The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 95,001-96,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
97749H2Sf9HUMANFunctionalHIS1200Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97750H2Sf9HUMANFunctionalUR-AK411400Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97751H2Sf9HUMANFunctionalUR-AK26150Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97752H2Sf9HUMANFunctionalUR-AK51100Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97753H2Sf9HUMANFunctionalUR-AK6767Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97754H2Sf9HUMANFunctionalUR-AK2272Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97755H2Sf9HUMANFunctionalUR-AK6875Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97756H2Sf9HUMANFunctionalUR-AK2467Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97757H2Sf9HUMANFunctionalUR-AK4638Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97758H2Sf9HUMANFunctionalUR-AK6262Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97759H2Sf9HUMANFunctionalUR-AK4946Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97760H2Sf9HUMANFunctionalUR-AK6423Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97761H2Sf9HUMANFunctionalUR-AK5999Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97762H2Sf9HUMANFunctionalUR-AK5723Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97763H2Sf9GUINEA PIGFunctionalUR-AK579Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97764H2Sf9GUINEA PIGFunctionalUR-AK5937Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97765H2Sf9GUINEA PIGFunctionalUR-AK6416Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97766H2Sf9GUINEA PIGFunctionalUR-AK4922Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97767H2Sf9GUINEA PIGFunctionalUR-AK41640Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97768H2Sf9GUINEA PIGFunctionalUR-AK2676Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97769H2Sf9GUINEA PIGFunctionalUR-AK5123Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97770H2Sf9GUINEA PIGFunctionalUR-AK6721Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97771H2Sf9GUINEA PIGFunctionalUR-AK2256Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97772H2Sf9GUINEA PIGFunctionalUR-AK6829Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97773H2Sf9GUINEA PIGFunctionalUR-AK2412Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97774H2Sf9GUINEA PIGFunctionalUR-AK4621Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97775H2Sf9GUINEA PIGFunctionalUR-AK6223Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97776H2Sf9GUINEA PIGFunctionalHIS1200Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97777H1Sf9HUMANFunctionalHIS190Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97778H1Sf9HUMANFunctionalUR-AK683500Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97779H1Sf9HUMANFunctionalUR-AK46>10000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97780H1Sf9HUMANFunctionalUR-AK592300Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97781H1Sf9HUMANFunctionalUR-AK57280Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97782H1Sf9HUMAN3H-MEPYRAMINEUR-AK57910Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97783H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK571600Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97784H1Sf9HUMAN3H-MEPYRAMINEHIS2000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97785H1Sf9GUINEA PIG3H-MEPYRAMINEHIS4600Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97786H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK672200Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97787H1Sf9HUMAN3H-MEPYRAMINEUR-AK67>10000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97788H1Sf9HUMAN3H-MEPYRAMINEUR-AK222900Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97789H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK22440Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97790H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK242600Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97791H1Sf9HUMAN3H-MEPYRAMINEUR-AK245300Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97792H1Sf9HUMAN3H-MEPYRAMINEUR-AK627000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97793H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK624700Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97794H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK64350Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97795H1Sf9HUMAN3H-MEPYRAMINEUR-AK64990Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97796H1Sf9HUMAN3H-MEPYRAMINEUR-AK596000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97797H1Sf9GUINEA PIG3H-MEPYRAMINEUR-AK59>10000Xie, S. et. al., 2006Jan 15, 2025Jan 15, 2025
97798L1210 cellsUNDEFINEDFunctionaldihydroMotu (3,3)c3000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97799L1210 cellsUNDEFINED14C-spermidinedihydroMotu (3,3)c9900Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97800L1210 cellsUNDEFINED14C-spermidinedihydroMotu (4,4)6200Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97801L1210 cellsUNDEFINEDFunctionaldihydroMotu (4,4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97802L1210 cellsUNDEFINEDFunctionalAnt-CH2 (3,3)d1800Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97803L1210 cellsUNDEFINED14C-spermidineAnt-CH2 (3,3)d>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97804L1210 cellsUNDEFINED14C-spermidineAnt-CH2 (4,4)1800Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97805L1210 cellsUNDEFINEDFunctionalAnt-CH2 (4,4)300Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97806L1210 cellsUNDEFINEDFunctionalAnt-CH2CH2 (4,4)3500Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97807L1210 cellsUNDEFINED14C-spermidineAnt-CH2CH2 (4,4)1600Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97808L1210 cellsUNDEFINED14C-spermidineAnt-CH2CH2CH2 (4, 4)1100Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97809L1210 cellsUNDEFINEDFunctionalAnt-CH2CH2CH2 (4, 4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97810L1210 cellsUNDEFINEDFunctionalN1-ethyl-N1-Ant-CH2 (3,3)2200Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97811L1210 cellsUNDEFINED14C-spermidineN1-ethyl-N1-Ant-CH2 (3,3)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97812L1210 cellsUNDEFINED14C-spermidineN1-ethyl-N1-Ant-CH2 (4,4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97813L1210 cellsUNDEFINEDFunctionalN1-ethyl-N1-Ant-CH2 (4,4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97814CLONEDUNDEFINEDFunctionalN1-ethyl-N1-Ant-CH2 (4,4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97815CLONEDUNDEFINEDFunctionalN1-ethyl-N1-Ant-CH2 (3,3)5300Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97816CLONEDUNDEFINEDFunctionalAnt-CH2CH2CH2 (4, 4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97817CLONEDUNDEFINEDFunctionalAnt-CH2CH2 (4,4)9800Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97818CLONEDUNDEFINEDFunctionalAnt-CH2 (4,4)450Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97819CLONEDUNDEFINEDFunctionalAnt-CH2 (3,3)d1900Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97820CLONEDUNDEFINEDFunctionaldihydroMotu (4,4)>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97821CLONEDUNDEFINEDFunctionaldihydroMotu (3,3)c>10000Breitbeil III F, et al., 2006Jan 15, 2025Jan 15, 2025
97822L1210 cellsUNDEFINEDFunctionalAntmethyl (3,3)1800Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97823L1210 cellsUNDEFINED14C-spermidineAntmethyl (3,3)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97824CHO (COX-1)cellsUNDEFINEDFunctionalAntmethyl (3,3)1900Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97825CHO (COX-1)cellsUNDEFINEDFunctionalAntmethyl(4,4)450Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97826L1210 cellsUNDEFINED14C-spermidineAntmethyl(4,4)1800Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97827L1210 cellsUNDEFINEDFunctionalAntmethyl(4,4)300Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97828L1210 cellsUNDEFINEDFunctionaldihydroMotu (3,3)3000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97829L1210 cellsUNDEFINED14C-spermidinedihydroMotu (3,3)9900Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97830CHO (COX-1)cellsUNDEFINEDFunctionaldihydroMotu (3,3)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97831CHO (COX-1)cellsUNDEFINEDFunctionaldihydroMotu (4,4)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97832L1210 cellsUNDEFINED14C-spermidinedihydroMotu (4,4)6200Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97833L1210 cellsUNDEFINEDFunctionaldihydroMotu (4,4)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97834L1210 cellsUNDEFINEDFunctionalN-ethyl-N-Antmethyl (4,4)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97835L1210 cellsUNDEFINED14C-spermidineN-ethyl-N-Antmethyl (4,4)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
97836CHO (COX-1)cellsUNDEFINEDFunctionalN-ethyl-N-Antmethyl (4,4)>10000Kaur N, et al., 2005Jan 15, 2025Jan 15, 2025
978375-HT2AMembranesHUMAN[3H]-ketanserinRITANSERIN0.0831764Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978385-HT2ACLONEDHUMANFunctionalRITANSERIN0.0691831Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978395-HT2ACLONEDHUMANFunctionalMDL 1009071.14815Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978405-HT2ACLONEDHUMANFunctionalEplivanserin1.04713Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978415-HT2ACLONEDHUMANFunctionalCLOZAPINE13.4896Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978425-HT2ACLONEDHUMANFunctionalACP-1031.86209Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978435-HT2AMembranesHUMAN[3H]-ketanserinMDL 1009070.0301995Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978445-HT2AMembranesHUMAN[3H]-ketanserinEplivanserin0.0457088Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978455-HT2AMembranesHUMAN[3H]-ketanserinACP-1030.501187Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978465-HT2AMembranesHUMAN[3H]-ketanserinCLOZAPINE0.549541Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978475-HT2CMembranesHUMAN3H-MESULERGINECLOZAPINE1.31826Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978485-HT2CMembranesHUMAN3H-MESULERGINEACP-1031.58489Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978495-HT2CMembranesHUMAN3H-MESULERGINEEplivanserin1.34896Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978505-HT2CMembranesHUMAN3H-MESULERGINEMDL 1009073.80189Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978515-HT2CMembranesHUMAN3H-MESULERGINERITANSERIN0.436516Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978525-HT2CCELLSHUMAN3H-MESULERGINERITANSERIN24.5471Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978535-HT2CCELLSHUMAN3H-MESULERGINEMDL 100907446.684Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978545-HT2CCELLSHUMAN3H-MESULERGINEEplivanserin741.31Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978555-HT2CCELLSHUMAN3H-MESULERGINEACP-10310Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978565-HT2CCELLSHUMAN3H-MESULERGINECLOZAPINE691.831Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978575-HT2ACELLSHUMAN[3H]-ketanserinCLOZAPINE1.31826Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978585-HT2ACELLSHUMAN[3H]-ketanserinMDL 1009070.17378Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978595-HT2ACELLSHUMAN[3H]-ketanserinEplivanserin0.398107Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978605-HT2ACELLSHUMAN[3H]-ketanserinACP-1030.199526Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
978615-HT2ACELLSHUMAN[3H]-ketanserinCLOZAPINE5.88844Vanover, K., et al., 2006Jan 15, 2025Jan 15, 2025
97862SLC6A3CORTICALRAT3H-DA UPTAKEBUPROPION550Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97863SLC6A3CORTICALRAT3H-DA UPTAKE(2RS,3RS)-Hydroxybupropion>10000Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97864SLC6A3CORTICALRAT3H-DA UPTAKE(2S,3S)-Hydroxybupropion790Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97865SLC6A3CORTICALRAT3H-DA UPTAKE(2R,3R)-Hydroxybupropion>10000Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97866NETCORTICALRAT3H-NE Uptake(2R,3R)-Hydroxybupropion>10000Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97867NETCORTICALRAT3H-NE Uptake(2S,3S)-Hydroxybupropion520Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97868NETCORTICALRAT3H-NE Uptake(2RS,3RS)-Hydroxybupropion1700Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97869NETCORTICALRAT3H-NE UptakeBUPROPION1900Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97870nAChRCLONEDHUMANFunctionalBUPROPION1800Damaj, I. et al., 2004Jan 15, 2025Jan 28, 2025
97871nAChRCLONEDHUMANFunctional(2S,3S) OH-bupropion>10000Damaj, I. et al., 2004Jan 15, 2025Jan 28, 2025
97872nAChRCLONEDHUMANFunctional(2R,3R)-OH-bupropion6500Damaj, I. et al., 2004Jan 15, 2025Jan 28, 2025
97873nAChRCLONEDHUMANFunctional(2R,3R)-OH-bupropion3100Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97874nAChRCLONEDHUMANFunctional(2S,3S) OH-bupropion3300Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97875nAChRCLONEDHUMANFunctionalBUPROPION>10000Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97876nAChRCLONEDHUMANFunctionalBUPROPION>10000Damaj, I. et al., 2004Jan 15, 2025Jan 27, 2025
97877nAChRCLONEDHUMANFunctional(2S,3S) OH-bupropion>10000Damaj, I. et al., 2004Jan 15, 2025Jan 27, 2025
97878nAChRCLONEDHUMANFunctional(2R,3R)-OH-bupropion>10000Damaj, I. et al., 2004Jan 15, 2025Jan 27, 2025
97879nAchR1CLONEDHUMANFunctionalBUPROPION7900Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97880nAchR1CLONEDHUMANFunctionalBUPROPION>10000Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97881nAchR1CLONEDHUMANFunctionalBUPROPION7600Damaj, I. et al., 2004Jan 15, 2025Jan 15, 2025
97882SLC6A3BRAINRAT3H-dopamineAmphetamine,(+)34Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97883SLC6A3BRAINRAT3H-dopaminediethylpropion>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97884SLC6A3BRAINRAT3H-dopamine(±)-2-ethylamino-1-phenyl-propan-1-one1014Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97885SLC6A3BRAINRAT3H-dopamine(1R,2S)-(−)-N,N-diethylnorephedrine>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97886SLC6A3BRAINRAT3H-dopamine(1S,2R)-(−)-N,N-diethylnorephedrine>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97887SLC6A4BRAINRAT3H-5HT(1S,2R)-(−)-N,N-diethylnorephedrine>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97888SLC6A4BRAINRAT3H-5HT(1R,2S)-(−)-N,N-diethylnorephedrine>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97889SLC6A4BRAINRAT3H-5HT(±)-2-ethylamino-1-phenyl-propan-1-one3840Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97890SLC6A4BRAINRAT3H-5HTdiethylpropion>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97891SLC6A4BRAINRAT3H-5HTAmphetamine,(+)>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97892NETBRAINRAT3H-NorepinephrineAmphetamine,(+)38.9Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97893NETBRAINRAT3H-Norepinephrinediethylpropion>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97894NETBRAINRAT3H-Norepinephrine(±)-2-ethylamino-1-phenyl-propan-1-one360Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97895NETBRAINRAT3H-Norepinephrine(1R,2S)-(−)-N,N-diethylnorephedrine>10000Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97896NETBRAINRAT3H-Norepinephrine(1S,2R)-(−)-N,N-diethylnorephedrine6820Yu, H, et al., 2000Jan 15, 2025Jan 15, 2025
97897HEK293 cellsHUMAN3H-AMPALY 2935589200Bleakman, D., et al., 1999Jan 15, 2025Jan 15, 2025
97898mGluR2HEK293 cellsHUMAN3H-AMPALY 2935583200Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97899AMPAHEK293 cellsHUMAN3H-AMPALY 293558>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 15, 2025
97900mGluR4HEK293 cellsHUMAN3H-AMPALY 293558>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97901Kainate receptorHEK293 cellsHUMAN3H-Kainic acidLY 2935584200Bleakman, D., et al., 1999Jan 15, 2025Jan 15, 2025
97902Kainate receptorHEK293 cellsHUMAN3H-Kainic acidLY 293558>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 28, 2025
97903mGluR6HEK293 cellsHUMAN3H-Kainic acidLY 293558>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97904mGluR7HEK293 cellsHUMAN3H-Kainic acidLY 293558>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97905HEK293 cellsHUMAN3H-AMPANBQX1600Bleakman, D., et al., 1999Jan 15, 2025Jan 15, 2025
97906mGluR2HEK293 cellsHUMAN3H-AMPANBQX260Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97907AMPAHEK293 cellsHUMAN3H-AMPANBQX900Bleakman, D., et al., 1999Jan 15, 2025Jan 15, 2025
97908mGluR4HEK293 cellsHUMAN3H-AMPANBQX600Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97909Kainate receptorHEK293 cellsHUMAN3H-Kainic acidNBQX>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 15, 2025
97910Kainate receptorHEK293 cellsHUMAN3H-Kainic acidNBQX>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 28, 2025
97911mGluR6HEK293 cellsHUMAN3H-Kainic acidNBQX600Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97912mGluR7HEK293 cellsHUMAN3H-Kainic acidNBQX>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 29, 2025
97913Kainate receptorHEK293 cellsHUMAN3H-Kainic acidNBQX>10000Bleakman, D., et al., 1999Jan 15, 2025Jan 28, 2025
97914NETBRAINRAT3H-NorepinephrineAmphetamine,(+)38.9Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97915NETBRAINRAT3H-NorepinephrineMETHAMPHETAMINE (+)48Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97916NETBRAINRAT3H-NorepinephrinePhentermine244Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97917NETBRAINRAT3H-Norepinephrinediethylpropion1810Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97918NETBRAINRAT3H-NorepinephrineN-dealkylated Diethylpropion360Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97919NETBRAINRAT3H-NorepinephrinePhendimetrazine8300Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97920NETBRAINRAT3H-NorepinephrinePhendimetrazine-(+)240Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97921NETBRAINRAT3H-NorepinephrinePhendimetrazine-(-)388Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97922SLC6A3BRAINRAT3H-dopaminePhendimetrazine-(-)1669Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97923SLC6A3BRAINRAT3H-dopaminePhendimetrazine-(+)359Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97924SLC6A3BRAINRAT3H-dopaminePhendimetrazine>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97925SLC6A3BRAINRAT3H-dopamineN-dealkylated Diethylpropion1014Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97926SLC6A3BRAINRAT3H-dopaminediethylpropion>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97927SLC6A3BRAINRAT3H-dopaminePhentermine1580Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97928SLC6A3BRAINRAT3H-dopamineMETHAMPHETAMINE (+)114Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97929SLC6A3BRAINRAT3H-dopamineAmphetamine,(+)34Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97930SLC6A4BRAINRAT3H-5HTAmphetamine,(+)3830Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97931SLC6A4BRAINRAT3H-5HTMETHAMPHETAMINE (+)2137Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97932SLC6A4BRAINRAT3H-5HTPhentermine>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97933SLC6A4BRAINRAT3H-5HTdiethylpropion>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97934SLC6A4BRAINRAT3H-5HTN-dealkylated Diethylpropion3840Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97935SLC6A4BRAINRAT3H-5HTPhendimetrazine>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97936SLC6A4BRAINRAT3H-5HTPhendimetrazine-(+)>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97937SLC6A4BRAINRAT3H-5HTPhendimetrazine-(-)>10000Nelson, D. et al., 2006Jan 15, 2025Jan 15, 2025
97938SLC6A3BRAINRAT3H-dopaminePhendimetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97939SLC6A3BRAINRAT3H-dopaminePhenmetrazine607Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97940SLC6A3BRAINRAT3H-dopamine(+)-Phenmetrazine359Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97941SLC6A3BRAINRAT3H-dopamine(-)-Phenmetrazine1669Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97942SLC6A3BRAINRAT3H-dopaminePseudophenmetrazine2630Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97943SLC6A3BRAINRAT3H-dopamine(-)-Pseudophenmetrazine2691Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97944SLC6A3BRAINRAT3H-dopamine(+)-Pseudophenmetrazine3320Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97945NETBRAINRAT3H-Norepinephrine(+)-Pseudophenmetrazine270Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97946NETBRAINRAT3H-Norepinephrine(-)-Pseudophenmetrazine2512Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97947NETBRAINRAT3H-NorepinephrinePseudophenmetrazine453Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97948NETBRAINRAT3H-Norepinephrine(-)-Phenmetrazine388Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97949NETBRAINRAT3H-Norepinephrine(+)-Phenmetrazine240Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97950NETBRAINRAT3H-NorepinephrinePhenmetrazine153Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97951NETBRAINRAT3H-NorepinephrinePhendimetrazine8300Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97952SLC6A4BRAINRAT3H-5HTPhendimetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97953SLC6A4BRAINRAT3H-5HTPhenmetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97954SLC6A4BRAINRAT3H-5HT(+)-Phenmetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97955SLC6A4BRAINRAT3H-5HT(-)-Phenmetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97956SLC6A4BRAINRAT3H-5HTPseudophenmetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97957SLC6A4BRAINRAT3H-5HT(+)-Pseudophenmetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97958SLC6A4BRAINRAT3H-5HT(-)-Pseudophenmetrazine>10000Rothman, R, et al., 2002Jan 15, 2025Jan 15, 2025
97959CGRP1neuroblastomaHUMANFunctionalCGRP 27-373000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97960CGRP1neuroblastomaHUMANFunctional[K35]CGRP 27-372700Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97961CGRP1neuroblastomaHUMANFunctionalCGRP Y0-28-373000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97962CGRP1neuroblastomaHUMANFunctional[K35]CGRP Y0-28-376500Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97963CGRP1neuroblastomaHUMANFunctionalCGRP Ac-27-374500Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97964CGRP1neuroblastomaHUMANFunctionalCGRP Y0-29-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97965CGRP1neuroblastomaHUMANFunctionalCGRP Y0-30-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97966CGRP1neuroblastomaHUMANFunctionalCGRP26-34, ADR50-52>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97967CGRP1neuroblastomaHUMANFunctionalADR40-43, CGRP30-34, ADR50-52>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97968CGRP1neuroblastomaHUMANFunctionalCGRP26-29, ADR44-52>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97969CGRP1neuroblastomaHUMANFunctionalCGRP26-29, ADR44-49, CGRP35-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97970CGRP1neuroblastomaHUMANFunctionalADR40-49, CGRP35-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97971CGRP1neuroblastomaHUMANFunctionalADR40-43, CGRP30-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97972CGRP1neuroblastomaHUMANFunctionalCGRP26-34, IAPP35-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97973CGRP1neuroblastomaHUMANFunctionalIAPP26-34, CGRP30-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97974CGRP1neuroblastomaHUMANFunctional[A27]CGRP 27-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97975CGRP1neuroblastomaHUMANFunctional[A28]CGRP Y0-28-378000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97976CGRP1neuroblastomaHUMANFunctional[A31]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97977CGRP1neuroblastomaHUMANFunctional[A34]CGRP Y0-28-374000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97978CGRP1neuroblastomaHUMANFunctional[A35]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97979CGRP1neuroblastomaHUMANFunctional[F28]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97980CGRP1neuroblastomaHUMANFunctional[F29]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97981CGRP1neuroblastomaHUMANFunctional[F31]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97982CGRP1neuroblastomaHUMANFunctional[F35]CGRP Y0-28-374790Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97983CGRP1neuroblastomaHUMANFunctionalCGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97984CGRP1neuroblastomaHUMANFunctional[v28]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97985CGRP1neuroblastomaHUMANFunctional[p29]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97986CGRP1neuroblastomaHUMANFunctional[n31]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97987CGRP1neuroblastomaHUMANFunctional[s34]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97988CGRP1neuroblastomaHUMANFunctional[a36]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97989CGRP1neuroblastomaHUMANFunctional[Hyp29]CGRP Y0-28-379000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97990CGRP1neuroblastomaHUMANFunctional[S30]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97991CGRP1neuroblastomaHUMANFunctional[L31]CGRP Y0-28-377000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97992CGRP1neuroblastomaHUMANFunctional[Q31]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97993CGRP1neuroblastomaHUMANFunctional[D31]CGRP Y0-28-375000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97994CGRP1neuroblastomaHUMANFunctional[H35]CGRP Y0-28-374275Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97995CGRP1neuroblastomaHUMANFunctional[Q35]CGRP Y0-28-376900Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97996CGRP1neuroblastomaHUMANFunctional[L35]CGRP Y0-28-378550Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97997CGRP1neuroblastomaHUMANFunctional[G36]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97998CGRP1neuroblastomaHUMANFunctional[Y37]CGRP Y0-28-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
97999CGRP1neuroblastomaHUMANFunctional[P28]CGRP 27-373400Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98000CGRP1neuroblastomaHUMANFunctional[P30]CGRP 27-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98001CGRP1neuroblastomaHUMANFunctional[P31]CGRP 27-374500Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98002CGRP1neuroblastomaHUMANFunctional[P32]CGRP 27-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98003CGRP1neuroblastomaHUMANFunctional[P33]CGRP 27-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98004CGRP1neuroblastomaHUMANFunctional[P34]CGRP 27-37280Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98005CGRP1neuroblastomaHUMANFunctional[P35]CGRP 27-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98006CGRP1neuroblastomaHUMANFunctional[P36]CGRP 27-37>10000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98007CGRP1neuroblastomaHUMANFunctional[D31]CGRP 27-373000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98008CGRP1neuroblastomaHUMANFunctional[D31,Q35]CGRP 27-371200Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98009CGRP1neuroblastomaHUMANFunctional[D31,P34]CGRP 27-37470Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98010CGRP1neuroblastomaHUMANFunctional[D31,A34,H35]CGRP 27-37360Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98011CGRP1neuroblastomaHUMANFunctional[D31,A34,F35]CGRP 27-37159Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98012CGRP1neuroblastomaHUMANFunctional[D31,P34,F35]CGRP 27-3729Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98013CGRP1neuroblastomaHUMANFunctional[D31,A34,F35]CGRP Ac-27-37205Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98014CGRP1neuroblastomaHUMANFunctional[D31,A34,F35]CGRP Ac-28-37300Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98015CGRP1neuroblastomaHUMANFunctional[D31,A34,F35]CGRP 28-37200Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98016CGRP1neuroblastomaHUMANFunctional[D31,A34,F35]CGRP Ac-29-37490Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98017CGRP1neuroblastomaHUMANFunctional[D31,A34,F35]CGRP 29-37220Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98018CGRP1neuroblastomaHUMANFunctional[D31,Acp34,F35]CGRP 27-373000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98019CGRP1neuroblastomaHUMANFunctional[D31,Pac34,F35]CGRP 27-373000Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98020CGRP1neuroblastomaHUMANFunctional[D31,Tic34,F35]CGRP 27-37146Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98021CGRP1neuroblastomaHUMANFunctional[D31,Hyp34,F35]CGRP 27-37620Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98022CGRP1neuroblastomaHUMANFunctional[D31,Hop34,F35]CGRP 27-37910Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98023CGRP1neuroblastomaHUMANFunctional[D31,Aib34,F35]CGRP 27-37170Rist, B., et al, 1998Jan 15, 2025Jan 15, 2025
98024SST1CLONEDHUMAN125I-LTT-SRIF28somatostatin-282.7Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98025SST2CLONEDHUMAN125I-LTT-SRIF28somatostatin-282.3Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98026SST3CLONEDHUMAN125I-LTT-SRIF28somatostatin-283.4Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98027SST4CLONEDHUMAN125I-LTT-SRIF28somatostatin-282.7Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98028SST5CLONEDHUMAN125I-LTT-SRIF28somatostatin-282.5Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98029SST5CLONEDHUMAN125I-LTT-SRIF28KE1080.65Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98030SST4CLONEDHUMAN125I-LTT-SRIF28KE1081.6Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98031SST3CLONEDHUMAN125I-LTT-SRIF28KE1081.5Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98032SST2CLONEDHUMAN125I-LTT-SRIF28KE1080.9Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98033SST1CLONEDHUMAN125I-LTT-SRIF28KE1082.6Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98034SST1CLONEDHUMAN125I-LTT-SRIF28KE1196.9Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98035SST2CLONEDHUMAN125I-LTT-SRIF28KE1191.1Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98036SST3CLONEDHUMAN125I-LTT-SRIF28KE1192.5Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98037SST4CLONEDHUMAN125I-LTT-SRIF28KE1193.8Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98038SST5CLONEDHUMAN125I-LTT-SRIF28KE1192.6Reubi JC, et.al.,2002Jan 15, 2025Jan 15, 2025
98039CB1CHO cellsHUMAN3H-CP-55940Otenabant0.7Amato G et al 2019Jan 15, 2025Jan 28, 2025
98040CB2CHO cellsHUMAN3H-CP-55940Otenabant7700Amato G et al 2019Jan 15, 2025Jan 28, 2025
98041CB1CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-phenylpiperidin-4-amine6Amato G et al 2019Jan 15, 2025Jan 28, 2025
98042CB2CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-phenylpiperidin-4-amine>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98043CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pyridin-2-amine2.4Amato G et al 2019Jan 15, 2025Jan 28, 2025
98044CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pyridin-2-amine3100Amato G et al 2019Jan 15, 2025Jan 28, 2025
98045CB1CHO cellsHUMAN3H-CP-55940N-Benzyl-1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-methylpiperidin-4-amine42Amato G et al 2019Jan 15, 2025Jan 28, 2025
98046CB2CHO cellsHUMAN3H-CP-55940N-Benzyl-1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-methylpiperidin-4-amine2700Amato G et al 2019Jan 15, 2025Jan 28, 2025
98047CB1CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime5Amato G et al 2019Jan 15, 2025Jan 28, 2025
98048CB2CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98049CB1CHO cellsHUMAN3H-CP-559401-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl(4-fluorophenyl)methanoneoxime7Amato G et al 2019Jan 15, 2025Jan 28, 2025
98050CB1CHO cellsHUMAN3H-CP-559406-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine47Amato G et al 2019Jan 15, 2025Jan 28, 2025
98051CB2CHO cellsHUMAN3H-CP-559406-[4-(1H-Benzimidazol-2-yl)piperidin-1-yl]-8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purine830Amato G et al 2019Jan 15, 2025Jan 28, 2025
98052CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide780Amato G et al 2019Jan 15, 2025Jan 28, 2025
98053CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzenecarboximidamide6000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98054CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide3Amato G et al 2019Jan 15, 2025Jan 28, 2025
98055CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}pentanamide420Amato G et al 2019Jan 15, 2025Jan 28, 2025
98056CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3-dimethylbutanamide0.2Amato G et al 2019Jan 15, 2025Jan 28, 2025
98057CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3-dimethylbutanamide15Amato G et al 2019Jan 15, 2025Jan 28, 2025
98058CB1CHO cellsHUMAN3H-CP-559403-Tert-butoxy-N-{1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}propanamide6Amato G et al 2019Jan 15, 2025Jan 28, 2025
98059CB2CHO cellsHUMAN3H-CP-559403-Tert-butoxy-N-{1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}propanamide4900Amato G et al 2019Jan 15, 2025Jan 28, 2025
98060CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}tetrahydro-2H-thiopyran-4-carboxamide3Amato G et al 2019Jan 15, 2025Jan 28, 2025
98061CB2CHO cellsHUMAN3H-CP55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}tetrahydro-2H-thiopyran-4-carboxamide1900Amato G et al 2019Jan 15, 2025Jan 28, 2025
98062CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}benzamide8Amato G et al 2019Jan 15, 2025Jan 28, 2025
98063CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}benzamide740Amato G et al 2019Jan 15, 2025Jan 28, 2025
98064CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzamide0.98Amato G et al 2019Jan 15, 2025Jan 28, 2025
98065CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzamide6000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98066CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzamide2Amato G et al 2019Jan 15, 2025Jan 28, 2025
98067CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzamide>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98068CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2,4-difluorobenzamide2Amato G et al 2019Jan 15, 2025Jan 28, 2025
98069CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2,4-difluorobenzamide7000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98070CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzamide3Amato G et al 2019Jan 15, 2025Jan 28, 2025
98071CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzamide5900Amato G et al 2019Jan 15, 2025Jan 28, 2025
98072CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-phenylpropanamide3Amato G et al 2019Jan 15, 2025Jan 28, 2025
98073CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-phenylpropanamide150Amato G et al 2019Jan 15, 2025Jan 28, 2025
98074CB1CHO cellsHUMAN3H-CP-559402-MethoxyethylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate17Amato G et al 2019Jan 15, 2025Jan 28, 2025
98075CB2CHO cellsHUMAN3H-CP-559402-MethoxyethylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate5000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98076CB1CHO cellsHUMAN3H-CP-55940CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate0.6Amato G et al 2019Jan 15, 2025Jan 28, 2025
98077CB2CHO cellsHUMAN3H-CP-55940CyclobutylN-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate1050Amato G et al 2019Jan 15, 2025Jan 28, 2025
98078CB1CHO cellsHUMAN3H-CP-55940Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate4Amato G et al 2019Jan 15, 2025Jan 28, 2025
98079CB2CHO cellsHUMAN3H-CP-55940Benzyl{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}carbamate710Amato G et al 2019Jan 15, 2025Jan 28, 2025
98080CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3,3-trifluoropropane-1-sulfonamide4Amato G et al 2019Jan 15, 2025Jan 28, 2025
98081CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,3,3-trifluoropropane-1-sulfonamide420Amato G et al 2019Jan 15, 2025Jan 28, 2025
98082CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pentylsulfonamide9Amato G et al 2019Jan 15, 2025Jan 28, 2025
98083CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}pentylsulfonamide570Amato G et al 2019Jan 15, 2025Jan 28, 2025
98084CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}cyclohexanesulfonamide9Amato G et al 2019Jan 15, 2025Jan 28, 2025
98085CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}cyclohexanesulfonamide>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98086CB1CHO cellsHUMAN3H-CP-55940N-Cyclohexyl({1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}amino)sulfonamide5Amato G et al 2019Jan 15, 2025Jan 28, 2025
98087CB2CHO cellsHUMAN3H-CP-55940N-Cyclohexyl({1-[8-(2-chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}amino)sulfonamide330Amato G et al 2019Jan 15, 2025Jan 28, 2025
98088CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide0.38Amato G et al 2019Jan 15, 2025Jan 28, 2025
98089CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide8500Amato G et al 2019Jan 15, 2025Jan 28, 2025
98090CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-fluorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide2.6Amato G et al 2019Jan 15, 2025Jan 28, 2025
98091CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-fluorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98092CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide4Amato G et al 2019Jan 15, 2025Jan 28, 2025
98093CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide400Amato G et al 2019Jan 15, 2025Jan 28, 2025
98094CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide1.6Amato G et al 2019Jan 15, 2025Jan 28, 2025
98095CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-2-fluorobenzene-1-sulfonamide190Amato G et al 2019Jan 15, 2025Jan 28, 2025
98096CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzene-1-sulfonamide3.3Amato G et al 2019Jan 15, 2025Jan 28, 2025
98097CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-4-fluorobenzene-1-sulfonamide9000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98098CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2,4-difluorobenzene-1-sulfonamide2Amato G et al 2019Jan 15, 2025Jan 28, 2025
98099CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-2,4-difluorobenzene-1-sulfonamide>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98100CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide1.7Amato G et al 2019Jan 15, 2025Jan 28, 2025
98101CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98102CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide10Amato G et al 2019Jan 15, 2025Jan 28, 2025
98103CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(trifluoromethyl)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide6000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98104CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide3Amato G et al 2019Jan 15, 2025Jan 28, 2025
98105CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-[6-(difluoromethoxy)pyridin-3-yl]-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamide860Amato G et al 2019Jan 15, 2025Jan 28, 2025
98106CB1CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(5-methyl-1,2-oxazol-3-yl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamid420Amato G et al 2019Jan 15, 2025Jan 28, 2025
98107CB2CHO cellsHUMAN3H-CP-55940N-{1-[8-(2-Chlorophenyl)-9-(5-methyl-1,2-oxazol-3-yl)-9H-purin-6-yl]piperidin-4-yl}-3,4-difluorobenzene-1-sulfonamid>10000Amato G et al 2019Jan 15, 2025Jan 28, 2025
98108CB1CLONEDHUMAN[3H]CP55940Otenabant9.7Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98109CB1CLONEDHUMAN[3H]CP559408-(2-chlorophenyl)-9-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)purine 3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98110CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(methylsulfonyl)piperazin-1-yl]-9H-purine24Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98111CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(ethylsulfonyl)piperazin-1-yl]-9H-purine3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98112CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(1-methylethyl)sulfonyl]piperazin-1-yl}-9H-purine1.4Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98113CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclopropylsulfonyl)piperazin-1-yl]-9H-purine5Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98114CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(propylsulfonyl)piperazin-1-yl]-9H-purine1.2Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98115CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(3,3,3-trifluoropropyl)sulfonyl]piperazin-1-yl}-9H-purine1.2Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98116CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(2-methylpropyl)sulfonyl]piperazin-1-yl}-9H-purine2Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98117CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(butylsulfonyl)piperazin-1-yl]-9H-purine0.6Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98118CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(cyclohexylmethyl)sulfonyl]piperazin-1-yl}-9H-purine3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98119CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(tetrahydro-2H-pyran-4-ylmethyl)sulfonyl]piperazin-1-yl}-9H-purine3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98120CB1CLONEDHUMAN[3H]CP55940tert-Butyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate5Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98121CB1CLONEDHUMAN[3H]CP55940Cyclobutyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98122CB1CLONEDHUMAN[3H]CP55940Cyclobutylmethyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98123CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(trifluoroacetyl)piperazin-1-yl]-9H-purine1Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98124CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-(4-pentanoylpiperazin-1-yl)-9H-purine6Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98125CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(ethoxyacetyl)piperazin-1-yl]-9H-purine11Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98126CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(3,3-dimethylbutanoyl)piperazin-1-yl]-9H-purine2Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98127CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(tetrahydro-2H-thiopyran-4-ylcarbonyl)piperazin-1-yl]-9H-purine2Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98128CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2,3-dihydro-1,4-benzodioxin-2-ylcarbonyl)piperazin-1-yl]-9H-purine5Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98129CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclopentylacetyl)piperazin-1-yl]-9H-purine0.4Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98130CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(tetrahydrofuran-3-ylacetyl)piperazin-1-yl]-9H-purine8Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98131CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(piperidin-1-ylacetyl)piperazin-1-yl]-9H-purine21Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98132CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2-phenylpropanoyl)piperazin-1-yl]-9H-purine3Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98133CB1CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(pyrrolidin-1-yl)carbonyl]piperazin-1-yl}-9H-purine13Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98134CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclopentylpiperazine-1-carboxamide5Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98135CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[1-(trifluoromethyl)cyclopentyl]-piperazine-1-carboxamide24Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98136CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclohexylpiperazine-1-carboxamide1.4Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98137CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(cyclohexylmethyl)piperazine-1-carboxamide43Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98138CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-phenylpiperazine-1-carboxamide6Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98139CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(pyridin-2-yl)piperazine-1-carboxamide6Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98140CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2-fluorophenyl)piperazine-1- carboxamide6Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98141CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2,4-difluorophenyl)piperazine-1-carboxamide5Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98142CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(3,4-difluorophenyl)piperazine-1-carboxamide5Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98143CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(4-fluorophenyl)piperazine-1-carboxamide19Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98144CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[6-(difluoromethoxy)pyridin-3-yl]piperazine-1-carboxamide4Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98145CB1CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[(2- fluorobenzene)sulfonyl]piperazine-1-carboxamide250Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98146CB2CLONEDHUMAN[3H]CP55940Otenabant7700Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98147CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(methylsulfonyl)piperazin-1-yl]-9H-purine1700Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98148CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(ethylsulfonyl)piperazin-1-yl]-9H-purine980Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98149CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(1-methylethyl)sulfonyl]piperazin-1-yl}-9H-purine980Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98150CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclopropylsulfonyl)piperazin-1-yl]-9H-purine2300Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98151CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(propylsulfonyl)piperazin-1-yl]-9H-purine850Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98152CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(3,3,3-trifluoropropyl)sulfonyl]piperazin-1-yl}-9H-purine500Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98153CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(2-methylpropyl)sulfonyl]piperazin-1-yl}-9H-purine2800Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98154CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(butylsulfonyl)piperazin-1-yl]-9H-purine500Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98155CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(cyclohexylmethyl)sulfonyl]piperazin-1-yl}-9H-purine91Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98156CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-{4-[(tetrahydro-2H-pyran-4-ylmethyl)sulfonyl]piperazin-1-yl}-9H-purine3000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98157CB2CLONEDHUMAN[3H]CP55940tert-Butyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate3400Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98158CB2CLONEDHUMAN[3H]CP55940Cyclobutyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate3400Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98159CB2CLONEDHUMAN[3H]CP55940Cyclobutylmethyl 4-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]piperazine-1-carboxylate1500Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98160CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(trifluoroacetyl)piperazin-1-yl]-9H-purine130Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98161CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-(4-pentanoylpiperazin-1-yl)-9H-purine400Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98162CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(ethoxyacetyl)piperazin-1-yl]-9H-purine>10000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98163CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(3,3-dimethylbutanoyl)piperazin-1-yl]-9H-purine5000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98164CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(tetrahydro-2H-thiopyran-4-ylcarbonyl)piperazin-1-yl]-9H-purine530Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98165CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2,3-dihydro-1,4-benzodioxin-2-ylcarbonyl)piperazin-1-yl]-9H-purine610Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98166CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(cyclopentylacetyl)piperazin-1-yl]-9H-purine>10000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98167CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(tetrahydrofuran-3-ylacetyl)piperazin-1-yl]-9H-purine3000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98168CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(piperidin-1-ylacetyl)piperazin-1-yl]-9H-purine5000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98169CB2CLONEDHUMAN[3H]CP559408-(2-Chlorophenyl)-9-(4-chlorophenyl)-6-[4-(2-phenylpropanoyl)piperazin-1-yl]-9H-purine560Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98170CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclopentylpiperazine-1-carboxamide740Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98171CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[1-(trifluoromethyl)cyclopentyl]-piperazine-1-carboxamide1300Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98172CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-cyclohexylpiperazine-1-carboxamide620Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98173CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(cyclohexylmethyl)piperazine-1-carboxamide740Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98174CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-phenylpiperazine-1-carboxamide2400Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98175CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(pyridin-2-yl)piperazine-1-carboxamide7100Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98176CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2-fluorophenyl)piperazine-1-carboxamide1300Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98177CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(2,4-difluorophenyl)piperazine-1-carboxamide3200Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98178CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(3,4-difluorophenyl)piperazine-1-carboxamide4200Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98179CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-(4-fluorophenyl)piperazine-1-carboxamide2000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98180CB2CLONEDHUMAN[3H]CP559404-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-N-[6-(difluoromethoxy)pyridin-3-yl]piperazine-1-carboxamide>10000Amato GS et al 2018Jan 15, 2025Jan 28, 2025
98181CLONEDHUMAN125I-HEATQuetiapine22Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98182Alpha2ACLONEDHUMAN125I-ClonidineQuetiapine3630Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98183Alpha2BCLONEDHUMAN125I-ClonidineQuetiapine747Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98184Alpha2CCLONEDHUMAN125I-ClonidineQuetiapine28.7Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98185Alpha2ACLONEDHUMAN125I-ClonidineN-Desalkylquetiapine237Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98186Alpha1ACLONEDHUMAN125I-HEATN-Desalkylquetiapine144Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98187Alpha2BCLONEDHUMAN125I-ClonidineN-Desalkylquetiapine378Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98188Alpha2CCLONEDHUMAN125I-ClonidineN-Desalkylquetiapine736Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981895-HT1ACLONEDHUMAN3H-8-OH-DPATN-Desalkylquetiapine45Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981905-HT1ACLONEDHUMAN3H-8-OH-DPATQuetiapine432Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981915-HT2ACLONEDHUMAN3H-KETANSERINQuetiapine101Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981925-HT2ACLONEDHUMAN3H-KETANSERINN-Desalkylquetiapine48Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981935-HT2CCLONEDHUMAN3H-MESULERGINEN-Desalkylquetiapine107Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981945-HT2CCLONEDHUMAN3H-MESULERGINEQuetiapine2502Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981955-HT6CLONEDHUMAN3H-LSDQuetiapine1865Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981965-HT6CLONEDHUMAN3H-LSDN-Desalkylquetiapine503Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981975-HT7CLONEDHUMAN3H-LSDN-Desalkylquetiapine76Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
981985-HT7CLONEDHUMAN3H-LSDQuetiapine307Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98199mGluR5CLONEDHUMAN3H-domperidoneQuetiapine245Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98200mGluR5CLONEDHUMAN3H-domperidoneN-Desalkylquetiapine196Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98201H1CLONEDHUMAN3H-PYRILAMINEN-Desalkylquetiapine3.5Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98202H1CLONEDHUMAN3H-PYRILAMINEQuetiapine11Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98203M3CLONEDHUMAN3H-QNBQuetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98204M3CLONEDHUMAN3H-QNBN-Desalkylquetiapine23Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98205Alpha1BCLONEDHUMAN125I-HEATN-Desalkylquetiapine95Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
982065-HT1BCLONEDHUMAN3H-GR-125743N-Desalkylquetiapine1117Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
982075-HT1DCLONEDHUMAN3H-GR-125743N-Desalkylquetiapine249Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
982085-HT1ECLONEDHUMAN3H-5HTN-Desalkylquetiapine97Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
982095-HT2BCLONEDHUMAN3H-LSDN-Desalkylquetiapine14Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
982105-HT3CLONEDHUMAN3H-LY 278584N-Desalkylquetiapine394Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98211CB1CLONEDHUMAN3H-LSDN-Desalkylquetiapine768Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98212mGluR5CLONEDHUMAN3H-SCH23390N-Desalkylquetiapine214Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98213D4CLONEDHUMAN3H-NMSPN-Desalkylquetiapine1297Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98214D5CLONEDHUMAN3H-SCH23390N-Desalkylquetiapine1419Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98215KORCLONEDHUMAN3H-MUSCIMOLN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98216H2CLONEDHUMAN3H-CimetidineN-Desalkylquetiapine298Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98217H3CLONEDHUMAN3H-NMSPN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98218H4CLONEDHUMAN3H-NMSPN-Desalkylquetiapine1660Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98219M1CLONEDHUMAN3H-QNBN-Desalkylquetiapine39Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98220M2CLONEDHUMAN3H-QNBN-Desalkylquetiapine453Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98221M4CLONEDHUMAN3H-QNBN-Desalkylquetiapine110Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98222M5CLONEDHUMAN3H-QNBN-Desalkylquetiapine23Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98223NETCLONEDHUMAN3H-NisoxetineN-Desalkylquetiapine58Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98224SERTCLONEDHUMAN3H-CITALOPRAMN-Desalkylquetiapine927Jensen NH, et al., 2008Jan 15, 2025Jan 28, 2025
98225Beta1CLONEDHUMAN125I-IodopindololN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98226Beta2CLONEDHUMAN125I-IodopindololN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 28, 2025
98227nAChRCLONEDHUMAN3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98228CCR5CLONEDHUMAN3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98229nAChRCLONEDHUMAN3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98230nAChRCLONEDHUMAN3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98231nAChRCLONEDHUMAN3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 28, 2025
98232nAChRCLONEDHUMAN3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 27, 2025
98233nAChRCLONEDRAT3H-EpibatidineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98234Sigma 1CLONEDHUMAN3H-Pentazocine(+)N-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98235Sigma 2CLONEDHUMAN3H-DTGN-Desalkylquetiapine1050Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98236SLC6A3CLONEDHUMAN3H-GBR 12935N-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98237DORCLONEDHUMAN3H-DiprenorphineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98238KORCLONEDHUMAN3H-DiprenorphineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98239MORCLONEDHUMAN3H-DiprenorphineN-Desalkylquetiapine>10000Jensen NH, et al., 2008Jan 15, 2025Jan 15, 2025
98240MORBRAINMOUSE3H-DAMGO(E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-3-yl)-N-methylacrylamide0.57Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98241MORBRAINMOUSE3H-DAMGONalfurafine0.431Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98242MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide0.51Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98243MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide0.42Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98244MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide2.7Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98245MORBRAINMOUSE3H-DAMGO(E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide13.9Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98246MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide4.36Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98247MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide12.2Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98248MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide47.6Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98249MORBRAINMOUSE3H-DAMGO(E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide0.232Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98250MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide0.229Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98251MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide0.197Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98252MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide0.28Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98253MORBRAINMOUSE3H-DAMGOE)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide47.9Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98254MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide11.5Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98255MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide59.6Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98256MORBRAINMOUSE3H-DAMGON-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide56Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98257DORBRAINMOUSE3H-DPDPENalfurafine51.3Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98258DORBRAINMOUSE3H-DPDPE(E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-3-yl)-N-methylacrylamide3.98Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98259DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide3.52Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98260DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide1.66Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98261DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide2.23Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98262DORBRAINMOUSE3H-DPDPE(E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide14.2Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98263DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide10.7Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98264DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide4.5Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98265DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide6.46Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98266DORBRAINMOUSE3H-DPDPE(E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide0.182Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98267DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide1.15Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98268DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide1.19Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98269DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide3.65Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98270DORBRAINMOUSE3H-DPDPE(E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide19.1Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98271DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide32.4Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98272DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide15Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98273DORBRAINMOUSE3H-DPDPEN-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide1.27Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98274KORCEREBELLUMGUINEA PIG3H-U69593Nalfurafine0.178Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98275KORCEREBELLUMGUINEA PIG3H-U69593(E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-3-yl)-N-methylacrylamide0.23Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98276KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide0.47Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98277KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide0.24Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98278KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide4.46Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98279KORCEREBELLUMGUINEA PIG3H-U69593(E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide0.82Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98280KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide1.86Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98281KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide1.73Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98282KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,4a,5,6,7,12-hexahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide13.1Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98283KORCEREBELLUMGUINEA PIG3H-U69593(E)-N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide0.204Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98284KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide0.113Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98285KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide0.136Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98286KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14R)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide0.543Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98287KORCEREBELLUMGUINEA PIG3H-U69593(E)-N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9- hydroxy-2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno- [1,2-d]quinolin-14-yl]-3-(furan-2-yl)-N-methylacrylamide8.36Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98288KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-3-phenylpropanamide11.9Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98289KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methyl-2-phenylacetamide11Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98290KORCEREBELLUMGUINEA PIG3H-U69593N-[(2S,4aS,7aR,12aR,14S)-5-(cyclopropylmethyl)-9-hydroxy2,3,4,4a,5,6,7,12-octahydro-1H-2,7a-ethanoindeno[1,2-d]- quinolin-14-yl]-N-methylbenzamide13.8Nakajima R et al 2015Jan 15, 2025Jan 28, 2025
98291H1CLONEDHUMAN[3H]-Pyrilamine2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98292H1CLONEDHUMAN[3H]-Pyrilamine2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline1437Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98293H1CLONEDHUMAN[3H]-Pyrilamine2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide998Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98294H1CLONEDHUMAN[3H]-Pyrilamine1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98295H1CLONEDHUMAN[3H]-Pyrilamine1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione3867Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98296H1CLONEDHUMAN[3H]-Pyrilamine4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one86.3Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98297H1CLONEDHUMAN[3H]-Pyrilamine1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 597Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98298H1CLONEDHUMAN[3H]-Pyrilamine1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98299H1CLONEDHUMAN[3H]-Pyrilamine1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98300H1CLONEDHUMAN[3H]-Pyrilamine1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride3224Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98301H1CLONEDHUMAN[3H]-Pyrilamine1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid1087Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98302H1CLONEDHUMAN[3H]-Pyrilamine5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98303H1CLONEDHUMAN[3H]-Pyrilamine2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride24Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98304H1CLONEDHUMAN[3H]-Pyrilamine5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride553Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98305D2CLONEDHUMAN[3H]-N-methylspiperone2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 167Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98306D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98307D2CLONEDHUMAN[3H]-N-methylspiperone2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole990Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98308D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline915Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98309D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride272Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98310D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride138Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98311D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride853Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98312D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride1087Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98313D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride418Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98314D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98315D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline5647Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98316D2CLONEDHUMAN[3H]-N-methylspiperone2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98317D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98318D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione2933Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98319D2CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one49Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98320D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 126Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98321D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98322D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98323D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride3578Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98324D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid1170Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98325D2CLONEDHUMAN[3H]-N-methylspiperone5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,5399Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98326D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,750Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98327D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride2583.5Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98328D2CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride946Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98329D3CLONEDHUMAN[3H]-N-methylspiperone2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 8.7Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98330D3CLONEDHUMAN[3H]-N-methylspiperone2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide80Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98331D3CLONEDHUMAN[3H]-N-methylspiperone2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole259Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98332D3CLONEDHUMAN[3H]-N-methylspiperone2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline2176Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98333D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride31Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98334D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride447Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98335D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride91Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98336D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride526Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98337D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride1083Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98338D3CLONEDHUMAN[3H]-N-methylspiperone2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline88Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98339D3CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline184Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98340D3CLONEDHUMAN[3H]-N-methylspiperone2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide150Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98341D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride1645Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98342D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98343D3CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one72Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98344D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 17Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98345D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98346D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98347D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride342Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98348D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid106Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98349D3CLONEDHUMAN[3H]-N-methylspiperone5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,66Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98350D3CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,223Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98351D3CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride866Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98352D3CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride783Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98353D4CLONEDHUMAN[3H]-N-methylspiperone2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 67Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98354D4CLONEDHUMAN[3H]-N-methylspiperone2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide41Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98355D4CLONEDHUMAN[3H]-N-methylspiperone2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole141Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98356D4CLONEDHUMAN[3H]-N-methylspiperone2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline127Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98357D4CLONEDHUMAN[3H]-N-methylspiperone2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride129Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98358D4CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride572Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98359D4CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride279Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98360D4CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride37Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98361D4CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride272Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98362D4CLONEDHUMAN[3H]-N-methylspiperone2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline194Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98363D4CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline140Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98364D4CLONEDHUMAN[3H]-N-methylspiperone2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98365D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98366D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98367D4CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one2.3Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98368D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 86Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98369D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98370D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98371D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride442Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98372D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid82Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98373D4CLONEDHUMAN[3H]-N-methylspiperone5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,3335Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98374D4CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,251Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98375D4CLONEDHUMAN[3H]-N-methylspiperone2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride1102Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98376D4CLONEDHUMAN[3H]-N-methylspiperone5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride50Ofon E et al 2016Jan 15, 2025Jan 28, 2025
983775-HT1ACLONEDHUMAN[3H]-Way1006352-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 10Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983785-HT1ACLONEDHUMAN[3H]-Way1006352-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide95Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983795-HT1ACLONEDHUMAN[3H]-Way1006352-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole111Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983805-HT1ACLONEDHUMAN[3H]-Way1006352-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline65Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983815-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride15Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983825-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride42Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983835-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride11Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983845-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride9.9Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983855-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline1109Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983865-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline138Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983875-HT1ACLONEDHUMAN[3H]-Way1006352-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983885-HT1ACLONEDHUMAN[3H]-Way1006351-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983895-HT1ACLONEDHUMAN[3H]-Way1006351-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione339Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983905-HT1ACLONEDHUMAN[3H]-Way1006354-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one19.5Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983915-HT1ACLONEDHUMAN[3H]-Way1006351-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 8.3Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983925-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983935-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983945-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride1712Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983955-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid214Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983965-HT1ACLONEDHUMAN[3H]-Way1006355-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,122Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983975-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,19Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983985-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride48.3Ofon E et al 2016Jan 15, 2025Jan 15, 2025
983995-HT1ACLONEDHUMAN[3H]-Way1006355-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride16Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984005-HT2ACLONEDHUMAN[3H]-ketanserin2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 1681Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984015-HT2ACLONEDHUMAN[3H]-ketanserin2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide2051Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984025-HT2ACLONEDHUMAN[3H]-ketanserin2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984035-HT2ACLONEDHUMAN[3H]-ketanserin2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984045-HT2ACLONEDHUMAN[3H]-ketanserin2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride258Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984055-HT2ACLONEDHUMAN[3H]-ketanserin5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride702Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984065-HT2ACLONEDHUMAN[3H]-ketanserin5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride483Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984075-HT2ACLONEDHUMAN[3H]-ketanserin5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride1144Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984085-HT2ACLONEDHUMAN[3H]-ketanserin5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride667Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984095-HT2ACLONEDHUMAN[3H]-ketanserin2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline1867Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984105-HT2ACLONEDHUMAN[3H]-ketanserin2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline975Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984115-HT2ACLONEDHUMAN[3H]-ketanserin2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984125-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984135-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984145-HT2ACLONEDHUMAN[3H]-ketanserin4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one21Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984155-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one >10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984165-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984175-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984185-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride120Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984195-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid281Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984205-HT2ACLONEDHUMAN[3H]-ketanserin5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,1022Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984215-HT2ACLONEDHUMAN[3H]-ketanserin2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,1204Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984225-HT2ACLONEDHUMAN[3H]-ketanserin2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride391.3Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984235-HT2ACLONEDHUMAN[3H]-ketanserin5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride748Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984245-HT7CLONEDHUMAN[3H]-LSD2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 22Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984255-HT7CLONEDHUMAN[3H]-LSD2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide37Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984265-HT7CLONEDHUMAN[3H]-LSD2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole211Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984275-HT7CLONEDHUMAN[3H]-LSD2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline91Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984285-HT7CLONEDHUMAN[3H]-LSD2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride45Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984295-HT7CLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride25Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984305-HT7CLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride144Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984315-HT7CLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride44Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984325-HT7CLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride67Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984335-HT7CLONEDHUMAN[3H]-LSD2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline132Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984345-HT7CLONEDHUMAN[3H]-LSD2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline65Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984355-HT7CLONEDHUMAN[3H]-LSD2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide497Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984365-HT7CLONEDHUMAN[3H]-LSD1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984375-HT7CLONEDHUMAN[3H]-LSD1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione739Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984385-HT7CLONEDHUMAN[3H]-LSD4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one381Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984395-HT7CLONEDHUMAN[3H]-LSD1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 3.6Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984405-HT7CLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984415-HT7CLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984425-HT7CLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride257Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984435-HT7CLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid138Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984445-HT7CLONEDHUMAN[3H]-LSD5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,127Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984455-HT7CLONEDHUMAN[3H]-LSD2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,1.6Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984465-HT7CLONEDHUMAN[3H]-LSD2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride265Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984475-HT7CLONEDHUMAN[3H]-LSD5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride0.5Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984485-HT2BCLONEDHUMAN[3H]-LSD2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 18Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984495-HT2BCLONEDHUMAN[3H]-LSD2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide18Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984505-HT2BCLONEDHUMAN[3H]-LSD2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole135Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984515-HT2BCLONEDHUMAN[3H]-LSD2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984525-HT2BCLONEDHUMAN[3H]-LSD2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride239Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984535-HT2BCLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride16Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984545-HT2BCLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride327Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984555-HT2BCLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride64Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984565-HT2BCLONEDHUMAN[3H]-LSD5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride7Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984575-HT2BCLONEDHUMAN[3H]-LSD2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline149Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984585-HT2BCLONEDHUMAN[3H]-LSD2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline126Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984595-HT2BCLONEDHUMAN[3H]-LSD2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984605-HT2BCLONEDHUMAN[3H]-LSD1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984615-HT2BCLONEDHUMAN[3H]-LSD1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione531Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984625-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one519Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984635-HT2BCLONEDHUMAN[3H]-LSD1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 232Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984645-HT2BCLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984655-HT2BCLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984665-HT2BCLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride501Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984675-HT2BCLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid549Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984685-HT2BCLONEDHUMAN[3H]-LSD5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,483Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984695-HT2BCLONEDHUMAN[3H]-LSD2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,294Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984705-HT2BCLONEDHUMAN[3H]-LSD2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride391Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984715-HT2BCLONEDHUMAN[3H]-LSD5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride109Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984725-HT2CCLONEDHUMAN[3H]-mesulergine2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 910Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984735-HT2CCLONEDHUMAN[3H]-mesulergine2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide1182Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984745-HT2CCLONEDHUMAN[3H]-mesulergine2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984755-HT2CCLONEDHUMAN[3H]-mesulergine2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984765-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride675Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984775-HT2CCLONEDHUMAN[3H]-mesulergine5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride759Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984785-HT2CCLONEDHUMAN[3H]-mesulergine5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride820Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984795-HT2CCLONEDHUMAN[3H]-mesulergine5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride501Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984805-HT2CCLONEDHUMAN[3H]-mesulergine5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride329Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984815-HT2CCLONEDHUMAN[3H]-mesulergine2-(2-(1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984825-HT2CCLONEDHUMAN[3H]-mesulergine2-(2-(3,4-Dihydronaphthalen-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline2903Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984835-HT2CCLONEDHUMAN[3H]-mesulergine2-(4,4-Bis(4-chlorophenyl)but-3-en-1-yl)-1,2,3,4-tetrahydroisoquinineol hydrobromide2028Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984845-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)-4,4-dimethylpiperidine-2,6-dione hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984855-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-(Isoindolin-2-yl)butyl)-4,4-dimethylpiperidine-2,6-dione305Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984865-HT2CCLONEDHUMAN[3H]-mesulergine4-(3,4-dihydro-1H-isoquinolin-2-yl)-1-(4-fluorophenyl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984875-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-chlorophenyl)-4-(3,4-dihydro-1H-isoquinolin-2-yl)butan-1-one 2976Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984885-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-Chlorophenyl)-4-(3,4-dihydroquinolin-1(2H)-yl)butan-1-one>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984895-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-Chlorophenyl)-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)butan-1-one hydrochloride>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984905-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[c]azepin-2(3H)-yl)butan-1-one hydrochloride348Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984915-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-Chlorophenyl)-4-(4,5-dihydro-1H-benzo[d]azepin-3(2H)-yl)butan-1-one hydrochlorid611Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984925-HT2CCLONEDHUMAN[3H]-mesulergine5-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)indolin-2-one,4234Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984935-HT2CCLONEDHUMAN[3H]-mesulergine2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-5-fluoro-2,3-dihydro-1H-inden-1-one,>10000Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984945-HT2CCLONEDHUMAN[3H]-mesulergine2-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride1184Ofon E et al 2016Jan 15, 2025Jan 15, 2025
984955-HT2CCLONEDHUMAN[3H]-mesulergine5-Chloro-2-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)-2,3-dihydro-1H-inden-1-one hydrochloride128Ofon E et al 2016Jan 15, 2025Jan 15, 2025
98496H1CLONEDHUMAN[3H]-Pyrilamine2-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]-1,3-benzothiazole 583Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98497H1CLONEDHUMAN[3H]-Pyrilamine2-(3-(3,4-Dihydroisoquinolin-2(1H)-yl)propyl)benzo[d]thiazole hydrobromide822Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98498H1CLONEDHUMAN[3H]-Pyrilamine2-[4-(1,3-dihydroisoindol-2-yl)butyl]-1,3-benzothiazole762Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98499H1CLONEDHUMAN[3H]-Pyrilamine2-(3-(1H-benzo[d]imidazol-2-yl)propyl)-1,2,3,4-tetra-hydroisoquinoline290Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98500H1CLONEDHUMAN[3H]-Pyrilamine2-(4-(8-Chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride293Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98501H1CLONEDHUMAN[3H]-Pyrilamine5-Chloro-2-(4-(3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride247Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98502H1CLONEDHUMAN[3H]-Pyrilamine5-Chloro-2-(4-(5-chloro-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride560Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98503H1CLONEDHUMAN[3H]-Pyrilamine5-Chloro-2-(4-(octahydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride268Ofon E et al 2016Jan 15, 2025Jan 28, 2025
98504H1CLONEDHUMAN[3H]-Pyrilamine5-Chloro-2-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)benzo[d]thiazole hydrochloride327Ofon E et al 2016Jan 15, 2025Jan 28, 2025
985055-HT1ACLONEDHUMAN[3H]-Way1006352-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione499Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985065-HT1ACLONEDHUMAN[3H]-Way1006352-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione533Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985075-HT1ACLONEDHUMAN[3H]-Way1006352-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985085-HT1ACLONEDHUMAN[3H]-Way1006352-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline1680Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985095-HT1ACLONEDHUMAN[3H]-Way1006352-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride193Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985105-HT1ACLONEDHUMAN[3H]-Way1006352-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride141Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985115-HT1ACLONEDHUMAN[3H]-Way1006352-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride244Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985125-HT1ACLONEDHUMAN[3H]-Way1006352-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride217Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985135-HT1ACLONEDHUMAN[3H]-Way1006352-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride41Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985145-HT1ACLONEDHUMAN[3H]-Way1006354-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one12Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985155-HT1ACLONEDHUMAN[3H]-Way1006354-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one710Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985165-HT1ACLONEDHUMAN[3H]-Way1006354-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile295Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985175-HT1ACLONEDHUMAN[3H]-Way1006354-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide38Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985185-HT1ACLONEDHUMAN[3H]-Way1006354-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,23Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985195-HT1ACLONEDHUMAN[3H]-Way1006354-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride33.5Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985205-HT1ACLONEDHUMAN[3H]-Way1006351-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride8.2Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985215-HT1ACLONEDHUMAN[3H]-Way100635ARIPIPRAZOLE5.6Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985225-HT2ACLONEDHUMAN[3H]-ketanserin2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985235-HT2ACLONEDHUMAN[3H]-ketanserin2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985245-HT2ACLONEDHUMAN[3H]-ketanserin2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985255-HT2ACLONEDHUMAN[3H]-ketanserin2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline926Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985265-HT2ACLONEDHUMAN[3H]-ketanserin2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride522.5Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985275-HT2ACLONEDHUMAN[3H]-ketanserin2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride726Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985285-HT2ACLONEDHUMAN[3H]-ketanserin2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride322Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985295-HT2ACLONEDHUMAN[3H]-ketanserin2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride317Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985305-HT2ACLONEDHUMAN[3H]-ketanserin2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride1779Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985315-HT2ACLONEDHUMAN[3H]-ketanserin4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one14Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985325-HT2ACLONEDHUMAN[3H]-ketanserin4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one3.9Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985335-HT2ACLONEDHUMAN[3H]-ketanserin4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile23Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985345-HT2ACLONEDHUMAN[3H]-ketanserin4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide404Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985355-HT2ACLONEDHUMAN[3H]-ketanserin4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,2993Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985365-HT2ACLONEDHUMAN[3H]-ketanserin4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride851Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985375-HT2ACLONEDHUMAN[3H]-ketanserin1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985385-HT2ACLONEDHUMAN[3H]-ketanserinARIPIPRAZOLE8.7Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985395-HT7CLONEDHUMAN[3H]-LSD2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione8.6Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985405-HT7CLONEDHUMAN[3H]-LSD2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione330Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985415-HT7CLONEDHUMAN[3H]-LSD2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985425-HT7CLONEDHUMAN[3H]-LSD2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline52Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985435-HT7CLONEDHUMAN[3H]-LSD2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride86Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985445-HT7CLONEDHUMAN[3H]-LSD2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride27Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985455-HT7CLONEDHUMAN[3H]-LSD2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride100Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985465-HT7CLONEDHUMAN[3H]-LSD2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride49Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985475-HT7CLONEDHUMAN[3H]-LSD2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride22.5Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985485-HT7CLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one364Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985495-HT7CLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one358Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985505-HT7CLONEDHUMAN[3H]-LSD4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile755Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985515-HT7CLONEDHUMAN[3H]-LSD4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide12Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985525-HT7CLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,17Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985535-HT7CLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride10Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985545-HT7CLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride3.6Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985555-HT7CLONEDHUMAN[3H]-LSDARIPIPRAZOLE10.3Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985565-HT2BCLONEDHUMAN[3H]-LSD2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985575-HT2BCLONEDHUMAN[3H]-LSD2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione400Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985585-HT2BCLONEDHUMAN[3H]-LSD2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985595-HT2BCLONEDHUMAN[3H]-LSD2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985605-HT2BCLONEDHUMAN[3H]-LSD2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride1247Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985615-HT2BCLONEDHUMAN[3H]-LSD2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride1713Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985625-HT2BCLONEDHUMAN[3H]-LSD2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride561Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985635-HT2BCLONEDHUMAN[3H]-LSD2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride204Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985645-HT2BCLONEDHUMAN[3H]-LSD2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride1166Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985655-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one614Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985665-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one273Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985675-HT2BCLONEDHUMAN[3H]-LSD4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile152Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985685-HT2BCLONEDHUMAN[3H]-LSD4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide587Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985695-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,723Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985705-HT2BCLONEDHUMAN[3H]-LSD4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride358Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985715-HT2BCLONEDHUMAN[3H]-LSD1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride232Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985725-HT2BCLONEDHUMAN[3H]-LSDARIPIPRAZOLE0.36Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985735-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985745-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione37Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985755-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione151Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985765-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985775-HT2CCLONEDHUMAN[3H]-mesulergine2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985785-HT2CCLONEDHUMAN[3H]-mesulergine2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride4440Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985795-HT2CCLONEDHUMAN[3H]-mesulergine2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985805-HT2CCLONEDHUMAN[3H]-mesulergine2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride2623Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985815-HT2CCLONEDHUMAN[3H]-mesulergine2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985825-HT2CCLONEDHUMAN[3H]-mesulergine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985835-HT2CCLONEDHUMAN[3H]-mesulergine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one603Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985845-HT2CCLONEDHUMAN[3H]-mesulergine4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile443Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985855-HT2CCLONEDHUMAN[3H]-mesulergine4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide1892Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985865-HT2CCLONEDHUMAN[3H]-mesulergine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,1404Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985875-HT2CCLONEDHUMAN[3H]-mesulergine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985885-HT2CCLONEDHUMAN[3H]-mesulergine1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride2976Ofon E et al 2016aJan 15, 2025Jan 15, 2025
985895-HT2CCLONEDHUMAN[3H]-mesulergineARIPIPRAZOLE76Ofon E et al 2016aJan 15, 2025Jan 15, 2025
98590D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98591D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98592D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98593D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline170Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98594D2CLONEDHUMAN[3H]-N-methylspiperone2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride1150Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98595D2CLONEDHUMAN[3H]-N-methylspiperone2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride319Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98596D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride166Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98597D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride123Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98598D2CLONEDHUMAN[3H]-N-methylspiperone2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride422Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98599D2CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one49Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98600D2CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one646Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98601D2CLONEDHUMAN[3H]-N-methylspiperone4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile1456Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98602D2CLONEDHUMAN[3H]-N-methylspiperone4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide218Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98603D2CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,249Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98604D2CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride366Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98605D2CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride126Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98606D2CLONEDHUMAN[3H]-N-methylspiperoneARIPIPRAZOLE3.3Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98607D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione491Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98608D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione630Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98609D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98610D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline469Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98611D3CLONEDHUMAN[3H]-N-methylspiperone2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride162Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98612D3CLONEDHUMAN[3H]-N-methylspiperone2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride6007Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98613D3CLONEDHUMAN[3H]-N-methylspiperone2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride769Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98614D3CLONEDHUMAN[3H]-N-methylspiperone2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride118Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98615D3CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one72Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98616D3CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one161Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98617D3CLONEDHUMAN[3H]-N-methylspiperone4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile336Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98618D3CLONEDHUMAN[3H]-N-methylspiperone4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide18Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98619D3CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,38Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98620D3CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride143Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98621D3CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride17Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98622D3CLONEDHUMAN[3H]-N-methylspiperoneARIPIPRAZOLE9.7Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98623D4CLONEDHUMAN[3H]-N-methylspiperone2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione240Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98624D4CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98625D4CLONEDHUMAN[3H]-N-methylspiperone2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione1361Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98626D4CLONEDHUMAN[3H]-N-methylspiperone2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline35Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98627D4CLONEDHUMAN[3H]-N-methylspiperone2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride123Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98628D4CLONEDHUMAN[3H]-N-methylspiperone2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride160Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98629D4CLONEDHUMAN[3H]-N-methylspiperone2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride83Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98630D4CLONEDHUMAN[3H]-N-methylspiperone2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride146Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98631D4CLONEDHUMAN[3H]-N-methylspiperone2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride460Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98632D4CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one2.3Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98633D4CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98634D4CLONEDHUMAN[3H]-N-methylspiperone4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile345Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98635D4CLONEDHUMAN[3H]-N-methylspiperone4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide205Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98636D4CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,210Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98637D4CLONEDHUMAN[3H]-N-methylspiperone4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride773Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98638D4CLONEDHUMAN[3H]-N-methylspiperone1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride86Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98639D4CLONEDHUMAN[3H]-N-methylspiperoneARIPIPRAZOLE510Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98640H1CLONEDHUMAN[3H]-Pyrilamine2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98641H1CLONEDHUMAN[3H]-Pyrilamine2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione3632Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98642H1CLONEDHUMAN[3H]-Pyrilamine2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98643H1CLONEDHUMAN[3H]-Pyrilamine2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline836Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98644H1CLONEDHUMAN[3H]-Pyrilamine2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride738Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98645H1CLONEDHUMAN[3H]-Pyrilamine2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride382Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98646H1CLONEDHUMAN[3H]-Pyrilamine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one86.3Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98647H1CLONEDHUMAN[3H]-Pyrilamine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one68Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98648H1CLONEDHUMAN[3H]-Pyrilamine4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile177Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98649H1CLONEDHUMAN[3H]-Pyrilamine4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide1427Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98650H1CLONEDHUMAN[3H]-Pyrilamine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,216Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98651H1CLONEDHUMAN[3H]-Pyrilamine4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98652H1CLONEDHUMAN[3H]-Pyrilamine1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride597Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98653H1CLONEDHUMAN[3H]-PyrilamineARIPIPRAZOLE25.1Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98654SERTCLONEDHUMAN[3H]Citalopram2-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98655SERTCLONEDHUMAN[3H]Citalopram2-(4-(Octahydroisoquinolin-2(1H)-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98656SERTCLONEDHUMAN[3H]Citalopram2-(4-(Isoindolin-2-yl)butyl)isoindoline-1,3-dione>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98657SERTCLONEDHUMAN[3H]Citalopram2-(4-(1H-Indol-3-yl)butyl)-1,2,3,4-tetrahydroisoquinoline113Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98658SERTCLONEDHUMAN[3H]Citalopram2-(2-(5-Fluoro-2,3-dihydro-1H-inden-2-yl)ethyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride163Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98659SERTCLONEDHUMAN[3H]Citalopram2-(4-(4-Fluorophenyl)butyl)-1,2,3,4-tetrahydroisoquinolinehydrochloride4284Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98660SERTCLONEDHUMAN[3H]Citalopram2-(3-(4-Fluorophenoxy)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98661SERTCLONEDHUMAN[3H]Citalopram2-(3-((4-Fluorophenyl)thio)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98662SERTCLONEDHUMAN[3H]Citalopram2-(3-((4-Fluorophenyl)sulfinyl)propyl)-1,2,3,4-tetrahydroisoquinoline hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98663SERTCLONEDHUMAN[3H]Citalopram4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-fluorophenyl)butan-1-one>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98664SERTCLONEDHUMAN[3H]Citalopram4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-phenylbutan-1-one1534Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98665SERTCLONEDHUMAN[3H]Citalopram4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzonitrile895Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98666SERTCLONEDHUMAN[3H]Citalopram4-(4-(3,4-Dihydroisoquinolin-2(1H)-yl)butanoyl)benzamide>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98667SERTCLONEDHUMAN[3H]Citalopram4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-methoxyphenyl)butan-1-one hydrochloride,2442Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98668SERTCLONEDHUMAN[3H]Citalopram4-(3,4-Dihydroisoquinolin-2(1H)-yl)-1-(4-hydroxyphenyl)butan-1-one hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98669SERTCLONEDHUMAN[3H]Citalopram1-(4-Chlorophenyl)-4-(3,4-dihydroisoquinolin-2(1H)-yl)butan-1-one hydrochloride>10000Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98670SERTCLONEDHUMAN[3H]CitalopramARIPIPRAZOLE1080Ofon E et al 2016aJan 15, 2025Jan 28, 2025
98671D3CLONEDHUMAN125I-IABN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane12Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98672D2CLONEDHUMAN125I-IABN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98673D2CLONEDHUMAN125I-IABN4-(5-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)-N,N-dimethylaniline>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98674D3CLONEDHUMAN125I-IABN4-(5-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)-N,N-dimethylaniline138Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98675D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-(2-methoxyphenyl)-4-methyl-4H1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane63Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98676D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-(2-methoxyphenyl)-4-methyl-4H1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane2112Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98677D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-(pyridin-3-yl)-4H-1,2,4- triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane213Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98678D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-(pyridin-3-yl)-4H-1,2,4- triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98679D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-(4-(thiophen-3-yl)- phenyl)-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]- undecane101Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98680D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-(4-(thiophen-3-yl)- phenyl)-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]- undecane3250Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98681D2CLONEDHUMAN125I-IABN2-(4-(5-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3- yl)propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)phenyl)oxazole1574Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98682D3CLONEDHUMAN125I-IABN2-(4-(5-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3- yl)propyl)thio)-4-methyl-4H-1,2,4-triazol-3-yl)phenyl)oxazole25.4Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98683D3CLONEDHUMAN125I-IABN3-(3-((5-(2-Fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane25.9Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98684D2CLONEDHUMAN125I-IABN3-(3-((5-(2-Fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98685D2CLONEDHUMAN125I-IABN3-(3-((5-(4-Fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98686D3CLONEDHUMAN125I-IABN3-(3-((5-(4-Fluorophenyl)-4-methyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane39.8Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98687D3CLONEDHUMAN125I-IABN3-(3-((5-Cyclohexyl-4-methyl-4H-1,2,4-triazol-3-yl)thio)propyl)- 9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane57Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98688D2CLONEDHUMAN125I-IABN3-(3-((5-Cyclohexyl-4-methyl-4H-1,2,4-triazol-3-yl)thio)propyl)- 9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98689D3CLONEDHUMAN125I-IABN3-(3-((4-Ethyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-9-(2- methoxyphenyl)-3,9-diazaspiro[5.5]undecane48.7Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98690D2CLONEDHUMAN125I-IABN3-(3-((4-Ethyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-9-(2- methoxyphenyl)-3,9-diazaspiro[5.5]undecane5650Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98691D2CLONEDHUMAN125I-IABN3-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propyl)thio)-5-phenyl-4H-1,2,4-triazol-4-amine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98692D3CLONEDHUMAN125I-IABN3-((3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propyl)thio)-5-phenyl-4H-1,2,4-triazol-4-amine75Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98693D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane32Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98694D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane1162Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98695D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-phenyl-1H-imidazol-2-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane5891Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98696D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-phenyl-1H-imidazol-2-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane383Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98697D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((1-methyl-5-phenyl-1H-imidazol-2- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane418Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98698D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((1-methyl-5-phenyl-1H-imidazol-2- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98699D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(2-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)ethyl)-3,9-diazaspiro[5.5]undecane9004Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98700D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(2-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)ethyl)-3,9-diazaspiro[5.5]undecane89.7Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98701D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(4-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)butyl)-3,9-diazaspiro[5.5]undecane59.2Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98702D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(4-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)butyl)-3,9-diazaspiro[5.5]undecane9248Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98703D2CLONEDHUMAN125I-IABN3-(2-Ethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane5165Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98704D3CLONEDHUMAN125I-IABN3-(2-Ethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane45.1Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98705D3CLONEDHUMAN125I-IABN2-(9-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- 3,9-diazaspiro[5.5]undecan-3-yl)phenol396Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98706D2CLONEDHUMAN125I-IABN2-(9-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- 3,9-diazaspiro[5.5]undecan-3-yl)phenol>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98707D2CLONEDHUMAN125I-IABN3-(2-(2-Fluoroethoxy)phenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4- triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane6379Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98708D3CLONEDHUMAN125I-IABN3-(2-(2-Fluoroethoxy)phenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4- triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane33.3Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98709D3CLONEDHUMAN125I-IABN3-(4-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane97.7Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98710D2CLONEDHUMAN125I-IABN3-(4-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98711D2CLONEDHUMAN125I-IABN3-(2,4-Dimethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98712D2CLONEDHUMAN125I-IABN3-(2,4-Dimethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane112Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98713D2CLONEDHUMAN125I-IABN3-(4-fluorophenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane9792Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98714D3CLONEDHUMAN125I-IABN3-(4-fluorophenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane25.6Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98715D3CLONEDHUMAN125I-IABN3-(2-Fluorophenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane208Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98716D2CLONEDHUMAN125I-IABN3-(2-Fluorophenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3- yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98717D2CLONEDHUMAN125I-IABN3-(2-Fluoro-4-(trifluoromethyl)phenyl)-9-(3-((4-methyl-5-phenyl4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98718D3CLONEDHUMAN125I-IABN3-(2-Fluoro-4-(trifluoromethyl)phenyl)-9-(3-((4-methyl-5-phenyl4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane370Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98719D3CLONEDHUMAN125I-IABN3-(4-Fluoro-2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane21Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98720D2CLONEDHUMAN125I-IABN3-(4-Fluoro-2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98721D2CLONEDHUMAN125I-IABN1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine260Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98722D3CLONEDHUMAN125I-IABN1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine6.5Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98723D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)propyl)-3,9-diazaspiro[5.5]undec-1-ene3.2Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98724D2CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)propyl)-3,9-diazaspiro[5.5]undec-1-ene197Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98725D2CLONEDHUMAN125I-IABN2-(2-methoxyphenyl)-8-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-2,8-diazaspiro[4.5]decane6168Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98726D3CLONEDHUMAN125I-IABN2-(2-methoxyphenyl)-8-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-2,8-diazaspiro[4.5]decane19.6Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98727D3CLONEDHUMAN125I-IABN8-(2-Methoxyphenyl)-2-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)propyl)-2,8-diazaspiro[4.5]decane27.8Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98728D2CLONEDHUMAN125I-IABN8-(2-Methoxyphenyl)-2-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol3-yl)thio)propyl)-2,8-diazaspiro[4.5]decane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98729D2CLONEDHUMAN125I-IABNN-(4-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- butyl)-4-(thiophen-3-yl)benzamide2766Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98730D3CLONEDHUMAN125I-IABNN-(4-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- butyl)-4-(thiophen-3-yl)benzamide92.9Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98731D3CLONEDHUMAN125I-IABN4-(Dimethylamino)-N-(4-(9-(2-methoxyphenyl)-3,9-diazaspiro- [5.5]undecan-3-yl)butyl)benzamide61.5Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98732D2CLONEDHUMAN125I-IABN4-(Dimethylamino)-N-(4-(9-(2-methoxyphenyl)-3,9-diazaspiro- [5.5]undecan-3-yl)butyl)benzamide3762Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98733D2CLONEDHUMAN125I-IABN7-(3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propoxy)-3,4-dihydroquinolin-2(1H)-one2630Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98734D3CLONEDHUMAN125I-IABN7-(3-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- propoxy)-3,4-dihydroquinolin-2(1H)-one>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98735D3CLONEDHUMAN125I-IABN2-(4-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- butyl)isoindoline-1,3-dione>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98736D2CLONEDHUMAN125I-IABN2-(4-(9-(2-Methoxyphenyl)-3,9-diazaspiro[5.5]undecan-3-yl)- butyl)isoindoline-1,3-dione>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98737D2CLONEDHUMAN125I-IABN3-Butyl-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98738D3CLONEDHUMAN125I-IABN3-Butyl-9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undecane2773Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98739D3CLONEDHUMAN125I-IABN8-Butyl-2-(2-methoxyphenyl)-2,8-diazaspiro[4.5]decane6647Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98740D2CLONEDHUMAN125I-IABN8-Butyl-2-(2-methoxyphenyl)-2,8-diazaspiro[4.5]decane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98741D2CLONEDHUMAN125I-IABN2-Butyl-7-(2-methoxyphenyl)-2,7-diazaspiro[4.4]nonane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98742D3CLONEDHUMAN125I-IABN2-Butyl-7-(2-methoxyphenyl)-2,7-diazaspiro[4.4]nonane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98743D2CLONEDHUMAN125I-IABN1-Butyl-4-(2-methoxyphenyl)piperazine20.6Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98744D3CLONEDHUMAN125I-IABN1-Butyl-4-(2-methoxyphenyl)piperazine23.9Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98745D3CLONEDHUMAN125I-IABN1-Butyl-4-(2-(2-fluoroethoxy)phenyl)piperazine14.7Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98746D2CLONEDHUMAN125I-IABN1-Butyl-4-(2-(2-fluoroethoxy)phenyl)piperazine22.3Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98747D2CLONEDHUMAN125I-IABN4-Methyl-3-phenyl-5-(propylthio)-4H-1,2,4-triazole>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98748D3CLONEDHUMAN125I-IABN4-Methyl-3-phenyl-5-(propylthio)-4H-1,2,4-triazole>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025