The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 92,001-93,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
947495-HT2CCLONEDHUMAN3H-MESULERGINE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947505-HT2CCLONEDHUMAN3H-MESULERGINE5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947515-HT2CCLONEDHUMAN3H-MESULERGINE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947525-HT2CCLONEDHUMAN3H-MESULERGINE4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947535-HT2CCLONEDHUMAN3H-MESULERGINE4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947545-HT2CCLONEDHUMAN3H-MESULERGINE4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947555-HT2CCLONEDHUMAN3H-MESULERGINE4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947565-HT2CCLONEDHUMAN3H-MESULERGINE4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947575-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947585-HT2CCLONEDHUMAN3H-MESULERGINE2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947595-HT2CCLONEDHUMAN3H-MESULERGINE2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947605-HT3CLONEDHUMAN3H-GR-656304-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947615-HT3CLONEDHUMAN3H-GR-656304-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947625-HT3CLONEDHUMAN3H-GR-656304′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947635-HT3CLONEDHUMAN3H-GR-656305-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947645-HT3CLONEDHUMAN3H-GR-656304′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947655-HT3CLONEDHUMAN3H-GR-656304′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947665-HT3CLONEDHUMAN3H-GR-656304′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947675-HT3CLONEDHUMAN3H-GR-656304′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947685-HT3CLONEDHUMAN3H-GR-656304′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947695-HT3CLONEDHUMAN3H-GR-656304′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947705-HT3CLONEDHUMAN3H-GR-656304-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947715-HT3CLONEDHUMAN3H-GR-656302-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947725-HT3CLONEDHUMAN3H-GR-656302-(Dimethylamino)-2-oxoethyl 4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947735-HT5ACLONEDHUMAN3H-LSD4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947745-HT5ACLONEDHUMAN3H-LSD4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947755-HT5ACLONEDHUMAN3H-LSD4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947765-HT5ACLONEDHUMAN3H-LSD5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947775-HT5ACLONEDHUMAN3H-LSD4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947785-HT5ACLONEDHUMAN3H-LSD4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947795-HT5ACLONEDHUMAN3H-LSD4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947805-HT5ACLONEDHUMAN3H-LSD4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947815-HT5ACLONEDHUMAN3H-LSD4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947825-HT5ACLONEDHUMAN3H-LSD4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947835-HT5ACLONEDHUMAN3H-LSD4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947845-HT5ACLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate2040Jung et al 2021Jan 15, 2025Jan 15, 2025
947855-HT5ACLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947865-HT6CLONEDHUMAN3H-LSD4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947875-HT6CLONEDHUMAN3H-LSD4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947885-HT6CLONEDHUMAN3H-LSD4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947895-HT6CLONEDHUMAN3H-LSD5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947905-HT6CLONEDHUMAN3H-LSD4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947915-HT6CLONEDHUMAN3H-LSD4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947925-HT6CLONEDHUMAN3H-LSD4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947935-HT6CLONEDHUMAN3H-LSD4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947945-HT6CLONEDHUMAN3H-LSD4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947955-HT6CLONEDHUMAN3H-LSD4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947965-HT6CLONEDHUMAN3H-LSD4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947975-HT6CLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947985-HT6CLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
947995-HT7CLONEDHUMAN3H-LSD4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948005-HT7CLONEDHUMAN3H-LSD4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948015-HT7CLONEDHUMAN3H-LSD4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948025-HT7CLONEDHUMAN3H-LSD5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948035-HT7CLONEDHUMAN3H-LSD4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948045-HT7CLONEDHUMAN3H-LSD4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948055-HT7CLONEDHUMAN3H-LSD4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948065-HT7CLONEDHUMAN3H-LSD4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948075-HT7CLONEDHUMAN3H-LSD4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948085-HT7CLONEDHUMAN3H-LSD4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948095-HT7CLONEDHUMAN3H-LSD4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
948105-HT7CLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate2220Jung et al 2021Jan 15, 2025Jan 15, 2025
948115-HT7CLONEDHUMAN3H-LSD2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94812Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate1230Jung et al 2021Jan 15, 2025Jan 28, 2025
94813Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94814Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94815Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94816Alpha1ACLONEDHUMAN3H-PRAZOSIN5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94817Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94818Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94819Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94820Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94821Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94822Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94823Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94824Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94825Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid2650Jung et al 2021Jan 15, 2025Jan 28, 2025
94826Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94827Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94828Alpha1BCLONEDHUMAN3H-PRAZOSIN5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94829Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94830Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94831Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94832Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94833Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94834Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94835Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94836Alpha1BCLONEDHUMAN3H-PRAZOSIN2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate2520Jung et al 2021Jan 15, 2025Jan 28, 2025
94837Alpha1BCLONEDHUMAN3H-PRAZOSIN2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94838Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94839Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94840Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94841Alpha1DCLONEDHUMAN3H-PRAZOSIN5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94842Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94843Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94844Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94845Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94846Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94847Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94848Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94849Alpha1DCLONEDHUMAN3H-PRAZOSIN2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94850Alpha1DCLONEDHUMAN3H-PRAZOSIN2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94851Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid3970Jung et al 2021Jan 15, 2025Jan 28, 2025
94852Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94853Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94854Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94855Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94856Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94857Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94858Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94859Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94860Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94861Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94862Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94863Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94864Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94865Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94866Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94867Alpha2BCLONEDHUMAN3H-RAUWOLSCINE5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94868Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94869Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94870Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94871Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94872Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94873Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94874Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94875Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate1810Jung et al 2021Jan 15, 2025Jan 28, 2025
94876Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94877Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid3930Jung et al 2021Jan 15, 2025Jan 28, 2025
94878Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94879Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94880Alpha2CCLONEDHUMAN3H-RAUWOLSCINE5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94881Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94882Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94883Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94884Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94885Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94886Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94887Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94888Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate790Jung et al 2021Jan 15, 2025Jan 28, 2025
94889Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94890Beta 1CLONEDHUMAN125I-Pindolol4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94891Beta 1CLONEDHUMAN125I-Pindolol4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94892Beta 1CLONEDHUMAN125I-Pindolol4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94893Beta 1CLONEDHUMAN125I-Pindolol5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94894Beta 1CLONEDHUMAN125I-Pindolol4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94895Beta 1CLONEDHUMAN125I-Pindolol4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94896Beta 1CLONEDHUMAN125I-Pindolol4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94897Beta 1CLONEDHUMAN125I-Pindolol4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94898Beta 1CLONEDHUMAN125I-Pindolol4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94899Beta 1CLONEDHUMAN125I-Pindolol4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94900Beta 1CLONEDHUMAN125I-Pindolol4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94901Beta 1CLONEDHUMAN125I-Pindolol2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94902Beta 1CLONEDHUMAN125I-Pindolol2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94903Beta3CLONEDHUMAN125I-Pindolol4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94904Beta3CLONEDHUMAN125I-Pindolol4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94905Beta3CLONEDHUMAN125I-Pindolol4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94906Beta3CLONEDHUMAN125I-Pindolol5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94907Beta3CLONEDHUMAN125I-Pindolol4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94908Beta3CLONEDHUMAN125I-Pindolol4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94909Beta3CLONEDHUMAN125I-Pindolol4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94910Beta3CLONEDHUMAN125I-Pindolol4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94911Beta3CLONEDHUMAN125I-Pindolol4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94912Beta3CLONEDHUMAN125I-Pindolol4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94913Beta3CLONEDHUMAN125I-Pindolol4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94914Beta3CLONEDHUMAN125I-Pindolol2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate1240Jung et al 2021Jan 15, 2025Jan 28, 2025
94915Beta3CLONEDHUMAN125I-Pindolol2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94916Beta3CLONEDHUMAN3H-CGP-121774-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94917Beta 2CLONEDHUMAN3H-CGP-121774-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94918Beta 2CLONEDHUMAN3H-CGP-121774-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94919Beta 2CLONEDHUMAN3H-CGP-121774′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94920Beta 2CLONEDHUMAN3H-CGP-121775-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94921Beta 2CLONEDHUMAN3H-CGP-121774′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94922Beta 2CLONEDHUMAN3H-CGP-121774′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94923Beta 2CLONEDHUMAN3H-CGP-121774′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94924Beta 2CLONEDHUMAN3H-CGP-121774′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94925Beta 2CLONEDHUMAN3H-CGP-121774′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94926Beta 2CLONEDHUMAN3H-CGP-121774′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94927Beta 2CLONEDHUMAN3H-CGP-121774-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94928Beta 2CLONEDHUMAN3H-CGP-121772-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate4180Jung et al 2021Jan 15, 2025Jan 15, 2025
94929Beta 2CLONEDHUMAN3H-CGP-121772-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
94930BZPCORTICAL MEMBRANESRATFNZ4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94931BZPCORTICAL MEMBRANESRATFNZ4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94932BZPCORTICAL MEMBRANESRATFNZ4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94933BZPCORTICAL MEMBRANESRATFNZ5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94934BZPCORTICAL MEMBRANESRATFNZ4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94935BZPCORTICAL MEMBRANESRATFNZ4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94936BZPCORTICAL MEMBRANESRATFNZ4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94937BZPCORTICAL MEMBRANESRATFNZ4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94938BZPCORTICAL MEMBRANESRATFNZ4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94939BZPCORTICAL MEMBRANESRATFNZ4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94940BZPCORTICAL MEMBRANESRATFNZ2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94941BZPCORTICAL MEMBRANESRATFNZ2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94942D1CLONEDHUMAN3H-SCH233904-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid520Jung et al 2021Jan 15, 2025Jan 28, 2025
94943D1CLONEDHUMAN3H-SCH233904-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94944D1CLONEDHUMAN3H-SCH233904′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94945D1CLONEDHUMAN3H-SCH233905-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94946D1CLONEDHUMAN3H-SCH233904′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94947D1CLONEDHUMAN3H-SCH233904′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94948D1CLONEDHUMAN3H-SCH233904′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94949D1CLONEDHUMAN3H-SCH233904′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94950D1CLONEDHUMAN3H-SCH233904′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94951D1CLONEDHUMAN3H-SCH233904′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94952D1CLONEDHUMAN3H-SCH233904-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94953D1CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94954D1CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94955D5CLONEDHUMAN3H-SCH233904-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid1440Jung et al 2021Jan 15, 2025Jan 28, 2025
94956D5CLONEDHUMAN3H-SCH233904-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94957D5CLONEDHUMAN3H-SCH233904′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94958D5CLONEDHUMAN3H-SCH233905-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94959D5CLONEDHUMAN3H-SCH233904′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94960D5CLONEDHUMAN3H-SCH233904′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94961D5CLONEDHUMAN3H-SCH233904′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94962D5CLONEDHUMAN3H-SCH233904′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94963D5CLONEDHUMAN3H-SCH233904′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94964D5CLONEDHUMAN3H-SCH233904′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94965D5CLONEDHUMAN3H-SCH233904-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94966D5CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate3010Jung et al 2021Jan 15, 2025Jan 28, 2025
94967D5CLONEDHUMAN3H-SCH233902-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94968D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94969D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94970D2CLONEDHUMAN3H-N-Methylspiperone4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94971D2CLONEDHUMAN3H-N-Methylspiperone5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94972D2CLONEDHUMAN3H-N-Methylspiperone4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94973D2CLONEDHUMAN3H-N-Methylspiperone4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94974D2CLONEDHUMAN3H-N-Methylspiperone4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94975D2CLONEDHUMAN3H-N-Methylspiperone4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94976D2CLONEDHUMAN3H-N-Methylspiperone4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94977D2CLONEDHUMAN3H-N-Methylspiperone4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94978D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94979D2CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94980D2CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94981D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94982D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94983D3CLONEDHUMAN3H-N-Methylspiperone4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94984D3CLONEDHUMAN3H-N-Methylspiperone5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94985D3CLONEDHUMAN3H-N-Methylspiperone4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94986D3CLONEDHUMAN3H-N-Methylspiperone4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94987D3CLONEDHUMAN3H-N-Methylspiperone4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94988D3CLONEDHUMAN3H-N-Methylspiperone4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94989D3CLONEDHUMAN3H-N-Methylspiperone4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94990D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94991D3CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate840Jung et al 2021Jan 15, 2025Jan 28, 2025
94992D3CLONEDHUMAN3H-N-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94993D4CLONEDHUMAN3H-Methylspiperone4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94994D4CLONEDHUMAN3H-Methylspiperone4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94995D4CLONEDHUMAN3H-Methylspiperone4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94996D4CLONEDHUMAN3H-Methylspiperone5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94997D4CLONEDHUMAN3H-Methylspiperone4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94998D4CLONEDHUMAN3H-Methylspiperone4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
94999D4CLONEDHUMAN3H-Methylspiperone4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95000D4CLONEDHUMAN3H-Methylspiperone4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95001D4CLONEDHUMAN3H-Methylspiperone4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95002D4CLONEDHUMAN3H-Methylspiperone4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95003D4CLONEDHUMAN3H-Methylspiperone4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95004D4CLONEDHUMAN3H-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95005D4CLONEDHUMAN3H-Methylspiperone2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95006KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95007KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95008KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95009KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95010KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95011KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95012KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95013KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95014KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95015KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95016KORCEREBRAL CORTEXRAT3H-MUSCIMOL2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95017KORCEREBRAL CORTEXRAT3H-MUSCIMOL2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95018H1CLONEDHUMAN3H-PYRILAMINE4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95019H1CLONEDHUMAN3H-PYRILAMINE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95020H1CLONEDHUMAN3H-PYRILAMINE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95021H1CLONEDHUMAN3H-PYRILAMINE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95022H1CLONEDHUMAN3H-PYRILAMINE4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95023H1CLONEDHUMAN3H-PYRILAMINE4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95024H1CLONEDHUMAN3H-PYRILAMINE4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95025H1CLONEDHUMAN3H-PYRILAMINE4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95026H1CLONEDHUMAN3H-PYRILAMINE4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95027H1CLONEDHUMAN3H-PYRILAMINE2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95028H1CLONEDHUMAN3H-PYRILAMINE2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95029H1CLONEDHUMAN3H-PYRILAMINE4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2650Jung et al 2021Jan 15, 2025Jan 28, 2025
950305-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950315-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950325-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950335-HT1DCLONEDHUMAN125I-iodoaminopotentidine5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950345-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950355-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950365-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950375-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950385-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950395-HT1DCLONEDHUMAN125I-iodoaminopotentidine4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950405-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950415-HT1DCLONEDHUMAN125I-iodoaminopotentidine2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
950425-HT1DCLONEDHUMAN125I-iodoaminopotentidine2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95043H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95044H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95045H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95046H3CLONEDHUMAN3H-Alpha-methylhistamine5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95047H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95048H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95049H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95050H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95051H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95052H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95053H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95054H3CLONEDHUMAN3H-Alpha-methylhistamine2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95055H3CLONEDHUMAN3H-Alpha-methylhistamine2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95056H4CLONEDHUMAN3H-Histamine4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid1700Jung et al 2021Jan 15, 2025Jan 28, 2025
95057H4CLONEDHUMAN3H-Histamine4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95058H4CLONEDHUMAN3H-Histamine4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95059H4CLONEDHUMAN3H-Histamine5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95060H4CLONEDHUMAN3H-Histamine4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95061H4CLONEDHUMAN3H-Histamine4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95062H4CLONEDHUMAN3H-Histamine4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95063H4CLONEDHUMAN3H-Histamine4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95064H4CLONEDHUMAN3H-Histamine4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95065H4CLONEDHUMAN3H-Histamine4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95066H4CLONEDHUMAN3H-Histamine4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95067H4CLONEDHUMAN3H-Histamine2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95068H4CLONEDHUMAN3H-Histamine2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95069M1CLONEDHUMAN3H-QNB4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95070M2CLONEDHUMAN3H-QNB4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95071M5CLONEDHUMAN3H-QNB4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95072M5CLONEDHUMAN3H-QNB4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95073M2CLONEDHUMAN3H-QNB4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95074M1CLONEDHUMAN3H-QNB4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95075M1CLONEDHUMAN3H-QNB4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95076M2CLONEDHUMAN3H-QNB4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95077M5CLONEDHUMAN3H-QNB4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95078M5CLONEDHUMAN3H-QNB5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95079M2CLONEDHUMAN3H-QNB5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95080M1CLONEDHUMAN3H-QNB5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95081M1CLONEDHUMAN3H-QNB4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95082M2CLONEDHUMAN3H-QNB4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95083M5CLONEDHUMAN3H-QNB4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95084M5CLONEDHUMAN3H-QNB4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95085M2CLONEDHUMAN3H-QNB4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95086M1CLONEDHUMAN3H-QNB4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95087M1CLONEDHUMAN3H-QNB4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95088M2CLONEDHUMAN3H-QNB4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95089M5CLONEDHUMAN3H-QNB4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95090M5CLONEDHUMAN3H-QNB4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95091M2CLONEDHUMAN3H-QNB4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95092M1CLONEDHUMAN3H-QNB4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95093M1CLONEDHUMAN3H-QNB4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95094M2CLONEDHUMAN3H-QNB4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95095M5CLONEDHUMAN3H-QNB4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95096M5CLONEDHUMAN3H-QNB4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95097M2CLONEDHUMAN3H-QNB4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95098M1CLONEDHUMAN3H-QNB4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95099M1CLONEDHUMAN3H-QNB4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95100M2CLONEDHUMAN3H-QNB4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95101M5CLONEDHUMAN3H-QNB4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95102M5CLONEDHUMAN3H-QNB2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95103M2CLONEDHUMAN3H-QNB2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95104M1CLONEDHUMAN3H-QNB2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95105M1CLONEDHUMAN3H-QNB2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95106M2CLONEDHUMAN3H-QNB2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95107M5CLONEDHUMAN3H-QNB2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95108DORCLONEDHUMAN3H-DADLE4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95109DORCLONEDHUMAN3H-DADLE4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95110DORCLONEDHUMAN3H-DADLE4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2000Jung et al 2021Jan 15, 2025Jan 28, 2025
95111DORCLONEDHUMAN3H-DADLE5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95112DORCLONEDHUMAN3H-DADLE4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95113DORCLONEDHUMAN3H-DADLE4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95114DORCLONEDHUMAN3H-DADLE4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95115DORCLONEDHUMAN3H-DADLE4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid6900Jung et al 2021Jan 15, 2025Jan 28, 2025
95116DORCLONEDHUMAN3H-DADLE4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2150Jung et al 2021Jan 15, 2025Jan 28, 2025
95117DORCLONEDHUMAN3H-DADLE4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid3300Jung et al 2021Jan 15, 2025Jan 28, 2025
95118DORCLONEDHUMAN3H-DADLE4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95119DORCLONEDHUMAN3H-DADLE2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95120DORCLONEDHUMAN3H-DADLE2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95121KORCLONEDHUMAN3H-U695934-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95122KORCLONEDHUMAN3H-U695934-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95123KORCLONEDHUMAN3H-U695934′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95124KORCLONEDHUMAN3H-U695935-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95125KORCLONEDHUMAN3H-U695934′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95126KORCLONEDHUMAN3H-U695934′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95127KORCLONEDHUMAN3H-U695934′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95128KORCLONEDHUMAN3H-U695934′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95129KORCLONEDHUMAN3H-U695934′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95130KORCLONEDHUMAN3H-U695934′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95131KORCLONEDHUMAN3H-U695934-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95132KORCLONEDHUMAN3H-U695932-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95133KORCLONEDHUMAN3H-U69593Methyl 4′-((tert-Butoxycarbonyl)amino)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95134MORCLONEDHUMAN3H-DAMGO4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95135MORCLONEDHUMAN3H-DAMGO4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95136MORCLONEDHUMAN3H-DAMGO4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95137MORCLONEDHUMAN3H-DAMGO5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95138MORCLONEDHUMAN3H-DAMGO4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95139MORCLONEDHUMAN3H-DAMGO4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95140MORCLONEDHUMAN3H-DAMGO4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95141MORCLONEDHUMAN3H-DAMGO4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95142MORCLONEDHUMAN3H-DAMGO4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95143MORCLONEDHUMAN3H-DAMGO4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95144MORCLONEDHUMAN3H-DAMGO4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95145MORCLONEDHUMAN3H-DAMGO2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95146MORCLONEDHUMAN3H-DAMGO2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95147Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid759Jung et al 2021Jan 15, 2025Jan 15, 2025
95148Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95149Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2330Jung et al 2021Jan 15, 2025Jan 15, 2025
95150Sigma 1CLONEDHUMAN3H-Pentazocine(+)5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95151Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95152Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95153Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95154Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95155Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95156Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95157Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid2680Jung et al 2021Jan 15, 2025Jan 15, 2025
95158Sigma 1CLONEDHUMAN3H-Pentazocine(+)2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate1330Jung et al 2021Jan 15, 2025Jan 15, 2025
95159Sigma 1CLONEDHUMAN3H-Pentazocine(+)2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95160Sigma 2CLONEDHUMAN3H-DTG4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95161Sigma 2CLONEDHUMAN3H-DTG4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95162Sigma 2CLONEDHUMAN3H-DTG4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95163Sigma 2CLONEDHUMAN3H-DTG5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95164Sigma 2CLONEDHUMAN3H-DTG4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid931Jung et al 2021Jan 15, 2025Jan 28, 2025
95165Sigma 2CLONEDHUMAN3H-DTG4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95166Sigma 2CLONEDHUMAN3H-DTG4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95167Sigma 2CLONEDHUMAN3H-DTG4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95168Sigma 2CLONEDHUMAN3H-DTG4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95169Sigma 2CLONEDHUMAN3H-DTG4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2260Jung et al 2021Jan 15, 2025Jan 28, 2025
95170Sigma 2CLONEDHUMAN3H-DTG4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid4780Jung et al 2021Jan 15, 2025Jan 28, 2025
95171Sigma 2CLONEDHUMAN3H-DTG4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid230Jung et al 2021Jan 15, 2025Jan 28, 2025
95172Sigma 2CLONEDHUMAN3H-DTG2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate585Jung et al 2021Jan 15, 2025Jan 28, 2025
95173DATCLONEDHUMAN3H-WIN 35,4284-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95174DATCLONEDHUMAN3H-WIN 35,4284-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95175DATCLONEDHUMAN3H-WIN 35,4284′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95176DATCLONEDHUMAN3H-WIN 35,4285-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95177DATCLONEDHUMAN3H-WIN 35,4284′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95178DATCLONEDHUMAN3H-WIN 35,4284′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95179DATCLONEDHUMAN3H-WIN 35,4284′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95180DATCLONEDHUMAN3H-WIN 35,4284′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95181DATCLONEDHUMAN3H-WIN 35,4284′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95182DATCLONEDHUMAN3H-WIN 35,4284′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95183DATCLONEDHUMAN3H-WIN 35,4284-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95184DATCLONEDHUMAN3H-WIN 35,4282-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate165Jung et al 2021Jan 15, 2025Jan 15, 2025
95185DATCLONEDHUMAN3H-WIN 35,4282-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95186NETCLONEDHUMAN3H-Nisoxetine4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95187NETCLONEDHUMAN3H-Nisoxetine4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95188NETCLONEDHUMAN3H-Nisoxetine4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95189NETCLONEDHUMAN3H-Nisoxetine5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95190NETCLONEDHUMAN3H-Nisoxetine4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95191NETCLONEDHUMAN3H-Nisoxetine4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95192NETCLONEDHUMAN3H-Nisoxetine4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95193NETCLONEDHUMAN3H-Nisoxetine4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95194NETCLONEDHUMAN3H-Nisoxetine4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95195NETCLONEDHUMAN3H-Nisoxetine4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95196NETCLONEDHUMAN3H-Nisoxetine4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95197NETCLONEDHUMAN3H-Nisoxetine2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate469Jung et al 2021Jan 15, 2025Jan 15, 2025
95198NETCLONEDHUMAN3H-Nisoxetine2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95199SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95200SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95201SERTCLONEDHUMAN3H-CITALOPRAM4′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95202SERTCLONEDHUMAN3H-CITALOPRAM5-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95203SERTCLONEDHUMAN3H-CITALOPRAM4′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95204SERTCLONEDHUMAN3H-CITALOPRAM4′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95205SERTCLONEDHUMAN3H-CITALOPRAM4′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95206SERTCLONEDHUMAN3H-CITALOPRAM4′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95207SERTCLONEDHUMAN3H-CITALOPRAM4′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95208SERTCLONEDHUMAN3H-CITALOPRAM4′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95209SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95210SERTCLONEDHUMAN3H-CITALOPRAM2-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate1800Jung et al 2021Jan 15, 2025Jan 28, 2025
95211SERTCLONEDHUMAN3H-CITALOPRAM2-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95212PBRKidney membranesRAT3H-PK111954-(4-(1-Formylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95213PBRKidney membranesRAT3H-PK111954-(4-(1-(2,2,2-Trifluoroacetyl)piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95214PBRKidney membranesRAT3H-PK111954′-(Piperidine-4-carboxamido)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95215PBRKidney membranesRAT3H-PK111955-(4-(4-(Trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3,4′-dicarboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95216PBRKidney membranesRAT3H-PK111954′-(2-Amino-2-oxoethyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2810Jung et al 2021Jan 15, 2025Jan 15, 2025
95217PBRKidney membranesRAT3H-PK111954′-(3-Aminopropyl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95218PBRKidney membranesRAT3H-PK111954′-(3-Aminoprop-1-yn-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95219PBRKidney membranesRAT3H-PK111954′-(5-(Hydroxymethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid751Jung et al 2021Jan 15, 2025Jan 15, 2025
95220PBRKidney membranesRAT3H-PK111954′-(5-(2-Hydroxyethyl)isoxazol-3-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid1930Jung et al 2021Jan 15, 2025Jan 15, 2025
95221PBRKidney membranesRAT3H-PK111954′-(1H-Tetrazol-5-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95222PBRKidney membranesRAT3H-PK111954-(4-(5-(Hydroxymethyl)isoxazol-3-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid4630Jung et al 2021Jan 15, 2025Jan 15, 2025
95223PBRKidney membranesRAT3H-PK111952-(Dimethylamino)-2-oxoethyl 4′-(Piperidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95224PBRKidney membranesRAT3H-PK111952-(Dimethylamino)-2-oxoethyl 4-(4-(1-Acetylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95225D2STRIATUMRAT3H-SPIPERONEN-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide3.3Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95226D2STRIATUMRAT3H-SPIPERONEN-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide118Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95227D2STRIATUMRAT3H-SPIPERONEN-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide0.4Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95228D2STRIATUMRAT3H-SPIPERONEN-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide76.9Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95229D2STRIATUMRAT3H-SPIPERONEN-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide25.7Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95230D2STRIATUMRAT3H-SPIPERONEN-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide0.6Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95231D2STRIATUMRAT3H-SPIPERONEN-[8-(2-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide34.8Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95232D2STRIATUMRAT3H-SPIPERONEN-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide3.6Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95233D2STRIATUMRAT3H-SPIPERONEN-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide0.4Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95234D2STRIATUMRAT3H-SPIPERONEN-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide22.8Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95235D2STRIATUMRAT3H-SPIPERONEN-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide11.6Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95236D2STRIATUMRAT3H-SPIPERONEN-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide4.5Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95237D2STRIATUMRAT3H-SPIPERONEN-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide714.5Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95238D2STRIATUMRAT3H-SPIPERONEN-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide214Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95239D2STRIATUMRAT3H-SPIPERONEN-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide137Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95240D2STRIATUMRAT3H-SPIPERONEN-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide536.7Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95241D2STRIATUMRAT3H-SPIPERONEN-[8-(3-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide217.3Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95242D2STRIATUMRAT3H-SPIPERONEN-[8-(4-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide629Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95243D2STRIATUMRAT3H-SPIPERONEN-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide2200Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95244D2STRIATUMRAT3H-SPIPERONEN-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide2400Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95245D2STRIATUMRAT3H-SPIPERONEN-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide2700Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95246D2STRIATUMRAT3H-SPIPERONEN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide588.6Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
95247D2STRIATUMRAT3H-SPIPERONEN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide>10000Stefanowicz J et al 2016aJan 15, 2025Jan 28, 2025
952485-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide192.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952495-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide182Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952505-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide728.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952515-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide82.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952525-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide212.6Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952535-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide2600Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952545-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide158Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952555-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide298Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952565-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide2500Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952575-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide196.3Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952585-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide199.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952595-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide229.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952605-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide365.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952615-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide210.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952625-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide218Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952635-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide476Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952645-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(3-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide130Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952655-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-[8-(4-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide2000Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952665-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide314.8Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952675-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide484.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952685-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide2300Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952695-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide62.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952705-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide30.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952715-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT5-Hydroxy Tryptamine9.4Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952725-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATDPAT2.3Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952735-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(2-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide854Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952745-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(3-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide231Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952755-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(4-Methylbenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide908Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952765-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(2-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide919.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952775-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(3-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide663Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952785-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(4-Methoxybenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide509Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952795-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(2-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide396.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952805-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(3-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide135.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952815-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(4-Chlorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide571Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952825-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(2-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide326.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952835-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(3-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide105.7Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952845-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(4-Bromobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide298.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952855-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(2-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide141Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952865-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(3-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide101.5Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952875-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(4-Fluorobenzyl)-8-azabicyclo[3.2.1]oct-3b-yl)]-2- naphthamide209Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952885-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(2-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide>10000Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952895-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(3-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide589Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952905-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-[8-(4-Trifluoromethylbenzyl)-8-azabicyclo[3.2.1]oct3b-yl)]-2-naphthamide484Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952915-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-(8-Pyridin-2-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide1116Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952925-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-(8-Pyridin-3-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide502Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952935-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-(8-Pyridin-4-ylmethyl-8-azabicyclo[3.2.1]oct-3b-yl)-2- naphthamide495Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952945-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-quinoline-2- carboxamide1291Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952955-HT2ACEREBRAL CORTEXRAT3H-KETANSERINN-(8-Benzyl-8-azabicyclo[3.2.1]oct-3b-yl)-4-methoxyquinoline-2-carboxamide2315Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952965-HT2ACEREBRAL CORTEXRAT3H-KETANSERINmianserine18.4Stefanowicz J et al 2016aJan 15, 2025Jan 15, 2025
952975-HT2ACLONEDHUMAN3H-KETANSERIN(+) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin470Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
952985-HT2ACLONEDHUMAN3H-KETANSERIN(-) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin100Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
95299H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95300H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95301H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine>10000Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95302H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine430Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95303H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine>10000Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95304H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine200Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95305CB1CLONEDUNDEFINED[3H]-CP 55,9401-(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-heptan-1-one>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95306CB1CLONEDUNDEFINED[3H]-CP 55,940Cyclohexyl-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone298.6Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95307CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-p-tolyl-methanone9429Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95308CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-m-tolyl-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95309CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3,5-dimethyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95310CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-trifluoromethyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95311CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3-trifluoromethyl-phenyl)-methanone4134Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95312CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-ethyl-phenyl)-methanone1138Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95313CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3-ethyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95314CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-propyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95315CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-isopropyl-phenyl)-methanone3326Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95316CB1CLONEDUNDEFINED[3H]-CP 55,940(4-Butyl-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95317CB1CLONEDUNDEFINED[3H]-CP 55,940(4-tert-Butyl-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone2529Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95318CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-hydroxyphenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95319CB1CLONEDUNDEFINED[3H]-CP 55,940(4-Chloro-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone4645Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95320CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-p-tolyl-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95321CB1CLONEDUNDEFINED[3H]-CP 55,940(4-Butyl-phenyl)-(30,50-dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95322CB1CLONEDUNDEFINED[3H]-CP 55,940(4-Chloro-phenyl)-(30,50-dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95323CB1CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dimethoxy-biphenyl-4-yl)-p-tolyl-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95324CB1CLONEDUNDEFINED[3H]-CP 55,940(4-Butyl-phenyl)-(30,50-dichloro-2,6-dimethoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95325CB1CLONEDUNDEFINED[3H]-CP 55,940(4-Chloro-phenyl)-(30,50-dichloro-2,6-dimethoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95326CB1CLONEDUNDEFINED[3H]-CP 55,940SMM-1894778Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95327CB1CLONEDUNDEFINED[3H]-CP 55,940SR144528>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95328CB2CLONEDUNDEFINED[3H]-CP 55,9401-(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-heptan-1-one>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95329CB2CLONEDUNDEFINED[3H]-CP 55,940Cyclohexyl-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone1589Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95330CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-p-tolyl-methanone257.6Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95331CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-m-tolyl-methanone2618Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95332CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3,5-dimethyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95333CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-trifluoromethyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95334CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3-trifluoromethyl-phenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95335CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-ethyl-phenyl)-methanone37.56Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95336CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(3-ethyl-phenyl)-methanone1717Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95337CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-propyl-phenyl)-methanone59.91Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95338CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-isopropyl-phenyl)-methanone160.7Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95339CB2CLONEDUNDEFINED[3H]-CP 55,940(4-Butyl-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone464.4Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95340CB2CLONEDUNDEFINED[3H]-CP 55,940(4-tert-Butyl-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone3166Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95341CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dihydroxy-biphenyl-4-yl)-(4-hydroxyphenyl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95342CB2CLONEDUNDEFINED[3H]-CP 55,940(4-Chloro-phenyl)-(30,50-dichloro-2,6-dihydroxy-biphenyl-4-yl)-methanone120.7Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95343CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-p-tolyl-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95344CB2CLONEDUNDEFINED[3H]-CP 55,940(4-Butyl-phenyl)-(30,50-dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95345CB2CLONEDUNDEFINED[3H]-CP 55,940(4-Chloro-phenyl)-(30,50-dichloro-2-hydroxy-6-methoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95346CB2CLONEDUNDEFINED[3H]-CP 55,940(30,50-Dichloro-2,6-dimethoxy-biphenyl-4-yl)-p-tolyl-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95347CB2CLONEDUNDEFINED[3H]-CP 55,940(4-Butyl-phenyl)-(30,50-dichloro-2,6-dimethoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95348CB2CLONEDUNDEFINED[3H]-CP 55,940(4-Chloro-phenyl)-(30,50-dichloro-2,6-dimethoxy-biphenyl-4-yl)-methanone>10000Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95349CB2CLONEDUNDEFINED[3H]-CP 55,940SMM-189121.3Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95350CB2CLONEDUNDEFINED[3H]-CP 55,940SR14452818.65Presley CS et al 2015Jan 15, 2025Jan 28, 2025
95351A1BRAINRAT[3H]DPCPX3-phenylisochromen-1-one7410Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95352A1BRAINRAT[3H]DPCPX2-phenyl-4H-3,1-benzoxazin-4-one6380Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95353A1BRAINRAT[3H]DPCPX2-(4-fluorophenyl)-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95354A1BRAINRAT[3H]DPCPX2-(4-chlorophenyl)-3,1-benzoxazin-4-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95355A1BRAINRAT[3H]DPCPX2-(4-bromophenyl)-4H-3,1-benzoxazin-4-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95356A1BRAINRAT[3H]DPCPX2-(4-methylphenyl)-3,1-benzoxazin-4-one 100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95357A1BRAINRAT[3H]DPCPX2-(4-methoxyphenyl)-4H-3,1-benzoxazin-4-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95358A1BRAINRAT[3H]DPCPX2-(4-ethoxyphenyl)-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95359A1BRAINRAT[3H]DPCPX2-(furan-2-yl)-4H-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95360A1BRAINRAT[3H]DPCPX2-(thiophen-2-yl)-4H-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95361A1BRAINRAT[3H]DPCPX2-(2-phenylethenyl)-3,1-benzoxazin-4-one >10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95362A1BRAINRAT[3H]DPCPX2-phenyl-3,1-benzoxazin-4-one5060Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95363A1BRAINRAT[3H]DPCPX3-phenylisoquinolin-1(2H)-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95364A1BRAINRAT[3H]DPCPX2-phenylquinazolin-4(3H)-one3670Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95365A1BRAINRAT[3H]DPCPX2-(4-fluorophenyl)quinazolin-4(3H)-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95366A1BRAINRAT[3H]DPCPX2-(4-chlorophenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95367A1BRAINRAT[3H]DPCPX2-(4-bromophenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95368A1BRAINRAT[3H]DPCPX2-(4-methylphenyl)quinazolin-4(3H)-one2500Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95369A1BRAINRAT[3H]DPCPX2-(4-methoxyphenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95370A1BRAINRAT[3H]DPCPX2-(3,4-dimethoxyphenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95371A1BRAINRAT[3H]DPCPX2-(furan-2-yl)quinazolin-4(3H)-one4620Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95372A1BRAINRAT[3H]DPCPX2-(thiophen-2-yl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95373A1BRAINRAT[3H]DPCPX2-[(E)-2-phenylethenyl]quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95374A1BRAINRAT[3H]DPCPX3-phenylchromen-2-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95375A1BRAINRAT[3H]DPCPX3-phenyl-1,4-benzoxazin-2-one >10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95376A1BRAINRAT[3H]DPCPXCPA5.1Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95377A1BRAINRAT[3H]DPCPXZM-241385420Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95378A2ASTRIATUMRAT[3H]NECA3-phenylisochromen-1-one3350Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95379A2ASTRIATUMRAT[3H]NECA2-phenyl-4H-3,1-benzoxazin-4-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95380A2ASTRIATUMRAT[3H]NECA2-(4-fluorophenyl)-3,1-benzoxazin-4-one100Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95381A2ASTRIATUMRAT[3H]NECA2-(4-chlorophenyl)-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95382A2ASTRIATUMRAT[3H]NECA2-(4-bromophenyl)-4H-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95383A2ASTRIATUMRAT[3H]NECA2-(4-methylphenyl)-3,1-benzoxazin-4-one >10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95384A2ASTRIATUMRAT[3H]NECA2-(4-methoxyphenyl)-4H-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95385A2ASTRIATUMRAT[3H]NECA2-(4-ethoxyphenyl)-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95386A2ASTRIATUMRAT[3H]NECA2-(furan-2-yl)-4H-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95387A2ASTRIATUMRAT[3H]NECA2-(thiophen-2-yl)-4H-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95388A2ASTRIATUMRAT[3H]NECA2-(2-phenylethenyl)-3,1-benzoxazin-4-one >10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95389A2ASTRIATUMRAT[3H]NECA2-phenyl-3,1-benzoxazin-4-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95390A2ASTRIATUMRAT[3H]NECA3-phenylisoquinolin-1(2H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95391A2ASTRIATUMRAT[3H]NECA2-phenylquinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95392A2ASTRIATUMRAT[3H]NECA2-(4-fluorophenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95393A2ASTRIATUMRAT[3H]NECA2-(4-chlorophenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95394A2ASTRIATUMRAT[3H]NECA2-(4-bromophenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95395A2ASTRIATUMRAT[3H]NECA2-(4-methylphenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95396A2ASTRIATUMRAT[3H]NECA2-(4-methoxyphenyl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95397A2ASTRIATUMRAT[3H]NECA2-(3,4-dimethoxyphenyl)quinazolin-4(3H)-one2810Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95398A2ASTRIATUMRAT[3H]NECA2-(furan-2-yl)quinazolin-4(3H)-one8110Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95399A2ASTRIATUMRAT[3H]NECA2-(thiophen-2-yl)quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95400A2ASTRIATUMRAT[3H]NECA2-[(E)-2-phenylethenyl]quinazolin-4(3H)-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95401A2ASTRIATUMRAT[3H]NECA3-phenylchromen-2-one>10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95402A2ASTRIATUMRAT[3H]NECA3-phenyl-1,4-benzoxazin-2-one >10000Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95403A2ASTRIATUMRAT[3H]NECACPA557Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95404A2ASTRIATUMRAT[3H]NECAZM-2413851.3Pieterse L et al 2020Jan 15, 2025Jan 15, 2025
95405D2CLONEDHUMAN[3H]-Raclopride5-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)quinoline1237Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95406D2CLONEDHUMAN[3H]-Raclopride4-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)isoquinoline1218Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95407D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline141Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95408D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline223Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95409D2CLONEDHUMAN[3H]-Raclopride4-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline418Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95410D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline76Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95411D2CLONEDHUMAN[3H]-Raclopride4-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline37Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95412D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline1821Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95413D2CLONEDHUMAN[3H]-Raclopride4-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline1022Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95414D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)quinoline149Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95415D2CLONEDHUMAN[3H]-Raclopride4-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)isoquinoline148Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95416D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline36Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95417D2CLONEDHUMAN[3H]-Raclopride4-({4-(2-[4-(2,3-Dichlorophenyl)iperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline30Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95418D2CLONEDHUMAN[3H]-Raclopride5-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline121Partyka A et al 2017Jan 15, 2025Jan 28, 2025
95419D2CLONEDHUMAN[3H]-Raclopride4-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl) isoquinoline145Partyka A et al 2017Jan 15, 2025Jan 28, 2025
954205-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)quinoline749Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954215-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)isoquinoline543Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954225-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline740Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954235-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline759Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954245-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline975Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954255-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline54Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954265-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline32Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954275-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline609Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954285-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline370Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954295-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)quinoline40Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954305-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)isoquinoline30Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954315-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline45Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954325-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-(2-[4-(2,3-Dichlorophenyl)iperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline29Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954335-HT1ACLONEDHUMAN[3H]-8-OH-DPAT5-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline257Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954345-HT1ACLONEDHUMAN[3H]-8-OH-DPAT4-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl) isoquinoline324Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954355-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)quinoline646Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954365-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)isoquinoline410Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954375-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline152Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954385-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline139Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954395-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline156Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954405-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline197Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954415-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline157Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954425-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline665Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954435-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline691Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954445-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)quinoline530Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954455-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)isoquinoline161Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954465-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline286Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954475-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-(2-[4-(2,3-Dichlorophenyl)iperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline371Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954485-HT2ACLONEDHUMAN[3H]-ketanserin5-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline336Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954495-HT2ACLONEDHUMAN[3H]-ketanserin4-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl) isoquinoline179Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954505-HT6CLONEDHUMAN[3H]-LSD5-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)quinoline6712Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954515-HT6CLONEDHUMAN[3H]-LSD4-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)isoquinoline2412Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954525-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline1020Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954535-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline1459Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954545-HT6CLONEDHUMAN[3H]-LSD4-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline1863Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954555-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline445Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954565-HT6CLONEDHUMAN[3H]-LSD4-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline1185Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954575-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline8279Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954585-HT6CLONEDHUMAN[3H]-LSD4-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline3802Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954595-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)quinoline640Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954605-HT6CLONEDHUMAN[3H]-LSD4-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)isoquinoline1016Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954615-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline401Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954625-HT6CLONEDHUMAN[3H]-LSD4-({4-(2-[4-(2,3-Dichlorophenyl)iperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline309Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954635-HT6CLONEDHUMAN[3H]-LSD5-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline791Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954645-HT6CLONEDHUMAN[3H]-LSD4-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl) isoquinoline1041Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954655-HT7CLONEDHUMAN[3H]-5-CT5-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)quinoline209Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954665-HT7CLONEDHUMAN[3H]-5-CT4-({4-[2-(4-Phenylpiperazin-1-yl)ethyl]piperidin-1-yl}sulfonyl)isoquinoline174Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954675-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline37Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954685-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline29Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954695-HT7CLONEDHUMAN[3H]-5-CT4-({4-(2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline14Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954705-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline37Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954715-HT7CLONEDHUMAN[3H]-5-CT4-({4-(2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline18Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954725-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline165Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954735-HT7CLONEDHUMAN[3H]-5-CT4-({4-(2-[4-(3-Fluorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline142Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954745-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)quinoline56Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954755-HT7CLONEDHUMAN[3H]-5-CT4-({4-(2-(4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl)ethyl)piperidin-1-yl}sulfonyl)isoquinoline52Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954765-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-[4-(2,3-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline55Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954775-HT7CLONEDHUMAN[3H]-5-CT4-({4-(2-[4-(2,3-Dichlorophenyl)iperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)isoquinoline39Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954785-HT7CLONEDHUMAN[3H]-5-CT5-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl)quinoline52Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954795-HT7CLONEDHUMAN[3H]-5-CT4-({4-(2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl)piperidin-1-yl}sulfonyl) isoquinoline36Partyka A et al 2017Jan 15, 2025Jan 15, 2025
954805-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT1,3-dimethyl-7-[2-(4-phenylpiperazin-1-yl)ethyl]purine-2,6-dione571Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954815-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione 119Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954825-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione  182Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954835-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione23Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954845-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione1.2Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954855-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione1Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954865-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride55Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954875-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride105Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954885-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione11Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954895-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione1Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954905-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione5Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954915-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride433Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954925-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride239Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954935-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPAT7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride171Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954945-HT1AHIPPOCAMPUSRAT[3H]-8-OH-DPATBUSPIRONE20Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954955-HT2ACORTEXRAT[3H]-ketanserin1,3-dimethyl-7-[2-(4-phenylpiperazin-1-yl)ethyl]purine-2,6-dione92Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954965-HT2ACORTEXRAT[3H]-ketanserin7-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione 927Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954975-HT2ACORTEXRAT[3H]-ketanserin7-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione  53Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954985-HT2ACORTEXRAT[3H]-ketanserin1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione507Partyka A et al 2015Jan 15, 2025Jan 15, 2025
954995-HT2ACORTEXRAT[3H]-ketanserin7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione1055Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955005-HT2ACORTEXRAT[3H]-ketanserin7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione102Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955015-HT2ACORTEXRAT[3H]-ketanserin7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride162Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955025-HT2ACORTEXRAT[3H]-ketanserin7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride460Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955035-HT2ACORTEXRAT[3H]-ketanserin1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione308Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955045-HT2ACORTEXRAT[3H]-ketanserin7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione598Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955055-HT2ACORTEXRAT[3H]-ketanserin7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione54Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955065-HT2ACORTEXRAT[3H]-ketanserin7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955075-HT2ACORTEXRAT[3H]-ketanserin7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955085-HT2ACORTEXRAT[3H]-ketanserin7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955095-HT2ACORTEXRAT[3H]-ketanserinOLANZAPINE4.6Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955105-HT6CLONEDHUMAN[3H]-LSD1,3-dimethyl-7-[2-(4-phenylpiperazin-1-yl)ethyl]purine-2,6-dione>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955115-HT6CLONEDHUMAN[3H]-LSD7-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione >10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955125-HT6CLONEDHUMAN[3H]-LSD7-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione  >10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955135-HT6CLONEDHUMAN[3H]-LSD1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955145-HT6CLONEDHUMAN[3H]-LSD7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione1970Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955155-HT6CLONEDHUMAN[3H]-LSD7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione5150Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955165-HT6CLONEDHUMAN[3H]-LSD7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride68Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955175-HT6CLONEDHUMAN[3H]-LSD7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride1902Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955185-HT6CLONEDHUMAN[3H]-LSD1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955195-HT6CLONEDHUMAN[3H]-LSD7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione8987Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955205-HT6CLONEDHUMAN[3H]-LSD7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione1195Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955215-HT6CLONEDHUMAN[3H]-LSD7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955225-HT6CLONEDHUMAN[3H]-LSD7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride>10000Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955235-HT6CLONEDHUMAN[3H]-LSD7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride9141Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955245-HT6CLONEDHUMAN[3H]-LSDOLANZAPINE7Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955255-HT7CLONEDHUMAN[3H]-5-CT1,3-dimethyl-7-[2-(4-phenylpiperazin-1-yl)ethyl]purine-2,6-dione1429Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955265-HT7CLONEDHUMAN[3H]-5-CT7-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione 2210Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955275-HT7CLONEDHUMAN[3H]-5-CT7-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione  2800Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955285-HT7CLONEDHUMAN[3H]-5-CT1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione1148Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955295-HT7CLONEDHUMAN[3H]-5-CT7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione434Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955305-HT7CLONEDHUMAN[3H]-5-CT7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione479Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955315-HT7CLONEDHUMAN[3H]-5-CT7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride73Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955325-HT7CLONEDHUMAN[3H]-5-CT7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride179Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955335-HT7CLONEDHUMAN[3H]-5-CT1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione346Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955345-HT7CLONEDHUMAN[3H]-5-CT7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione294Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955355-HT7CLONEDHUMAN[3H]-5-CT7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione131Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955365-HT7CLONEDHUMAN[3H]-5-CT7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride3616Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955375-HT7CLONEDHUMAN[3H]-5-CT7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride629Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955385-HT7CLONEDHUMAN[3H]-5-CT7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride1009Partyka A et al 2015Jan 15, 2025Jan 15, 2025
955395-HT7CLONEDHUMAN[3H]-5-CTCLOZAPINE18Partyka A et al 2015Jan 15, 2025Jan 15, 2025
95540D2STRIATUMRAT[3H]-spiperone1,3-dimethyl-7-[2-(4-phenylpiperazin-1-yl)ethyl]purine-2,6-dione1088Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95541D2STRIATUMRAT[3H]-spiperone7-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione 944Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95542D2STRIATUMRAT[3H]-spiperone7-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]-1,3-dimethylpurine-2,6-dione  3187Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95543D2STRIATUMRAT[3H]-spiperone1,3-dimethyl-7-[3-(4-phenylpiperazin-1-yl)propyl]purine-2,6-dione1006Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95544D2STRIATUMRAT[3H]-spiperone7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione65Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95545D2STRIATUMRAT[3H]-spiperone7-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,3-dimethylpurine-2,6-dione195Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95546D2STRIATUMRAT[3H]-spiperone7-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride15Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95547D2STRIATUMRAT[3H]-spiperone7-{4-[4-(3,4-Dichlorophenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-purine-2,6-dione hydrochloride73Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95548D2STRIATUMRAT[3H]-spiperone1,3-dimethyl-7-[4-(4-phenylpiperazin-1-yl)butyl]purine-2,6-dione356Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95549D2STRIATUMRAT[3H]-spiperone7-[4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione33Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95550D2STRIATUMRAT[3H]-spiperone7-[4-[4-(3-chlorophenyl)piperazin-1-yl]butyl]-1,3-dimethylpurine-2,6-dione40Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95551D2STRIATUMRAT[3H]-spiperone7-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-1,3-dimethyl-purine-2,6-dione hydrochloride2705Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95552D2STRIATUMRAT[3H]-spiperone7-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-1,3-dimethyl-purine-2,6-dione hydrochloride7823Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95553D2STRIATUMRAT[3H]-spiperone7-[5-(3,4-Dihydro-1H-isoquinolin-2-yl)-pentyl]-1,3-dimethyl-purine-2,6-dione hydrochloride1222Partyka A et al 2015Jan 15, 2025Jan 28, 2025
95554D2CLONEDRAT[3H]-spiperoneOLANZAPINE7Partyka A et al 2015Jan 15, 2025Jan 28, 2025
955555-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine320Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955565-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine110Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955575-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine130Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955585-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine40Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955595-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine260Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955605-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine20Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955615-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine1300Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955625-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine80Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955635-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine500Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955645-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine74Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955655-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine71Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955665-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine140Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955675-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine50Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955685-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine250Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955695-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine60Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955705-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine220Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955715-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine210Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955725-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine2000Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955735-HT2ACLONEDHUMAN3H-KETANSERIN(+/-)trans-4-(4' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine8100Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955745-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine760Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955755-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1100Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955765-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine80Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955775-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine20Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955785-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine370Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955795-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine30Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955805-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine650Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955815-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine44Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955825-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2800Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955835-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2400Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955845-HT2ACLONEDHUMAN3H-KETANSERIN(+)trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine700Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955855-HT2ACLONEDHUMAN3H-KETANSERIN(-)trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1000Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955865-HT2BCLONEDHUMAN3H-MESULERGINE(+) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin240Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955875-HT2BCLONEDHUMAN3H-MESULERGINE(-) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin94Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955885-HT2BCLONEDHUMAN3H-MESULERGINE(+) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine110Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955895-HT2BCLONEDHUMAN3H-MESULERGINE(-) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine70Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955905-HT2BCLONEDHUMAN3H-MESULERGINE(+) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine50Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955915-HT2BCLONEDHUMAN3H-MESULERGINE(-) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine30Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955925-HT2BCLONEDHUMAN3H-MESULERGINE(+) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine40Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955935-HT2BCLONEDHUMAN3H-MESULERGINE(-) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine8Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955945-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine200Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955955-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine60Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955965-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine20Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955975-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine70Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955985-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine66Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
955995-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine400Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956005-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine80Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956015-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine300Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956025-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine30Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956035-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine210Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956045-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine250Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956055-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine540Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956065-HT2BCLONEDHUMAN[3H] Mesulergine(+/-) trans-4-(4' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine4100Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956075-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine4100Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956085-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine650Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956095-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine170Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956105-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine20Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956115-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine40Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956125-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine10Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956135-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine200Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956145-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine73Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956155-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine710Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956165-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine300Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956175-HT2BCLONEDHUMAN[3H] Mesulergine(+) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine6000Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956185-HT2BCLONEDHUMAN[3H] Mesulergine(-) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine800Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956195-HT2CCLONEDHUMAN[3H] Mesulergine(+) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin430Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956205-HT2CCLONEDHUMAN[3H] Mesulergine(-) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin30Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956215-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine200Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956225-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine43Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956235-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine170Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956245-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine8Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956255-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine200Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956265-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine4Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956275-HT2CCLONEDHUMAN[3H] Mesulergine(+)trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine230Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956285-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine10Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956295-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine120Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956305-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine10Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956315-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine75Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956325-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4'-Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine68Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956335-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine55Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956345-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine120Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956355-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine70Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956365-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine100Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956375-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine220Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956385-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine520Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956395-HT2CCLONEDHUMAN[3H] Mesulergine(+/-) trans-4-(4' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1000Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956405-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine78Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956415-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine70Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956425-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine30Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956435-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-Cyclohexyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine7Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956445-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine800Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956455-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-Cyclooctyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine30Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956465-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1000Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956475-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(Biphenyl-3-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine5Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956485-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine50Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956495-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine290Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956505-HT2CCLONEDHUMAN[3H] Mesulergine(+) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2000Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
956515-HT2CCLONEDHUMAN[3H] Mesulergine(-) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1600Sakhuja R et al 2015Jan 15, 2025Jan 15, 2025
95652H1CLONEDHUMAN3H-MEPYRAMINE(+) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin30Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95653H1CLONEDHUMAN3H-MEPYRAMINE(-) (2S,4R)-()-trans-4-phenyl-N, N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine (4-phenyl2-dimethylaminotetralin2Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95654H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine94Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95655H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(3' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine3Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95656H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine80Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95657H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(3' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine10Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95658H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine60Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95659H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(3' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine30Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95660H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(3' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine4100Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95661H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(3'-Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine230Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95662H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1000Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95663H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(3' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine800Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95664H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine8Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95665H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(4' -Fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine4Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95666H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine6Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95667H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(4' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine8Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95668H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine530Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95669H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(4' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine1100Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95670H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine230Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95671H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(4' -Trifluoromethylphenyl)-N,N-dimethyl-1,2,3,4- tetrahydronaphthalen-2-amine5100Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95672H1CLONEDHUMAN3H-MEPYRAMINE(+/-) trans-4-(4' -Nitrophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine680Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95673H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine2600Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95674H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(2' -Bromophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine4200Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95675H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine60Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95676H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(2' -Chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine190Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95677H1CLONEDHUMAN3H-MEPYRAMINE(+) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine120Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
95678H1CLONEDHUMAN3H-MEPYRAMINE(-) trans-4-(2' -Methylphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine400Sakhuja R et al 2015Jan 15, 2025Jan 28, 2025
956795-HT1ACLONEDHUMAN3H-WAY1006356-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956805-HT1ACLONEDHUMAN3H-WAY100635Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956815-HT1ACLONEDHUMAN3H-WAY100635Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956825-HT1ACLONEDHUMAN3H-WAY1006356-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956835-HT1ACLONEDHUMAN3H-WAY100635N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956845-HT1ACLONEDHUMAN3H-WAY100635tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956855-HT1ACLONEDHUMAN3H-WAY1006354-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956865-HT1ACLONEDHUMAN3H-WAY1006352-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956875-HT1BCLONEDHUMAN3H-GR1257436-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956885-HT1BCLONEDHUMAN3H-GR125743Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956895-HT1BCLONEDHUMAN3H-GR125743Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956905-HT1BCLONEDHUMAN3H-GR1257436-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956915-HT1BCLONEDHUMAN3H-GR125743N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956925-HT1BCLONEDHUMAN3H-GR125743tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956935-HT1BCLONEDHUMAN3H-GR1257434-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956945-HT1BCLONEDHUMAN3H-GR1257432-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956955-HT1DCLONEDHUMAN3H-GR1257436-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956965-HT1DCLONEDHUMAN3H-GR125743Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956975-HT1DCLONEDHUMAN3H-GR125743Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956985-HT1DCLONEDHUMAN3H-GR1257436-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
956995-HT1DCLONEDHUMAN3H-GR125743N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957005-HT1DCLONEDHUMAN3H-GR125743tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957015-HT1DCLONEDHUMAN3H-GR1257434-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957025-HT1DCLONEDHUMAN3H-GR1257432-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957035-HT1ECLONEDHUMAN3H-5-HT6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957045-HT1ECLONEDHUMAN3H-5-HTTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957055-HT1ECLONEDHUMAN3H-5-HTTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957065-HT1ECLONEDHUMAN3H-5-HT6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957075-HT1ECLONEDHUMAN3H-5-HTN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957085-HT1ECLONEDHUMAN3H-5-HTtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957095-HT1ECLONEDHUMAN3H-5-HT4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957105-HT1ECLONEDHUMAN3H-5-HT2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957115-HT2ACLONEDHUMAN3H-KETANSERIN6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957125-HT2ACLONEDHUMAN3H-KETANSERINTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957135-HT2ACLONEDHUMAN3H-KETANSERINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957145-HT2ACLONEDHUMAN3H-KETANSERIN6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957155-HT2ACLONEDHUMAN3H-KETANSERINN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957165-HT2ACLONEDHUMAN3H-KETANSERINtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957175-HT2ACLONEDHUMAN3H-KETANSERIN4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957185-HT2ACLONEDHUMAN3H-KETANSERIN2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957195-HT2BCLONEDHUMAN3H-LSD6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957205-HT2BCLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957215-HT2BCLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957225-HT2BCLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957235-HT2BCLONEDHUMAN3H-LSDN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957245-HT2BCLONEDHUMAN3H-LSDtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957255-HT2BCLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957265-HT2BCLONEDHUMAN3H-LSD2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957275-HT2CCLONEDHUMAN3H-MESULERGINE6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957285-HT2CCLONEDHUMAN3H-MESULERGINETrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957295-HT2CCLONEDHUMAN3H-MESULERGINETriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957305-HT2CCLONEDHUMAN3H-MESULERGINE6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957315-HT2CCLONEDHUMAN3H-MESULERGINEN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957325-HT2CCLONEDHUMAN3H-MESULERGINEtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957335-HT2CCLONEDHUMAN3H-MESULERGINE4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957345-HT2CCLONEDHUMAN3H-MESULERGINE2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957355-HT3CLONEDHUMAN3H-GR656306-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957365-HT3CLONEDHUMAN3H-GR65630Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957375-HT3CLONEDHUMAN3H-GR65630Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957385-HT3CLONEDHUMAN3H-GR656306-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957395-HT3CLONEDHUMAN3H-GR65630N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957405-HT3CLONEDHUMAN3H-GR65630tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957415-HT3CLONEDHUMAN3H-GR656304-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957425-HT3CLONEDHUMAN3H-GR656302-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957435-HT5ACLONEDHUMAN3H-LSD6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957445-HT6CLONEDHUMAN3H-LSD6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957455-HT7CLONEDHUMAN3H-LSD6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957465-HT5ACLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957475-HT6CLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957485-HT7CLONEDHUMAN3H-LSDTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025