The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 83,001-84,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
857495-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)picolinamide59.5Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857505-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)picolinamide80.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857515-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)picolinamide101Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857525-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl)picolinamide39.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857535-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl)picolinamide371Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857545-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl)picolinamide68Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857555-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) picolinamide181Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857565-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) picolinamide90.4Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857575-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) picolinamide9.57Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857585-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857595-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide327Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857605-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl)picolinamide230Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857615-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857625-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide161Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857635-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl)picolinamide11.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857645-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide140Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857655-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857665-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl)picolinamide495Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857675-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide500Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857685-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide16.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857695-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857705-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857715-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide45.3Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857725-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(piperonyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857735-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857745-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide1.68Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857755-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(furoyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857765-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857775-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide725Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857785-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) picolinamide443Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857795-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide52.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857805-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide77.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857815-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) picolinamide117Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857825-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857835-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl)picolinamide213Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857845-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl)picolinamide44.1Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857855-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-OH-DPAT0.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857865-HT2AFR. CORTEXRAT3H-KETANSERINKETANSERIN0.85Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857875-HT2CFR. CORTEXRAT3H-MESULERGINEMESULERGINE1.9Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85788CEREBRAL CORTEXRAT3H-PRAZOSINN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide76Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85789CEREBRAL CORTEXRAT3H-RX821002N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85790D1CLONEDHUMAN3H-SCH23390N-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
85791D2CLONEDHUMAN3H-N-MethylspiperoneN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide2300Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
85792D2CLONEDHUMAN3H-N-MethylspiperoneN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide250Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
85793D1CLONEDHUMAN3H-SCH23390N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide610Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
85794CEREBRAL CORTEXRAT3H-RX821002N-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide4200Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85795CEREBRAL CORTEXRAT3H-PRAZOSINN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide31Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85796CEREBRAL CORTEXRAT3H-PRAZOSINN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85797CEREBRAL CORTEXRAT3H-RX821002N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
85798D1CLONEDHUMAN3H-SCH23390N-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
85799D2CLONEDHUMAN3H-N-MethylspiperoneN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide>10000Fiorino F et al 2017Jan 15, 2025Jan 28, 2025
858005-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-1542Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858015-HT2AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-1630Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858025-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-14800Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858035-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-22145Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858045-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-22943Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858055-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-29871Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858065-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-3158Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858075-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-31317Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858085-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-34181Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858095-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-4204Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858105-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-4567Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858115-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-41082Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858125-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-51246Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858135-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-553Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858145-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-51209Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858155-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-7479Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858165-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-7987Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858175-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-72573Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858185-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-81241Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858195-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-819Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858205-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-8233Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858215-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-102326Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858225-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-1079Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858235-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-102114Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858245-HT1ACLONEDHUMAN3H-8-OH-DPAT2C-BI-11931Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858255-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-1142Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858265-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-111702Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858275-HT1AHEK293 cellsHUMAN3H-8-OH-DPAT2C-BI-122313Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858285-HT2AHEK293 cellsHUMAN3H- Ketanserin2C-BI-1221Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858295-HT2CHEK293 cellsHUMAN3H-MESULERGINE2C-BI-12279Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858305-HT1AHEK293 cellsHUMAN3H-8-OH-DPATBiscaline4021Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858315-HT2AHEK293 cellsHUMAN3H- KetanserinBiscaline>10000Luethi D et al 2019Jan 15, 2025Jan 15, 2025
858325-HT2CHEK293 cellsHUMAN3H-MESULERGINEBiscaline>10000Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85833TAAR1HEK293 cellsRAT3H-RO51660172C-BI-16.1Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85834TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-1221Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85835Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-11040Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85836Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-1401Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85837D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-1>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85838NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-12882Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85839DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-18450Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85840SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-17580Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85841TAAR1HEK293 cellsRAT3H-RO51660172C-BI-2264Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85842TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-24520Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85843Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-28770Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85844Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-21164Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85845D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-2>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85846NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-28800Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85847DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-28450Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85848SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-27580Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85849TAAR1HEK293 cellsRAT3H-RO51660172C-BI-315Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85850TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-3604Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85851Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-36945Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85852Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-3157Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85853D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-3>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85854NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-3352Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85855DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-33933Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85856SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-33835Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85857TAAR1HEK293 cellsRAT3H-RO51660172C-BI-46.8Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85858TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-4512Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85859Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-48212Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85860Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-4320Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85861D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-4>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85862NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-41106Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85863DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-46332Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85864SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-43407Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85865TAAR1HEK293 cellsRAT3H-RO51660172C-BI-510Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85866TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-5235Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85867Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-52545Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85868Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-51326Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85869D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-5>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85870NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-57705Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85871DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-57689Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85872SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-56011Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85873TAAR1HEK293 cellsRAT3H-RO51660172C-BI-74.6Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85874TAAR1HEK293 cellsRAT3H-RO51660172C-BI-7251Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85875Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-72018Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85876Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-7519Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85877D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-7>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85878NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-78800Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85879DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-76286Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85880SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-72593Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85881TAAR1HEK293 cellsRAT3H-RO51660172C-BI-838Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85882TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-8446Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85883Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-86938Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85884Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-8634Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85885D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-8>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85886NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-86335Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85887DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-88450Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85888SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-87580Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85889TAAR1HEK293 cellsRAT3H-RO51660172C-BI-1013Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85890TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-1093Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85891Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-106226Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85892Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-102088Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85893D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-10>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85894NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-108800Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85895DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-108450Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85896SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-107580Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85897TAAR1HEK293 cellsRAT3H-RO51660172C-BI-111.4Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85898TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-1113Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85899Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-114174Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85900Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-113860Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85901D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-11>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85902NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-114337Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85903DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-118450Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85904SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-117580Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85905TAAR1HEK293 cellsRAT3H-RO51660172C-BI-12192Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85906TAAR1HEK293 cellsMOUSE3H-RO51660172C-BI-124172Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85907Alpha1ACHO cellsHUMAN3H-PRAZOSIN2C-BI-128018Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85908Alpha2ACHLHUMAN3H-RAUWOLSCINE2C-BI-12657Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85909D2HEK293 cellsHUMAN3H-SPIPERONE2C-BI-12>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85910NETHEK293 cellsHUMAN3H-Nisoxetine2C-BI-128800Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85911DATHEK293 cellsHUMAN3H-WIN 35,4282C-BI-128450Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85912SERTHEK293 cellsHUMAN3H-CITALOPRAM2C-BI-127580Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85913TAAR1HEK293 cellsRAT3H-RO5166017Biscaline586Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85914TAAR1HEK293 cellsMOUSE3H-RO5166017Biscaline4270Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85915Alpha1ACHO cellsHUMAN3H-PRAZOSINBiscaline8770Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85916Alpha2ACHLHUMAN3H-RAUWOLSCINEBiscaline797Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85917D2HEK293 cellsHUMAN3H-SPIPERONEBiscaline8520Luethi D et al 2019Jan 15, 2025Jan 28, 2025
85918NETHEK293 cellsHUMAN3H-NisoxetineBiscaline7510Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85919DATHEK293 cellsHUMAN3H-WIN 35,428Biscaline9720Luethi D et al 2019Jan 15, 2025Jan 15, 2025
85920SERTHEK293 cellsHUMAN3H-CITALOPRAMBiscaline>10000Luethi D et al 2019Jan 15, 2025Jan 28, 2025
859215-HT1ACLONEDHUMAN3H-WAY100635delta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859225-HT1BCLONEDHUMAN3H-5-CTdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859235-HT1DCLONEDHUMAN3H-5-CTdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859245-HT2ACLONEDHUMAN3H-KETANSERINdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859255-HT2BCLONEDHUMAN3H-LSDdelta9 -tetrahydrocannabinol (THC)765Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859265-HT2CCLONEDHUMAN3H-MESULERGINEdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859275-HT3CLONEDHUMAN3H-GR65630delta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859285-HT5ACLONEDHUMAN3H-LSDdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859295-HT6CLONEDHUMAN3H-LSDdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859305-HT7CLONEDHUMAN3H-LSDdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85931SERTCLONEDHUMAN3H-CITALOPRAMdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85932D1CLONEDHUMAN3H-SCH23390delta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85933D5CLONEDHUMAN3H-SCH23390delta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85934D2CLONEDHUMAN3H-N-Methylspiperonedelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85935D3CLONEDHUMAN3H-N-Methylspiperonedelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85936D4CLONEDHUMAN3H-N-Methylspiperonedelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85937DATCLONEDHUMAN3H-WIN35428delta9 -tetrahydrocannabinol (THC)1575Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85938M1CLONEDHUMAN3H-QNBdelta9 -tetrahydrocannabinol (THC)1673Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85939M2CLONEDHUMAN3H-QNBdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85940M3CLONEDHUMAN3H-QNBdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85941M4CLONEDHUMAN3H-QNBdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85942M5CLONEDHUMAN3H-QNBdelta9 -tetrahydrocannabinol (THC)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859435-HT1ACLONEDHUMAN3H-WAY1006351-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859445-HT1BCLONEDHUMAN3H-5-CT1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859455-HT1DCLONEDHUMAN3H-5-CT1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859465-HT2ACLONEDHUMAN3H-KETANSERIN1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859475-HT2BCLONEDHUMAN3H-LSD1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)192Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859485-HT2CCLONEDHUMAN3H-MESULERGINE1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859495-HT5ACLONEDHUMAN3H-LSD1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859505-HT6CLONEDHUMAN3H-LSD1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)693Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
859515-HT7CLONEDHUMAN3H-LSD1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85952D1CLONEDHUMAN3H-SCH233901-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85953D5CLONEDHUMAN3H-SCH233901-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85954D2CLONEDHUMAN3H-N-Methylspiperone1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85955D3CLONEDHUMAN3H-N-Methylspiperone1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85956D4CLONEDHUMAN3H-N-Methylspiperone1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85957DATCLONEDHUMAN3H-WIN 35,4281-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85958SERTCLONEDHUMAN3H-CITALOPRAM1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85959NETCLONEDHUMAN3H-Nisoxetine1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85960M1CLONEDHUMAN3H-QNB1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85961M2CLONEDHUMAN3H-QNB1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85962M3CLONEDHUMAN3H-QNB1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85963M4CLONEDHUMAN3H-QNB1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85964M5CLONEDHUMAN3H-QNB1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85965GABAACORTICAL MEMBRANESRAT3H-MUSCIMOL1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85966PBRKidney membranesRAT3H-PK111951-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)3291Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85967Alpha1ACLONEDHUMAN3H-PRAZOSIN1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85968Alpha1BCLONEDHUMAN3H-PRAZOSIN1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85969Alpha1DCLONEDHUMAN3H-PRAZOSIN1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85970Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85971Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85972Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85973Beta 1CLONEDHUMAN125I-Pindolol1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85974Beta3CLONEDHUMAN125I-Pindolol1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85975Beta 2CLONEDHUMAN3H-CGP-121771-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85976H1CLONEDHUMAN3H-PYRILAMINE1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
859775-HT1DCLONEDHUMAN125I-aminopotentidine1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85978H3CLONEDHUMAN3H-Alpha-methylhistamine1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85979H4CLONEDHUMAN3H-Histamine1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85980KORCLONEDHUMAN3H-U695931-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85981MORCLONEDHUMAN3H-DAMGO1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85982DORCLONEDHUMAN3H-DADLE1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85983Sigma 1CLONEDHUMAN3H-Pentazocine(+)1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85984Sigma 2CLONEDHUMAN3H-DTG1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85985BZPCORTICAL MEMBRANESRATFNZ1-(5-fluoropentyl)-3-(1-naphthoyl)indole) (AM-2201)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
85986BZPCORTICAL MEMBRANESRATFNZDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
85987Alpha1ACLONEDHUMAN3H-PRAZOSINDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85988Alpha1BCLONEDHUMAN3H-PRAZOSINDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85989Alpha1DCLONEDHUMAN3H-PRAZOSINDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85990Alpha2ACLONEDHUMAN3H-RAUWOLSCINEDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85991Alpha2BCLONEDHUMAN3H-RAUWOLSCINEDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85992Alpha2CCLONEDHUMAN3H-RAUWOLSCINEDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85993Beta 1CLONEDHUMAN125I-PindololDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85994Beta3CLONEDHUMAN125I-PindololDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85995Beta 2CLONEDHUMAN3H-CGP-12177Delta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85996NETCLONEDHUMAN3H-NisoxetineDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
85997H1CLONEDHUMAN3H-PYRILAMINEDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
859985-HT1DCLONEDHUMAN125I-aminopotentidineDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
85999H3CLONEDHUMAN3H-Alpha-methylhistamineDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86000H4CLONEDHUMAN3H-HistamineDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86001KORCLONEDHUMAN3H-U69593Delta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86002MORCLONEDHUMAN3H-DAMGODelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86003DORCLONEDHUMAN3H-DADLEDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86004Sigma 1CLONEDHUMAN3H-Pentazocine(+)Delta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86005Sigma 2CLONEDHUMAN3H-DTGDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86006KORCORTICAL MEMBRANESRAT3H-MUSCIMOLDelta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
86007PBRKidney membranesRAT3H-PK11195Delta9 -tetrahydrocannabinol (THC))>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860085-HT1ACLONEDHUMAN3H-WAY100635(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860095-HT1BCLONEDHUMAN3H-5-CT(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860105-HT1DCLONEDHUMAN3H-5-CT(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860115-HT1ECLONEDHUMAN3H-5-HT(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860125-HT2ACLONEDHUMAN3H-KETANSERIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860135-HT2BCLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)316Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860145-HT2CCLONEDHUMAN3H-MESULERGINE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860155-HT3CLONEDHUMAN3H-GR-65630(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860165-HT5ACLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860175-HT6CLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860185-HT7CLONEDHUMAN3H-LSD(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86019SERTCLONEDHUMAN3H-CITALOPRAM(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86020DATCLONEDHUMAN3H-WIN 35,428(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86021D1CLONEDHUMAN3H-SCH23390(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86022D5CLONEDHUMAN3H-SCH23390(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86023D2CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86024D3CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86025D4CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86026M1CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86027M2CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86028M3CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86029M4CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86030M5CLONEDHUMAN3H-QNB(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86031PBRKidney membranesRAT3H-PK11195(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)673Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86032Alpha1ACLONEDHUMAN3H-PRAZOSIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86033Alpha1BCLONEDHUMAN3H-PRAZOSIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86034Alpha1DCLONEDHUMAN3H-PRAZOSIN(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86035Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86036Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86037Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86038Beta 1CLONEDHUMAN125I-Pindolol(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86039Beta3CLONEDHUMAN125I-Pindolol(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86040Beta 2CLONEDHUMAN3H-CGP-12177(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86041NETCLONEDHUMAN3H-Nisoxetine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86042H1CLONEDHUMAN3H-PYRILAMINE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
860435-HT1DCLONEDHUMAN125I-aminopotentidine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86044H3CLONEDHUMAN3H-Alpha-methylhistamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86045H4CLONEDHUMAN3H-Histamine(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86046KORCLONEDHUMAN3H-U69593(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86047MORCLONEDHUMAN3H-DAMGO(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86048DORCLONEDHUMAN3H-DADLE(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86049Sigma 1CLONEDHUMAN3H-Pentazocine(+)(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86050Sigma 2CLONEDHUMAN3H-DTG(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86051KORCORTICAL MEMBRANESRAT3H-MUSCIMOL(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
86052BZPCORTICAL MEMBRANESRATFNZ(1-pentyl-3-(1-naphthoyl)indole) (JWH-018)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
860535-HT1ACLONEDHUMAN3H-WAY100635Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860545-HT1BCLONEDHUMAN3H-5CTNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860555-HT1DCLONEDHUMAN3H-5CTNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860565-HT1ECLONEDHUMAN3H-5HTNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860575-HT2ACLONEDHUMAN3H-KETANSERINNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860585-HT2BCLONEDHUMAN3H-LSDNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)184Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860595-HT2CCLONEDHUMAN3H-MESULERGINENaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860605-HT3CLONEDHUMAN3H-GR-65630Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860615-HT5ACLONEDHUMAN3H-LSDNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860625-HT6CLONEDHUMAN3H-LSDNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
860635-HT7CLONEDHUMAN3H-LSDNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86064SERTCLONEDHUMAN3H-CITALOPRAMNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86065D1CLONEDHUMAN3H-SCH23390Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86066D5CLONEDHUMAN3H-SCH23390Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86067D2CLONEDHUMAN3H-N-MethylspiperoneNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86068D3CLONEDHUMAN3H-N-MethylspiperoneNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86069D4CLONEDHUMAN3H-N-MethylspiperoneNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86070DATCLONEDHUMAN3H-WIN 35,428Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86071M1CLONEDHUMAN3H-QNBNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86072M2CLONEDHUMAN3H-QNBNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86073M3CLONEDHUMAN3H-QNBNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86074M4CLONEDHUMAN3H-QNBNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86075M5CLONEDHUMAN3H-QNBNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86076PBRKidney membranesRAT3H-PK11195Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86077Alpha1ACLONEDHUMAN3H-PRAZOSINNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86078Alpha1BCLONEDHUMAN3H-PRAZOSINNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86079Alpha1DCLONEDHUMAN3H-PRAZOSINNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86080Alpha2ACLONEDHUMAN3H-RAUWOLSCINENaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86081Alpha2BCLONEDHUMAN3H-RAUWOLSCINENaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86082Alpha2CCLONEDHUMAN3H-RAUWOLSCINENaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86083Beta 1CLONEDHUMAN125I-PindololNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86084Beta3CLONEDHUMAN125I-PindololNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86085Beta 2CLONEDHUMAN3H-CGP12177Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86086NETCLONEDHUMAN3H-NisoxetineNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86087H1CLONEDHUMAN3H-PYRILAMINENaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
860885-HT1DCLONEDHUMAN125I-aminopotentidineNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86089H3CLONEDHUMAN3H-Alpha-methylhistamineNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86090H4CLONEDHUMAN3H-HistamineNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86091KORCLONEDHUMAN3H-U69593Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86092MORCLONEDHUMAN3H-DAMGONaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86093DORCLONEDHUMAN3H-DADLENaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86094Sigma 1CLONEDHUMAN3H-Pentazocine(+)Naphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86095Sigma 2CLONEDHUMAN3H-DTGNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86096KORCORTICAL MEMBRANESRAT3H-MUSCIMOLNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
86097BZPCORTICAL MEMBRANESRATFNZNaphthalen-1-yl-(1-butylindol-3-yl)methanone (JWH-073)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
86098BZPCORTICAL MEMBRANESRATFNZ4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
86099KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
861005-HT1ACLONEDHUMAN3H-WAY1006354-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861015-HT1BCLONEDHUMAN3H-5-CT4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861025-HT1DCLONEDHUMAN3H-5-CT4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861035-HT1ECLONEDHUMAN3H-5-HT4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861045-HT2ACLONEDHUMAN3H-KETANSERIN4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861055-HT2BCLONEDHUMAN3H-LSD4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861065-HT2CCLONEDHUMAN3H-MESULERGINE4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861075-HT3CLONEDHUMAN3H-GR-656304-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861085-HT5ACLONEDHUMAN3H-LSD4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861095-HT6CLONEDHUMAN3H-LSD4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861105-HT7CLONEDHUMAN3H-LSD4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86111SERTCLONEDHUMAN3H-CITALOPRAM4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86112D1CLONEDHUMAN3H-SCH233904-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86113D5CLONEDHUMAN3H-SCH233904-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86114D2CLONEDHUMAN3H-N-Methylspiperone4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86115D3CLONEDHUMAN3H-N-Methylspiperone4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86116D4CLONEDHUMAN3H-N-Methylspiperone4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86117DATCLONEDHUMAN3H-WIN354284-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86118M1CLONEDHUMAN3H-QNB4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86119M2CLONEDHUMAN3H-QNB4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86120M3CLONEDHUMAN3H-QNB4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86121M4CLONEDHUMAN3H-QNB4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86122M5CLONEDHUMAN3H-QNB4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86123PBRKidney membranesRAT3H-PK111954-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86124Alpha1ACLONEDHUMAN3H-PRAZOSIN4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86125Alpha1BCLONEDHUMAN3H-PRAZOSIN4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86126Alpha1DCLONEDHUMAN3H-PRAZOSIN4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86127Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86128Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86129Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86130Beta 1CLONEDHUMAN125I-Pindolol4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86131Beta3CLONEDHUMAN125I-Pindolol4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86132Beta 2CLONEDHUMAN3H-CGP-121774-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86133NETCLONEDHUMAN3H-Nisoxetine4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86134H1CLONEDHUMAN3H-PYRILAMINE4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
861355-HT1DCLONEDHUMAN125I-aminopotentidine4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86136H3CLONEDHUMAN3H-Alpha-methylhistamine4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86137H4CLONEDHUMAN3H-Histamine4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86138KORCLONEDHUMAN3H-U695934-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86139MORCLONEDHUMAN3H-DAMGO4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86140DORCLONEDHUMAN3H-DADLE4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86141Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86142Sigma 2CLONEDHUMAN3H-DTG4-Methoxynaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-081)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
861435-HT1ACLONEDHUMAN3H-WAY1006352-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861445-HT1BCLONEDHUMAN3H-5CT2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861455-HT1DCLONEDHUMAN3H-5CT2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861465-HT1ECLONEDHUMAN3H-5HT2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861475-HT2ACLONEDHUMAN3H-KETANSERIN2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861485-HT2BCLONEDHUMAN3H-LSD2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)1249Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861495-HT2CCLONEDHUMAN3H-MESULERGINE2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)4815Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861505-HT3CLONEDHUMAN3H-GR-656302-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861515-HT5ACLONEDHUMAN3H-LSD2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861525-HT6CLONEDHUMAN3H-LSD2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861535-HT7CLONEDHUMAN3H-LSD2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86154SERTCLONEDHUMAN3H-CITALOPRAM2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86155D1CLONEDHUMAN3H-SCH233902-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86156D5CLONEDHUMAN3H-SCH233902-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86157D2CLONEDHUMAN3H-N-Methylspiperone2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86158D3CLONEDHUMAN3H-N-Methylspiperone2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86159D4CLONEDHUMAN3H-N-Methylspiperone2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86160DATCLONEDHUMAN3H-WIN 35,4282-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86161M1CLONEDHUMAN3H-QNB2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86162M2CLONEDHUMAN3H-QNB2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86163M3CLONEDHUMAN3H-QNB2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86164M4CLONEDHUMAN3H-QNB2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86165M5CLONEDHUMAN3H-QNB2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86166PBRKidney membranesRAT3H-PK111952-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86167BZPCEREBRAL CORTEXRATFNZ2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
86168Alpha1ACLONEDHUMAN3H-PRAZOSIN2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86169Alpha1BCLONEDHUMAN3H-PRAZOSIN2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86170Alpha1DCLONEDHUMAN3H-PRAZOSIN2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86171Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86172Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86173Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86174Beta 1CLONEDHUMAN125I-Pindolol2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86175Beta3CLONEDHUMAN125I-Pindolol2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86176Beta 2CLONEDHUMAN3H-CGP121772-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86177NETCLONEDHUMAN3H-Nisoxetine2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86178H1CLONEDHUMAN3H-PYRILAMINE2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
861795-HT1DCLONEDHUMAN125I-aminopotentidine2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86180H3CLONEDHUMAN3H-Alpha-methylhistamine2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86181H4CLONEDHUMAN3H-Histamine2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86182KORCLONEDHUMAN3H-U695932-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86183MORCLONEDHUMAN3H-DAMGO2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86184DORCLONEDHUMAN3H-DADLE2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86185Sigma 1CLONEDHUMAN3H-Pentazocine(+)2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86186Sigma 2CLONEDHUMAN3H-DTG2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86187GABAACORTICAL MEMBRANESRAT3H-MUSCIMOL2-Phenyl-1-(1-pentylindol-3-yl)ethanone (JWH-167)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
861885-HT1ACLONEDHUMAN3H-WAY1006354-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861895-HT1BCLONEDHUMAN3H-5-CT4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861905-HT1DCLONEDHUMAN3H-5-CT4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861915-HT1ECLONEDHUMAN3H-5-HT4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861925-HT2ACLONEDHUMAN3H-KETANSERIN4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861935-HT2BCLONEDHUMAN3H-LSD4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861945-HT2CCLONEDHUMAN3H-MESULERGINE4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861955-HT3CLONEDHUMAN3H-GR-656304-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861965-HT5ACLONEDHUMAN3H-LSD4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861975-HT6CLONEDHUMAN3H-LSD4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
861985-HT7CLONEDHUMAN3H-LSD4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86199SERTCLONEDHUMAN3H-CITALOPRAM4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86200D1CLONEDHUMAN3H-SCH233904-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86201D5CLONEDHUMAN3H-SCH233904-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86202D2CLONEDHUMAN3H-N-Methylspiperone4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86203D3CLONEDHUMAN3H-N-Methylspiperone4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86204D4CLONEDHUMAN3H-N-Methylspiperone4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86205DATCLONEDHUMAN3H-WIN 35,4284-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86206M1CLONEDHUMAN3H-QNB4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86207M2CLONEDHUMAN3H-QNB4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86208M3CLONEDHUMAN3H-QNB4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86209M4CLONEDHUMAN3H-QNB4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86210M5CLONEDHUMAN3H-QNB4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86211PBRKidney membranesRAT3H-PK111954-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86212Alpha1ACLONEDHUMAN3H-PRAZOSIN4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86213Alpha1BCLONEDHUMAN3H-PRAZOSIN4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86214Alpha1DCLONEDHUMAN3H-PRAZOSIN4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86215Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86216Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86217Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86218Beta 1CLONEDHUMAN125I-Pindolol4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86219Beta3CLONEDHUMAN125I-Pindolol4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86220Beta 2CLONEDHUMAN3H-CGP-121774-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86221NETCLONEDHUMAN3H-Nisoxetine4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86222H1CLONEDHUMAN3H-PYRILAMINE4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
862235-HT1DCLONEDHUMAN125I-aminopotentidine4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86224H3CLONEDHUMAN3H-Alpha-methylhistamine4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86225H4CLONEDHUMAN3H-Histamine4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86226KORCLONEDHUMAN3H-U695934-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86227MORCLONEDHUMAN3H-DAMGO4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86228DORCLONEDHUMAN3H-DADLE4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86229Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86230Sigma 2CLONEDHUMAN3H-DTG4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86231KORCORTICAL MEMBRANESRAT3H-MUSCIMOL4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
86232BZPCORTICAL MEMBRANESRATFNZ4-Ethylnaphthalen-1-yl-(1-pentylindol-3-yl)methanone (JWH-210)>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
862335-HT1ACLONEDHUMAN3H-WAY100635JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862345-HT1BCLONEDHUMAN3H-5-CTJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862355-HT1DCLONEDHUMAN3H-5-CTJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862365-HT1ECLONEDHUMAN3H-5-HTJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862375-HT2ACLONEDHUMAN3H-KETANSERINJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862385-HT2BCLONEDHUMAN3H-LSDJWH-391368Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862395-HT2CCLONEDHUMAN3H-MESULERGINEJWH-3911899Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862405-HT3CLONEDHUMAN3H-GR-65630JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862415-HT5ACLONEDHUMAN3H-LSDJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862425-HT6CLONEDHUMAN3H-LSDJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
862435-HT7CLONEDHUMAN3H-LSDJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86244SERTCLONEDHUMAN3H-CITALOPRAMJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86245D1CLONEDHUMAN3H-SCH23390JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86246D5CLONEDHUMAN3H-SCH23390JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86247D2CLONEDHUMAN3H-N-MethylspiperoneJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86248D3CLONEDHUMAN3H-N-MethylspiperoneJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86249D4CLONEDHUMAN3H-N-MethylspiperoneJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86250D5CLONEDHUMAN3H-N-MethylspiperoneJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86251DATCLONEDHUMAN3H-WIN 35,428JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86252M1CLONEDHUMAN3H-QNBJWH-391461Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86253M2CLONEDHUMAN3H-QNBJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86254M3CLONEDHUMAN3H-QNBJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86255M4CLONEDHUMAN3H-QNBJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86256M5CLONEDHUMAN3H-QNBJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86257PBRKidney membranesRAT3H-PK11195JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86258Alpha1ACLONEDHUMAN3H-PRAZOSINJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86259Alpha1BCLONEDHUMAN3H-PRAZOSINJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86260Alpha1DCLONEDHUMAN3H-PRAZOSINJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86261Alpha2ACLONEDHUMAN3H-RAUWOLSCINEJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86262Alpha2BCLONEDHUMAN3H-RAUWOLSCINEJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86263Alpha2CCLONEDHUMAN3H-RAUWOLSCINEJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86264Beta 1CLONEDHUMAN125I-PindololJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86265Beta3CLONEDHUMAN125I-PindololJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86266Beta 2CLONEDHUMAN3H-CGP12177JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86267NETCLONEDHUMAN3H-NisoxetineJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 15, 2025
86268H1CLONEDHUMAN3H-PYRILAMINEJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
862695-HT1DCLONEDHUMAN125I-aminopotentidineJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86270H3CLONEDHUMAN3H-Alpha-methylhistamineJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86271H4CLONEDHUMAN3H-HistamineJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86272KORCLONEDHUMAN3H-U69593JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86273MORCLONEDHUMAN3H-DAMGOJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86274DORCLONEDHUMAN3H-DADLEJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86275Sigma 1CLONEDHUMAN3H-Pentazocine(+)JWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86276Sigma 2CLONEDHUMAN3H-DTGJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 28, 2025
86277KORCORTICAL MEMBRANESRAT3H-MUSCIMOLJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 27, 2025
86278BZPCORTICAL MEMBRANESRATFNZJWH-391>10000Wiley JL et al 2016Jan 15, 2025Jan 29, 2025
86279mGluR5HEK293 cellsRAT3H-methoxyPEPyMPEP35Hammond AS et al 2010Jan 15, 2025Jan 28, 2025
86280mGluR5HEK293 cellsRAT3H-methoxyPEPy5-MPEP388Hammond AS et al 2010Jan 15, 2025Jan 28, 2025
86281A1CLONEDHUMAN3H-CCPA8-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione41.7Koch P et al 2018Jan 15, 2025Jan 15, 2025
86282A2ASTRIATUMRAT3H-MSX-28-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione497Koch P et al 2018Jan 15, 2025Jan 15, 2025
86283A2BCLONEDHUMAN3H-PSB-6038-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86284A3CLONEDHUMAN3H-PSB-118-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86285A1BRAIN CORTEXRAT3H-CCPA8-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione123Koch P et al 2018Jan 15, 2025Jan 15, 2025
86286A2ACLONEDHUMAN3H-MSX-28-(2-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione408Koch P et al 2018Jan 15, 2025Jan 15, 2025
86287A1CLONEDHUMAN3H-CCPA8-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione70.7Koch P et al 2018Jan 15, 2025Jan 15, 2025
86288A2BCLONEDHUMAN3H-PSB-6038-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86289A3CLONEDHUMAN3H-PSB-118-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86290A1CORTEXRAT3H-CCPA8-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione28.8Koch P et al 2018Jan 15, 2025Jan 15, 2025
86291A2ASTRIATUMRAT3H-MSX-28-(3-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1140Koch P et al 2018Jan 15, 2025Jan 15, 2025
86292A1CLONEDHUMAN3H-CCPA8-(4-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1350Koch P et al 2018Jan 15, 2025Jan 15, 2025
86293A2BCLONEDHUMAN3H-PSB-6038-(4-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86294A3CLONEDHUMAN3H-PSB-118-(4-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione9390Koch P et al 2018Jan 15, 2025Jan 15, 2025
86295A1CORTEXRAT3H-CCPA8-(4-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione156Koch P et al 2018Jan 15, 2025Jan 15, 2025
86296A2ASTRIATUMRAT3H-MSX-28-(4-Bromobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86297A1CLONEDHUMAN3H-CCPA3-Ethyl-1-methyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione244Koch P et al 2018Jan 15, 2025Jan 15, 2025
86298A2BCLONEDHUMAN3H-PSB-6033-Ethyl-1-methyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86299A3CLONEDHUMAN3H-PSB-113-Ethyl-1-methyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione8760Koch P et al 2018Jan 15, 2025Jan 15, 2025
86300A1CORTEXRAT3H-CCPA3-Ethyl-1-methyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione114Koch P et al 2018Jan 15, 2025Jan 15, 2025
86301A2ASTRIATUMRAT3H-MSX-23-Ethyl-1-methyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86302A1CLONEDHUMAN3H-CCPA3-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione156Koch P et al 2018Jan 15, 2025Jan 15, 2025
86303A2ACLONEDHUMAN3H-MSX-23-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1780Koch P et al 2018Jan 15, 2025Jan 15, 2025
86304A2BCLONEDHUMAN3H-PSB-6033-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione100Koch P et al 2018Jan 15, 2025Jan 15, 2025
86305A3CLONEDHUMAN3H-PSB-113-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86306A1CORTEXRAT3H-CCPA3-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione49.1Koch P et al 2018Jan 15, 2025Jan 15, 2025
86307A2ASTRIATUMRAT3H-MSX-23-Ethyl-1-methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione708Koch P et al 2018Jan 15, 2025Jan 15, 2025
86308A1CORTEXRAT3H-CCPA3-Ethyl-1-methyl-8-(4-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86309A2ASTRIATUMRAT3H-MSX-23-Ethyl-1-methyl-8-(4-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86310A2BCLONEDHUMAN3H-PSB-6033-Ethyl-1-methyl-8-(4-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione100Koch P et al 2018Jan 15, 2025Jan 15, 2025
86311A3CLONEDHUMAN3H-PSB-113-Ethyl-1-methyl-8-(4-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86312A3CLONEDHUMAN3H-PSB-113-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86313A2BCLONEDHUMAN3H-PSB-6033-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione100Koch P et al 2018Jan 15, 2025Jan 15, 2025
86314A1CLONEDHUMAN3H-CCPA3-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione85.3Koch P et al 2018Jan 15, 2025Jan 15, 2025
86315A1CORTEXRAT3H-CCPA3-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione59.4Koch P et al 2018Jan 15, 2025Jan 15, 2025
86316A2ASTRIATUMRAT3H-MSX-23-Ethyl-8-(4-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86317A1CORTEXRAT3H-CCPA3-Ethyl-8-(4-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione164Koch P et al 2018Jan 15, 2025Jan 15, 2025
86318A1CLONEDHUMAN3H-CCPA3-Ethyl-8-(4-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione5120Koch P et al 2018Jan 15, 2025Jan 15, 2025
86319A2BCLONEDHUMAN3H-PSB-6033-Ethyl-8-(4-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86320A3CLONEDHUMAN3H-PSB-113-Ethyl-8-(4-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86321A2ASTRIATUMRAT3H-MSX-23-Ethyl-8-(3-fluorobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86322A2ASTRIATUMRAT3H-MSX-28-(3-Chlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86323A1CORTEXRAT3H-CCPA8-(3-Chlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione53Koch P et al 2018Jan 15, 2025Jan 15, 2025
86324A1CLONEDHUMAN3H-CCPA8-(3-Chlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione121Koch P et al 2018Jan 15, 2025Jan 15, 2025
86325A2ACLONEDHUMAN3H-MSX-28-(3-Chlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86326A2BCLONEDHUMAN3H-PSB-6038-(3-Chlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86327A1CLONEDHUMAN3H-CCPA8-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione391Koch P et al 2018Jan 15, 2025Jan 15, 2025
86328A2ACLONEDHUMAN3H-MSX-28-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione906Koch P et al 2018Jan 15, 2025Jan 15, 2025
86329A2BCLONEDHUMAN3H-PSB-6038-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86330A3CLONEDHUMAN3H-PSB-118-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86331A1CORTEXRAT3H-CCPA8-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione36.9Koch P et al 2018Jan 15, 2025Jan 15, 2025
86332A2ASTRIATUMRAT3H-MSX-28-(2,5-Dichlorobenzyl)-3-ethyl-1-dimethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione617Koch P et al 2018Jan 15, 2025Jan 15, 2025
86333A2ASTRIATUMRAT3H-MSX-28-(2,6-Dichlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1100Koch P et al 2018Jan 15, 2025Jan 15, 2025
86334A1CORTEXRAT3H-CCPA8-(2,6-Dichlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione142Koch P et al 2018Jan 15, 2025Jan 15, 2025
86335A1CLONEDHUMAN3H-CCPA8-(2,6-Dichlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione197Koch P et al 2018Jan 15, 2025Jan 15, 2025
86336A2BCLONEDHUMAN3H-PSB-6038-(2,6-Dichlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86337A3CLONEDHUMAN3H-PSB-118-(2,6-Dichlorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86338A3CLONEDHUMAN3H-PSB-113-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86339A2BCLONEDHUMAN3H-PSB-6033-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86340A2ACLONEDHUMAN3H-MSX-23-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione2020Koch P et al 2018Jan 15, 2025Jan 15, 2025
86341A1CLONEDHUMAN3H-CCPA3-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione495Koch P et al 2018Jan 15, 2025Jan 15, 2025
86342A1CORTEXRAT3H-CCPA3-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione236Koch P et al 2018Jan 15, 2025Jan 15, 2025
86343A2ASTRIATUMRAT3H-MSX-23-Ethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione667Koch P et al 2018Jan 15, 2025Jan 15, 2025
86344A2ASTRIATUMRAT3H-MSX-28-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione592Koch P et al 2018Jan 15, 2025Jan 15, 2025
86345A1CORTEXRAT3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione76.2Koch P et al 2018Jan 15, 2025Jan 15, 2025
86346A1CLONEDHUMAN3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione55.9Koch P et al 2018Jan 15, 2025Jan 15, 2025
86347A2ACLONEDHUMAN3H-MSX-28-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione881Koch P et al 2018Jan 15, 2025Jan 15, 2025
86348A2BCLONEDHUMAN3H-PSB-6038-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86349A3CLONEDHUMAN3H-PSB-118-(2-Chloro-5-(trifluoromethyl)benzyl)-3-ethyl-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86350A3CLONEDHUMAN3H-PSB-118-(3-Chloro-5-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86351A2BCLONEDHUMAN3H-PSB-6038-(3-Chloro-5-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86352A1CLONEDHUMAN3H-CCPA8-(3-Chloro-5-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione298Koch P et al 2018Jan 15, 2025Jan 15, 2025
86353A1CORTEXRAT3H-CCPA8-(3-Chloro-5-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione36.2Koch P et al 2018Jan 15, 2025Jan 15, 2025
86354A2ASTRIATUMRAT3H-MSX-28-(3-Chloro-5-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione981Koch P et al 2018Jan 15, 2025Jan 15, 2025
86355A2ASTRIATUMRAT3H-MSX-28-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione880Koch P et al 2018Jan 15, 2025Jan 15, 2025
86356A1CORTEXRAT3H-CCPA8-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione36Koch P et al 2018Jan 15, 2025Jan 15, 2025
86357A1CLONEDHUMAN3H-CCPA8-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione116Koch P et al 2018Jan 15, 2025Jan 15, 2025
86358A2ACLONEDHUMAN3H-MSX-28-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1700Koch P et al 2018Jan 15, 2025Jan 15, 2025
86359A2BCLONEDHUMAN3H-PSB-6038-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86360A3CLONEDHUMAN3H-PSB-118-(5-Bromo-2-fluorobenzyl)-3-ethyl-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86361A1CLONEDHUMAN3H-CCPA3-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione330Koch P et al 2018Jan 15, 2025Jan 15, 2025
86362A2ACLONEDHUMAN3H-MSX-23-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione503Koch P et al 2018Jan 15, 2025Jan 15, 2025
86363A2BCLONEDHUMAN3H-PSB-6033-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86364A3CLONEDHUMAN3H-PSB-113-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86365A2ASTRIATUMRAT3H-MSX-23-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione801Koch P et al 2018Jan 15, 2025Jan 15, 2025
86366A1CORTEXRAT3H-CCPA3-Ethyl-8-(3-fluoro-5-(trifluoromethyl)benzyl)-1- methyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione111Koch P et al 2018Jan 15, 2025Jan 15, 2025
86367A1CORTEXRAT3H-CCPA8-(3,5-Bis(trifluoromethyl)benzyl)-3-ethyl-1-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86368A2ASTRIATUMRAT3H-MSX-28-(3,5-Bis(trifluoromethyl)benzyl)-3-ethyl-1-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86369A2BCLONEDHUMAN3H-PSB-6038-(3,5-Bis(trifluoromethyl)benzyl)-3-ethyl-1-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86370A3CLONEDHUMAN3H-PSB-118-(3,5-Bis(trifluoromethyl)benzyl)-3-ethyl-1-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86371A3CLONEDHUMAN3H-PSB-118-(2-Bromobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86372A2BCLONEDHUMAN3H-PSB-6038-(2-Bromobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86373A2ASTRIATUMRAT3H-MSX-28-(2-Bromobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86374A1CORTEXRAT3H-CCPA8-(2-Bromobenzyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86375A1CORTEXRAT3H-CCPA1-Methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86376A2ASTRIATUMRAT3H-MSX-21-Methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86377A2BCLONEDHUMAN3H-PSB-6031-Methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86378A3CLONEDHUMAN3H-PSB-111-Methyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86379A3CLONEDHUMAN3H-PSB-118-(3-Chlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86380A2BCLONEDHUMAN3H-PSB-6038-(3-Chlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86381A2ASTRIATUMRAT3H-MSX-28-(3-Chlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86382A1CORTEXRAT3H-CCPA8-(3-Chlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86383A1CORTEXRAT3H-CCPA8-(3-Bromophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86384A2ASTRIATUMRAT3H-MSX-28-(3-Bromophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86385A2BCLONEDHUMAN3H-PSB-6038-(3-Bromophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86386A3CLONEDHUMAN3H-PSB-118-(3-Bromophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86387A3CLONEDHUMAN3H-PSB-111-Methyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86388A2BCLONEDHUMAN3H-PSB-6031-Methyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione300Koch P et al 2018Jan 15, 2025Jan 15, 2025
86389A2ASTRIATUMRAT3H-MSX-21-Methyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86390A1CORTEXRAT3H-CCPA1-Methyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86391A1CORTEXRAT3H-CCPA8-(2,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86392A2ASTRIATUMRAT3H-MSX-28-(2,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86393A2BCLONEDHUMAN3H-PSB-6038-(2,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86394A3CLONEDHUMAN3H-PSB-118-(2,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86395A3CLONEDHUMAN3H-PSB-118-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86396A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86397A2ASTRIATUMRAT3H-MSX-28-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86398A1CORTEXRAT3H-CCPA8-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86399A1CORTEXRAT3H-CCPA8-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86400A2ASTRIATUMRAT3H-MSX-28-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86401A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86402A3CLONEDHUMAN3H-PSB-118-(3,4-Dichlorophenethyl)-1-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86403A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(2-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7820Koch P et al 2018Jan 15, 2025Jan 15, 2025
86404A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(2-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86405A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(2-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione156Koch P et al 2018Jan 15, 2025Jan 15, 2025
86406A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(2-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione32Koch P et al 2018Jan 15, 2025Jan 15, 2025
86407A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(2-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione2000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86408A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(3-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1580Koch P et al 2018Jan 15, 2025Jan 15, 2025
86409A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(3-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione47.2Koch P et al 2018Jan 15, 2025Jan 15, 2025
86410A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(3-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione207Koch P et al 2018Jan 15, 2025Jan 15, 2025
86411A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(3-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86412A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(3-fluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7020Koch P et al 2018Jan 15, 2025Jan 15, 2025
86413A3CLONEDHUMAN3H-PSB-118-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione5410Koch P et al 2018Jan 15, 2025Jan 15, 2025
86414A2BCLONEDHUMAN3H-PSB-6038-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86415A2ACLONEDHUMAN3H-MSX-28-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione2380Koch P et al 2018Jan 15, 2025Jan 15, 2025
86416A1CLONEDHUMAN3H-CCPA8-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione128Koch P et al 2018Jan 15, 2025Jan 15, 2025
86417A1CORTEXRAT3H-CCPA8-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione85.9Koch P et al 2018Jan 15, 2025Jan 15, 2025
86418A2ASTRIATUMRAT3H-MSX-28-(3-Chlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86419A2ASTRIATUMRAT3H-MSX-28-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1040Koch P et al 2018Jan 15, 2025Jan 15, 2025
86420A1CORTEXRAT3H-CCPA8-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione21.5Koch P et al 2018Jan 15, 2025Jan 15, 2025
86421A1CLONEDHUMAN3H-CCPA8-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione13.6Koch P et al 2018Jan 15, 2025Jan 15, 2025
86422A2ACLONEDHUMAN3H-MSX-28-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1050Koch P et al 2018Jan 15, 2025Jan 15, 2025
86423A2BCLONEDHUMAN3H-PSB-6038-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione496Koch P et al 2018Jan 15, 2025Jan 15, 2025
86424A3CLONEDHUMAN3H-PSB-118-(3-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7220Koch P et al 2018Jan 15, 2025Jan 15, 2025
86425A3CLONEDHUMAN3H-PSB-118-(4-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86426A2BCLONEDHUMAN3H-PSB-6038-(4-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86427A2ACLONEDHUMAN3H-MSX-28-(4-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione4420Koch P et al 2018Jan 15, 2025Jan 15, 2025
86428A2ASTRIATUMRAT3H-MSX-28-(4-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1140Koch P et al 2018Jan 15, 2025Jan 15, 2025
86429A1CORTEXRAT3H-CCPA8-(4-Bromobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione54Koch P et al 2018Jan 15, 2025Jan 15, 2025
86430A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione51.4Koch P et al 2018Jan 15, 2025Jan 15, 2025
86431A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86432A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione129Koch P et al 2018Jan 15, 2025Jan 15, 2025
86433A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86434A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(2-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione4060Koch P et al 2018Jan 15, 2025Jan 15, 2025
86435A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86436A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86437A2ACLONEDHUMAN3H-MSX-21,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione277Koch P et al 2018Jan 15, 2025Jan 15, 2025
86438A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione84.8Koch P et al 2018Jan 15, 2025Jan 15, 2025
86439A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione30Koch P et al 2018Jan 15, 2025Jan 15, 2025
86440A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(3-(trifluoromethyl)benzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1030Koch P et al 2018Jan 15, 2025Jan 15, 2025
86441A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione895Koch P et al 2018Jan 15, 2025Jan 15, 2025
86442A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione172Koch P et al 2018Jan 15, 2025Jan 15, 2025
86443A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione189Koch P et al 2018Jan 15, 2025Jan 15, 2025
86444A2ACLONEDHUMAN3H-MSX-21,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione663Koch P et al 2018Jan 15, 2025Jan 15, 2025
86445A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86446A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(2-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86447A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(4-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86448A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(4-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86449A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(4-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86450A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(4-fluoro-3-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86451A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione124Koch P et al 2018Jan 15, 2025Jan 15, 2025
86452A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione600Koch P et al 2018Jan 15, 2025Jan 15, 2025
86453A2ACLONEDHUMAN3H-MSX-21,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione781Koch P et al 2018Jan 15, 2025Jan 15, 2025
86454A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione39.4Koch P et al 2018Jan 15, 2025Jan 15, 2025
86455A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86456A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(2-fluoro-5-(trifluoromethyl)benzyl)- 6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86457A3CLONEDHUMAN3H-PSB-118-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7190Koch P et al 2018Jan 15, 2025Jan 15, 2025
86458A2BCLONEDHUMAN3H-PSB-6038-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86459A2ACLONEDHUMAN3H-MSX-28-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione756Koch P et al 2018Jan 15, 2025Jan 15, 2025
86460A1CLONEDHUMAN3H-CCPA8-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione362Koch P et al 2018Jan 15, 2025Jan 15, 2025
86461A1CORTEXRAT3H-CCPA8-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione270Koch P et al 2018Jan 15, 2025Jan 15, 2025
86462A2ASTRIATUMRAT3H-MSX-28-(3-Bromo-4-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86463A1CLONEDHUMAN3H-CCPA8-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione75.4Koch P et al 2018Jan 15, 2025Jan 15, 2025
86464A2ACLONEDHUMAN3H-MSX-28-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione598Koch P et al 2018Jan 15, 2025Jan 15, 2025
86465A2BCLONEDHUMAN3H-PSB-6038-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86466A3CLONEDHUMAN3H-PSB-118-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86467A2ASTRIATUMRAT3H-MSX-28-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione756Koch P et al 2018Jan 15, 2025Jan 15, 2025
86468A1CORTEXRAT3H-CCPA8-(5-Bromo-2-fluorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione33.5Koch P et al 2018Jan 15, 2025Jan 15, 2025
86469A1CORTEXRAT3H-CCPA8-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione89.6Koch P et al 2018Jan 15, 2025Jan 15, 2025
86470A2ASTRIATUMRAT3H-MSX-28-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione2200Koch P et al 2018Jan 15, 2025Jan 15, 2025
86471A1CLONEDHUMAN3H-CCPA8-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione207Koch P et al 2018Jan 15, 2025Jan 15, 2025
86472A2ACLONEDHUMAN3H-MSX-28-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione631Koch P et al 2018Jan 15, 2025Jan 15, 2025
86473A2BCLONEDHUMAN3H-PSB-6038-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86474A3CLONEDHUMAN3H-PSB-118-(3,5-Dichlorobenzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione4720Koch P et al 2018Jan 15, 2025Jan 15, 2025
86475A3CLONEDHUMAN3H-PSB-118-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86476A2BCLONEDHUMAN3H-PSB-6038-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86477A2ACLONEDHUMAN3H-MSX-28-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione613Koch P et al 2018Jan 15, 2025Jan 15, 2025
86478A1CLONEDHUMAN3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione22.6Koch P et al 2018Jan 15, 2025Jan 15, 2025
86479A1CORTEXRAT3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione19.6Koch P et al 2018Jan 15, 2025Jan 15, 2025
86480A2ASTRIATUMRAT3H-MSX-28-(2-Chloro-5-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione871Koch P et al 2018Jan 15, 2025Jan 15, 2025
86481A2ASTRIATUMRAT3H-MSX-28-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86482A1CORTEXRAT3H-CCPA8-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86483A2BCLONEDHUMAN3H-PSB-6038-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86484A3CLONEDHUMAN3H-PSB-118-(4-Chloro-2-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1690Koch P et al 2018Jan 15, 2025Jan 15, 2025
86485A3CLONEDHUMAN3H-PSB-118-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7180Koch P et al 2018Jan 15, 2025Jan 15, 2025
86486A2BCLONEDHUMAN3H-PSB-6038-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86487A1CLONEDHUMAN3H-CCPA8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione129Koch P et al 2018Jan 15, 2025Jan 15, 2025
86488A1CORTEXRAT3H-CCPA8-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione588Koch P et al 2018Jan 15, 2025Jan 15, 2025
86489A2ASTRIATUMRAT3H-MSX-28-(4-Chloro-3-(trifluoromethyl)benzyl)-1,3-diethyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86490A2ASTRIATUMRAT3H-MSX-28-(3,5-Bis(trifluoromethyl)benzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86491A1CORTEXRAT3H-CCPA8-(3,5-Bis(trifluoromethyl)benzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86492A2BCLONEDHUMAN3H-PSB-6038-(3,5-Bis(trifluoromethyl)benzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86493A3CLONEDHUMAN3H-PSB-118-(3,5-Bis(trifluoromethyl)benzyl)-1,3-diethyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86494A3CLONEDHUMAN3H-PSB-111,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86495A2BCLONEDHUMAN3H-PSB-6031,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86496A2ACLONEDHUMAN3H-MSX-21,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione4110Koch P et al 2018Jan 15, 2025Jan 15, 2025
86497A1CLONEDHUMAN3H-CCPA1,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1190Koch P et al 2018Jan 15, 2025Jan 15, 2025
86498A1CORTEXRAT3H-CCPA1,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1500Koch P et al 2018Jan 15, 2025Jan 15, 2025
86499A2ASTRIATUMRAT3H-MSX-21,3-Diethyl-8-(3,4,5-trifluorobenzyl)-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86500A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(2-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1380Koch P et al 2018Jan 15, 2025Jan 15, 2025
86501A1CORTEXRAT3H-CCPA1-Ethyl-8-(2-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1140Koch P et al 2018Jan 15, 2025Jan 15, 2025
86502A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(2-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86503A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(2-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione4270Koch P et al 2018Jan 15, 2025Jan 15, 2025
86504A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione2390Koch P et al 2018Jan 15, 2025Jan 15, 2025
86505A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86506A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione378Koch P et al 2018Jan 15, 2025Jan 15, 2025
86507A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1530Koch P et al 2018Jan 15, 2025Jan 15, 2025
86508A1CORTEXRAT3H-CCPA1-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione410Koch P et al 2018Jan 15, 2025Jan 15, 2025
86509A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(4-fluorophenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione128Koch P et al 2018Jan 15, 2025Jan 15, 2025
86510A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione250Koch P et al 2018Jan 15, 2025Jan 15, 2025
86511A1CORTEXRAT3H-CCPA1-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione328Koch P et al 2018Jan 15, 2025Jan 15, 2025
86512A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione946Koch P et al 2018Jan 15, 2025Jan 15, 2025
86513A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione289Koch P et al 2018Jan 15, 2025Jan 15, 2025
86514A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86515A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(3-methoxyphenyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7160Koch P et al 2018Jan 15, 2025Jan 15, 2025
86516A3CLONEDHUMAN3H-PSB-118-(3,4-Dimethoxyphenyl)-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione3640Koch P et al 2018Jan 15, 2025Jan 15, 2025
86517A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dimethoxyphenyl)-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86518A2ASTRIATUMRAT3H-MSX-28-(3,4-Dimethoxyphenyl)-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1580Koch P et al 2018Jan 15, 2025Jan 15, 2025
86519A1CORTEXRAT3H-CCPA8-(3,4-Dimethoxyphenyl)-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1670Koch P et al 2018Jan 15, 2025Jan 15, 2025
86520A1CORTEXRAT3H-CCPA8-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione118Koch P et al 2018Jan 15, 2025Jan 15, 2025
86521A2ASTRIATUMRAT3H-MSX-28-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione245Koch P et al 2018Jan 15, 2025Jan 15, 2025
86522A1CLONEDHUMAN3H-CCPA8-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione180Koch P et al 2018Jan 15, 2025Jan 15, 2025
86523A2ACLONEDHUMAN3H-MSX-28-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione282Koch P et al 2018Jan 15, 2025Jan 15, 2025
86524A2BCLONEDHUMAN3H-PSB-6038-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86525A3CLONEDHUMAN3H-PSB-118-Benzyl-1-ethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86526A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7640Koch P et al 2018Jan 15, 2025Jan 15, 2025
86527A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86528A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione311Koch P et al 2018Jan 15, 2025Jan 15, 2025
86529A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione210Koch P et al 2018Jan 15, 2025Jan 15, 2025
86530A1CORTEXRAT3H-CCPA1-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione32.7Koch P et al 2018Jan 15, 2025Jan 15, 2025
86531A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(2-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1200Koch P et al 2018Jan 15, 2025Jan 15, 2025
86532A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione769Koch P et al 2018Jan 15, 2025Jan 15, 2025
86533A1CORTEXRAT3H-CCPA1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione118Koch P et al 2018Jan 15, 2025Jan 15, 2025
86534A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione124Koch P et al 2018Jan 15, 2025Jan 15, 2025
86535A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione542Koch P et al 2018Jan 15, 2025Jan 15, 2025
86536A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86537A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(3-methoxybenzyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86538A1CLONEDHUMAN3H-CCPA1-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione2440Koch P et al 2018Jan 15, 2025Jan 15, 2025
86539A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione149Koch P et al 2018Jan 15, 2025Jan 15, 2025
86540A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86541A3CLONEDHUMAN3H-PSB-111-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86542A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione1700Koch P et al 2018Jan 15, 2025Jan 15, 2025
86543A1CORTEXRAT3H-CCPA1-Ethyl-8-phenethyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1h,3h)- dione117Koch P et al 2018Jan 15, 2025Jan 15, 2025
86544A1CORTEXRAT3H-CCPA1-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione701Koch P et al 2018Jan 15, 2025Jan 15, 2025
86545A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione883Koch P et al 2018Jan 15, 2025Jan 15, 2025
86546A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione3230Koch P et al 2018Jan 15, 2025Jan 15, 2025
86547A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1260Koch P et al 2018Jan 15, 2025Jan 15, 2025
86548A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86549A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(2-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione5830Koch P et al 2018Jan 15, 2025Jan 15, 2025
86550A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86551A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86552A2ACLONEDHUMAN3H-MSX-21-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86553A1CLONEDHUMAN3H-CCPA1-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1020Koch P et al 2018Jan 15, 2025Jan 15, 2025
86554A1CORTEXRAT3H-CCPA1-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione669Koch P et al 2018Jan 15, 2025Jan 15, 2025
86555A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(3-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione798Koch P et al 2018Jan 15, 2025Jan 15, 2025
86556A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione2700Koch P et al 2018Jan 15, 2025Jan 15, 2025
86557A1CORTEXRAT3H-CCPA1-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1600Koch P et al 2018Jan 15, 2025Jan 15, 2025
86558A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86559A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(4-methoxyphenethyl)-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86560A3CLONEDHUMAN3H-PSB-111-Ethyl-8-(2,3-dimethoxyphenethyl)-3-propargyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86561A2BCLONEDHUMAN3H-PSB-6031-Ethyl-8-(2,3-dimethoxyphenethyl)-3-propargyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86562A2ASTRIATUMRAT3H-MSX-21-Ethyl-8-(2,3-dimethoxyphenethyl)-3-propargyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione7400Koch P et al 2018Jan 15, 2025Jan 15, 2025
86563A1CORTEXRAT3H-CCPA1-Ethyl-8-(2,3-dimethoxyphenethyl)-3-propargyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione3800Koch P et al 2018Jan 15, 2025Jan 15, 2025
86564A1CORTEXRAT3H-CCPA8-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione236Koch P et al 2018Jan 15, 2025Jan 15, 2025
86565A2ASTRIATUMRAT3H-MSX-28-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1100Koch P et al 2018Jan 15, 2025Jan 15, 2025
86566A2ACLONEDHUMAN3H-MSX-28-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1620Koch P et al 2018Jan 15, 2025Jan 15, 2025
86567A1CLONEDHUMAN3H-CCPA8-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione396Koch P et al 2018Jan 15, 2025Jan 15, 2025
86568A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86569A3CLONEDHUMAN3H-PSB-118-(3,4-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86570A3CLONEDHUMAN3H-PSB-118-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86571A2BCLONEDHUMAN3H-PSB-6038-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86572A2ACLONEDHUMAN3H-MSX-28-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione2230Koch P et al 2018Jan 15, 2025Jan 15, 2025
86573A1CLONEDHUMAN3H-CCPA8-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione143Koch P et al 2018Jan 15, 2025Jan 15, 2025
86574A1CORTEXRAT3H-CCPA8-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione49.3Koch P et al 2018Jan 15, 2025Jan 15, 2025
86575A2ASTRIATUMRAT3H-MSX-28-(3,5-Dichlorobenzyl)-1-ethyl-3-methyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1490Koch P et al 2018Jan 15, 2025Jan 15, 2025
86576A2ASTRIATUMRAT3H-MSX-28-(3,4-Dichlorobenzyl)-1-cyclopropyl-3-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione3940Koch P et al 2018Jan 15, 2025Jan 15, 2025
86577A1CORTEXRAT3H-CCPA8-(3,4-Dichlorobenzyl)-1-cyclopropyl-3-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione584Koch P et al 2018Jan 15, 2025Jan 15, 2025
86578A1CLONEDHUMAN3H-CCPA8-(3,4-Dichlorobenzyl)-1-cyclopropyl-3-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1130Koch P et al 2018Jan 15, 2025Jan 15, 2025
86579A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dichlorobenzyl)-1-cyclopropyl-3-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione100Koch P et al 2018Jan 15, 2025Jan 15, 2025
86580A3CLONEDHUMAN3H-PSB-118-(3,4-Dichlorobenzyl)-1-cyclopropyl-3-methyl6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86581A3CLONEDHUMAN3H-PSB-118-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86582A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86583A2ACLONEDHUMAN3H-MSX-28-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione2110Koch P et al 2018Jan 15, 2025Jan 15, 2025
86584A1CLONEDHUMAN3H-CCPA8-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione475Koch P et al 2018Jan 15, 2025Jan 15, 2025
86585A1CORTEXRAT3H-CCPA8-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione152Koch P et al 2018Jan 15, 2025Jan 15, 2025
86586A2ASTRIATUMRAT3H-MSX-28-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione675Koch P et al 2018Jan 15, 2025Jan 15, 2025
86587A2ASTRIATUMRAT3H-MSX-28-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione642Koch P et al 2018Jan 15, 2025Jan 15, 2025
86588A1CORTEXRAT3H-CCPA8-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione292Koch P et al 2018Jan 15, 2025Jan 15, 2025
86589A1CLONEDHUMAN3H-CCPA8-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione967Koch P et al 2018Jan 15, 2025Jan 15, 2025
86590A2ACLONEDHUMAN3H-MSX-28-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1580Koch P et al 2018Jan 15, 2025Jan 15, 2025
86591A2BCLONEDHUMAN3H-PSB-6038-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86592A3CLONEDHUMAN3H-PSB-118-(3,4-Dichlorobenzyl)-1-methyl-3-propargyl-6,7,8,9- tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)- dione5630Koch P et al 2018Jan 15, 2025Jan 15, 2025
86593A3CLONEDHUMAN3H-PSB-118-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione>10000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86594A2BCLONEDHUMAN3H-PSB-6038-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione1000Koch P et al 2018Jan 15, 2025Jan 15, 2025
86595A2ACLONEDHUMAN3H-MSX-28-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione712Koch P et al 2018Jan 15, 2025Jan 15, 2025
86596A1CLONEDHUMAN3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione110Koch P et al 2018Jan 15, 2025Jan 15, 2025
86597A1CORTEXRAT3H-CCPA8-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione153Koch P et al 2018Jan 15, 2025Jan 15, 2025
86598A2ASTRIATUMRAT3H-MSX-28-(2-Chloro-5-(trifluoromethyl)benzyl)-1-methyl-3- propargyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine2,4(1H,3H)-dione414Koch P et al 2018Jan 15, 2025Jan 15, 2025
865995-HT4CLONEDHUMAN3H-GR-1138081-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide0.0794328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866005-HT2ACLONEDHUMAN3H-KETANSERIN1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide31.6228Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866015-HT2ACLONEDHUMAN3H-KETANSERINN-[[1-(2-Phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866025-HT4CLONEDHUMAN3H-GR113808N-[[1-(2-Phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide0.630957Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866035-HT4CLONEDHUMAN3H-GR1138081-Isopropyl-N-[[1-(2-pyridin-2-ylethyl)-4-piperidinyl]methyl]-1Hindazole-3-carboxamide0.1Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866045-HT2ACLONEDHUMAN3H-KETANSERIN1-Isopropyl-N-[[1-(2-pyridin-2-ylethyl)-4-piperidinyl]methyl]-1Hindazole-3-carboxamide100Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866055-HT2ACLONEDHUMAN3H-KETANSERIN4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]-1- methyl-1-(2-phenylethyl)piperidinium Iodide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866065-HT4CLONEDHUMAN3H-GR1138084-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]-1- methyl-1-(2-phenylethyl)piperidinium Iodide31.6228Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866075-HT4CLONEDHUMAN3H-GR113808N-[[1-(2-Cyclohexylethyl)-4-piperidinyl]methyl]-1-isopropyl-1Hindazole-3-carboxamide0.158489Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866085-HT2ACLONEDHUMAN3H-KETANSERINN-[[1-(2-Cyclohexylethyl)-4-piperidinyl]methyl]-1-isopropyl-1Hindazole-3-carboxamide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866095-HT2ACLONEDHUMAN3H-KETANSERIN1-Isopropyl-N-[[1-(2-morpholin-4-ylethyl]-4-piperidinyl]methyl]- 1H-indazole-3-carboxamide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866105-HT4CLONEDHUMAN3H-GR1138081-Isopropyl-N-[[1-(2-morpholin-4-ylethyl]-4-piperidinyl]methyl]- 1H-indazole-3-carboxamide0.398107Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866115-HT4CLONEDHUMAN3H-GR113808N-[[1-[3-(Dimethylamino)propyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide0.794328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866125-HT2ACLONEDHUMAN3H-KETANSERINN-[[1-[3-(Dimethylamino)propyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866135-HT2ACLONEDHUMAN3H-KETANSERIN1-Isopropyl-N-[[1-[2-[(methylsulfonyl)amino]ethyl]-4- piperidinyl]methyl]-1H-indazole-3-carboxamide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866145-HT4CLONEDHUMAN3H-GR1138081-Isopropyl-N-[[1-[3-(methylamino)-3-oxo-1-propyl]-4- piperidinyl]methyl]-1H-indazole-3-carboxamide0.501187Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866155-HT4CLONEDHUMAN3H-GR1138081-Isopropyl-N-[[1-[2-(4-hydroxyphenyl)ethyl]-4-piperidinyl]- methyl]-1H-indazole-3-carboxamide0.251189Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866165-HT2ACLONEDHUMAN3H-KETANSERIN1-Isopropyl-N-[[1-[2-(4-hydroxyphenyl)ethyl]-4-piperidinyl]- methyl]-1H-indazole-3-carboxamide10Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866175-HT2ACLONEDHUMAN3H-KETANSERIN1-Isopropyl-N-[[1-[2-(4-nitrophenyl)ethyl]-4-piperidinyl]methyl]- 1H-indazole-3-carboxamide1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866185-HT4CLONEDHUMAN3H-GR1138081-Isopropyl-N-[[1-[2-(4-nitrophenyl)ethyl]-4-piperidinyl]methyl]- 1H-indazole-3-carboxamide1.25893Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866195-HT4CLONEDHUMAN3H-GR113808N-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide0.199526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866205-HT2ACLONEDHUMAN3H-KETANSERINN-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methyl]-1-isopropyl-1H-indazole-3-carboxamide79.4328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866215-HT2ACLONEDHUMAN3H-KETANSERIN4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866225-HT4CLONEDHUMAN3H-GR-1138084-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid0.794328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866235-HT4CLONEDHUMAN3H-GR-113808piboserod0.158489Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866245-HT2ACLONEDHUMAN3H-KETANSERINMETHYSERGIDE1.58489Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866255-HT4CLONEDHUMAN3H-GR1138082-Methyl-4-(4-piperidinylmethoxy)-2H-pyrrolo[3,4-c]quinoline398.107Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866265-HT4CLONEDHUMAN3H-GR1138084-[(1-Butyl-4-piperidinyl)methoxy]-2-methyl-2H-pyrrolo[3,4-c]- quinoline7.94328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866275-HT2ACLONEDHUMAN3H-KETANSERIN4-[(1-Butyl-4-piperidinyl)methoxy]-2-methyl-2H-pyrrolo[3,4-c]- quinoline1000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866285-HT2ACLONEDHUMAN3H-KETANSERIN2-Methyl-4-[[1-(2-phenylethyl)-4-piperidinyl]methoxy]-2Hpyrrolo[3,4-c]quinoline79.4328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866295-HT4CLONEDHUMAN3H-GR1138082-Methyl-4-[[1-(2-phenylethyl)-4-piperidinyl]methoxy]-2Hpyrrolo[3,4-c]quinoline1.99526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866305-HT4CLONEDHUMAN3H-GR1138082-Isopropyl-4-[[1-(2-phenylethyl)-4-piperidinyl]methoxy]-2Hpyrrolo[3,4-c]quinoline125.893Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866315-HT2ACLONEDHUMAN3H-KETANSERIN2-Isopropyl-4-[[1-(2-phenylethyl)-4-piperidinyl]methoxy]-2Hpyrrolo[3,4-c]quinoline100Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866325-HT2ACLONEDHUMAN3H-KETANSERIN2-Methyl-4-[[1-(2-morpholin-4-ylethyl)-4-piperidinyl]methoxy]- 2H-pyrrolo[3,4-c]quinoline>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866335-HT2ACLONEDHUMAN3H-KETANSERIN2-Methyl-4-[[1-(2-morpholin-4-ylethyl)-4-piperidinyl]methoxy]- 2H-pyrrolo[3,4-c]quinoline>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866345-HT4CLONEDHUMAN3H-GR1138082-Methyl-4-[[1-(2-morpholin-4-ylethyl)-4-piperidinyl]methoxy]- 2H-pyrrolo[3,4-c]quinoline2.51189Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866355-HT4CLONEDHUMAN3H-GR1138084-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methoxy]-2-methyl2H-pyrrolo[3,4-c]quinoline5.01187Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866365-HT2ACLONEDHUMAN3H-KETANSERIN4-[[1-[2-(4-Aminophenyl)ethyl]-4-piperidinyl]methoxy]-2-methyl2H-pyrrolo[3,4-c]quinoline251.189Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866375-HT2ACLONEDHUMAN3H-KETANSERIN4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866385-HT4CLONEDHUMAN3H-GR1138084-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid1.99526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866395-HT4CLONEDHUMAN3H-GR1138082-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid199.526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866405-HT2ACLONEDHUMAN3H-KETANSERIN2-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid794.328Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866415-HT2ACLONEDHUMAN3H-KETANSERIN4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzenemethanol31.6228Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866425-HT4CLONEDHUMAN3H-GR1138084-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzenemethanol10Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866435-HT4CLONEDHUMAN3H-GR1138084-[[1-[2-[4-(Methoxymethyl)phenyl]ethyl]-4-piperidinyl]- methoxy]-2-methyl-2H-pyrrolo[3,4-c]quinoline19.9526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866445-HT2ACLONEDHUMAN3H-KETANSERIN4-[[1-[2-[4-(Methoxymethyl)phenyl]ethyl]-4-piperidinyl]- methoxy]-2-methyl-2H-pyrrolo[3,4-c]quinoline199.526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866455-HT2ACLONEDHUMAN3H-KETANSERIN4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]phenylacetamide3162.28Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866465-HT4CLONEDHUMAN3H-GR1138084-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]phenylacetamide1.99526Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866475-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866485-HT1BSTRIATUMRAT125I-ICYPN-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866495-HT1DSTRIATUMBOVINE3H-5-CTN-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866505-HT2CCLONEDHUMAN3H-MESULERGINEN-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866515-HT3CLONEDHUMAN3H-GR-65630N-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866525-HT6CLONEDHUMAN3H-LSDN-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866535-HT7CLONEDHUMAN3H-LSDN-[(1-Butyl-4-piperidinyl)methyl]-1-methyl-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866545-HT1ACLONEDHUMAN3H-8-OH-DPAT1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866555-HT1BSTRIATUMRAT125I-ICYP1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866565-HT1DSTRIATUMBOVINE3H-5-CT1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866575-HT3CLONEDHUMAN3H-GR656301-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866585-HT6CLONEDHUMAN3H-LSD1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866595-HT7CLONEDHUMAN3H-LSD1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
86660SERTCLONEDHUMAN3H-N-Me-citalopram1-Methyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
866615-HT1ACLONEDHUMAN3H-8-OH-DPAT1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866625-HT1BSTRIATUMRAT125I-ICYP1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866635-HT1DSTRIATUMBOVINE3H-5-CT1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866645-HT2CCLONEDHUMAN3H-MESULERGINE1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866655-HT3CLONEDHUMAN3H-GR-656301-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866665-HT6CLONEDHUMAN3H-LSD1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866675-HT7CLONEDHUMAN3H-LSD1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
86668SERTCLONEDHUMAN3H-N-Me-citalopram1-Isopropyl-N-[[1-(2-phenylethyl)-4-piperidinyl]methyl]-1H-indazole-3-carboxamide>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86669Alpha1ASUBMAXILLARY GLANDRAT3H-PRAZOSIN4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86670Alpha1BLIVERRAT3H-PRAZOSIN4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86671Alpha1DCLONEDHUMAN3H-PRAZOSIN4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86672CORTEXRAT3H-QNB4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866735-HT1ACLONEDHUMAN3H-8-OH-DPAT4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866745-HT1BCORTEXRAT125I-ICYP4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866755-HT2BCLONEDHUMAN3H-LSD4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866765-HT2CCLONEDHUMAN3H-MESULERGINE4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866775-HT3CLONEDHUMAN3H-GR-656304-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866785-HT5ACLONEDHUMAN3H-LSD4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866795-HT6CLONEDHUMAN3H-LSD4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866805-HT7CLONEDHUMAN3H-LSD4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
86681Sigma 1Jurkat cellsHUMAN3H-Pentazocine(+)4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86682Sigma 2BRAINRAT3H-DTG4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86683BRAINRAT3H-Alpha-Bungarotoxin4-[2-[4-[[[(1-Isopropyl-1H-indazol-3-yl)carbonyl]amino]methyl]- 1-piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
86684BRAINRAT3H-Alpha-Bungarotoxin4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
86685Alpha1ASUBMAXILLARY GLANDRAT3H-PRAZOSIN4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86686Alpha1BLIVERRAT3H-PRAZOSIN4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86687Alpha1DCLONEDHUMAN3H-PRAZOSIN4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86688CORTEXRAT3H-QNB4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866895-HT1ACLONEDHUMAN3H-8-OH-DPAT4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866905-HT1BCORTEXRAT125I-ICYP4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866915-HT2BCLONEDHUMAN3H-LSD4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866925-HT2CCLONEDHUMAN3H-MESULERGINE4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866935-HT3CLONEDHUMAN3H-GR-656304-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866945-HT5ACLONEDHUMAN3H-LSD4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866955-HT6CLONEDHUMAN3H-LSD4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
866965-HT7CLONEDHUMAN3H-LSD4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 15, 2025
86697Sigma 1Jurkat cellsHUMAN3H-Pentazocine(+)4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
86698SERTCLONEDHUMAN3H-N-Me-citalopram4-[2-[4-[[(2-Methyl-2H-pyrrolo[3,4-c]-4-quinolinyl)oxy]methyl]-1- piperidinyl]ethyl]benzoic Acid>10000Furlotti G et al 2012Jan 15, 2025Jan 28, 2025
866995-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-phenylpiperazin-1-yl)ethyl)isonicotinamide8.74Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867005-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-phenylpiperazin-1-yl)ethyl)isonicotinamide199Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867015-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-phenylpiperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867025-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide0.933Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867035-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide587Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867045-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide0.36Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867055-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide1270Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867065-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide911Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867075-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide1330Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867085-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide5.1Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867095-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide16.2Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867105-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide4.77Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867115-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl) isonicotinamide15.2Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867125-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl) isonicotinamide54.6Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867135-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867145-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(o-tolyl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867155-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(o-tolyl)piperazin-1-yl)ethyl)isonicotinamide631Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867165-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(o-tolyl)piperazin-1-yl)ethyl)isonicotinamide549Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867175-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) isonicotinamide16.7Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867185-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) isonicotinamide70.7Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867195-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) isonicotinamide2.23Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867205-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide6.79Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867215-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide469Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867225-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide2.85Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867235-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide0.82Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867245-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide35.5Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867255-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide0.156Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867265-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867275-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide664Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867285-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide334Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867295-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) isonicotinamide455Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867305-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) isonicotinamide9.85Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867315-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867325-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide100Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867335-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide0.0126Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867345-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide10.6Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867355-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide549Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867365-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide0.046Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867375-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867385-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867395-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867405-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1.08Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867415-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl) isonicotinamide157Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867425-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl) isonicotinamide2770Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867435-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867445-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(piperonyl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867455-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(piperonyl)piperazin-1-yl)ethyl)isonicotinamide0.793Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867465-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(piperonyl)piperazin-1-yl)ethyl)isonicotinamide36.2Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867475-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(furoyl)piperazin-1-yl)ethyl)isonicotinamide72.5Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867485-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(furoyl)piperazin-1-yl)ethyl)isonicotinamide3660Fiorino F et al 2016Jan 15, 2025Jan 15, 2025