88749 H1 CLONED HUMAN 3H-PYRILAMINE 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 1009 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88750 M1 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88751 M2 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88752 M3 CLONED HUMAN 3H-QNB 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol >10000 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88753 DAT CLONED HUMAN 3H-WIN 35,428 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 354 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88754 NET CLONED HUMAN 3H-Nisoxetine 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 462 Sampson D et al 2014 Jan 15, 2025 Jan 15, 2025
88755 SERT CLONED HUMAN 3H-CITALOPRAM 3-(4-chlorophenyl)-8-(3-((2-fluorophenyl)thio)propyl)-8-azabicyclo[3.2.1]octan-3-ol 102 Sampson D et al 2014 Jan 15, 2025 Jan 28, 2025
88756 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-diphenylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88757 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-diphenylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88758 A2B CHO cells HUMAN 3H-DPCPX N-(4,6-diphenylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88759 A3 HeLa HUMAN 3H-NECA N-(4,6-diphenylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88760 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-diphenylpyrimidin-2-yl)propionamide 31.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88761 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-diphenylpyrimidin-2-yl)propionamide 554 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88762 A2A HEK293 cells HUMAN 3H-DPCPX N-(4,6-diphenylpyrimidin-2-yl)propionamide 42.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88763 A3 HeLa HUMAN 3H-NECA N-(4,6-diphenylpyrimidin-2-yl)propionamide 531 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88764 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-diphenylpyrimidin-2-yl)butyramide 10.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88765 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-diphenylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88766 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-diphenylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88767 A3 HeLa HUMAN 3H-NECA N-(4,6-diphenylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88768 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-dip-tolylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88769 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-dip-tolylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88770 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-dip-tolylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88771 A3 HeLa HUMAN 3H-NECA N-(4,6-dip-tolylpyrimidin-2-yl)acetamide 47.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88772 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di-tolylpyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88773 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di-tolylpyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88774 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di-tolylpyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88775 A3 HeLa HUMAN 3H-NECA N-(4,6-di-tolylpyrimidin-2-yl)propionamide 157 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88776 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-dip-tolylpyrimidin-2-yl)butyramide 3760 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88777 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-dip-tolylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88778 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-dip-tolylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88779 A3 HeLa HUMAN 3H-NECA N-(4,6-dip-tolylpyrimidin-2-yl)butyramide 131 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88780 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88781 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88782 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88783 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88784 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88785 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88786 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88787 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88788 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88789 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88790 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88791 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88792 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88793 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88794 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88795 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88796 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88797 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88798 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88799 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88800 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88801 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88802 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88803 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88804 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88805 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88806 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88807 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88808 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide 505 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88809 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide 183 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88810 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide 374 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88811 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)propionamide 4435 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88812 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88813 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88814 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88815 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-(methylthio)phenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88816 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88817 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88818 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88819 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88820 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88821 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88822 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88823 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88824 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88825 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88826 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88827 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-acetylphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88828 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88829 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88830 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88831 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88832 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88833 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88834 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88835 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88836 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88837 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88838 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88839 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88840 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88841 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88842 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88843 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88844 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88845 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88846 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88847 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88848 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88849 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88850 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88851 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(4-chlorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88852 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88853 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88854 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88855 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88856 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide 48.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88857 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide 424 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88858 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide 307 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88859 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)propionamide 279 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88860 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 23.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88861 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 647 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88862 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88863 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-methoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88864 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88865 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88866 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88867 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88868 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88869 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88870 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88871 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88872 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88873 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88874 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88875 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2-fluorophenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88876 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88877 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88878 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88879 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88880 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88881 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88882 A2B HeLa HUMAN 3H-DPCPX N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88883 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88884 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88885 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88886 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88887 A3 HeLa HUMAN 3H-NECA N-(4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88888 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88889 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88890 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88891 A3 HeLa HUMAN 3H-NECA N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)acetamide 101 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88892 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide 535 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88893 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88894 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88895 A3 HeLa HUMAN 3H-NECA N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)propionamide 127 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88896 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide 678 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88897 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88898 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88899 A3 HeLa HUMAN 3H-NECA N-(4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-yl)butyramide 751 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88900 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-distyrylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88901 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-distyrylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88902 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-distyrylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88903 A3 HeLa HUMAN 3H-NECA N-(4,6-distyrylpyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88904 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-distyrylpyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88905 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-distyrylpyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88906 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-distyrylpyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88907 A3 HeLa HUMAN 3H-NECA N-(4,6-distyrylpyrimidin-2-yl)propionamide 142 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88908 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-distyrylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88909 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-distyrylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88910 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-distyrylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88911 A3 HeLa HUMAN 3H-NECA N-(4,6-distyrylpyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88912 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88913 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88914 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88915 A3 HeLa HUMAN 3H-NECA N-(4,6-di(furan-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88916 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88917 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88918 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88919 A3 HeLa HUMAN 3H-NECA N-(4,6-di(furan-2-yl)pyrimidin-2-yl)propionamide 1903 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88920 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88921 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88922 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88923 A3 HeLa HUMAN 3H-NECA N-(4,6-di(furan-2-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88924 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88925 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88926 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88927 A3 HeLa HUMAN 3H-NECA N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88928 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88929 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88930 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88931 A3 HeLa HUMAN 3H-NECA N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88932 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide 255 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88933 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide 201 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88934 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88935 A3 HeLa HUMAN 3H-NECA N-(4,6-di(thiophen-2-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88936 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88937 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88938 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88939 A3 HeLa HUMAN 3H-NECA N-(4,6-di(furan-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88940 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88941 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88942 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88943 A3 HeLa HUMAN 3H-NECA N-(4,6-di(furan-3-yl)pyrimidin-2-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88944 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88945 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88946 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88947 A3 HeLa HUMAN 3H-NECA N-(4,6-di(furan-3-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88948 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88949 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88950 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88951 A3 HeLa HUMAN 3H-NECA N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88952 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide 367 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88953 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide 1893 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88954 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide 3250 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88955 A3 HeLa HUMAN 3H-NECA N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)propionamide 1279 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88956 A1 CHO cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide 85.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88957 A2A HeLa HUMAN 3H-ZM241385 N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide 4568 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88958 A2B HEK293 cells HUMAN 3H-DPCPX N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88959 A3 HeLa HUMAN 3H-NECA N-(4,6-di(thiophen-3-yl)pyrimidin-2-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88960 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-diphenylpyrimidin-4-yl)acetamide 31.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88961 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-diphenylpyrimidin-4-yl)acetamide 255.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88962 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-diphenylpyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88963 A3 HeLa HUMAN 3H-NECA N-(2,6-diphenylpyrimidin-4-yl)acetamide 12.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88964 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-diphenylpyrimidin-4-yl)propionamide 22.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88965 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-diphenylpyrimidin-4-yl)propionamide 84.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88966 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-diphenylpyrimidin-4-yl)propionamide 76.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88967 A3 HeLa HUMAN 3H-NECA N-(2,6-diphenylpyrimidin-4-yl)propionamide 45.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88968 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-diphenylpyrimidin-4-yl)butyramide 19.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88969 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-diphenylpyrimidin-4-yl)butyramide 103 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88970 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-diphenylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88971 A3 HeLa HUMAN 3H-NECA N-(2,6-diphenylpyrimidin-4-yl)butyramide 171 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88972 A1 CHO cells HUMAN 3H-DPCPX ISVY133 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88973 A2A HeLa HUMAN 3H-ZM241385 ISVY133 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88974 A2B HEK293 cells HUMAN 3H-DPCPX ISVY133 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88975 A3 HeLa HUMAN 3H-NECA ISVY133 4.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88976 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di-p-tolylpyrimidin-4-yl)propionamide 36.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88977 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di-p-tolylpyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88978 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di-p-tolylpyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88979 A3 HeLa HUMAN 3H-NECA N-(2,6-di-p-tolylpyrimidin-4-yl)propionamide 18.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88980 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di-p-tolylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88981 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di-p-tolylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88982 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di-p-tolylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88983 A3 HeLa HUMAN 3H-NECA N-(2,6-di-p-tolylpyrimidin-4-yl)butyramide 59 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88984 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88985 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88986 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88987 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)acetamide 126 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88988 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88989 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88990 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88991 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88992 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88993 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88994 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88995 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88996 A1 CHO cells HUMAN 3H-DPCPX ISVY130 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88997 A2A HeLa HUMAN 3H-ZM241385 ISVY130 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88998 A2B HEK293 cells HUMAN 3H-DPCPX ISVY130 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
88999 A3 HeLa HUMAN 3H-NECA ISVY130 3.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89000 A1 CHO cells HUMAN 3H-DPCPX ISVY074 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89001 A2A HeLa HUMAN 3H-ZM241385 ISVY074 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89002 A2B HEK293 cells HUMAN 3H-DPCPX ISVY074 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89003 A3 HeLa HUMAN 3H-NECA ISVY074 3.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89004 A1 CHO cells HUMAN 3H-DPCPX ISVY071 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89005 A2A HeLa HUMAN 3H-ZM241385 ISVY071 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89006 A2B HEK293 cells HUMAN 3H-DPCPX ISVY071 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89007 A3 HeLa HUMAN 3H-NECA ISVY071 11 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89008 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89009 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89010 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89011 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)acetamide 71.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89012 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89013 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89014 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89015 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)propionamide 43.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89016 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89017 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89018 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89019 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-(methylthio)phenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89020 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89021 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89022 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89023 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)acetamide 25.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89024 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89025 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89026 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89027 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)propionamide 43.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89028 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89029 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89030 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89031 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-acetylphenyl)pyrimidin-4-yl)butyramide 133 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89032 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89033 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide 1334 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89034 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89035 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)acetamide 16.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89036 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide 83.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89037 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide 429 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89038 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89039 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)propionamide 12.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89040 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide 82.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89041 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide 1829 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89042 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89043 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-fluorophenyl)pyrimidin-4-yl)butyramide 34.8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89044 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89045 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89046 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89047 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)acetamide 63.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89048 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89049 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89050 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89051 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)propionamide 25.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89052 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89053 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89054 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89055 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-chlorophenyl)pyrimidin-4-yl)butyramide 103 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89056 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89057 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide 73.8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89058 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89059 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2-methoxyphenyl)p ]yrimidin-4-yl)acetamide 18.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89060 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide 31.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89061 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide 103 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89062 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89063 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)propionamide 160 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89064 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide 18.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89065 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide 142 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89066 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89067 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2-methoxyphenyl)pyrimidin-4-yl)butyramide 135 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89068 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89069 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89070 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89071 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)acetamide 24.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89072 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide 113 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89073 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89074 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89075 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)propionamide 23.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89076 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide 41.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89077 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89078 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89079 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2-fluorophenyl)pyrimidin-4-yl)butyramide 110 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89080 A1 CHO cells HUMAN 3H-DPCPX ISVY127 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89081 A2A HeLa HUMAN 3H-ZM241385 ISVY127 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89082 A2B HEK293 cells HUMAN 3H-DPCPX ISVY127 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89083 A3 HeLa HUMAN 3H-NECA ISVY127 5.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89084 A1 CHO cells HUMAN 3H-DPCPX ISVY169 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89085 A2A HeLa HUMAN 3H-ZM241385 ISVY169 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89086 A2B HEK293 cells HUMAN 3H-DPCPX ISVY169 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89087 A3 HeLa HUMAN 3H-NECA ISVY169 11.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89088 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89089 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89090 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89091 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)butyramide 10.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89092 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 17.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89093 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 3345 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89094 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89095 A3 HeLa HUMAN 3H-NECA N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)acetamide 3.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89096 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide 5.28 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89097 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide 2541 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89098 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide 1668 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89099 A3 HeLa HUMAN 3H-NECA N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)propionamide 14.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89100 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide 9.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89101 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89102 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89103 A3 HeLa HUMAN 3H-NECA N-(2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-yl)butyramide 59 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89104 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-distyrylpyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89105 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-distyrylpyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89106 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-distyrylpyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89107 A3 HeLa HUMAN 3H-NECA N-(2,6-distyrylpyrimidin-4-yl)acetamide 15.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89108 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-distyrylpyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89109 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-distyrylpyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89110 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-distyrylpyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89111 A3 HeLa HUMAN 3H-NECA N-(2,6-distyrylpyrimidin-4-yl)propionamide 46.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89112 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-distyrylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89113 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-distyrylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89114 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-distyrylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89115 A3 HeLa HUMAN 3H-NECA N-(2,6-distyrylpyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89116 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 40.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89117 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 8.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89118 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 12 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89119 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-2-yl)pyrimidin-4-yl)acetamide 3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89120 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide 15.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89121 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide 6.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89122 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide 20.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89123 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-2-yl)pyrimidin-4-yl)propionamide 6.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89124 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide 7.8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89125 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide 5.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89126 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide 16.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89127 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-2-yl)pyrimidin-4-yl)butyramide 9.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89128 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89129 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide 24.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89130 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89131 A3 HeLa HUMAN 3H-NECA N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)acetamide 8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89132 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide 32.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89133 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide 114 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89134 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89135 A3 HeLa HUMAN 3H-NECA N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)propionamide 21.8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89136 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide 33.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89137 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide 153 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89138 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89139 A3 HeLa HUMAN 3H-NECA N-(2,6-di(thiophen-2-yl)pyrimidin-4-yl)butyramide 23 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89140 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89141 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide 74 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89142 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide 302 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89143 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-3-yl)pyrimidin-4-yl)acetamide 10.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89144 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide 132 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89145 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide 82.8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89146 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide 49 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89147 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-3-yl)pyrimidin-4-yl)propionamide 12.6 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89148 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide 65.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89149 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide 544 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89150 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89151 A3 HeLa HUMAN 3H-NECA N-(2,6-di(furan-3-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89152 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89153 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide 39.8 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89154 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89155 A3 HeLa HUMAN 3H-NECA N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)acetamide 20.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89156 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide 39.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89157 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide 63.5 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89158 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide 164.7 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89159 A3 HeLa HUMAN 3H-NECA N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)propionamide 64.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89160 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide 65.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89161 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89162 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89163 A3 HeLa HUMAN 3H-NECA N-(2,6-di(thiophen-3-yl)pyrimidin-4-yl)butyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89164 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89165 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89166 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89167 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)isobutyramide 12.2 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89168 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89169 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89170 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89171 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 58.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89172 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89173 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89174 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89175 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(4-methoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 32.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89176 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89177 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89178 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89179 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)isobutyramide 15.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89180 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89181 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89182 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89183 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)-2-ethylbutanamide 52.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89184 A1 CHO cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89185 A2A HeLa HUMAN 3H-ZM241385 N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89186 A2B HEK293 cells HUMAN 3H-DPCPX N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89187 A3 HeLa HUMAN 3H-NECA N-(2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-yl)cyclohexanecarboxamide 56.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89188 A1 CHO cells HUMAN 3H-DPCPX 4,6-diphenylpyrimidin-2-amine 64 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89189 A2A CHO cells HUMAN 3H-DPCPX 4,6-diphenylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89190 A2B CHO cells HUMAN 3H-DPCPX 4,6-diphenylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89191 A3 HeLa HUMAN 3H-NECA 4,6-diphenylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89192 A1 CHO cells HUMAN 3H-DPCPX 4,6-di-p-tolylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89193 A2A HeLa HUMAN 3H-ZM241385 4,6-di-p-tolylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89194 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-di-p-tolylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89195 A3 HeLa HUMAN 3H-NECA 4,6-di-p-tolylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89196 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89197 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89198 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89199 A3 HeLa HUMAN 3H-NECA 4,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89200 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(4-methoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89201 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(4-methoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89202 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(4-methoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89203 A3 HeLa HUMAN 3H-NECA 4,6-bis(4-methoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89204 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89205 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89206 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89207 A3 HeLa HUMAN 3H-NECA 4,6-bis(4-(methylthio)phenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89208 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(acetylphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89209 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(acetylphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89210 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(acetylphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89211 A3 HeLa HUMAN 3H-NECA 4,6-bis(acetylphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89212 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(4-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89213 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(4-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89214 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(4-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89215 A3 HeLa HUMAN 3H-NECA 4,6-bis(4-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89216 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(4-chlorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89217 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(4-chlorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89218 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(4-chlorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89219 A3 HeLa HUMAN 3H-NECA 4,6-bis(4-chlorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89220 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(2-methoxyphenyl)pyrimidin-2-amine 76.1 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89221 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(2-methoxyphenyl)pyrimidin-2-amine 369 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89222 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(2-methoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89223 A3 HeLa HUMAN 3H-NECA 4,6-bis(2-methoxyphenyl)pyrimidin-2-amine 667 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89224 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(2-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89225 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(2-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89226 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(2-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89227 A3 HeLa HUMAN 3H-NECA 4,6-bis(2-fluorophenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89228 A1 CHO cells HUMAN 3H-DPCPX 4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89229 A2A HeLa HUMAN 3H-ZM241385 4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89230 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89231 A3 HeLa HUMAN 3H-NECA 4,6-bis(2,4-dimethoxyphenyl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89232 A1 CHO cells HUMAN 3H-DPCPX 4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine 538 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89233 A2A HeLa HUMAN 3H-ZM241385 4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89234 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89235 A3 HeLa HUMAN 3H-NECA 4,6-di(benzo[d][1,3]dioxol-5-yl)pyrimidin-2-amine 5306 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89236 A1 CHO cells HUMAN 3H-DPCPX 4,6-distyrylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89237 A2A HeLa HUMAN 3H-ZM241385 4,6-distyrylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89238 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-distyrylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89239 A3 HeLa HUMAN 3H-NECA 4,6-distyrylpyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89240 A1 CHO cells HUMAN 3H-DPCPX 4,6-di(furan-2-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89241 A2A HeLa HUMAN 3H-ZM241385 4,6-di(furan-2-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89242 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-di(furan-2-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89243 A3 HeLa HUMAN 3H-NECA 4,6-di(furan-2-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89244 A1 CHO cells HUMAN 3H-DPCPX 4,6-di(thiophen-2-yl)pyrimidin-2-amine 174 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89245 A2A HeLa HUMAN 3H-ZM241385 4,6-di(thiophen-2-yl)pyrimidin-2-amine 361 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89246 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-di(thiophen-2-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89247 A3 HeLa HUMAN 3H-NECA 4,6-di(thiophen-2-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89248 A1 CHO cells HUMAN 3H-DPCPX 4,6-di(furan-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89249 A2A HeLa HUMAN 3H-ZM241385 4,6-di(furan-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89250 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-di(furan-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89251 A3 HeLa HUMAN 3H-NECA 4,6-di(furan-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89252 A1 CHO cells HUMAN 3H-DPCPX 4,6-di(thiophen-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89253 A2A HeLa HUMAN 3H-ZM241385 4,6-di(thiophen-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89254 A2B HEK293 cells HUMAN 3H-DPCPX 4,6-di(thiophen-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89255 A3 HeLa HUMAN 3H-NECA 4,6-di(thiophen-3-yl)pyrimidin-2-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89256 A1 CHO cells HUMAN 3H-DPCPX 2,6-diphenylpyrimidin-4-amine 48.3 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89257 A2A HeLa HUMAN 3H-ZM241385 2,6-diphenylpyrimidin-4-amine 459 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89258 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-diphenylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89259 A3 HeLa HUMAN 3H-NECA 2,6-diphenylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89260 A1 CHO cells HUMAN 3H-DPCPX 2,6-di-p-tolylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89261 A2A HeLa HUMAN 3H-ZM241385 2,6-di-p-tolylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89262 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-di-p-tolylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89263 A3 HeLa HUMAN 3H-NECA 2,6-di-p-tolylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89264 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89265 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89266 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89267 A3 HeLa HUMAN 3H-NECA 2,6-bis(4-(trifluoromethyl)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89268 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(4-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89269 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(4-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89270 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(4-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89271 A3 HeLa HUMAN 3H-NECA 2,6-bis(4-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89272 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89273 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89274 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89275 A3 HeLa HUMAN 3H-NECA 2,6-bis(4-(methylthio)phenyl)pyrimidin-4-amine 3600 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89276 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(4-acetylphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89277 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(4-acetylphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89278 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(4-acetylphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89279 A3 HeLa HUMAN 3H-NECA 2,6-bis(4-acetylphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89280 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(4-fluorophenyl)pyrimidin-4-amine 110 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89281 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(4-fluorophenyl)pyrimidin-4-amine 1304 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89282 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(4-fluorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89283 A3 HeLa HUMAN 3H-NECA 2,6-bis(4-fluorophenyl)pyrimidin-4-amine 3107 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89284 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(4-chlorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89285 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(4-chlorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89286 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(4-chlorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89287 A3 HeLa HUMAN 3H-NECA 2,6-bis(4-chlorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89288 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(2-methoxyphenyl)pyrimidin-4-amine 184 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89289 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(2-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89290 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(2-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89291 A3 HeLa HUMAN 3H-NECA 2,6-bis(2-methoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89292 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(2-fluorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89293 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(2-fluorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89294 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(2-fluorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89295 A3 HeLa HUMAN 3H-NECA 2,6-bis(2-fluorophenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89296 A1 CHO cells HUMAN 3H-DPCPX 2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89297 A2A HeLa HUMAN 3H-ZM241385 2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89298 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89299 A3 HeLa HUMAN 3H-NECA 2,6-bis(2,4-dimethoxyphenyl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89300 A1 CHO cells HUMAN 3H-DPCPX 2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine 7.9 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89301 A2A HeLa HUMAN 3H-ZM241385 2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89302 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89303 A3 HeLa HUMAN 3H-NECA 2,6-di(benzo[d][1,3]dioxol-6-yl)pyrimidin-4-amine 299 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89304 A1 CHO cells HUMAN 3H-DPCPX 2,6-distyrylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89305 A2A HeLa HUMAN 3H-ZM241385 2,6-distyrylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89306 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-distyrylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89307 A3 HeLa HUMAN 3H-NECA 2,6-distyrylpyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89308 A1 CHO cells HUMAN 3H-DPCPX 2,6-di(furan-2-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89309 A2A HeLa HUMAN 3H-ZM241385 2,6-di(furan-2-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89310 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-di(furan-2-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89311 A3 HeLa HUMAN 3H-NECA 2,6-di(furan-2-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89312 A1 CHO cells HUMAN 3H-DPCPX 2,6-di(thiophen-2-yl)pyrimidin-4-amine 85.4 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89313 A2A HeLa HUMAN 3H-ZM241385 2,6-di(thiophen-2-yl)pyrimidin-4-amine 164 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89314 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-di(thiophen-2-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89315 A3 HeLa HUMAN 3H-NECA 2,6-di(thiophen-2-yl)pyrimidin-4-amine 831 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89316 A1 CHO cells HUMAN 3H-DPCPX 2,6-di(furan-3-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89317 A2A HeLa HUMAN 3H-ZM241385 2,6-di(furan-3-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89318 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-di(furan-3-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89319 A3 HeLa HUMAN 3H-NECA 2,6-di(furan-3-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89320 A1 CHO cells HUMAN 3H-DPCPX 2,6-di(thiophen-3-yl)pyrimidin-4-amine 194 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89321 A2A HeLa HUMAN 3H-ZM241385 2,6-di(thiophen-3-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89322 A2B HEK293 cells HUMAN 3H-DPCPX 2,6-di(thiophen-3-yl)pyrimidin-4-amine 100 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89323 A3 HeLa HUMAN 3H-NECA 2,6-di(thiophen-3-yl)pyrimidin-4-amine 1178 Yaziji V et al 2011 Jan 15, 2025 Jan 15, 2025
89324 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide 16 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89325 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide 437 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89326 5-HT6 CLONED HUMAN 3H-LSD 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide 148 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89327 D2 CLONED HUMAN 3H-RACLOPRIDE 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide 631 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89328 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-cyanophenyl)methyl]propanamide 9.3 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89329 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide 245 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89330 D2 CLONED HUMAN 3H-RACLOPRIDE 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide 345 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89331 5-HT6 CLONED HUMAN 3H-LSD 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide 830 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89332 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide 582 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89333 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-[(4-trifluoromethylpnenyl)methyl]propanamide 35 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89334 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide 53 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89335 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide 1055 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89336 5-HT6 CLONED HUMAN 3H-LSD 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide 2518 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89337 D2 CLONED HUMAN 3H-RACLOPRIDE 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide 2450 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89338 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-{2-[4-(2-Biphenyl)piperazin-1-yl]ethoxy}-N-(pyridin-4-ylmethyl)propanamide 94 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89339 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide 288 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89340 D2 CLONED HUMAN 3H-RACLOPRIDE N-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide 537 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89341 5-HT6 CLONED HUMAN 3H-LSD N-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide 1633 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89342 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide 595 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89343 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(3-phenyl-2-pyridyl)piperazin-1-yl]ethoxy}propanamide 76 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89344 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 52 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89345 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 365 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89346 5-HT6 CLONED HUMAN 3H-LSD 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 1039 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89347 D2 CLONED HUMAN 3H-RACLOPRIDE 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 268 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89348 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-{2-[4-(3-Phenyl-2-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 1221 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89349 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 310 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89350 D2 CLONED HUMAN 3H-RACLOPRIDE N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 4346 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89351 5-HT6 CLONED HUMAN 3H-LSD N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 3441 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89352 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 3842 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89353 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Cyanophenyl)methyl]-3-{2-[4-(2-phenyl-3-pyridyl)piperazin-1-yl]ethoxy}propanamide 87 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89354 5-HT7 CLONED HUMAN 3H-5-CT 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 44 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89355 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 802 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89356 5-HT6 CLONED HUMAN 3H-LSD 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 2215 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89357 D2 CLONED HUMAN 3H-RACLOPRIDE 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 2766 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89358 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-{2-[4-(2-Phenyl-3-pyridyl)piperazin-1-yl]ethoxy}N-[(4-trifluoromethylphenyl)methyl] propanamide 471 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89359 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 914 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89360 D2 CLONED HUMAN 3H-RACLOPRIDE N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 1959 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89361 5-HT6 CLONED HUMAN 3H-LSD N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 2815 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89362 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 6631 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89363 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[2-(4-fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy) propanamide 108 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89364 5-HT7 CLONED HUMAN 3H-5-CT 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 254 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89365 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 6064 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89366 5-HT6 CLONED HUMAN 3H-LSD 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 2634 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89367 D2 CLONED HUMAN 3H-RACLOPRIDE 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 3460 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89368 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-(2-{4-[2-(4-Fluorophenyl)-3-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 263 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89369 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 156 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89370 D2 CLONED HUMAN 3H-RACLOPRIDE N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 685 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89371 5-HT6 CLONED HUMAN 3H-LSD N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 1621 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89372 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 2630 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89373 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Cyanophenyl)methyl]-3-(2-{4-[3-(4-fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy) propanamide 54 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89374 5-HT7 CLONED HUMAN 3H-5-CT 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 32 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89375 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 1836 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89376 5-HT6 CLONED HUMAN 3H-LSD 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 1074 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89377 D2 CLONED HUMAN 3H-RACLOPRIDE 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 393 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89378 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 3-(2-{4-[3-(4-Fluorophenyl)-2-pyridyl]piperazin-1-yl}ethoxy)-N-[(4-trifluoromethylphenyl)methyl] propanamide 1369 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89379 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 5.9 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89380 D2 CLONED HUMAN 3H-RACLOPRIDE N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 321 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89381 5-HT6 CLONED HUMAN 3H-LSD N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 640 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 160 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89383 5-HT7 CLONED HUMAN 3H-5-CT N-[(4-Methoxymethoxyphenyl)methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 6.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89384 5-HT7 CLONED HUMAN 3H-5-CT N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 14.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 152 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89386 5-HT6 CLONED HUMAN 3H-LSD N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 1336 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89387 D2 CLONED HUMAN 3H-RACLOPRIDE N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 419 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89388 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-[[4-(2-Hydroxyethoxy)phenyl]methyl]- 4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 53 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89389 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 26 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89390 D2 CLONED HUMAN 3H-RACLOPRIDE 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 375 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89391 5-HT6 CLONED HUMAN 3H-LSD 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 1706 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 163 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89393 5-HT7 CLONED HUMAN 3H-5-CT 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 25 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89394 5-HT7 CLONED HUMAN 3H-5-CT 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 18.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89395 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 105 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89396 5-HT6 CLONED HUMAN 3H-LSD 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 1623 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89397 D2 CLONED HUMAN 3H-RACLOPRIDE 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 260 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89398 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-[2-(4-Methoxyphenyl)phenyl]-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 53 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89399 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 30 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89400 D2 CLONED HUMAN 3H-RACLOPRIDE N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 293 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89401 5-HT6 CLONED HUMAN 3H-LSD N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 745 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89402 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 126 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89403 5-HT7 CLONED HUMAN 3H-5-CT N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 8 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89404 5-HT7 CLONED HUMAN 3H-5-CT 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 4.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89405 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 86 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89406 5-HT6 CLONED HUMAN 3H-LSD 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 413 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89407 D2 CLONED HUMAN 3H-RACLOPRIDE 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 36 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89408 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-(2-Biphenyl)-N-[(4-methoxymethoxyphenyl)methyl]-1-piperazinehexanamide 20 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89409 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-(2-Biphenyl)-N-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-piperazinehexanamide 4.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89410 5-HT7 CLONED HUMAN 3H-5-CT 4-(2-Biphenyl)-N-[[4-(2-hydroxyethoxy)phenyl]methyl]-1-piperazinehexanamide 259 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89411 5-HT7 CLONED HUMAN 3H-5-CT 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 16 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89412 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 160 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89413 5-HT6 CLONED HUMAN 3H-LSD 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 1724 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89414 D2 CLONED HUMAN 3H-RACLOPRIDE 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 136 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89415 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)ethoxy]phenyl]methyl]-1-piperazinehexanamide 7.4 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89416 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 12.3 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89417 D2 CLONED HUMAN 3H-RACLOPRIDE 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 64 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89418 5-HT6 CLONED HUMAN 3H-LSD 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 1152 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89419 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 149 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89420 5-HT7 CLONED HUMAN 3H-5-CT 4-(2-Biphenyl)-N-[[4-[2-(4-morpholinyl)propoxy]phenyl]methyl]-1-piperazinehexanamide 9.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89421 5-HT7 CLONED HUMAN 3H-5-CT 4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide 21 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89422 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide 74 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89423 5-HT6 CLONED HUMAN 3H-LSD 4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide 1506 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89424 D2 CLONED HUMAN 3H-RACLOPRIDE 4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide 75 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89425 CORTICAL MEMBRANES PIG 3H-PRAZOSIN 4-(2-Biphenyl)-N-[[4-(dimethylaminomethyl)phenyl]methyl]-1-piperazinehexanamide 23 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89426 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide 6.6 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89427 D2 CLONED HUMAN 3H-RACLOPRIDE N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide 522 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89428 5-HT6 CLONED HUMAN 3H-LSD N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide 614 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89429 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide 771 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89430 5-HT7 CLONED HUMAN 3H-5-CT N-(4-Cyanophenylmethyl)-4-[2-(4-methoxyphenyl)-4-fluorophenyl]-1-piperazinehexanamide 25.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89431 5-HT7 CLONED HUMAN 3H-5-CT N-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide 27 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89432 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide 2870 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89433 5-HT6 CLONED HUMAN 3H-LSD N-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide 927 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89434 D2 CLONED HUMAN 3H-RACLOPRIDE N-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide 1385 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89435 CORTICAL MEMBRANES PIG 3H-PRAZOSIN N-(4-Cyanophenylmethyl)-4-[2-(4-cyanophenyl)-4-fluorophenyl]-1-piperazinehexanamide 3.2 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89436 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 12.9 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89437 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 308 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89438 5-HT6 CLONED HUMAN 3H-LSD (S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 700 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89439 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 147 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89440 5-HT7 CLONED HUMAN 3H-5-CT (S)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 19 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89441 5-HT7 CLONED HUMAN 3H-5-CT (R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 12 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89442 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 109 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89443 5-HT6 CLONED HUMAN 3H-LSD (R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 843 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89444 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 243 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89445 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (R)-N-(4-Cyano-1-phenylethyl)-4-[2-(4-methoxyphenyl)phenyl]-1-piperazinehexanamide 17.8 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89446 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 46.4 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89447 D2 CORTICAL MEMBRANES PIG 3H-RACLOPRIDE (S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 53 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89448 5-HT6 CLONED HUMAN 3H-LSD (S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 480 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89449 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 66 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89450 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 10 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89451 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 10.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89452 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 80 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89453 5-HT6 CLONED HUMAN 3H-LSD (R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 561 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89454 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 116 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89455 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (R)-4-(2-Biphenyl)-N-(1-phenylethyl)-1-piperazinehexanamide 36.6 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89456 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 36 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89457 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 295 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89458 5-HT6 CLONED HUMAN 3H-LSD (R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 721 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89459 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 134 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89460 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 11.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89461 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 15.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89462 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 103 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89463 5-HT6 CLONED HUMAN 3H-LSD (S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 652 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89464 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 177 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89465 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (S)-4-[2-(4-Methoxyphenyl)phenyl]-N-(1-phenylethyl)-1-piperazinehexanamide 22.1 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89466 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 11.6 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89467 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 178 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89468 5-HT6 CLONED HUMAN 3H-LSD (R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 434 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89469 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 101 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89470 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 14 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89471 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 36.5 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89472 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 202 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89473 5-HT6 CLONED HUMAN 3H-LSD (S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 395 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89474 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 243 Lacivita E et al 2016 Jan 15, 2025 Jan 28, 2025
89475 CORTICAL MEMBRANES PIG 3H-PRAZOSIN (S)-4-(2-Biphenyl)-N-[(4-cyanophenyl)methyl]-2-methyl-1-piperazinehexanamide 42.6 Lacivita E et al 2016 Jan 15, 2025 Jan 15, 2025
89476 M1 CLONED HUMAN 3H-NMS 1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89477 M2 CLONED HUMAN 3H-NMS 1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89478 M3 CLONED HUMAN 3H-NMS 1-(2-Methoxyphenyl)-N,N,N-trimethylmethanaminium iodide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89479 M3 CLONED HUMAN 3H-NMS 2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 4700 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89480 M2 CLONED HUMAN 3H-NMS 2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 5700 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89481 M1 CLONED HUMAN 3H-NMS 2-(2-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 4900 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89482 M1 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89483 M2 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89484 M3 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89485 M3 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide 620 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89486 M2 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide 630 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89487 M1 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylpropan-1-aminium iodide 330 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89488 M1 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89489 M2 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89490 M3 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-en-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89491 M3 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89492 M2 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89493 M1 CLONED HUMAN 3H-NMS 3-(3-Methoxyphenyl)-N,N,N-trimethylprop-2-yn-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89494 M1 CLONED HUMAN 3H-NMS 1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate 7300 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89495 M2 CLONED HUMAN 3H-NMS 1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89496 M3 CLONED HUMAN 3H-NMS 1-(2-(3-Methoxyphenyl)cyclopropyl)-N,N,N-trimethylmethanaminium formate 8700 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89497 M3 CLONED HUMAN 3H-NMS 5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89498 M2 CLONED HUMAN 3H-NMS 5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89499 M1 CLONED HUMAN 3H-NMS 5-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89500 M1 CLONED HUMAN 3H-NMS 8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89501 M2 CLONED HUMAN 3H-NMS 8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate 6300 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89502 M3 CLONED HUMAN 3H-NMS 8-Methoxy-2,2-dimethyl-1,2,3,4-tetrahydroisoquinolin-2-ium formate 5800 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89503 M3 CLONED HUMAN 3H-NMS 8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 2000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89504 M2 CLONED HUMAN 3H-NMS 8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 930 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89505 M1 CLONED HUMAN 3H-NMS 8-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 1000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89506 M1 CLONED HUMAN 3H-NMS 8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 2900 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89507 M2 CLONED HUMAN 3H-NMS 8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 4200 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89508 M3 CLONED HUMAN 3H-NMS 8-Hydroxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89509 M3 CLONED HUMAN 3H-NMS 1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate 3900 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89510 M2 CLONED HUMAN 3H-NMS 1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate 1300 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89511 M1 CLONED HUMAN 3H-NMS 1-(8-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate 1800 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89512 M1 CLONED HUMAN 3H-NMS 5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 2500 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89513 M2 CLONED HUMAN 3H-NMS 5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 4400 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89514 M3 CLONED HUMAN 3H-NMS 5-Methoxy-N,N,N-trimethyl-1,2,3,4-tetrahydronaphthalen-2-aminium iodide 4000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89515 M3 CLONED HUMAN 3H-NMS 1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89516 M2 CLONED HUMAN 3H-NMS 1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89517 M1 CLONED HUMAN 3H-NMS 1-(5-Methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N,N,N-trimethylmethanaminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89518 M1 CLONED HUMAN 3H-NMS 8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 2000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89519 M2 CLONED HUMAN 3H-NMS 8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 1200 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89520 M3 CLONED HUMAN 3H-NMS 8-Methoxy-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 830 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89521 M3 CLONED HUMAN 3H-NMS 7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89522 M2 CLONED HUMAN 3H-NMS 7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89523 M1 CLONED HUMAN 3H-NMS 7-(Dimethylamino)-5,6,7,8-tetrahydronaphthalen-1-ol >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89524 M1 CLONED HUMAN 3H-NMS 2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 23 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89525 M2 CLONED HUMAN 3H-NMS 2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 140 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89526 M3 CLONED HUMAN 3H-NMS 2-(Benzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 41 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89527 M3 CLONED HUMAN 3H-NMS 3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate 140 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89528 M2 CLONED HUMAN 3H-NMS 3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate 230 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89529 M1 CLONED HUMAN 3H-NMS 3-(Benzofuran-6-yl)-N,N,N-trimethylpropan-1-aminium formate 63 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89530 M1 CLONED HUMAN 3H-NMS N,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate 380 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89531 M2 CLONED HUMAN 3H-NMS N,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate 790 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89532 M3 CLONED HUMAN 3H-NMS N,N,N-Trimethyl-6,7,8,9-tetrahydronaphtho[1,2-b]furan-8-aminium formate 690 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89533 M3 CLONED HUMAN 3H-NMS iperoxo 550 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89534 M2 CLONED HUMAN 3H-NMS iperoxo 4.9 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89535 M1 CLONED HUMAN 3H-NMS iperoxo 350 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89536 M1 CLONED HUMAN 3H-NMS Acetylcholine 5.8 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89537 M2 CLONED HUMAN 3H-NMS Acetylcholine 0.39 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89538 M3 CLONED HUMAN 3H-NMS Acetylcholine 4.7 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89539 M3 CLONED HUMAN 3H-NMS CARBACHOL 51 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89540 M2 CLONED HUMAN 3H-NMS CARBACHOL 4.1 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89541 M1 CLONED HUMAN 3H-NMS CARBACHOL 63 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89542 M1 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N-methylethan-1-amine 740 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89543 M2 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N-methylethan-1-amine 1000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89544 M3 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N-methylethan-1-amine 780 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89545 M3 CLONED HUMAN 3H-NMS 2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89546 M2 CLONED HUMAN 3H-NMS 2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89547 M1 CLONED HUMAN 3H-NMS 2-(3-Hydroxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89548 M1 CLONED HUMAN 3H-NMS 2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 7100 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89549 M2 CLONED HUMAN 3H-NMS 2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate 980 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89550 M3 CLONED HUMAN 3H-NMS 2-(2-Fluoro-5-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89551 M3 CLONED HUMAN 3H-NMS 2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89552 M2 CLONED HUMAN 3H-NMS 2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89553 M1 CLONED HUMAN 3H-NMS 2-Hydroxy-2-(3-methoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89554 M1 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate 170 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89555 M2 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate 2400 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89556 M3 CLONED HUMAN 3H-NMS 2-(3-Methoxyphenyl)-N,N,N-trimethyl-2-oxoethan-1-aminium formate 210 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89557 M3 CLONED HUMAN 3H-NMS 2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89558 M2 CLONED HUMAN 3H-NMS 2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89559 M1 CLONED HUMAN 3H-NMS 2-(3-Ethoxyphenyl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89560 M1 CLONED HUMAN 3H-NMS 2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate 4500 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89561 M2 CLONED HUMAN 3H-NMS 2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate 4800 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89562 M3 CLONED HUMAN 3H-NMS 2-(3-Chlorophenyl)-N,N,N-trimethylethan-1-aminium formate 5800 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89563 M3 CLONED HUMAN 3H-NMS N,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89564 M2 CLONED HUMAN 3H-NMS N,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate 9200 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89565 M1 CLONED HUMAN 3H-NMS N,N,N-Trimethyl-2-(3-(trifluoromethoxy)phenyl)ethan-1-aminium formate 7800 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89566 M1 CLONED HUMAN 3H-NMS 2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 6400 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89567 M2 CLONED HUMAN 3H-NMS 2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89568 M3 CLONED HUMAN 3H-NMS 2-(2,3-Dihydrobenzofuran-6-yl)-N,N,N-trimethylethan-1-aminium formate 6300 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89569 M3 CLONED HUMAN 3H-NMS 3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89570 M2 CLONED HUMAN 3H-NMS 3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89571 M1 CLONED HUMAN 3H-NMS 3-[[(3R)-pyrrolidin-3-yl]methoxymethyl]pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89572 M1 CLONED HUMAN 3H-NMS 2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole 4200 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89573 M2 CLONED HUMAN 3H-NMS 2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole 6000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89574 M3 CLONED HUMAN 3H-NMS 2-[[(3R)-pyrrolidin-3-yl]oxymethyl]-1,3-thiazole 4100 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89575 M1 CLONED HUMAN 3H-NMS (3R)-3-(imidazol-1-ylmethyl)piperidine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89576 M2 CLONED HUMAN 3H-NMS (3R)-3-(imidazol-1-ylmethyl)piperidine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89577 M3 CLONED HUMAN 3H-NMS (3R)-3-(imidazol-1-ylmethyl)piperidine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89578 M3 CLONED HUMAN 3H-NMS 2-(1,3-benzodioxol-5-yl)guanidine 9700 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89579 M2 CLONED HUMAN 3H-NMS 2-(1,3-benzodioxol-5-yl)guanidine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89580 M1 CLONED HUMAN 3H-NMS 2-(1,3-benzodioxol-5-yl)guanidine 8300 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89581 M1 CLONED HUMAN 3H-NMS 3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89582 M2 CLONED HUMAN 3H-NMS 3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89583 M3 CLONED HUMAN 3H-NMS 3-[[(3R)-piperidin-3-yl]oxymethyl]pyridine 9500 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89584 M3 CLONED HUMAN 3H-NMS 2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89585 M2 CLONED HUMAN 3H-NMS 2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89586 M1 CLONED HUMAN 3H-NMS 2-(8-methoxyimidazo[1,2-a]pyridin-2-yl)ethanamine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89587 M1 CLONED HUMAN 3H-NMS 2-(3-methoxyphenyl)ethanimidamide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89588 M2 CLONED HUMAN 3H-NMS 2-(3-methoxyphenyl)ethanimidamide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89589 M3 CLONED HUMAN 3H-NMS 2-(3-methoxyphenyl)ethanimidamide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89590 M3 CLONED HUMAN 3H-NMS 2-(3-methoxyphenoxy)ethanimidamide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89591 M2 CLONED HUMAN 3H-NMS 2-(3-methoxyphenoxy)ethanimidamide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89592 M1 CLONED HUMAN 3H-NMS 2-(3-methoxyphenoxy)ethanimidamide >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89593 M1 CLONED HUMAN 3H-NMS (2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89594 M2 CLONED HUMAN 3H-NMS (2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89595 M3 CLONED HUMAN 3H-NMS (2R)-1-imidazo[2,1-b][1,3]thiazol-6-ylpropan-2-amine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89596 M3 CLONED HUMAN 3H-NMS 4-[(3R)-piperidin-3-yl]oxypyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89597 M2 CLONED HUMAN 3H-NMS 4-[(3R)-piperidin-3-yl]oxypyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89598 M1 CLONED HUMAN 3H-NMS 4-[(3R)-piperidin-3-yl]oxypyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89599 M1 CLONED HUMAN 3H-NMS 1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium 6100 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89600 M2 CLONED HUMAN 3H-NMS 1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89601 M3 CLONED HUMAN 3H-NMS 1,1-Dimethyl-3-(thiazol-2-ylmethoxy)pyrrolidin-1-ium >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89602 M3 CLONED HUMAN 3H-NMS 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89603 M2 CLONED HUMAN 3H-NMS 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89604 M1 CLONED HUMAN 3H-NMS 3-(((1-Methylpyrrolidin-3-yl)methoxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89605 M1 CLONED HUMAN 3H-NMS 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89606 M2 CLONED HUMAN 3H-NMS 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89607 M3 CLONED HUMAN 3H-NMS 3-(((1-Methylpiperidin-3-yl)oxy)methyl)pyridine >10000 Fish I et al 2017 Jan 15, 2025 Jan 15, 2025
89608 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 0.47863 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89609 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89610 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89611 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89612 Alpha1A CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 177.828 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89613 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 2.5704 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89614 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.86209 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89615 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89616 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89617 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89618 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 54.9541 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89619 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1.25893 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89620 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.562341 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89621 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89622 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89623 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 23.4423 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89624 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 0.616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89625 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0616595 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89626 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 512.861 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89627 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89628 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89629 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 165.959 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89630 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0645654 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89631 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 0.0147911 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89632 D2 CLONED HUMAN 3H-Methylspiperone (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89633 D2 CLONED HUMAN 3H-Methylspiperone (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89634 CORTEX RAT 3H-PRAZOSIN (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 128.825 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89635 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 0.0338844 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89636 5-HT1A CLONED HUMAN 3H-8-OH-DPAT NLX-101 2.18776 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89637 CORTEX RAT 3H-PRAZOSIN NLX-101 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89638 D2 CLONED HUMAN 3H-Methylspiperone NLX-101 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89639 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 8-OH-DPAT 0.812831 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89640 5-HT1A CLONED HUMAN 3H-8-OH-DPAT BUSPIRONE 5.01187 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89641 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1.51356 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89642 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89643 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89644 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89645 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89646 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 389.045 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89647 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 0.524807 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89648 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89649 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89650 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 35.4813 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89651 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 208.93 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89652 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89653 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89654 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89655 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89656 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 199.526 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89657 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 3.80189 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89658 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89659 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89660 D2 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89661 CORTEX RAT 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89662 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 13.8038 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89663 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89664 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89665 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl) (4-fluoro-4-(((3-phenylpropyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89666 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89667 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89668 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((3-(pyridin-2-yl)propyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89669 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89670 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89671 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylamino)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89672 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89673 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89674 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylamino)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89675 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89676 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89677 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(phenylthio)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89678 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89679 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89680 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-ylthio)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89681 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89682 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89683 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89684 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89685 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89686 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89687 5-HT2A CLONED HUMAN 3H-KETANSERIN (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89688 M1 CLONED HUMAN 3H-NMS (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89689 H1 CLONED HUMAN 3H-PYRILAMINE (3,4-Dichlorophenyl)(4-fluoro-4-(((2-phenoxyethyl)amino)- methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89690 H1 CLONED HUMAN 3H-PYRILAMINE (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89691 M1 CLONED HUMAN 3H-NMS (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89692 5-HT2A CLONED HUMAN 3H-KETANSERIN (3,4-Dichlorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89693 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89694 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89695 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-3-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89696 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89697 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89698 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-4-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89699 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89700 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89701 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrazin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89702 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89703 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89704 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-2-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89705 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89706 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89707 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyrimidin-5-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89708 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89709 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89710 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridazin-4-yloxy)- ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89711 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89712 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89713 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyridin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89714 H1 CLONED HUMAN 3H-PYRILAMINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89715 M1 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89716 5-HT2A CLONED HUMAN 3H-KETANSERIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-((5-methylpyrimidin-2- yl)oxy)ethyl)amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89717 A2A CLONED HUMAN 3H-NECA (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89718 Alpha1A CLONED HUMAN 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 165.959 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89719 Alpha1B CLONED HUMAN 3H-PRAZOSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89720 Beta 1 CLONED HUMAN 125I-Pindolol (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89721 Beta 2 CLONED HUMAN 3H-CGP12177 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89722 CB1 CLONED HUMAN 3H-CP55940 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89723 CB2 CLONED HUMAN 3H-CP55940 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89724 CCK1 CLONED HUMAN 125I-BH-CCK-8 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89725 D1 CLONED HUMAN 3H-SCH23390 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89726 D3 CLONED HUMAN 3H-Methylspiperone (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89727 ETA CLONED HUMAN 125I-ENDOTHELIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89728 5-HT1D CLONED HUMAN 125I-aminopotentidine (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89729 H3 CLONED HUMAN 3H-Alpha-methylhistamine (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89730 H4 CLONED HUMAN 3H-Histamine (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89731 M2 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89732 M3 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89733 M4 CLONED HUMAN 3H-NMS (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89734 DOR CLONED HUMAN 3H-DADLE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89735 KOR CLONED HUMAN 3H-U69593 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89736 MOR CLONED HUMAN 3H-DAMGO (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89737 V1A CLONED HUMAN 3H-VASOPRESSIN (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89738 5-HT1B CLONED HUMAN 3H-5-CT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89739 5-HT1D CLONED HUMAN 3H-5-CT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89740 5-HT2B CLONED HUMAN 3H-LSD (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89741 5-HT2C CLONED HUMAN 3H-MESULERGINE (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89742 5-HT6 CLONED HUMAN 3H-LSD (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89743 5-HT6 CLONED HUMAN 3H-5-CT (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone 1000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89744 DAT CLONED HUMAN 3H-WIN 35,428 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89745 NET CLONED HUMAN 3H-Nisoxene (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89746 SERT CLONED HUMAN 3H-CITALOPRAM (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89747 BZP CORTEX RAT FNZ (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 29, 2025
89748 NMDA CORTEX RAT 3H-MK-801 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025