The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 86,001-87,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
88749H1CLONEDHUMAN3H-PYRILAMINE3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol1009Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88750M1CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88751M2CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88752M3CLONEDHUMAN3H-QNB3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol>10000Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88753DATCLONEDHUMAN3H-WIN 35,4283-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol354Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88754NETCLONEDHUMAN3H-Nisoxetine3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol462Sampson D et al 2014Jan 15, 2025Jan 15, 2025
88755SERTCLONEDHUMAN3H-CITALOPRAM3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol102Sampson D et al 2014Jan 15, 2025Jan 28, 2025
88756A1CHO cellsHUMAN3H-DPCPXN-(4,6-diphenylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88757A2AHeLaHUMAN3H-ZM241385N-(4,6-diphenylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88758A2BCHO cellsHUMAN3H-DPCPXN-(4,6-diphenylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88759A3HeLaHUMAN3H-NECAN-(4,6-diphenylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88760A1CHO cellsHUMAN3H-DPCPXN-(4,6-diphenylpyrimidin-2-yl)propionamide31.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88761A2AHeLaHUMAN3H-ZM241385N-(4,6-diphenylpyrimidin-2-yl)propionamide554Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88762A2AHEK293 cellsHUMAN3H-DPCPXN-(4,6-diphenylpyrimidin-2-yl)propionamide42.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88763A3HeLaHUMAN3H-NECAN-(4,6-diphenylpyrimidin-2-yl)propionamide531Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88764A1CHO cellsHUMAN3H-DPCPXN-(4,6-diphenylpyrimidin-2-yl)butyramide10.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88765A2AHeLaHUMAN3H-ZM241385N-(4,6-diphenylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88766A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-diphenylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88767A3HeLaHUMAN3H-NECAN-(4,6-diphenylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88768A1CHO cellsHUMAN3H-DPCPXN-(4,6-dip-tolylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88769A2AHeLaHUMAN3H-ZM241385N-(4,6-dip-tolylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88770A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-dip-tolylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88771A3HeLaHUMAN3H-NECAN-(4,6-dip-tolylpyrimidin-2-yl)acetamide47.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88772A1CHO cellsHUMAN3H-DPCPXN-(4,6-di-tolylpyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88773A2AHeLaHUMAN3H-ZM241385N-(4,6-di-tolylpyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88774A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di-tolylpyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88775A3HeLaHUMAN3H-NECAN-(4,6-di-tolylpyrimidin-2-yl)propionamide157Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88776A1CHO cellsHUMAN3H-DPCPXN-(4,6-dip-tolylpyrimidin-2-yl)butyramide3760Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88777A2AHeLaHUMAN3H-ZM241385N-(4,6-dip-tolylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88778A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-dip-tolylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88779A3HeLaHUMAN3H-NECAN-(4,6-dip-tolylpyrimidin-2-yl)butyramide131Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88780A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88781A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88782A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88783A3HeLaHUMAN3H-NECAN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88784A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88785A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88786A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88787A3HeLaHUMAN3H-NECAN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88788A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88789A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88790A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88791A3HeLaHUMAN3H-NECAN-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88792A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88793A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88794A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88795A3HeLaHUMAN3H-NECAN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88796A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88797A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88798A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88799A3HeLaHUMAN3H-NECAN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88800A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88801A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88802A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88803A3HeLaHUMAN3H-NECAN-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88804A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88805A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88806A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88807A3HeLaHUMAN3H-NECAN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88808A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide505Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88809A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide183Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88810A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide374Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88811A3HeLaHUMAN3H-NECAN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide4435Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88812A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88813A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88814A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88815A3HeLaHUMAN3H-NECAN-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88816A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88817A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88818A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88819A3HeLaHUMAN3H-NECAN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88820A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88821A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88822A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88823A3HeLaHUMAN3H-NECAN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88824A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88825A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88826A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88827A3HeLaHUMAN3H-NECAN-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88828A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88829A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88830A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88831A3HeLaHUMAN3H-NECAN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88832A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88833A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88834A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88835A3HeLaHUMAN3H-NECAN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88836A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88837A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88838A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88839A3HeLaHUMAN3H-NECAN-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88840A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88841A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88842A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88843A3HeLaHUMAN3H-NECAN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88844A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88845A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88846A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88847A3HeLaHUMAN3H-NECAN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88848A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88849A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88850A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88851A3HeLaHUMAN3H-NECAN-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88852A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88853A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88854A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88855A3HeLaHUMAN3H-NECAN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88856A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide48.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88857A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide424Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88858A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide307Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88859A3HeLaHUMAN3H-NECAN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide279Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88860A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide23.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88861A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide647Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88862A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88863A3HeLaHUMAN3H-NECAN-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88864A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88865A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88866A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88867A3HeLaHUMAN3H-NECAN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88868A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88869A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88870A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88871A3HeLaHUMAN3H-NECAN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88872A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88873A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88874A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88875A3HeLaHUMAN3H-NECAN-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88876A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88877A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88878A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88879A3HeLaHUMAN3H-NECAN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88880A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88881A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88882A2BHeLaHUMAN3H-DPCPXN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88883A3HeLaHUMAN3H-NECAN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88884A1CHO cellsHUMAN3H-DPCPXN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88885A2AHeLaHUMAN3H-ZM241385N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88886A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88887A3HeLaHUMAN3H-NECAN-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88888A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88889A2AHeLaHUMAN3H-ZM241385N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88890A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88891A3HeLaHUMAN3H-NECAN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide101Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88892A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide535Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88893A2AHeLaHUMAN3H-ZM241385N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88894A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88895A3HeLaHUMAN3H-NECAN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide127Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88896A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide678Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88897A2AHeLaHUMAN3H-ZM241385N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88898A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88899A3HeLaHUMAN3H-NECAN-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide751Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88900A1CHO cellsHUMAN3H-DPCPXN-(4,6-distyrylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88901A2AHeLaHUMAN3H-ZM241385N-(4,6-distyrylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88902A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-distyrylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88903A3HeLaHUMAN3H-NECAN-(4,6-distyrylpyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88904A1CHO cellsHUMAN3H-DPCPXN-(4,6-distyrylpyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88905A2AHeLaHUMAN3H-ZM241385N-(4,6-distyrylpyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88906A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-distyrylpyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88907A3HeLaHUMAN3H-NECAN-(4,6-distyrylpyrimidin-2-yl)propionamide142Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88908A1CHO cellsHUMAN3H-DPCPXN-(4,6-distyrylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88909A2AHeLaHUMAN3H-ZM241385N-(4,6-distyrylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88910A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-distyrylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88911A3HeLaHUMAN3H-NECAN-(4,6-distyrylpyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88912A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88913A2AHeLaHUMAN3H-ZM241385N-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88914A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88915A3HeLaHUMAN3H-NECAN-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88916A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88917A2AHeLaHUMAN3H-ZM241385N-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88918A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88919A3HeLaHUMAN3H-NECAN-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide1903Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88920A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88921A2AHeLaHUMAN3H-ZM241385N-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88922A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88923A3HeLaHUMAN3H-NECAN-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88924A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88925A2AHeLaHUMAN3H-ZM241385N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88926A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88927A3HeLaHUMAN3H-NECAN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88928A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88929A2AHeLaHUMAN3H-ZM241385N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88930A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88931A3HeLaHUMAN3H-NECAN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88932A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide255Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88933A2AHeLaHUMAN3H-ZM241385N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide201Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88934A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88935A3HeLaHUMAN3H-NECAN-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88936A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88937A2AHeLaHUMAN3H-ZM241385N-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88938A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88939A3HeLaHUMAN3H-NECAN-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88940A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88941A2AHeLaHUMAN3H-ZM241385N-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88942A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88943A3HeLaHUMAN3H-NECAN-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88944A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88945A2AHeLaHUMAN3H-ZM241385N-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88946A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88947A3HeLaHUMAN3H-NECAN-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88948A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88949A2AHeLaHUMAN3H-ZM241385N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88950A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88951A3HeLaHUMAN3H-NECAN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88952A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide367Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88953A2AHeLaHUMAN3H-ZM241385N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide1893Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88954A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide3250Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88955A3HeLaHUMAN3H-NECAN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide1279Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88956A1CHO cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide85.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88957A2AHeLaHUMAN3H-ZM241385N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide4568Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88958A2BHEK293 cellsHUMAN3H-DPCPXN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88959A3HeLaHUMAN3H-NECAN-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88960A1CHO cellsHUMAN3H-DPCPXN-(2,6-diphenylpyrimidin-4-yl)acetamide31.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88961A2AHeLaHUMAN3H-ZM241385N-(2,6-diphenylpyrimidin-4-yl)acetamide255.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88962A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-diphenylpyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88963A3HeLaHUMAN3H-NECAN-(2,6-diphenylpyrimidin-4-yl)acetamide12.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88964A1CHO cellsHUMAN3H-DPCPXN-(2,6-diphenylpyrimidin-4-yl)propionamide22.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88965A2AHeLaHUMAN3H-ZM241385N-(2,6-diphenylpyrimidin-4-yl)propionamide84.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88966A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-diphenylpyrimidin-4-yl)propionamide76.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88967A3HeLaHUMAN3H-NECAN-(2,6-diphenylpyrimidin-4-yl)propionamide45.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88968A1CHO cellsHUMAN3H-DPCPXN-(2,6-diphenylpyrimidin-4-yl)butyramide19.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88969A2AHeLaHUMAN3H-ZM241385N-(2,6-diphenylpyrimidin-4-yl)butyramide103Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88970A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-diphenylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88971A3HeLaHUMAN3H-NECAN-(2,6-diphenylpyrimidin-4-yl)butyramide171Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88972A1CHO cellsHUMAN3H-DPCPXISVY133100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88973A2AHeLaHUMAN3H-ZM241385ISVY133100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88974A2BHEK293 cellsHUMAN3H-DPCPXISVY133100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88975A3HeLaHUMAN3H-NECAISVY1334.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88976A1CHO cellsHUMAN3H-DPCPXN-(2,6-di-p-tolylpyrimidin-4-yl)propionamide36.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88977A2AHeLaHUMAN3H-ZM241385N-(2,6-di-p-tolylpyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88978A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di-p-tolylpyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88979A3HeLaHUMAN3H-NECAN-(2,6-di-p-tolylpyrimidin-4-yl)propionamide18.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88980A1CHO cellsHUMAN3H-DPCPXN-(2,6-di-p-tolylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88981A2AHeLaHUMAN3H-ZM241385N-(2,6-di-p-tolylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88982A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di-p-tolylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88983A3HeLaHUMAN3H-NECAN-(2,6-di-p-tolylpyrimidin-4-yl)butyramide59Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88984A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88985A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88986A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88987A3HeLaHUMAN3H-NECAN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide126Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88988A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88989A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88990A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88991A3HeLaHUMAN3H-NECAN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88992A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88993A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88994A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88995A3HeLaHUMAN3H-NECAN-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88996A1CHO cellsHUMAN3H-DPCPXISVY130100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88997A2AHeLaHUMAN3H-ZM241385ISVY130100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88998A2BHEK293 cellsHUMAN3H-DPCPXISVY130100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
88999A3HeLaHUMAN3H-NECAISVY1303.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89000A1CHO cellsHUMAN3H-DPCPXISVY074100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89001A2AHeLaHUMAN3H-ZM241385ISVY074100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89002A2BHEK293 cellsHUMAN3H-DPCPXISVY074100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89003A3HeLaHUMAN3H-NECAISVY0743.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89004A1CHO cellsHUMAN3H-DPCPXISVY071100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89005A2AHeLaHUMAN3H-ZM241385ISVY071100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89006A2BHEK293 cellsHUMAN3H-DPCPXISVY071100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89007A3HeLaHUMAN3H-NECAISVY07111Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89008A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89009A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89010A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89011A3HeLaHUMAN3H-NECAN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide71.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89012A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89013A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89014A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89015A3HeLaHUMAN3H-NECAN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide43.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89016A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89017A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89018A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89019A3HeLaHUMAN3H-NECAN-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89020A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89021A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89022A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89023A3HeLaHUMAN3H-NECAN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide25.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89024A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89025A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89026A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89027A3HeLaHUMAN3H-NECAN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide43.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89028A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89029A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89030A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89031A3HeLaHUMAN3H-NECAN-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide133Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89032A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89033A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide1334Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89034A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89035A3HeLaHUMAN3H-NECAN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide16.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89036A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide83.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89037A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide429Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89038A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89039A3HeLaHUMAN3H-NECAN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide12.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89040A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide82.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89041A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide1829Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89042A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89043A3HeLaHUMAN3H-NECAN-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide34.8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89044A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89045A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89046A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89047A3HeLaHUMAN3H-NECAN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide63.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89048A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89049A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89050A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89051A3HeLaHUMAN3H-NECAN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide25.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89052A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89053A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89054A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89055A3HeLaHUMAN3H-NECAN-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide103Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89056A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89057A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide73.8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89058A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89059A3HeLaHUMAN3H-NECAN-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide18.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89060A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide31.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89061A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide103Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89062A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89063A3HeLaHUMAN3H-NECAN-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide160Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89064A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide18.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89065A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide142Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89066A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89067A3HeLaHUMAN3H-NECAN-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide135Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89068A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89069A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89070A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89071A3HeLaHUMAN3H-NECAN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide24.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89072A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide113Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89073A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89074A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89075A3HeLaHUMAN3H-NECAN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide23.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89076A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide41.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89077A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89078A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89079A3HeLaHUMAN3H-NECAN-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide110Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89080A1CHO cellsHUMAN3H-DPCPXISVY127100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89081A2AHeLaHUMAN3H-ZM241385ISVY127100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89082A2BHEK293 cellsHUMAN3H-DPCPXISVY127100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89083A3HeLaHUMAN3H-NECAISVY1275.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89084A1CHO cellsHUMAN3H-DPCPXISVY169100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89085A2AHeLaHUMAN3H-ZM241385ISVY169100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89086A2BHEK293 cellsHUMAN3H-DPCPXISVY169100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89087A3HeLaHUMAN3H-NECAISVY16911.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89088A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89089A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89090A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89091A3HeLaHUMAN3H-NECAN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide10.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89092A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide17.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89093A2AHeLaHUMAN3H-ZM241385N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide3345Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89094A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89095A3HeLaHUMAN3H-NECAN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide3.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89096A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide5.28Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89097A2AHeLaHUMAN3H-ZM241385N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide2541Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89098A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide1668Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89099A3HeLaHUMAN3H-NECAN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide14.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89100A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide9.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89101A2AHeLaHUMAN3H-ZM241385N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89102A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89103A3HeLaHUMAN3H-NECAN-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide59Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89104A1CHO cellsHUMAN3H-DPCPXN-(2,6-distyrylpyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89105A2AHeLaHUMAN3H-ZM241385N-(2,6-distyrylpyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89106A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-distyrylpyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89107A3HeLaHUMAN3H-NECAN-(2,6-distyrylpyrimidin-4-yl)acetamide15.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89108A1CHO cellsHUMAN3H-DPCPXN-(2,6-distyrylpyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89109A2AHeLaHUMAN3H-ZM241385N-(2,6-distyrylpyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89110A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-distyrylpyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89111A3HeLaHUMAN3H-NECAN-(2,6-distyrylpyrimidin-4-yl)propionamide46.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89112A1CHO cellsHUMAN3H-DPCPXN-(2,6-distyrylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89113A2AHeLaHUMAN3H-ZM241385N-(2,6-distyrylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89114A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-distyrylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89115A3HeLaHUMAN3H-NECAN-(2,6-distyrylpyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89116A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide40.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89117A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide8.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89118A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide12Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89119A3HeLaHUMAN3H-NECAN-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89120A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide15.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89121A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide6.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89122A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide20.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89123A3HeLaHUMAN3H-NECAN-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide6.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89124A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide7.8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89125A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide5.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89126A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide16.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89127A3HeLaHUMAN3H-NECAN-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide9.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89128A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89129A2AHeLaHUMAN3H-ZM241385N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide24.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89130A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89131A3HeLaHUMAN3H-NECAN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89132A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide32.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89133A2AHeLaHUMAN3H-ZM241385N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide114Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89134A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89135A3HeLaHUMAN3H-NECAN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide21.8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89136A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide33.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89137A2AHeLaHUMAN3H-ZM241385N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide153Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89138A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89139A3HeLaHUMAN3H-NECAN-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide23Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89140A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89141A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide74Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89142A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide302Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89143A3HeLaHUMAN3H-NECAN-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide10.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89144A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide132Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89145A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide82.8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89146A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide49Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89147A3HeLaHUMAN3H-NECAN-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide12.6Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89148A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide65.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89149A2AHeLaHUMAN3H-ZM241385N-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide544Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89150A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89151A3HeLaHUMAN3H-NECAN-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89152A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89153A2AHeLaHUMAN3H-ZM241385N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide39.8Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89154A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89155A3HeLaHUMAN3H-NECAN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide20.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89156A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide39.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89157A2AHeLaHUMAN3H-ZM241385N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide63.5Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89158A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide164.7Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89159A3HeLaHUMAN3H-NECAN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide64.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89160A1CHO cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide65.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89161A2AHeLaHUMAN3H-ZM241385N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89162A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89163A3HeLaHUMAN3H-NECAN-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89164A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89165A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89166A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89167A3HeLaHUMAN3H-NECAN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide12.2Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89168A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89169A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89170A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89171A3HeLaHUMAN3H-NECAN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide58.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89172A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89173A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89174A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89175A3HeLaHUMAN3H-NECAN-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide32.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89176A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89177A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89178A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89179A3HeLaHUMAN3H-NECAN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide15.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89180A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89181A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89182A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89183A3HeLaHUMAN3H-NECAN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide52.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89184A1CHO cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89185A2AHeLaHUMAN3H-ZM241385N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89186A2BHEK293 cellsHUMAN3H-DPCPXN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89187A3HeLaHUMAN3H-NECAN-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide56.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89188A1CHO cellsHUMAN3H-DPCPX4,6-diphenylpyrimidin-2-amine64Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89189A2ACHO cellsHUMAN3H-DPCPX4,6-diphenylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89190A2BCHO cellsHUMAN3H-DPCPX4,6-diphenylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89191A3HeLaHUMAN3H-NECA4,6-diphenylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89192A1CHO cellsHUMAN3H-DPCPX4,6-di-p-tolylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89193A2AHeLaHUMAN3H-ZM2413854,6-di-p-tolylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89194A2BHEK293 cellsHUMAN3H-DPCPX4,6-di-p-tolylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89195A3HeLaHUMAN3H-NECA4,6-di-p-tolylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89196A1CHO cellsHUMAN3H-DPCPX4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89197A2AHeLaHUMAN3H-ZM2413854,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89198A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89199A3HeLaHUMAN3H-NECA4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89200A1CHO cellsHUMAN3H-DPCPX4,6-bis(4-methoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89201A2AHeLaHUMAN3H-ZM2413854,6-bis(4-methoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89202A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(4-methoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89203A3HeLaHUMAN3H-NECA4,6-bis(4-methoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89204A1CHO cellsHUMAN3H-DPCPX4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89205A2AHeLaHUMAN3H-ZM2413854,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89206A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89207A3HeLaHUMAN3H-NECA4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89208A1CHO cellsHUMAN3H-DPCPX4,6-bis(acetylphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89209A2AHeLaHUMAN3H-ZM2413854,6-bis(acetylphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89210A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(acetylphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89211A3HeLaHUMAN3H-NECA4,6-bis(acetylphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89212A1CHO cellsHUMAN3H-DPCPX4,6-bis(4-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89213A2AHeLaHUMAN3H-ZM2413854,6-bis(4-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89214A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(4-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89215A3HeLaHUMAN3H-NECA4,6-bis(4-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89216A1CHO cellsHUMAN3H-DPCPX4,6-bis(4-chlorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89217A2AHeLaHUMAN3H-ZM2413854,6-bis(4-chlorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89218A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(4-chlorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89219A3HeLaHUMAN3H-NECA4,6-bis(4-chlorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89220A1CHO cellsHUMAN3H-DPCPX4,6-bis(2-methoxyphenyl)pyrimidin-2-amine76.1Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89221A2AHeLaHUMAN3H-ZM2413854,6-bis(2-methoxyphenyl)pyrimidin-2-amine369Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89222A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(2-methoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89223A3HeLaHUMAN3H-NECA4,6-bis(2-methoxyphenyl)pyrimidin-2-amine667Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89224A1CHO cellsHUMAN3H-DPCPX4,6-bis(2-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89225A2AHeLaHUMAN3H-ZM2413854,6-bis(2-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89226A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(2-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89227A3HeLaHUMAN3H-NECA4,6-bis(2-fluorophenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89228A1CHO cellsHUMAN3H-DPCPX4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89229A2AHeLaHUMAN3H-ZM2413854,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89230A2BHEK293 cellsHUMAN3H-DPCPX4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89231A3HeLaHUMAN3H-NECA4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89232A1CHO cellsHUMAN3H-DPCPX4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine538Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89233A2AHeLaHUMAN3H-ZM2413854,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89234A2BHEK293 cellsHUMAN3H-DPCPX4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89235A3HeLaHUMAN3H-NECA4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine5306Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89236A1CHO cellsHUMAN3H-DPCPX4,6-distyrylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89237A2AHeLaHUMAN3H-ZM2413854,6-distyrylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89238A2BHEK293 cellsHUMAN3H-DPCPX4,6-distyrylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89239A3HeLaHUMAN3H-NECA4,6-distyrylpyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89240A1CHO cellsHUMAN3H-DPCPX4,6-di(furan-2-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89241A2AHeLaHUMAN3H-ZM2413854,6-di(furan-2-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89242A2BHEK293 cellsHUMAN3H-DPCPX4,6-di(furan-2-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89243A3HeLaHUMAN3H-NECA4,6-di(furan-2-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89244A1CHO cellsHUMAN3H-DPCPX4,6-di(thiophen-2-yl)pyrimidin-2-amine174Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89245A2AHeLaHUMAN3H-ZM2413854,6-di(thiophen-2-yl)pyrimidin-2-amine361Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89246A2BHEK293 cellsHUMAN3H-DPCPX4,6-di(thiophen-2-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89247A3HeLaHUMAN3H-NECA4,6-di(thiophen-2-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89248A1CHO cellsHUMAN3H-DPCPX4,6-di(furan-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89249A2AHeLaHUMAN3H-ZM2413854,6-di(furan-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89250A2BHEK293 cellsHUMAN3H-DPCPX4,6-di(furan-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89251A3HeLaHUMAN3H-NECA4,6-di(furan-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89252A1CHO cellsHUMAN3H-DPCPX4,6-di(thiophen-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89253A2AHeLaHUMAN3H-ZM2413854,6-di(thiophen-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89254A2BHEK293 cellsHUMAN3H-DPCPX4,6-di(thiophen-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89255A3HeLaHUMAN3H-NECA4,6-di(thiophen-3-yl)pyrimidin-2-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89256A1CHO cellsHUMAN3H-DPCPX2,6-diphenylpyrimidin-4-amine48.3Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89257A2AHeLaHUMAN3H-ZM2413852,6-diphenylpyrimidin-4-amine459Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89258A2BHEK293 cellsHUMAN3H-DPCPX2,6-diphenylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89259A3HeLaHUMAN3H-NECA2,6-diphenylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89260A1CHO cellsHUMAN3H-DPCPX2,6-di-p-tolylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89261A2AHeLaHUMAN3H-ZM2413852,6-di-p-tolylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89262A2BHEK293 cellsHUMAN3H-DPCPX2,6-di-p-tolylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89263A3HeLaHUMAN3H-NECA2,6-di-p-tolylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89264A1CHO cellsHUMAN3H-DPCPX2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89265A2AHeLaHUMAN3H-ZM2413852,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89266A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89267A3HeLaHUMAN3H-NECA2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89268A1CHO cellsHUMAN3H-DPCPX2,6-bis(4-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89269A2AHeLaHUMAN3H-ZM2413852,6-bis(4-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89270A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(4-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89271A3HeLaHUMAN3H-NECA2,6-bis(4-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89272A1CHO cellsHUMAN3H-DPCPX2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89273A2AHeLaHUMAN3H-ZM2413852,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89274A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89275A3HeLaHUMAN3H-NECA2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine3600Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89276A1CHO cellsHUMAN3H-DPCPX2,6-bis(4-acetylphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89277A2AHeLaHUMAN3H-ZM2413852,6-bis(4-acetylphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89278A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(4-acetylphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89279A3HeLaHUMAN3H-NECA2,6-bis(4-acetylphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89280A1CHO cellsHUMAN3H-DPCPX2,6-bis(4-fluorophenyl)pyrimidin-4-amine110Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89281A2AHeLaHUMAN3H-ZM2413852,6-bis(4-fluorophenyl)pyrimidin-4-amine1304Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89282A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(4-fluorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89283A3HeLaHUMAN3H-NECA2,6-bis(4-fluorophenyl)pyrimidin-4-amine3107Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89284A1CHO cellsHUMAN3H-DPCPX2,6-bis(4-chlorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89285A2AHeLaHUMAN3H-ZM2413852,6-bis(4-chlorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89286A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(4-chlorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89287A3HeLaHUMAN3H-NECA2,6-bis(4-chlorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89288A1CHO cellsHUMAN3H-DPCPX2,6-bis(2-methoxyphenyl)pyrimidin-4-amine184Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89289A2AHeLaHUMAN3H-ZM2413852,6-bis(2-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89290A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(2-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89291A3HeLaHUMAN3H-NECA2,6-bis(2-methoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89292A1CHO cellsHUMAN3H-DPCPX2,6-bis(2-fluorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89293A2AHeLaHUMAN3H-ZM2413852,6-bis(2-fluorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89294A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(2-fluorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89295A3HeLaHUMAN3H-NECA2,6-bis(2-fluorophenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89296A1CHO cellsHUMAN3H-DPCPX2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89297A2AHeLaHUMAN3H-ZM2413852,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89298A2BHEK293 cellsHUMAN3H-DPCPX2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89299A3HeLaHUMAN3H-NECA2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89300A1CHO cellsHUMAN3H-DPCPX2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine7.9Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89301A2AHeLaHUMAN3H-ZM2413852,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89302A2BHEK293 cellsHUMAN3H-DPCPX2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89303A3HeLaHUMAN3H-NECA2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine299Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89304A1CHO cellsHUMAN3H-DPCPX2,6-distyrylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89305A2AHeLaHUMAN3H-ZM2413852,6-distyrylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89306A2BHEK293 cellsHUMAN3H-DPCPX2,6-distyrylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89307A3HeLaHUMAN3H-NECA2,6-distyrylpyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89308A1CHO cellsHUMAN3H-DPCPX2,6-di(furan-2-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89309A2AHeLaHUMAN3H-ZM2413852,6-di(furan-2-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89310A2BHEK293 cellsHUMAN3H-DPCPX2,6-di(furan-2-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89311A3HeLaHUMAN3H-NECA2,6-di(furan-2-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89312A1CHO cellsHUMAN3H-DPCPX2,6-di(thiophen-2-yl)pyrimidin-4-amine85.4Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89313A2AHeLaHUMAN3H-ZM2413852,6-di(thiophen-2-yl)pyrimidin-4-amine164Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89314A2BHEK293 cellsHUMAN3H-DPCPX2,6-di(thiophen-2-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89315A3HeLaHUMAN3H-NECA2,6-di(thiophen-2-yl)pyrimidin-4-amine831Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89316A1CHO cellsHUMAN3H-DPCPX2,6-di(furan-3-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89317A2AHeLaHUMAN3H-ZM2413852,6-di(furan-3-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89318A2BHEK293 cellsHUMAN3H-DPCPX2,6-di(furan-3-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89319A3HeLaHUMAN3H-NECA2,6-di(furan-3-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89320A1CHO cellsHUMAN3H-DPCPX2,6-di(thiophen-3-yl)pyrimidin-4-amine194Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89321A2AHeLaHUMAN3H-ZM2413852,6-di(thiophen-3-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89322A2BHEK293 cellsHUMAN3H-DPCPX2,6-di(thiophen-3-yl)pyrimidin-4-amine100Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
89323A3HeLaHUMAN3H-NECA2,6-di(thiophen-3-yl)pyrimidin-4-amine1178Yaziji V et al 2011Jan 15, 2025Jan 15, 2025
893245-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide16Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893255-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide437Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893265-HT6CLONEDHUMAN3H-LSD3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide148Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89327D2CLONEDHUMAN3H-RACLOPRIDE3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide631Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89328CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide9.3Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89329CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide245Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89330D2CLONEDHUMAN3H-RACLOPRIDE3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide345Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893315-HT6CLONEDHUMAN3H-LSD3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide830Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893325-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide582Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893335-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide35Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893345-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide53Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893355-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide1055Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893365-HT6CLONEDHUMAN3H-LSD3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide2518Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89337D2CLONEDHUMAN3H-RACLOPRIDE3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide2450Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89338CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide94Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89339CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide288Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89340D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide537Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893415-HT6CLONEDHUMAN3H-LSDN-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide1633Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893425-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide595Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893435-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide76Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893445-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide52Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893455-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide365Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893465-HT6CLONEDHUMAN3H-LSD3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide1039Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89347D2CLONEDHUMAN3H-RACLOPRIDE3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide268Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89348CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide1221Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89349CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide310Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89350D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide4346Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893515-HT6CLONEDHUMAN3H-LSDN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide3441Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893525-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide3842Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893535-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide87Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893545-HT7CLONEDHUMAN3H-5-CT3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide44Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893555-HT1ACLONEDHUMAN3H-8-OH-DPAT3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide802Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893565-HT6CLONEDHUMAN3H-LSD3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide2215Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89357D2CLONEDHUMAN3H-RACLOPRIDE3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide2766Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89358CORTICAL MEMBRANESPIG3H-PRAZOSIN3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide471Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89359CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide914Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89360D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide1959Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893615-HT6CLONEDHUMAN3H-LSDN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide2815Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893625-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide6631Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893635-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide108Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893645-HT7CLONEDHUMAN3H-5-CT3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide254Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893655-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide6064Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893665-HT6CLONEDHUMAN3H-LSD3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide2634Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89367D2CLONEDHUMAN3H-RACLOPRIDE3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide3460Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89368CORTICAL MEMBRANESPIG3H-PRAZOSIN3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide263Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89369CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide156Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89370D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide685Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893715-HT6CLONEDHUMAN3H-LSDN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide1621Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893725-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide2630Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893735-HT7CLONEDHUMAN3H-5-CTN-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide54Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893745-HT7CLONEDHUMAN3H-5-CT3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide32Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893755-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1836Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893765-HT6CLONEDHUMAN3H-LSD3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1074Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89377D2CLONEDHUMAN3H-RACLOPRIDE3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide393Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89378CORTICAL MEMBRANESPIG3H-PRAZOSIN3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide1369Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89379CORTICAL MEMBRANESPIG3H-PRAZOSINN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide5.9Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89380D2CLONEDHUMAN3H-RACLOPRIDEN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide321Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893815-HT6CLONEDHUMAN3H-LSDN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide640Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893825-HT1ACLONEDHUMAN3H-8-OH-DPATN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide160Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893835-HT7CLONEDHUMAN3H-5-CTN-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide6.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893845-HT7CLONEDHUMAN3H-5-CTN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide14.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893855-HT1ACLONEDHUMAN3H-8-OH-DPATN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide152Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893865-HT6CLONEDHUMAN3H-LSDN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide1336Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89387D2CLONEDHUMAN3H-RACLOPRIDEN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide419Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89388CORTICAL MEMBRANESPIG3H-PRAZOSINN-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide53Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89389CORTICAL MEMBRANESPIG3H-PRAZOSIN4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide26Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89390D2CLONEDHUMAN3H-RACLOPRIDE4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide375Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
893915-HT6CLONEDHUMAN3H-LSD4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide1706Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893925-HT1ACLONEDHUMAN3H-8-OH-DPAT4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide163Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893935-HT7CLONEDHUMAN3H-5-CT4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide25Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893945-HT7CLONEDHUMAN3H-5-CT4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide18.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893955-HT1ACLONEDHUMAN3H-8-OH-DPAT4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide105Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
893965-HT6CLONEDHUMAN3H-LSD4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide1623Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89397D2CLONEDHUMAN3H-RACLOPRIDE4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide260Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89398CORTICAL MEMBRANESPIG3H-PRAZOSIN4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide53Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89399CORTICAL MEMBRANESPIG3H-PRAZOSINN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide30Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89400D2CLONEDHUMAN3H-RACLOPRIDEN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide293Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894015-HT6CLONEDHUMAN3H-LSDN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide745Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894025-HT1ACLONEDHUMAN3H-8-OH-DPATN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide126Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894035-HT7CLONEDHUMAN3H-5-CTN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide8Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894045-HT7CLONEDHUMAN3H-5-CT4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide4.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894055-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide86Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894065-HT6CLONEDHUMAN3H-LSD4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide413Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89407D2CLONEDHUMAN3H-RACLOPRIDE4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide36Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89408CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide20Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89409CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-piperazinehexanamide4.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894105-HT7CLONEDHUMAN3H-5-CT4-(2-Biphenyl)-N-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-piperazinehexanamide259Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894115-HT7CLONEDHUMAN3H-5-CT4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide16Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894125-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide160Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894135-HT6CLONEDHUMAN3H-LSD4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide1724Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89414D2CLONEDHUMAN3H-RACLOPRIDE4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide136Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89415CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide7.4Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89416CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide12.3Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89417D2CLONEDHUMAN3H-RACLOPRIDE4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide64Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894185-HT6CLONEDHUMAN3H-LSD4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide1152Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894195-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide149Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894205-HT7CLONEDHUMAN3H-5-CT4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide9.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894215-HT7CLONEDHUMAN3H-5-CT4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide21Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894225-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide74Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894235-HT6CLONEDHUMAN3H-LSD4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide1506Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89424D2CLONEDHUMAN3H-RACLOPRIDE4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide75Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89425CORTICAL MEMBRANESPIG3H-PRAZOSIN4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide23Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89426CORTICAL MEMBRANESPIG3H-PRAZOSINN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide6.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89427D2CLONEDHUMAN3H-RACLOPRIDEN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide522Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894285-HT6CLONEDHUMAN3H-LSDN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide614Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894295-HT1ACLONEDHUMAN3H-8-OH-DPATN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide771Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894305-HT7CLONEDHUMAN3H-5-CTN-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide25.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894315-HT7CLONEDHUMAN3H-5-CTN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide27Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894325-HT1ACLONEDHUMAN3H-8-OH-DPATN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide2870Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894335-HT6CLONEDHUMAN3H-LSDN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide927Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89434D2CLONEDHUMAN3H-RACLOPRIDEN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide1385Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89435CORTICAL MEMBRANESPIG3H-PRAZOSINN-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide3.2Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89436CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide12.9Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89437D2CLONEDHUMAN3H-RACLOPRIDE(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide308Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894385-HT6CLONEDHUMAN3H-LSD(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide700Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894395-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide147Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894405-HT7CLONEDHUMAN3H-5-CT(S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide19Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894415-HT7CLONEDHUMAN3H-5-CT(R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide12Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894425-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide109Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894435-HT6CLONEDHUMAN3H-LSD(R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide843Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89444D2CLONEDHUMAN3H-RACLOPRIDE(R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide243Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89445CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide17.8Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89446CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide46.4Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89447D2CORTICAL MEMBRANESPIG3H-RACLOPRIDE(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide53Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894485-HT6CLONEDHUMAN3H-LSD(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide480Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894495-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide66Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894505-HT7CLONEDHUMAN3H-5-CT(S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide10Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894515-HT7CLONEDHUMAN3H-5-CT(R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide10.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894525-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide80Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894535-HT6CLONEDHUMAN3H-LSD(R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide561Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89454D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide116Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89455CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide36.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89456CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide36Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89457D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide295Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894585-HT6CLONEDHUMAN3H-LSD(R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide721Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894595-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide134Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894605-HT7CLONEDHUMAN3H-5-CT(R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide11.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894615-HT7CLONEDHUMAN3H-5-CT(S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide15.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894625-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide103Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894635-HT6CLONEDHUMAN3H-LSD(S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide652Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89464D2CLONEDHUMAN3H-RACLOPRIDE(S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide177Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89465CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide22.1Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89466CORTICAL MEMBRANESPIG3H-PRAZOSIN(R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide11.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89467D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide178Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
894685-HT6CLONEDHUMAN3H-LSD(R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide434Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894695-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide101Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894705-HT7CLONEDHUMAN3H-5-CT(R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide14Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894715-HT7CLONEDHUMAN3H-5-CT(S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide36.5Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894725-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide202Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
894735-HT6CLONEDHUMAN3H-LSD(S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide395Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89474D2CLONEDHUMAN3H-RACLOPRIDE(S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide243Lacivita E et al 2016Jan 15, 2025Jan 28, 2025
89475CORTICAL MEMBRANESPIG3H-PRAZOSIN(S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide42.6Lacivita E et al 2016Jan 15, 2025Jan 15, 2025
89476M1CLONEDHUMAN3H-NMS1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89477M2CLONEDHUMAN3H-NMS1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89478M3CLONEDHUMAN3H-NMS1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89479M3CLONEDHUMAN3H-NMS2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate4700Fish I et al 2017Jan 15, 2025Jan 15, 2025
89480M2CLONEDHUMAN3H-NMS2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate5700Fish I et al 2017Jan 15, 2025Jan 15, 2025
89481M1CLONEDHUMAN3H-NMS2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate4900Fish I et al 2017Jan 15, 2025Jan 15, 2025
89482M1CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89483M2CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89484M3CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89485M3CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide620Fish I et al 2017Jan 15, 2025Jan 15, 2025
89486M2CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide630Fish I et al 2017Jan 15, 2025Jan 15, 2025
89487M1CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide330Fish I et al 2017Jan 15, 2025Jan 15, 2025
89488M1CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89489M2CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89490M3CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89491M3CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89492M2CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89493M1CLONEDHUMAN3H-NMS3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89494M1CLONEDHUMAN3H-NMS1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate7300Fish I et al 2017Jan 15, 2025Jan 15, 2025
89495M2CLONEDHUMAN3H-NMS1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89496M3CLONEDHUMAN3H-NMS1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate8700Fish I et al 2017Jan 15, 2025Jan 15, 2025
89497M3CLONEDHUMAN3H-NMS5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89498M2CLONEDHUMAN3H-NMS5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89499M1CLONEDHUMAN3H-NMS5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89500M1CLONEDHUMAN3H-NMS8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89501M2CLONEDHUMAN3H-NMS8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate6300Fish I et al 2017Jan 15, 2025Jan 15, 2025
89502M3CLONEDHUMAN3H-NMS8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate5800Fish I et al 2017Jan 15, 2025Jan 15, 2025
89503M3CLONEDHUMAN3H-NMS8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide2000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89504M2CLONEDHUMAN3H-NMS8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide930Fish I et al 2017Jan 15, 2025Jan 15, 2025
89505M1CLONEDHUMAN3H-NMS8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide1000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89506M1CLONEDHUMAN3H-NMS8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide2900Fish I et al 2017Jan 15, 2025Jan 15, 2025
89507M2CLONEDHUMAN3H-NMS8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide4200Fish I et al 2017Jan 15, 2025Jan 15, 2025
89508M3CLONEDHUMAN3H-NMS8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89509M3CLONEDHUMAN3H-NMS1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate3900Fish I et al 2017Jan 15, 2025Jan 15, 2025
89510M2CLONEDHUMAN3H-NMS1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate1300Fish I et al 2017Jan 15, 2025Jan 15, 2025
89511M1CLONEDHUMAN3H-NMS1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate1800Fish I et al 2017Jan 15, 2025Jan 15, 2025
89512M1CLONEDHUMAN3H-NMS5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide2500Fish I et al 2017Jan 15, 2025Jan 15, 2025
89513M2CLONEDHUMAN3H-NMS5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide4400Fish I et al 2017Jan 15, 2025Jan 15, 2025
89514M3CLONEDHUMAN3H-NMS5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide4000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89515M3CLONEDHUMAN3H-NMS1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89516M2CLONEDHUMAN3H-NMS1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89517M1CLONEDHUMAN3H-NMS1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89518M1CLONEDHUMAN3H-NMS8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89519M2CLONEDHUMAN3H-NMS8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1200Fish I et al 2017Jan 15, 2025Jan 15, 2025
89520M3CLONEDHUMAN3H-NMS8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine830Fish I et al 2017Jan 15, 2025Jan 15, 2025
89521M3CLONEDHUMAN3H-NMS7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89522M2CLONEDHUMAN3H-NMS7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89523M1CLONEDHUMAN3H-NMS7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89524M1CLONEDHUMAN3H-NMS2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate23Fish I et al 2017Jan 15, 2025Jan 15, 2025
89525M2CLONEDHUMAN3H-NMS2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate140Fish I et al 2017Jan 15, 2025Jan 15, 2025
89526M3CLONEDHUMAN3H-NMS2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate41Fish I et al 2017Jan 15, 2025Jan 15, 2025
89527M3CLONEDHUMAN3H-NMS3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate140Fish I et al 2017Jan 15, 2025Jan 15, 2025
89528M2CLONEDHUMAN3H-NMS3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate230Fish I et al 2017Jan 15, 2025Jan 15, 2025
89529M1CLONEDHUMAN3H-NMS3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate63Fish I et al 2017Jan 15, 2025Jan 15, 2025
89530M1CLONEDHUMAN3H-NMSN,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate380Fish I et al 2017Jan 15, 2025Jan 15, 2025
89531M2CLONEDHUMAN3H-NMSN,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate790Fish I et al 2017Jan 15, 2025Jan 15, 2025
89532M3CLONEDHUMAN3H-NMSN,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate690Fish I et al 2017Jan 15, 2025Jan 15, 2025
89533M3CLONEDHUMAN3H-NMSiperoxo550Fish I et al 2017Jan 15, 2025Jan 15, 2025
89534M2CLONEDHUMAN3H-NMSiperoxo4.9Fish I et al 2017Jan 15, 2025Jan 15, 2025
89535M1CLONEDHUMAN3H-NMSiperoxo350Fish I et al 2017Jan 15, 2025Jan 15, 2025
89536M1CLONEDHUMAN3H-NMSAcetylcholine5.8Fish I et al 2017Jan 15, 2025Jan 15, 2025
89537M2CLONEDHUMAN3H-NMSAcetylcholine0.39Fish I et al 2017Jan 15, 2025Jan 15, 2025
89538M3CLONEDHUMAN3H-NMSAcetylcholine4.7Fish I et al 2017Jan 15, 2025Jan 15, 2025
89539M3CLONEDHUMAN3H-NMSCARBACHOL51Fish I et al 2017Jan 15, 2025Jan 15, 2025
89540M2CLONEDHUMAN3H-NMSCARBACHOL4.1Fish I et al 2017Jan 15, 2025Jan 15, 2025
89541M1CLONEDHUMAN3H-NMSCARBACHOL63Fish I et al 2017Jan 15, 2025Jan 15, 2025
89542M1CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N-methylethan-1-amine740Fish I et al 2017Jan 15, 2025Jan 15, 2025
89543M2CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N-methylethan-1-amine1000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89544M3CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N-methylethan-1-amine780Fish I et al 2017Jan 15, 2025Jan 15, 2025
89545M3CLONEDHUMAN3H-NMS2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89546M2CLONEDHUMAN3H-NMS2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89547M1CLONEDHUMAN3H-NMS2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89548M1CLONEDHUMAN3H-NMS2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate7100Fish I et al 2017Jan 15, 2025Jan 15, 2025
89549M2CLONEDHUMAN3H-NMS2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate980Fish I et al 2017Jan 15, 2025Jan 15, 2025
89550M3CLONEDHUMAN3H-NMS2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89551M3CLONEDHUMAN3H-NMS2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89552M2CLONEDHUMAN3H-NMS2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89553M1CLONEDHUMAN3H-NMS2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89554M1CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate170Fish I et al 2017Jan 15, 2025Jan 15, 2025
89555M2CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate2400Fish I et al 2017Jan 15, 2025Jan 15, 2025
89556M3CLONEDHUMAN3H-NMS2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate210Fish I et al 2017Jan 15, 2025Jan 15, 2025
89557M3CLONEDHUMAN3H-NMS2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89558M2CLONEDHUMAN3H-NMS2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89559M1CLONEDHUMAN3H-NMS2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89560M1CLONEDHUMAN3H-NMS2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate4500Fish I et al 2017Jan 15, 2025Jan 15, 2025
89561M2CLONEDHUMAN3H-NMS2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate4800Fish I et al 2017Jan 15, 2025Jan 15, 2025
89562M3CLONEDHUMAN3H-NMS2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate5800Fish I et al 2017Jan 15, 2025Jan 15, 2025
89563M3CLONEDHUMAN3H-NMSN,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89564M2CLONEDHUMAN3H-NMSN,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate9200Fish I et al 2017Jan 15, 2025Jan 15, 2025
89565M1CLONEDHUMAN3H-NMSN,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate7800Fish I et al 2017Jan 15, 2025Jan 15, 2025
89566M1CLONEDHUMAN3H-NMS2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate6400Fish I et al 2017Jan 15, 2025Jan 15, 2025
89567M2CLONEDHUMAN3H-NMS2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89568M3CLONEDHUMAN3H-NMS2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate6300Fish I et al 2017Jan 15, 2025Jan 15, 2025
89569M3CLONEDHUMAN3H-NMS3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89570M2CLONEDHUMAN3H-NMS3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89571M1CLONEDHUMAN3H-NMS3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89572M1CLONEDHUMAN3H-NMS2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole4200Fish I et al 2017Jan 15, 2025Jan 15, 2025
89573M2CLONEDHUMAN3H-NMS2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole6000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89574M3CLONEDHUMAN3H-NMS2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole4100Fish I et al 2017Jan 15, 2025Jan 15, 2025
89575M1CLONEDHUMAN3H-NMS(3R)-3-(imidazol-1-ylmethyl)piperidine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89576M2CLONEDHUMAN3H-NMS(3R)-3-(imidazol-1-ylmethyl)piperidine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89577M3CLONEDHUMAN3H-NMS(3R)-3-(imidazol-1-ylmethyl)piperidine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89578M3CLONEDHUMAN3H-NMS2-(1,3-benzodioxol-5-yl)guanidine9700Fish I et al 2017Jan 15, 2025Jan 15, 2025
89579M2CLONEDHUMAN3H-NMS2-(1,3-benzodioxol-5-yl)guanidine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89580M1CLONEDHUMAN3H-NMS2-(1,3-benzodioxol-5-yl)guanidine8300Fish I et al 2017Jan 15, 2025Jan 15, 2025
89581M1CLONEDHUMAN3H-NMS3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89582M2CLONEDHUMAN3H-NMS3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89583M3CLONEDHUMAN3H-NMS3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine9500Fish I et al 2017Jan 15, 2025Jan 15, 2025
89584M3CLONEDHUMAN3H-NMS2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89585M2CLONEDHUMAN3H-NMS2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89586M1CLONEDHUMAN3H-NMS2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89587M1CLONEDHUMAN3H-NMS2-(3-methoxyphenyl)ethanimidamide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89588M2CLONEDHUMAN3H-NMS2-(3-methoxyphenyl)ethanimidamide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89589M3CLONEDHUMAN3H-NMS2-(3-methoxyphenyl)ethanimidamide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89590M3CLONEDHUMAN3H-NMS2-(3-methoxyphenoxy)ethanimidamide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89591M2CLONEDHUMAN3H-NMS2-(3-methoxyphenoxy)ethanimidamide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89592M1CLONEDHUMAN3H-NMS2-(3-methoxyphenoxy)ethanimidamide>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89593M1CLONEDHUMAN3H-NMS(2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89594M2CLONEDHUMAN3H-NMS(2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89595M3CLONEDHUMAN3H-NMS(2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89596M3CLONEDHUMAN3H-NMS4-[(3R)-piperidin-3-yl]oxypyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89597M2CLONEDHUMAN3H-NMS4-[(3R)-piperidin-3-yl]oxypyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89598M1CLONEDHUMAN3H-NMS4-[(3R)-piperidin-3-yl]oxypyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89599M1CLONEDHUMAN3H-NMS1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium6100Fish I et al 2017Jan 15, 2025Jan 15, 2025
89600M2CLONEDHUMAN3H-NMS1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89601M3CLONEDHUMAN3H-NMS1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89602M3CLONEDHUMAN3H-NMS3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89603M2CLONEDHUMAN3H-NMS3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89604M1CLONEDHUMAN3H-NMS3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89605M1CLONEDHUMAN3H-NMS3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89606M2CLONEDHUMAN3H-NMS3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
89607M3CLONEDHUMAN3H-NMS3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine>10000Fish I et al 2017Jan 15, 2025Jan 15, 2025
896085-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone0.47863Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89609CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89610D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89611D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89612Alpha1ACORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone177.828Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
896135-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone2.5704Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896145-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1.86209Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89615CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89616D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89617D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89618CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone54.9541Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896195-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1.25893Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896205-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone0.562341Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89621D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89622D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89623CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone23.4423Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896245-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone0.616595Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896255-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0616595Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89626CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone512.861Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89627D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89628D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89629CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone165.959Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896305-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone0.0645654Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896315-HT1ACLONEDHUMAN3H-8-OH-DPAT(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone0.0147911Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89632D2CLONEDHUMAN3H-Methylspiperone(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89633D2CLONEDHUMAN3H-Methylspiperone(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89634CORTEXRAT3H-PRAZOSIN(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone128.825Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896355-HT1ACLONEDHUMAN3H-8-OH-DPAT(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone0.0338844Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896365-HT1ACLONEDHUMAN3H-8-OH-DPATNLX-1012.18776Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89637CORTEXRAT3H-PRAZOSINNLX-1011000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89638D2CLONEDHUMAN3H-MethylspiperoneNLX-1011000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
896395-HT1ACLONEDHUMAN3H-8-OH-DPAT8-OH-DPAT0.812831Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896405-HT1ACLONEDHUMAN3H-8-OH-DPATBUSPIRONE5.01187Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896415-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1.51356Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89642CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89643D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89644D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89645CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896465-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone389.045Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896475-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone0.524807Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89648CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89649D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
896505-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone35.4813Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896515-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone208.93Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89652CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89653D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89654D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89655CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896565-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone199.526Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896575-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone3.80189Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89658CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89659D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89660D2CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89661CORTEXRAT3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896625-HT1ACLONEDHUMAN3H-8-OH-DPAT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone13.8038Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896635-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89664M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89665H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89666H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89667M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896685-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896695-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89670M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89671H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89672H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89673M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896745-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896755-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89676M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89677H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89678H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89679M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896805-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896815-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89682M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89683H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89684H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89685M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896865-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896875-HT2ACLONEDHUMAN3H-KETANSERIN(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89688M1CLONEDHUMAN3H-NMS(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89689H1CLONEDHUMAN3H-PYRILAMINE(3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89690H1CLONEDHUMAN3H-PYRILAMINE(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89691M1CLONEDHUMAN3H-NMS(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896925-HT2ACLONEDHUMAN3H-KETANSERIN(3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896935-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89694M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89695H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89696H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89697M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896985-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
896995-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89700M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89701H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89702H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89703M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897045-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897055-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89706M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89707H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89708H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89709M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897105-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897115-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89712M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89713H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89714H1CLONEDHUMAN3H-PYRILAMINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89715M1CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897165-HT2ACLONEDHUMAN3H-KETANSERIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89717A2ACLONEDHUMAN3H-NECA(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89718Alpha1ACLONEDHUMAN3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone165.959Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89719Alpha1BCLONEDHUMAN3H-PRAZOSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89720Beta 1CLONEDHUMAN125I-Pindolol(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89721Beta 2CLONEDHUMAN3H-CGP12177(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89722CB1CLONEDHUMAN3H-CP55940(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89723CB2CLONEDHUMAN3H-CP55940(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89724CCK1CLONEDHUMAN125I-BH-CCK-8(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89725D1CLONEDHUMAN3H-SCH23390(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89726D3CLONEDHUMAN3H-Methylspiperone(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89727ETACLONEDHUMAN125I-ENDOTHELIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897285-HT1DCLONEDHUMAN125I-aminopotentidine(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89729H3CLONEDHUMAN3H-Alpha-methylhistamine(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89730H4CLONEDHUMAN3H-Histamine(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89731M2CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89732M3CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89733M4CLONEDHUMAN3H-NMS(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89734DORCLONEDHUMAN3H-DADLE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89735KORCLONEDHUMAN3H-U69593(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89736MORCLONEDHUMAN3H-DAMGO(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89737V1ACLONEDHUMAN3H-VASOPRESSIN(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897385-HT1BCLONEDHUMAN3H-5-CT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897395-HT1DCLONEDHUMAN3H-5-CT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897405-HT2BCLONEDHUMAN3H-LSD(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897415-HT2CCLONEDHUMAN3H-MESULERGINE(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897425-HT6CLONEDHUMAN3H-LSD(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
897435-HT6CLONEDHUMAN3H-5-CT(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone1000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89744DATCLONEDHUMAN3H-WIN 35,428(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89745NETCLONEDHUMAN3H-Nisoxene(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89746SERTCLONEDHUMAN3H-CITALOPRAM(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89747BZPCORTEXRATFNZ(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 29, 2025
89748NMDACORTEXRAT3H-MK-801(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025