82749 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82750 5-HT1B CLONED HUMAN 3H-5-CT (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82751 5-HT1D CLONED HUMAN 3H-5-CT (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82752 5-HT1E CLONED HUMAN 3H-5-HT (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82753 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82754 5-HT2B CLONED HUMAN 3H-LSD (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82755 5-HT2C CLONED HUMAN 3H-MESULERGINE (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82756 5-HT3 CLONED HUMAN 3H-GR65630 (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82757 5-HT4 CLONED HUMAN 3H-GR113808 (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82758 5-HT5A CLONED HUMAN 3H-LSD (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82759 5-HT6 CLONED HUMAN 3H-LSD (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82760 5-HT7 CLONED HUMAN 3H-LSD (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82761 Alpha1A CLONED HUMAN 3H-PRAZOSIN (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82762 Alpha1B CLONED HUMAN 3H-PRAZOSIN (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82763 Alpha1D CLONED HUMAN 3H-PRAZOSIN (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82764 D1 CLONED HUMAN 3H-SCH23390 (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine 5852 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82765 D5 CLONED HUMAN 3H-SCH23390 (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82766 D2 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82767 D3 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82768 D4 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(((5-Chloropyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine 90 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82769 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82770 5-HT1B CLONED HUMAN 3H-5-CT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82771 5-HT1D CLONED HUMAN 3H-5-CT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82772 5-HT1E CLONED HUMAN 3H-5-HT (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82773 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine 1482 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82774 5-HT2B CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82775 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82776 5-HT3 CLONED HUMAN 3H-GR65630 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82777 5-HT4 CLONED HUMAN 3H-GR113808 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82778 5-HT5A CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82779 5-HT6 CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82780 5-HT7 CLONED HUMAN 3H-LSD (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82781 Alpha1A CLONED HUMAN 3H-PRAZOSIN (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82782 Alpha1B CLONED HUMAN 3H-PRAZOSIN (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82783 Alpha1D CLONED HUMAN 3H-PRAZOSIN (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82784 D1 CLONED HUMAN 3H-SCH23390 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82785 D5 CLONED HUMAN 3H-SCH23390 (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82786 D2 CLONED HUMAN 3H-N-Methylspiperone (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82787 D3 CLONED HUMAN 3H-N-Methylspiperone (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82788 D4 CLONED HUMAN 3H-N-Methylspiperone (R)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82789 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82790 5-HT1B CLONED HUMAN 3H-5-CT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82791 5-HT1D CLONED HUMAN 3H-5-CT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82792 5-HT1E CLONED HUMAN 3H-5-HT (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82793 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82794 5-HT2B CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82795 5-HT2C CLONED HUMAN 3H-MESULERGINE (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82796 5-HT3 CLONED HUMAN 3H-GR65630 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82797 5-HT4 CLONED HUMAN 3H-GR113808 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82798 5-HT5A CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82799 5-HT6 CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82800 5-HT7 CLONED HUMAN 3H-LSD (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82801 Alpha1A CLONED HUMAN 3H-PRAZOSIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82802 Alpha1B CLONED HUMAN 3H-PRAZOSIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82803 Alpha1D CLONED HUMAN 3H-PRAZOSIN (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82804 D1 CLONED HUMAN 3H-SCH23390 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82805 D5 CLONED HUMAN 3H-SCH23390 (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82806 D2 CLONED HUMAN 3H-N-Methylspiperone (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82807 D3 CLONED HUMAN 3H-N-Methylspiperone (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82808 D4 CLONED HUMAN 3H-N-Methylspiperone (S)-4-(2-(Indolin-1-yl)ethyl)-2-(((6-methylpyridin-3-yl)oxy)methyl)morpholine 502.9 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82809 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82810 5-HT1B CLONED HUMAN 3H-5-CT (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82811 5-HT1D CLONED HUMAN 3H-5-CT (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82812 5-HT1E CLONED HUMAN 3H-5-HT (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82813 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82814 5-HT2B CLONED HUMAN 3H-LSD (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine 1326 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82815 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82816 5-HT3 CLONED HUMAN 3H-GR65630 (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82817 5-HT4 CLONED HUMAN 3H-GR113808 (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82818 5-HT5A CLONED HUMAN 3H-LSD (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82819 5-HT6 CLONED HUMAN 3H-LSD (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82820 5-HT7 CLONED HUMAN 3H-LSD (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 15, 2025
82821 Alpha1A CLONED HUMAN 3H-PRAZOSIN (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82822 Alpha1B CLONED HUMAN 3H-PRAZOSIN (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82823 Alpha1D CLONED HUMAN 3H-PRAZOSIN (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82824 D1 CLONED HUMAN 3H-SCH23390 (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82825 D5 CLONED HUMAN 3H-SCH23390 (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82826 D2 CLONED HUMAN 3H-N-Methylspiperone (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82827 D3 CLONED HUMAN 3H-N-Methylspiperone (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine >10000 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82828 D4 CLONED HUMAN 3H-N-Methylspiperone (R)-2-(((2,4-Dimethylpyridin-3-yl)oxy)methyl)-4-(2-(indolin-1-yl)ethyl)morpholine 4947 Besnard J et al 2012 Jan 15, 2025 Jan 28, 2025
82829 A1 CHO cells HUMAN 3H-CCPA Istradefylline 841 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82830 A1 CORTICAL MEMBRANES RAT 3H-CCPA Istradefylline 230 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82831 A2A CHO cells HUMAN 3H-MSX-2 Istradefylline 12 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82832 A2A Striatal Membranes RAT 3H-MSX-2 Istradefylline 4.46 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82833 A2B CHO cells HUMAN 3H-PSB-603 Istradefylline >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82834 A3 CHO cells HUMAN 3H-PSB-11 Istradefylline 4470 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82835 A1 CHO cells HUMAN 3H-CCPA CSC >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82836 A1 CORTICAL MEMBRANES RAT 3H-CCPA CSC >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82837 A2A CHO cells HUMAN 3H-MSX-2 CSC 38 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82838 A2A Striatal Membranes RAT 3H-MSX-2 CSC 54 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82839 A2B CHO cells HUMAN 3H-PSB-603 CSC 8200 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82840 A3 CHO cells HUMAN 3H-PSB-11 CSC >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82841 A1 CHO cells HUMAN 3H-CCPA 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 265 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82842 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 79.3 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82843 A2A CHO cells HUMAN 3H-MSX-2 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1060 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82844 A2A Striatal Membranes RAT 3H-MSX-2 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 598 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82845 A2B CHO cells HUMAN 3H-PSB-603 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82846 A3 CHO cells HUMAN 3H-PSB-11 8-Benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82847 A1 CHO cells HUMAN 3H-CCPA 8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 152 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82848 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 40.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82849 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1260 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82850 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82851 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82852 A1 CHO cells HUMAN 3H-CCPA 8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 80.6 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82853 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 42 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82854 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1330 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82855 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82856 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82857 A1 CHO cells HUMAN 3H-CCPA 8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 427 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82858 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 54.2 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82859 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1250 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82860 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82861 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Chlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82862 A1 CHO cells HUMAN 3H-CCPA 8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 218 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82863 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 15.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82864 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82865 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82866 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82867 A1 CHO cells HUMAN 3H-CCPA 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 215 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82868 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 61.9 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82869 A2A CHO cells HUMAN 3H-MSX-2 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 962 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82870 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82871 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82872 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82873 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82874 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82875 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82876 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82877 A1 CHO cells HUMAN 3H-CCPA 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 85.7 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82878 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 40.1 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82879 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 291 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82880 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 257 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82881 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82882 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82883 A1 CHO cells HUMAN 3H-CCPA 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 64.4 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82884 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 52.8 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82885 A2A CHO cells HUMAN 3H-MSX-2 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 769 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82886 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 621 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82887 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82888 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82889 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82890 A2A CHO cells HUMAN 3H-MSX-2 8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3860 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82891 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1060 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82892 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82893 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Bromobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82894 A1 CHO cells HUMAN 3H-CCPA 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 87.7 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82895 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 25.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82896 A2A CHO cells HUMAN 3H-MSX-2 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 834 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82897 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 384 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82898 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82899 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Iodobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82900 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82901 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82902 A2B CHO cells HUMAN 3H-PSB-603 8-(2-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82903 A3 CHO cells HUMAN 3H-PSB-11 8-(2-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82904 A1 CHO cells HUMAN 3H-CCPA 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 127 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82905 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 26 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82906 A2A CHO cells HUMAN 3H-MSX-2 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 533 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82907 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 476 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82908 A2B CHO cells HUMAN 3H-PSB-603 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82909 A3 CHO cells HUMAN 3H-PSB-11 8-(3-(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82910 A1 CHO cells HUMAN 3H-CCPA 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 216 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82911 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 74.4 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82912 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 653 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82913 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 387 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82914 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82915 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82916 A1 CHO cells HUMAN 3H-CCPA 8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 392 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82917 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 51.1 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82918 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82919 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82920 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82921 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82922 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82923 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82924 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82925 A1 CHO cells HUMAN 3H-CCPA 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 76.2 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82926 A1 CORTICAL MEMBRANES RAT 3H-CCPA 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 98.8 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82927 A2A CHO cells HUMAN 3H-MSX-2 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1020 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82928 A2A Striatal Membranes RAT 3H-MSX-2 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 558 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82929 A2B CHO cells HUMAN 3H-PSB-603 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82930 A3 CHO cells HUMAN 3H-PSB-11 1,3-Dimethyl-8-(3-(thiazol-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82931 A1 CHO cells HUMAN 3H-CCPA 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 21.8 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82932 A1 CORTICAL MEMBRANES RAT 3H-CCPA 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 10.1 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82933 A2A CHO cells HUMAN 3H-MSX-2 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 426 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82934 A2A Striatal Membranes RAT 3H-MSX-2 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 375 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82935 A2B CHO cells HUMAN 3H-PSB-603 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82936 A3 CHO cells HUMAN 3H-PSB-11 1,3-Dimethyl-8-(3-(thiophen-2-yl)benzyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 6490 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82937 A1 CHO cells HUMAN 3H-CCPA 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 59.1 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82938 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 21.4 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82939 A2A CHO cells HUMAN 3H-MSX-2 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 437 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82940 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 184 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82941 A2B CHO cells HUMAN 3H-PSB-603 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82942 A3 CHO cells HUMAN 3H-PSB-11 8-(3-(1H-Pyrrol-1-yl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82943 A1 CHO cells HUMAN 3H-CCPA 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 61.8 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82944 A1 CORTICAL MEMBRANES RAT 3H-CCPA 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 32.9 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82945 A2A CHO cells HUMAN 3H-MSX-2 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 569 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82946 A2A Striatal Membranes RAT 3H-MSX-2 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 335 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82947 A2B CHO cells HUMAN 3H-PSB-603 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82948 A3 CHO cells HUMAN 3H-PSB-11 1,3-Dimethyl-8-(thiophen-3-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]-purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82949 A1 CORTICAL MEMBRANES RAT 3H-CCPA (R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82950 A2A Striatal Membranes RAT 3H-MSX-2 (R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1210 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82951 A2B CHO cells HUMAN 3H-PSB-603 (R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82952 A3 CHO cells HUMAN 3H-PSB-11 (R,S)-8-(1-(4-Fluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82953 A1 CHO cells HUMAN 3H-CCPA 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 116 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82954 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 86.8 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82955 A2A CHO cells HUMAN 3H-MSX-2 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 94.3 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82956 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 993 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82957 A2B CHO cells HUMAN 3H-PSB-603 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82958 A3 CHO cells HUMAN 3H-PSB-11 8-(2,3-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82959 A1 CHO cells HUMAN 3H-CCPA 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 227 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82960 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 25.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82961 A2A CHO cells HUMAN 3H-MSX-2 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 782 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82962 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 402 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82963 A3 CHO cells HUMAN 3H-PSB-603 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82964 A3 CHO cells HUMAN 3H-PSB-11 8-(2,6-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82965 A1 CHO cells HUMAN 3H-CCPA 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 296 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82966 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 33.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82967 A2A CHO cells HUMAN 3H-MSX-2 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 662 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82968 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 174 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82969 A2B CHO cells HUMAN 3H-PSB-603 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82970 A3 CHO cells HUMAN 3H-PSB-11 8-(2,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 7840 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82971 A1 CHO cells HUMAN 3H-CCPA 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 257 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82972 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 44.4 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82973 A2A CHO cells HUMAN 3H-MSX-2 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 2440 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82974 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 927 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82975 A2B CHO cells HUMAN 3H-PSB-603 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82976 A3 CHO cells HUMAN 3H-PSB-11 8-(3,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82977 A1 CHO cells HUMAN 3H-CCPA 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 89.8 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82978 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 14.1 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82979 A2A CHO cells HUMAN 3H-MSX-2 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 320 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82980 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 484 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82981 A2B CHO cells HUMAN 3H-PSB-603 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82982 A3 CHO cells HUMAN 3H-PSB-11 8-(2,5-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82983 A1 CHO cells HUMAN 3H-CCPA 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 791 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82984 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 351 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82985 A2A CHO cells HUMAN 3H-MSX-2 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1510 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82986 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 322 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82987 A2B CHO cells HUMAN 3H-PSB-603 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82988 A3 CHO cells HUMAN 3H-PSB-11 8-(3,4-Dichlorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82989 A1 CHO cells HUMAN 3H-CCPA 8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 376 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82990 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 238 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82991 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 3660 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82992 A2B CHO cells HUMAN 3H-PSB-603 8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82993 A3 CHO cells HUMAN 3H-PSB-11 8-(2,6-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82994 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82995 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82996 A2B CHO cells HUMAN 3H-PSB-603 8-(2,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82997 A3 CHO cells HUMAN 3H-PSB-11 8-(2,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82998 A1 CHO cells HUMAN 3H-CCPA 8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 687 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
82999 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 77.1 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83000 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83001 A2B CHO cells HUMAN 3H-PSB-603 8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83002 A3 CHO cells HUMAN 3H-PSB-11 8-(2,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83003 A1 CHO cells HUMAN 3H-CCPA 8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 794 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83004 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 85.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83005 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1220 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83006 A2B CHO cells HUMAN 3H-PSB-603 8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83007 A3 CHO cells HUMAN 3H-PSB-11 8-(3,5-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83008 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83009 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83010 A2B CHO cells HUMAN 3H-PSB-603 8-(3,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83011 A3 CHO cells HUMAN 3H-PSB-11 8-(3,4-Difluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83012 A1 CHO cells HUMAN 3H-CCPA 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 231 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83013 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 107 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83014 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1270 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83015 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 518 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83016 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83017 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Chloro-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83018 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83019 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83020 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83021 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Chloro-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83022 A1 CHO cells HUMAN 3H-CCPA 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 243 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83023 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 54.4 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83024 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 812 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83025 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 624 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83026 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83027 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83028 A1 CHO cells HUMAN 3H-CCPA 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 186 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83029 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 99.9 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83030 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83031 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 758 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83032 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83033 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Chloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83034 A1 CHO cells HUMAN 3H-CCPA 8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 384 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83035 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 95.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83036 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1070 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83037 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83038 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Chloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83039 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83040 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1330 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83041 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83042 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Chloro-3-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83043 A1 CHO cells HUMAN 3H-CCPA 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 150 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83044 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 28.9 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83045 A2A CHO cells HUMAN 3H-MSX-2 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1150 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83046 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 681 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83047 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83048 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83049 A1 CHO cells HUMAN 3H-CCPA 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 247 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83050 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 144 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83051 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1420 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83052 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 652 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83053 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83054 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83055 A1 CHO cells HUMAN 3H-CCPA 8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 84.3 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83056 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 151 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83057 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1020 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83058 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83059 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Fluoro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83060 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83061 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 2570 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83062 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83063 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83064 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83065 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1870 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83066 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83067 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Fluoro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83068 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83069 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83070 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 100 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83071 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83072 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83073 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83074 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Fluoro-4-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83075 A1 CHO cells HUMAN 3H-CCPA 8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 678 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83076 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 611 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83077 A2A Striatal Membranes RAT 3H-MSX-2 8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83078 A2B CHO cells HUMAN 3H-PSB-603 8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83079 A3 CHO cells HUMAN 3H-PSB-11 8-(5-Fluoro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83080 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83081 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1160 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83082 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83083 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83084 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83085 A2A Striatal Membranes RAT 3H-MSX-2 8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83086 A2B CHO cells HUMAN 3H-PSB-603 8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83087 A3 CHO cells HUMAN 3H-PSB-11 8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83088 A1 CHO cells HUMAN 3H-CCPA 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 67.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83089 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 23 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83090 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 261 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83091 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 358 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83092 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83093 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83094 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Fluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83095 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Fluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83096 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Fluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83097 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Fluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83098 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83099 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83100 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83101 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Bromo-4-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83102 A1 CHO cells HUMAN 3H-CCPA 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 76.5 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83103 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 36 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83104 A2A CHO cells HUMAN 3H-MSX-2 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 4730 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83105 A2A Striatal Membranes RAT 3H-MSX-2 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 991 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83106 A2B CHO cells HUMAN 3H-PSB-603 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83107 A3 CHO cells HUMAN 3H-PSB-11 8-(5-Bromo-2-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83108 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83109 A2A CHO cells HUMAN 3H-MSX-2 8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1910 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83110 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 729 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83111 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83112 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Fluoro-4-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83113 A1 CHO cells HUMAN 3H-CCPA 8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 51.9 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83114 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 46 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83115 A2A Striatal Membranes RAT 3H-MSX-2 8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1100 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83116 A2B CHO cells HUMAN 3H-PSB-603 8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83117 A3 CHO cells HUMAN 3H-PSB-11 8-(3-Fluoro-5-methylbenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83118 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,5-bis(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83119 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,5-bis(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83120 A2B CHO cells HUMAN 3H-PSB-603 8-(3,5-bis(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83121 A3 CHO cells HUMAN 3H-PSB-11 8-(3,5-bis(Trifluoromethyl)benzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83122 A1 CHO cells HUMAN 3H-CCPA 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 217 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83123 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 134 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83124 A2A CHO cells HUMAN 3H-MSX-2 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1120 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83125 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 236 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83126 A2B CHO cells HUMAN 3H-PSB-603 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83127 A3 CHO cells HUMAN 3H-PSB-11 8-(2,3-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83128 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,4-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83129 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,4-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83130 A2B CHO cells HUMAN 3H-PSB-603 8-(2,4-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 100 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83131 A3 CHO cells HUMAN 3H-PSB-11 8-(2,4-Dimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83132 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(Benzo[d][1,3]dioxol-5-ylmethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83133 A2A Striatal Membranes RAT 3H-MSX-2 8-(Benzo[d][1,3]dioxol-5-ylmethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83134 A2B CHO cells HUMAN 3H-PSB-603 8-(Benzo[d][1,3]dioxol-5-ylmethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83135 A3 CHO cells HUMAN 3H-PSB-11 8-(Benzo[d][1,3]dioxol-5-ylmethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83136 A1 CORTICAL MEMBRANES RAT 3H-CCPA (R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1530 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83137 A2A CHO cells HUMAN 3H-MSX-2 (R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 692 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83138 A2A Striatal Membranes RAT 3H-MSX-2 (R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 688 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83139 A2B CHO cells HUMAN 3H-PSB-603 (R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83140 A3 CHO cells HUMAN 3H-PSB-11 (R,S)-8-(1-(3,4-Dichlorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83141 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,4,5-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83142 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,4,5-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1670 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83143 A2B CHO cells HUMAN 3H-PSB-603 8-(3,4,5-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83144 A3 CHO cells HUMAN 3H-PSB-11 8-(3,4,5-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 100 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83145 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,4,6-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83146 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,4,6-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1880 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83147 A2B CHO cells HUMAN 3H-PSB-603 8-(2,4,6-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83148 A3 CHO cells HUMAN 3H-PSB-11 8-(2,4,6-Trifluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83149 A1 CHO cells HUMAN 3H-CCPA 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 91.4 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83150 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 73 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83151 A2A CHO cells HUMAN 3H-MSX-2 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1080 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83152 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 897 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83153 A2B CHO cells HUMAN 3H-PSB-603 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83154 A3 CHO cells HUMAN 3H-PSB-11 8-(2,3-Dichloro-6-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 100 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83155 A1 CHO cells HUMAN 3H-CCPA 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 217 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83156 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 111 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83157 A2A CHO cells HUMAN 3H-MSX-2 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 268 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83158 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 603 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83159 A2B CHO cells HUMAN 3H-PSB-603 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83160 A3 CHO cells HUMAN 3H-PSB-11 8-(2,4-Dichloro-5-fluorobenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83161 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(4,5-Difluoro-2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83162 A2A Striatal Membranes RAT 3H-MSX-2 8-(4,5-Difluoro-2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1390 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83163 A2B CHO cells HUMAN 3H-PSB-603 8-(4,5-Difluoro-2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83164 A3 CHO cells HUMAN 3H-PSB-11 8-(4,5-Difluoro-2-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83165 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,3-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83166 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,3-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83167 A2B CHO cells HUMAN 3H-PSB-603 8-(2,3-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83168 A3 CHO cells HUMAN 3H-PSB-11 8-(2,3-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 300 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83169 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,5-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83170 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,5-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 2670 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83171 A2B CHO cells HUMAN 3H-PSB-603 8-(3,5-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83172 A3 CHO cells HUMAN 3H-PSB-11 8-(3,5-Difluoro-4-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione >10000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83173 A1 CHO cells HUMAN 3H-CCPA 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 752 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83174 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 170 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83175 A2A CHO cells HUMAN 3H-MSX-2 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 3810 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83176 A2A Striatal Membranes RAT 3H-MSX-2 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 823 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83177 A2B CHO cells HUMAN 3H-PSB-603 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83178 A3 CHO cells HUMAN 3H-PSB-11 8-(2-Chloro-6-fluoro-3-methoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione 100 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83179 A1 CHO cells HUMAN 3H-CCPA 8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 3040 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83180 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 343 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83181 A2A Striatal Membranes RAT 3H-MSX-2 8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1700 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83182 A2B CHO cells HUMAN 3H-PSB-603 8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83183 A3 CHO cells HUMAN 3H-PSB-11 8-(2,4,6-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83184 A1 CORTICAL MEMBRANES RAT 3H-CCPA 8-(3,4,5-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1500 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83185 A2A Striatal Membranes RAT 3H-MSX-2 8-(3,4,5-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83186 A2B CHO cells HUMAN 3H-PSB-603 8-(3,4,5-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83187 A3 CHO cells HUMAN 3H-PSB-11 8-(3,4,5-Trimethoxybenzyl)-1,3-dimethyl-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione 1000 Brunschweiger A et al 2014 Jan 15, 2025 Jan 15, 2025
83188 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-Mefloquine 9100 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83189 5-HT2A CLONED HUMAN 125I-DOI (+)-Mefloquine 341 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83190 5-HT2C CLONED HUMAN 125I-DOI (+)-Mefloquine 5730 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83191 5-HT2C CLONED HUMAN 125I-DOI (-)-Mefloquine 3870 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83192 5-HT2A CLONED HUMAN 125I-DOI (-)-Mefloquine 1510 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83193 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83194 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Chloroquine 6000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83195 5-HT2A CLONED HUMAN 125I-DOI Chloroquine 6300 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83196 5-HT2C CLONED HUMAN 125I-DOI Chloroquine 6200 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83197 5-HT2C CLONED HUMAN 125I-DOI 5-Hydroxy Tryptamine 4.31 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83198 5-HT2A CLONED HUMAN 125I-DOI 5-Hydroxy Tryptamine 9.1 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83199 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 5-Hydroxy Tryptamine 2.67 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83200 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LSD 2.78 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83201 5-HT2A CLONED HUMAN 125I-DOI LSD 0.71 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83202 5-HT2C CLONED HUMAN 125I-DOI LSD 2.91 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83203 5-HT2C CLONED HUMAN 125I-DOI DMT 166 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83204 5-HT2A CLONED HUMAN 125I-DOI DMT 210 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83205 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DMT 450 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83206 5-HT1A CLONED HUMAN 3H-8-OH-DPAT DOM >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83207 5-HT2A CLONED HUMAN 125I-DOI DOM 4.3 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83208 5-HT2C CLONED HUMAN 125I-DOI DOM 25.7 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83209 5-HT2C CLONED HUMAN 125I-DOI KETANSERIN 117 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83210 5-HT2A CLONED HUMAN 125I-DOI KETANSERIN 7.6 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83211 5-HT1A CLONED HUMAN 3H-8-OH-DPAT KETANSERIN 6510 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83212 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ro 60-0175 6680 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83213 5-HT2A CLONED HUMAN 125I-DOI Ro 60-0175 13.1 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83214 5-HT2C CLONED HUMAN 125I-DOI Ro 60-0175 7.3 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83215 5-HT2C CLONED HUMAN 125I-DOI SB242087 11.4 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83216 5-HT2A CLONED HUMAN 125I-DOI SB242087 120 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83217 5-HT1A CLONED HUMAN 3H-8-OH-DPAT SB242087 9300 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83218 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide 1.21 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83219 5-HT2A CLONED HUMAN 125I-DOI Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide 331 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83220 5-HT2C CLONED HUMAN 125I-DOI Cyclohexanecarboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-pyridin-2-yl-amide 3000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83221 5-HT2A CLONED HUMAN 125I-DOI 5-Hydroxy Tryptamine 3.734 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83222 5-HT2A CLONED HUMAN 125I-DOI (+)-Mefloquine 2400 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83223 5-HT2A CLONED HUMAN 125I-DOI (-)-Mefloquine 4260 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83224 5-HT2A CLONED HUMAN 125I-DOI Chloroquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83225 5-HT2A CLONED HUMAN 125I-DOI LSD 0.72 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83226 5-HT2A CLONED HUMAN 125I-DOI DOM 2.06 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83227 5-HT2A CLONED HUMAN 125I-DOI DMT 53 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83228 5-HT2A CLONED HUMAN 125I-DOI KETANSERIN 4.1 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83229 5-HT2A CLONED HUMAN 125I-DOI MDL 100907 0.67 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83230 5-HT2A CLONED HUMAN 3H-KETANSERIN MDL 100907 0.048 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83231 5-HT2A CLONED HUMAN 3H-KETANSERIN KETANSERIN 0.77 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83232 5-HT2A CLONED HUMAN 3H-KETANSERIN DMT 175 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83233 5-HT2A CLONED HUMAN 3H-KETANSERIN DOM 13.7 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83234 5-HT2A CLONED HUMAN 3H-KETANSERIN LSD 0.475 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83235 5-HT2A CLONED HUMAN 3H-KETANSERIN Chloroquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83236 5-HT2A CLONED HUMAN 3H-KETANSERIN (-)-Mefloquine 3280 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83237 5-HT2A CLONED HUMAN 3H-KETANSERIN (+)-Mefloquine 2940 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83238 5-HT2A CLONED HUMAN 3H-KETANSERIN 5-Hydroxy Tryptamine 12.6 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83239 DAT CLONED HUMAN 125I-RTI-55 (+)-Mefloquine 6400 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83240 NET CLONED HUMAN 125I-RTI-55 (+)-Mefloquine 5300 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83241 SERT CLONED HUMAN 125I-RTI-55 (+)-Mefloquine 229 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83242 SERT CLONED HUMAN 125I-RTI-55 (-)-Mefloquine 2900 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83243 NET CLONED HUMAN 125I-RTI-55 (-)-Mefloquine 5280 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83244 DAT CLONED HUMAN 125I-RTI-55 (-)-Mefloquine 6500 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83245 DAT CLONED HUMAN 125I-RTI-55 Chloroquine 8000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83246 NET CLONED HUMAN 125I-RTI-55 Chloroquine 1052 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83247 SERT CLONED HUMAN 125I-RTI-55 Chloroquine 8300 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83248 SERT CLONED HUMAN 125I-RTI-55 Quinine 4000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83249 NET CLONED HUMAN 125I-RTI-55 Quinine 5500 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83250 DAT CLONED HUMAN 125I-RTI-55 Quinine 8300 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83251 DAT CLONED HUMAN 125I-RTI-55 LSD >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83252 NET CLONED HUMAN 125I-RTI-55 LSD 5600 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83253 SERT CLONED HUMAN 125I-RTI-55 LSD >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83254 SERT CLONED HUMAN 125I-RTI-55 COCAINE 450 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83255 NET CLONED HUMAN 125I-RTI-55 COCAINE 410 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83256 DAT CLONED HUMAN 125I-RTI-55 COCAINE 416 Janowsky A et al 2014 Jan 15, 2025 Jan 15, 2025
83257 D1 CLONED HUMAN 3H-SCH23390 (+)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83258 D1 CLONED HUMAN 3H-SCH23390 (-)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83259 D1 CLONED HUMAN 3H-SCH23390 Chloroquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83260 D1 CLONED HUMAN 3H-SCH23390 LSD 273 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83261 D1 CLONED HUMAN 3H-SCH23390 DOPAMINE 4300 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83262 D1 CLONED HUMAN 3H-SCH23390 SKF 38393 258 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83263 D1 CLONED HUMAN 3H-SCH23390 SCH 23390 0.491 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83264 D1 CLONED HUMAN 3H-SCH23390 QUINPIROLE >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83265 D1 CLONED HUMAN 3H-SCH23390 BUTACLAMOL 4.1 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83266 D2 CLONED HUMAN 3H-YM 09151-2 BUTACLAMOL 2.04 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83267 D3 CLONED HUMAN 3H-YM 09151-2 BUTACLAMOL 4 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83268 D4 CLONED HUMAN 3H-YM 09151-2 BUTACLAMOL 255 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83269 D4 CLONED HUMAN 3H-YM 09151-2 QUINPIROLE 262 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83270 D3 CLONED HUMAN 3H-YM 09151-2 QUINPIROLE 52.8 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83271 D2 CLONED HUMAN 3H-YM 09151-2 QUINPIROLE 2780 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83272 D2 CLONED HUMAN 3H-YM 09151-2 SCH 23390 887 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83273 D3 CLONED HUMAN 3H-YM 09151-2 SCH 23390 1920 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83274 D4 CLONED HUMAN 3H-YM 09151-2 SCH 23390 9700 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83275 D4 CLONED HUMAN 3H-YM 09151-2 SKF 38393 >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83276 D3 CLONED HUMAN 3H-YM 09151-2 SKF 38393 4300 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83277 D2 CLONED HUMAN 3H-YM 09151-2 SKF 38393 4800 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83278 D2 CLONED HUMAN 3H-YM 09151-2 DOPAMINE 1710 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83279 D3 CLONED HUMAN 3H-YM 09151-2 DOPAMINE 61 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83280 D4 CLONED HUMAN 3H-YM 09151-2 DOPAMINE 630 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83281 D4 CLONED HUMAN 3H-YM 09151-2 LSD 330 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83282 D3 CLONED HUMAN 3H-YM 09151-2 LSD 27.1 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83283 D2 CLONED HUMAN 3H-YM 09151-2 LSD 38.8 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83284 D2 CLONED HUMAN 3H-YM 09151-2 Chloroquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83285 D3 CLONED HUMAN 3H-YM 09151-2 Chloroquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83286 D4 CLONED HUMAN 3H-YM 09151-2 Chloroquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83287 D4 CLONED HUMAN 3H-YM 09151-2 (-)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83288 D3 CLONED HUMAN 3H-YM 09151-2 (-)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83289 D2 CLONED HUMAN 3H-YM 09151-2 (-)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83290 D2 CLONED HUMAN 3H-YM 09151-2 (+)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83291 D3 CLONED HUMAN 3H-YM 09151-2 (+)-Mefloquine 1960 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83292 D4 CLONED HUMAN 3H-YM 09151-2 (+)-Mefloquine >10000 Janowsky A et al 2014 Jan 15, 2025 Jan 28, 2025
83293 M1 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 9.33254 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83294 M2 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 43.6516 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83295 M3 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 14.4544 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83296 M4 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 30.903 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83297 M5 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 54.9541 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83298 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3.89045 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83299 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.933254 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83300 M3 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.851138 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83301 M2 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 12.3027 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83302 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.524807 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83303 M1 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83304 M2 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 8709.64 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83305 M3 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83306 M4 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83307 M5 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83308 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83309 M2 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 5370.32 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83310 M3 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83311 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83312 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83313 M5 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide and 1-((2R*,6R*)-6-(4-Benzylphenyl)- 1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 7413.1 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83314 M4 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide and 1-((2R*,6R*)-6-(4-Benzylphenyl)- 1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83315 M3 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide and 1-((2R*,6R*)-6-(4-Benzylphenyl)- 1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83316 M2 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide and 1-((2R*,6R*)-6-(4-Benzylphenyl)- 1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 4897.79 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83317 M1 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide and 1-((2R*,6R*)-6-(4-Benzylphenyl)- 1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83318 M1 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3162.28 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83319 M2 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3388.44 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83320 M3 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83321 M4 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3715.35 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83322 M5 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2630.27 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83323 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1122.02 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83324 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1995.26 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83325 M3 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1698.24 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83326 M2 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 194.984 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83327 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3090.3 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83328 M1 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83329 M2 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 3019.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83330 M3 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83331 M4 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83332 M5 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 6165.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83333 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1819.7 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83334 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 3801.89 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83335 M3 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1318.26 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83336 M2 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 416.869 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83337 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 6760.83 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83338 M1 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 8317.64 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83339 M2 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 7413.1 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83340 M3 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83341 M4 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83342 M5 CLONED HUMAN 3H-NMS 1-((2R*,6S*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 6165.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83343 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1584.89 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83344 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 6309.57 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83345 M3 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 2344.23 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83346 M2 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 199.526 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83347 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 5128.61 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83348 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2344.23 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83349 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 8709.64 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83350 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 7244.36 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83351 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 7943.28 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83352 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83353 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83354 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83355 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83356 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83357 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83358 M1 CLONED HUMAN 3H-NMS 1-(5,5-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 36.3078 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83359 M2 CLONED HUMAN 3H-NMS 1-(5,5-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 177.828 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83360 M3 CLONED HUMAN 3H-NMS 1-(5,5-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 134.896 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83361 M4 CLONED HUMAN 3H-NMS 1-(5,5-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 154.882 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83362 M5 CLONED HUMAN 3H-NMS 1-(5,5-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 158.489 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83363 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 35.4813 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83364 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 70.7946 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83365 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 37.1535 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83366 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 54.9541 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83367 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 9.77237 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83368 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 15.4882 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83369 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 60.256 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83370 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 43.6516 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83371 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 58.8844 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83372 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Cyclohexyl-5-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 47.863 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83373 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3235.94 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83374 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2511.89 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83375 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1698.24 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83376 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1348.96 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83377 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 524.807 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83378 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 831.764 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83379 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 870.964 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83380 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2398.83 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83381 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3019.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83382 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-Benzhydryl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 6309.57 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83383 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83384 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83385 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83386 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83387 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83388 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83389 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3235.94 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83390 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83391 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83392 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-([1,1′-Biphenyl]-4-yl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83393 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2951.21 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83394 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83395 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2238.72 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83396 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2238.72 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83397 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83398 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83399 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83400 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83401 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83402 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-Benzylphenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83403 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83404 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1995.26 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83405 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 977.237 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83406 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 199.526 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83407 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3715.35 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83408 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2691.53 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83409 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1380.38 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83410 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 4466.84 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83411 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 7244.36 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83412 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylthio)phenyl)-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3981.07 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83413 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 6165.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83414 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83415 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83416 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 3019.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83417 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83418 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 6760.83 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83419 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 416.869 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83420 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1318.26 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83421 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 3801.89 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83422 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfinyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 1905.46 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83423 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 8912.51 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83424 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83425 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 7244.36 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83426 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide 407.38 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83427 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83428 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83429 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83430 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83431 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83432 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5-(4-(Phenylsulfonyl)phenyl)-1,4-dioxan-2-yl)- N,N,N-trimethylmethanaminium Iodide >10000 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83433 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6S*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 4570.88 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83434 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6S*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 5623.41 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83435 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6S*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 4677.35 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83436 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6S*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1905.46 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83437 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6S*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1412.54 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83438 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 501.187 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83439 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2238.72 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83440 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1548.82 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83441 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3981.07 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83442 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3019.95 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83443 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 616.595 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83444 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 398.107 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83445 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 354.813 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83446 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 239.883 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83447 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*,6R*)-5,6-Diphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 64.5654 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83448 M1 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 676.083 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83449 M2 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 4365.16 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83450 M3 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1995.26 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83451 M4 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3890.45 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83452 M5 CLONED HUMAN 3H-NMS 1-((2R*,5S*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 3981.07 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83453 M5 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1445.44 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83454 M4 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1174.9 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83455 M3 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 1096.48 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83456 M2 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 2137.96 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83457 M1 CLONED HUMAN 3H-NMS 1-((2R*,5R*)-5,6,6-Triphenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 549.541 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83458 M1 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.301995 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83459 M2 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 6.0256 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83460 M3 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.891251 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83461 M4 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.676083 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83462 M5 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide 0.660693 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83463 M5 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 20.893 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83464 M4 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 35.4813 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83465 M3 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 30.903 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83466 M2 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 13.8038 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83467 M1 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N,N-trimethylmethanaminium Iodide [(2R,6R)-(+) 5.01187 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83468 M1 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 1.38038 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83469 M2 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 13.1826 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83470 M3 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 1.90546 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83471 M4 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 2.39883 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83472 M5 CLONED HUMAN 3H-NMS 1-((2R*,6R*)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine 2.39883 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83473 M5 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+) 69.1831 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83474 M4 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+) 97.7237 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83475 M3 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+) 186.209 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83476 M2 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+) 67.6083 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83477 M1 CLONED HUMAN 3H-NMS 1-((2R,6R)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (+) 20.893 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83478 M1 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 0.794328 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83479 M2 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 7.94328 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83480 M3 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 0.954993 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83481 M4 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 0.812831 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83482 M5 CLONED HUMAN 3H-NMS 1-((2S,6S)-6-Cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine (-) 1.47911 Del Bello F et al 2020 Jan 15, 2025 Jan 15, 2025
83483 NET HEK293 cells HUMAN 3H-Nisoxetine MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83484 DAT HEK293 cells HUMAN 3H-WIN 35,428 MDMA 6500 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83485 SERT HEK293 cells HUMAN 3H-CITALOPRAM MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83486 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83487 5-HT2A HEK293 cells HUMAN 3H-KETANSERIN MDMA 7800 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83488 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83489 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN MDMA 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83490 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83491 D1 HEK293 cells HUMAN 3H-SCH23390 MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83492 D2 HEK293 cells HUMAN 3H-SPIPERONE MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83493 D3 HEK293 cells HUMAN 3H-SPIPERONE MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83494 H1 HEK293 cells HUMAN 3H-PYRILAMINE MDMA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83495 D1 HEK293 cells RAT 3H-RO5166017 MDMA 370 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83496 D1 HEK293 cells MOUSE 3H-RO5166017 MDMA 2400 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83497 NET HEK293 cells HUMAN 3H-Nisoxetine MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83498 DAT HEK293 cells HUMAN 3H-WIN 35,428 MBDB 3100 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83499 SERT HEK293 cells HUMAN 3H-CITALOPRAM MBDB 5800 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83500 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83501 5-HT2A HEK293 cells HUMAN 3H- Ketanserin MBDB 6620 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83502 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83503 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN MBDB 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83504 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83505 D1 HEK293 cells HUMAN 3H-SCH23390 MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83506 D3 HEK293 cells HUMAN 3H-SPIPERONE MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83507 H1 HEK293 cells HUMAN 3H-PYRILAMINE MBDB >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83508 D1 HEK293 cells RAT 3H-RO5166017 MBDB 1200 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83509 D1 HEK293 cells MOUSE 3H-RO166017 MBDB 3600 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83510 NET HEK293 cells HUMAN 3H-Nisoxetine MDEA 6170 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83511 DAT HEK293 cells HUMAN 3H-WIN 35,428 MDEA 1350 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83512 SERT HEK293 cells HUMAN 3H-CITALOPRAM MDEA 4320 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83513 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83514 5-HT2A HEK293 cells HUMAN 3H-KETANSERIN MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83515 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83516 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN MDEA 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83517 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83518 D1 HEK293 cells HUMAN 3H-SCH23390 MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83519 D3 HEK293 cells HUMAN 3H-SPIPERONE MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83520 H1 HEK293 cells HUMAN 3H-PYRILAMINE MDEA >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83521 D1 HEK293 cells RAT 3H-RO5166017 MDEA 320 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83522 D1 HEK293 cells MOUSE 3H-RO5166017 MDEA 4900 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83523 NET HEK293 cells HUMAN 3H-Nisoxetine Ethylone 9890 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83524 DAT HEK293 cells HUMAN 3H-WIN 35,428 Ethylone 1430 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83525 SERT HEK293 cells HUMAN 3H-CITALOPRAM Ethylone 9040 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83526 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83527 5-HT2A HEK293 cells HUMAN 3H-KETANSERIN Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83528 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83529 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Ethylone 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83530 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83531 D1 HEK293 cells HUMAN 3H-SCH23390 Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83532 D3 HEK293 cells HUMAN 3H-SPIPERONE Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83533 H1 HEK293 cells HUMAN 3H-PYRILAMINE Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83534 D1 HEK293 cells RAT 3H-RO5166017 Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83535 D1 HEK293 cells MOUSE 3H-RO5166017 Ethylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83536 NET HEK293 cells HUMAN 3H-Nisoxetine mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83537 DAT HEK293 cells HUMAN 3H-WIN 35,428 mephedrone 3400 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83538 SERT HEK293 cells HUMAN 3H-CITALOPRAM mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83539 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83540 5-HT2A HEK293 cells HUMAN 3H- Ketanserin mephedrone 2100 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83541 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83542 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN mephedrone 3480 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83543 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83544 D1 HEK293 cells HUMAN 3H-SCH23390 mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83545 D2 HEK293 cells HUMAN 3H-SPIPERONE mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83546 D3 HEK293 cells HUMAN 3H-SPIPERONE mephedrone 9200 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83547 H1 HEK293 cells HUMAN 3H-PYRILAMINE mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83548 D1 HEK293 cells RAT 3H-RO5166017 mephedrone 4300 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83549 D1 HEK293 cells MOUSE 3H-RO5166017 mephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83550 NET HEK293 cells HUMAN 3H-Nisoxetine Naphyrone 180 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83551 DAT HEK293 cells HUMAN 3H-WIN 35,428 Naphyrone 40 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83552 SERT HEK293 cells HUMAN 3H-CITALOPRAM Naphyrone 180 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83553 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Naphyrone 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83554 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Naphyrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83555 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Naphyrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83556 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Naphyrone 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83557 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Naphyrone 8000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83558 D1 HEK293 cells HUMAN 3H-SCH23390 Naphyrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83559 D3 HEK293 cells HUMAN 3H-SPIPERONE Naphyrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83560 H1 HEK293 cells HUMAN 3H-PYRILAMINE Naphyrone 2280 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83561 D1 HEK293 cells RAT 3H-RO5166017 Naphyrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83562 D1 HEK293 cells MOUSE 3H-RO5166017 Naphyrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83563 NET HEK293 cells HUMAN 3H-Nisoxetine Butylone 8130 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83564 DAT HEK293 cells HUMAN 3H-WIN 35,428 Butylone 440 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83565 SERT HEK293 cells HUMAN 3H-CITALOPRAM Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83566 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83567 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83568 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83569 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Butylone 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83570 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83571 D1 HEK293 cells HUMAN 3H-SCH23390 Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83572 D3 HEK293 cells HUMAN 3H-SPIPERONE Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83573 H1 HEK293 cells HUMAN 3H-PYRILAMINE Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83574 D1 HEK293 cells RAT 3H-RO5166017 Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83575 D1 HEK293 cells MOUSE 3H-RO5166017 Butylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83576 NET HEK293 cells HUMAN 3H-Nisoxetine COCAINE 4470 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83577 DAT HEK293 cells HUMAN 3H-WIN 35,428 COCAINE 280 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83578 SERT HEK293 cells HUMAN 3H-CITALOPRAM COCAINE 1100 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83579 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83580 5-HT2A HEK293 cells HUMAN 3H- Ketanserin COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83581 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83582 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN COCAINE 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83583 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83584 D1 HEK293 cells HUMAN 3H-SCH23390 COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83585 D2 HEK293 cells HUMAN 3H-SPIPERONE COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83586 D3 HEK293 cells HUMAN 3H-SPIPERONE COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83587 H1 HEK293 cells HUMAN 3H-PYRILAMINE COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83588 D1 HEK293 cells RAT 3H-RO5166017 COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83589 D1 HEK293 cells MOUSE 3H-RO5166017 COCAINE >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83590 NET HEK293 cells HUMAN 3H-Nisoxetine Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83591 DAT HEK293 cells HUMAN 3H-WIN 35,428 Methylone 2730 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83592 SERT HEK293 cells HUMAN 3H-CITALOPRAM Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83593 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83594 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83595 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83596 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Methylone 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83597 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83598 D1 HEK293 cells HUMAN 3H-SCH23390 Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83599 D2 HEK293 cells HUMAN 3H-SPIPERONE Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83600 D3 HEK293 cells HUMAN 3H-SPIPERONE Methylone 9200 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83601 H1 HEK293 cells HUMAN 3H-PYRILAMINE Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83602 D1 HEK293 cells RAT 3H-RO5166017 Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83603 D1 HEK293 cells MOUSE 3H-RO5166017 Methylone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83604 NET HEK293 cells HUMAN 3H-Nisoxetine Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83605 DAT HEK293 cells HUMAN 3H-WIN 35,428 Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83606 SERT HEK293 cells HUMAN 3H-CITALOPRAM Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83607 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83608 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Flephedrone 1400 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83609 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83610 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Flephedrone 1520 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83611 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83612 D1 HEK293 cells HUMAN 3H-SCH23390 Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83613 D2 HEK293 cells HUMAN 3H-SPIPERONE Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83614 D3 HEK293 cells HUMAN 3H-SPIPERONE Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83615 H1 HEK293 cells HUMAN 3H-PYRILAMINE Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83616 D1 HEK293 cells RAT 3H-RO5166017 Flephedrone 5400 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83617 D1 HEK293 cells MOUSE 3H-RO5166017 Flephedrone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83618 NET HEK293 cells HUMAN 3H-Nisoxetine Cathinone 3500 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83619 DAT HEK293 cells HUMAN 3H-WIN 35,428 Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83620 SERT HEK293 cells HUMAN 3H-CITALOPRAM Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83621 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83622 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83623 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83624 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Cathinone 5400 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83625 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Cathinone 8900 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83626 D1 HEK293 cells HUMAN 3H-SCH23390 Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83627 D2 HEK293 cells HUMAN 3H-SPIPERONE Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83628 D3 HEK293 cells HUMAN 3H-SPIPERONE Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83629 H1 HEK293 cells HUMAN 3H-PYRILAMINE Cathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83630 D1 HEK293 cells RAT 3H-RO5166017 Cathinone 2200 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83631 D1 HEK293 cells MOUSE 3H-RO5166017 Cathinone 2100 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83632 NET HEK293 cells HUMAN 3H-Nisoxetine Methcathinone 1450 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83633 DAT HEK293 cells HUMAN 3H-WIN 35,428 Methcathinone 1280 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83634 SERT HEK293 cells HUMAN 3H-CITALOPRAM Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83635 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83636 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Methcathinone 3000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83637 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83638 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Methcathinone 3930 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83639 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83640 D1 HEK293 cells HUMAN 3H-SCH23390 Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83641 D2 HEK293 cells HUMAN 3H-SPIPERONE Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83642 D3 HEK293 cells HUMAN 3H-SPIPERONE Methcathinone 9200 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83643 H1 HEK293 cells HUMAN 3H-PYRILAMINE Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83644 D1 HEK293 cells RAT 3H-RO5166017 Methcathinone 4100 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83645 D1 HEK293 cells MOUSE 3H-RO5166017 Methcathinone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83646 NET HEK293 cells HUMAN 3H-Nisoxetine Amphetamine 1000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83647 DAT HEK293 cells HUMAN 3H-WIN 35,428 Amphetamine 5680 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83648 SERT HEK293 cells HUMAN 3H-CITALOPRAM Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83649 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Amphetamine 6740 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83650 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83651 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83652 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Amphetamine 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83653 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Amphetamine 2800 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83654 D1 HEK293 cells HUMAN 3H-SCH23390 Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83655 D2 HEK293 cells HUMAN 3H-SPIPERONE Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83656 D3 HEK293 cells HUMAN 3H-SPIPERONE Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83657 H1 HEK293 cells HUMAN 3H-PYRILAMINE Amphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83658 D1 HEK293 cells RAT 3H-RO5166017 Amphetamine 230 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83659 D1 HEK293 cells MOUSE 3H-RO5166017 Amphetamine 90 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83660 NET HEK293 cells HUMAN 3H-Nisoxetine Methamphetamine 4280 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83661 DAT HEK293 cells HUMAN 3H-WIN 35,428 Methamphetamine 1850 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83662 SERT HEK293 cells HUMAN 3H-CITALOPRAM Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83663 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT Methamphetamine 8070 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83664 5-HT2A HEK293 cells HUMAN 3H- Ketanserin Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83665 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83666 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN Methamphetamine 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83667 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE Methamphetamine 6100 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83668 D1 HEK293 cells HUMAN 3H-SCH23390 Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83669 D2 HEK293 cells HUMAN 3H-SPIPERONE Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83670 D3 HEK293 cells HUMAN 3H-SPIPERONE Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83671 H1 HEK293 cells HUMAN 3H-PYRILAMINE Methamphetamine >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83672 D1 HEK293 cells RAT 3H-RO5166017 Methamphetamine 350 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83673 D1 HEK293 cells MOUSE 3H-RO5166017 Methamphetamine 550 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83674 NET HEK293 cells HUMAN 3H-Nisoxetine pyrovalerone 60 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83675 DAT HEK293 cells HUMAN 3H-WIN 35,428 pyrovalerone 30 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83676 SERT HEK293 cells HUMAN 3H-CITALOPRAM pyrovalerone 4970 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83677 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83678 5-HT2A HEK293 cells HUMAN 3H- Ketanserin pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83679 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83680 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN pyrovalerone 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83681 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83682 D1 HEK293 cells HUMAN 3H-SCH23390 pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83683 D2 HEK293 cells HUMAN 3H-SPIPERONE pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83684 D3 HEK293 cells HUMAN 3H-SPIPERONE pyrovalerone 9200 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83685 H1 HEK293 cells HUMAN 3H-PYRILAMINE pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83686 D1 HEK293 cells RAT 3H-RO5166017 pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83687 D1 HEK293 cells MOUSE 3H-RO5166017 pyrovalerone >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83688 NET HEK293 cells HUMAN 3H-Nisoxetine MDPV 80 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83689 DAT HEK293 cells HUMAN 3H-WIN 35,428 MDPV 10 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83690 SERT HEK293 cells HUMAN 3H-CITALOPRAM MDPV 2860 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83691 5-HT1A HEK293 cells HUMAN 3H-8-OH-DPAT MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83692 5-HT2A HEK293 cells HUMAN 3H- Ketanserin MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83693 5-HT2C HEK293 cells HUMAN 3H-MESULERGINE MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 15, 2025
83694 Alpha1A HEK293 cells HUMAN 3H-PRAZOSIN MDPV 6000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83695 Alpha2A HEK293 cells HUMAN 3H-RAUWOLSCINE MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83696 D1 HEK293 cells HUMAN 3H-SCH23390 MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83697 D2 HEK293 cells HUMAN 3H-SPIPERONE MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83698 D3 HEK293 cells HUMAN 3H-SPIPERONE MDPV 9200 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83699 H1 HEK293 cells HUMAN 3H-PYRILAMINE MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 28, 2025
83700 D1 HEK293 cells RAT 3H-RO5166017 MDPV 7200 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83701 D1 HEK293 cells MOUSE 3H-RO5166017 MDPV >10000 Simmler LD et al 2013 Jan 15, 2025 Jan 27, 2025
83702 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid 4560 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83703 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) ±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid 6549 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83704 KOR CLONED HUMAN 3H-U69593 ±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid 6549 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83705 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 4802 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83706 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5189 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83707 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 1334 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83708 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5973 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83709 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3320 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83710 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5195 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83711 Sigma 2 CLONED HUMAN 3H-DTG (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 9813 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83712 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2961 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83713 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 4655 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83714 5-HT2B CLONED HUMAN 3H-LSD (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 453 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83715 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3596 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83716 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 8396 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83717 SERT CLONED HUMAN 3H-CITALOPRAM (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2284 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83718 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-N-(3,4-difluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2961 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83719 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83720 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83721 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83722 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 9987 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83723 NET CLONED HUMAN 3H-Nisoxetine (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5904 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83724 SERT CLONED HUMAN 3H-Nisoxetine (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3137 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83725 KOR CLONED HUMAN 3H-U69593 methyl (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 668 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83726 5-HT2B CLONED HUMAN 3H-LSD methyl (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 6021 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83727 NET CLONED HUMAN 3H-Nisoxetine methyl (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 9209 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83728 SERT CLONED HUMAN 3H-CITALOPRAM methyl (±)-(4aS,8R,8aS)-2-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate 372 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83729 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 5.3 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83730 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3552 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83731 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 2950 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83732 A1 CLONED HUMAN 3H-DPCPX (±)-(4aS,8R,8aS)-2-cyclohexyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 6394 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83733 SERT CLONED HUMAN 3H-CITALOPRAM ±)-(4aS,8R,8aS)-2-butyl-8-(morpholine-4-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 6260 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83734 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 4803 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83735 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 2396 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83736 5-HT1B CLONED HUMAN 3H-5-CT (±)-(4aS,8R,8aS)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 8143 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83737 DAT CLONED HUMAN 3H-WIN 35,428 (±)-(4aS,8R,8aS)-2-benzyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 3854 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83738 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 3194 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83739 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (±)-(4aS,8R,8aS)-2-cyclopropyl-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 8590 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83740 DOR CLONED HUMAN 3H-DADLE (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 4693 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83741 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 8897 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83742 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 5536 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83743 5-HT1D CLONED HUMAN 3H-5-CT (±)-(4aS,8R,8aS)-2-(3,4-dimethoxybenzyl)-8-(4-phenylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one 3230 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83744 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 561 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83745 MOR CLONED HUMAN 3H-DAMGO (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 4599 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
83746 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 8411 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83747 5-HT2C CLONED HUMAN 3H-MESULERGINE (±)-(4aS,8R,8aS)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 2246 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
83748 KOR CLONED HUMAN 3H-U69593 (±)-(4aS,8R,8aS)-2-butyl-1-oxo-N-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide 3271 PDSP Certified Data Jan 15, 2025 Jan 28, 2025