759755-HT1DCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759765-HT1ECLONEDHUMAN3H-5-HTEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759775-HT2ACLONEDHUMAN3H-KETANSERINEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759785-HT2BCLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759795-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759805-HT3CLONEDHUMAN3H-GR65630Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759815-HT5ACLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759825-HT6CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
759835-HT7CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75984Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75985Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75986Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75987Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75988Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75989Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75990Beta 1CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75991Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75992Beta 2CLONEDHUMAN3H-CGP-12177Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
75993BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
75994D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75995D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75996D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75997D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75998D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
75999DORCLONEDHUMAN3H-DADLEEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76000KORCLONEDHUMAN3H-U69593Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate1400Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76001MORCLONEDHUMAN3H-DAMGOEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate1300Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76002KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76003M1CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76004M2CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76005M3CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76006M4CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76007M5CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76008Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76009Sigma 2CLONEDHUMAN3H-DTGEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76010SERTCLONEDHUMAN3H-CITALOPRAMEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76011NETCLONEDHUMAN3H-NisoxetineEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76012NOPCLONEDHUMAN3H-NociceptinEthyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76013PBRKidney membranesRAT3H-PK11195Ethyl(1S,2R,3S,4R,5S)-4-(4-((cyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-2,3- dihydroxybicyclo[3.1.0]hexane-1-carboxylate4470Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760145-HT1ACLONEDHUMAN3H-WAY100635Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760155-HT1BCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760165-HT1DCLONEDHUMAN3H-5-CTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760175-HT1ECLONEDHUMAN3H-5-HTEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760185-HT2ACLONEDHUMAN3H-KETANSERINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760195-HT2BCLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760205-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760215-HT3CLONEDHUMAN3H-GR-65630Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760225-HT5ACLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760235-HT6CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760245-HT7CLONEDHUMAN3H-LSDEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76025Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76026Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76027Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76028Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76029Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76030Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76031Beta 1CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76032Beta3CLONEDHUMAN125I-PindololEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76033Beta 2CLONEDHUMAN3H-CGP-12177Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76034BZPCORTICAL MEMBRANESRATFNZEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76035D1CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76036D5CLONEDHUMAN3H-SCH23390Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76037D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76038D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76039D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76040DORCLONEDHUMAN3H-DADLEEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate627Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76041KORCLONEDHUMAN3H-U69593Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate207Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76042MORCLONEDHUMAN3H-DAMGOEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate1770Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76043KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76044M1CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76045M2CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76046M3CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76047M4CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76048M5CLONEDHUMAN3H-QNBEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76049Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76050Sigma 2CLONEDHUMAN3H-DTGEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76051SERTCLONEDHUMAN3H-CITALOPRAMEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76052NETCLONEDHUMAN3H-NisoxetineEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76053NOPCLONEDHUMAN3H-NociceptinEthyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76054PBRKidney membranesRAT3H-PK11195Ethyl(1S,2R,3S,4R,5S)-2,3-dihydroxy-4-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- bicyclo[3.1.0]hexane-1-carboxylate480Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760555-HT1ACLONEDHUMAN3H-WAY100635Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760565-HT1BCLONEDHUMAN3H-5-CTEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760575-HT1DCLONEDHUMAN3H-5-CTEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760585-HT1ECLONEDHUMAN3H-5-HTEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760595-HT2ACLONEDHUMAN3H-KETANSERINEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760605-HT2BCLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760615-HT2CCLONEDHUMAN3H-MESULERGINEEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760625-HT3CLONEDHUMAN3H-GR-65630Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760635-HT5ACLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760645-HT6CLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760655-HT7CLONEDHUMAN3H-LSDEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76066Alpha1ACLONEDHUMAN3H-PRAZOSINEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76067Alpha1BCLONEDHUMAN3H-PRAZOSINEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76068Alpha1DCLONEDHUMAN3H-PRAZOSINEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76069Alpha2ACLONEDHUMAN3H-RAUWOLSCINEEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76070Alpha2BCLONEDHUMAN3H-RAUWOLSCINEEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76071Alpha2CCLONEDHUMAN3H-RAUWOLSCINEEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76072Beta 1CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76073Beta3CLONEDHUMAN125I-PindololEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76074Beta 2CLONEDHUMAN3H-CGP12177Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76075BZPCORTICAL MEMBRANESRATFNZEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76076D1CLONEDHUMAN3H-SCH23390Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76077D5CLONEDHUMAN3H-SCH23390Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76078D2CLONEDHUMAN3H-N-MethylspiperoneEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76079D3CLONEDHUMAN3H-N-MethylspiperoneEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76080D4CLONEDHUMAN3H-N-MethylspiperoneEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76081DORCLONEDHUMAN3H-DADLEEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate881Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76082KORCLONEDHUMAN3H-U69593Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate217Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76083MORCLONEDHUMAN3H-DAMGOEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76084KORCORTICAL MEMBRANESRAT3H-MUSCIMOLEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76085M1CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76086M2CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76087M3CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76088M4CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76089M5CLONEDHUMAN3H-QNBEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76090Sigma 1CLONEDHUMAN3H-Pentazocine(+)Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76091Sigma 2CLONEDHUMAN3H-DTGEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76092SERTCLONEDHUMAN3H-CITALOPRAMEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76093NETCLONEDHUMAN3H-NisoxetineEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76094NOPCLONEDHUMAN3H-NociceptinEthyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76095PBRKidney membranesRAT3H-PK11195Ethyl(3aR,3bS,4aS,5R,5aS)-2,2-dimethyl-5-(4-(phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)- tetrahydrocyclopropa[3,4]cyclopenta[1,2-d][1,3]dioxole-3b- (3aH)-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760965-HT1ACLONEDHUMAN3H-WAY1006352S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760975-HT1BCLONEDHUMAN3H-5-CT2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760985-HT1DCLONEDHUMAN3H-5-CT2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
760995-HT1ECLONEDHUMAN3H-5-HT2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761005-HT2ACLONEDHUMAN3H-KETANSERIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761015-HT2BCLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761025-HT2CCLONEDHUMAN3H-MESULERGINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761035-HT3CLONEDHUMAN3H-GR-656302S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761045-HT5ACLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761055-HT6CLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761065-HT7CLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76107Alpha1ACLONEDHUMAN3H-PRAZOSIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76108Alpha1BCLONEDHUMAN3H-PRAZOSIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76109Alpha1DCLONEDHUMAN3H-PRAZOSIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76110Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76111Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76112Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76113Beta 1CLONEDHUMAN125I-Pindolol2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76114Beta3CLONEDHUMAN125I-Pindolol2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76115Beta 2CLONEDHUMAN3H-CGP-121772S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76116BZPCORTICAL MEMBRANESRATFNZ2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76117D1CLONEDHUMAN3H-SCH233902S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76118D5CLONEDHUMAN3H-SCH233902S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76119D2CLONEDHUMAN3H-N-Methylspiperone2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76120D3CLONEDHUMAN3H-N-Methylspiperone2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76121D4CLONEDHUMAN3H-N-Methylspiperone2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76122DORCLONEDHUMAN3H-DADLE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76123KORCLONEDHUMAN3H-U695932S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide2610Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76124MORCLONEDHUMAN3H-DAMGO2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76125KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76126M1CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76127M2CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76128M3CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76129M4CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76130M5CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76131Sigma 1CLONEDHUMAN3H-Pentazocine(+)2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76132Sigma 2CLONEDHUMAN3H-DTG2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76133SERTCLONEDHUMAN3H-CITALOPRAM2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76134NETCLONEDHUMAN3H-Nisoxetine2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76135NOPCLONEDHUMAN3H-Nociceptin2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76136PBRKidney membranesRAT3H-PK111952S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761375-HT1ACLONEDHUMAN3H-WAY1006352S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761385-HT1BCLONEDHUMAN3H-5-CT2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761395-HT1DCLONEDHUMAN3H-5-CT2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761405-HT1ECLONEDHUMAN3H-5-HT2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761415-HT2ACLONEDHUMAN3H-KETANSERIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761425-HT2BCLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761435-HT2CCLONEDHUMAN3H-MESULERGINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761445-HT3CLONEDHUMAN3H-GR-656302S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761455-HT5ACLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761465-HT6CLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761475-HT7CLONEDHUMAN3H-LSD2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76148Alpha1ACLONEDHUMAN3H-PRAZOSIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76149Alpha1BCLONEDHUMAN3H-PRAZOSIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76150Alpha1DCLONEDHUMAN3H-PRAZOSIN2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76151Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76152Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76153Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76154Beta 1CLONEDHUMAN125I-Pindolol2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76155Beta3CLONEDHUMAN125I-Pindolol2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76156Beta 2CLONEDHUMAN3H-CGP121772S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76157BZPCORTICAL MEMBRANESRATFNZ2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76158D1CLONEDHUMAN3H-SCH233902S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76159D5CLONEDHUMAN3H-SCH233902S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76160D2CLONEDHUMAN3H-N-Methylspiperone2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76161D3CLONEDHUMAN3H-N-Methylspiperone2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76162D4CLONEDHUMAN3H-N-Methylspiperone2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76163DORCLONEDHUMAN3H-DADLE2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76164KORCLONEDHUMAN3H-U695932S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76165MORCLONEDHUMAN3H-DAMGO2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76166KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76167M1CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76168M2CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76169M3CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76170M4CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76171M5CLONEDHUMAN3H-QNB2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76172Sigma 1CLONEDHUMAN3H-Pentazocine(+)2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76173Sigma 2CLONEDHUMAN3H-DTG2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76174SERTCLONEDHUMAN3H-CITALOPRAM2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76175NETCLONEDHUMAN3H-Nisoxetine2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76176NOPCLONEDHUMAN3H-Nociceptin2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76177PBRKidney membranesRAT3H-PK111952S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxy-N-methyloxolane-2-carboxamide>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761785-HT1ACLONEDHUMAN3H-WAY100635(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761795-HT1BCLONEDHUMAN3H-5-CT(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761805-HT1DCLONEDHUMAN3H-5-CT(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761815-HT1ECLONEDHUMAN3H-5-HT(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761825-HT2ACLONEDHUMAN3H-KETANSERIN(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761835-HT2BCLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761845-HT2CCLONEDHUMAN3H-MESULERGINE(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761855-HT3CLONEDHUMAN3H-GR-65630(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761865-HT5ACLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761875-HT6CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
761885-HT7CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76189Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76190Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76191Alpha1DCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76192Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76193Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76194Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76195Beta 1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76196Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76197Beta 2CLONEDHUMAN3H-CGP-12177(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76198BZPCORTICAL MEMBRANESRATFNZ(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76199D1CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76200D5CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76201D2CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76202D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76203D4CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76204DORCLONEDHUMAN3H-DADLE(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76205KORCLONEDHUMAN3H-U69593(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76206MORCLONEDHUMAN3H-DAMGO(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76207KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76208M1CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76209M2CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76210M3CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76211M4CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76212M5CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76213Sigma 1CLONEDHUMAN3H-Pentazocine(+)(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76214Sigma 2CLONEDHUMAN3H-DTG(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76215SERTCLONEDHUMAN3H-CITALOPRAM(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76216NETCLONEDHUMAN3H-Nisoxetine(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76217NOPCLONEDHUMAN3H-Nociceptin(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76218PBRKidney membranesRAT3H-PK11195(2S,3S,4R,5R)-5-[2-[2-(5-chlorothiophen-2-yl)ethynyl]-6-(methylamino)purin-9-yl]-3,4-dihydroxyoxolane-2-carboxylate>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762195-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762205-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762215-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762225-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762235-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762245-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762255-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762265-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762275-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762285-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762295-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76230Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76231Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76232Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76233Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76234Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76235Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76236Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76237Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76238Beta 2CLONEDHUMAN3H-CGP-12177(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76239BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76240D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76241D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76242D2CLONEDHUMAN3H-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76243D3CLONEDHUMAN3H-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76244D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76245DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76246KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76247MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76248KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76249M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76250M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76251M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76252M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76253M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76254Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76255Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76256SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76257NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76258NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76259PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-[2-(3,4-difluorophenyl)ethynyl]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol1750Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762605-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762615-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762625-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762635-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762645-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762655-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762665-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762675-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762685-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762695-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
762705-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76271Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76272Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76273Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76274Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76275Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76276Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76277Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76278Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76279Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76280D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76281D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76282D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76283D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76284D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76285DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol8000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76286KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76287MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76288KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76289M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76290M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76291M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76292M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76293M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76294Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76295Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76296SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76297NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76298NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76299PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol1640Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763005-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763015-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763025-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763035-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763045-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763055-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763065-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763075-HT3CLONEDHUMAN3H-GR65630(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763085-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763095-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763105-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76311Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76312Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76313Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76314Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76315Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76316Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76317Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76318Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76319Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76320BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76321D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76322D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76323D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76324D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76325D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76326DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76327KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76328MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76329KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76330M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76331M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76332M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76333M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76334M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76335Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76336Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76337SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76338NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76339NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76340PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-[(3-chlorophenyl)methylamino]purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763415-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763425-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763435-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763445-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763455-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763465-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763475-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763485-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763495-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763505-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763515-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76352Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76353Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76354Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76355Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76356Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76357Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76358Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76359Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76360Beta 2CLONEDHUMAN3H-CGP-12177(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76361BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76362D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76363D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76364D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76365D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76366D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76367DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76368KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76369MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76370KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76371M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76372M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76373M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76374M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76375M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76376Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76377Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76378SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76379NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76380PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-(methylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763815-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763825-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763835-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763845-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763855-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763865-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763875-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763885-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763895-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763905-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
763915-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76392Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76393Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76394Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76395Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76396Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76397Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76398Beta1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76399Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76400Beta2CLONEDHUMAN3H-CGP-12177(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76401BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76402D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76403D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76404D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76405D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76406D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76407DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76408KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76409MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76410KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76411M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76412M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76413M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76414M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76415M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76416Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76417Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76418SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76419NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol8660Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76420NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76421PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-(ethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764225-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764235-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764245-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764255-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764265-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764275-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764285-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764295-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764305-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764315-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764325-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76433Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76434Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76435Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76436Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76437Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76438Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76439Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76440Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76441Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76442BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76443D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76444D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76445D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76446D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76447D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76448DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76449KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76450MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76451KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76452M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76453M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76454M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76455M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76456M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76457Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76458Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76459SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76460NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol2800Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76461NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76462PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-(2-phenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764635-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764645-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764655-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764665-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764675-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764685-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764695-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764705-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764715-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764725-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
764735-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76474Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76475Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76476Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76477Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76478Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76479Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76480Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76481Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76482Beta 2CLONEDHUMAN3H-CGP-12177(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76483BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76484D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76485D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76486D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76487D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76488D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76489DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76490KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76491MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76492KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76493M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76494M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76495M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76496M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76497M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76498Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76499Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76500SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76501NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76502NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76503PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[2-[2-(2-chlorophenyl)ethynyl]-6-(2-phenylethylamino)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol877Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765045-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765055-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765065-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765075-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765085-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765095-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765105-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765115-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765125-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765135-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765145-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76515Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76516Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76517Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76518Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76519Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76520Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76521Beta1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76522Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76523Beta2CLONEDHUMAN3H-CGP-12177(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76524BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76525D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76526D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76527D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76528D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76529D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76530DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76531KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76532MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76533KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76534M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76535M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76536M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76537M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76538M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76539Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76540Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76541SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76542NETCLONEDHUMAN[3 H](R,S)-3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-amine(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol5780Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76543NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76544PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-[6-(2,2-diphenylethylamino)-2-(2-phenylethynyl)purin-9-yl]bicyclo[3.1.0]hexane-2,3-diol3570Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765455-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765465-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765475-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765485-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765495-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765505-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765515-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765525-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765535-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765545-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765555-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76556Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76557Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76558Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76559Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76560Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76561Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76562Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76563Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76564Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76565BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76566D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76567D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76568D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76569D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76570D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76571DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76572KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol1120Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76573MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol2670Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76574KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76575M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76576M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76577M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76578M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76579M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76580Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76581Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76582SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76583NETCLONEDHUMAN3H-Nisoxetine(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76584NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76585PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-(4-(Methylamino)-2-(phenylethynyl)- 7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane-2,3- diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765865-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765875-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765885-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765895-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765905-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765915-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765925-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765935-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765945-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765955-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
765965-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76597Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76598Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76599Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76600Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76601Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76602Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76603Beta1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76604Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76605Beta2CLONEDHUMAN3H-CGP-12177(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76606BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76607D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76608D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76609D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76610D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76611D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76612DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol3660Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76613KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol1370Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76614MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol4020Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76615KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76616M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76617M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76618M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76619M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76620M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76621Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76622Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76623SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76624NETCLONEDHUMAN3H-Nisoxetine(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol5560Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76625NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76626PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-(4-(Phenethylamino)-2-(phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol2120Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766275-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766285-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766295-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766305-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766315-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766325-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766335-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766345-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766355-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766365-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766375-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76638Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76639Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76640Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76641Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76642Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76643Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76644Beta1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76645Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76646Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76647BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76648D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76649D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76650D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76651D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76652D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76653DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol2550Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76654KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76655MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol1440Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76656KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76657M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76658M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76659M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76660M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76661M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76662Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76663Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76664SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76665NETCLONEDHUMAN3H-Nisoxetine(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76666DATCLONEDHUMAN3H-WIN 35,428(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76667NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76668PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- (phenylethynyl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo- [3.1.0]hexane-2,3-diol4210Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766695-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766705-HT1BCLONEDHUMAN3H-5CT(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766715-HT1DCLONEDHUMAN3H-5CT(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766725-HT1ECLONEDHUMAN3H-5HT(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766735-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766745-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766755-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766765-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766775-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766785-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
766795-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76680Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76681Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76682Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76683Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76684Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76685Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76686Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76687Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76688Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76689BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76690D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76691D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76692D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76693D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76694D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76695DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76696KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol3020Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76697MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76698KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76699M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76700M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76701M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76702M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76703M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76704Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76705Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76706SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76707NETCLONEDHUMAN3H-Nisoxetine(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76708NOPCLONEDHUMAN3H-Nociceptin(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76709DATCLONEDHUMAN3H-WIN 35,428(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76710PBRKidney membranesRAT3H-PK11195(1R,2R,3S,4R,5S)-4-(2-((5-Bromothiophen-2-yl)ethynyl)-4- ((dicyclopropylmethyl)amino)-7H-pyrrolo[2,3-d]pyrimidin7-yl)bicyclo[3.1.0]hexane-2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767115-HT1ACLONEDHUMAN3H-WAY100635(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767125-HT1BCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767135-HT1DCLONEDHUMAN3H-5-CT(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767145-HT1ECLONEDHUMAN3H-5-HT(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767155-HT2ACLONEDHUMAN3H-KETANSERIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767165-HT2BCLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767175-HT2CCLONEDHUMAN3H-MESULERGINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767185-HT3CLONEDHUMAN3H-GR-65630(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767195-HT5ACLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767205-HT6CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
767215-HT7CLONEDHUMAN3H-LSD(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76722Alpha1ACLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76723Alpha1BCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76724Alpha1DCLONEDHUMAN3H-PRAZOSIN(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76725Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76726Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76727Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76728Beta 1CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76729Beta3CLONEDHUMAN125I-Pindolol(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76730Beta 2CLONEDHUMAN3H-CGP12177(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76731BZPCORTICAL MEMBRANESRATFNZ(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 29, 2025
76732D1CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76733D5CLONEDHUMAN3H-SCH23390(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76734D2CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76735D3CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76736D4CLONEDHUMAN3H-N-Methylspiperone(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76737DORCLONEDHUMAN3H-DADLE(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76738KORCLONEDHUMAN3H-U69593(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76739MORCLONEDHUMAN3H-DAMGO(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76740KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 27, 2025
76741M1CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76742M2CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76743M3CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76744M4CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76745M5CLONEDHUMAN3H-QNB(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 15, 2025
76746Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76747Sigma 2CLONEDHUMAN3H-DTG(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025
76748SERTCLONEDHUMAN3H-CITALOPRAM(1R,2R,3S,4R,5S)-4-(4-((Dicyclopropylmethyl)amino)-2- iodo-7H-pyrrolo[2,3-d]pyrimidin-7-yl)bicyclo[3.1.0]hexane2,3-diol>10000Tosh DK et al 2018Jan 15, 2025Jan 28, 2025