47615 ADK recombinant HUMAN Functional 4-N-Benzylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 30 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47616 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47617 ADK recombinant HUMAN Functional 4-N-(4-Methoxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 6 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47618 ADK recombinant HUMAN Functional 4-N-(4-Hydroxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47619 ADK recombinant HUMAN Functional 4-N-Cyclohexylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 250 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47620 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 0.8 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47621 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-(4-fluorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine  26 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47622 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.2 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47623 ADK recombinant HUMAN Functional 4-N-(4-Chlorophenyl)amino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2.7 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47624 ADK recombinant HUMAN Functional 4-N-(4-Cyanophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 14 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47625 ADK recombinant HUMAN Functional 4-N-(4-Cyanophenyl)amino-5-(4-methoxyphenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47626 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 3.6 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47627 ADK recombinant HUMAN Functional 4-N-(4-Methoxyphenyl)amino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 9 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47628 ADK recombinant HUMAN Functional 4-N-(3-Pyridyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 25 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47629 ADK recombinant HUMAN Functional 4-N-(4-Chlorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2.3 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47630 ADK recombinant HUMAN Functional 4-N-(4-Methylphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47631 ADK recombinant HUMAN Functional 2-Methyl-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 47 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47632 ADK recombinant HUMAN Functional 6-Bromo-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47633 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(5-azido-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47634 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(5-amino-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 6.3 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47635 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(2-deoxy-beta-D-erythropentofuranosyl)pyrrolo[2,3-d]pyrimidine 300 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47636 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(2,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 100 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47637 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(3,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 44 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025  
47638 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 13 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47639 GABAA CLONED HUMAN 3H-RO-15-1788 NS-2710 2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47640 GABAA CLONED HUMAN 3H-RO-15-1788 7-trifluoromethyl-3-(2'-cyano-2,4'-difluorobiphenyl-5-yl) analogue 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47641 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1-hydroxy-1-methylethyl)-3-[4-fluoro-3-(pyridine-3-yl)phenyl derivative  0.85 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47642 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(7-Methyl-imidazo[1,2-b]pyridazin-3-yl)-biphenyl-2-carbonitrile 13 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47643 GABAA CLONED HUMAN 3H-RO-15-1788 7-Methyl-3-[3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]imidazo-[1,2-a]pyridine 0.4 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47644 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 1.5 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47645 GABAA CLONED HUMAN 3H-RO-15-1788 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.25 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47646 GABAA CLONED HUMAN 3H-RO-15-1788 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47647 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.73 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47648 GABAA CLONED HUMAN 3H-RO-15-1788 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.15 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47649 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 33 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47650 GABAA CLONED HUMAN 3H-RO-15-1788 NS-2710 14 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47651 GABAA CLONED HUMAN 3H-RO-15-1788 7-trifluoromethyl-3-(2'-cyano-2,4'-difluorobiphenyl-5-yl) analogue 0.73 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47652 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1-hydroxy-1-methylethyl)-3-[4-fluoro-3-(pyridine-3-yl)phenyl derivative  4 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47653 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(7-Methyl-imidazo[1,2-b]pyridazin-3-yl)-biphenyl-2-carbonitrile 19 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47654 GABAA CLONED HUMAN 3H-RO-15-1788 7-Methyl-3-[3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]imidazo-[1,2-a]pyridine 0.4 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47655 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47656 GABAA CLONED HUMAN 3H-RO-15-1788 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.8 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47657 GABAA CLONED HUMAN 3H-RO-15-1788 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 2.1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47658 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 1.8 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47659 GABAA CLONED HUMAN 3H-RO-15-1788 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47660 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47661 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 1.1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025  
47662 OT CLONED HUMAN 3H-Oxytocin (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 28 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47663 OT CLONED HEK293 3H-Oxytocin (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 17 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47664 V1A CLONED HUMAN 3H-AVP (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 170 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47665 V1B CLONED HUMAN 3H-AVP (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide >10000 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47666 V2 CLONED HUMAN 3H-AVP (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide >10000 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47667 OT CLONED RAT 3H-Oxytocin (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 135 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47668 OT CLONED HUMAN 3H-Oxytocin Atosiban 81 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47669 OT CLONED HEK293 3H-Oxytocin Atosiban 27 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47670 V1A CLONED HUMAN 3H-AVP Atosiban 3.5 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47671 V1B CLONED HUMAN 3H-AVP Atosiban 657 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47672 V2 CLONED HUMAN 3H-AVP Atosiban 954 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47673 OT CLONED RAT 3H-Oxytocin Atosiban 76 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47674 OT CLONED HUMAN 3H-Oxytocin Oxytocin 0.5 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47675 OT CLONED HEK293 3H-Oxytocin Oxytocin 0.71 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47676 V1A CLONED HUMAN 3H-AVP Oxytocin 123 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47677 V1B CLONED HUMAN 3H-AVP Oxytocin 1782 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47678 V2 CLONED HUMAN 3H-AVP Oxytocin 1544 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47679 OT CLONED RAT 3H-Oxytocin Oxytocin 1.9 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47680 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE PAROXETINE 0.019 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47681 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE SERTRALINE 0.047 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47682 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Indatraline 0.13 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47683 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE CLOMIPRAMINE 0.14 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47684 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE CITALOPRAM 0.65 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47685 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE FLUOXETINE 1.96 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47686 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Desmethylsertraline 2.29 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47687 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE NORFLUOXETINE 3.15 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47688 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE IMIPRAMINE 14.2 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47689 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE AMITRIPTYLINE 17.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47690 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Dothiepin 31.3 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47691 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Zimeldine 67.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47692 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE NORTRYPTYLINE 60.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47693 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE DOXEPIN 126 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47694 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE northiaden 130 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47695 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE DESIPRAMINE 152 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47696 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE AMOXAPINE 290 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47697 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Fenfluramine (+) 855 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47698 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Fenfluramine (-) 2784 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47699 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE sibutramine 2135 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47700 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake PAROXETINE 0.48 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47701 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake SERTRALINE 2.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47702 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Indatraline 1.5 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47703 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake CLOMIPRAMINE 5.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47704 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake CITALOPRAM 3.51 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47705 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake FLUOXETINE 10.9 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47706 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Desmethylsertraline 53.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47707 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake NORFLUOXETINE 13.9 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47708 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Fluvoxamine 3.57 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47709 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake AMITRIPTYLINE 48.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47710 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake BTS 54 505 26.2 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47711 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake BTS 54 354 18.2 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47712 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Dothiepin 77.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47713 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Zimeldine 56.7 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47714 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake NORTRYPTYLINE 197 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47715 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake DOXEPIN 201 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47716 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake northiaden 192 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47717 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake DESIPRAMINE 200 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47718 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake AMOXAPINE 409 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47719 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Fenfluramine (+) 279 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47720 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Fenfluramine (-) 809 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47721 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake sibutramine 3131 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47722 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Fluvoxamine 4.17 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47723 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE BTS 54 505 18 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47724 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE BTS 54 354 19.3 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47725 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake IMIPRAMINE 30.9 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025  
47726 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY, porcine 0.043 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47727 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY, porcine 0.048 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47728 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY, zebrafish 0.066 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47729 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY, zebrafish 0.11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47730 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.035 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47731 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY,[leu31,Pro34], human 0.035 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47732 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY2-36, porcine 0.26 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47733 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY 3-36, porcine 2 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47734 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY18-36 260 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47735 Y1 CLONED GUINEA PIG [125I] - Peptide YY PP, guinea pig 3.2 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47736 Y1 CLONED GUINEA PIG [125I] - Peptide YY SR 120819A 0.8 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47737 Y1 CLONED GUINEA PIG [125I] - Peptide YY BIBP3226 4.9 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47738 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY 28-36, [P30, Y32, L34] 2.4 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47739 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY D-Trp32, porcine 1000 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47740 Y1 CLONED RAT [125I] - Peptide YY NPY, porcine 0.06 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47741 Y1 CLONED RAT [125I] - Peptide YY PYY, porcine 0.13 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47742 Y1 CLONED RAT [125I] - Peptide YY NPY, zebrafish 0.1 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47743 Y1 CLONED RAT [125I] - Peptide YY PYY, zebrafish 0.18 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47744 Y1 CLONED RAT [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.061 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47745 Y1 CLONED RAT [125I] - Peptide YY PYY,[leu31,Pro34], human 0.11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47746 Y1 CLONED RAT [125I] - Peptide YY NPY2-36, porcine 0.38 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47747 Y1 CLONED RAT [125I] - Peptide YY NPY 3-36, porcine 4.1 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47748 Y1 CLONED RAT [125I] - Peptide YY NPY18-36 100 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47749 Y1 CLONED RAT [125I] - Peptide YY PP, guinea pig 11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47750 Y1 CLONED RAT [125I] - Peptide YY SR 120819A 1.3 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47751 Y1 CLONED RAT [125I] - Peptide YY BIBP3226 3.2 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47752 Y1 CLONED RAT [125I] - Peptide YY NPY 28-36, [P30, Y32, L34] 1.4 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47753 Y1 CLONED RAT [125I] - Peptide YY NPY D-Trp32, porcine 1000 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025  
47754 CEREBRAL CORTEX RAT Functional Val-D-Pro-NHBu >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47755 CEREBRAL CORTEX RAT Functional L-Valyl-L-Proline hexylamide hydrogen oxalate 900 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47756 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline benzylamide hydrogen oxalate 3300 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47757 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline cyclohexylmethylamide hydrogen oxalate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47758 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline-N- β-naphthylamide trifluroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47759 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline piperidinylamide hydrogen oxalate hemihydrate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47760 CEREBRAL CORTEX RAT Functional L-Valyl-L-prolinamide trifluoroacetate 6000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47761 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-prolinamide trifluoroacetate hemihydrate 570 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47762 CEREBRAL CORTEX RAT Functional L-Norvalyl-L-prolinamide trifluoroacetate hemihydrate 1600 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47763 CEREBRAL CORTEX RAT Functional L-Norleucyl-L-prolinamide hydrogen oxalate hemihydrate 2000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47764 CEREBRAL CORTEX RAT Functional L-Leucyl-L-prolinamide trifluoroacetate 2100 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47765 CEREBRAL CORTEX RAT Functional L-Isoleucyl-L-prolinamide trifluoroacetate 4300 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47766 CEREBRAL CORTEX RAT Functional L-Phenylalanyl-L-prolinamide trifluoroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47767 CEREBRAL CORTEX RAT Functional α-Methylalanyl-L-proline butylamide hydrochloride hemihydrate 5000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47768 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline n-propylamide trifluoroacetate 80 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47769 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline n-butylamide hydrogen oxalate 80 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47770 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline n-pentylamide hydrogen oxalate 270 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47771 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline isobutylamide trifluoroacetate 320 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47772 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline (R)-sec-butylamide hydrogen oxalate 4500 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47773 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline-(2S)-methylbutylamide hydrogen oxalate hemihydrate 500 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47774 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline 3-methylthiopropylamide hydrogen oxalate hemihydrate 300 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47775 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-azetidine carboxamide trifluoroacetate hydrate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47776 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(R)-pipecolinic acid amide trifluoroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47777 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-pipecolinic acid n-butylamide trifluoroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47778 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(S)-nipecotamide hydrogen oxalate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47779 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-4-thia-L-prolinamide trifluoroacetate hemihydrate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47780 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(4S)-fluoro-L-proline n-Butylamide Trifluoroacetate 320 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47781 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-4-cis-benzyl-L-proline n-butylamide Hydrogen Oxalate 140 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47782 CEREBRAL CORTEX RAT Functional butabindide 7 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47783 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-indoline carboxylic acid methylamide hydrogen oxalate hydrate 340 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47784 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-indoline carboxylic acid ethylamide hydrogen oxalate hydrate 12 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47785 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-indoline carboxylic acid propylamide hydrogen oxalate hydrate 6 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025  
47786 MOR CLONED HUMAN 3H-DAMGO Enadoline 22 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47787 MOR CLONED HUMAN 3H-DAMGO Cyclorphan 0.062 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47788 MOR CLONED HUMAN 3H-DAMGO MCL-101 0.23 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47789 MOR CLONED HUMAN 3H-DAMGO Levorphanol 0.21 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47790 MOR CLONED HUMAN 3H-DAMGO MCL-133 48 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47791 MOR CLONED HUMAN 3H-DAMGO MCL-134 52 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47792 MOR CLONED HUMAN 3H-DAMGO MCL-153 29 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47793 MOR CLONED HUMAN 3H-DAMGO MCL-154 66 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47794 MOR CLONED HUMAN 3H-DAMGO MCL-135 0.14 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47795 MOR CLONED HUMAN 3H-DAMGO MCL-136 0.93 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47796 MOR CLONED HUMAN 3H-DAMGO MCL-176 0.23 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47797 MOR CLONED HUMAN 3H-DAMGO MCL-139 0.16 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47798 MOR CLONED HUMAN 3H-DAMGO MCL-140 3.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47799 MOR CLONED HUMAN 3H-DAMGO MCL-177 0.89 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47800 MOR CLONED HUMAN 3H-DAMGO MCL-179 0.97 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47801 MOR CLONED HUMAN 3H-DAMGO MCL-144 0.09 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47802 MOR CLONED HUMAN 3H-DAMGO MCL-178 1.8 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47803 MOR CLONED HUMAN 3H-DAMGO MCL-145 0.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47804 MOR CLONED HUMAN 3H-DAMGO MCL-141 4.7 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47805 MOR CLONED HUMAN 3H-DAMGO MCL-142 3.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47806 MOR CLONED HUMAN 3H-DAMGO MCL-143 0.28 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47807 DOR CLONED HUMAN 3H-Naltrindole Enadoline 1000 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47808 DOR CLONED HUMAN 3H-Naltrindole Cyclorphan 1.9 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47809 DOR CLONED HUMAN 3H-Naltrindole MCL-101 5.9 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47810 DOR CLONED HUMAN 3H-Naltrindole Levorphanol 4.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47811 DOR CLONED HUMAN 3H-Naltrindole MCL-133 600 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47812 DOR CLONED HUMAN 3H-Naltrindole MCL-134 370 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47813 DOR CLONED HUMAN 3H-Naltrindole MCL-153 730 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47814 DOR CLONED HUMAN 3H-Naltrindole MCL-154 2500 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47815 DOR CLONED HUMAN 3H-Naltrindole MCL-135 3.8 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47816 DOR CLONED HUMAN 3H-Naltrindole MCL-136 32 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47817 DOR CLONED HUMAN 3H-Naltrindole MCL-176 44 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47818 DOR CLONED HUMAN 3H-Naltrindole MCL-139 9.4 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47819 DOR CLONED HUMAN 3H-Naltrindole MCL-140 80 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47820 DOR CLONED HUMAN 3H-Naltrindole MCL-177 24 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47821 DOR CLONED HUMAN 3H-Naltrindole MCL-179 21 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47822 DOR CLONED HUMAN 3H-Naltrindole MCL-144 4.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47823 DOR CLONED HUMAN 3H-Naltrindole MCL-178 82 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47824 DOR CLONED HUMAN 3H-Naltrindole MCL-145 9.4 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47825 DOR CLONED HUMAN 3H-Naltrindole MCL-141 400 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47826 DOR CLONED HUMAN 3H-Naltrindole MCL-142 920 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47827 DOR CLONED HUMAN 3H-Naltrindole MCL-143 16 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47828 KOR CLONED HUMAN 3H-U69,593 Enadoline 0.27 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47829 KOR CLONED HUMAN 3H-U69,593 Cyclorphan 0.034 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47830 KOR CLONED HUMAN 3H-U69,593 MCL-101 0.079 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47831 KOR CLONED HUMAN 3H-U69,593 Levorphanol 2.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47832 KOR CLONED HUMAN 3H-U69,593 MCL-133 24 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47833 KOR CLONED HUMAN 3H-U69,593 MCL-134 50 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47834 KOR CLONED HUMAN 3H-U69,593 MCL-153 18 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47835 KOR CLONED HUMAN 3H-U69,593 MCL-154 120 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47836 KOR CLONED HUMAN 3H-U69,593 MCL-135 0.1 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47837 KOR CLONED HUMAN 3H-U69,593 MCL-136 0.41 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47838 KOR CLONED HUMAN 3H-U69,593 MCL-176 0.07 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47839 KOR CLONED HUMAN 3H-U69,593 MCL-139 0.076 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47840 KOR CLONED HUMAN 3H-U69,593 MCL-140 1.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47841 KOR CLONED HUMAN 3H-U69,593 MCL-177 0.65 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47842 KOR CLONED HUMAN 3H-U69,593 MCL-179 0.59 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47843 KOR CLONED HUMAN 3H-U69,593 MCL-144 0.049 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47844 KOR CLONED HUMAN 3H-U69,593 MCL-178 1.1 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47845 KOR CLONED HUMAN 3H-U69,593 MCL-145 0.078 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47846 KOR CLONED HUMAN 3H-U69,593 MCL-141 4.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47847 KOR CLONED HUMAN 3H-U69,593 MCL-142 3.4 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47848 KOR CLONED HUMAN 3H-U69,593 MCL-143 0.17 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47849 BRAIN RAT 3H-MK912 MCL-202 3000 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025  
47850 CLONED HUMAN 1251-CGRP h-alpha-CGRP 8-37 1.3 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47851 CLONED HUMAN 1251-CGRP h-alpha-CGRP 0.18 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47852 CLONED HUMAN 1251-CGRP [D31,p34,F35]-h-alpha-CGRP 27-37 14 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47853 CLONED HUMAN 1251-CGRP [D31,Tic34,F35]-h-alpha-CGRP 27-37 70.5 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47854 CLONED HUMAN 1251-CGRP [D31,A34,F35]-h-alpha-CGRP 27-37 76.8 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47855 CLONED HUMAN 3H-CGRP 8-37 [propionyl-K24]-h-alpha-CGRP 8-37 0.6 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47856 CLONED HUMAN 3H-CGRP 8-37 h-alpha-CGRP 8-37 0.06 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47857 CLONED HUMAN 3H-CGRP 8-37 h-alpha-CGRP 0.29 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47858 CLONED HUMAN 3H-CGRP 8-37 [D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47859 CLONED HUMAN 3H-CGRP 8-37 [D31,Tic34,F35]-h-alpha-CGRP 27-37 1.8 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47860 CLONED HUMAN 3H-CGRP 8-37 [D31,A34,F35]-h-alpha-CGRP 27-37 13.6 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47861 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 h-alpha-CGRP 0.29 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47862 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 h-alpha-CGRP  (reduced) 10.2 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47863 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47864 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47865 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47866 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47867 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34,F35]-h-alpha-CGRP 8-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47868 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 (1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47869 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1S,2S,3S)-beta-aminocyclopropane carboxylic acid, F35]-h-alpha-CGRP 8-37 31 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47870 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 65.3 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47871 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Hop29,D31,p34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47872 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Tic29,D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47873 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Hyp29,D31,p34,F35]-h-alpha-CGRP 27-37 0.006 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47874 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Aib29,D31,p34,F35]-h-alpha-CGRP 27-37 0.002 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47875 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [A29,D31,p34,F35]-h-alpha-CGRP 27-37 8.4 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47876 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47877 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 0.7 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47878 PDE5 AORTA RAT Functional sildenafil 7.94328 Teixeira CE, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47879 PDE5 AORTA RAT Functional vardenafil 2.95121 Teixeira CE, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47880 PDE5 AORTA RAT Functional tadalafil 9.77237 Teixeira CE, et al., 2006 Jan 15, 2025 Jan 15, 2025  
47881 SST1 CLONED HUMAN 3H-thymidine BIM-23926 3.6 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47882 SST2 CLONED HUMAN 3H-thymidine BIM-23926 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47883 SST3 CLONED HUMAN 3H-thymidine BIM-23926 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47884 SST4 CLONED HUMAN 3H-thymidine BIM-23926 833 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47885 SST5 CLONED HUMAN 3H-thymidine BIM-23926 788 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47886 SST1 CLONED HUMAN 3H-thymidine BIM-23745 42 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47887 SST2 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47888 SST3 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47889 SST4 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47890 SST5 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025  
47891 P2X1 CLONED Xenopus Functional NF279 19 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025  
47892 P2X2 CLONED Xenopus Functional NF279 770 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025  
47893 P2X3 CLONED Xenopus Functional NF279 1620 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025  
47894 P2X4 CLONED Xenopus Functional NF279 >10000 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025  
47895 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 2.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47896 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 10 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47897 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 13 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47898 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 7.5 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47899 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47900 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 66 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47901 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 56 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47902 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 21 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47903 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47904 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 12 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47905 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 16 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47906 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 16 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47907 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 4.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47908 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 22 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47909 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 28 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47910 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 41 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47911 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 18 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47912 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 57 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47913 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 184 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47914 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 182 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47915 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47916 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47917 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 12 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47918 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47919 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 170 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47920 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47921 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47922 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47923 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2.9 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47924 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 31 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47925 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 21 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47926 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 24 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47927 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 4.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47928 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 60 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47929 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 46 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47930 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 50 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47931 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 1.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47932 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 4.3 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47933 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 19 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47934 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 48 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47935 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 2.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47936 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 10 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47937 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 7.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47938 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 18 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47939 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 67 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47940 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47941 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47942 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47943 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 15 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47944 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 119 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47945 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 182 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47946 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 69 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47947 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 132 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47948 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47949 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47950 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47951 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 3.9 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47952 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 72 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47953 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 44 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47954 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 87 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47955 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 78 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47956 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47957 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47958 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47959 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 11 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47960 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 211 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47961 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 162 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47962 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 240 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47963 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47964 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47965 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47966 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47967 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47968 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 45 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47969 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 26 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47970 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 25 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47971 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5.8 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47972 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 165 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47973 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 31 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47974 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 33 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47975 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 9.1 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47976 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 172 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47977 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 43 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47978 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 35 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47979 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 15 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47980 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 175 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47981 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 161 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47982 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 159 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47983 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47984 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47985 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47986 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47987 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 85 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47988 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47989 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47990 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47991 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 0.5 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47992 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 3.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47993 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47994 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 10 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47995 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 37 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47996 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47997 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47998 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 185 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
47999 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48000 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 61 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48001 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 44 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48002 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 47 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48003 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 19 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48004 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 267 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48005 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 49 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48006 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 102 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48007 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48008 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 20 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48009 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 16 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48010 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 20 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48011 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 4.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48012 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 79 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48013 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 48 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48014 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 48 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48015 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 1.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48016 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 24 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48017 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 39 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48018 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 28 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025  
48019 AORTA RAT 3H-PRAZOSIN N-(1-Benzylpiperidin-4-yl)-1-isopropylindazole-3-carboxamide Hydrochloride >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025  
48020 AORTA RAT 3H-PRAZOSIN N-(1-(2-((N-Methylsulfonyl)amino)ethyl)piperidin-4-yl)-1-isopropylindazole-3-carboxamide Maleate >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025  
48021 AORTA RAT 3H-PRAZOSIN CISAPRIDE 199.526 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025  
48022 AORTA RAT 3H-PRAZOSIN N-(2-(4-((Benzyloxycarbonyl)amino)-1-piperidinyl)-ethyl)-1-isopropylindazole-3-carboxamide Oxalate >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025  
48023 AORTA RAT 3H-PRAZOSIN N-(2-(4-(1-Adamantylcarboxamido)-1-piperidinyl)ethyl)-1-isopropylindazole-3-carboxamide Oxalate >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025  
48024 AMPA CORTEX RAT 3H-AMPA AMPA 40 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48025 AMPA CORTEX RAT 3H-AMPA Br-HIBO,(RS) 650 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48026 AMPA CORTEX RAT 3H-AMPA C1-HIBO 220 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48027 KA CORTEX RAT 3H-Kainic acid C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48028 KA CORTEX RAT 3H-Kainic acid Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48029 KA CORTEX RAT 3H-Kainic acid AMPA >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48030 NMDA CORTEX RAT 3H-CGP39653 AMPA >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 27, 2025  
48031 NMDA CORTEX RAT 3H-CGP39653 Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 27, 2025  
48032 NMDA CORTEX RAT 3H-CGP39653 C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 27, 2025  
48033 GRIA1 CLONED RAT 3H-AMPA AMPA 22 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48034 GRIA1 CLONED RAT 3H-AMPA Br-HIBO,(RS) 170 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48035 GRIA2 CLONED RAT 3H-AMPA AMPA 17 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48036 GRIA1 CLONED RAT 3H-AMPA C1-HIBO 130 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48037 GRIA2 CLONED RAT 3H-AMPA Br-HIBO,(RS) 250 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48038 GRIA2 CLONED RAT 3H-AMPA C1-HIBO 370 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48039 AMPA CLONED RAT 3H-AMPA AMPA 21 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48040 AMPA CLONED RAT 3H-AMPA Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48041 AMPA CLONED RAT 3H-AMPA C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48042 GRIA4 CLONED RAT 3H-AMPA C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48043 GRIA4 CLONED RAT 3H-AMPA Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48044 GRIA4 CLONED RAT 3H-AMPA AMPA 40 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48045 CLONED RAT 3H-AMPA AMPA 740 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48046 CLONED RAT 3H-AMPA Br-HIBO,(RS) 4800 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48047 CLONED RAT 3H-AMPA C1-HIBO 6800 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48048 CLONED RAT 3H-AMPA C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48049 CLONED RAT 3H-AMPA Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48050 CLONED RAT 3H-AMPA AMPA >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025  
48051 CLONED HUMAN 3H-25-OHC paxilline 660 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025  
48052 CLONED HUMAN 3H-25-OHC paxilline 1100 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025  
48053 CLONED HUMAN 3H-25-OHC [22(R)-hydroxycholesterol 250 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025  
48054 CLONED HUMAN 3H-25-OHC [22(R)-hydroxycholesterol 490 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025  
48055 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 1 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48056 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 7 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48057 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 7 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48058 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48059 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48060 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.05 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48061 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48062 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.8 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48063 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.3 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48064 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.09 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48065 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.1 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48066 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48067 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.9 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48068 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.7 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48069 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.3 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48070 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48071 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48072 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48073 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48074 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48075 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48076 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.4 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48077 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48078 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48079 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.3 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025  
48080 CLONED RAT Functional (S)-Glu >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48081 mGluR2 CLONED RAT Functional (S)-Glu 4400 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48082 mGluR4 CLONED RAT Functional (S)-Glu >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48083 mGluR5 CLONED RAT Functional (S)-Glu 7400 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48084 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48085 mGluR2 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48086 mGluR4 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48087 mGluR5 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48088 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48089 mGluR2 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48090 mGluR4 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48091 mGluR5 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48092 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48093 mGluR2 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48094 mGluR4 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48095 mGluR5 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48096 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48097 mGluR2 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48098 mGluR4 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48099 mGluR5 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48100 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48101 mGluR2 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48102 mGluR4 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48103 mGluR5 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48104 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48105 mGluR2 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48106 mGluR4 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48107 mGluR5 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48108 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48109 mGluR2 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48110 mGluR4 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48111 mGluR5 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48112 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48113 mGluR2 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48114 mGluR4 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48115 mGluR5 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48116 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48117 mGluR2 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48118 mGluR4 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48119 mGluR5 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48120 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48121 mGluR2 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48122 mGluR4 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48123 mGluR5 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48124 CLONED RAT Functional (S)-4-Carboxyphenylglycine >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025  
48125 mGluR5 CLONED RAT Functional (S)-4-Carboxyphenylglycine >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025  
48126 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.23 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48127 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 700 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48128 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48129 Y1 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 530 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48130 Y1 CLONED HUMAN 3H-Propionyl-NPY PP, human 170 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48131 Y1 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 760 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48132 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48133 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 29 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48134 Y2 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 0.03 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48135 Y2 CLONED HUMAN 3H-Propionyl-NPY PP, human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48136 Y2 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48137 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48138 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48139 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.04 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48140 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY, human 5.8 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48141 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48142 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 170 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48143 Y4 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 51 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48144 Y4 CLONED HUMAN 3H-Propionyl-NPY PP, human 0.06 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48145 Y4 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 15 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48146 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48147 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 35 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48148 Y5 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 17 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48149 Y5 CLONED HUMAN 3H-Propionyl-NPY PP, human 1.4 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48150 Y5 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 0.24 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48151 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 0.92 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48152 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 6 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48153 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.6 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025  
48154 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(Pyrrol-1-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 61.5 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025  
48155 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(Thien-2-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 10.3 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025  
48156 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(Thien-3-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 36.3 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025  
48157 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(N-Formylcarbamoyl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 844.2 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025  
48158 GABAA BRAIN BOVINE 3H-RO-15-1788 DIAZEPAM 10 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025  
48159 A1 BRAIN RAT 3H-cyclohexyladenosine BS-DMPX 1200 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48160 A1 BRAIN RAT 3H-cyclohexyladenosine MS-DMPX 1280 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48161 A1 BRAIN RAT 3H-cyclohexyladenosine 3-(2-Hydroxyethyl)-8-(m-methoxystyryl)-7-methyl-1-propargylxanthine 1040 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48162 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(m-Bromostyryl)-3-(2-hydroxyethyl)-7-methyl-1-propargylxanthine 1280 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48163 A1 CLONED HUMAN 3H-CCPA MSX-2 2500 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48164 A1 BRAIN RAT 3H-cyclohexyladenosine MSX-2 900 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48165 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(m-Bromostyryl)-3-(3-hydroxypropyl)-7-methyl-1-propargylxanthine 625 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48166 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(m-Aminostyryl)-3,7-dimethyl-1-propargylxanthine 1070 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48167 A1 BRAIN RAT 3H-cyclohexyladenosine 3,7-Dimethyl-8-(m-hydroxystyryl)-1-propargylxanthine 940 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48168 A2A BRAIN RAT 3H-CGS-21680 BS-DMPX 8.2 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48169 A2A BRAIN RAT 3H-CGS-21680 MS-DMPX 12 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48170 A2A BRAIN RAT 3H-CGS-21680 3-(2-Hydroxyethyl)-8-(m-methoxystyryl)-7-methyl-1-propargylxanthine 39 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48171 A2A BRAIN RAT 3H-CGS-21680 8-(m-Bromostyryl)-3-(2-hydroxyethyl)-7-methyl-1-propargylxanthine 25 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48172 A2A CLONED HUMAN 3H-CGS-21680 MSX-2 5 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48173 A2A BRAIN HUMAN 3H-CGS-21680 MSX-2 15 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48174 A2A BRAIN RAT 3H-CGS-21680 MSX-2 8 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48175 A2A BRAIN RAT 3H-CGS-21680 8-(m-Bromostyryl)-3-(3-hydroxypropyl)-7-methyl-1-propargylxanthine 13 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48176 A2A BRAIN RAT 3H-CGS-21680 8-(m-Aminostyryl)-3,7-dimethyl-1-propargylxanthine 42 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48177 A2A BRAIN RAT 3H-CGS-21680 3,7-Dimethyl-8-(m-hydroxystyryl)-1-propargylxanthine 21 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48178 A3 CLONED HUMAN 3H-NECA BS-DMPX >10000 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48179 A3 CLONED HUMAN 3H-NECA MSX-2 >10000 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025  
48180 Y4 CLONED GUINEA PIG 125I-hPP PP, guinea pig 0.046 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48181 Y4 CLONED GUINEA PIG 125I-hPP PP, human 0.031 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48182 Y4 CLONED GUINEA PIG 125I-hPP PP, rat 0.044 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48183 Y4 CLONED GUINEA PIG 125I-hPP PP, BOVINE 0.013 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48184 Y4 CLONED HUMAN 125I-hPP PP, guinea pig 0.06 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48185 Y4 CLONED HUMAN 125I-hPP PP, human 0.039 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48186 Y4 CLONED HUMAN 125I-hPP PP, rat 0.071 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48187 Y4 CLONED HUMAN 125I-hPP PP, BOVINE 0.031 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48188 Y4 CLONED RAT 125I-hPP PP, guinea pig 0.007 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48189 Y4 CLONED RAT 125I-hPP PP, human 0.003 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48190 Y4 CLONED RAT 125I-hPP PP, rat 0.0027 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48191 Y4 CLONED RAT 125I-hPP PP, BOVINE 0.006 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48192 Y4 CLONED GUINEA PIG 125I-hPP NPY, porcine 25 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48193 Y4 CLONED GUINEA PIG 125I-hPP PYY, porcine 26 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48194 Y4 CLONED GUINEA PIG 125I-hPP NPY,[leu31,Pro34], porcine 20 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48195 Y4 CLONED GUINEA PIG 125I-hPP PYY,[leu31,Pro34], human 16 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48196 Y4 CLONED GUINEA PIG 125I-hPP NPY2-36, porcine 130 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48197 Y4 CLONED GUINEA PIG 125I-hPP NPY13-36, porcine 29 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48198 Y4 CLONED GUINEA PIG 125I-hPP NPY D-Trp32, porcine 1000 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48199 Y4 CLONED HUMAN 125I-hPP NPY, porcine 6 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48200 Y4 CLONED HUMAN 125I-hPP PYY, porcine 4 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48201 Y4 CLONED HUMAN 125I-hPP NPY,[leu31,Pro34], porcine 6.6 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48202 Y4 CLONED HUMAN 125I-hPP PYY,[leu31,Pro34], human 11 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48203 Y4 CLONED HUMAN 125I-hPP NPY2-36, porcine 17 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48204 Y4 CLONED HUMAN 125I-hPP NPY13-36, porcine 9 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48205 Y4 CLONED HUMAN 125I-hPP NPY D-Trp32, porcine 1000 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48206 Y4 CLONED RAT 125I-hPP NPY, porcine 18 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48207 Y4 CLONED RAT 125I-hPP PYY, porcine 11 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48208 Y4 CLONED RAT 125I-hPP PYY,[leu31,Pro34], human 0.62 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48209 Y4 CLONED RAT 125I-hPP NPY2-36, porcine 29 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48210 Y4 CLONED RAT 125I-hPP NPY13-36, porcine 2.2 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48211 Y4 CLONED RAT 125I-hPP NPY D-Trp32, porcine 60 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025  
48212 nAChR BRAIN RAT 3H-NICOTINE Nicotine 1.26 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48213 nAChR BRAIN RAT 3H-NICOTINE 6-Bromonicotine 0.45 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48214 nAChR BRAIN RAT 3H-NICOTINE 6-Fluoro-3-( l-methyl-2-pyrrohdinyl )pyridme maleate 1.03 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48215 nAChR BRAIN RAT 3H-NICOTINE 6-Methyl-3-(1 -methyl-2-pyrrohdmyl)pyridme dthydrochlortde 1.8 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48216 nAChR BRAIN RAT 3H-NICOTINE 6-methoxynicotine 22 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48217 nAChR BRAIN RAT 3H-NICOTINE 5-(N-Ethyl)amino-5,0,7,8-tetrahydroquinoline maleate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48218 nAChR BRAIN RAT 3H-NICOTINE 1,2,3.4-Tetrahydro[2,7]naphthyrldine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48219 nAChR BRAIN RAT 3H-NICOTINE 2-Methyl-l,2,3.4-tetrahydro[2,7]naphthyridine oxalate 18 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48220 nAChR BRAIN RAT 3H-NICOTINE 2-Ethyl-l,2,3,4-tetrahydro[2,7]naphthyrtdme oxalate 52 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48221 nAChR BRAIN RAT 3H-NICOTINE 2-Propyl-l,2,3,4-tetrahydro[2,7]naphthyrMme oxalate 1640 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48222 nAChR BRAIN RAT 3H-NICOTINE 2-1sopropyl-l.2,3,4-tetrahydro[2.7]naphthyridine oxalate 123 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48223 nAChR BRAIN RAT 3H-NICOTINE 5,6,7,9-Tetrahydro-8H-pyrldo[3,4-c]azepine oxalate 1100 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48224 nAChR BRAIN RAT 3H-NICOTINE 8-Methyl-5.6,7,9-tetrahydro-8H-pyrido[3,4-c]azepine oxalate 780 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48225 nAChR BRAIN RAT 3H-NICOTINE 2-Methyl- 2.3-dihydro-l H-pyrrolo[3,4-c]pyrMine oxalate 85 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48226 nAChR BRAIN RAT 3H-NICOTINE 6-Chloro-3-(N-ethyl-N-methyl)aminomethylpyridine oxalat 41 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48227 nAChR BRAIN RAT 3H-NICOTINE 6-Methyl-3-(N-ethyl-N-methylammomethyl)pyridme oxalate 66 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48228 nAChR BRAIN RAT 3H-NICOTINE 6-Metho,D'-3-(N-ethyl-N-methylamtnomethyl)pyndine oxalate 640 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48229 nAChR BRAIN RAT 3H-NICOTINE 6-Fluoro-3-(N-ethyl-N-methyl)aminomethylpyridine oxalate 93 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48230 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Methyl-N-n-propylammomethyl)-2-methylpyridine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48231 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Methyl-N-n-propylaminomethyl)pyridine oxalate 1140 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48232 nAChR BRAIN RAT 3H-NICOTINE 3-(N-n-Butyl-N-methylaminornethyl)pyridine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48233 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Methyl-N-n-peno, laminomethyl)pyrtdine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48234 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Cyclopropyl-N-methylaminornethyl)pyrMine oxalate 840 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025  
48235 SLC6A4 CLONED HUMAN 3H-CITALOPRAM stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48236 5-HT1A CLONED HUMAN 3H-8-OH-DPAT stepholidine 143.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48237 5-HT1B CLONED HUMAN 3H-GR-125743 stepholidine 6984 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48238 5-HT1D CLONED HUMAN 3H-GR-125743 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48239 5-HT1E CLONED HUMAN 3H-5HT stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48240 5-HT2A CLONED HUMAN 3H-KETANSERIN stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48241 5-HT2C CLONED RAT 3H-MESULERGINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48242 5-HT3 CLONED HUMAN 3H-LY 278584 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48243 CB1 CLONED HUMAN 3H-LSD stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025  
48244 5-HT6 CLONED HUMAN 3H-LSD stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48245 5-HT7 CLONED HUMAN 3H-LSD stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48246 5-HT2B CLONED HUMAN 3H-LSD stepholidine 226 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48247 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48248 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48249 5-HT1B CLONED HUMAN 3H-GR-125743 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48250 5-HT1D CLONED HUMAN 3H-GR-125743 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48251 5-HT1E CLONED HUMAN 3H-5HT PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48252 5-HT2A CLONED HUMAN 3H-KETANSERIN PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48253 5-HT2C CLONED RAT 3H-MESULERGINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48254 5-HT3 CLONED HUMAN 3H-ZACOPRIDE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48255 CB1 CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025  
48256 5-HT6 CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48257 5-HT7 CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48258 5-HT2B CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48259 Alpha1A CLONED HUMAN 3H-PRAZOSIN PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48260 Alpha1B CLONED HUMAN 3H-PRAZOSIN PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48261 Alpha2A CLONED HUMAN 3H-CLONIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48262 Alpha2B CLONED HUMAN 3H-CLONIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48263 Alpha2C CLONED HUMAN 3H-CLONIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48264 Beta1 CLONED HUMAN 125I-Pindolol PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48265 Beta2 CLONED HUMAN 125I-Pindolol PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025  
48266 H1 CLONED HUMAN 3H-PYRILAMINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48267 H2 CLONED HUMAN 3H-TIOTIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48268 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48269 H4 CLONED HUMAN 3H-Histamine PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48270 D1 CLONED HUMAN 3H-SCH23390 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48271 D2 CLONED HUMAN 3H-NMSP PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48272 D3 CLONED RAT 3H-NMSP PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48273 D4 CLONED HUMAN 3H-NMSP PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48274 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48275 NET CLONED HUMAN 3H-Nisoxetine PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48276 M2 CLONED HUMAN 3H-QNB PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48277 M5 CLONED HUMAN 3H-QNB PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48278 KOR CLONED HUMAN 3H-Diprenorphine PBR28 2.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48279 Alpha1A CLONED HUMAN 3H-PRAZOSIN stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48280 Alpha1B CLONED HUMAN 3H-PRAZOSIN stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48281 Alpha2A CLONED HUMAN 3H-CLONIDINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48282 Alpha2B CLONED HUMAN 3H-CLONIDINE stepholidine 6884 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48283 Alpha2C CLONED HUMAN 3H-CLONIDINE stepholidine 214.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48284 Beta1 CLONED HUMAN 125I-Pindolol stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48285 Beta2 CLONED HUMAN 125I-Pindolol stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025  
48286 H1 CLONED HUMAN 3H-PYRILAMINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48287 H2 CLONED HUMAN 3H-TIOTIDINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48288 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48289 H4 CLONED HUMAN 3H-Histamine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48290 D1 CLONED HUMAN 3H-SCH23390 stepholidine 5.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48291 D2 CLONED HUMAN 3H-NMSP stepholidine 974.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48292 D3 CLONED RAT 3H-NMSP stepholidine 30.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48293 D4 CLONED HUMAN 3H-NMSP stepholidine 3748 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48294 D5 CLONED HUMAN 3H-SCH23390 stepholidine 4.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48295 SLC6A3 CLONED HUMAN 3H-WIN 35,428 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48296 NET CLONED HUMAN 3H-Nisoxetine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48297 MOR CLONED HUMAN 3H-Diprenorphine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48298 M2 CLONED HUMAN 3H-QNB stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48299 DOR CLONED HUMAN 3H-DADLE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48300 KOR CLONED HUMAN 3H-Diprenorphine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48301 M5 CLONED HUMAN 3H-QNB stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48302 KOR FOREBRAIN RAT 3H-MUSCIMOL stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025  
48303 HEART RAT 3H-Nitrendipine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48304 CB2 CLONED HUMAN 3H-CP-55940 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48305 CB1 CLONED HUMAN 3H-CP-55940 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48306 I1 PC12 RAT 125I-Pindolol stepholidine 8909 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48307 Sigma 1 BRAIN RAT 3H-Pentazocine(+) stepholidine 1600 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48308 Sigma 2 PC12 RAT 3H-DTG stepholidine 53.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48309 NMDA FOREBRAIN RAT 3H-MK-801 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48310 mGluR5 LLC-PK1 cells PORCINE Functional Glutamate 9750 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48311 LLC-PK1 cells PORCINE Functional Glutamate 7670 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48312 LLC-PK1 cells PORCINE Functional Quisqualate 260 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48313 mGluR5 LLC-PK1 cells PORCINE Functional Quisqualate 22 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48314 LLC-PK1 cells PORCINE Functional Quisqualate 47 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48315 LLC-PK1 cells PORCINE Functional Ibotenate >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48316 mGluR5 LLC-PK1 cells PORCINE Functional Ibotenate 2870 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48317 LLC-PK1 cells PORCINE Functional Ibotenate 1930 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48318 LLC-PK1 cells PORCINE Functional (+/-)-trans-ACPD 2880 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48319 mGluR5 LLC-PK1 cells PORCINE Functional (+/-)-trans-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48320 LLC-PK1 cells PORCINE Functional (+/-)-trans-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48321 LLC-PK1 cells PORCINE Functional 1S, 3R-ACPD 9300 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48322 mGluR5 LLC-PK1 cells PORCINE Functional 1S, 3R-ACPD 6700 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48323 LLC-PK1 cells PORCINE Functional 1S, 3R-ACPD 5300 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48324 LLC-PK1 cells PORCINE Functional 1R,3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48325 mGluR5 LLC-PK1 cells PORCINE Functional 1R,3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48326 LLC-PK1 cells PORCINE Functional 1R,3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48327 LLC-PK1 cells PORCINE Functional 1S, 3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48328 mGluR5 LLC-PK1 cells PORCINE Functional 1S, 3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48329 LLC-PK1 cells PORCINE Functional 1S, 3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48330 LLC-PK1 cells PORCINE Functional 1R,3R-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48331 mGluR5 LLC-PK1 cells PORCINE Functional 1R,3R-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025  
48332 LLC-PK1 cells PORCINE Functional 1R,3R-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48333 LLC-PK1 cells PORCINE Functional Glutamate >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025  
48334 5-HT2A CLONED RAT 3H-KETANSERIN  1-(Aminomethyl)dibenzo[b,e]bicyclo[2.2.2]octadiene Hydrochloride 770 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48335 5-HT2A CLONED RAT 3H-KETANSERIN  9-Aminomethyl-9,10-dihydro-9,10-methanoanthracene Hydrochloride 6780 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48336 5-HT2A CLONED RAT 3H-KETANSERIN  9-Methyl-9-aminomethyl-9,10-dihydroanthracene Oxalate 65 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48337 5-HT2A CLONED RAT 3H-KETANSERIN  9-Aminomethyl-10,10-dimethyl-9,10-dihydroanthracene Oxalate  330 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48338 5-HT2A CLONED RAT 3H-KETANSERIN 11-Amino-9,10-dihydro-9,10-ethanoanthracene Oxalate >10000 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48339 5-HT2A CLONED RAT 3H-KETANSERIN 9-(1-Aminoethyl)-9,10-dihydroanthracene Hydrochloride 193 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48340 5-HT2A CLONED RAT 3H-KETANSERIN 2,3,7,11b-Tetrahydrodibenzo[d,e,h]isoquinoline Oxalate 296 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48341 5-HT2A CLONED RAT 3H-KETANSERIN AMDA 20 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48342 5-HT2A CLONED RAT 3H-KETANSERIN 2,2-diphenylethylamine 4610 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48343 5-HT2A CLONED RAT 3H-KETANSERIN tetrahydronaphthalene >10000 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48344 5-HT2A CLONED RAT 3H-KETANSERIN 2-(2-benzylphenyl)-ethylamine 1810 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48345 5-HT2A CLONED RAT 3H-KETANSERIN [a,d]dibenz-fused cycloheptane 112 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025  
48346 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PERGOLIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48347 Sigma 2 PC12 RAT 3H-DTG PERGOLIDE 922.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48348 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Memantine 4131 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48349 Sigma 2 PC12 RAT 3H-DTG Memantine 9450 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48350 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Chloroquine 108.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48351 Sigma 2 PC12 RAT 3H-DTG Chloroquine 1129 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48352 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PPP, S(-)-3 774.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48353 Sigma 2 PC12 RAT 3H-DTG PPP, S(-)-3 1415 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48354 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PPP, R(+)-3 192.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48355 Sigma 2 PC12 RAT 3H-DTG PPP, R(+)-3 181.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48356 Sigma 1 BRAIN RAT 3H-Pentazocine(+) FLUOXETINE 1911 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48357 Sigma 2 PC12 RAT 3H-DTG FLUOXETINE 1121 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48358 Sigma 2 PC12 RAT 3H-DTG DESIPRAMINE 1611 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48359 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Amiodarone 791.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48360 Sigma 1 BRAIN RAT 3H-Pentazocine(+) SKF 82957 1444 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48361 Sigma 2 PC12 RAT 3H-DTG PHENYLEPHRINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48363 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 6-(((6-chloro-4H-1,3-benzodioxin-8-yl)methyl)thio)-3-(cyclopropylmethyl)-1,2,3,4-tetrahydro-1,3,5-triazine 410.83 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48364 Sigma 2 PC12 RAT 3H-DTG R-(+) staurosine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48365 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Lofepramine 2520 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48366 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Rimonabant 4350 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48367 Sigma 2 PC12 RAT 3H-DTG CLOZAPINE-N-OXIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48368 Sigma 1 BRAIN RAT 3H-Pentazocine(+) CLOZAPINE-N-OXIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48369 Sigma 1 BRAIN RAT 3H-Pentazocine(+) L-DOPA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48370 Sigma 2 PC12 RAT 3H-DTG L-DOPA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48371 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Picrotoxin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48372 Sigma 2 PC12 RAT 3H-DTG Picrotoxin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48373 Sigma 1 BRAIN RAT 3H-Pentazocine(+) YOHIMBINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48374 Sigma 2 PC12 RAT 3H-DTG YOHIMBINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48375 Sigma 1 BRAIN RAT 3H-Pentazocine(+) SKF 75670 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48376 Sigma 2 PC12 RAT 3H-DTG SKF 75670 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48377 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Arecoline >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48378 Sigma 2 PC12 RAT 3H-DTG Arecoline >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48379 Sigma 1 BRAIN RAT 3H-Pentazocine(+) DESIPRAMINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48380 Sigma 2 PC12 RAT 3H-DTG Amiodarone >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48381 Sigma 2 PC12 RAT 3H-DTG SKF 82957 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48382 Sigma 2 PC12 RAT 3H-DTG Tramadol(+-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48383 Sigma 2 PC12 RAT 3H-DTG Pramipexole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48384 Sigma 2 PC12 RAT 3H-DTG Amantadine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48385 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Agomelatine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48386 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Tramadol(+-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48387 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Amantadine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48388 Sigma 1 BRAIN RAT 3H-Pentazocine(+) topiramate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48389 Sigma 2 PC12 RAT 3H-DTG topiramate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48390 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PHENYLEPHRINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48391 Sigma 1 BRAIN RAT 3H-Pentazocine(+) DDMV >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48392 Sigma 2 PC12 RAT 3H-DTG Menthol-(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48393 Sigma 2 PC12 RAT 3H-DTG Menthol-(-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48394 Sigma 2 PC12 RAT 3H-DTG Neomenthol-(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48395 Sigma 2 PC12 RAT 3H-DTG Neomenthol-(-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48396 Sigma 2 PC12 RAT 3H-DTG Isomenthol-(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48397 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Thujone >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48398 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Acetyl-L-Carnitine HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48399 Sigma 1 BRAIN RAT 3H-Pentazocine(+) L-Carnitine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48400 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Triamcinolone (Fluoxyprednisolone) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48401 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Phenobarbitol sodium salt >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48402 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Dieldrin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48403 Sigma 1 BRAIN RAT 3H-Pentazocine(+) D,L Kavain >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48404 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Myristicin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48405 Sigma 1 BRAIN RAT 3H-Pentazocine(+) alpha-Estradiol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48406 Sigma 1 BRAIN RAT 3H-Pentazocine(+) MTEP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48407 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Indinavir sulphate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48408 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Efavirenz >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48409 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Stavudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48410 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Ritonavir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48411 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Nelfinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48412 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Nevirapine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48413 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Zalcitabine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48414 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Saquinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48415 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Zidovudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48416 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Tenofovir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48417 Sigma 1 BRAIN RAT 3H-Pentazocine(+) DHL >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48418 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4OHBA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48419 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4OHMNA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48420 Sigma 1 BRAIN RAT 3H-Pentazocine(+) securinine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48421 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 3-(2,4-dithioxo-1,3-thiazolidin-3-yl)propanoic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48422 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4-methyl[1]benzofuro[3,2-g]quinolin-2-ol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48423 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Gitoxigenin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48424 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Triciribine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48425 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 6-Benzylthioinosine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48426 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Hoodia Extract >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48427 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Galnon >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48428 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Glaucine HBr >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48429 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Glaucium fl. extract >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48430 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Acamprosate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48431 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Oseltamivir PO4 - Tamiflu >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48432 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Oseltamivir Acid - tamiflu metabolite >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48444 Sigma 2 PC12 RAT 3H-DTG Thujone >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48445 Sigma 2 PC12 RAT 3H-DTG Acetyl-L-Carnitine HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48446 Sigma 2 PC12 RAT 3H-DTG L-Carnitine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48447 Sigma 2 PC12 RAT 3H-DTG Triamcinolone (Fluoxyprednisolone) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48448 Sigma 2 PC12 RAT 3H-DTG Phenobarbitol sodium salt >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48449 Sigma 2 PC12 RAT 3H-DTG Dieldrin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48450 Sigma 2 PC12 RAT 3H-DTG D,L Kavain >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48451 Sigma 2 PC12 RAT 3H-DTG 1-phenlsemicarbazide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48452 Sigma 2 PC12 RAT 3H-DTG Myristicin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48453 Sigma 2 PC12 RAT 3H-DTG alpha-Estradiol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48454 Sigma 2 PC12 RAT 3H-DTG Indinavir sulphate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48455 Sigma 2 PC12 RAT 3H-DTG Efavirenz >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48456 Sigma 2 PC12 RAT 3H-DTG Stavudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48457 Sigma 2 PC12 RAT 3H-DTG Ritonavir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48458 Sigma 2 PC12 RAT 3H-DTG Nelfinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48459 Sigma 2 PC12 RAT 3H-DTG Nevirapine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48460 Sigma 2 PC12 RAT 3H-DTG Zalcitabine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48461 Sigma 2 PC12 RAT 3H-DTG Saquinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48462 Sigma 2 PC12 RAT 3H-DTG Zidovudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48463 Sigma 2 PC12 RAT 3H-DTG Tenofovir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48464 Sigma 2 PC12 RAT 3H-DTG DHL >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48465 Sigma 2 PC12 RAT 3H-DTG 4OHBA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48466 Sigma 2 PC12 RAT 3H-DTG 4OHMNA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48467 Sigma 2 PC12 RAT 3H-DTG securinine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48468 Sigma 2 PC12 RAT 3H-DTG 3-(2,4-dithioxo-1,3-thiazolidin-3-yl)propanoic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48469 Sigma 2 PC12 RAT 3H-DTG 4-methyl[1]benzofuro[3,2-g]quinolin-2-ol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48470 Sigma 2 PC12 RAT 3H-DTG Gitoxigenin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48471 Sigma 2 PC12 RAT 3H-DTG Triciribine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48472 Sigma 2 PC12 RAT 3H-DTG 6-Benzylthioinosine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48473 Sigma 2 PC12 RAT 3H-DTG Hoodia Extract >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48474 Sigma 2 PC12 RAT 3H-DTG Galnon >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48475 Sigma 2 PC12 RAT 3H-DTG MTEP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48476 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 1-phenlsemicarbazide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48555 5-HT2B CLONED HUMAN 3H-LSD METHAMPHETAMINE (+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48556 NET CLONED HUMAN 3H-Nisoxetine METHAMPHETAMINE (+) 965.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48557 Alpha2A CLONED HUMAN 3H-CLONIDINE METHAMPHETAMINE (+) 4142 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48558 Alpha2B CLONED HUMAN 3H-CLONIDINE METHAMPHETAMINE (+) 744.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48559 Alpha2C CLONED HUMAN 3H-CLONIDINE METHAMPHETAMINE (+) 813.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48560 5-HT1A CLONED HUMAN 3H-8-OH-DPAT mCPP 43.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48561 5-HT1B CLONED HUMAN 3H-5CT mCPP 163.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48562 5-HT2A CLONED HUMAN 3H-KETANSERIN mCPP 196.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48563 5-HT2B CLONED HUMAN 3H-LSD mCPP 19.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48564 5-HT2C CLONED RAT 3H-MESULERGINE mCPP 108 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48565 5-HT3 CLONED HUMAN 3H-LY 278584 mCPP 427 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48566 5-HT5A CLONED HUMAN 3H-LSD mCPP 1354 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48567 5-HT6 CLONED HUMAN 3H-LSD mCPP 1748 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48568 5-HT7 CLONED HUMAN 3H-LSD mCPP 162.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48569 Alpha1A CLONED HUMAN 3H-PRAZOSIN mCPP 1386 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48570 Alpha1B CLONED HUMAN 3H-PRAZOSIN mCPP 914.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48571 Alpha2A CLONED HUMAN 3H-CLONIDINE mCPP 145.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48572 Alpha2B CLONED HUMAN 3H-CLONIDINE mCPP 105.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48573 Alpha2C CLONED HUMAN 3H-CLONIDINE mCPP 123.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48574 Beta1 CLONED HUMAN 125I-Pindolol mCPP 2359 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48575 Beta2 CLONED HUMAN 125I-Pindolol mCPP 3474 PDSP Certified Data Jan 15, 2025 Jan 28, 2025  
48576 HEART RAT 3H-Nitrendipine mCPP 6043 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48577 D3 CLONED RAT 3H-NMSP mCPP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48578 D5 CLONED HUMAN 3H-SCH23390 mCPP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48579 H1 CLONED HUMAN 3H-PYRILAMINE mCPP 326.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48580 I1 PC12 RAT 125I-Pindolol mCPP 758.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48581 NET CLONED HUMAN 3H-Nisoxetine mCPP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48582 SLC6A4 CLONED HUMAN 3H-CITALOPRAM mCPP 328.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48583 Sigma 2 PC12 RAT 3H-DTG mCPP 8350 PDSP Certified Data Jan 15, 2025 Jan 15, 2025  
48585 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 800 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48586 CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 475 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48587 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2400 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48588 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 330 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48589 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 700 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48590 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 417 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48591 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 7700 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48592 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48593 CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48594 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48595 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48596 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48597 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.25 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48598 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.9 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48599 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 17.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48600 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 158 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48601 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 18.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48602 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 42.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48603 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 35 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48604 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 18.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48605 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 1.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48606 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48607 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48608 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48609 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48610 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48611 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48612 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 30 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48613 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 1.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48614 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 9 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48615 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 4.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48616 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48617 GNRHR CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48618 GNRHR CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48619 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48620 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48621 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 1.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48622 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.55 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48623 GNRHR CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48624 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 435 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48625 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48626 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 18.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48627 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48628 GNRHR CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.15 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48629 CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 1140 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48630 CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48631 GNRHR CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48632 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 1060 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48633 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 0.22 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48634 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 59 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48635 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 3.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48636 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48637 GNRHR CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 0.37 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48638 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 464 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48639 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48640 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.29 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48641 GNRHR CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48642 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 350 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48643 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48644 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48645 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 9.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48646 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48647 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48648 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 400 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48649 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48650 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48651 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 12.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48652 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48653 GNRHR CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48654 CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 770 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48655 CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48656 GNRHR CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48657 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 274 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48658 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.13 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48659 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 12.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48660 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.85 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48661 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48662 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.22 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48663 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 464 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48664 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48665 GNRHR CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48666 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 800 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48667 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48668 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48669 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48670 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48671 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48672 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 39.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48673 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 11.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48674 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 9.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48675 GNRHR CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.68 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48676 CLONED HUMAN Functional 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48677 CLONED HUMAN Functional 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48678 GNRHR CLONED HUMAN Functional 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48679 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48680 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48681 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 20 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48682 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48683 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48684 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48685 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48686 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48687 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 23.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48688 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 3.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48689 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 2.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48690 GNRHR CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48691 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48692 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride 0.15 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48693 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48694 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 8660 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48695 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.33 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48696 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 13 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48697 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 1.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48698 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 1.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48699 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48700 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 7300 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48701 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48702 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 23 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48703 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48704 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025  
48705 GNRHR CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025