The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 88,001-89,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
90749Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine9.4Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90750Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine7.6Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90751Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90752Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine33Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90753Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine12Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90754Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine5.5Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90755Sigma 2CLONEDHUMAN3H-DTGDTG20Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90756MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine258Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90757MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90758MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine163Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90759MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine391Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90760MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine185Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90761MORbrain membranesGUINEA PIG3H-DAMGOcis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine495Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90762MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine879Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90763MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine297Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90764MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine354Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90765MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine462Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90766MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine299Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90767MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine391Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90768MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine273Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90769MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine501Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90770MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine231Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90771MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90772MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine114Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90773MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine841Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90774MORbrain membranesGUINEA PIG3H-DAMGOcis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90775MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine115Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90776MORbrain membranesGUINEA PIG3H-DAMGOcis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine768Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90777MORbrain membranesGUINEA PIG3H-DAMGOtrans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine31Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90778MORbrain membranesGUINEA PIG3H-DAMGOcis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90779MORbrain membranesGUINEA PIG3H-DAMGONALOXONE2.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90780MORbrain membranesGUINEA PIG3H-DAMGOMorphine3.9Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90781DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine479Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90782DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine209Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90783DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90784DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90785DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine185Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90786DORbrain membranesRAT3H-DPDPEcis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine432Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90787DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90788DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine356Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90789DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine228Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90790DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90791DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine150Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90792DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine364Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90793DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine114Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90794DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine143Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90795DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine254Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90796DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine559Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90797DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine178Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90798DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90799DORbrain membranesRAT3H-DPDPEtrans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine187Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90800DORbrain membranesRAT3H-DPDPEcis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine565Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90801DORbrain membranesRAT3H-DPDPEtrans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90802DORbrain membranesRAT3H-DPDPEcis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine655Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90803DORbrain membranesRAT3H-DPDPEtrans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine14Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90804DORbrain membranesRAT3H-DPDPEcis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90805DORbrain membranesRAT3H-DPDPENALOXONE2.4Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90806DORbrain membranesRAT3H-DPDPEMorphine2Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90807KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine604Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90808KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90809KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine85Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90810KORbrain membranesGUINEA PIG3H-U69593cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine745Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90811KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90812KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90813KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine96Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90814KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90815KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine980Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90816KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90817KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine506Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90818KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90819KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine639Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90820KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90821KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine236Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90822KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90823KORbrain membranesGUINEA PIG3H-U69593trans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90824KORbrain membranesGUINEA PIG3H-U69593cis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90825KORbrain membranesGUINEA PIG3H-U69593trans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine413Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90826KORbrain membranesGUINEA PIG3H-U69593cis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine1140Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90827KORbrain membranesGUINEA PIG3H-U69593trans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine85Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90828KORbrain membranesGUINEA PIG3H-U69593cis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90829KORbrain membranesGUINEA PIG3H-U69593NALOXONE6.9Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90830KORbrain membranesGUINEA PIG3H-U69593Morphine35Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90831NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90832NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90833NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90834NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90835NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-Benzyl-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90836NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-Benzyl-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90837NMDACORTICAL MEMBRANESPIG3H-MK-801trans-N-Benzyl-3-methoxy-N-methyl-3,4-dihydrospiro-[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90838NMDACORTICAL MEMBRANESPIG3H-MK-801cis-N-Benzyl-3-methoxy-N-methyl-3,4-dihydrospiro-[[2]benzopyran-1,1′-cyclohexan]-4′-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90839Alpha1ACHO cellsHUMAN3H-PRAZOSIN1-(1,4-dioxaspiro[4,5]dec-2-ylmethyl)-4-(2-methoxyphenyl)piperazine91.2011Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90840Alpha1BCHO cellsHUMAN3H-PRAZOSIN1-(1,4-dioxaspiro[4,5]dec-2-ylmethyl)-4-(2-methoxyphenyl)piperazine125.893Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90841Alpha1DCHO cellsHUMAN3H-PRAZOSIN1-(1,4-dioxaspiro[4,5]dec-2-ylmethyl)-4-(2-methoxyphenyl)piperazine1000Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908425-HT1AHeLaHUMAN3H-8-OH-DPAT1-(1,4-dioxaspiro[4,5]dec-2-ylmethyl)-4-(2-methoxyphenyl)piperazine5.12861Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90843Alpha1ACHO cellsHUMAN3H-PRAZOSIN1-{1,4-Dioxa-8-thiaspiro[4.5]decan-2-ylmethyl}-4-(2-methoxyphenyl)piperazine8.51138Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90844Alpha1BCHO cellsHUMAN3H-PRAZOSIN1-{1,4-Dioxa-8-thiaspiro[4.5]decan-2-ylmethyl}-4-(2-methoxyphenyl)piperazine141.254Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90845Alpha1DCHO cellsHUMAN3H-PRAZOSIN1-{1,4-Dioxa-8-thiaspiro[4.5]decan-2-ylmethyl}-4-(2-methoxyphenyl)piperazine14.7911Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908465-HT1AHeLaHUMAN3H-8-OH-DPAT1-{1,4-Dioxa-8-thiaspiro[4.5]decan-2-ylmethyl}-4-(2-methoxyphenyl)piperazine9.33254Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90847Alpha1ACHO cellsHUMAN3H-PRAZOSIN1-(2-Methoxyphenyl)-4-{1,4,8-trioxaspiro[4.5]decan-2-ylmethyl}piperazine16.9824Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90848Alpha1BCHO cellsHUMAN3H-PRAZOSIN1-(2-Methoxyphenyl)-4-{1,4,8-trioxaspiro[4.5]decan-2-ylmethyl}piperazine323.594Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90849Alpha1DCHO cellsHUMAN3H-PRAZOSIN1-(2-Methoxyphenyl)-4-{1,4,8-trioxaspiro[4.5]decan-2-ylmethyl}piperazine25.1189Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908505-HT1AHeLaHUMAN3H-8-OH-DPAT1-(2-Methoxyphenyl)-4-{1,4,8-trioxaspiro[4.5]decan-2-ylmethyl}piperazine46.7735Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90851Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-Benzyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane6.76083Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90852Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-Benzyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane16.5959Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90853Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-Benzyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane4.67735Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908545-HT1AHeLaHUMAN3H-8-OH-DPAT8-Benzyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane14.4544Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90855Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l4-thiaspiro[4.5]decan-8-one478.63Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90856Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l4-thiaspiro[4.5]decan-8-one42.658Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908575-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l4-thiaspiro[4.5]decan-8-one117.49Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90858Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l6-thiaspiro[4.5]decane-8,8-dione9.77237Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90859Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l6-thiaspiro[4.5]decane-8,8-dione288.403Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90860Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l6-thiaspiro[4.5]decane-8,8-dione51.2861Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908615-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4- dioxa-8l6-thiaspiro[4.5]decane-8,8-dione81.2831Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90862Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane48.9779Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90863Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane42.658Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90864Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane37.1535Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908655-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane158.489Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90866Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-phenyl-1,4-dioxa-8-azaspiro[4.5]decane6.45654Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90867Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-phenyl-1,4-dioxa-8-azaspiro[4.5]decane154.882Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90868Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-phenyl-1,4-dioxa-8-azaspiro[4.5]decane8.12831Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908695-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-phenyl-1,4-dioxa-8-azaspiro[4.5]decane15.8489Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90870Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyridin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane17.7828Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90871Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyridin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane1000Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90872Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyridin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane22.9087Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908735-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyridin-2-yl)-1,4-dioxa-8-azaspiro[4.5]decane8.91251Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90874Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-Benzoyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane10.7152Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90875Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-Benzoyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane67.6083Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90876Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-Benzoyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane20.4174Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908775-HT1AHeLaHUMAN3H-8-OH-DPAT8-Benzoyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane58.8844Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90878Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane10.2329Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90879Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane63.0957Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90880Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane10.9648Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908815-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4-(trifluoromethyl)benzoyl]-1,4-dioxa-8-azaspiro[4.5]decane50.1187Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90882Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane21.3796Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90883Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane158.489Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90884Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane28.1838Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908855-HT1AHeLaHUMAN3H-8-OH-DPAT8-(Furan-2-carbonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane42.658Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90886Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane30.903Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90887Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane109.648Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90888Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane39.8107Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908895-HT1AHeLaHUMAN3H-8-OH-DPAT8-Cyclohexanecarbonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane20.4174Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90890Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane11.749Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90891Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane158.489Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90892Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane26.9153Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908935-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(pyrrolidine-2-carbonyl)-1,4-dioxa-8-azaspiro[4.5]decane36.3078Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90894Alpha1ACHO cellsHUMAN3H-PRAZOSIN1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one60.256Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90895Alpha1BCHO cellsHUMAN3H-PRAZOSIN1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one1000Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90896Alpha1DCHO cellsHUMAN3H-PRAZOSIN1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one89.1251Franchini S et al 2014Jan 15, 2025Jan 28, 2025
908975-HT1AHeLaHUMAN3H-8-OH-DPAT1-(2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one64.5654Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90898Alpha1ACHO cellsHUMAN3H-PRAZOSIN2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one1000Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90899Alpha1BCHO cellsHUMAN3H-PRAZOSIN2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one1000Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90900Alpha1DCHO cellsHUMAN3H-PRAZOSIN2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one416.869Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909015-HT1AHeLaHUMAN3H-8-OH-DPAT2,2,2-Trifluoro-1-(2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decan-8-yl)ethan-1-one323.594Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90902Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane7.94328Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90903Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane85.1138Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90904Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane12.3027Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909055-HT1AHeLaHUMAN3H-8-OH-DPAT8-(Benzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane52.4807Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90906Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane4.57088Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90907Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane8.31764Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90908Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane10.7152Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909095-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-methylbenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane26.9153Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90910Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane6.45654Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90911Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane69.1831Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90912Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane7.07946Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909135-HT1AHeLaHUMAN3H-8-OH-DPAT8-(4-Chlorobenzenesulfonyl)-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane37.1535Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90914Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane8.91251Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90915Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane147.911Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90916Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane26.3027Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909175-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-[4(trifluoromethoxy)benzenesulfonyl]-1,4-dioxa-8-azaspiro[4.5]decane69.1831Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90918Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane5.24807Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90919Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane109.648Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90920Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane5.7544Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909215-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(4-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane24.5471Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90922Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane3.01995Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90923Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane69.1831Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90924Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane0.912011Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909255-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(3-nitrobenzenesulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane43.6516Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90926Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane7.94328Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90927Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane85.1138Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90928Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane9.77237Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909295-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-8-(thiophene-2-sulfonyl)-1,4-dioxa-8-azaspiro[4.5]decane60.256Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90930Alpha1ACHO cellsHUMAN3H-PRAZOSIN8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane18.6209Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90931Alpha1BCHO cellsHUMAN3H-PRAZOSIN8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane363.078Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90932Alpha1DCHO cellsHUMAN3H-PRAZOSIN8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane23.4423Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909335-HT1AHeLaHUMAN3H-8-OH-DPAT8-Methanesulfonyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane144.544Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90934Alpha1ACHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-N-phenyl-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide12.0226Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90935Alpha1BCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-N-phenyl-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide81.2831Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90936Alpha1DCHO cellsHUMAN3H-PRAZOSIN2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-N-phenyl-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide13.1826Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909375-HT1AHeLaHUMAN3H-8-OH-DPAT2-{[4-(2-Methoxyphenyl)piperazin-1-yl]methyl}-N-phenyl-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide33.1131Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90938Alpha1ACHO cellsHUMAN3H-PRAZOSINN-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide19.9526Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90939Alpha1BCHO cellsHUMAN3H-PRAZOSINN-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide239.883Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90940Alpha1DCHO cellsHUMAN3H-PRAZOSINN-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide19.0546Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909415-HT1AHeLaHUMAN3H-8-OH-DPATN-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide79.4328Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90942Alpha1ACHO cellsHUMAN3H-PRAZOSINN-tert-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide12.5893Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90943Alpha1BCHO cellsHUMAN3H-PRAZOSINN-tert-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide128.825Franchini S et al 2014Jan 15, 2025Jan 28, 2025
90944Alpha1DCHO cellsHUMAN3H-PRAZOSINN-tert-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide35.4813Franchini S et al 2014Jan 15, 2025Jan 28, 2025
909455-HT1AHeLaHUMAN3H-8-OH-DPATN-tert-butyl-2-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-1,4-dioxa-8-azaspiro[4.5]decane-8-carboxamide87.0964Franchini S et al 2014Jan 15, 2025Jan 15, 2025
90946Sigma 1BRAINRAT3H-Pentazocine(+)HALOPERIDOL7Sun H et al 2016Jan 15, 2025Jan 28, 2025
90947Sigma 2PC12RAT3H-DTGHALOPERIDOL19.6Sun H et al 2016Jan 15, 2025Jan 28, 2025
90948Sigma 1BRAINRAT3H-Pentazocine(+)(S)-N-Phenyl-3-(pyrrolidin-2-ylmethoxy)isoxazole-5-carbox-amide Hydrochloride130Sun H et al 2016Jan 15, 2025Jan 28, 2025
90949Sigma 1BRAINRAT3H-Pentazocine(+)(S)-Indolin-1-yl(3-(pyrrolidin-2-ylmethoxy)isoxazol-5-yl)-methanone Hydrochloride13.9Sun H et al 2016Jan 15, 2025Jan 28, 2025
90950Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((Phenylthio)methyl)-3-(pyrrolidin-2-ylmethoxy)-isoxazole Trifluoroacetate65.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90951Sigma 2PC12RAT3H-DTG(S)-5-((Phenylthio)methyl)-3-(pyrrolidin-2-ylmethoxy)-isoxazole Trifluoroacetate1033Sun H et al 2016Jan 15, 2025Jan 28, 2025
90952Sigma 1BRAINRAT3H-Pentazocine(+)(S)-(3-(Pyrrolidin-2-ylmethoxy)isoxazol-5-yl)methyl Phenyl-carbamate Trifluoroacetate299Sun H et al 2016Jan 15, 2025Jan 28, 2025
90953Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((2-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride6Sun H et al 2016Jan 15, 2025Jan 28, 2025
90954Sigma 2PC12RAT3H-DTG(S)-5-((2-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride396Sun H et al 2016Jan 15, 2025Jan 28, 2025
90955Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((3-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride1.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90956Sigma 2PC12RAT3H-DTG(S)-5-((3-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride277Sun H et al 2016Jan 15, 2025Jan 28, 2025
90957Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((4-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride4.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90958Sigma 2PC12RAT3H-DTG(S)-5-((4-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride471Sun H et al 2016Jan 15, 2025Jan 28, 2025
90959Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((2-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride2.7Sun H et al 2016Jan 15, 2025Jan 28, 2025
90960Sigma 2PC12RAT3H-DTG(S)-5-((2-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride165Sun H et al 2016Jan 15, 2025Jan 28, 2025
90961Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((3-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate2.6Sun H et al 2016Jan 15, 2025Jan 28, 2025
90962Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((4-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride13Sun H et al 2016Jan 15, 2025Jan 28, 2025
90963Sigma 2PC12RAT3H-DTG(S)-5-((4-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride139Sun H et al 2016Jan 15, 2025Jan 28, 2025
90964Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((3-Bromophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride3.2Sun H et al 2016Jan 15, 2025Jan 28, 2025
90965Sigma 2PC12RAT3H-DTG(S)-5-((3-Bromophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride85.9Sun H et al 2016Jan 15, 2025Jan 28, 2025
90966Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((4-Bromophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride18.3Sun H et al 2016Jan 15, 2025Jan 28, 2025
90967Sigma 2PC12RAT3H-DTG(S)-5-((4-Bromophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride137Sun H et al 2016Jan 15, 2025Jan 28, 2025
90968Sigma 1BRAINRAT3H-Pentazocine(+)(S)-3-(Pyrrolidin-2-ylmethoxy)-5-((3-(trifluoromethyl)-phenoxy)methyl)isoxazole Trifluoroacetate6.6Sun H et al 2016Jan 15, 2025Jan 28, 2025
90969Sigma 2PC12RAT3H-DTG(S)-3-(Pyrrolidin-2-ylmethoxy)-5-((3-(trifluoromethyl)-phenoxy)methyl)isoxazole Trifluoroacetate88Sun H et al 2016Jan 15, 2025Jan 28, 2025
90970Sigma 1BRAINRAT3H-Pentazocine(+)(S)-3-(Pyrrolidin-2-ylmethoxy)-5-((4-(trifluoromethyl)-phenoxy)methyl)isoxazole Trifluoroacetate13.3Sun H et al 2016Jan 15, 2025Jan 28, 2025
90971Sigma 2PC12RAT3H-DTG(S)-3-(Pyrrolidin-2-ylmethoxy)-5-((4-(trifluoromethyl)-phenoxy)methyl)isoxazole Trifluoroacetate91.7Sun H et al 2016Jan 15, 2025Jan 28, 2025
90972Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((3-Methoxyphenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride31.1Sun H et al 2016Jan 15, 2025Jan 28, 2025
90973Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((4-Methoxyphenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride210Sun H et al 2016Jan 15, 2025Jan 28, 2025
90974Sigma 2PC12RAT3H-DTG(S)-5-((4-Methoxyphenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride675Sun H et al 2016Jan 15, 2025Jan 28, 2025
90975Sigma 1BRAINRAT3H-Pentazocine(+)(S)-3-(Pyrrolidin-2-ylmethoxy)-5-((m-tolyloxy)methyl)-isoxazole Hydrochloride4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90976Sigma 2PC12RAT3H-DTG(S)-3-(Pyrrolidin-2-ylmethoxy)-5-((m-tolyloxy)methyl)-isoxazole Hydrochloride341Sun H et al 2016Jan 15, 2025Jan 28, 2025
90977Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((Naphthalen-2-yloxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate36.6Sun H et al 2016Jan 15, 2025Jan 28, 2025
90978Sigma 2PC12RAT3H-DTG(S)-5-((Naphthalen-2-yloxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate153Sun H et al 2016Jan 15, 2025Jan 28, 2025
90979Sigma 1BRAINRAT3H-Pentazocine(+)(R)-5-(Phenoxymethyl)-3-(pyrrolidin-2-ylmethoxy)isoxazoleHydrochloride37.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90980Sigma 2PC12RAT3H-DTG(R)-5-(Phenoxymethyl)-3-(pyrrolidin-2-ylmethoxy)isoxazoleHydrochloride508Sun H et al 2016Jan 15, 2025Jan 28, 2025
90981Sigma 1BRAINRAT3H-Pentazocine(+)5-(Phenoxymethyl)-3-(piperidin-4-ylmethoxy)isoxazole Tri-fluoroacetate356Sun H et al 2016Jan 15, 2025Jan 28, 2025
90982Sigma 2PC12RAT3H-DTG5-(Phenoxymethyl)-3-(piperidin-4-ylmethoxy)isoxazole Tri-fluoroacetate284Sun H et al 2016Jan 15, 2025Jan 28, 2025
90983Sigma 1BRAINRAT3H-Pentazocine(+)2-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hy-drochloride63.9Sun H et al 2016Jan 15, 2025Jan 28, 2025
90984Sigma 1BRAINRAT3H-Pentazocine(+)3-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)propan-1-amineHydrochloride2312Sun H et al 2016Jan 15, 2025Jan 28, 2025
90985Sigma 1BRAINRAT3H-Pentazocine(+)N-Methyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride80.8Sun H et al 2016Jan 15, 2025Jan 28, 2025
90986Sigma 1BRAINRAT3H-Pentazocine(+)N-Ethyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride3.7Sun H et al 2016Jan 15, 2025Jan 28, 2025
90987Sigma 2PC12RAT3H-DTGN-Ethyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride987Sun H et al 2016Jan 15, 2025Jan 28, 2025
90988Sigma 1BRAINRAT3H-Pentazocine(+)(S)-3-((1-Methylpyrrolidin-2-yl)methoxy)-5-(phenoxymethyl)isoxazole Hydrochloride3.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90989Sigma 2PC12RAT3H-DTG(S)-3-((1-Methylpyrrolidin-2-yl)methoxy)-5-(phenoxymethyl)isoxazole Hydrochloride665Sun H et al 2016Jan 15, 2025Jan 28, 2025
90990Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((3-Fluorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride0.7Sun H et al 2016Jan 15, 2025Jan 28, 2025
90991Sigma 2PC12RAT3H-DTG(S)-5-((3-Fluorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride687Sun H et al 2016Jan 15, 2025Jan 28, 2025
90992Sigma 1BRAINRAT3H-Pentazocine(+)(S)-5-((3-Chlorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride1.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90993Sigma 2PC12RAT3H-DTG(S)-5-((3-Chlorophenoxy)methyl)-3-((1-methylpyrrolidin-2-yl)methoxy)isoxazole Hydrochloride371Sun H et al 2016Jan 15, 2025Jan 28, 2025
90994Sigma 1BRAINRAT3H-Pentazocine(+)(R)-3-((1-Methylpyrrolidin-2-yl)methoxy)-5-(phenoxymethyl)isoxazole Hydrochloride23.1Sun H et al 2016Jan 15, 2025Jan 28, 2025
90995Sigma 2PC12RAT3H-DTG(R)-3-((1-Methylpyrrolidin-2-yl)methoxy)-5-(phenoxymethyl)isoxazole Hydrochloride411Sun H et al 2016Jan 15, 2025Jan 28, 2025
90996Sigma 1BRAINRAT3H-Pentazocine(+)3-((1-Methylpiperidin-4-yl)methoxy)-5-(phenoxymethyl)-isoxazole Hydrochloride96.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90997Sigma 2PC12RAT3H-DTG3-((1-Methylpiperidin-4-yl)methoxy)-5-(phenoxymethyl)-isoxazole Hydrochloride216Sun H et al 2016Jan 15, 2025Jan 28, 2025
90998Sigma 1BRAINRAT3H-Pentazocine(+)N-Ethyl-N-methyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)-ethan-1-amine Hydrochloride18.4Sun H et al 2016Jan 15, 2025Jan 28, 2025
90999Sigma 2PC12RAT3H-DTGN-Ethyl-N-methyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)-ethan-1-amine Hydrochloride820Sun H et al 2016Jan 15, 2025Jan 28, 2025
91000Sigma 1BRAINRAT3H-Pentazocine(+)N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclobutanamine Hydrochloride1.8Sun H et al 2016Jan 15, 2025Jan 28, 2025
91001Sigma 2PC12RAT3H-DTGN-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclobutanamine Hydrochloride307Sun H et al 2016Jan 15, 2025Jan 28, 2025
91002Sigma 1BRAINRAT3H-Pentazocine(+)N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclopentanamine Hydrochloride0.5Sun H et al 2016Jan 15, 2025Jan 28, 2025
91003Sigma 2PC12HUMAN3H-DTGN-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclopentanamine Hydrochloride73.7Sun H et al 2016Jan 15, 2025Jan 28, 2025
91004Sigma 1BRAINRAT3H-Pentazocine(+)N-(Cyclopropylmethyl)-N-methyl-2-((5-(phenoxymethyl)-isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride0.8Sun H et al 2016Jan 15, 2025Jan 28, 2025
91005Sigma 2PC12RAT3H-DTGN-(Cyclopropylmethyl)-N-methyl-2-((5-(phenoxymethyl)-isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride225Sun H et al 2016Jan 15, 2025Jan 28, 2025
91006Sigma 1BRAINRAT3H-Pentazocine(+)N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclohexanamine Hydrochloride0.3Sun H et al 2016Jan 15, 2025Jan 28, 2025
91007Sigma 2BRAINRAT3H-DTGN-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclohexanamine Hydrochloride18.7Sun H et al 2016Jan 15, 2025Jan 28, 2025
91008Sigma 1BRAINRAT3H-Pentazocine(+)N-(Cyclopropylmethyl)-2-((5-((3-fluorophenoxy)methyl)-isoxazol-3-yl)oxy)-N-methylethan-1-amine Hydrochloride0.9Sun H et al 2016Jan 15, 2025Jan 28, 2025
91009Sigma 2PC12RAT3H-DTGN-(Cyclopropylmethyl)-2-((5-((3-fluorophenoxy)methyl)-isoxazol-3-yl)oxy)-N-methylethan-1-amine Hydrochloride314Sun H et al 2016Jan 15, 2025Jan 28, 2025
91010Sigma 1BRAINRAT3H-Pentazocine(+)2-((5-((3-Chlorophenoxy)methyl)isoxazol-3-yl)oxy)-N-(cyclo-propylmethyl)-N-methylethan-1-amine Hydrochloride1.1Sun H et al 2016Jan 15, 2025Jan 28, 2025
91011Sigma 2PC12RAT3H-DTG2-((5-((3-Chlorophenoxy)methyl)isoxazol-3-yl)oxy)-N-(cyclo-propylmethyl)-N-methylethan-1-amine Hydrochloride123Sun H et al 2016Jan 15, 2025Jan 28, 2025
91012Sigma 2PC12RAT3H-DTGN-(2-((5-((3-Fluorophenoxy)methyl)isoxazol-3-yl)oxy)ethyl)-N-methylcyclohexanamine Hydrochloride24.5Sun H et al 2016Jan 15, 2025Jan 28, 2025
91013Sigma 1BRAINRAT3H-Pentazocine(+)N-(2-((5-((3-Fluorophenoxy)methyl)isoxazol-3-yl)oxy)ethyl)-N-methylcyclohexanamine Hydrochloride0.5Sun H et al 2016Jan 15, 2025Jan 28, 2025
91014Sigma 1BRAINRAT3H-Pentazocine(+)N-(2-((5-((3-Chlorophenoxy)methyl)isoxazol-3-yl)oxy)ethyl)-N-methylcyclohexanamine Hydrochloride0.5Sun H et al 2016Jan 15, 2025Jan 28, 2025
91015Sigma 2PC12RAT3H-DTGN-(2-((5-((3-Chlorophenoxy)methyl)isoxazol-3-yl)oxy)ethyl)-N-methylcyclohexanamine Hydrochloride15.1Sun H et al 2016Jan 15, 2025Jan 28, 2025
91016Sigma 1BRAINRAT3H-Pentazocine(+)4-(2-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-morpholine Hydrochloride403Sun H et al 2016Jan 15, 2025Jan 28, 2025
91017Sigma 1BRAINRAT3H-Pentazocine(+)5-(Phenoxymethyl)-3-(piperazin-1-yl)isoxazole Hydrochlor-ide5.3Sun H et al 2016Jan 15, 2025Jan 28, 2025
91018Sigma 2PC12RAT3H-DTG5-(Phenoxymethyl)-3-(piperazin-1-yl)isoxazole Hydrochlor-ide221Sun H et al 2016Jan 15, 2025Jan 28, 2025
91019Sigma 1BRAINRAT3H-Pentazocine(+)N-(Cyclopropylmethyl)-2-((5-((3-fluorophenoxy)methyl)-isoxazol-3-yl)oxy)-N-methylethan-1-amine Hydrochloride36.5Sun H et al 2016Jan 15, 2025Jan 28, 2025
91020Sigma 2PC12RAT3H-DTGN-(Cyclopropylmethyl)-2-((5-((3-fluorophenoxy)methyl)-isoxazol-3-yl)oxy)-N-methylethan-1-amine Hydrochloride687Sun H et al 2016Jan 15, 2025Jan 28, 2025
91021Sigma 1BRAINRAT3H-Pentazocine(+)3-(4-Methylpiperazin-1-yl)-5-(phenoxymethyl)isoxazole Hy-drochloride63.9Sun H et al 2016Jan 15, 2025Jan 28, 2025
91022Sigma 2PC12RAT3H-DTG3-(4-Methylpiperazin-1-yl)-5-(phenoxymethyl)isoxazole Hy-drochloride2202Sun H et al 2016Jan 15, 2025Jan 28, 2025
91023Sigma 1BRAINRAT3H-Pentazocine(+)Phenyl (S)-3-(Pyrrolidin-2-ylmethoxy)isoxazole-5-carboxy-late Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91024Sigma 2PC12RAT3H-DTGPhenyl (S)-3-(Pyrrolidin-2-ylmethoxy)isoxazole-5-carboxy-late Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91025Sigma 2PC12RAT3H-DTG(S)-N-Phenyl-3-(pyrrolidin-2-ylmethoxy)isoxazole-5-carbox-amide Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91026Sigma 2PC12RAT3H-DTG(S)-Indolin-1-yl(3-(pyrrolidin-2-ylmethoxy)isoxazol-5-yl)-methanone Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91027Sigma 2PC12RAT3H-DTG(S)-(3-(Pyrrolidin-2-ylmethoxy)isoxazol-5-yl)methyl Phenyl-carbamate Trifluoroacetate>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91028Sigma 2PC12RAT3H-DTG(S)-5-((3-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Trifluoroacetate>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91029Sigma 2PC12RAT3H-DTG(S)-5-((3-Methoxyphenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91030Sigma 2PC12RAT3H-DTG2-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hy-drochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91031Sigma 2PC12RAT3H-DTG3-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)propan-1-amineHydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91032Sigma 2PC12RAT3H-DTGN-Methyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91033Sigma 1BRAINRAT3H-Pentazocine(+)N,N-Dimethyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)-ethan-1-amine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91034Sigma 2PC12RAT3H-DTGN,N-Dimethyl-2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)-ethan-1-amine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91035Sigma 2PC12RAT3H-DTG4-(2-((5-(Phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-morpholine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91036Sigma 1BRAINRAT3H-Pentazocine(+)4-(5-(Phenoxymethyl)isoxazol-3-yl)morpholine Hydrochlor-ide>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91037Sigma 2PC12RAT3H-DTG4-(5-(Phenoxymethyl)isoxazol-3-yl)morpholine Hydrochlor-ide>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91038Sigma 1BRAINRAT3H-Pentazocine(+)5-(Phenoxymethyl)-3-(piperidin-1-yl)isoxazole Hydrochlor-ide>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91039Sigma 2PC12RAT3H-DTG5-(Phenoxymethyl)-3-(piperidin-1-yl)isoxazole Hydrochlor-ide>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91040DATCLONEDHUMAN3H-WIN 35,428(S)-5-((2-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 15, 2025
91041NETCLONEDHUMAN3H-Nisoxetine(S)-5-((2-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride1082Sun H et al 2016Jan 15, 2025Jan 15, 2025
91042SERTCLONEDHUMAN3H-CITALOPRAM(S)-5-((2-Fluorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91043DATCLONEDHUMAN3H-WIN 35,428(S)-5-((2-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 15, 2025
91044NETCLONEDHUMAN3H-Nisoxetine(S)-5-((2-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride2109Sun H et al 2016Jan 15, 2025Jan 15, 2025
91045SERTCLONEDHUMAN3H-CITALOPRAM(S)-5-((2-Chlorophenoxy)methyl)-3-(pyrrolidin-2-ylmethoxy)isoxazole Hydrochloride2946Sun H et al 2016Jan 15, 2025Jan 28, 2025
91046DATCLONEDHUMAN3H-WIN 35,428N-(Cyclopropylmethyl)-N-methyl-2-((5-(phenoxymethyl)-isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 15, 2025
91047NETCLONEDHUMAN3H-NisoxetineN-(Cyclopropylmethyl)-N-methyl-2-((5-(phenoxymethyl)-isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 15, 2025
91048SERTCLONEDHUMAN3H-CITALOPRAMN-(Cyclopropylmethyl)-N-methyl-2-((5-(phenoxymethyl)-isoxazol-3-yl)oxy)ethan-1-amine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91049DATCLONEDHUMAN3H-WIN 35,428N-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclohexanamine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 15, 2025
91050NETCLONEDHUMAN3H-NisoxetineN-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclohexanamine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 15, 2025
91051SERTCLONEDHUMAN3H-CITALOPRAMN-Methyl-N-(2-((5-(phenoxymethyl)isoxazol-3-yl)oxy)ethyl)-cyclohexanamine Hydrochloride>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91052DATCLONEDHUMAN3H-WIN 35,4285-(Phenoxymethyl)-3-(piperazin-1-yl)isoxazole Hydrochlor-ide497Sun H et al 2016Jan 15, 2025Jan 15, 2025
91053NETCLONEDHUMAN3H-Nisoxetine5-(Phenoxymethyl)-3-(piperazin-1-yl)isoxazole Hydrochlor-ide163Sun H et al 2016Jan 15, 2025Jan 15, 2025
91054SERTCLONEDHUMAN3H-CITALOPRAM5-(Phenoxymethyl)-3-(piperazin-1-yl)isoxazole Hydrochlor-ide>10000Sun H et al 2016Jan 15, 2025Jan 28, 2025
91055A1CHO cellsHUMAN3H-CCPA4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91056A2ACHO cellsHUMAN3H-NECA4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine9100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91057A3CHO cellsHUMAN3H-HEMADO4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91058A1CHO cellsHUMAN3H-CCPA4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine9000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91059A2ACHO cellsHUMAN3H-NECA4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine3300Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91060A3CHO cellsHUMAN3H-HEMADO4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91061A1CHO cellsHUMAN3H-CCPA4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91062A2ACHO cellsHUMAN3H-NECA4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine4100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91063A3CHO cellsHUMAN3H-HEMADO4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91064A1CHO cellsHUMAN3H-CCPA4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine4300Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91065A2ACHO cellsHUMAN3H-NECA4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine3700Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91066A3CHO cellsHUMAN3H-HEMADO4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-amine>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91067A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91068A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91069A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91070A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91071A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91072A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91073A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91074A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91075A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91076A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91077A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91078A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91079A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91080A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide4600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91081A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91082A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide3400Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91083A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide1600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91084A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91085A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91086A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide2700Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91087A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91088A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide4100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91089A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide1100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91090A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91091A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91092A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide3500Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91093A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91094A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91095A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide2200Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91096A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide5900Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91097A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91098A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91099A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide6600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91100A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91101A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide2100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91102A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide5000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91103A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl) benzamide3800Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91104A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl) benzamide3100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91105A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl) benzamide8600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91106A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide2700Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91107A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide2060Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91108A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-fluorobenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91109A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91110A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91111A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-(trifluoromethyl)benzamide2800Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91112A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91113A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide9900Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91114A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-4-methylbenzamide1500Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91115A1CHO cellsHUMAN3H-CCPAN-Benzoyl-N-(4-chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91116A2ACHO cellsHUMAN3H-NECAN-Benzoyl-N-(4-chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91117A3CHO cellsHUMAN3H-HEMADON-Benzoyl-N-(4-chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide7100Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91118A1CHO cellsHUMAN3H-CCPAN-Benzoyl-N-(4-chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide7900Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91119A2ACHO cellsHUMAN3H-NECAN-Benzoyl-N-(4-chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide800Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91120A3CHO cellsHUMAN3H-HEMADON-Benzoyl-N-(4-chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide6700Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91121A1CHO cellsHUMAN3H-CCPAN-Benzoyl-N-(4-chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91122A2ACHO cellsHUMAN3H-NECAN-Benzoyl-N-(4-chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91123A3CHO cellsHUMAN3H-HEMADON-Benzoyl-N-(4-chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide6500Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91124A1CHO cellsHUMAN3H-CCPAN-Benzoyl-N-(4-chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91125A2ACHO cellsHUMAN3H-NECAN-Benzoyl-N-(4-chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide5400Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91126A3CHO cellsHUMAN3H-HEMADON-Benzoyl-N-(4-chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)benzamide2900Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91127A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91128A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91129A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-methyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide6600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91130A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide1900Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91131A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide4700Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91132A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-isopropyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91133A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91134A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91135A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91136A1CHO cellsHUMAN3H-CCPAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide6500Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91137A2ACHO cellsHUMAN3H-NECAN-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide8600Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91138A3CHO cellsHUMAN3H-HEMADON-(4-Chloro-2-phenethyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl)-2-phenylacetamide>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91139A1CHO cellsHUMAN3H-CCPAEthyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91140A2AH9HUMAN3H-NECAEthyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91141A3CHO cellsHUMAN3H-HEMADOEthyl-2-neopentyl-6-(4-(trifluoromethyl)benzamido)-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate1300Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91142A1CHO cellsHUMAN3H-CCPAEthyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91143A2ACHO cellsHUMAN3H-NECAEthyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate>10000Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91144A3CHO cellsHUMAN3H-HEMADOEthyl-6-(4-methylbenzamido)-2-neopentyl-2H-pyrazolo[3,4-d]pyrimidine-4-carboxylate900Venkatesan G et al 2014Jan 15, 2025Jan 15, 2025
91145A1CLONEDHUMAN3H-DPCPXN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91146A2ACLONEDHUMAN3H-CGS-21680N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide3310Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91147A3CLONEDHUMAN125I-AB-MECAN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91148A3CLONEDHUMAN125I-AB-MECA3-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91149A2ACLONEDHUMAN3H-CGS-216803-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91150A1CLONEDHUMAN3H-DPCPX3-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide3460Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91151A1CLONEDHUMAN3H-DPCPX2-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methylsulfanyl]-N-(2-methylphenyl)acetamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91152A2ACLONEDHUMAN3H-CGS-216802-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methylsulfanyl]-N-(2-methylphenyl)acetamide2360Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91153A3CLONEDHUMAN125I-AB-MECA2-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methylsulfanyl]-N-(2-methylphenyl)acetamide4860Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91154A3CLONEDHUMAN125I-AB-MECAN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide9060Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91155A2ACLONEDHUMAN3H-CGS-21680N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91156A3CLONEDHUMAN125I-AB-MECAN-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91157A3CLONEDHUMAN125I-AB-MECA4-methoxy-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide2780Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91158A2ACLONEDHUMAN3H-CGS-216804-methoxy-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide3655Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91159A1CLONEDHUMAN3H-DPCPX4-methoxy-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91160A1CLONEDHUMAN3H-DPCPX2,6-diphenyl-8-propan-2-yl-7H-purine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91161A2ACLONEDHUMAN3H-CGS-216802,6-diphenyl-8-propan-2-yl-7H-purine6540Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91162A3CLONEDHUMAN125I-AB-MECA2,6-diphenyl-8-propan-2-yl-7H-purine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91163A3CLONEDHUMAN125I-AB-MECA2-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine9330Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91164A2ACLONEDHUMAN3H-CGS-216802-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91165A1CLONEDHUMAN3H-DPCPX2-(3-fluorophenyl)pyrazolo[3,4-c]quinolin-4-amine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91166A1CLONEDHUMAN3H-DPCPXN-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91167A2ACLONEDHUMAN3H-CGS21680N-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91168A3CLONEDHUMAN125I-AB-MECAN-(4-pyridin-2-yl-1,3-thiazol-2-yl)cyclopentanecarboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91169A3CLONEDHUMAN125I-AB-MECA2-amino-6-(2-ethoxyphenyl)-N-(pyridin-2-ylmethyl)pyrimidine-4-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91170A2ACLONEDHUMAN3H-CGS216802-amino-6-(2-ethoxyphenyl)-N-(pyridin-2-ylmethyl)pyrimidine-4-carboxamide740Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91171A1CLONEDHUMAN3H-DPCPX2-amino-6-(2-ethoxyphenyl)-N-(pyridin-2-ylmethyl)pyrimidine-4-carboxamide400Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91172A1CLONEDHUMAN3H-DPCPXN-(4,6-dithiophen-2-ylpyrimidin-2-yl)propanamide3430Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91173A2ACLONEDHUMAN3H-CGS21680N-(4,6-dithiophen-2-ylpyrimidin-2-yl)propanamide2130Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91174A3CLONEDHUMAN125I-AB-MECAN-(4,6-dithiophen-2-ylpyrimidin-2-yl)propanamide1760Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91175A3CLONEDHUMAN125I-AB-MECA3-(oxolan-2-ylmethyl)-8-phenyl-1-propyl-7H-purine-2,6-dione>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91176A2ACLONEDHUMAN3H-CGS216803-(oxolan-2-ylmethyl)-8-phenyl-1-propyl-7H-purine-2,6-dione6660Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91177A1CLONEDHUMAN3H-DPCPX3-(oxolan-2-ylmethyl)-8-phenyl-1-propyl-7H-purine-2,6-dione3340Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91178A1CLONEDHUMAN3H-DPCPX3-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91179A2ACLONEDHUMAN3H-CGS216803-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide3560Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91180A3CLONEDHUMAN125I-AB-MECA3-chloro-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzamide1520Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91181A3CLONEDHT29125I-AB-MECA3-[(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)carbamoyl]benzenesulfonyl fluoride205Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91182A2ACLONEDHUMAN3H-CGS216803-[(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)carbamoyl]benzenesulfonyl fluoride1340Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91183A1CLONEDHUMAN3H-DPCPX3-[(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)carbamoyl]benzenesulfonyl fluoride980Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91184A1CLONEDHUMAN3H-DPCPX1-[2-(diethylamino)quinazolin-4-yl]-3-phenylurea>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91185A2ACLONEDHUMAN3H-CGS216801-[2-(diethylamino)quinazolin-4-yl]-3-phenylurea9300Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91186A3CLONEDHUMAN125I-AB-MECA1-[2-(diethylamino)quinazolin-4-yl]-3-phenylurea>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91187A3CLONEDHUMAN125I-AB-MECA3,4-dichloro-N-(4-phenyl-1,3-thiazol-2-yl)benzamide70Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91188A2ACLONEDHUMAN3H-CGS216803,4-dichloro-N-(4-phenyl-1,3-thiazol-2-yl)benzamide3780Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91189A1CLONEDHUMAN3H-DPCPX3,4-dichloro-N-(4-phenyl-1,3-thiazol-2-yl)benzamide1220Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91190A1CLONEDHUMAN3H-DPCPX6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-N-(4-fluorophenyl)-1,3,5-triazine-2,4-diamine>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91191A2ACLONEDHUMAN3H-CGS216806-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-N-(4-fluorophenyl)-1,3,5-triazine-2,4-diamine6140Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91192A3CLONEDHUMAN125I-AB-MECA6-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-2-N-(4-fluorophenyl)-1,3,5-triazine-2,4-diamine40Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91193A3CLONEDHUMAN125I-AB-MECA5-ethyl-1-hydroxy-3-(3-prop-2-enoxyphenyl)imidazo[5,1-a]phthalazin-6-one550Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91194A2ACLONEDHUMAN3H-CGS216805-ethyl-1-hydroxy-3-(3-prop-2-enoxyphenyl)imidazo[5,1-a]phthalazin-6-one1450Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91195A1CLONEDHUMAN3H-DPCPX5-ethyl-1-hydroxy-3-(3-prop-2-enoxyphenyl)imidazo[5,1-a]phthalazin-6-one2930Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91196A1CLONEDHUMAN3H-DPCPXN-(5-methyl-1,2-oxazol-3-yl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,2-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide3940Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91197A2ACLONEDHUMAN3H-CGS21680N-(5-methyl-1,2-oxazol-3-yl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,2-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide1370Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91198A3CLONEDHUMAN125I-AB-MECAN-(5-methyl-1,2-oxazol-3-yl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,2-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide3850Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91199A3CLONEDHUMAN125I-AB-MECAethyl 5-[(3,4-dimethoxyphenyl)methylamino]-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91200A2ACLONEDHUMAN3H-CGS21680ethyl 5-[(3,4-dimethoxyphenyl)methylamino]-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91201A1CLONEDHUMAN3H-DPCPXethyl 5-[(3,4-dimethoxyphenyl)methylamino]-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91202A1CLONEDHUMAN3H-DPCPXethyl 2-[2-(4-chlorophenyl)-5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91203A2ACLONEDHUMAN3H-CGS21680ethyl 2-[2-(4-chlorophenyl)-5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91204A1CLONEDHUMAN125I-AB-MECAethyl 2-[2-(4-chlorophenyl)-5-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91205A1CLONEDHUMAN125I-AB-MECApropan-2-yl (2S)-2-[(5-cyano-6-oxo-4-phenyl-1H-pyrimidin-2-yl)sulfanyl]propanoate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91206A2ACLONEDHUMAN3H-CGS21680propan-2-yl (2S)-2-[(5-cyano-6-oxo-4-phenyl-1H-pyrimidin-2-yl)sulfanyl]propanoate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91207A1CLONEDHUMAN3H-DPCPXpropan-2-yl (2S)-2-[(5-cyano-6-oxo-4-phenyl-1H-pyrimidin-2-yl)sulfanyl]propanoate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91208A1CLONEDHUMAN3H-DPCPXethyl 2-[5-methyl-2-(4-methylphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91209A2ACLONEDHUMAN3H-CGS21680ethyl 2-[5-methyl-2-(4-methylphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91210A3CLONEDHUMAN125I-AB-MECAethyl 2-[5-methyl-2-(4-methylphenyl)-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-6-yl]acetate>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91211A3CLONEDHUMAN125I-AB-MECA2-[4-(1H-benzimidazol-2-ylamino)-6-methyl-1,3,5-triazin-2-yl]phenol>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91212A2ACLONEDHUMAN3H-CGS216802-[4-(1H-benzimidazol-2-ylamino)-6-methyl-1,3,5-triazin-2-yl]phenol>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91213A1CLONEDHUMAN3H-DPCPX2-[4-(1H-benzimidazol-2-ylamino)-6-methyl-1,3,5-triazin-2-yl]phenol>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91214A1CLONEDHUMAN3H-DPCPX1-(1-methylpyrrol-2-yl)-2-(3H-[1,2,4]triazolo[4,3-a]benzimidazol-1-ylsulfanyl)ethanone>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91215A2ACLONEDHUMAN3H-CGS216801-(1-methylpyrrol-2-yl)-2-(3H-[1,2,4]triazolo[4,3-a]benzimidazol-1-ylsulfanyl)ethanone>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91216A3CLONEDHUMAN125I-AB-MECA1-(1-methylpyrrol-2-yl)-2-(3H-[1,2,4]triazolo[4,3-a]benzimidazol-1-ylsulfanyl)ethanone>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91217A3CLONEDHUMAN125I-AB-MECAN-[7-[(1S)-1-(3-methoxyphenoxy)ethyl]-1H-[1,2,4]triazolo[1,5-a]pyrimidin-8-ium-2-yl]-N,N-dimethylmethanimidamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91218A2ACLONEDHUMAN3H-CGS21680N-[7-[(1S)-1-(3-methoxyphenoxy)ethyl]-1H-[1,2,4]triazolo[1,5-a]pyrimidin-8-ium-2-yl]-N,N-dimethylmethanimidamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91219A1CLONEDHUMAN3H-DPCPXN-[7-[(1S)-1-(3-methoxyphenoxy)ethyl]-1H-[1,2,4]triazolo[1,5-a]pyrimidin-8-ium-2-yl]-N,N-dimethylmethanimidamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91220A1CLONEDHUMAN3H-DPCPX5-cyano-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-6-methylpyridine-2-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91221A2ACLONEDHUMAN3H-CGS216805-cyano-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-6-methylpyridine-2-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91222A3CLONEDHUMAN125I-AB-MECA5-cyano-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-6-methylpyridine-2-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91223A3CLONEDHUMAN125I-AB-MECA(E)-3-(3-cyanophenyl)-N-methyl-N-[(4-oxo-3H-quinazolin-2-yl)methyl]prop-2-enamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91224A2ACLONEDHUMAN3H-CGS21680(E)-3-(3-cyanophenyl)-N-methyl-N-[(4-oxo-3H-quinazolin-2-yl)methyl]prop-2-enamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91225A1CLONEDHUMAN3H-DPCPX(E)-3-(3-cyanophenyl)-N-methyl-N-[(4-oxo-3H-quinazolin-2-yl)methyl]prop-2-enamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91226A1CLONEDHUMAN3H-DPCPX1-(2-phenoxyphenyl)-3-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]urea>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91227A2ACLONEDHUMAN3H-CGS216801-(2-phenoxyphenyl)-3-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]urea>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91228A3CLONEDHUMAN125I-AB-MECA1-(2-phenoxyphenyl)-3-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]urea>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91229A3CLONEDHUMAN125I-AB-MECA2-[(Z)-1-chloro-2-(3-hydroxy-4-methoxyphenyl)ethenyl]-8-methyl-3H-quinazolin-4-one>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91230A2ACLONEDHUMAN3H-CGS216802-[(Z)-1-chloro-2-(3-hydroxy-4-methoxyphenyl)ethenyl]-8-methyl-3H-quinazolin-4-one>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91231A1CLONEDHUMAN3H-DPCPX2-[(Z)-1-chloro-2-(3-hydroxy-4-methoxyphenyl)ethenyl]-8-methyl-3H-quinazolin-4-one>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91232A1CLONEDHUMAN3H-DPCPXN-(1H-benzimidazol-2-yl)-3-(4-oxo-3H-quinazolin-2-yl)propanamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91233A2ACLONEDHUMAN3H-CGS21680N-(1H-benzimidazol-2-yl)-3-(4-oxo-3H-quinazolin-2-yl)propanamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91234A3CLONEDHUMAN125I-AB-MECAN-(1H-benzimidazol-2-yl)-3-(4-oxo-3H-quinazolin-2-yl)propanamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91235A3CLONEDHUMAN125I-AB-MECA4-oxo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)chromene-2-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91236A2ACLONEDHUMAN3H-CGS216804-oxo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)chromene-2-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91237A1CLONEDHUMAN3H-DPCPX4-oxo-N-(4-pyridin-2-yl-1,3-thiazol-2-yl)chromene-2-carboxamide>10000Kolb P et al 2012Jan 15, 2025Jan 15, 2025
91238MORCLONEDHUMAN3H-NALOXONE17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan28.26Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91239DORCLONEDHUMAN3H-Diprenorphine17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan9860Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91240KORCLONEDHUMAN3H-Diprenorphine17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan20.11Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91241KORCLONEDHUMAN3H-Diprenorphine17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan3.09Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91242DORCLONEDHUMAN3H-Diprenorphine17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan603.8Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91243MORCLONEDHUMAN3H-NALOXONE17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan2.85Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91244NETCLONEDHUMAN3H-Nisoxetine17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91245PBRKidney membranesRAT3H-PK1119517-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91246SERTCLONEDHUMAN3H-CITALOPRAM17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91247Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91248Sigma 2PC12RAT3H-DTG17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91249H1CLONEDHUMAN3H-PYRILAMINE17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
912505-HT1DCLONEDHUMAN125I-aminopotentidine17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91251H3CLONEDHUMAN3H-Alpha-methylhistamine17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91252H4CLONEDHUMAN3H-Histamine17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91253M1CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91254M2CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91255M3CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91256M4CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91257D1CLONEDHUMAN3H-SCH2339017-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91258D5CLONEDHUMAN3H-SCH2339017-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91259D2CLONEDHUMAN3H-N-Methylspiperone17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91260D3CLONEDHUMAN3H-N-Methylspiperone17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91261D4CLONEDHUMAN3H-N-Methylspiperone17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91262DATCLONEDHUMAN3H-WIN 35,42817-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91263KORCORTICAL MEMBRANESRAT3H-MUSCIMOL17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 27, 2025
912645-HT1ACLONEDHUMAN3H-WAY10063517-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912655-HT1BCLONEDHUMAN3H-5-CT17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912665-HT1DCLONEDHUMAN3H-5-CT17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912675-HT1ECLONEDHUMAN3H-5-HT17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912685-HT2ACLONEDHUMAN3H-KETANSERIN17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912695-HT2BCLONEDHUMAN3H-LSD17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912705-HT2CCLONEDHUMAN3H-MESULERGINE17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912715-HT3CLONEDHUMAN3H-GR-6563017-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
912725-HT7CLONEDHUMAN3H-LSD17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91273Alpha1ACLONEDHUMAN3H-PRAZOSIN17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91274Alpha1BCLONEDHUMAN3H-PRAZOSIN17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91275Alpha1DCLONEDHUMAN3H-PRAZOSIN17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91276Alpha2ACLONEDHUMAN3H-RAUWOLSCINE17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91277Alpha2BCLONEDHUMAN3H-RAUWOLSCINE17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91278Alpha2CCLONEDHUMAN3H-RAUWOLSCINE17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91279Beta 1CLONEDHUMAN125I-Pindolol17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91280Beta3CLONEDHUMAN125I-Pindolol17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91281BZPCORTICAL MEMBRANESRATFNZ17-Cyclopropylmethyl-3,14β-dihydroxy-4,5α-epoxy-6β-{[4′-methyl-(3′-methylpy ridyl)]carboxamido} morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91282NETCLONEDHUMAN3H-Nisoxetine17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91283PBRKidney membranesRAT3H-PK1119517-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91284SERTCLONEDHUMAN3H-CITALOPRAM17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91285Sigma 1CEREBRAL CORTEXGUINEA PIG3H-Pentazocine(+)17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91286Sigma 2PC12RAT3H-DTG17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91287H1CLONEDHUMAN3H-PYRILAMINE17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
912885-HT1DCLONEDHUMAN125I-aminopotentidine17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91289H3CLONEDHUMAN3H-Alpha-methylhistamine17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91290H4CLONEDHUMAN3H-Histamine17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91291M1CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91292M2CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91293M3CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91294M4CLONEDHUMAN3H-QNB17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91295D1CLONEDHUMAN3H-SCH2339017-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91296D5CLONEDHUMAN3H-SCH2339017-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91297D2CLONEDHUMAN3H-N-Methylspiperone17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91298D3CLONEDHUMAN3H-N-Methylspiperone17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91299D4CLONEDHUMAN3H-N-Methylspiperone17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91300DATCLONEDHUMAN3H-WIN 35,42817-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91301KORCORTICAL MEMBRANESRAT3H-MUSCIMOL17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 27, 2025
913025-HT1ACLONEDHUMAN3H-WAY10063517-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913035-HT1BCLONEDHUMAN3H-5-CT17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913045-HT1DCLONEDHUMAN3H-5-CT17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913055-HT1ECLONEDHUMAN3H-5-HT17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913065-HT2ACLONEDHUMAN3H-KETANSERIN17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913075-HT2BCLONEDHUMAN3H-LSD17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913085-HT2CCLONEDHUMAN3H-MESULERGINE17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913095-HT3CLONEDHUMAN3H-GR-6563017-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
913105-HT7CLONEDHUMAN3H-LSD17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91311Alpha1ACLONEDHUMAN3H-PRAZOSIN17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91312Alpha1BCLONEDHUMAN3H-PRAZOSIN17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91313Alpha1DCLONEDHUMAN3H-PRAZOSIN17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91314Alpha2ACLONEDHUMAN3H-RAUWOLSCINE17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91315Alpha2BCLONEDHUMAN3H-RAUWOLSCINE17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91316Alpha2CCLONEDHUMAN3H-RAUWOLSCINE17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91317Beta 1CLONEDHUMAN125I-Pindolol17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 15, 2025
91318Beta3CLONEDHUMAN125I-Pindolol17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91319BZPCORTICAL MEMBRANESRATFNZ17-Cyclopropylmethyl-3,14β-dhydroxy-4,5α-epoxy-17-methyl-6β-[(4′-methylpyri dyl)acetamido] morphinan>10000Zheng Y et al 2018Jan 15, 2025Jan 28, 2025
91320CB1CLONEDHUMAN3H-CP55940Rimonabant6Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91321CB1CLONEDHUMAN3H-SR144528Rimonabant2Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91322CB2CLONEDHUMAN3H-CP55940Rimonabant702Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91323CB2CLONEDHUMAN3H-CP55940THC, delta 936Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91324CB1CLONEDHUMAN3H-SR144528THC, delta 9764Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91325CB1CLONEDHUMAN3H-CP55940THC, delta 967Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91326CB1CLONEDHUMAN3H-CP55940CP 55,9401Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91327CB1CLONEDHUMAN3H-SR144528CP 55,94031Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91328CB2CLONEDHUMAN3H-CP-55940CP 55,9400.7Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91329CB2CLONEDHUMAN3H-CP-55940O-43341035Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91330CB1CLONEDHUMAN3H-CP-55940O-433419Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91331CB1CLONEDHUMAN3H-SR144528O-43346Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91332CB1CLONEDHUMAN3H-SR144528O-433311Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91333CB1CLONEDHUMAN3H-CP55940O-433334Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91334CB2CLONEDHUMAN3H-CP55940O-4333862Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91335CB2CLONEDHUMAN3H-CP55940O-43322263Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91336CB1CLONEDHUMAN3H-CP55940O-4332484Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91337CB1CLONEDHUMAN3H-SR144528O-4332299Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91338CB1CLONEDHUMAN3H-SR144528O-4331145Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91339CB1CLONEDHUMAN3H-CP55940O-4331249Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91340CB2CLONEDHUMAN3H-CP55940O-4331742Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91341CB2CLONEDHUMAN3H-CP55940O-43352341Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91342CB1CLONEDHUMAN3H-CP55940O-4335172Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91343CB1CLONEDHUMAN3H-SR144528O-433556Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91344CB1CLONEDHUMAN3H-SR144528O-215410Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91345CB1CLONEDHUMAN3H-CP55940O-215438Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91346CB2CLONEDHUMAN3H-CP55940O-2154731Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91347CB2CLONEDHUMAN3H-CP55940O-4336669Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91348CB1CLONEDHUMAN3H-CP55940O-433661Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91349CB1CLONEDHUMAN3H-SR144528O-433615Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91350CB1CLONEDHUMAN3H-SR144528O-43719Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91351CB1CLONEDHUMAN3H-CP55940O-437139Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91352CB2CLONEDHUMAN3H-CP55940O-4371555Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91353CB2CLONEDHUMAN3H-CP55940O-43731703Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91354CB1CLONEDHUMAN3H-CP55940O-4373147Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91355CB1CLONEDHUMAN3H-SR144528O-437344Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91356CB1CLONEDHUMAN3H-SR144528O-4337153Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91357CB1CLONEDHUMAN3H-CP55940O-4337420Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91358CB2CLONEDHUMAN3H-CP55940O-43371593Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91359CB2CLONEDHUMAN3H-CP55940O-21551848Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91360CB1CLONEDHUMAN3H-CP55940O-2155222Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91361CB1CLONEDHUMAN3H-SR144528O-215547Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91362CB1CLONEDHUMAN3H-SR144528O-433950Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91363CB1CLONEDHUMAN3H-CP55940O-4339162Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91364CB2CLONEDHUMAN3H-CP55940O-4339947Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91365CB2CLONEDHUMAN3H-CP55940O-4372298Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91366CB1CLONEDHUMAN3H-CP55940O-437277Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91367CB1CLONEDHUMAN3H-SR144528O-437227Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91368CB1CLONEDHUMAN3H-SR144528O-442373Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91369CB1CLONEDHUMAN3H-CP55940O-4423318Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91370CB2CLONEDHUMAN3H-CP55940O-44233658Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91371CB2CLONEDHUMAN3H-CP55940O-4338>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91372CB1CLONEDHUMAN3H-CP55940O-4338680Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91373CB1CLONEDHUMAN3H-SR144528O-4338290Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91374CB1CLONEDHUMAN3H-SR144528O-666845Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91375CB1CLONEDHUMAN3H-CP55940O-666868Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91376CB2CLONEDHUMAN3H-CP55940O-6668>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91377CB2CLONEDHUMAN3H-CP55940O-67305415Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91378CB1CLONEDHUMAN3H-CP55940O-673083Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91379CB1CLONEDHUMAN3H-SR144528O-673089Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91380CB1CLONEDHUMAN3H-SR144528O-6729120Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91381CB1CLONEDHUMAN3H-CP-55940O-6729185Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91382CB2CLONEDHUMAN3H-CP-55940O-67294573Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91383CB2CLONEDHUMAN3H-CP-55940O-67315342Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91384CB1CLONEDHUMAN3H-CP-55940O-6731117Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91385CB1CLONEDHUMAN3H-SR144528O-6731247Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91386CB1CLONEDHUMAN3H-SR144528O-6740265Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91387CB1CLONEDHUMAN3H-CP55940O-6740159Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91388CB2CLONEDHUMAN3H-CP55940O-6740>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91389CB2CLONEDHUMAN3H-CP55940O-4424>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91390CB1CLONEDHUMAN3H-CP55940O-4424169Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91391CB1CLONEDHUMAN3H-SR144528O-442445Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91392CB1CLONEDHUMAN3H-SR144528O-621152Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91393CB1CLONEDHUMAN3H-CP55940O-6211138Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91394CB2CLONEDHUMAN3H-CP55940O-6211>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91395CB2CLONEDHUMAN3H-CP55940O-6212>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91396CB1CLONEDHUMAN3H-CP55940O-621286Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91397CB1CLONEDHUMAN3H-SR144528O-621241Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91398CB1CLONEDHUMAN3H-SR144528O-661743Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91399CB1CLONEDHUMAN3H-CP55940O-661785Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91400CB2CLONEDHUMAN3H-CP55940O-6617>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91401CB2CLONEDHUMAN3H-CP55940O-6618>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91402CB1CLONEDHUMAN3H-CP55940O-661889Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91403CB1CLONEDHUMAN3H-SR144528O-661844Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91404CB1CLONEDHUMAN3H-SR144528O-621391Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91405CB1CLONEDHUMAN3H-CP55940O-6213182Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91406CB2CLONEDHUMAN3H-CP55940O-6213>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91407CB2CLONEDHUMAN3H-CP55940O-6215>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91408CB1CLONEDHUMAN3H-CP55940O-6215332Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91409CB1CLONEDHUMAN3H-SR144528O-6215221Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91410CB1CLONEDHUMAN3H-SR144528O-621456Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91411CB1CLONEDHUMAN3H-CP55940O-621488Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91412CB2CLONEDHUMAN3H-CP55940O-6214>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91413CB2CLONEDHUMAN3H-CP55940O-6629>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91414CB1CLONEDHUMAN3H-CP55940O-662924Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91415CB1CLONEDHUMAN3H-SR144528O-662920Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91416CB1CLONEDHUMAN3H-SR144528O-665846Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91417CB1CLONEDHUMAN3H-CP55940O-665857Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91418CB2CLONEDHUMAN3H-CP55940O-6658>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91419CB2CLONEDHUMAN3H-CP55940O-6659>10000Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91420CB1CLONEDHUMAN3H-CP55940O-6659109Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
91421CB1CLONEDHUMAN3H-SR144528O-6659128Wiley JL et al 2012Jan 15, 2025Jan 28, 2025
914225-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate0.54Li P et al 2014Jan 15, 2025Jan 15, 2025
914235-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone0.94Li P et al 2014Jan 15, 2025Jan 15, 2025
914245-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Ethyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone2.1Li P et al 2014Jan 15, 2025Jan 15, 2025
914255-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Isopropyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone7.5Li P et al 2014Jan 15, 2025Jan 15, 2025
914265-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Butyl-2,3,6b,9,10,10ahexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone14Li P et al 2014Jan 15, 2025Jan 15, 2025
914275-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-benzyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone4.7Li P et al 2014Jan 15, 2025Jan 15, 2025
914285-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-5-Bromo-3-methyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone4Li P et al 2014Jan 15, 2025Jan 15, 2025
914295-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-5-Methoxy-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone (3.5Li P et al 2014Jan 15, 2025Jan 15, 2025
914305-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate172Li P et al 2014Jan 15, 2025Jan 15, 2025
914315-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone280Li P et al 2014Jan 15, 2025Jan 15, 2025
914325-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Ethyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone287Li P et al 2014Jan 15, 2025Jan 15, 2025
914335-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Isopropyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone498Li P et al 2014Jan 15, 2025Jan 15, 2025
914345-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Butyl-2,3,6b,9,10,10ahexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone240Li P et al 2014Jan 15, 2025Jan 15, 2025
914355-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-benzyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone (385Li P et al 2014Jan 15, 2025Jan 15, 2025
914365-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-5-Bromo-3-methyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone582Li P et al 2014Jan 15, 2025Jan 15, 2025
914375-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-5-Methoxy-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone (1090Li P et al 2014Jan 15, 2025Jan 15, 2025
91438D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate32Li P et al 2014Jan 15, 2025Jan 29, 2025
91439D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone30Li P et al 2014Jan 15, 2025Jan 29, 2025
91440D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-3-Ethyl-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone66Li P et al 2014Jan 15, 2025Jan 29, 2025
91441D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-3-benzyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone (86Li P et al 2014Jan 15, 2025Jan 29, 2025
91442D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-5-Methoxy-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone (46Li P et al 2014Jan 15, 2025Jan 29, 2025
914435-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-phenyl-butan-1-one5.8Li P et al 2014Jan 15, 2025Jan 15, 2025
914445-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-( 4-pyridinyl)-1-butanone (4.7Li P et al 2014Jan 15, 2025Jan 15, 2025
914455-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4,4-difluoro-piperidin-1-yl)-butan-1-one1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914465-HT2ACLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(4-Fluorophenoxy)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahy-dro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxaline2.4Li P et al 2014Jan 15, 2025Jan 15, 2025
914475-HT2ACLONEDHUMAN125I-DOI4-Fluoro-N-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-benzamide671Li P et al 2014Jan 15, 2025Jan 15, 2025
914485-HT2ACLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(1,2-Benzisoxazol-3yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline hydrochloride3.3Li P et al 2014Jan 15, 2025Jan 15, 2025
914495-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline2.5Li P et al 2014Jan 15, 2025Jan 15, 2025
914505-HT2ACLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(6-Fluoro-1H-indazol-3-yl)-propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline formate18Li P et al 2014Jan 15, 2025Jan 15, 2025
914515-HT2ACLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(4-Fluoro-phenyl)-4,5-dihydro-isoxazol-5-ylmethyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline50Li P et al 2014Jan 15, 2025Jan 15, 2025
914525-HT2ACLONEDHUMAN125I-DOI6-Chloro-5-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-1,3-dihydro-indol-2-one1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914535-HT2ACLONEDHUMAN125I-DOI2,8-Dimethyl-3-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-pyrido[1,2-a]pyrimidin-4-one702Li P et al 2014Jan 15, 2025Jan 15, 2025
914545-HT2ACLONEDHUMAN125I-DOI(3aR,7aS)-2-[4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-butyl]-hexahydro-isoindole-1,3-dione1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914555-HT2ACLONEDHUMAN125I-DOI(3aR,7aS)-2-[3-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-propyl]-hexahydro-isoindole-1,3-dione1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914565-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-phenyl-butan-1-one (89Li P et al 2014Jan 15, 2025Jan 15, 2025
914575-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-( 4-pyridinyl)-1-butanone1090Li P et al 2014Jan 15, 2025Jan 15, 2025
914585-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4,4-difluoro-piperidin-1-yl)-butan-1-one1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914595-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(4-Fluorophenoxy)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahy-dro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxaline259Li P et al 2014Jan 15, 2025Jan 15, 2025
914605-HT2CCLONEDHUMAN125I-DOI4-Fluoro-N-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-benzamide1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914615-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(1,2-Benzisoxazol-3yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline hydrochloride287Li P et al 2014Jan 15, 2025Jan 15, 2025
914625-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline300Li P et al 2014Jan 15, 2025Jan 15, 2025
914635-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-8-[3-(4-Fluoro-phenyl)-4,5-dihydro-isoxazol-5-ylmethyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline3280Li P et al 2014Jan 15, 2025Jan 15, 2025
914645-HT2CCLONEDHUMAN125I-DOI6-Chloro-5-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-1,3-dihydro-indol-2-one1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914655-HT2CCLONEDHUMAN125I-DOI(3aR,7aS)-2-[4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-butyl]-hexahydro-isoindole-1,3-dione1000Li P et al 2014Jan 15, 2025Jan 15, 2025
91466D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-phenyl-butan-1-one (43Li P et al 2014Jan 15, 2025Jan 29, 2025
91467D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-( 4-pyridinyl)-1-butanone1000Li P et al 2014Jan 15, 2025Jan 29, 2025
91468D2CLONEDRAT3H-SPIPERONE4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4,4-difluoro-piperidin-1-yl)-butan-1-one1000Li P et al 2014Jan 15, 2025Jan 29, 2025
91469D2CLONEDRAT3H-SPIPERONE(6bR,10aS)-8-[3-(4-Fluorophenoxy)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahy-dro-1H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxaline213Li P et al 2014Jan 15, 2025Jan 29, 2025
91470D2CLONEDRAT3H-SPIPERONE4-Fluoro-N-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-benzamide767Li P et al 2014Jan 15, 2025Jan 29, 2025
91471D2CLONEDRAT3H-SPIPERONE(6bR,10aS)-8-[3-(1,2-Benzisoxazol-3yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline hydrochloride174Li P et al 2014Jan 15, 2025Jan 29, 2025
91472D2CLONEDRAT3H-SPIPERONE(6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline192Li P et al 2014Jan 15, 2025Jan 29, 2025
91473D2CLONEDRAT3H-SPIPERONE(6bR,10aS)-8-[3-(6-Fluoro-1H-indazol-3-yl)-propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline formate27Li P et al 2014Jan 15, 2025Jan 29, 2025
91474D2CLONEDRAT3H-SPIPERONE6-Chloro-5-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-1,3-dihydro-indol-2-one1000Li P et al 2014Jan 15, 2025Jan 29, 2025
91475D2CLONEDRAT3H-SPIPERONE2,8-Dimethyl-3-[2-((6bR,10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-ethyl]-pyrido[1,2-a]pyrimidin-4-one3000Li P et al 2014Jan 15, 2025Jan 29, 2025
91476D2CLONEDRAT3H-SPIPERONE(3aR,7aS)-2-[4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-butyl]-hexahydro-isoindole-1,3-dione1000Li P et al 2014Jan 15, 2025Jan 29, 2025
91477D2CLONEDRAT3H-SPIPERONE(3aR,7aS)-2-[3-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-propyl]-hexahydro-isoindole-1,3-dione1000Li P et al 2014Jan 15, 2025Jan 29, 2025
914785-HT2ACLONEDHUMAN125I-DOI4-((6bS,10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-butan-1-one (4.6Li P et al 2014Jan 15, 2025Jan 15, 2025
914795-HT2ACLONEDHUMAN125I-DOI4-(rel-(6bS,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-1-butanone1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914805-HT2ACLONEDHUMAN125I-DOI4-(rel-(6bR, 10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-1-butanone324Li P et al 2014Jan 15, 2025Jan 15, 2025
914815-HT2ACLONEDHUMAN125I-DOI4-((6bS,10aR)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone5.5Li P et al 2014Jan 15, 2025Jan 15, 2025
914825-HT2ACLONEDHUMAN125I-DOI(6bS,11aS)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophenyl)-1-butanone1.7Li P et al 2014Jan 15, 2025Jan 15, 2025
914835-HT2ACLONEDHUMAN125I-DOI(6bR,11aR)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophenyl)-1-butanone17Li P et al 2014Jan 15, 2025Jan 15, 2025
914845-HT2ACLONEDHUMAN125I-DOI(6bR,10aS)-1-(4-fluorophenyl)-4-(1,3-dimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-butanone5.7Li P et al 2014Jan 15, 2025Jan 15, 2025
914855-HT2ACLONEDHUMAN125I-DOI(6bR,10aS)-1-(4-Fluorophenyl)-4-(1,1,3-trimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-butanone5.2Li P et al 2014Jan 15, 2025Jan 15, 2025
914865-HT2ACLONEDHUMAN125I-DOI4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone1Li P et al 2014Jan 15, 2025Jan 15, 2025
914875-HT2ACLONEDHUMAN125I-DOI4-((7aR,11aS)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone (7.7Li P et al 2014Jan 15, 2025Jan 15, 2025
914885-HT2ACLONEDHUMAN125I-DOI4-((6aS,10aR)-4,5,7,8,10,10a-Hexahydro-6aH-pyrido[4,3-b]pyrrolo[3,2,1-hi]indol-9-yl)-1-(4-Fluoro-phenyl)-butan-1-one2.9Li P et al 2014Jan 15, 2025Jan 15, 2025
914895-HT2ACLONEDHUMAN125I-DOI4-((8aS,12aR)-4,5,6,7,9,10,12,12a-Octahydroazepino[3,2,1-hi]pyrido[4,3-b]-indol-11(8aH)-yl)-1-(4-fluorophenyl)-1-butanone1.1Li P et al 2014Jan 15, 2025Jan 15, 2025
914905-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-thia-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)-butan-1-one1.3Li P et al 2014Jan 15, 2025Jan 15, 2025
914915-HT2ACLONEDHUMAN125I-DOI4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one (0.89Li P et al 2014Jan 15, 2025Jan 15, 2025
914925-HT2ACLONEDHUMAN125I-DOI(6bS, 11aS)-4-(1,2,6b,7,8,10,11,11a-Octahydro-9H-azepino[4,5-b][1,4]oxazino[2,3,4-hi]indol-9-yl)-1-(4-fluorophenyl)-1-butanone14Li P et al 2014Jan 15, 2025Jan 15, 2025
914935-HT2CCLONEDHUMAN125I-DOI4-((6bS,10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-butan-1-one (532Li P et al 2014Jan 15, 2025Jan 15, 2025
914945-HT2CCLONEDHUMAN125I-DOI4-(rel-(6bS,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-1-butanone1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914955-HT2CCLONEDHUMAN125I-DOI4-(rel-(6bR, 10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-1-butanone1000Li P et al 2014Jan 15, 2025Jan 15, 2025
914965-HT2CCLONEDHUMAN125I-DOI4-((6bS,10aR)-2,3,6b,9,10,10a-Hexahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-(4-fluorophenyl)-1-butanone702Li P et al 2014Jan 15, 2025Jan 15, 2025
914975-HT2CCLONEDHUMAN125I-DOI(6bS,11aS)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophenyl)-1-butanone503Li P et al 2014Jan 15, 2025Jan 15, 2025
914985-HT2CCLONEDHUMAN125I-DOI(6bR,11aR)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophenyl)-1-butanone1280Li P et al 2014Jan 15, 2025Jan 15, 2025
914995-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-1-(4-fluorophenyl)-4-(1,3-dimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-butanone (280Li P et al 2014Jan 15, 2025Jan 15, 2025
915005-HT2CCLONEDHUMAN125I-DOI(6bR,10aS)-1-(4-Fluorophenyl)-4-(1,1,3-trimethyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]-pyrrolo[1,2,3-de]quinoxalin-8(7H)-yl)-1-butanone862Li P et al 2014Jan 15, 2025Jan 15, 2025
915015-HT2CCLONEDHUMAN125I-DOI4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone83Li P et al 2014Jan 15, 2025Jan 15, 2025
915025-HT2CCLONEDHUMAN125I-DOI4-((7aR,11aS)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone (110Li P et al 2014Jan 15, 2025Jan 15, 2025
915035-HT2CCLONEDHUMAN125I-DOI4-((6aS,10aR)-4,5,7,8,10,10a-Hexahydro-6aH-pyrido[4,3-b]pyrrolo[3,2,1-hi]indol-9-yl)-1-(4-Fluoro-phenyl)-butan-1-one507Li P et al 2014Jan 15, 2025Jan 15, 2025
915045-HT2CCLONEDHUMAN125I-DOI4-((8aS,12aR)-4,5,6,7,9,10,12,12a-Octahydroazepino[3,2,1-hi]pyrido[4,3-b]-indol-11(8aH)-yl)-1-(4-fluorophenyl)-1-butanone195Li P et al 2014Jan 15, 2025Jan 15, 2025
915055-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-thia-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)-butan-1-one150Li P et al 2014Jan 15, 2025Jan 15, 2025
915065-HT2CCLONEDHUMAN125I-DOI4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one (520Li P et al 2014Jan 15, 2025Jan 15, 2025
915075-HT2CCLONEDHUMAN125I-DOI(6bS, 11aS)-4-(1,2,6b,7,8,10,11,11a-Octahydro-9H-azepino[4,5-b][1,4]oxazino[2,3,4-hi]indol-9-yl)-1-(4-fluorophenyl)-1-butanone641Li P et al 2014Jan 15, 2025Jan 15, 2025
91508D2CLONEDRAT3H-Methylspiperone4-((6bS,10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-butan-1-one95Li P et al 2014Jan 15, 2025Jan 29, 2025
91509D2CLONEDRAT3H-Methylspiperone4-(rel-(6bS,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-1-butanone97Li P et al 2014Jan 15, 2025Jan 29, 2025
91510D2CLONEDRAT3H-Methylspiperone4-(rel-(6bR, 10aR)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)-1-butanone52Li P et al 2014Jan 15, 2025Jan 29, 2025
91511D2CLONEDRAT3H-Methylspiperone(6bS,11aS)-4-(3-Methyl-2,3,6b,7,8,10,11,11a-octahydro-1H,9H-azepino[4,5:4,5]pyrrolo[1,2,3-de]quinoxalin-9-yl)-1-(4-fluorophenyl)-1-butanone148Li P et al 2014Jan 15, 2025Jan 29, 2025
91512D2CLONEDRAT3H-Methylspiperone4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone27Li P et al 2014Jan 15, 2025Jan 29, 2025
91513D2CLONEDRAT3H-Methylspiperone4-((6aS,10aR)-4,5,7,8,10,10a-Hexahydro-6aH-pyrido[4,3-b]pyrrolo[3,2,1-hi]indol-9-yl)-1-(4-Fluoro-phenyl)-butan-1-one71Li P et al 2014Jan 15, 2025Jan 29, 2025
91514D2CLONEDRAT3H-Methylspiperone4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-thia-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)-butan-1-one50Li P et al 2014Jan 15, 2025Jan 29, 2025
91515D2CLONEDRAT3H-Methylspiperone4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one (41Li P et al 2014Jan 15, 2025Jan 29, 2025
91516D2CLONEDRAT3H-Methylspiperone(6bS, 11aS)-4-(1,2,6b,7,8,10,11,11a-Octahydro-9H-azepino[4,5-b][1,4]oxazino[2,3,4-hi]indol-9-yl)-1-(4-fluorophenyl)-1-butanone69Li P et al 2014Jan 15, 2025Jan 29, 2025
91517SERTPlateletsHUMAN3H-N-Me-citalopram4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate61Li P et al 2014Jan 15, 2025Jan 28, 2025
91518SERTPlateletsHUMAN3H-N-Me-citalopram4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate31Li P et al 2014Jan 15, 2025Jan 28, 2025
91519SERTPlateletsHUMAN3H-N-Me-citalopram4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone98Li P et al 2014Jan 15, 2025Jan 28, 2025
915205-HT1AUNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate1480Li P et al 2014Jan 15, 2025Jan 15, 2025
915215-HT1AUNDEFINEDUNDEFINEDUNDEFINED(6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline364Li P et al 2014Jan 15, 2025Jan 15, 2025
915225-HT1AUNDEFINEDUNDEFINEDUNDEFINED4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone206Li P et al 2014Jan 15, 2025Jan 15, 2025
915235-HT1AUNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one1330Li P et al 2014Jan 15, 2025Jan 15, 2025
915245-HT1AUNDEFINEDUNDEFINEDUNDEFINEDCLOZAPINE140Li P et al 2014Jan 15, 2025Jan 15, 2025
915255-HT1AUNDEFINEDUNDEFINEDUNDEFINEDOLANZAPINE2720Li P et al 2014Jan 15, 2025Jan 15, 2025
91526H1UNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate1000Li P et al 2014Jan 15, 2025Jan 28, 2025
91527Alpha1AUNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate73Li P et al 2014Jan 15, 2025Jan 15, 2025
91528Alpha1AUNDEFINEDUNDEFINEDUNDEFINED(6bR,10aS)-8-[3-(1,2-Benzisoxazol-3yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline hydrochloride314Li P et al 2014Jan 15, 2025Jan 15, 2025
91529Alpha1AUNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one262Li P et al 2014Jan 15, 2025Jan 15, 2025
91530Alpha1AUNDEFINEDUNDEFINEDUNDEFINEDCLOZAPINE19Li P et al 2014Jan 15, 2025Jan 15, 2025
91531Alpha1AUNDEFINEDUNDEFINEDUNDEFINEDOLANZAPINE60Li P et al 2014Jan 15, 2025Jan 15, 2025
91532Alpha1BUNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate31Li P et al 2014Jan 15, 2025Jan 15, 2025
91533Alpha1BUNDEFINEDUNDEFINEDUNDEFINED(6bR,10aS)-8-[3-(1,2-Benzisoxazol-3yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido-[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline hydrochloride294Li P et al 2014Jan 15, 2025Jan 15, 2025
91534Alpha1BUNDEFINEDUNDEFINEDUNDEFINED(6bR,10aS)-8-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxaline66Li P et al 2014Jan 15, 2025Jan 15, 2025
91535Alpha1BUNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one (104Li P et al 2014Jan 15, 2025Jan 15, 2025
91536D1UNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate52Li P et al 2014Jan 15, 2025Jan 28, 2025
91537D1UNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate110Li P et al 2014Jan 15, 2025Jan 28, 2025
91538D4UNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-3-Methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3,4:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluoro-phenyl)-butan-1-one 4-methylbenzenesulfonate108Li P et al 2014Jan 15, 2025Jan 28, 2025
91539D4UNDEFINEDUNDEFINEDUNDEFINED4-((7aS,11aR)-5,6,8,9,11,11a-Hexahydro-4H,7aH-pyrido[3,4:4,5]pyrrolo[3,2,1-ij]quinoline-10(7aH)-yl)-1-(4-fluorophenyl)-1-butanone60Li P et al 2014Jan 15, 2025Jan 28, 2025
91540D4UNDEFINEDUNDEFINEDUNDEFINED4-((6bR,10aS)-1,2,6b,9,10,10a-Hexahydro-7H-3-oxa-8,10b-diaza-fluoranthen-8-yl)-1-(4-Fluoro-phenyl)--butan-1-one320Li P et al 2014Jan 15, 2025Jan 28, 2025
91541D4UNDEFINEDUNDEFINEDUNDEFINEDCLOZAPINE40Li P et al 2014Jan 15, 2025Jan 28, 2025
91542D4UNDEFINEDUNDEFINEDUNDEFINEDOLANZAPINE28Li P et al 2014Jan 15, 2025Jan 28, 2025
91543A1CLONEDHUMAN3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide55.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91544A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide2.79Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91545A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide3.47Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91546A1CLONEDHUMAN3H-CCPAN-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide90.8Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91547A1CLONEDHUMAN3H-CCPAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide24.4Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91548A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide0.939Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91549A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91550A1CLONEDHUMAN3H-CCPAN-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91551A1CLONEDHUMAN3H-CCPAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91552A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91553A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91554A1CLONEDHUMAN3H-CCPAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91555A1CLONEDHUMAN3H-CCPAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91556A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91557A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide1.47Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91558A1CLONEDHUMAN3H-CCPAN-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide36.7Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91559A1CLONEDHUMAN3H-CCPAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide32.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91560A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1.01Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91561A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide1.77Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91562A1CLONEDHUMAN3H-CCPA4-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide13.6Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91563A1CLONEDHUMAN3H-CCPA4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide9.69Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91564A1CLONEDHUMAN3H-CCPA4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide0.529Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91565A1CLONEDHUMAN3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91566A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91567A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91568A1CLONEDHUMAN3H-CCPA4-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91569A1CLONEDHUMAN3H-CCPA4-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91570A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91571A1CORTICAL MEMBRANESRAT3H-CCPA4-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91572A1CLONEDHUMAN3H-CCPA4-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91573A1CLONEDHUMAN3H-CCPAN-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide7.57Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91574A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide0.348Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91575A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide6.69Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91576A1CLONEDHUMAN3H-CCPAN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide178Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91577A1CLONEDHUMAN3H-CCPAN-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91578A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91579A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91580A1CLONEDHUMAN3H-CCPAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91581A1CLONEDHUMAN3H-CCPAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91582A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91583A1CORTICAL MEMBRANESRAT3H-CCPAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91584A1CLONEDHUMAN3H-CCPAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91585A2ACLONEDHUMAN3H-MSX-2N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide77.7Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91586A2AStriatal MembranesRAT3H-MSX-2N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91587A2AStriatal MembranesRAT3H-MSX-2N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide391Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91588A2ACLONEDHUMAN3H-MSX-2N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide83.6Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91589A2ACLONEDHUMAN3H-MSX-2N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide39.1Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91590A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide1670Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91591A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91592A2ACLONEDHUMAN3H-MSX-2N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91593A2ACLONEDHUMAN3H-MSX-2N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91594A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91595A2AStriatal MembranesRAT3H-MSX-2N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91596A2ACLONEDHUMAN3H-MSX-2N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91597A2ACLONEDHUMAN3H-MSX-2N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91598A2AStriatal MembranesRAT3H-MSX-2N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91599A2AStriatal MembranesRAT3H-MSX-2N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91600A2ACLONEDHUMAN3H-MSX-2N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91601A2ACLONEDHUMAN3H-MSX-2N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91602A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91603A2AStriatal MembranesRAT3H-MSX-24-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91604A2ACLONEDHUMAN3H-MSX-24-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91605A2ACLONEDHUMAN3H-MSX-24-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91606A2AStriatal MembranesRAT3H-MSX-24-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91607A2AStriatal MembranesRAT3H-MSX-2N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91608A2ACLONEDHUMAN3H-MSX-2N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91609A2ACLONEDHUMAN3H-MSX-24-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91610A2AStriatal MembranesRAT3H-MSX-24-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91611A2AStriatal MembranesRAT3H-MSX-24-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91612A2ACLONEDHUMAN3H-MSX-24-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91613A2ACLONEDHUMAN3H-MSX-24-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91614A2AStriatal MembranesRAT3H-MSX-24-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91615A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide1210Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91616A2AStriatal MembranesRAT3H-MSX-2N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide73.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91617A2ACLONEDHUMAN3H-MSX-2N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide132Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91618A2ACLONEDHUMAN3H-MSX-2N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91619A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91620A2AStriatal MembranesRAT3H-MSX-2N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91621A2ACLONEDHUMAN3H-MSX-2N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91622A2ACLONEDHUMAN3H-MSX-2N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91623A2AStriatal MembranesRAT3H-MSX-2N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91624A2AStriatal MembranesRAT3H-MSX-2N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91625A2ACLONEDHUMAN3H-MSX-2N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91626A2BCLONEDHUMAN3H-PSB-603N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91627A2BCLONEDHUMAN3H-PSB-603N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91628A2BCLONEDHUMAN3H-PSB-603N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91629A2BCLONEDHUMAN3H-PSB-603N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91630A2BCLONEDHUMAN3H-PSB-603N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91631A2BCLONEDHUMAN3H-PSB-603N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91632A2BCLONEDHUMAN3H-PSB-603N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91633A2BCLONEDHUMAN3H-PSB-603N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91634A2BCLONEDHUMAN3H-PSB-603N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91635A2BCLONEDHUMAN3H-PSB-6034-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91636A2BCLONEDHUMAN3H-PSB-6034-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91637A2BCLONEDHUMAN3H-PSB-603N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91638A2BCLONEDHUMAN3H-PSB-6034-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91639A2BCLONEDHUMAN3H-PSB-6034-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91640A2BCLONEDHUMAN3H-PSB-6034-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91641A2BCLONEDHUMAN3H-PSB-603N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91642A2BCLONEDHUMAN3H-PSB-603N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91643A2BCLONEDHUMAN3H-PSB-603N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91644A2BCLONEDHUMAN3H-PSB-603N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91645A2BCLONEDHUMAN3H-PSB-603N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91646A2BCLONEDHUMAN3H-PSB-603N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide100Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91647A3CLONEDHUMAN3H-PSB-11N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide67.8Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91648A3CLONEDHUMAN3H-PSB-11N-(4-phenyl-5-(pyridin-2-yl)thiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91649A3CLONEDHUMAN3H-PSB-11N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide428Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91650A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide111Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91651A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide9.05Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91652A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide8.23Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91653A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide83.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91654A3CLONEDHUMAN3H-PSB-11N-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide25.4Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91655A3CLONEDHUMAN3H-PSB-11N-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91656A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-methoxybenzoyl)4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91657A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91658A3CLONEDHUMAN3H-PSB-11N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91659A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide174Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91660A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide27.8Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91661A3CLONEDHUMAN3H-PSB-114-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide4.63Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91662A3CLONEDHUMAN3H-PSB-11N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide42.2Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91663A3CLONEDHUMAN3H-PSB-11N-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide124Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91664A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide129Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91665A3CLONEDHUMAN3H-PSB-11N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide25.4Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91666A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide6.45Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91667A3CLONEDHUMAN3H-PSB-11N-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide48.3Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91668A3CLONEDRAT3H-NECAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide806Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91669A3CLONEDRAT3H-NECAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benz- 1 amide1320Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91670A3CLONEDRAT3H-NECAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide>10000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91671A3CLONEDRAT3H-NECAN-(5-benzoyl-4-phenylthiazol-2-yl)-4-methoxybenzamide1000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91672A3CLONEDRAT3H-NECAN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)-4-methoxybenzamide>10000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91673A3CLONEDRAT3H-NECA4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide>10000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91674A3CLONEDRAT3H-NECA4-Methoxy-N-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide>10000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91675A3CLONEDRAT3H-NECA4-Methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide>10000Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91676A3CLONEDRAT3H-NECAN-(5-(4-oxo-3-p-tolyl-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide1840Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91677A3CLONEDRAT3H-NECAN-(5-(3-(4-methoxyphenyl)-4-oxo-3,4dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide973Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91678A3CLONEDRAT3H-NECAN-(5-(3-(4-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)furan-2- 1 carboxamide607Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91679A1CORTICAL MEMBRANESRAT3H-DPCPXN-(5-(2,4-difluorobenzoyl)-4-phenylthiazol-2-yl)benzamide2.93Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91680A1CORTICAL MEMBRANESRAT3H-DPCPXN-(5-(4-chlorobenzoyl)-4-phenylthiazol-2-yl)benzamide0.0867Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91681A1CORTICAL MEMBRANESRAT3H-DPCPX4-Methoxy-N-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)benzamide0.0709Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91682A1CORTICAL MEMBRANESRAT3H-DPCPXN-(5-(4-methylbenzoyl)-4-phenylthiazol-2-yl)furan-2-carboxamide0.0628Abdelrahman A et al 2020Jan 15, 2025Jan 15, 2025
91683A3HEK293 cellsHUMAN3H-HEMADO1-Propyl-8-{1-[3-(3-trifluoromethyl-phenyl)-prop-2-ynyl]-1H-pyrazol-4-yl}-3, 7-dihydro-purine-2, 6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91684A1CLONEDHUMAN3H-DPCPX8-[1-(5-Oxo-1-m-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91685A1CLONEDHUMAN3H-DPCPX8-[1-(5-Oxo-1-p-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91686A1CLONEDHUMAN3H-DPCPX8-{1-[1-(3-Methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91687A1CLONEDHUMAN3H-DPCPX8-{1-[1-(4-Methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91688A1CLONEDHUMAN3H-DPCPX8-{1-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91689A1CLONEDHUMAN3H-DPCPX8-{1-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91690A1CLONEDHUMAN3H-DPCPX8-{1-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91691A1CLONEDHUMAN3H-DPCPX8-{1-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91692A1CLONEDHUMAN3H-DPCPX8-{1-[5-Oxo-1-(3-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91693A1CLONEDHUMAN3H-DPCPX8-{1-[5-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91694A1CLONEDHUMAN3H-DPCPX4-{4-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-pyrazol-1-ylmethyl]-2-oxo-pyrrolidin-1-yl}-benzonitrile1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91695A1CLONEDHUMAN3H-DPCPX8-{1-[1-(2,4-Difluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91696A1CLONEDHUMAN3H-DPCPX3-Ethyl-8-{1-[1-(3-fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91697A1CLONEDHUMAN3H-DPCPX3-Ethyl-8-{1-[1-(4-fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91698A1CLONEDHUMAN3H-DPCPX3-Ethyl-8-{1-[5-oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91699A1CLONEDHUMAN3H-DPCPX3-Ethyl-8-{1-[5-oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91700A1CLONEDHUMAN3H-DPCPX3-Ethyl-8-{1-[5-oxo-1-(3-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91701A1CLONEDHUMAN3H-DPCPX3-Ethyl-8-{1-[1-(4-methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91702A1CLONEDHUMAN3H-DPCPX8-{1-[2-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91703A1CLONEDHUMAN3H-DPCPX8-{1-[2-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91704A1CLONEDHUMAN3H-DPCPX1,3-Dipropyl-8-[1-(1-p-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91705A1CLONEDHUMAN3H-DPCPX8-{1-[1-(3-Methoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91706A1CLONEDHUMAN3H-DPCPX8-{1-[1-(4-Methoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91707A1CLONEDHUMAN3H-DPCPX1,3-Dipropyl-8-{1-[1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91708A1CLONEDHUMAN3H-DPCPX1,3-Dipropyl-8-{1-[1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91709A1CLONEDHUMAN3H-DPCPX8-(1-{2-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91710A1CLONEDHUMAN3H-DPCPX8-(1-{1-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91711A1CLONEDHUMAN3H-DPCPX8-(1-{2-Hydroxy-2-[5-oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91712A1CLONEDHUMAN3H-DPCPX8-(1-{2-Oxo-2-[4-(3-trifluoromethyl-phenyl)-piperazin-1-yl]-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91713A1CLONEDHUMAN3H-DPCPX8-(1-{2-[4-(2,4-Difluoro-phenyl)-piperazin-1-yl]-2-oxo-ethyl}-1H-pyrazol-4-yl)-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91714A1CLONEDHUMAN3H-DPCPX8-{4-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91715A1CLONEDHUMAN3H-DPCPX8-{4-[1-(4-Fluorophenyl)-5-oxo-pyrrolidin-3-ylmethoxy]phenyl}-1,3-dipropyl-3,7-dihydropurine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91716A1CLONEDHUMAN3H-DPCPX8-{4-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-phenyl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91717A1CLONEDHUMAN3H-DPCPX8-{6-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91718A1CLONEDHUMAN3H-DPCPX8-{6-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91719A1CLONEDHUMAN3H-DPCPX8-{6-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-pyridin-3-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91720A1CLONEDHUMAN3H-DPCPX8-{3-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91721A1CLONEDHUMAN3H-DPCPX8-{3-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91722A1CLONEDHUMAN3H-DPCPX8-{3-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91723A1CLONEDHUMAN3H-DPCPX8-{3-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethoxy]-isoxazol-5-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1000Basu S et al 2017Jan 15, 2025Jan 15, 2025
91724A2BCLONEDHUMAN3H-MRS-17548-[1-(5-Oxo-1-m-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione10.7Basu S et al 2017Jan 15, 2025Jan 15, 2025
91725A2BCLONEDHUMAN3H-MRS-17548-[1-(5-Oxo-1-p-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-1,3-dipropyl-3,7-dihydro-purine-2,6-dione8Basu S et al 2017Jan 15, 2025Jan 15, 2025
91726A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(3-Methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione21.6Basu S et al 2017Jan 15, 2025Jan 15, 2025
91727A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(4-Methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione9Basu S et al 2017Jan 15, 2025Jan 15, 2025
91728A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(3-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione41Basu S et al 2017Jan 15, 2025Jan 15, 2025
91729A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(4-Fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione9.7Basu S et al 2017Jan 15, 2025Jan 15, 2025
91730A2BCLONEDHUMAN3H-MRS-17548-{1-[5-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione6.5Basu S et al 2017Jan 15, 2025Jan 15, 2025
91731A2BCLONEDHUMAN3H-MRS-17548-{1-[5-Oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione1Basu S et al 2017Jan 15, 2025Jan 15, 2025
91732A2BCLONEDHUMAN3H-MRS-17548-{1-[5-Oxo-1-(3-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione9Basu S et al 2017Jan 15, 2025Jan 15, 2025
91733A2BCLONEDHUMAN3H-MRS-17548-{1-[5-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione4Basu S et al 2017Jan 15, 2025Jan 15, 2025
91734A2BCLONEDHUMAN3H-MRS-17548-{1-[5-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione23Basu S et al 2017Jan 15, 2025Jan 15, 2025
91735A2BCLONEDHUMAN3H-MRS-17544-{4-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-pyrazol-1-ylmethyl]-2-oxo-pyrrolidin-1-yl}-benzoic acid77Basu S et al 2017Jan 15, 2025Jan 15, 2025
91736A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(2,4-Difluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione19Basu S et al 2017Jan 15, 2025Jan 15, 2025
91737A2BCLONEDHUMAN3H-MRS-17543-Ethyl-8-{1-[1-(3-fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione24Basu S et al 2017Jan 15, 2025Jan 15, 2025
91738A2BCLONEDHUMAN3H-MRS-17543-Ethyl-8-{1-[1-(4-fluoro-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione12Basu S et al 2017Jan 15, 2025Jan 15, 2025
91739A2BCLONEDHUMAN3H-MRS-17543-Ethyl-8-{1-[5-oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione4.5Basu S et al 2017Jan 15, 2025Jan 15, 2025
91740A2BCLONEDHUMAN3H-MRS-17543-Ethyl-8-{1-[5-oxo-1-(4-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione4Basu S et al 2017Jan 15, 2025Jan 15, 2025
91741A2BCLONEDHUMAN3H-MRS-17543-Ethyl-8-{1-[5-oxo-1-(3-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione17.5Basu S et al 2017Jan 15, 2025Jan 15, 2025
91742A2BCLONEDHUMAN3H-MRS-17543-Ethyl-8-{1-[1-(4-methoxy-phenyl)-5-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1-propyl-3,7-dihydro-purine-2,6-dione16Basu S et al 2017Jan 15, 2025Jan 15, 2025
91743A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(3-Fluoro-phenyl)-2-oxo-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione43Basu S et al 2017Jan 15, 2025Jan 15, 2025
91744A2BCLONEDHUMAN3H-MRS-17548-{1-[2-Oxo-1-(3-trifluoromethyl-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione6Basu S et al 2017Jan 15, 2025Jan 15, 2025
91745A2BCLONEDHUMAN3H-MRS-17548-{1-[2-Oxo-1-(4-trifluoromethoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione8Basu S et al 2017Jan 15, 2025Jan 15, 2025
91746A2BCLONEDHUMAN3H-MRS-17541,3-Dipropyl-8-[1-(1-p-tolyl-pyrrolidin-3-ylmethyl)-1H-pyrazol-4-yl]-3,7-dihydro-purine-2,6-dione12Basu S et al 2017Jan 15, 2025Jan 15, 2025
91747A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(3-Methoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione13.7Basu S et al 2017Jan 15, 2025Jan 15, 2025
91748A2BCLONEDHUMAN3H-MRS-17548-{1-[1-(4-Methoxy-phenyl)-pyrrolidin-3-ylmethyl]-1H-pyrazol-4-yl}-1,3-dipropyl-3,7-dihydro-purine-2,6-dione13Basu S et al 2017Jan 15, 2025Jan 15, 2025