The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 91,001-92,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
93749A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3,4-dimethoxy-benzylamide102Federico S et al 2018Jan 15, 2025Jan 15, 2025
93750A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3,4-dimethoxy-benzylamide141Federico S et al 2018Jan 15, 2025Jan 15, 2025
93751A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid 3,4-dimethoxy-benzylamide246Federico S et al 2018Jan 15, 2025Jan 15, 2025
93752A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid phenethyl-amide73.1Federico S et al 2018Jan 15, 2025Jan 15, 2025
93753A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid phenethyl-amide29.7Federico S et al 2018Jan 15, 2025Jan 15, 2025
93754A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid phenethyl-amide6.82Federico S et al 2018Jan 15, 2025Jan 15, 2025
93755A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid [2-(3,4-dimethoxy-phenyl)-ethyl]-amide107Federico S et al 2018Jan 15, 2025Jan 15, 2025
93756A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid [2-(3,4-dimethoxy-phenyl)-ethyl]-amide169Federico S et al 2018Jan 15, 2025Jan 15, 2025
93757A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid [2-(3,4-dimethoxy-phenyl)-ethyl]-amide177Federico S et al 2018Jan 15, 2025Jan 15, 2025
93758A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (1,1-dimethyl-2-phenyl-ethyl)-amide38Federico S et al 2018Jan 15, 2025Jan 15, 2025
93759A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (1,1-dimethyl-2-phenyl-ethyl)-amide6.12Federico S et al 2018Jan 15, 2025Jan 15, 2025
93760A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (1,1-dimethyl-2-phenyl-ethyl)-amide6.52Federico S et al 2018Jan 15, 2025Jan 15, 2025
93761A3CLONEDHUMAN3H-HEMADO2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (2-phenoxy-ethyl)-amide16.4Federico S et al 2018Jan 15, 2025Jan 15, 2025
93762A2ACLONEDHUMAN3H-NECA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (2-phenoxy-ethyl)-amide38.2Federico S et al 2018Jan 15, 2025Jan 15, 2025
93763A1CLONEDHUMAN3H-CCPA2-Furan-2-yl-5-methylamino-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylic acid (2-phenoxy-ethyl)-amide172Federico S et al 2018Jan 15, 2025Jan 15, 2025
93764A1CLONEDHUMAN3H-CCPA2-furan-2-yl-5-methylamino- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid N0 -phenylhydrazide58.7Federico S et al 2018Jan 15, 2025Jan 15, 2025
93765A2ACLONEDHUMAN3H-NECA2-furan-2-yl-5-methylamino- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid N0 -phenylhydrazide342Federico S et al 2018Jan 15, 2025Jan 15, 2025
93766A3CLONEDHUMAN3H-HEMADO2-furan-2-yl-5-methylamino- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid N0 -phenylhydrazide15.1Federico S et al 2018Jan 15, 2025Jan 15, 2025
93767A3CLONEDHUMAN3H-HEMADO5-(3,4-dimethoxy-benzylamino)-2-furan-2-yl- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid benzhydryl-amide69.9Federico S et al 2018Jan 15, 2025Jan 15, 2025
93768A2ACLONEDHUMAN3H-NECA5-(3,4-dimethoxy-benzylamino)-2-furan-2-yl- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid benzhydryl-amide137Federico S et al 2018Jan 15, 2025Jan 15, 2025
93769A1CLONEDHUMAN3H-CCPA5-(3,4-dimethoxy-benzylamino)-2-furan-2-yl- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid benzhydryl-amide122Federico S et al 2018Jan 15, 2025Jan 15, 2025
93770A1CLONEDHUMAN3H-CCPAEthyl 2-(5-((2-ethoxy-2-oxoethyl)amino)-2-(furan-2-yl)-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxamido)acetate>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93771A2ACLONEDHUMAN3H-NECAEthyl 2-(5-((2-ethoxy-2-oxoethyl)amino)-2-(furan-2-yl)-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxamido)acetate1540Federico S et al 2018Jan 15, 2025Jan 15, 2025
93772A3CLONEDHUMAN3H-HEMADOEthyl 2-(5-((2-ethoxy-2-oxoethyl)amino)-2-(furan-2-yl)-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxamido)acetate646Federico S et al 2018Jan 15, 2025Jan 15, 2025
93773A3CLONEDHUMAN3H-HEMADOEthyl 2-(furan-2-yl)-5-(2-phenylhydrazinyl)-[1,2,4]triazolo[1,5-c] pyrimidine-8-carboxylate339Federico S et al 2018Jan 15, 2025Jan 15, 2025
93774A2ACLONEDHUMAN3H-NECAEthyl 2-(furan-2-yl)-5-(2-phenylhydrazinyl)-[1,2,4]triazolo[1,5-c] pyrimidine-8-carboxylate41.8Federico S et al 2018Jan 15, 2025Jan 15, 2025
93775A1CLONEDHUMAN3H-CCPAEthyl 2-(furan-2-yl)-5-(2-phenylhydrazinyl)-[1,2,4]triazolo[1,5-c] pyrimidine-8-carboxylate1360Federico S et al 2018Jan 15, 2025Jan 15, 2025
93776A1CLONEDHUMAN3H-CCPA5-(2-tert-Butoxycarbonylamino-ethylamino)-2-furan-2-yl-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxylic acid ethyl ester>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93777A2ACLONEDHUMAN3H-NECA5-(2-tert-Butoxycarbonylamino-ethylamino)-2-furan-2-yl-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxylic acid ethyl ester376Federico S et al 2018Jan 15, 2025Jan 15, 2025
93778A3CLONEDHUMAN3H-HEMADO5-(2-tert-Butoxycarbonylamino-ethylamino)-2-furan-2-yl-[1,2,4] triazolo[1,5-c]pyrimidine-8-carboxylic acid ethyl ester129Federico S et al 2018Jan 15, 2025Jan 15, 2025
93779A3CLONEDHUMAN3H-HEMADOEthyl 5-(4-(tert-butoxycarbonyl)piperazin-1-yl)-2-(furan-2-yl)- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93780A2ACLONEDHUMAN3H-NECAEthyl 5-(4-(tert-butoxycarbonyl)piperazin-1-yl)-2-(furan-2-yl)- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93781A1CLONEDHUMAN3H-CCPAEthyl 5-(4-(tert-butoxycarbonyl)piperazin-1-yl)-2-(furan-2-yl)- [1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93782A1CLONEDHUMAN3H-CCPAEthyl 5-(2-(tert-butoxycarbonyl)hydrazinyl)-2-(furan-2-yl)-[1,2,4triazolo[1,5-c]pyrimidine-8-carboxylate>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93783A2ACLONEDHUMAN3H-NECAEthyl 5-(2-(tert-butoxycarbonyl)hydrazinyl)-2-(furan-2-yl)-[1,2,4triazolo[1,5-c]pyrimidine-8-carboxylate827Federico S et al 2018Jan 15, 2025Jan 15, 2025
93784A3CLONEDHUMAN3H-HEMADOEthyl 5-(2-(tert-butoxycarbonyl)hydrazinyl)-2-(furan-2-yl)-[1,2,4triazolo[1,5-c]pyrimidine-8-carboxylate89Federico S et al 2018Jan 15, 2025Jan 15, 2025
93785A3CLONEDHUMAN3H-HEMADO2-(8-Ethoxycarbonyl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin5-ylamino)-ethyl-amine hydrochloride2000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93786A2ACLONEDHUMAN3H-NECA2-(8-Ethoxycarbonyl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin5-ylamino)-ethyl-amine hydrochloride829Federico S et al 2018Jan 15, 2025Jan 15, 2025
93787A1CLONEDHUMAN3H-CCPA2-(8-Ethoxycarbonyl-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidin5-ylamino)-ethyl-amine hydrochloride2340Federico S et al 2018Jan 15, 2025Jan 15, 2025
93788A1CLONEDHUMAN3H-CCPAEthyl 2-(furan-2-yl)-5-(piperazin-1-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93789A2ACLONEDHUMAN3H-NECAEthyl 2-(furan-2-yl)-5-(piperazin-1-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93790A3CLONEDHUMAN3H-HEMADOEthyl 2-(furan-2-yl)-5-(piperazin-1-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93791A3CLONEDHUMAN3H-HEMADOEthyl 2-(furan-2-yl)-5-hydrazinyl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride159Federico S et al 2018Jan 15, 2025Jan 15, 2025
93792A2ACLONEDHUMAN3H-NECAEthyl 2-(furan-2-yl)-5-hydrazinyl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride63.1Federico S et al 2018Jan 15, 2025Jan 15, 2025
93793A1CLONEDHUMAN3H-CCPAEthyl 2-(furan-2-yl)-5-hydrazinyl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylate hydrochloride2080Federico S et al 2018Jan 15, 2025Jan 15, 2025
93794A1CLONEDHUMAN3H-CCPA5-(2-tert-butoxycarbonylamino-ethylamino)-2- furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93795A2ACLONEDHUMAN3H-NECA5-(2-tert-butoxycarbonylamino-ethylamino)-2- furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid>10000Federico S et al 2018Jan 15, 2025Jan 15, 2025
93796A3CLONEDHUMAN3H-HEMADO5-(2-tert-butoxycarbonylamino-ethylamino)-2- furan-2-yl-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxylic acid7750Federico S et al 2018Jan 15, 2025Jan 15, 2025
93797A3CLONEDHUMAN3H-HEMADOEthyl 5-ethoxy-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylate108Federico S et al 2018Jan 15, 2025Jan 15, 2025
93798A2ACLONEDHUMAN3H-NECAEthyl 5-ethoxy-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylate1860Federico S et al 2018Jan 15, 2025Jan 15, 2025
93799A1CLONEDHUMAN3H-CCPAEthyl 5-ethoxy-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]pyrimidine-8- carboxylate4100Federico S et al 2018Jan 15, 2025Jan 15, 2025
938005-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione6.3Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938015-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione4.9Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938025-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion2.3Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938035-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione204.1Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938045-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione246Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938055-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion68.7Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938065-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione48.7Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938075-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione222Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938085-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione240Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938095-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione13Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938105-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione7Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938115-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione3.2Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938125-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione143.2Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938135-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione336Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938145-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dion157Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938155-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione320Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938165-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione700Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938175-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione5000Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938185-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione122Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938195-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[3-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione183Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938205-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyrrolidine-2,5-dione78Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938215-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[3-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione52Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938225-HT1ACLONEDHUMAN3H-8-OH-DPAT5-Hydroxy Tryptamine5.5Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
93823SERTCLONEDHUMAN3H-IMIPRAMINE1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione705Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93824SERTCLONEDHUMAN3H-IMIPRAMINE1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione17.5Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93825SERTCLONEDHUMAN3H-IMIPRAMINE1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion308Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93826SERTCLONEDHUMAN3H-IMIPRAMINE1-{3-[4-(1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione523Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93827SERTCLONEDHUMAN3H-IMIPRAMINE1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione30Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93828SERTCLONEDHUMAN3H-IMIPRAMINE1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion111Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93829SERTCLONEDHUMAN3H-IMIPRAMINE1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione141.8Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93830SERTCLONEDHUMAN3H-IMIPRAMINE1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione221Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93831SERTCLONEDHUMAN3H-IMIPRAMINE1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione63Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93832SERTCLONEDHUMAN3H-IMIPRAMINE1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione51Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93833SERTCLONEDHUMAN3H-IMIPRAMINE1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione32.4Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93834SERTCLONEDHUMAN3H-IMIPRAMINE1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione201Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93835SERTCLONEDHUMAN3H-IMIPRAMINE1-{3-[4-(1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione150.5Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93836SERTCLONEDHUMAN3H-IMIPRAMINE1-{3-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione140Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93837SERTCLONEDHUMAN3H-IMIPRAMINE1-{3-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]propyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dion156Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93838SERTCLONEDHUMAN3H-IMIPRAMINE1-{2-[4-(1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione102Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93839SERTCLONEDHUMAN3H-IMIPRAMINE1-{2-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione314Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93840SERTCLONEDHUMAN3H-IMIPRAMINE1-{2-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]ethyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione1313Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93841SERTCLONEDHUMAN3H-IMIPRAMINEIMIPRAMINE2.5Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
938425-HT1ACLONEDHUMAN3H-8-OH-DPAT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyr-rolidine-2,5-dione7.5Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938435-HT1ACLONEDHUMAN3H-8-OH-DPATMW0112.2Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
93844D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyr-rolidine-2,5-dione14Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93845D2CLONEDHUMAN3H-RACLOPRIDEMW011161Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93846D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione16Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93847D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione62Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93848D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion217Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93849D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione190Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93850D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione19Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
93851D2CLONEDHUMAN3H-RACLOPRIDE1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione20Wrobel MZ et al 2019Jan 15, 2025Jan 28, 2025
938525-HT6CLONEDHUMAN3H-LSD1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyr-rolidine-2,5-dione63Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938535-HT6CLONEDHUMAN3H-LSDMW011159Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938545-HT6CLONEDHUMAN3H-LSD1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione81Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938555-HT6CLONEDHUMAN3H-LSD1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione85Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938565-HT6CLONEDHUMAN3H-LSD1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dion427Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938575-HT6CLONEDHUMAN3H-LSD1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione29Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938585-HT6CLONEDHUMAN3H-LSD1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione301Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938595-HT6CLONEDHUMAN3H-LSD1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione71Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938605-HT7BCLONEDHUMAN3H-5CT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(1H-indol-3-yl)pyr-rolidine-2,5-dione196Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938615-HT7BCLONEDHUMAN3H-5-CTMW011345Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938625-HT7BCLONEDHUMAN3H-5-CT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione25Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938635-HT7BCLONEDHUMAN3H-5-CT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-methoxy-1H-indol-3-yl)pyrrolidine-2,5-dione641Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938645-HT7BCLONEDHUMAN3H-5CT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione320Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938655-HT7BCLONEDHUMAN3H-5CT1-{4-[4-(1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione50Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938665-HT7BCLONEDHUMAN3H-5-CT1-{4-[4-(5-fluoro-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione1158Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938675-HT7BCLONEDHUMAN3H-5CT1-{4-[4-(5-methoxy-1H-indol-3-yl)piperidin-1-yl]butyl}-3-(5-fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione458Wrobel MZ et al 2019Jan 15, 2025Jan 15, 2025
938685-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione22Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938695-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione50Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938705-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione53Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938715-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione102Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938725-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione132Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938735-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion294Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938745-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion46Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938755-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione63Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938765-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione42Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938775-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione209Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938785-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-chlorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione378Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938795-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-fluorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione218Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938805-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione376Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938815-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione80Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938825-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione155Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938835-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-fluorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione147Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938845-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione136Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938855-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dion140Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938865-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione261Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938875-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-chlorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione176Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938885-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2-fluorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione130Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938895-HT1BCLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione476Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938905-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione69Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938915-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-chlorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione257Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938925-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(4-fluorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione281Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938935-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione333Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938945-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione62Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
938955-HT1ACLONEDHUMAN3H-8-OH-DPAT5-Hydroxy Tryptamine3Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
93896SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione68Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93897SERTCORTEXRAT3H-CITALOPRAM4-(2-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione103Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93898SERTCORTEXRAT3H-CITALOPRAM4-(2-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione240Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93899SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione76Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93900SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione411Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93901SERTCORTEXRAT3H-CITALOPRAM4-(4-chlorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion82Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93902SERTCORTEXRAT3H-CITALOPRAM4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion46Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93903SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione207Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93904SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione41Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93905SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione8Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93906SERTCORTEXRAT3H-CITALOPRAM4-(2-chlorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione255Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93907SERTCORTEXRAT3H-CITALOPRAM4-(2-fluorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione115Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93908SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione338Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93909SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione118Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93910SERTCORTEXRAT3H-CITALOPRAM4-(4-chlorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione86Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93911SERTCORTEXRAT3H-CITALOPRAM4-(4-fluorophenyl)-2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione30Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93912SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione135Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93913SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-fluoro-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dion27Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93914SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione248Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93915SERTCORTEXRAT3H-CITALOPRAM4-(2-chlorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione459Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93916SERTCORTEXRAT3H-CITALOPRAM4-(2-fluorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione1670Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93917SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(o-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione87Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93918SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(2-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione386Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93919SERTCORTEXRAT3H-CITALOPRAM4-(4-chlorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione490Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93920SERTCORTEXRAT3H-CITALOPRAM4-(4-fluorophenyl)-2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dione192Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93921SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(p-tolyl)pyrido[1,2-c]pyrimidine-1,3-dione173Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93922SERTCORTEXRAT3H-CITALOPRAM2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione86Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93923SERTCORTEXRAT3H-CITALOPRAMIMIPRAMINE29Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
939245-HT2ACLONEDHUMAN3H-KETANSERIN2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione433Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939255-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion435Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939265-HT2ACLONEDHUMAN3H-KETANSERIN2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione21Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939275-HT2ACLONEDHUMAN3H-KETANSERIN2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione314Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939285-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE4.6Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939295-HT2ACLONEDHUMAN3H-KETANSERINmianserine2.8Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939305-HT6CLONEDHUMAN3H-LSD2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione435Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939315-HT6CLONEDHUMAN3H-LSD4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion697Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939325-HT6CLONEDHUMAN3H-LSD2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione1709Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939335-HT6CLONEDHUMAN3H-LSD2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione690Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939345-HT6CLONEDHUMAN3H-LSDOLANZAPINE7Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939355-HT7CLONEDHUMAN3H-5CT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione1115Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939365-HT7CLONEDHUMAN3H-5-CT4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion1444Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939375-HT7CLONEDHUMAN3H-5CT2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione1922Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939385-HT7CLONEDHUMAN3H-5-CT2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione958Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
939395-HT7CLONEDHUMAN3H-5-CTCLOZAPINE18Slifirski G et al 2019Jan 15, 2025Jan 15, 2025
93940D2CLONEDHUMAN3H-RACLOPRIDE2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-phenyl-pyrido[1,2-c]pyrimidine-1,3-dione>10000Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93941D2CLONEDHUMAN3H-RACLOPRIDE4-(4-fluorophenyl)-2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]pyrido[1,2-c]pyrimidine-1,3-dion963Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93942D2CLONEDHUMAN3H-RACLOPRIDE2-[4-[3-(1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione1129Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93943D2CLONEDHUMAN3H-RACLOPRIDE2-[4-[3-(5-methoxy-1H-indol-3-yl)-1-piperidyl]butyl]-4-(4-methoxyphenyl)pyrido[1,2-c]pyrimidine-1,3-dione>10000Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93944D2CLONEDHUMAN3H-RACLOPRIDEHALOPERIDOL4.5Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93945D2CLONEDHUMAN3H-RACLOPRIDEAPOMORPHINE42Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93946D2CLONEDHUMAN3H-RACLOPRIDECHLORPROMAZINE1.8Slifirski G et al 2019Jan 15, 2025Jan 28, 2025
93947D1STRIATUMPIG3H-SCH23390compound 422500Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93948D1STRIATUMPIG3H-SCH23390compound 432900Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93949D1STRIATUMPIG3H-SCH233903,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one2100Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93950D1STRIATUMPIG3H-SCH233907-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one2300Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93951D1STRIATUMPIG3H-SCH233903,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one640Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93952D1STRIATUMPIG3H-SCH233903,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one220Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93953D1STRIATUMPIG3H-SCH233903,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one580Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93954D1STRIATUMPIG3H-SCH233903,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one480Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93955D1STRIATUMPIG3H-SCH233902-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one920Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93956D1STRIATUMPIG3H-SCH233903,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one380Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93957D1STRIATUMPIG3H-SCH233902-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile3200Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93958D1STRIATUMPIG3H-SCH233903,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one1900Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93959D2CLONEDHUMAN3H-SPIPERONEcompound 4221Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93960D2CLONEDHUMAN3H-SPIPERONEcompound 433.9Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93961D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one3.2Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93962D2CLONEDHUMAN3H-SPIPERONE7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one26Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93963D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one38Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93964D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one52Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93965D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one16Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93966D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one11Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93967D2CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one5.1Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93968D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one7.1Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93969D2CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile38Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93970D2CLONEDHUMAN3H-SPIPERONE40 3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one24Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93971D2CLONEDHUMAN3H-SPIPERONEcompound 427Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93972D2CLONEDHUMAN3H-SPIPERONEcompound 431.5Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93973D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one0.93Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93974D2CLONEDHUMAN3H-SPIPERONE7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one9.2Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93975D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one15Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93976D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one63Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93977D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one4.8Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93978D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one6.9Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93979D2CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one2.1Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93980D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one13Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93981D2CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile22Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93982D2CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one8.8Ortega R et al 2011Jan 15, 2025Jan 29, 2025
93983D3CLONEDHUMAN3H-SPIPERONEcompound 421.7Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93984D3CLONEDHUMAN3H-SPIPERONEcompound 430.27Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93985D3CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one0.27Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93986D3CLONEDHUMAN3H-SPIPERONE7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one1.6Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93987D3CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one0.25Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93988D3CLONEDHUMAN3H-SCH233903,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one12Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93989D3CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one0.21Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93990D3CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one0.12Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93991D3CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one0.29Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93992D3CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one0.12Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93993D3CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile1.3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93994D3CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one0.5Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93995D4CLONEDHUMAN3H-SPIPERONEcompound 421.9Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93996D4CLONEDHUMAN3H-SPIPERONEcompound 431.3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93997D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93998D4CLONEDHUMAN3H-SPIPERONE7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one2.8Ortega R et al 2011Jan 15, 2025Jan 28, 2025
93999D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one3.4Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94000D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one9.8Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94001D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one3.3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94002D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one2.3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94003D4CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one2.9Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94004D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one3.4Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94005D4CLONEDHUMAN3H-SPIPERONE2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile6.1Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94006D4CLONEDHUMAN3H-SPIPERONE3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one4.1Ortega R et al 2011Jan 15, 2025Jan 28, 2025
940075-HT1ACORTEXPIG[3H]WAY 600135compound 422.4Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940085-HT1ACORTEXPIG[3H]WAY 600135compound 431.7Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940095-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one2.5Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940105-HT1ACORTEXPIG[3H]WAY 6001357-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one1.7Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940115-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one38Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940125-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one47Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940135-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one19Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940145-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one6.2Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940155-HT1ACORTEXPIG[3H]WAY 6001352-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one68Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940165-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one13Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940175-HT1ACORTEXPIG[3H]WAY 6001352-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile3.8Ortega R et al 2011Jan 15, 2025Jan 15, 2025
940185-HT1ACORTEXPIG[3H]WAY 6001353,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one14Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94019CORTEXPIG3H-KETANSERINcompound 42990Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94020CORTEXPIG3H-KETANSERINcompound 431100Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94021CORTEXPIG3H-KETANSERIN3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one810Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94022CORTEXPIG3H-KETANSERIN7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one840Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94023CORTEXPIG3H-KETANSERIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one330Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94024CORTEXPIG3H-KETANSERIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one230Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94025CORTEXPIG3H-KETANSERIN3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one330Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94026CORTEXPIG3H-KETANSERIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one190Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94027CORTEXPIG3H-KETANSERIN2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one530Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94028CORTEXPIG3H-KETANSERIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one160Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94029CORTEXPIG3H-KETANSERIN2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile430Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94030CORTEXPIG3H-KETANSERIN3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one920Ortega R et al 2011Jan 15, 2025Jan 15, 2025
94031Alpha1ACORTEXPIG3H-PRAZOSINcompound 422.3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94032Alpha1ACORTEXPIG3H-PRAZOSINcompound 435.7Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94033Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-6-fluoro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one3.7Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94034Alpha1ACORTEXPIG3H-PRAZOSIN7-Methoxy-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydrobenzo[c]azepin-1-one3.1Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94035Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-phenylisoquinolin-1(2H)-one5.4Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94036Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-5-phenylisoquinolin-1(2H)-one1.3Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94037Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one1.6Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94038Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(2-thienyl)isoquinolin-1(2H)-one3.7Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94039Alpha1ACORTEXPIG3H-PRAZOSIN2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3,4,5-tetrahydro-7-(2-thienyl)benzo[c]azepin-1-one9.7Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94040Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]-6-(4-pyridyl)isoquinolin-1(2H)-one2.2Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94041Alpha1ACORTEXPIG3H-PRAZOSIN2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-6-carbonitrile3.8Ortega R et al 2011Jan 15, 2025Jan 28, 2025
94042Alpha1ACORTEXPIG3H-PRAZOSIN3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl]isoquinolin-1(2H)-one2.4Ortega R et al 2011Jan 15, 2025Jan 28, 2025
940435-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-methylthiophenethylamine1035Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940445-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-dimethoxy-4-(b-methallyl)thio-phenethylamine812Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940455-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-isopropylthiophenethylamine916Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940465-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-propylthiophenethylamine878Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940475-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-allylthiophenethylamine660Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940485-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-n-butylthiophenethylamine1019Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940495-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine1321Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940505-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine1915Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940515-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-isobutylthiophenethylamine1036Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940525-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-benzylthiophenethylamine,1166Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940535-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine1904Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940545-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine2368Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940555-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine1063Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940565-HT1ACLONEDHUMAN[3H]-8-OH-DPAT2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine1411Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940575-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-Bromo-2,5-dimethoxyphenethylamine311Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940585-HT1ACLONEDHUMAN[3H]-8-OH-DPATLSD1.5Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940595-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-methylthiophenethylamine49Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940605-HT2ACLONEDHUMAN[3H]-ketanserin5-dimethoxy-4-(b-methallyl)thio-phenethylamine11Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940615-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-isopropylthiophenethylamine54Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940625-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-propylthiophenethylamine5.3Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940635-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-allylthiophenethylamine9.2Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940645-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-n-butylthiophenethylamine6.98Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940655-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine14Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940665-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine16Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940675-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-isobutylthiophenethylamine21Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940685-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-benzylthiophenethylamine1.6Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940695-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine17Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940705-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine9.5Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940715-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine3.8Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940725-HT2ACLONEDHUMAN[3H]-ketanserin2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine17Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940735-HT2ACLONEDHUMAN[3H]-ketanserin4-Bromo-2,5-dimethoxyphenethylamine6.9Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940745-HT2ACLONEDHUMAN[3H]-ketanserinLSD5.3Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940755-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-methylthiophenethylamine347Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940765-HT2CCLONEDHUMAN[3H]-mesulergine5-dimethoxy-4-(b-methallyl)thio-phenethylamine40Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940775-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-isopropylthiophenethylamine295Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940785-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-propylthiophenethylamine54Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940795-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-allylthiophenethylamine67Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940805-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-n-butylthiophenethylamine101Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940815-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine159Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940825-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine151Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940835-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-isobutylthiophenethylamine80Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940845-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-benzylthiophenethylamine52Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940855-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine135Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940865-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine158Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940875-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine157Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940885-HT2CCLONEDHUMAN[3H]-mesulergine2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine75Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940895-HT2CCLONEDHUMAN[3H]-mesulergine4-Bromo-2,5-dimethoxyphenethylamine43Luethi D et al 2018Jan 15, 2025Jan 15, 2025
940905-HT2CCLONEDHUMAN[3H]-mesulergineLSD14Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94091TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-methylthiophenethylamine52Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94092TAAR1CLONEDRAT[3H]-RO51660175-dimethoxy-4-(b-methallyl)thio-phenethylamine8Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94093TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-isopropylthiophenethylamine19Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94094TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-propylthiophenethylamine10Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94095TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-allylthiophenethylamine17Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94096TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-n-butylthiophenethylamine4.8Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94097TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine68Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94098TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine38Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94099TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-isobutylthiophenethylamine11Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94100TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-benzylthiophenethylamine10Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94101TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine62Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94102TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine29Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94103TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine5.2Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94104TAAR1CLONEDRAT[3H]-RO51660172,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine38Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94105TAAR1CLONEDRAT[3H]-RO5166017d-Methamphetamine257Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94106TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-methylthiophenethylamine1877Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94107TAAR1CLONEDMOUSE[3H]-RO51660175-dimethoxy-4-(b-methallyl)thio-phenethylamine465Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94108TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-isopropylthiophenethylamine2337Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94109TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-propylthiophenethylamine311Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94110TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-allylthiophenethylamine453Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94111TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-n-butylthiophenethylamine96Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94112TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine1674Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94113TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine974Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94114TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-isobutylthiophenethylamine359Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94115TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-benzylthiophenethylamine596Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94116TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine426Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94117TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine182Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94118TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine55Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94119TAAR1CLONEDMOUSE[3H]-RO51660172,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine761Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94120TAAR1CLONEDMOUSE[3H]-RO5166017d-Methamphetamine889Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94121Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-methylthiophenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94122Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-isopropylthiophenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94123Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-propylthiophenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94124Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-n-butylthiophenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94125Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94126Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94127Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-isobutylthiophenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94128Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-benzylthiophenethylamine6510Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94129Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine2730Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94130Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine2297Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94131Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine2534Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94132Alpha1ACLONEDHUMAN[3H]-prazosin2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine3628Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94133Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-methylthiophenethylamine334Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94134Alpha2ACLONEDHUMAN[3H]-rauwolscine5-dimethoxy-4-(b-methallyl)thio-phenethylamine97Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94135Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-isopropylthiophenethylamine217Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94136Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-propylthiophenethylamine335Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94137Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-allylthiophenethylamine229Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94138Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-n-butylthiophenethylamine458Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94139Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine383Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94140Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine592Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94141Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-isobutylthiophenethylamine279Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94142Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-benzylthiophenethylamine351Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94143Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine331Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94144Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine408Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94145Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine804Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94146Alpha2ACLONEDHUMAN[3H]-rauwolscine2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine343Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94147D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-methylthiophenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94148D2CLONEDHUMAN[3H]-spiperone5-dimethoxy-4-(b-methallyl)thio-phenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94149D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-isopropylthiophenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94150D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-propylthiophenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94151D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-allylthiophenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94152D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-n-butylthiophenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94153D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94154D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine4400Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94155D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-isobutylthiophenethylamine6270Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94156D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-benzylthiophenethylamine6270Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94157D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine6270Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94158D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine6270Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94159D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine6270Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94160D2CLONEDHUMAN[3H]-spiperone2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine6270Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94161NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-methylthiophenethylamine9710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94162NETCLONEDHUMANN-methyl-[3H]-nisoxetine5-dimethoxy-4-(b-methallyl)thio-phenethylamine9710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94163NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-isopropylthiophenethylamine9710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94164NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-propylthiophenethylamine9710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94165NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-allylthiophenethylamine9710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94166NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-n-butylthiophenethylamine9710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94167NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94168NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94169NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-isobutylthiophenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94170NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-benzylthiophenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94171NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94172NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94173NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94174NETCLONEDHUMANN-methyl-[3H]-nisoxetine2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine9720Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94175DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-methylthiophenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94176DATCLONEDHUMAN[3H]-citalopram5-dimethoxy-4-(b-methallyl)thio-phenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94177DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-isopropylthiophenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94178DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-propylthiophenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94179DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-allylthiophenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94180DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-n-butylthiophenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94181DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94182DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94183DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-isobutylthiophenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94184DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-benzylthiophenethylamine4760Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94185DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94186DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine8710Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94187DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine5474Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94188DATCLONEDHUMAN[3H]-citalopram2,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine7706Luethi D et al 2018Jan 15, 2025Jan 15, 2025
94189SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-methylthiophenethylamine8580Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94190SERTCLONEDHUMAN[3H]-WIN35,4285-dimethoxy-4-(b-methallyl)thio-phenethylamine7221Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94191SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-isopropylthiophenethylamine8580Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94192SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-propylthiophenethylamine8580Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94193SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-allylthiophenethylamine8580Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94194SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-n-butylthiophenethylamine8580Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94195SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-(2,2-difluoroethylthio)phenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94196SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-(2,2,2-trifluoroethylthio)phenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94197SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-isobutylthiophenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94198SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-benzylthiophenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94199SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-(3-fluoropropylthio)phene-thylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94200SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-(4-fluorobutylthio)phenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94201SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-(4-trifluoromethylbenzylthio)phenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
94202SERTCLONEDHUMAN[3H]-WIN35,4282,5-dimethoxy-4-(3-methoxybenzylthio)phenethylamine7510Luethi D et al 2018Jan 15, 2025Jan 28, 2025
942035-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-ethoxyphenethylamine3600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942045-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-methallyloxyphenethylamine2700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942055-HT1ACLONEDHUMAN3H-8-OH-DPAT4-allyloxy-2,5-dimethoxyphenethylamine4500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942065-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine5500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942075-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine2900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942085-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine3300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942095-HT1ACLONEDHUMAN3H-8-OH-DPAT4-benzyloxy-2,5-dimethoxyphenethylamine2700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942105-HT1ACLONEDHUMAN3H-8-OH-DPAT4-allyloxy-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942115-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942125-HT1ACLONEDHUMAN3H-8-OH-DPAT4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942135-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942145-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-isopropoxyamphetamine5600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942155-HT1ACLONEDHUMAN3H-8-OH-DPAT2,4,5-trimethoxyamphetamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942165-HT1ACLONEDHUMAN3H-8-OH-DPAT4-Bromo-2,5-dimethoxyphenethylamine311Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942175-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-ethoxyphenethylamine670Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942185-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-methallyloxyphenethylamine40Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942195-HT2ACLONEDHUMAN3H-KETANSERIN4-allyloxy-2,5-dimethoxyphenethylamine140Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942205-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine1700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942215-HT2ACLONEDHUMAN3H-KETANSERIN4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine1000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942225-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine440Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942235-HT2ACLONEDHUMAN3H-KETANSERIN4-benzyloxy-2,5-dimethoxyphenethylamine8.1Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942245-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-methallyloxyamphetamine61Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942255-HT2ACLONEDHUMAN3H-KETANSERIN4-allyloxy-2,5-dimethoxyamphetamine150Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942265-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine1900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942275-HT2ACLONEDHUMAN3H-KETANSERIN4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine980Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942285-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine460Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942295-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-isopropoxyamphetamine4400Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942305-HT2ACLONEDHUMAN3H-KETANSERIN2,4,5-trimethoxyamphetamine1300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942315-HT2ACLONEDHUMAN3H-KETANSERIN4-Bromo-2,5-dimethoxyphenethylamine6.9Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942325-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-ethoxyphenethylamine2300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942335-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-methallyloxyphenethylamine150Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942345-HT2CCLONEDHUMAN3H-MESULERGINE4-allyloxy-2,5-dimethoxyphenethylamine470Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942355-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine3600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942365-HT2CCLONEDHUMAN3H-MESULERGINE4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine4200Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942375-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine1900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942385-HT2CCLONEDHUMAN3H-MESULERGINE4-benzyloxy-2,5-dimethoxyphenethylamine110Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942395-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-methallyloxyamphetamine290Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942405-HT2CCLONEDHUMAN3H-MESULERGINE4-allyloxy-2,5-dimethoxyamphetamine900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942415-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942425-HT2CCLONEDHUMAN3H-MESULERGINE4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine6700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942435-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine2400Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942445-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-isopropoxyamphetamine9030Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942455-HT2CCLONEDHUMAN3H-MESULERGINE2,4,5-trimethoxyamphetamine5300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
942465-HT2CCLONEDHUMAN3H-MESULERGINE4-Bromo-2,5-dimethoxyphenethylamine43Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94247TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-ethoxyphenethylamine340Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94248TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-methallyloxyphenethylamine130Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94249TAAR1CLONEDRAT3H-RO51660174-allyloxy-2,5-dimethoxyphenethylamine260Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94250TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine410Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94251TAAR1CLONEDRAT3H-RO51660174-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine250Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94252TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine240Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94253TAAR1CLONEDRAT3H-RO51660174-benzyloxy-2,5-dimethoxyphenethylamine21Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94254TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-methallyloxyamphetamine630Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94255TAAR1CLONEDRAT3H-RO51660174-allyloxy-2,5-dimethoxyamphetamine1100Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94256TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-(2-fluoroethoxy)amphetamine1640Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94257TAAR1CLONEDRAT3H-RO51660174-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine1200Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94258TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine1300Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94259TAAR1CLONEDRAT3H-RO51660172,5-dimethoxy-4-isopropoxyamphetamine2900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94260TAAR1CLONEDHUMAN3H-RO51660172,4,5-trimethoxyamphetamine3100Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94261TAAR1CLONEDRAT3H-RO51660174-Bromo-2,5-dimethoxyphenethylamine370Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94262TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-ethoxyphenethylamine4000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94263TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-methallyloxyphenethylamine1100Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94264TAAR1CLONEDMOUSE3H-RO51660174-allyloxy-2,5-dimethoxyphenethylamine2500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94265TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine4900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94266TAAR1CLONEDMOUSE3H-RO51660174-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94267TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine2500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94268TAAR1CLONEDMOUSE3H-RO51660174-benzyloxy-2,5-dimethoxyphenethylamine650Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94269TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-methallyloxyamphetamine1700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94270TAAR1CLONEDMOUSE3H-RO51660174-allyloxy-2,5-dimethoxyamphetamine2000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94271TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-(2-fluoroethoxy)amphetamine4900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94272TAAR1CLONEDMOUSE3H-RO51660174-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94273TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine4500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94274TAAR1CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-isopropoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94275TAAR1CLONEDMOUSE3H-RO51660172,4,5-trimethoxyamphetamine4400Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94276TAAR1CLONEDMOUSE3H-RO51660174-Bromo-2,5-dimethoxyphenethylamine2400Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94277Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-ethoxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94278Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-methallyloxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94279Alpha1ACLONEDHUMAN3H-PRAZOSIN4-allyloxy-2,5-dimethoxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94280Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94281Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94282Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94283Alpha1ACLONEDHUMAN3H-PRAZOSIN4-benzyloxy-2,5-dimethoxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94284Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-methallyloxyamphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94285Alpha1ACLONEDHUMAN3H-PRAZOSIN4-allyloxy-2,5-dimethoxyamphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94286Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94287Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94288Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94289Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-isopropoxyamphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94290Alpha1ACLONEDHUMAN3H-PRAZOSIN2,4,5-trimethoxyamphetamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94291Alpha1ACLONEDHUMAN3H-PRAZOSIN4-Bromo-2,5-dimethoxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94292Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-ethoxyphenethylamine2600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94293Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-methallyloxyphenethylamine180Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94294Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-allyloxy-2,5-dimethoxyphenethylamine620Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94295Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine3600Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94296Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine1900Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94297Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine1800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94298Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-benzyloxy-2,5-dimethoxyphenethylamine570Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94299Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-methallyloxyamphetamine2400Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94300Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-allyloxy-2,5-dimethoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94301Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94302Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94303Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94304Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-isopropoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94305Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,4,5-trimethoxyamphetamine4700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94306Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-Bromo-2,5-dimethoxyphenethylamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94307D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-ethoxyphenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94308D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-methallyloxyphenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94309D2CLONEDHUMAN3H-SPIPERONE4-allyloxy-2,5-dimethoxyphenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94310D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94311D2CLONEDHUMAN3H-SPIPERONE4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94312D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94313D2CLONEDHUMAN3H-SPIPERONE4-benzyloxy-2,5-dimethoxyphenethylamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94314D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-methallyloxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94315D2CLONEDHUMAN3H-SPIPERONE4-allyloxy-2,5-dimethoxyamphetamine4400Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94316D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94317D2CLONEDHUMAN3H-SPIPERONE4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94318D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94319D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-isopropoxyamphetamine4800Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94320D2CLONEDHT293H-SPIPERONE2,4,5-trimethoxyamphetamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94321D2CLONEDHUMAN3H-SPIPERONE4-Bromo-2,5-dimethoxyphenethylamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94322NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-ethoxyphenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94323NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-methallyloxyphenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94324NETCLONEDHUMANn-methyl-[3h]nisoxetine4-allyloxy-2,5-dimethoxyphenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94325NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94326NETCLONEDHUMANn-methyl-[3h]nisoxetine4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94327NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94328NETCLONEDHUMANn-methyl-[3h]nisoxetine4-benzyloxy-2,5-dimethoxyphenethylamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94329NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-methallyloxyamphetamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94330NETCLONEDHUMANn-methyl-[3h]nisoxetine4-allyloxy-2,5-dimethoxyamphetamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94331NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94332NETCLONEDHUMANn-methyl-[3h]nisoxetine4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94333NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94334NETCLONEDHUMANn-methyl-[3h]nisoxetine2,5-dimethoxy-4-isopropoxyamphetamine9700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94335NETCLONEDHUMANn-methyl-[3h]nisoxetine2,4,5-trimethoxyamphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94336NETCLONEDHUMANn-methyl-[3h]nisoxetine4-Bromo-2,5-dimethoxyphenethylamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94337DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-ethoxyphenethylamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94338DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-methallyloxyphenethylamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94339DATCLONEDHUMAN3H-WIN 35,4284-allyloxy-2,5-dimethoxyphenethylamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94340DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94341DATCLONEDHUMAN3H-WIN 35,4284-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94342DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94343DATCLONEDHUMAN3H-WIN 35,4284-benzyloxy-2,5-dimethoxyphenethylamine6100Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94344DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-methallyloxyamphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94345DATCLONEDHUMAN3H-WIN 35,4284-allyloxy-2,5-dimethoxyamphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94346DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-(2-fluoroethoxy)amphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94347DATCLONEDHUMAN3H-WIN 35,4284-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94348DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94349DATCLONEDHUMAN3H-WIN354282,5-dimethoxy-4-isopropoxyamphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94350DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-isopropoxyamphetamine8700Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94351DATCLONEDHUMAN3H-WIN 35,4282,4,5-trimethoxyamphetamine8500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94352DATCLONEDHUMAN3H-WIN 35,4284-Bromo-2,5-dimethoxyphenethylamine6500Kolaczynska KE et al 2019Jan 15, 2025Jan 15, 2025
94353SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-ethoxyphenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94354SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-methallyloxyphenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94355SERTCLONEDHUMAN3H-CITALOPRAM4-allyloxy-2,5-dimethoxyphenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94356SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-(2-fluoroethoxy)phenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94357SERTCLONEDHUMAN3H-CITALOPRAM4-(2,2-difluoroethoxy)-2,5-dimethoxyphenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94358SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)phenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94359SERTCLONEDHUMAN3H-CITALOPRAM4-benzyloxy-2,5-dimethoxyphenethylamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94360SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-methallyloxyamphetamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94361SERTCLONEDHUMAN3H-CITALOPRAM4-allyloxy-2,5-dimethoxyamphetamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94362SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-(2-fluoroethoxy)amphetamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94363SERTCLONEDHUMAN3H-CITALOPRAM4-(2,2-difluoroethoxy)-2,5-dimethoxyamphetamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94364SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-(2,2,2-trifluoroethoxy)amphetamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94365SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-isopropoxyamphetamine8600Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94366SERTCLONEDHUMAN3H-CITALOPRAM2,4,5-trimethoxyamphetamine7500Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94367SERTCLONEDHUMAN3H-CITALOPRAM4-Bromo-2,5-dimethoxyphenethylamine>10000Kolaczynska KE et al 2019Jan 15, 2025Jan 28, 2025
94368A1CLONEDHUMAN3H-CCPAEthyl 2-(4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94369A1CLONEDHUMAN3H-CCPAEthyl 2-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94370A1CLONEDHUMAN3H-CCPAEthyl 2-(4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94371A1CLONEDHUMAN3H-CCPAEthyl 2-(2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94372A1CLONEDHUMAN3H-CCPAEthyl 2-(2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate7750Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94373A1CLONEDHUMAN3H-CCPAEthyl 2-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94374A1CLONEDHUMAN3H-CCPAEthyl 2-(4-(dimethylamino)-2-((methoxycarbonyl)amino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94375A1CLONEDHUMAN3H-CCPAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94376A1CLONEDHUMAN3H-CCPAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4- (dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94377A1CLONEDHUMAN3H-CCPAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94378A1CLONEDHUMAN3H-CCPAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamide2380Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94379A1CLONEDHUMAN3H-CCPAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94380A1CLONEDHUMAN3H-CCPAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94381A1CLONEDHUMAN3H-CCPAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94382A1CLONEDHUMAN3H-CCPAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-methyl-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94383A1CLONEDHUMAN3H-CCPA4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-((4-methoxyphenyl)amino) thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94384A1CLONEDHUMAN3H-CCPA4-Ethyl 2-methyl 3-methyl-5-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)thiophene-2,4-dicarboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94385A1CLONEDHUMAN3H-CCPA4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94386A2ACLONEDHUMAN3H-NECAEthyl 2-(4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate6450Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94387A2ACLONEDHUMAN3H-NECAEthyl 2-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94388A2ACLONEDHUMAN3H-NECAEthyl 2-(4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94389A2ACLONEDHUMAN3H-NECAEthyl 2-(2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94390A2ACLONEDHUMAN3H-NECAEthyl 2-(2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94391A2ACLONEDHUMAN3H-NECAEthyl 2-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94392A2ACLONEDHUMAN3H-NECAEthyl 2-(4-(dimethylamino)-2-((methoxycarbonyl)amino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94393A2ACLONEDHUMAN3H-NECAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94394A2ACLONEDHUMAN3H-NECAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4- (dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94395A2ACLONEDHUMAN3H-NECAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94396A2ACLONEDHUMAN3H-NECAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamide3440Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94397A2ACLONEDHUMAN3H-NECAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94398A2ACLONEDHUMAN3H-NECAN-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94399A2ACLONEDHUMAN3H-NECAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94400A2ACLONEDHUMAN3H-NECAN-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-methyl-2-(p-tolylamino)thiazole-5-carboxamide5670Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94401A2ACLONEDHUMAN3H-NECA4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-((4-methoxyphenyl)amino) thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate9660Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94402A2ACLONEDHUMAN3H-NECA4-Ethyl 2-methyl 3-methyl-5-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)thiophene-2,4-dicarboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94403A2ACLONEDHUMAN3H-NECA4-Ethyl 2-methyl 3-methyl-5-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)thiophene-2,4-dicarboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94404A3CLONEDHUMAN3H-HEMADOEthyl 2-(4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate4120Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94405A3CLONEDHUMAN3H-HEMADOEthyl 2-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate8220Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94406A3CLONEDHUMAN3H-HEMADOEthyl 2-(4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate2160Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94407A3CLONEDHUMAN3H-HEMADOEthyl 2-(2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate520Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94408A3CLONEDHUMAN3H-HEMADOEthyl 2-(2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate4090Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94409A3CLONEDHUMAN3H-HEMADOEthyl 2-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate4710Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94410A3CLONEDHUMAN3H-HEMADOEthyl 2-(4-(dimethylamino)-2-((methoxycarbonyl)amino)thiazole-5-carboxamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94411A3CLONEDHUMAN3H-HEMADON-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94412A3CLONEDHUMAN3H-HEMADON-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(phenylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94413A3CLONEDHUMAN3H-HEMADON-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4- (dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94414A3CLONEDHUMAN3H-HEMADON-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamide7130Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94415A3CLONEDHUMAN3H-HEMADON-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-(phenylamino)-4-(p-tolyl)thiazole-5-carboxamide334Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94416A3CLONEDHUMAN3H-HEMADON-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94417A3CLONEDHUMAN3H-HEMADON-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-2-((4-methoxyphenyl)amino)-4-(p-tolyl)thiazole-5-carboxamide9560Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94418A3CLONEDHUMAN3H-HEMADON-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-(p-tolyl)-2-(p-tolylamino)thiazole-5-carboxamide330Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94419A3CLONEDHUMAN3H-HEMADON-(3-carbamoyl-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)-4-methyl-2-(p-tolylamino)thiazole-5-carboxamide3870Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94420A3CLONEDHUMAN3H-HEMADO4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-((4-methoxyphenyl)amino) thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate2730Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94421A3CLONEDHUMAN3H-HEMADO4-Ethyl 2-methyl 3-methyl-5-(4-methyl-2-(p-tolylamino)thiazole-5-carboxamido)thiophene-2,4-dicarboxylate>10000Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94422A3CLONEDHUMAN3H-HEMADO4-Ethyl 2-methyl 5-(4-(dimethylamino)-2-(p-tolylamino)thiazole-5-carboxamido)-3-methylthiophene-2,4-dicarboxylate3910Pandya DH et al 2015Jan 15, 2025Jan 15, 2025
94423A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-methyl2-(phenylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94424A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94425A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-phenyl-2- (phenylamino)thiazol-5-yl)methanone6710Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94426A1CLONEDHUMAN3H-CCPAN-(5-(2-Amino-1-(4-chlorophenyl)-1H-imidazole-5-carbonyl)-4-(dimethylamino)thiazol-2-yl)benzamide>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94427A1CLONEDHUMAN3H-CCPAN-(5-(2-Amino-1-(4-(trifluoromethyl)phenyl)-1H-imidazole5-carbonyl)-4IJdimethylamino)thiazol-2-yl)benzamide>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94428A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (p-tolylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94429A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-phenyl2-(phenylamino) thiazol-5-yl)methanone3670Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94430A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2- morpholino-4-phenylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94431A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ2-(4-chlorophenylamino)-4-methylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94432A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2-(4- chlorophenylamino)-4-methylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94433A1CLONEDHUMAN3H-CCPA(2-Amino-1-p-tolyl-1H-imidazol-5-yl)IJ2-morpholino-4- phenylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94434A1CLONEDHUMAN3H-CCPA(2-Amino-1-(4-chlorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94435A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-methyl2-(phenylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94436A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone8040Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94437A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-phenyl-2- (phenylamino)thiazol-5-yl)methanone7410Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94438A2ACLONEDHUMAN3H-NECAN-(5-(2-Amino-1-(4-chlorophenyl)-1H-imidazole-5-carbonyl)-4-(dimethylamino)thiazol-2-yl)benzamide>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94439A2ACLONEDHUMAN3H-NECAN-(5-(2-Amino-1-(4-(trifluoromethyl)phenyl)-1H-imidazole5-carbonyl)-4IJdimethylamino)thiazol-2-yl)benzamide>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94440A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (p-tolylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94441A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-phenyl2-(phenylamino) thiazol-5-yl)methanone8840Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94442A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2- morpholino-4-phenylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94443A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ2-(4-chlorophenylamino)-4-methylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94444A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2-(4- chlorophenylamino)-4-methylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94445A2ACLONEDHUMAN3H-NECA(2-Amino-1-p-tolyl-1H-imidazol-5-yl)IJ2-morpholino-4- phenylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94446A2ACLONEDHUMAN3H-NECA(2-Amino-1-(4-chlorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94447A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-methyl2-(phenylamino)thiazol-5-yl)methanone574Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94448A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone190Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94449A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-phenyl-2- (phenylamino)thiazol-5-yl)methanone305Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94450A3CLONEDHUMAN3H-HEMADON-(5-(2-Amino-1-(4-chlorophenyl)-1H-imidazole-5-carbonyl)-4-(dimethylamino)thiazol-2-yl)benzamide4320Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94451A3CLONEDHUMAN3H-HEMADON-(5-(2-Amino-1-(4-(trifluoromethyl)phenyl)-1H-imidazole5-carbonyl)-4IJdimethylamino)thiazol-2-yl)benzamide4920Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94452A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (p-tolylamino)thiazol-5-yl)methanone487Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94453A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ4-phenyl2-(phenylamino) thiazol-5-yl)methanone326Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94454A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2- morpholino-4-phenylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94455A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-fluorophenyl)-1H-imidazol-5-yl)IJ2-(4-chlorophenylamino)-4-methylthiazol-5-yl)methanone871Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94456A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-methoxyphenyl)-1H-imidazol-5-yl)IJ2-(4- chlorophenylamino)-4-methylthiazol-5-yl)methanone1600Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94457A3CLONEDHUMAN3H-HEMADO(2-Amino-1-p-tolyl-1H-imidazol-5-yl)IJ2-morpholino-4- phenylthiazol-5-yl)methanone>10000Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94458A3CLONEDHUMAN3H-HEMADO(2-Amino-1-(4-chlorophenyl)-1H-imidazol-5-yl)IJ4-methyl-2- (phenylamino)thiazol-5-yl)methanone802Pandya AN et al 2018Jan 15, 2025Jan 15, 2025
94459A3C.H.O.? HUMAN3H-HEMADO{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indol-7-yl}azinic acid>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94460A3C.H.O.? HUMAN3H-HEMADO2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94461A3C.H.O.? HUMAN3H-HEMADO2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94462A3C.H.O.? HUMAN3H-HEMADO2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-fluoro-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94463A3C.H.O.? HUMAN3H-HEMADO2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94464A3C.H.O.? HUMAN3H-HEMADO3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-7-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94465A3C.H.O.? HUMAN3H-HEMADO1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(6-fluoro-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94466A3C.H.O.? HUMAN3H-HEMADO1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(1H-indol-3-yl)ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94467A3C.H.O.? HUMAN3H-HEMADO2-(5-Bromo-7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94468A3C.H.O.? HUMAN3H-HEMADO5-Chloro-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94469A3C.H.O.? HUMAN3H-HEMADO1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl) ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94470A3C.H.O.? HUMAN3H-HEMADO3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94471A3C.H.O.? HUMAN3H-HEMADO3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-4-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94472A3C.H.O.? HUMAN3H-HEMADO3-{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]ethyl}-2-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94473A3C.H.O.? HUMAN3H-HEMADO3-{[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94474A3C.H.O.? HUMAN3H-HEMADO1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94475A3C.H.O.? HUMAN3H-HEMADO3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94476A2BC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94477A2AC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94478A2AC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1- one8710Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94479A2BC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94480A2BC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-3-(1H-indol-3-yl)propan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94481A2AC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-3-(1H-indol-3-yl)propan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94482A2AC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-4-(1H-indol-3-yl)butan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94483A2BC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-4-(1H-indol-3-yl)butan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94484A2BC.H.O.? HUMAN3H-NECA3-{[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94485A2AC.H.O.? HUMAN3H-NECA3-{[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94486A2AC.H.O.? HUMAN3H-NECA3-{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]ethyl}-2-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94487A2BC.H.O.? HUMAN3H-NECA3-{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]ethyl}-2-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94488A2BC.H.O.? HUMAN3H-NECA3-{3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]propyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94489A2AC.H.O.? HUMAN3H-NECA3-{3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]propyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94490A2AC.H.O.? HUMAN3H-NECA3-{4-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]butyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94491A2BC.H.O.? HUMAN3H-NECA3-{4-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]butyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94492A2BC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-4-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94493A2AC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-4-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94494A2AC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94495A2BC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94496A2BC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl) ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94497A2AC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl) ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94498A2AC.H.O.? HUMAN3H-NECA5-Chloro-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94499A2BC.H.O.? HUMAN3H-NECA5-Chloro-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94500A2BC.H.O.? HUMAN3H-NECA2-(5-Bromo-7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94501A2AC.H.O.? HUMAN3H-NECA2-(5-Bromo-7-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94502A2AC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(1H-indol-3-yl)ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94503A2BC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(1H-indol-3-yl)ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94504A2BC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(6-fluoro-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94505A2AC.H.O.? HUMAN3H-NECA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(6-fluoro-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94506A2AC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-7-methoxy-1H-indole3630Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94507A2BC.H.O.? HUMAN3H-NECA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-7-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94508A2BC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94509A2AC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94510A2AC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-fluoro-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94511A2BC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-fluoro-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94512A2BC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94513A2AC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94514A2AC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94515A2BC.H.O.? HUMAN3H-NECA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94516A2BC.H.O.? HUMAN3H-NECA{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indol-7-yl}azinic acid>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94517A2AC.H.O.? HUMAN3H-NECA{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indol-7-yl}azinic acid>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94518A1C.H.O.? HUMAN3H-CCPA{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indol-7-yl}azinic acid4820Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94519A1C.H.O.? HUMAN3H-CCPA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94520A1C.H.O.? HUMAN3H-CCPA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94521A1C.H.O.? HUMAN3H-CCPA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-fluoro-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94522A1C.H.O.? HUMAN3H-CCPA2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94523A1C.H.O.? HUMAN3H-CCPA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-7-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94524A1C.H.O.? HUMAN3H-CCPA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(6-fluoro-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94525A1C.H.O.? HUMAN3H-CCPA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(1H-indol-3-yl)ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94526A1C.H.O.? HUMAN3H-CCPA5-Chloro-3-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94527A1C.H.O.? HUMAN3H-CCPA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl) ethan-1-one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94528A1C.H.O.? HUMAN3H-CCPA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94529A1C.H.O.? HUMAN3H-CCPA3-[4-(4,6-Dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-4-methoxy-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94530A1C.H.O.? HUMAN3H-CCPA3-{[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]methyl}-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94531A1C.H.O.? HUMAN3H-CCPA3-{2-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]ethyl}-2-methyl-1H-indole>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94532A1C.H.O.? HUMAN3H-CCPA1-[4-(4,6-Dimethylpyrimidin-2-yl)piperazin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1- one>10000Shao YM et al 2018Jan 15, 2025Jan 15, 2025
94533A1C.H.O.? HUMAN3H-CCPA5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine0.59Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94534A1C.H.O.? HUMAN3H-CCPA2-chloro-5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine1.56Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94535A1C.H.O.? HUMAN3H-CCPA5′-Chloro-5′- deoxy-N6 -(±)-endo-norbornyl-adenosine (5′Cl5′d-(±)-ENBA0.51Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94536A1C.H.O.? HUMAN3H-CCPA2-chloro-5′-chloro-5′-deoxyN6 -(±)-endo-norbornyl-adenosine1.61Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94537A1C.H.O.? HUMAN3H-CCPAN6-(R)-3-Tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine1.89Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94538A1C.H.O.? HUMAN3H-CCPA2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-Dribofuranosyl)adenine3.5Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94539A1C.H.O.? HUMAN3H-CCPAN6 -(4-Chloro-2-fluorophenyl)amino-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine1.87Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94540A1C.H.O.? HUMAN3H-CCPA2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-chloro-5- deoxy-β-D-ribofuranosyl)adenine11.2Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94541A1C.H.O.? HUMAN3H-CCPAN6 -Cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β- D-ribofuranosyl)adenine115Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94542A1C.H.O.? HUMAN3H-CCPA2-Chloro-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine18.6Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94543A1C.H.O.? HUMAN3H-CCPAN6 -(±)-endo-Norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine25.6Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94544A1C.H.O.? HUMAN3H-CCPA2-Chloro-N6 -(±)-endo-norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine4.35Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94545A1C.H.O.? HUMAN3H-CCPAN6 -(R)-3-Tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1- yl)-5-deoxy-β-D-ribofuranosyl)adenine491Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94546A1C.H.O.? HUMAN3H-CCPA2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine438Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94547A1C.H.O.? HUMAN3H-CCPAN6 -(4-Chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine158Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94548A1C.H.O.? HUMAN3H-CCPA2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine139Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94549A1C.H.O.? HUMAN3H-CCPA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine8.02Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94550A1C.H.O.? HUMAN3H-CCPA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(±)-endo-norbornyl-9H-(5- (3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine59.4Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94551A1C.H.O.? HUMAN3H-CCPA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(R)-3-tetrahydrofuranyl-9H- (5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)- adenine24.6Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94552A1C.H.O.? HUMAN3H-CCPA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(4-chloro-2-fluorophenyl)- amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-Dribofuranosyl)adenine91.4Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94553A2AC.H.O.? HUMAN3H-NECA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(4-chloro-2-fluorophenyl)- amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-Dribofuranosyl)adenine4320Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94554A2AC.H.O.? HUMAN3H-NECA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(R)-3-tetrahydrofuranyl-9H- (5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)- adenine5090Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94555A2AC.H.O.? HUMAN3H-NECA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(±)-endo-norbornyl-9H-(5- (3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94556A2AC.H.O.? HUMAN3H-NECA2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine5870Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94557A2AC.H.O.? HUMAN3H-NECA2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94558A2AC.H.O.? HUMAN3H-NECAN6 -(4-Chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine6830Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94559A2AC.H.O.? HUMAN3H-NECA2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94560A2AC.H.O.? HUMAN3H-NECAN6 -(R)-3-Tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1- yl)-5-deoxy-β-D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94561A2AC.H.O.? HUMAN3H-NECA2-Chloro-N6 -(±)-endo-norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine9430Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94562A2AC.H.O.? HUMAN3H-NECAN6 -(±)-endo-Norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94563A2AC.H.O.? HUMAN3H-NECA2-Chloro-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94564A2AC.H.O.? HUMAN3H-NECAN6 -Cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β- D-ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94565A2AC.H.O.? HUMAN3H-NECA2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-chloro-5- deoxy-β-D-ribofuranosyl)adenine1960Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94566A2AC.H.O.? HUMAN3H-NECAN6 -(4-Chloro-2-fluorophenyl)amino-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine1360Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94567A2AC.H.O.? HUMAN3H-NECA2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-Dribofuranosyl)adenine8680Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94568A2AC.H.O.? HUMAN3H-NECAN6-(R)-3-Tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine>10000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94569A2AC.H.O.? HUMAN3H-NECA2-chloro-5′-chloro-5′-deoxyN6 -(±)-endo-norbornyl-adenosine2050Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94570A2AC.H.O.? HUMAN3H-NECA5′-Chloro-5′- deoxy-N6 -(±)-endo-norbornyl-adenosine1340Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94571A2AC.H.O.? HUMAN3H-NECA2-chloro-5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine2160Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94572A2AC.H.O.? HUMAN3H-NECA5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine837Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94573A3C.H.O.? HUMAN3H-HEMADO5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine376Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94574A3C.H.O.? HUMAN3H-HEMADO2-chloro-5′-chloro-5′-deoxy-N6 -cyclopentyl-adenosine417Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94575A3C.H.O.? HUMAN3H-HEMADO5′-Chloro-5′- deoxy-N6 -(±)-endo-norbornyl-adenosine1290Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94576A3C.H.O.? HUMAN3H-HEMADO2-chloro-5′-chloro-5′-deoxyN6 -(±)-endo-norbornyl-adenosine1410Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94577A3C.H.O.? HUMAN3H-HEMADON6-(R)-3-Tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine1200Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94578A3C.H.O.? HUMAN3H-HEMADO2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-chloro-5-deoxy-β-Dribofuranosyl)adenine1100Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94579A3C.H.O.? HUMAN3H-HEMADON6 -(4-Chloro-2-fluorophenyl)amino-9H-(5-chloro-5-deoxy-β-D- ribofuranosyl)adenine136Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94580A3C.H.O.? HUMAN3H-HEMADO2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-chloro-5- deoxy-β-D-ribofuranosyl)adenine232Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94581A3C.H.O.? HUMAN3H-HEMADON6 -Cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β- D-ribofuranosyl)adenine5640Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94582A3C.H.O.? HUMAN3H-HEMADO2-Chloro-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine343Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94583A3C.H.O.? HUMAN3H-HEMADON6 -(±)-endo-Norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5- deoxy-β-D-ribofuranosyl)adenine5450Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94584A3C.H.O.? HUMAN3H-HEMADO2-Chloro-N6 -(±)-endo-norbornyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine1451Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94585A3C.H.O.? HUMAN3H-HEMADON6 -(R)-3-Tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1- yl)-5-deoxy-β-D-ribofuranosyl)adenine5280Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94586A3C.H.O.? HUMAN3H-HEMADO2-Chloro-N6 -(R)-3-tetrahydrofuranyl-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine996Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94587A3C.H.O.? HUMAN3H-HEMADON6 -(4-Chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1Hpyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine2730Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94588A3C.H.O.? HUMAN3H-HEMADO2-Chloro-N6 -(4-chloro-2-fluorophenyl)amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine139Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94589A3C.H.O.? HUMAN3H-HEMADO2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -cyclopentyl-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine562Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94590A3C.H.O.? HUMAN3H-HEMADO2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(±)-endo-norbornyl-9H-(5- (3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)adenine667Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94591A3C.H.O.? HUMAN3H-HEMADO2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(R)-3-tetrahydrofuranyl-9H- (5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-D-ribofuranosyl)- adenine1000Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94592A3C.H.O.? HUMAN3H-HEMADO2-(3,5-Dimethyl-1H-pyrazol-1-yl)-N6 -(4-chloro-2-fluorophenyl)- amino)-9H-(5-(3,5-dimethyl-1H-pyrazol-1-yl)-5-deoxy-β-Dribofuranosyl)adenine636Petrelli R et al 2018Jan 15, 2025Jan 15, 2025
94593CB1BRAINMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide440Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94594CB1BRAINMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-(homopiperidinyl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide442Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94595CB1BRAINMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide1386Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94596CB1BRAINMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide447Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94597CB1BRAINMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide6.5Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94598CB1BRAINMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide3918Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94599CB1BRAINMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-(homopiperidinyl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide3798Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94600CB1BRAINMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide4731Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94601CB1BRAINMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide3076Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94602CB1BRAINMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-morpholinyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide4705Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94603CB1BRAINMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide3255Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94604CB1BRAINMOUSE3H-CP559407-methyl-1-(2,4-dichlorophenyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide2245Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94605CB1BRAINMOUSE3H-CP559406-Methyl-1-(4-methylbenzyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide180Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94606CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide377Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94607CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-(homopiperidin-yl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide1276Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94608CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide4500Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94609CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide1977Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94610CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-morpholinyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide4500Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94611CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide160Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94612CB1BRAINMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide420Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94613CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide2.4Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94614CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide2.7Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94615CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-morpholinyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide1758Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94616CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide191Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94617CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide515Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94618CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-(homopiperidin-yl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide69Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94619CB2SPLEENMOUSE3H-CP559407-Methyl-1-(4-methylbenzyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide125Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94620CB2SPLEENMOUSE3H-CP559406-Methyl-1-(4-methylbenzyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide4.8Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94621CB2SPLEENMOUSE3H-CP559407-methyl-1-(2,4-dichlorophenyl)-N-fenchyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide5.3Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94622CB2SPLEENMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide6.7Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94623CB2SPLEENMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-morpholinyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide747Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94624CB2SPLEENMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide501Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94625CB2SPLEENMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide817Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94626CB2SPLEENMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-(homopiperidinyl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide321Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94627CB2SPLEENMOUSE3H-CP559407-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide578Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94628CB2SPLEENMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-menthyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide5.1Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94629CB2SPLEENMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-cyclohexyl-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide7.2Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94630CB2SPLEENMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-(pyrrolidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide38.3Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94631CB2SPLEENMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-(homopiperidinyl)- 1,4-dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide1.1Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94632CB2SPLEENMOUSE3H-CP559406-Methyl-1-(2,4-dichlorophenyl)-N-(piperidinyl)-1,4- dihydrothieno[20 ,30 -4,5]cyclopenta[1,2c]pyrazole-3-carboxamide2.3Pinna G et al 2014Jan 15, 2025Jan 28, 2025
94633CB2?CLONED? HUMAN3H-CP-55940N-(1)-(S)-Fenchyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5.7Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94634CB1?CLONED? HUMAN3H-CP-55940N-(1)-(S)-Fenchyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide1470Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94635CB2?CLONED? HUMAN3H-CP-559401-(5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-yl)methyl)-fenchylamine343Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94636CB2?CLONED? HUMAN3H-CP-55940N-(R)-(þ)-Bornyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide164Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94637CB1?CLONED? HUMAN3H-CP-55940N-(R)-(þ)-Bornyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide368Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94638CB2?CLONED? HUMAN3H-CP-55940N-(1R,2R,3R,5S)-Isopinocampheyl-5-(4-chloro-3- methylphenyl)-1-(4-methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94639CB1?CLONED? HUMAN3H-CP-55940N-(1S,2R)-Myrtanyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94640CB2?CLONED? HUMAN3H-CP-55940N-(1S,2R)-Myrtanyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide72.2Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94641CB2?CLONED? HUMAN3H-CP-55940N-(Adamantan-1-yl)-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94642CB1?CLONED? HUMAN3H-CP-55940N-(Adamantan-1-yl)-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94643CB1?CLONED? HUMAN3H-CP-55940N-Adamantylmethane-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94644CB2?CLONED? HUMAN3H-CP-55940N-Adamantylmethane-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94645CB1?CLONED? HUMAN3H-CP-55940N-Menthyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94646CB2?CLONED? HUMAN3H-CP-55940N-Menthyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide1100Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94647CB2?CLONED? HUMAN3H-CP-55940N-(R)-()-Cyclohexylethyl-5-(4-chloro-3-methylphenyl)-1- (4-methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94648CB1?CLONED? HUMAN3H-CP-55940N-(R)-()-Cyclohexylethyl-5-(4-chloro-3-methylphenyl)-1- (4-methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94649CB2?CLONED? HUMAN3H-CP-55940N-(S)-(þ)-Cyclohexylethyl-5-(4-chloro-3-methylphenyl)-1- (4-methylbenzyl)-1H-pyrrole-3-carboxamide492Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94650CB2?CLONED? HUMAN3H-CP-55940N-Cyclohexyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide244Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94651CB1?CLONED? HUMAN3H-CP-55940N-Cyclohexyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94652CB1?CLONED? HUMAN3H-CP-55940N-Piperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide3070Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94653CB2?CLONED? HUMAN3H-CP-55940N-Piperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide106Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94654CB2?CLONED? HUMAN3H-CP-55940N-(4-(2-Chlorophenyl)piperazin-1-yl)-(5-(4-chloro-3- methylphenyl)-1-(4-methylbenzyl)-1H-pyrrole-3-carboxamide1707Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94655CB1?CLONED? HUMAN3H-CP-55940N-(4-(2-Chlorophenyl)piperazin-1-yl)-(5-(4-chloro-3- methylphenyl)-1-(4-methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94656CB1?CLONED? HUMAN3H-CP-55940N-Pyrrolidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94657CB2?CLONED? HUMAN3H-CP-55940N-Pyrrolidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94658CB2?CLONED? HUMAN3H-CP-55940N-Piperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94659CB1?CLONED? HUMAN3H-CP-55940N-Piperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94660CB1?CLONED? HUMAN3H-CP-55940N-Homopiperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94661CB2?CLONED? HUMAN3H-CP-55940N-Homopiperidinyl-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carbohydrazide575Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94662CB2?CLONED? HUMAN3H-CP-55940N-(Naphthalen-1-yl)-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94663CB1?CLONED? HUMAN3H-CP-55940N-(Naphthalen-1-yl)-5-(4-chloro-3-methylphenyl)-1-(4- methylbenzyl)-1H-pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94664CB1?CLONED? HUMAN3H-CP-559401-{[5-(4-Chloro-3-methylphenyl)-1-(4-methylbenzyl)-1Hpyrrol-3-yl]methyl}-4-(4-chlorophenyl)piperazine5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94665CB2?CLONED? HUMAN3H-CP-559401-{[5-(4-Chloro-3-methylphenyl)-1-(4-methylbenzyl)-1Hpyrrol-3-yl]methyl}-4-(4-chlorophenyl)piperazine5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94666CB2?CLONED? HUMAN3H-CP-559401-{[5-(4-Chloro-3-methylphenyl)-1-(4-methylbenzyl)-1Hpyrrol-3-yl]methyl}-4-(3,4-dichlorophenyl)piperazine5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94667CB1?CLONED? HUMAN3H-CP-559401-{[5-(4-Chloro-3-methylphenyl)-1-(4-methylbenzyl)-1Hpyrrol-3-yl]methyl}-4-(3,4-dichlorophenyl)piperazine5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94668CB1?CLONED? HUMAN3H-CP-55940N-(1)-(S)-fenchyl-6-chloro-2,5-dimethyl-1-(4- methylbenzyl)-1,4-dihydroindeno[1,2-b]pyrrole-3-carboxamide5000Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
94669CB2?CLONED? HUMAN3H-CP-55940N-(1)-(S)-fenchyl-6-chloro-2,5-dimethyl-1-(4- methylbenzyl)-1,4-dihydroindeno[1,2-b]pyrrole-3-carboxamide346Ragusa G et al 2015Jan 15, 2025Jan 28, 2025
946705-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946715-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946725-HT1ACLONEDHUMAN3H-WAY1006354′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946735-HT1ACLONEDHUMAN3H-WAY1006355-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946745-HT1ACLONEDHUMAN3H-WAY1006354′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946755-HT1ACLONEDHUMAN3H-WAY1006354′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946765-HT1ACLONEDHUMAN3H-WAY1006354′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946775-HT1ACLONEDHUMAN3H-WAY1006354′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946785-HT1ACLONEDHUMAN3H-WAY1006354′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946795-HT1ACLONEDHUMAN3H-WAY1006354′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946805-HT1ACLONEDHUMAN3H-WAY1006354-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946815-HT1ACLONEDHUMAN3H-WAY1006352-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946825-HT1ACLONEDHUMAN3H-WAY1006352-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946835-HT1BCLONEDHUMAN3H-GR1257434-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946845-HT1BCLONEDHUMAN3H-GR1257434-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946855-HT1BCLONEDHUMAN3H-GR1257434′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946865-HT1BCLONEDHUMAN3H-GR1257435-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946875-HT1BCLONEDHUMAN3H-GR1257434′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946885-HT1BCLONEDHUMAN3H-GR1257434′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946895-HT1BCLONEDHUMAN3H-GR1257434′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946905-HT1BCLONEDHUMAN3H-GR1257434′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946915-HT1BCLONEDHUMAN3H-GR1257434′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946925-HT1BCLONEDHUMAN3H-GR1257434-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946935-HT1BCLONEDHUMAN3H-GR1257432-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946945-HT1DCLONEDHUMAN3H-GR1257434-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946955-HT1DCLONEDHUMAN3H-GR1257434-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946965-HT1DCLONEDHUMAN3H-GR1257434′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946975-HT1DCLONEDHUMAN3H-GR1257435-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946985-HT1DCLONEDHUMAN3H-GR1257434′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
946995-HT1DCLONEDHUMAN3H-GR1257434′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947005-HT1DCLONEDHUMAN3H-GR1257434′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947015-HT1DCLONEDHUMAN3H-GR1257434′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947025-HT1DCLONEDHUMAN3H-GR1257434′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947035-HT1DCLONEDHUMAN3H-GR1257434′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947045-HT1DCLONEDHUMAN3H-GR1257434-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947055-HT1DCLONEDHUMAN3H-GR1257432-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate2390Jung et al 2021Jan 15, 2025Jan 15, 2025
947065-HT1DCLONEDHUMAN3H-GR1257432-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947075-HT1BCLONEDHUMAN3H-GR1257432-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate5570Jung et al 2021Jan 15, 2025Jan 15, 2025
947085-HT1ECLONEDHUMAN3H-5-HT4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947095-HT1ECLONEDHUMAN3H-5-HT4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947105-HT1ECLONEDHUMAN3H-5-HT4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947115-HT1ECLONEDHUMAN3H-5-HT5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947125-HT1ECLONEDHUMAN3H-5-HT4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947135-HT1ECLONEDHUMAN3H-5-HT4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947145-HT1ECLONEDHUMAN3H-5-HT4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947155-HT1ECLONEDHUMAN3H-5-HT4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947165-HT1ECLONEDHUMAN3H-5-HT4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947175-HT1ECLONEDHUMAN3H-5-HT4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947185-HT1ECLONEDHUMAN3H-5-HT4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947195-HT1ECLONEDHUMAN3H-5-HT2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947205-HT1ECLONEDHUMAN3H-5-HT2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947215-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947225-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947235-HT2ACLONEDHUMAN3H-KETANSERIN4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947245-HT2ACLONEDHUMAN3H-KETANSERIN5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947255-HT2ACLONEDHUMAN3H-KETANSERIN4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947265-HT2ACLONEDHUMAN3H-KETANSERIN4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947275-HT2ACLONEDHUMAN3H-KETANSERIN4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947285-HT2ACLONEDHUMAN3H-KETANSERIN4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947295-HT2ACLONEDHUMAN3H-KETANSERIN4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947305-HT2ACLONEDHUMAN3H-KETANSERIN4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947315-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947325-HT2ACLONEDHUMAN3H-KETANSERIN2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947335-HT2ACLONEDHUMAN3H-KETANSERIN2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947345-HT2BCLONEDHUMAN3H-LSD4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947355-HT2BCLONEDHUMAN3H-LSD4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947365-HT2BCLONEDHUMAN3H-LSD4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947375-HT2BCLONEDHUMAN3H-LSD5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947385-HT2BCLONEDHUMAN3H-LSD4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947395-HT2BCLONEDHUMAN3H-LSD4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947405-HT2BCLONEDHUMAN3H-LSD4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947415-HT2BCLONEDHUMAN3H-LSD4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947425-HT2BCLONEDHUMAN3H-LSD4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947435-HT2BCLONEDHUMAN3H-LSD4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947445-HT2BCLONEDHUMAN3H-LSD4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947455-HT2BCLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947465-HT2BCLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947475-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947485-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025