39486 5-HT2C CLONED RAT 3H-MESULERGINE 4-Hydroxy-3-(2-[N-1,2,3,4 tetrahydroquinolino]ethyl)indole 1446 Sard H, et al., 2005 Jan 15, 2025 Jan 15, 2025
39487 5-HT2C CLONED RAT 3H-MESULERGINE 4-Hydroxygramine 49 Sard H, et al., 2005 Jan 15, 2025 Jan 15, 2025
39488 5-HT2C CLONED RAT 3H-MESULERGINE 1-(2-Dimethylaminoethyl)-4-hydroxyindole 9351 Sard H, et al., 2005 Jan 15, 2025 Jan 15, 2025
39489 5-HT4 CLONED HUMAN 3H-GR-113808 ML10302 5 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39490 5-HT4 CLONED HUMAN 3H-GR-113808 C36H50Cl2N6O9•0.75H2O), C, H, N 19 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39491 5-HT4 CLONED HUMAN 3H-GR-113808 (C38H54Cl2N6O10•H2O), C, H, N 3 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39492 5-HT4 CLONED HUMAN 3H-GR-113808 (C34H46Cl2N6O8•1.5H2O), C, H, N 24 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39493 5-HT4 CLONED HUMAN 3H-GR-113808 (C35H48Cl2N6O8•2.5H2O), C, H, N 31 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39494 5-HT4 CLONED HUMAN 3H-GR-113808 (C37H52Cl2N6O8), C, H, N 7 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39495 5-HT4 CLONED HUMAN 3H-GR-113808 C42H62Cl2N6O8•0.75H2O), C, H, N 20 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39496 5-HT4 CLONED HUMAN 3H-GR-113808 (C34H46Cl2N6O8•H2O), C, H, N 21 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39497 5-HT4 CLONED HUMAN 3H-GR-113808 (C35H48Cl2N6O8), C, H, N 5 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39498 5-HT4 CLONED HUMAN 3H-GR-113808 (C37H52Cl2N6O8•1.5H2O), C, H, N 9 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39499 5-HT4 CLONED HUMAN 3H-GR-113808 (C42H62Cl2N6O8•0.5H2O), C, H, N 16 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39500 5-HT4 CLONED HUMAN 3H-GR-113808 (C34H46Cl2N6O8•3H2O), C, H, N 37 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39501 5-HT4 CLONED HUMAN 3H-GR-113808 (C35H48Cl2N6O8•H2O), C, H, N 13 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39502 5-HT4 CLONED HUMAN 3H-GR-113808 (C37H52Cl2N6O8•2.5H2O), C, H, N 5 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39503 5-HT4 CLONED HUMAN 3H-GR-113808 (C42H62Cl2N6O8•1.5H2O), C, H, N 8 Soulier JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39504 5-HT6 CLONED HUMAN 3H-LSD 3-benzyl-N1-(N,N-dimethylaminoethyl)indole 32 Kolanos R, et al., 2005 Jan 15, 2025 Jan 15, 2025
39505 5-HT6 CLONED HUMAN 3H-LSD 1-benzyl-3-(N,N-dimethylaminoethyl)indene 3 Kolanos R, et al., 2005 Jan 15, 2025 Jan 15, 2025
39506 5-HT6 CLONED HUMAN 3H-LSD 3-(4-aminobenzyl)indene >10000 Kolanos R, et al., 2005 Jan 15, 2025 Jan 15, 2025
39507 5-HT6 CLONED HUMAN 3H-LSD 1-(4-aminobenzyl)indene 4470 Kolanos R, et al., 2005 Jan 15, 2025 Jan 15, 2025
39508 5-HT6 CLONED HUMAN 3H-LSD 3-(4-aminobenzyl)indole 2530 Kolanos R, et al., 2005 Jan 15, 2025 Jan 15, 2025
39509 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 3.8 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39510 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid 1.3 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39511 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1.3 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39512 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 2.9 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39513 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 29 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39514 S1P1 CLONED HUMAN 35S-GTPGammaS 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 0.6 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39515 S1P1 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 3.8 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39516 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1.8 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39517 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 4.5 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39518 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 2.2 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39519 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 0.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39520 S1P1 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39521 S1P1 CLONED HUMAN 35S-GTPGammaS 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid 1.7 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39522 S1P1 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 0.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39523 S1P1 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 0.9 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39524 S1P1 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 0.8 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39525 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39526 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid 3086 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39527 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39528 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39529 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39530 S1P3 CLONED HUMAN 35S-GTPGammaS 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39531 S1P3 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39532 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39533 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39534 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39535 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39536 S1P3 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39537 S1P3 CLONED HUMAN 35S-GTPGammaS 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39538 S1P3 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39539 S1P3 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 4282 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39540 S1P3 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 4018 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39541 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 370 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39542 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid 75 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39543 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 150 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39544 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 350 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39545 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid >10000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39546 SIP4 CLONED HUMAN 35S-GTPGammaS 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 70 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39547 SIP4 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 90 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39548 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 370 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39549 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1000 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39550 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 520 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39551 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 49 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39552 SIP4 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 40 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39553 SIP4 CLONED HUMAN 35S-GTPGammaS 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid 240 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39554 SIP4 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 430 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39555 SIP4 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 68 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39556 SIP4 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 89 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39557 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 5.2 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39558 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid 1.8 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39559 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 1.6 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39560 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 2.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39561 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 6.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39562 S1P5 CLONED HUMAN 35S-GTPGammaS 1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid 1 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39563 S1P5 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 6.6 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39564 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 12 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39565 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 12 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39566 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39567 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 0.5 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39568 S1P5 CLONED HUMAN 35S-GTPGammaS 1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid 0.8 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39569 S1P5 CLONED HUMAN 35S-GTPGammaS 1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid 11 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39570 S1P5 CLONED HUMAN 35S-GTPGammaS 1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid 0.3 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39571 S1P5 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 0.5 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39572 S1P5 CLONED HUMAN 35S-GTPGammaS 1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid 0.4 Li Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
39573 5-HT2A CLONED HUMAN Functional BW-723C86 218.776 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39574 5-HT2B CLONED HUMAN Functional BW-723C86 1.07152 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39575 5-HT2C CLONED HUMAN Functional BW-723C86 93.3254 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39576 5-HT2A CLONED HUMAN Functional 5-Hydroxy Tryptamine 30.903 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39577 5-HT2A CLONED HUMAN Functional 5-HT,a-Me 40.738 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39578 5-HT2A CLONED HUMAN Functional TRYPTAMINE 257.04 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39579 5-HT2A CLONED HUMAN Functional 5-CT 549.541 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39580 5-HT2A CLONED HUMAN Functional 5-HT,20Me 2398.83 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39581 5-HT2A CLONED HUMAN Functional mCPP 223.872 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39582 5-HT2A CLONED HUMAN Functional TFMPP 162.181 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39583 5-HT2A CLONED HUMAN Functional ORG-12962 416.869 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39584 5-HT2A CLONED HUMAN Functional Ro 60-0175 446.684 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39585 5-HT2A CLONED HUMAN Functional 5,6-difluoroindol-methylethylamine 758.578 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39586 5-HT2A CLONED HUMAN Functional Nor-d-fenfluramine 1047.13 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39587 5-HT2A CLONED HUMAN Functional ORG-37684 77.6247 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39588 5-HT2A CLONED HUMAN Functional DOI 0.891251 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39589 5-HT2A CLONED HUMAN Functional DOB 1.51356 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39590 5-HT2A CLONED HUMAN Functional LSD 21.3796 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39591 5-HT2A CLONED HUMAN Functional lisuride, (S) 6918.31 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39592 5-HT2A CLONED HUMAN Functional lisuride, R 1096.48 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39593 5-HT2A CLONED HUMAN Functional QUIPAZINE 309.03 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39594 5-HT2A CLONED HUMAN Functional 8-OH-DPAT,(-) >10000 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39595 5-HT2A CLONED HUMAN Functional RU 24969 81.2831 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39596 5-HT2A CLONED HUMAN Functional SCH 23390 13.1826 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39597 5-HT2B CLONED HUMAN Functional 5-Hydroxy Tryptamine 2.0893 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39598 5-HT2B CLONED HUMAN Functional 5-HT,a-Me 1.99526 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39599 5-HT2B CLONED HUMAN Functional TRYPTAMINE 29.5121 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39600 5-HT2B CLONED HUMAN Functional 5-CT 15.4882 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39601 5-HT2B CLONED HUMAN Functional 5-HT,20Me 169.824 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39602 5-HT2B CLONED HUMAN Functional mCPP 63.0957 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39603 5-HT2B CLONED HUMAN Functional TFMPP 288.403 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39604 5-HT2B CLONED HUMAN Functional ORG-12962 524.807 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39605 5-HT2B CLONED HUMAN Functional MK 212 295.121 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39606 5-HT2B CLONED HUMAN Functional Ro 60-0175 0.891251 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39607 5-HT2B CLONED HUMAN Functional 5,6-difluoroindol-methylethylamine 0.977237 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39608 5-HT2B CLONED HUMAN Functional Nor-d-fenfluramine 8.70964 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39609 5-HT2B CLONED HUMAN Functional ORG-37684 10.9648 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39610 5-HT2B CLONED HUMAN Functional DOI 1.41254 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39611 5-HT2B CLONED HUMAN Functional DOB 2.88403 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39612 5-HT2B CLONED HUMAN Functional LSD 8.91251 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39613 5-HT2B CLONED HUMAN Functional QUIPAZINE 177.828 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39614 5-HT2B CLONED HUMAN Functional 8-OH-DPAT,(-) 891.251 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39615 5-HT2B CLONED HUMAN Functional RU 24969 26.3027 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39616 5-HT2B CLONED HUMAN Functional SCH 23390 70.7946 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39617 5-HT2C CLONED HUMAN Functional 5-Hydroxy Tryptamine 5.7544 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39618 5-HT2C CLONED HUMAN Functional 5-HT,a-Me 11.4815 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39619 5-HT2C CLONED HUMAN Functional TRYPTAMINE 45.7088 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39620 5-HT2C CLONED HUMAN Functional 5-CT 407.38 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39621 5-HT2C CLONED HUMAN Functional 5-HT,20Me 1202.26 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39622 5-HT2C CLONED HUMAN Functional mCPP 81.2831 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39623 5-HT2C CLONED HUMAN Functional TFMPP 74.131 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39624 5-HT2C CLONED HUMAN Functional ORG-12962 97.7237 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39625 5-HT2C CLONED HUMAN Functional MK 212 213.796 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39626 5-HT2C CLONED HUMAN Functional Ro 60-0175 32.3594 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39627 5-HT2C CLONED HUMAN Functional 5,6-difluoroindol-methylethylamine 37.1535 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39628 5-HT2C CLONED HUMAN Functional Nor-d-fenfluramine 169.824 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39629 5-HT2C CLONED HUMAN Functional ORG-37684 6.76083 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39630 5-HT2C CLONED HUMAN Functional DOI 7.94328 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39631 5-HT2C CLONED HUMAN Functional DOB 7.76247 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39632 5-HT2C CLONED HUMAN Functional LSD 45.7088 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39633 5-HT2C CLONED HUMAN Functional QUIPAZINE 338.844 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39634 5-HT2C CLONED HUMAN Functional RU 24969 281.838 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39635 5-HT2C CLONED HUMAN Functional SCH 23390 40.738 Porter RH, et.al., 1999 Jan 15, 2025 Jan 15, 2025
39636 D1 STRIATUM RAT 3H-SCH23390 SCH 39166 3.6 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39637 D1 STRIATUM RAT 3H-SCH23390 SCH 23390 0.4 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39638 D1 STRIATUM RAT 3H-SCH23390 HALOPERIDOL 781 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39639 D2 STRIATUM RAT 3H-SPIPERONE SCH 39166 4268 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39640 D2 STRIATUM RAT 3H-SPIPERONE SCH 23390 359 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39641 D2 STRIATUM RAT 3H-SPIPERONE HALOPERIDOL 3.6 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39642 FR. CORTEX RAT 3H-KETANSERIN SCH 39166 320.8 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39643 FR. CORTEX RAT 3H-KETANSERIN SCH 23390 13.1 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39644 FR. CORTEX RAT 3H-KETANSERIN HALOPERIDOL 160.6 Chipkin RE, et al., 1988 Jan 15, 2025 Jan 15, 2025
39645 5-HT2B jugular vein RAT Functional BW-723C86 12.5893 Ellis ES, et al., 1995 Jan 15, 2025 Jan 15, 2025
39646 5-HT2A caudal artery RAT Functional BW-723C86 5011.87 Ellis ES, et al., 1995 Jan 15, 2025 Jan 15, 2025
39647 5-HT2C CLONED HUMAN Functional BW-723C86 316.228 Ellis ES, et al., 1995 Jan 15, 2025 Jan 15, 2025
39648 5-HT2C CLONED RAT UNDEFINED YOHIMBINE 5011.87 Ellis ES, et al., 1995 Jan 15, 2025 Jan 15, 2025
39649 5-HT2A CLONED HUMAN 125I-DOI 5-CT 316.228 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39650 5-HT2A CLONED HUMAN 125I-DOI 5-Hydroxy Tryptamine 16.2181 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39651 5-HT2A CLONED HUMAN 125I-DOI 8-OH-DPAT 2691.53 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39652 5-HT2A CLONED HUMAN 125I-DOI 5-HT,a-Me 15.8489 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39653 5-HT2A CLONED HUMAN 125I-DOI BW-723C86 63.0957 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39654 5-HT2A CLONED HUMAN 125I-DOI CGS 12066B 4265.8 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39655 5-HT2A CLONED HUMAN 125I-DOI LSD 0.758578 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39656 5-HT2A CLONED HUMAN 125I-DOI DOB 1.1749 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39657 5-HT2A CLONED HUMAN 125I-DOI DOI,(+) 0.933254 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39658 5-HT2A CLONED HUMAN 125I-DOI DOI,(-) 0.645654 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39659 5-HT2A CLONED HUMAN 125I-DOI ERGOTAMINE 0.977237 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39660 5-HT2A CLONED HUMAN 125I-DOI mCPP 54.9541 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39661 5-HT2A CLONED HUMAN 125I-DOI METHYLERGONOVINE 0.354813 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39662 5-HT2A CLONED HUMAN 125I-DOI MK 212 1023.29 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39663 5-HT2A CLONED HUMAN 125I-DOI ORG-12962 30.1995 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39664 5-HT2A CLONED HUMAN 125I-DOI ORG-37684 32.3594 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39665 5-HT2A CLONED HUMAN 125I-DOI PINDOLOL,(+/-) 9332.54 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39666 5-HT2A CLONED HUMAN 125I-DOI QUINPIROLE 3311.31 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39667 5-HT2A CLONED HUMAN 125I-DOI QUIPAZINE 128.825 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39668 5-HT2A CLONED HUMAN 125I-DOI Ro 60-0175 36.3078 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39669 5-HT2A CLONED HUMAN 125I-DOI RU 24969 125.893 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39670 5-HT2A CLONED HUMAN 125I-DOI TFMPP 31.6228 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39671 5-HT2A CLONED HUMAN 125I-DOI TRYPTAMINE 218.776 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39672 5-HT2A CLONED HUMAN 125I-DOI VER-3323 354.813 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39673 5-HT2B CLONED HUMAN 3H-5HT 5-CT 186.209 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39674 5-HT2B CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 13.4896 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39675 5-HT2B CLONED HUMAN 3H-5HT 8-OH-DPAT 4073.8 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39676 5-HT2B CLONED HUMAN 3H-5HT 5-HT,a-Me 6.91831 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39677 5-HT2B CLONED HUMAN 3H-5HT BW-723C86 46.7735 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39678 5-HT2B CLONED HUMAN 3H-5HT CGS 12066B 870.964 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39679 5-HT2B CLONED HUMAN 3H-5HT LSD 0.977237 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39680 5-HT2B CLONED HUMAN 3H-5HT DOB 43.6516 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39681 5-HT2B CLONED HUMAN 3H-5HT DOI,(+) 28.1838 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39682 5-HT2B CLONED HUMAN 3H-5HT DOI,(-) 53.7032 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39683 5-HT2B CLONED HUMAN 3H-5HT ERGOTAMINE 1.28825 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39684 5-HT2B CLONED HUMAN 3H-5HT mCPP 40.738 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39685 5-HT2B CLONED HUMAN 3H-5HT METHYLERGONOVINE 0.457088 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39686 5-HT2B CLONED HUMAN 3H-5HT MK 212 616.595 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39687 5-HT2B CLONED HUMAN 3H-5HT ORG-12962 91.2011 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39688 5-HT2B CLONED HUMAN 3H-5HT ORG-37684 42.658 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39689 5-HT2B CLONED HUMAN 3H-5HT PINDOLOL,(+/-) 2187.76 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39690 5-HT2B CLONED HUMAN 3H-5HT QUINPIROLE 301.995 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39691 5-HT2B CLONED HUMAN 3H-5HT QUIPAZINE 85.1138 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39692 5-HT2B CLONED HUMAN 3H-5HT Ro 60-0175 5.37032 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39693 5-HT2B CLONED HUMAN 3H-5HT RU 24969 134.896 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39694 5-HT2B CLONED HUMAN 3H-5HT TFMPP 58.8844 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39695 5-HT2B CLONED HUMAN 3H-5HT TRYPTAMINE 102.329 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39696 5-HT2B CLONED HUMAN 3H-5HT VER-3323 30.1995 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39697 5-HT2C CLONED HUMAN 3H-5HT 5-CT 204.174 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39698 5-HT2C CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 5.7544 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39699 5-HT2C CLONED HUMAN 3H-5HT 8-OH-DPAT 2511.89 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39700 5-HT2C CLONED HUMAN 3H-5HT 5-HT,a-Me 2.69153 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39701 5-HT2C CLONED HUMAN 3H-5HT BW-723C86 77.6247 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39702 5-HT2C CLONED HUMAN 3H-5HT CGS 12066B 2511.89 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39703 5-HT2C CLONED HUMAN 3H-5HT LSD 1.09648 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39704 5-HT2C CLONED HUMAN 3H-5HT DOB 6.30957 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39705 5-HT2C CLONED HUMAN 3H-5HT DOI,(+) 8.31764 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39706 5-HT2C CLONED HUMAN 3H-5HT DOI,(-) 5.37032 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39707 5-HT2C CLONED HUMAN 3H-5HT ERGOTAMINE 1.90546 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39708 5-HT2C CLONED HUMAN 3H-5HT mCPP 14.1254 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39709 5-HT2C CLONED HUMAN 3H-5HT METHYLERGONOVINE 4.57088 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39710 5-HT2C CLONED HUMAN 3H-5HT MK 212 97.7237 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39711 5-HT2C CLONED HUMAN 3H-5HT ORG-12962 14.7911 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39712 5-HT2C CLONED HUMAN 3H-5HT ORG-37684 7.58578 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39713 5-HT2C CLONED HUMAN 3H-5HT PINDOLOL,(+/-) >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39714 5-HT2C CLONED HUMAN 3H-5HT QUINPIROLE 3311.31 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39715 5-HT2C CLONED HUMAN 3H-5HT QUIPAZINE 53.7032 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39716 5-HT2C CLONED HUMAN 3H-5HT Ro 60-0175 6.0256 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39717 5-HT2C CLONED HUMAN 3H-5HT RU 24969 173.78 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39718 5-HT2C CLONED HUMAN 3H-5HT TFMPP 14.4544 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39719 5-HT2C CLONED HUMAN 3H-5HT TRYPTAMINE 2344.23 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39720 5-HT2C CLONED HUMAN 3H-5HT VER-3323 5.62341 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39721 5-HT2A CLONED HUMAN 125I-DOI d-Fenfluramine 3801.89 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39722 5-HT2A CLONED HUMAN 125I-DOI d-Norfenfluramine 151.356 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39723 5-HT2A CLONED HUMAN 125I-DOI FLUOXETINE 245.471 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39724 5-HT2A CLONED HUMAN 125I-DOI sibutramine >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39725 5-HT2A CLONED HUMAN 125I-DOI BTS 54 505 >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39726 5-HT2B CLONED HUMAN 3H-5HT d-Fenfluramine 5495.41 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39727 5-HT2B CLONED HUMAN 3H-5HT d-Norfenfluramine 100 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39728 5-HT2B CLONED HUMAN 3H-5HT FLUOXETINE >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39729 5-HT2B CLONED HUMAN 3H-5HT sibutramine >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39730 5-HT2B CLONED HUMAN 3H-5HT BTS 54 505 >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39731 5-HT2C CLONED HUMAN 3H-5HT d-Fenfluramine 1412.54 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39732 5-HT2C CLONED HUMAN 3H-5HT d-Norfenfluramine 51.2861 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39733 5-HT2C CLONED HUMAN 3H-5HT FLUOXETINE 398.107 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39734 5-HT2C CLONED HUMAN 3H-5HT sibutramine >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39735 5-HT2C CLONED HUMAN 3H-5HT BTS 54 505 >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39736 5-HT2A CLONED HUMAN 125I-DOI AMI-193 22.3872 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39737 5-HT2A CLONED HUMAN 125I-DOI CLOZAPINE 25.1189 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39738 5-HT2A CLONED HUMAN 125I-DOI KETANSERIN 8.12831 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39739 5-HT2A CLONED HUMAN 125I-DOI MDL 100907 1.86209 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39740 5-HT2A CLONED HUMAN 125I-DOI MDL 11,939 26.3027 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39741 5-HT2A CLONED HUMAN 125I-DOI MESULERGINE 45.7088 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39742 5-HT2A CLONED HUMAN 125I-DOI METERGOLINE 2.29087 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39743 5-HT2A CLONED HUMAN 125I-DOI METHIOTHEPIN 3.16228 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39744 5-HT2A CLONED HUMAN 125I-DOI METHYSERGIDE 3.98107 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39745 5-HT2A CLONED HUMAN 125I-DOI MIANSERIN 18.197 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39746 5-HT2A CLONED HUMAN 125I-DOI RITANSERIN 4.57088 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39747 5-HT2A CLONED HUMAN 125I-DOI RS-102221 2884.03 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39748 5-HT2A CLONED HUMAN 125I-DOI RS-127445 933.254 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39749 5-HT2A CLONED HUMAN 125I-DOI SB204741 >10000 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39750 5-HT2A CLONED HUMAN 125I-DOI SB 206553 2290.87 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39751 5-HT2A CLONED HUMAN 125I-DOI SB 221284 549.541 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39752 5-HT2A CLONED HUMAN 125I-DOI SB-224289 5011.87 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39753 5-HT2A CLONED HUMAN 125I-DOI SB 242084 851.138 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39754 5-HT2A CLONED HUMAN 125I-DOI SDZ SER-082 512.861 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39755 5-HT2A CLONED HUMAN 125I-DOI SPIPERONE 15.4882 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39756 5-HT2A CLONED HUMAN 125I-DOI TRAZODONE 44.6684 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39757 5-HT2B CLONED HUMAN 3H-5HT AMI-193 977.237 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39758 5-HT2B CLONED HUMAN 3H-5HT CLOZAPINE 10.2329 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39759 5-HT2B CLONED HUMAN 3H-5HT KETANSERIN 741.31 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39760 5-HT2B CLONED HUMAN 3H-5HT MDL 100907 1023.29 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39761 5-HT2B CLONED HUMAN 3H-5HT MDL 11,939 3311.31 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39762 5-HT2B CLONED HUMAN 3H-5HT MESULERGINE 3.46737 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39763 5-HT2B CLONED HUMAN 3H-5HT METERGOLINE 1.77828 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39764 5-HT2B CLONED HUMAN 3H-5HT METHIOTHEPIN 2.0893 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39765 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 0.363078 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39766 5-HT2B CLONED HUMAN 3H-5HT MIANSERIN 12.0226 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39767 5-HT2B CLONED HUMAN 3H-5HT RITANSERIN 2.13796 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39768 5-HT2B CLONED HUMAN 3H-5HT RS-102221 2884.03 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39769 5-HT2B CLONED HUMAN 3H-5HT RS-127445 1.07152 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39770 5-HT2B CLONED HUMAN 3H-5HT SB204741 125.893 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39771 5-HT2B CLONED HUMAN 3H-5HT SB 206553 22.3872 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39772 5-HT2B CLONED HUMAN 3H-5HT SB 221284 2.45471 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39773 5-HT2B CLONED HUMAN 3H-5HT SB-224289 1348.96 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39774 5-HT2B CLONED HUMAN 3H-5HT SB 242084 144.544 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39775 5-HT2B CLONED HUMAN 3H-5HT SDZ SER-082 204.174 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39776 5-HT2B CLONED HUMAN 3H-5HT SPIPERONE 1318.26 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39777 5-HT2B CLONED HUMAN 3H-5HT TRAZODONE 83.1764 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39778 5-HT2C CLONED HUMAN 3H-5HT AMI-193 1548.82 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39779 5-HT2C CLONED HUMAN 3H-5HT CLOZAPINE 13.4896 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39780 5-HT2C CLONED HUMAN 3H-5HT KETANSERIN 61.6595 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39781 5-HT2C CLONED HUMAN 3H-5HT MDL 100907 30.1995 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39782 5-HT2C CLONED HUMAN 3H-5HT MDL 11,939 263.027 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39783 5-HT2C CLONED HUMAN 3H-5HT MESULERGINE 1.8197 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39784 5-HT2C CLONED HUMAN 3H-5HT METERGOLINE 1.77828 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39785 5-HT2C CLONED HUMAN 3H-5HT METHIOTHEPIN 4.46684 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39786 5-HT2C CLONED HUMAN 3H-5HT METHYSERGIDE 4.46684 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39787 5-HT2C CLONED HUMAN 3H-5HT MIANSERIN 5.49541 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39788 5-HT2C CLONED HUMAN 3H-5HT RITANSERIN 6.60693 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39789 5-HT2C CLONED HUMAN 3H-5HT RS-102221 5.01187 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39790 5-HT2C CLONED HUMAN 3H-5HT RS-127445 467.735 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39791 5-HT2C CLONED HUMAN 3H-5HT SB204741 2754.23 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39792 5-HT2C CLONED HUMAN 3H-5HT SB 206553 16.2181 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39793 5-HT2C CLONED HUMAN 3H-5HT SB 221284 2.18776 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39794 5-HT2C CLONED HUMAN 3H-5HT SB-224289 1995.26 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39795 5-HT2C CLONED HUMAN 3H-5HT SB 242084 7.07946 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39796 5-HT2C CLONED HUMAN 3H-5HT SDZ SER-082 7.58578 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39797 5-HT2C CLONED HUMAN 3H-5HT SPIPERONE 602.56 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39798 5-HT2C CLONED HUMAN 3H-5HT TRAZODONE 223.872 Knight AR, et al., 2004 Jan 15, 2025 Jan 15, 2025
39799 CLONED HUMAN 3H-CCK8 Cyclosporin A 1200 Letschert K, et al., 2005 Jan 15, 2025 Jan 15, 2025
39800 CLONED HUMAN 3H-CCK8 Cyclosporin A >10000 Letschert K, et al., 2005 Jan 15, 2025 Jan 15, 2025
39801 CLONED HUMAN 3H-CCK8 MK 571 600 Letschert K, et al., 2005 Jan 15, 2025 Jan 15, 2025
39802 CLONED HUMAN 3H-CCK8 MK 571 8500 Letschert K, et al., 2005 Jan 15, 2025 Jan 15, 2025
39803 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-Hydroxy Tryptamine 18.197 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39804 5-HT2C CLONED HUMAN 3H-MESULERGINE mCPP 85.1138 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39805 5-HT2C CLONED HUMAN 3H-MESULERGINE MK 212 891.251 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39806 5-HT2C CLONED HUMAN 3H-MESULERGINE Ro 600332 13.8038 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39807 5-HT2C CLONED HUMAN 3H-MESULERGINE DOI 18.6209 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39808 5-HT2C CLONED HUMAN 3H-MESULERGINE BW-723C86 114.815 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39809 5-HT2C CLONED HUMAN 3H-MESULERGINE Ro 60-0175 26.9153 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39810 5-HT2C CLONED HUMAN 3H-MESULERGINE LISURIDE 6.45654 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39811 5-HT2C CLONED HUMAN 3H-MESULERGINE Ro 600869 2.75423 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39812 5-HT2B CLONED HUMAN 3H-MESULERGINE 5-Hydroxy Tryptamine 2.81838 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39813 5-HT2B CLONED HUMAN 3H-MESULERGINE mCPP 12.0226 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39814 5-HT2B CLONED HUMAN 3H-MESULERGINE MK 212 151.356 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39815 5-HT2B CLONED HUMAN 3H-MESULERGINE Ro 600332 15.8489 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39816 5-HT2B CLONED HUMAN 3H-MESULERGINE DOI 7.07946 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39817 5-HT2B CLONED HUMAN 3H-MESULERGINE BW-723C86 3.16228 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39818 5-HT2B CLONED HUMAN 3H-MESULERGINE Ro 60-0175 0.549541 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39819 5-HT2B CLONED HUMAN 3H-MESULERGINE LISURIDE 1.38038 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39820 5-HT2B CLONED HUMAN 3H-MESULERGINE Ro 600869 7.94328 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39821 5-HT2C CLONED HUMAN 3H-MESULERGINE RS-102221 1.47911 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39822 5-HT2C CLONED HUMAN 3H-MESULERGINE SB 242084 0.47863 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39823 5-HT2C CLONED HUMAN 3H-MESULERGINE KETANSERIN 16.9824 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39824 5-HT2C CLONED HUMAN 3H-MESULERGINE MESULERGINE 1.12202 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39825 5-HT2C CLONED HUMAN 3H-MESULERGINE METERGOLINE 0.467735 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39826 5-HT2C CLONED HUMAN 3H-MESULERGINE SB 206553 3.16228 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39827 5-HT2C CLONED HUMAN 3H-MESULERGINE MIANSERIN 1.51356 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39828 5-HT2C CLONED HUMAN 3H-MESULERGINE RITANSERIN 1.62181 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39829 5-HT2C CLONED HUMAN 3H-MESULERGINE SB-215505 11.2202 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39830 5-HT2C CLONED HUMAN 3H-MESULERGINE SB204741 2137.96 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39831 5-HT2C CLONED HUMAN 3H-MESULERGINE S33526 457.088 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39832 5-HT2C CLONED HUMAN 3H-MESULERGINE LY 266097 67.6083 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39833 5-HT2B CLONED HUMAN 3H-MESULERGINE RS-102221 234.423 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39834 5-HT2B CLONED HUMAN 3H-MESULERGINE SB 242084 45.7088 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39835 5-HT2B CLONED HUMAN 3H-MESULERGINE KETANSERIN 234.423 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39836 5-HT2B CLONED HUMAN 3H-MESULERGINE MESULERGINE 1.94984 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39837 5-HT2B CLONED HUMAN 3H-MESULERGINE METERGOLINE 0.707946 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39838 5-HT2B CLONED HUMAN 3H-MESULERGINE SB 206553 5.49541 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39839 5-HT2B CLONED HUMAN 3H-MESULERGINE MIANSERIN 5.49541 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39840 5-HT2B CLONED HUMAN 3H-MESULERGINE RITANSERIN 1.25893 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39841 5-HT2B CLONED HUMAN 3H-MESULERGINE SB-215505 1.47911 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39842 5-HT2B CLONED HUMAN 3H-MESULERGINE SB204741 51.2861 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39843 5-HT2B CLONED HUMAN 3H-MESULERGINE S33526 4.0738 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39844 5-HT2B CLONED HUMAN 3H-MESULERGINE LY 266097 0.199526 Cussac D, et al., 2002 Jan 15, 2025 Jan 15, 2025
39845 MOR CLONED HUMAN 3H-DAMGO MCL-145 200 Mathews JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39846 MOR CLONED HUMAN 3H-DAMGO MCL-101 230 Mathews JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39847 DOR CLONED HUMAN 3H-Naltrindole MCL-145 9400 Mathews JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39848 DOR CLONED HUMAN 3H-Naltrindole MCL-101 5900 Mathews JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39849 KOR CLONED HUMAN 3H-U69,593 MCL-145 78 Mathews JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39850 KOR CLONED HUMAN 3H-U69,593 MCL-101 79 Mathews JL, et al., 2005 Jan 15, 2025 Jan 15, 2025
39851 AT1 LIVER RAT 125I-Angiotensin II Angiotensin II 0.95 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39852 AT1 LIVER RAT 125I-Angiotensin II Ang II Sar1 0.16 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39853 AT1 LIVER RAT 125I-Angiotensin II Ang II 4-NH2-Phe6 >10000 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39854 AT1 LIVER RAT 125I-Angiotensin II C45H56N11O10 >10000 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39855 AT1 LIVER RAT 125I-Angiotensin II C51H67N12O11 >10000 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39856 AT1 LIVER RAT 125I-Angiotensin II C50H65N12O11 >10000 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39857 AT1 LIVER RAT 125I-Angiotensin II C44H54N11O10 >10000 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39858 AT1 LIVER RAT 125I-Angiotensin II C49H63N12O11 30.3 Georgsson J, et al., 2005 Jan 15, 2025 Jan 15, 2025
39859 AT2 Uterus PIG 125I-Angiotensin II Angiotensin II 0.2 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39860 AT2 Uterus PIG 125I-Angiotensin II Ang II Sar1 0.18 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39861 AT2 Uterus PIG 125I-Angiotensin II Ang II 4-NH2-Phe6 0.7 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39862 AT2 Uterus PIG 125I-Angiotensin II C45H56N11O10 10.1 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39863 AT2 Uterus PIG 125I-Angiotensin II C51H67N12O11 463.7 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39864 AT2 Uterus PIG 125I-Angiotensin II C50H65N12O11 1.85 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39865 AT2 Uterus PIG 125I-Angiotensin II C44H54N11O10 41.3 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39866 AT2 Uterus PIG 125I-Angiotensin II C49H63N12O11 9.8 Georgsson J, et al., 2005 Jan 15, 2025 Jan 28, 2025
39938 5-HT2B CLONED HUMAN UNDEFINED BW-723C86 79.4328 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39939 5-HT2B Stomach RAT Functional BW-723C86 12.5893 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39940 5-HT2C CLONED HUMAN Functional BW-723C86 501.187 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39941 5-HT2C UNDEFINED RAT UNDEFINED BW-723C86 125.893 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39942 5-HT2A CLONED HUMAN Functional BW-723C86 100 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39943 5-HT2A UNDEFINED RAT Functional BW-723C86 251.189 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39944 5-HT1A UNDEFINED RAT UNDEFINED BW-723C86 1258.93 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39945 5-HT1B UNDEFINED HUMAN UNDEFINED BW-723C86 125.893 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39946 5-HT1D UNDEFINED HUMAN UNDEFINED BW-723C86 630.957 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39947 5-HT1E UNDEFINED HUMAN UNDEFINED BW-723C86 3162.28 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39948 5-HT1F CLONED HUMAN UNDEFINED BW-723C86 7943.28 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39949 5-HT3 UNDEFINED RAT UNDEFINED BW-723C86 316.228 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39950 5-HT4 UNDEFINED RAT Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39951 5-HT7 CLONED HUMAN UNDEFINED BW-723C86 3162.28 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39952 5-HT7 CLONED RAT Functional BW-723C86 1000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39953 D1 UNDEFINED UNDEFINED UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39954 D2 UNDEFINED UNDEFINED UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39955 D4 CLONED HUMAN UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39956 UNDEFINED UNDEFINED Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39957 UNDEFINED UNDEFINED Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39958 Beta1 UNDEFINED UNDEFINED Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39959 Beta2 UNDEFINED UNDEFINED Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 28, 2025
39960 H1 UNDEFINED UNDEFINED Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39961 H2 UNDEFINED UNDEFINED Functional BW-723C86 >10000 Kennett GA, et al., 1996a Jan 15, 2025 Jan 15, 2025
39962 CEREBRAL CORTEX RAT 3H-PRAZOSIN FLUOXETINE 3981.07 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39963 CEREBRAL CORTEX RAT 3H-RX821002 FLUOXETINE 5011.87 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39964 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE FLUOXETINE 10 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39965 NET FR. CORTEX RAT 3H-Nisoxetine FLUOXETINE 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39966 CEREBRAL CORTEX RAT 3H-PRAZOSIN Napamezole 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39967 CEREBRAL CORTEX RAT 3H-RX821002 Napamezole 3.16228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39968 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Napamezole 199.526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39969 NET FR. CORTEX RAT 3H-Nisoxetine Napamezole 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39970 CEREBRAL CORTEX RAT 3H-PRAZOSIN ATIPAMEZOLE 1995.26 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39971 CEREBRAL CORTEX RAT 3H-RX821002 ATIPAMEZOLE 0.125893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39972 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE ATIPAMEZOLE 3162.28 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39973 NET FR. CORTEX RAT 3H-Nisoxetine ATIPAMEZOLE >10000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39974 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39975 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39976 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 39.8107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39977 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39978 CEREBRAL CORTEX RAT 3H-PRAZOSIN C14H15ClN2·C4H4O4 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39979 CEREBRAL CORTEX RAT 3H-RX821002 C14H15ClN2·C4H4O4 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39980 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C14H15ClN2·C4H4O4 19.9526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39981 NET FR. CORTEX RAT 3H-Nisoxetine C14H15ClN2·C4H4O4 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39982 CEREBRAL CORTEX RAT 3H-PRAZOSIN C14H15FN2·C4H4O4 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39983 CEREBRAL CORTEX RAT 3H-RX821002 C14H15FN2·C4H4O4 39.8107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39984 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C14H15FN2·C4H4O4 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39985 NET FR. CORTEX RAT 3H-Nisoxetine C14H15FN2·C4H4O4 125.893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39986 CEREBRAL CORTEX RAT 3H-PRAZOSIN C15H16N2O·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39987 CEREBRAL CORTEX RAT 3H-RX821002 C15H16N2O·C4H4O4 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39988 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H16N2O·C4H4O4 15.8489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39989 NET FR. CORTEX RAT 3H-Nisoxetine C15H16N2O·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39990 CEREBRAL CORTEX RAT 3H-PRAZOSIN C15H16N2·C4H4O4 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39991 CEREBRAL CORTEX RAT 3H-RX821002 C15H16N2·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39992 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H16N2·C4H4O4 12.5893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39993 NET FR. CORTEX RAT 3H-Nisoxetine C15H16N2·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39994 CEREBRAL CORTEX RAT 3H-PRAZOSIN C14H15FN2·C4H4O4 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39995 CEREBRAL CORTEX RAT 3H-RX821002 C14H15FN2·C4H4O4 199.526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39996 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C14H15FN2·C4H4O4 1.58489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39997 NET FR. CORTEX RAT 3H-Nisoxetine C14H15FN2·C4H4O4 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39998 CEREBRAL CORTEX RAT 3H-PRAZOSIN C15H15F3N2·C4H4O4 1258.93 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
39999 CEREBRAL CORTEX RAT 3H-RX821002 C15H15F3N2·C4H4O4 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40000 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H15F3N2·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40001 NET FR. CORTEX RAT 3H-Nisoxetine C15H15F3N2·C4H4O4 >10000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40002 CEREBRAL CORTEX RAT 3H-PRAZOSIN C15H18N2O·C4H4O4 2511.89 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40003 CEREBRAL CORTEX RAT 3H-RX821002 C15H18N2O·C4H4O4 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40004 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H18N2O·C4H4O4 199.526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40005 NET FR. CORTEX RAT 3H-Nisoxetine C15H18N2O·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40006 CEREBRAL CORTEX RAT 3H-PRAZOSIN C15H18N2·C4H4O4 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40007 CEREBRAL CORTEX RAT 3H-RX821002 C15H18N2·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40008 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H18N2·C4H4O4 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40009 NET FR. CORTEX RAT 3H-Nisoxetine C15H18N2·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40010 CEREBRAL CORTEX RAT 3H-RX821002 C15H18N2·C4H4O4 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40011 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H18N2·C4H4O4 15.8489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40012 NET FR. CORTEX RAT 3H-Nisoxetine C15H18N2·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40013 CEREBRAL CORTEX RAT 3H-PRAZOSIN 2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40014 CEREBRAL CORTEX RAT 3H-RX821002 2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate 316.228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40015 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate 39.8107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40016 NET FR. CORTEX RAT 3H-Nisoxetine 2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40017 CEREBRAL CORTEX RAT 3H-RX821002 2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40018 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40019 NET FR. CORTEX RAT 3H-Nisoxetine 2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40020 CEREBRAL CORTEX RAT 3H-RX821002 2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40021 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40022 NET FR. CORTEX RAT 3H-Nisoxetine 2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40023 CEREBRAL CORTEX RAT 3H-PRAZOSIN 2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 316.228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40024 CEREBRAL CORTEX RAT 3H-RX821002 2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40025 NET FR. CORTEX RAT 3H-Nisoxetine 2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40026 CEREBRAL CORTEX RAT 3H-PRAZOSIN 2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40027 CEREBRAL CORTEX RAT 3H-RX821002 2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 1584.89 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40028 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40029 NET FR. CORTEX RAT 3H-Nisoxetine 2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40030 CEREBRAL CORTEX RAT 3H-RX821002 2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate 1584.89 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40031 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40032 NET FR. CORTEX RAT 3H-Nisoxetine 2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40033 CEREBRAL CORTEX RAT 3H-PRAZOSIN C14H14N2·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40034 CEREBRAL CORTEX RAT 3H-RX821002 C14H14N2·C4H4O4 125.893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40035 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C14H14N2·C4H4O4 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40036 NET FR. CORTEX RAT 3H-Nisoxetine C14H14N2·C4H4O4 15.8489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40037 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40038 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40039 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40040 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 19.9526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40041 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40042 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate 15.8489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40043 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate 10 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40044 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40045 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H14N2O·C4H4O4 1584.89 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40046 CEREBRAL CORTEX RAT 3H-RX821002 C13H14N2O·C4H4O4 125.893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40047 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H14N2O·C4H4O4 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40048 NET FR. CORTEX RAT 3H-Nisoxetine C13H14N2O·C4H4O4 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40049 CEREBRAL CORTEX RAT 3H-PRAZOSIN C12H14N2O2·C4H4O4 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40050 CEREBRAL CORTEX RAT 3H-RX821002 C12H14N2O2·C4H4O4 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40051 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C12H14N2O2·C4H4O4 1258.93 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40052 NET FR. CORTEX RAT 3H-Nisoxetine C12H14N2O2·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40053 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H16N2O·C4H4O4 316.228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40054 CEREBRAL CORTEX RAT 3H-RX821002 C13H16N2O·C4H4O4 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40055 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H16N2O·C4H4O4 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40056 NET FR. CORTEX RAT 3H-Nisoxetine C13H16N2O·C4H4O4 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40057 CEREBRAL CORTEX RAT 3H-PRAZOSIN C16H20N2·0.5C4H4O4 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40058 CEREBRAL CORTEX RAT 3H-RX821002 C16H20N2·0.5C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40059 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C16H20N2·0.5C4H4O4 >10000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40060 NET FR. CORTEX RAT 3H-Nisoxetine C16H20N2·0.5C4H4O4 39.8107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40061 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H14N2·C4H4O4 1258.93 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40062 CEREBRAL CORTEX RAT 3H-RX821002 C13H14N2·C4H4O4 15.8489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40063 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H14N2·C4H4O4 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40064 NET FR. CORTEX RAT 3H-Nisoxetine C13H14N2·C4H4O4 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40065 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H16N2·0.5C4H4O4 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40066 CEREBRAL CORTEX RAT 3H-RX821002 C13H16N2·0.5C4H4O4 1.99526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40067 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H16N2·0.5C4H4O4 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40068 NET FR. CORTEX RAT 3H-Nisoxetine C13H16N2·0.5C4H4O4 39.8107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40069 CEREBRAL CORTEX RAT 3H-PRAZOSIN C12H12N2O·C4H4O4 2511.89 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40070 CEREBRAL CORTEX RAT 3H-RX821002 C12H12N2O·C4H4O4 12.5893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40071 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C12H12N2O·C4H4O4 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40072 NET FR. CORTEX RAT 3H-Nisoxetine C12H12N2O·C4H4O4 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40073 CEREBRAL CORTEX RAT 3H-RX821002 C12H11FN2O·C4H4O4 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40074 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C12H11FN2O·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40075 NET FR. CORTEX RAT 3H-Nisoxetine C12H11FN2O·C4H4O4 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40076 CEREBRAL CORTEX RAT 3H-PRAZOSIN C18H16N2O·C4H4O4 3162.28 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40077 CEREBRAL CORTEX RAT 3H-RX821002 C18H16N2O·C4H4O4 >10000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40078 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C18H16N2O·C4H4O4 >10000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40079 NET FR. CORTEX RAT 3H-Nisoxetine C18H16N2O·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40080 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H15FN2·0.5C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40081 CEREBRAL CORTEX RAT 3H-RX821002 C13H15FN2·0.5C4H4O4 1.25893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40082 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H15FN2·0.5C4H4O4 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40083 NET FR. CORTEX RAT 3H-Nisoxetine C13H15FN2·0.5C4H4O4 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40084 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H15FN2·0.5C4H4O4 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40085 CEREBRAL CORTEX RAT 3H-RX821002 C13H15FN2·0.5C4H4O4 7.94328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40086 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H15FN2·0.5C4H4O4 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40087 NET FR. CORTEX RAT 3H-Nisoxetine C13H15FN2·0.5C4H4O4 316.228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40088 CEREBRAL CORTEX RAT 3H-PRAZOSIN C13H14F2N2·0.5C4H4O4 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40089 CEREBRAL CORTEX RAT 3H-RX821002 C13H14F2N2·0.5C4H4O4 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40090 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C13H14F2N2·0.5C4H4O4 12.5893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40091 NET FR. CORTEX RAT 3H-Nisoxetine C13H14F2N2·0.5C4H4O4 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40092 CEREBRAL CORTEX RAT 3H-PRAZOSIN C15H20N2·C4H4O4 199.526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40093 CEREBRAL CORTEX RAT 3H-RX821002 C15H20N2·C4H4O4 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40094 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE C15H20N2·C4H4O4 19.9526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40095 NET FR. CORTEX RAT 3H-Nisoxetine C15H20N2·C4H4O4 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40096 CEREBRAL CORTEX RAT 3H-PRAZOSIN Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40097 CEREBRAL CORTEX RAT 3H-RX821002 Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 10 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40098 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 15.8489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40099 NET FR. CORTEX RAT 3H-Nisoxetine Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 199.526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40100 CEREBRAL CORTEX RAT 3H-PRAZOSIN Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40101 CEREBRAL CORTEX RAT 3H-RX821002 Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40102 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40103 NET FR. CORTEX RAT 3H-Nisoxetine Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40104 CEREBRAL CORTEX RAT 3H-PRAZOSIN Spiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate 5011.87 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40105 CEREBRAL CORTEX RAT 3H-RX821002 Spiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40106 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Spiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate 6309.57 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40107 NET FR. CORTEX RAT 3H-Nisoxetine Spiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate >10000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40108 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate 1258.93 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40109 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40110 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40111 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate 316.228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40112 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40113 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40114 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 10 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40115 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 199.526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40116 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 1995.26 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40117 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40118 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40119 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40120 CLONED HUMAN 3H-RX821002 Napamezole 6.30957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40121 CLONED HUMAN 3H-RX821002 ATIPAMEZOLE 3.16228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40122 CLONED HUMAN 3H-RX821002 4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40123 CLONED HUMAN 3H-RX821002 C14H15ClN2·C4H4O4 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40124 CLONED HUMAN 3H-RX821002 C14H15FN2·C4H4O4 39.8107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40125 CLONED HUMAN 3H-RX821002 C14H15FN2·C4H4O4 158.489 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40126 CLONED HUMAN 3H-RX821002 C14H14N2·C4H4O4 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40127 CLONED HUMAN 3H-RX821002 4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40128 CLONED HUMAN 3H-RX821002 C13H16N2·0.5C4H4O4 3.98107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40129 CLONED HUMAN 3H-RX821002 C12H12N2O·C4H4O4 19.9526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40130 CLONED HUMAN 3H-RX821002 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 63.0957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40131 CLONED HUMAN 3H-RX821002 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 3.16228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40132 CLONED HUMAN 3H-RX821002 Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate 1.25893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40133 NMDA CORTICAL MEMBRANES RAT 3H-CPP (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40134 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40135 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40136 NMDA CORTICAL MEMBRANES RAT 3H-CPP (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid 490 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40137 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40138 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40139 NMDA CORTICAL MEMBRANES RAT 3H-CPP (+/-)-AP5 290 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40140 NMDA CORTICAL MEMBRANES RAT 3H-CPP (R)-AP5 880 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40141 NMDA CORTICAL MEMBRANES RAT 3H-CPP (S)-AP5 >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40142 NMDA CORTICAL MEMBRANES RAT 3H-CPP (R)-CPPene 40 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40143 mGluR5 CLONED RAT UNDEFINED (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40144 mGluR5 CLONED RAT UNDEFINED (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40145 mGluR2 CLONED RAT Functional (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40146 mGluR4 CLONED RAT UNDEFINED (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40147 mGluR5 CLONED RAT UNDEFINED (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40148 mGluR5 CLONED RAT UNDEFINED (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40149 mGluR4 CLONED RAT UNDEFINED (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40150 mGluR5 CLONED RAT Functional (+/-)-trans-ACPD >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 15, 2025
40151 mGluR5 CLONED RAT Functional (+/-)-trans-ACPD >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40152 mGluR2 CLONED RAT Functional (+/-)-trans-ACPD 2000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40153 mGluR4 CLONED RAT Functional (+/-)-trans-ACPD >10000 Conti P, et al., 2003 Jan 15, 2025 Jan 28, 2025
40154 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluoroacetic Acid Salt 0.057 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40155 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluoroacetic Acid Salt 3.3 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40156 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.047 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40157 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 64 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40158 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.05 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40159 TNFα whole blood assay (WBA) HUMAN Functional 3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 17 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40160 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.15 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40161 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 42 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40162 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 16 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40163 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 250 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40164 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(propylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.97 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40165 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(propylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 158 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40166 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.61 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40167 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 4.6 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40168 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 0.42 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40169 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide 4.1 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40170 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 0.41 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40171 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 8.7 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40172 MAPK14 CLONED HUMAN Functional 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 1.6 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40173 TNFα whole blood assay (WBA) HUMAN Functional 3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 3.5 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40174 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide 0.057 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40175 TNFα whole blood assay (WBA) HUMAN Functional 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide 18 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40176 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 0.16 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40177 TNFα whole blood assay (WBA) HUMAN Functional 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide 1.5 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40178 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 1.5 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40179 TNFα whole blood assay (WBA) HUMAN Functional 3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 67 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40180 MAPK14 CLONED HUMAN Functional 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 1.9 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40181 TNFα whole blood assay (WBA) HUMAN Functional 3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide 21 Liu C, et al., 2005 Jan 15, 2025 Jan 15, 2025
40182 5-HT1A UNDEFINED RAT UNDEFINED mCPP 316.228 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40183 5-HT1B UNDEFINED RAT UNDEFINED mCPP 251.189 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40184 5-HT1D UNDEFINED RAT UNDEFINED mCPP 1584.89 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40185 5-HT2A UNDEFINED RAT UNDEFINED mCPP 199.526 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40186 5-HT2B UNDEFINED RAT UNDEFINED mCPP 25.1189 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40187 5-HT2C UNDEFINED RAT UNDEFINED mCPP 19.9526 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40188 5-HT3 UNDEFINED RAT UNDEFINED mCPP 100 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40189 5-HT6 UNDEFINED RAT UNDEFINED mCPP 2511.89 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40190 5-HT7 UNDEFINED RAT UNDEFINED mCPP 251.189 Martin RS, et al., 2001 Jan 15, 2025 Jan 15, 2025
40191 DP2 BRAIN RAT 3H-PGD2 PGD2 19 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40192 DP2 BRAIN RAT 3H-PGD2 PGD2-methyl ester 27 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40193 DP2 BRAIN RAT 3H-PGD2 PGD1 523 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40194 DP2 BRAIN RAT 3H-PGD2 PGF2Alpha 693 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40195 DP2 BRAIN RAT 3H-PGD2 PGE1 3758 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40196 DP2 BRAIN RAT 3H-PGD2 PGE2 2948 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40197 DP2 BRAIN RAT 3H-PGD2 PGI2 3537 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40198 DP2 BRAIN RAT 3H-PGD2 PG Thromboxane B2 4200 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40199 DP2 BRAIN RAT 3H-PGD2 PG 13,14-dihydro-15-keto-D2 >10000 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40200 DP2 BRAIN RAT 3H-PGD2 PGF1 alpha 6-keto >10000 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40201 DP2 BRAIN RAT 3H-PGD2 PGA2 >10000 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40202 DP2 BRAIN RAT 3H-PGD2 PGB2 >10000 Shimizu T, et al., 1982 Jan 15, 2025 Jan 15, 2025
40203 IP NCB-20 MOUSE 3H-PGI2 PGI2 16.6 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40204 IP NCB-20 MOUSE 3H-PGI2 PGE1 137 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40205 IP NCB-20 MOUSE 3H-PGI2 PGE1, 13,14-dihydro 315 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40206 IP NCB-20 MOUSE 3H-PGI2 PGE1, 8-iso 735 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40207 IP NCB-20 MOUSE 3H-PGI2 PGE2, 5,6-trans 735 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40208 IP NCB-20 MOUSE 3H-PGI2 PGE2,17-Phenyl 4370 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40209 IP NCB-20 MOUSE 3H-PGI2 PGI1, 6beta 7350 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40210 IP NCB-20 MOUSE 3H-PGI2 PGE2 >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40211 IP NCB-20 MOUSE 3H-PGI2 PGE2, 13,14-dihydro15-oxo >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40212 IP NCB-20 MOUSE 3H-PGI2 PGE2, 15-epi >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40213 IP NCB-20 MOUSE 3H-PGI2 PGF1alpha >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40214 IP NCB-20 MOUSE 3H-PGI2 PGF1alpha, 6-oxo >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40215 IP NCB-20 MOUSE 3H-PGI2 PGF2Alpha >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40216 IP NCB-20 MOUSE 3H-PGI2 PGD1 >10000 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40217 IP NCB-20 MOUSE 3H-PGI2 PGE2 13,14-dihydro 8410 MacDermot J, et al., 1981 Jan 15, 2025 Jan 28, 2025
40218 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 1258.93 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40219 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40220 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40221 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40222 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40223 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate 3162.28 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40224 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40225 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40226 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40227 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 630.957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40228 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 794.328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40229 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 3162.28 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40230 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40231 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40232 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 501.187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40233 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 6.30957 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40234 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 1.99526 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40235 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 100 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40236 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 1000 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40237 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 251.189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40238 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 25.1189 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40239 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40240 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 6309.57 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40241 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 79.4328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40242 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 398.107 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40243 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 316.228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40244 CEREBRAL CORTEX RAT 3H-PRAZOSIN 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 125.893 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40245 CEREBRAL CORTEX RAT 3H-RX821002 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 0.794328 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40246 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 50.1187 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40247 NET FR. CORTEX RAT 3H-Nisoxetine 4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate 31.6228 Cordi AA, et al., 2001 Jan 15, 2025 Jan 15, 2025
40248 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid 210 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40249 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40250 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40251 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid 960 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40252 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40253 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40254 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40255 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40256 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40257 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid 370 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40258 NMDA CORTICAL MEMBRANES RAT 3H-D-APV (-)-2-aminoadipic acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40259 NMDA CORTICAL MEMBRANES RAT 3H-CPP CGS 19755 95 Conti P, et al., 2004 Jan 15, 2025 Jan 28, 2025
40260 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40261 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2004 Jan 15, 2025 Jan 15, 2025
40262 5-HT2B CLONED HUMAN 3H-5HT METHYSERGIDE 7.94328 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40263 5-HT2B CLONED HUMAN 3H-5HT YOHIMBINE 398.107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40264 5-HT2B CLONED HUMAN 3H-5HT MIANSERIN 19.9526 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40265 5-HT2B CLONED HUMAN 3H-5HT SPIPERONE 1584.89 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40266 5-HT2B CLONED HUMAN 3H-5HT KETANSERIN 630.957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40267 5-HT2B CLONED HUMAN 3H-5HT RITANSERIN 5.01187 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40268 5-HT2B CLONED HUMAN 3H-5HT SB204741 79.4328 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40269 5-HT2B CLONED RAT 3H-5HT LY 53857 6.30957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40270 5-HT2B CLONED RAT 3H-5HT MESULERGINE 39.8107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40271 5-HT2B CLONED RAT 3H-5HT METHYSERGIDE 6.30957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40272 5-HT2B CLONED RAT 3H-5HT RAUWOLSCINE 39.8107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40273 5-HT2B CLONED RAT 3H-5HT YOHIMBINE 50.1187 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40274 5-HT2B CLONED RAT 3H-5HT MIANSERIN 50.1187 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40275 5-HT2B CLONED RAT 3H-5HT SPIPERONE 3162.28 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40276 5-HT2B CLONED RAT 3H-5HT KETANSERIN 3162.28 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40277 5-HT2B CLONED RAT 3H-5HT RITANSERIN 5.01187 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40278 5-HT2C Choroid Plexus PIG 3H-MESULERGINE LY 53857 7.94328 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40279 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MESULERGINE 1.58489 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40280 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHYSERGIDE 2.51189 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40281 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METERGOLINE 0.630957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40282 5-HT2C Choroid Plexus PIG 3H-MESULERGINE RAUWOLSCINE 1584.89 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40283 5-HT2C Choroid Plexus PIG 3H-MESULERGINE YOHIMBINE >10000 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40284 5-HT2C Choroid Plexus PIG 3H-MESULERGINE CHLORPROMAZINE 15.8489 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40285 5-HT2C Choroid Plexus PIG 3H-MESULERGINE MIANSERIN 10 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40286 5-HT2C Choroid Plexus PIG 3H-MESULERGINE SPIPERONE 1258.93 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40287 5-HT2C Choroid Plexus PIG 3H-MESULERGINE KETANSERIN 100 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40288 5-HT2C Choroid Plexus PIG 3H-MESULERGINE METHIOTHEPIN 25.1189 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40289 5-HT2C Choroid Plexus PIG 3H-MESULERGINE PIZOTIFEN 7.94328 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40290 5-HT2C Choroid Plexus PIG 3H-KETANSERIN RITANSERIN 2.51189 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40291 5-HT2C Choroid Plexus PIG 3H-MESULERGINE SB204741 1000 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40292 5-HT6 CLONED RAT 3H-LSD MESULERGINE 1584.89 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40293 5-HT6 CLONED RAT 3H-LSD METHYSERGIDE 398.107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40294 5-HT6 CLONED RAT 3H-LSD METERGOLINE 31.6228 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40295 5-HT6 CLONED RAT 3H-LSD AMITRIPTYLINE 63.0957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40296 5-HT6 CLONED RAT 3H-LSD AMOXAPINE 6.30957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40297 5-HT6 CLONED RAT 3H-LSD CHLORPROMAZINE 3.98107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40298 5-HT6 CLONED RAT 3H-LSD CHLORPROTHIXENE 3.16228 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40299 5-HT6 CLONED RAT 3H-LSD FLUPHENAZINE 15.8489 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40300 5-HT6 CLONED RAT 3H-LSD LOXAPINE 15.8489 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40301 5-HT6 CLONED RAT 3H-LSD MIANSERIN 50.1187 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40302 5-HT6 CLONED RAT 3H-LSD PERPHENAZINE 15.8489 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40303 5-HT6 CLONED RAT 3H-LSD SPIPERONE 1584.89 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40304 5-HT6 CLONED RAT 3H-LSD THIORIDAZINE 6.30957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40305 5-HT6 CLONED RAT 3H-LSD KETANSERIN >10000 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40306 5-HT6 CLONED RAT 3H-LSD METHIOTHEPIN 1.99526 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40307 5-HT6 CLONED RAT 3H-LSD RITANSERIN 39.8107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40308 5-HT7 CLONED RAT 3H-LSD MESULERGINE 6.30957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40309 5-HT7 CLONED RAT 3H-LSD METHYSERGIDE 12.5893 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40310 5-HT7 CLONED RAT 3H-LSD METERGOLINE 1.99526 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40311 5-HT7 CLONED RAT 3H-LSD AMITRIPTYLINE 125.893 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40312 5-HT7 CLONED RAT 3H-LSD AMOXAPINE 39.8107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40313 5-HT7 CLONED RAT 3H-LSD CHLORPROMAZINE 19.9526 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40314 5-HT7 CLONED RAT 3H-LSD CHLORPROTHIXENE 5.01187 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40315 5-HT7 CLONED RAT 3H-LSD FLUPHENAZINE 7.94328 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40316 5-HT7 CLONED RAT 3H-LSD LOXAPINE 39.8107 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40317 5-HT7 CLONED RAT 3H-LSD MIANSERIN 100 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40318 5-HT7 CLONED RAT 3H-LSD PERPHENAZINE 25.1189 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40319 5-HT7 CLONED RAT 3H-LSD SPIPERONE 10 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40320 5-HT7 CLONED RAT 3H-LSD THIORIDAZINE 63.0957 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40321 5-HT7 CLONED RAT 3H-LSD KETANSERIN 199.526 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40322 5-HT7 CLONED RAT 3H-LSD METHIOTHEPIN 1 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40323 5-HT7 CLONED RAT 3H-LSD RITANSERIN 19.9526 Glusa E, et al., 2000 Jan 15, 2025 Jan 15, 2025
40324 recombinant HUMAN Functional 6-phenylsulfonylpyridazin-2H-3-one 600 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40325 recombinant HUMAN Functional 6-(2-Bromobenzenesulfonyl)-2H-pyridazin-3-one 210 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40326 recombinant HUMAN Functional 6-(4-Bromobenzenesulfonyl)-2H-pyridazin-3-one 350 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40327 recombinant HUMAN Functional 6-(2-Chlorobenzenesulfonyl)-2H-pyridazin-3-one 170 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40328 recombinant HUMAN Functional 6-(3-Chlorobenzenesulfonyl)-2H-pyridazin-3-one 240 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40329 recombinant HUMAN Functional 6-(4-Chlorobenzenesulfonyl)-2H-pyridazin-3-one 380 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40330 recombinant HUMAN Functional 6-(2-Fluorobenzenesulfonyl)-2H-pyridazin-3-one 540 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40331 recombinant HUMAN Functional 6-(4-Fluorobenzenesulfonyl)-2H-pyridazin-3-one 474 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40332 recombinant HUMAN Functional 6-(4-Methoxybenzenesulfonyl)-2H-pyridazin-3-one 2000 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40333 recombinant HUMAN Functional 6-(Biphenylyl-2-sulfonyl)-2H-pyridazin-3-one 2200 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40334 recombinant HUMAN Functional 6-(2,3-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 55 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40335 recombinant HUMAN Functional 6-(2,4-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 190 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40336 recombinant HUMAN Functional 6-(2,5-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 73 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40337 recombinant HUMAN Functional 6-(2,6-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one 50 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40338 recombinant HUMAN Functional 6-(2,3-Difluorobenzenesulfonyl)-2H-pyridazin-3-one 390 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40339 recombinant HUMAN Functional 6-(2,4-Difluorobenzenesulfonyl)-2H-pyridazin-3-one 870 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40340 recombinant HUMAN Functional 6-(2-Chloro-4-fluorobenzenesulfonyl)-2H-pyridazin-3-one 280 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40341 recombinant HUMAN Functional 6-(4-Bromo-2-fluorobenzenesulfonyl)-2H-pyridazin-3-one 140 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40342 recombinant HUMAN Functional 6-(3-Trifluoromethylbenzenesulfonyl)-2H-pyridazin-3-one 175 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40343 recombinant HUMAN Functional 6-(4-Trifluoromethylbenzenesulfonyl)-2H-pyridazin-3-one 360 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40344 recombinant HUMAN Functional 6-(alpha-Naphthylmethylbenzenesulfonyl)-2H-pyridazin-3-one 150 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40345 recombinant HUMAN Functional 6-(beta-Naphthylmethylbenzenesulfonyl)-2H-pyridazin-3-one 360 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40346 recombinant HUMAN Functional sorbinil 140 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40347 recombinant HUMAN Functional zopolrestat 4 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40348 recombinant HUMAN Functional 6-(2-Cl-phenylmethanesulfonyl)-2H-pyridazin-3-one 118 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40349 recombinant HUMAN Functional 6-(2-F-phenylmethanesulfonyl)-2H-pyridazin-3-one 422 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40350 recombinant HUMAN Functional 6-(2-CF3-phenylmethanesulfonyl)-2H-pyridazin-3-one 500 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40351 recombinant HUMAN Functional 6-(3-CF3-phenylmethanesulfonyl-2H-pyridazin-3-one 72 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40352 recombinant HUMAN Functional 6-(2,3-Cl2-phenylmethanesulfonyl)-2H-pyridazin-3-one 35 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40353 recombinant HUMAN Functional 6-(2,6-Cl2-phenylmethanesulfonyl)-2H-pyridazin-3-one 52 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40354 recombinant HUMAN Functional 6-(2,3-F2-phenylmethanesulfonyl)-2H-pyridazin-3-one 257 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40355 recombinant HUMAN Functional 6-(2F,4Br-phenylmethanesulfonyl)-2H-pyridazin-3-one 667 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40356 recombinant HUMAN Functional 6-(2Cl,6F-phenylmethanesulfonyl)-2H-pyridazin-3-one 26 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40357 recombinant HUMAN Functional 6-(2F,3-Cl-phenylmethanesulfonyl)-2H-pyridazin-3-one 54 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40358 recombinant HUMAN Functional 6-(2F,3-CF3-phenylmethanesulfonyl)-2H-pyridazin-3-one 44 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40359 recombinant HUMAN Functional 6-(Indole-2-sulfonyl)-2H-pyridazin-3-one 590 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40360 recombinant HUMAN Functional 6-(5-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one 1100 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40361 recombinant HUMAN Functional 6-(6-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one 645 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40362 recombinant HUMAN Functional 6-(7-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one 450 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40363 recombinant HUMAN Functional 6-(6-Fluoroindole-2-sulfonyl)-2H-pyridazin-3-one 1400 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40364 recombinant HUMAN Functional 6-(5,6-Methylenedioxyindole-2-sulfonyl)-2H-pyridazin-3-one 3800 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40365 recombinant HUMAN Functional 6-(5,7-Dichloroindole-2-sulfonyl)-2H-pyridazin-3-one 200 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40366 recombinant HUMAN Functional 6-(Benzofuran-2-sulfonyl)-2H-pyridazin-3-one 150 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40367 recombinant HUMAN Functional 6-(5-Chlorobenzofuran-2-sulfonyl)-2H-pyridazin-3-one 25 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40368 recombinant HUMAN Functional 6-(3-Methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 140 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40369 recombinant HUMAN Functional 6-(5-Methoxybenzofuran-2-sulfonyl)-2H-pyridazin-3-one 230 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40370 recombinant HUMAN Functional 6-(5,7-Dichlorobenzofuran-2-sulfonyl)-2H-pyridazin-3-one 87 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40371 recombinant HUMAN Functional 6-(5-Chloro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 1 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40372 recombinant HUMAN Functional 6-(6-Chloro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 190 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40373 recombinant HUMAN Functional 6-(5-Fluoro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 3 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40374 recombinant HUMAN Functional 6-(3,5-Dimethylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 13 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40375 recombinant HUMAN Functional 6-(5-Chloro-3-ethylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 6 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40376 recombinant HUMAN Functional 6-(5-Chloro-3-isopropylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 92 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40377 recombinant HUMAN Functional 6-(3-Phenylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 23 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40378 recombinant HUMAN Functional 6-(3-[4-Fluorophenyl]benzofuran-2-methylsulfonyl)-2H-pyridazin-3-one 49 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40379 recombinant HUMAN Functional 6-(5-Chloro-3-phenylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one 34 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40380 recombinant HUMAN Functional 6-(Benzothiophene-2-sulfonyl)-2H-pyridazin-3-one 180 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40381 recombinant HUMAN Functional 6-(5-Methylbenzothiophene-2-sulfonyl)-2H-pyridazin-3-one 160 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40382 recombinant HUMAN Functional 6-(Benzothiazole-2-sulfonyl)-2H-pyridazin-3-one 450 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40383 recombinant HUMAN Functional 6-(5-Chloro-3-methylbenzothiophene-2-sulfonyl)-2H-pyridazin-3-one 55 Mylari BL, et al., 2005 Jan 15, 2025 Jan 15, 2025
40384 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-D-Pro-Gln-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40385 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-alphaMe-Pro-Gln-Thr-NH 1870 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40386 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-4-hydroxy-Pro-Gln-Thr-NH2 484 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40387 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-cis-3,4-methanoPro-Gln-Thr-NH2–1 265 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40388 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-cis-3,4-methanoPro-Gln-Thr-NH2–2 3110 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40389 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Azt-Gln-Thr-NH2 1660 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40390 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pip-Gln-Thr-NH2 1240 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40391 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Nip-Gln-Thr-NH2-1 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40392 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Nip-Gln-Thr-NH2-2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40393 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Inp-Gln-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40394 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Cmpi-Gln-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40395 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-1Ac6c-Gln-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40396 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gaba 1780 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40397 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Ahx 9780 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40398 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-3-carboxamidoanilide >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40399 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-3Ac6c-NH2 9810 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40400 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Nip-NH2 3020 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40401 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Inp-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40402 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Cmpi-NH2 1400 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40403 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-PyA-NH2 1690 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40404 LIVER RAT Functional 2-{1-[2,5-Di(trifluoromethyl)phenyl]methylidene}-6-methoxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40405 LIVER RAT Functional 6-Methoxy-2-[1-(2-methylphenyl)methylidene]-3,4-dihydro-2H-naphthlalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40406 LIVER RAT Functional 2-[1-(2-Bromophenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40407 LIVER RAT Functional 2-[1-(4-Hydroxyphenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40408 LIVER RAT Functional 6-Hydroxy-2-[1-(4-hydroxyphenyl)methylidene]-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40409 LIVER RAT Functional 2-{1-[4-(Dimethylamino)phenyl]methylidene}-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40410 LIVER RAT Functional 2-[1-(2-Bromophenyl)methylidene]-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one 2400 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40411 LIVER RAT Functional 2-Biphenyl-2-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40412 LIVER RAT Functional 2-Biphenyl-4-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40413 LIVER RAT Functional Ketoconazole >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40414 LIVER RAT Functional R 115866 9000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40415 MCF7 RAT Functional 2-{1-[2,5-Di(trifluoromethyl)phenyl]methylidene}-6-methoxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40416 MCF7 RAT Functional 6-Methoxy-2-[1-(2-methylphenyl)methylidene]-3,4-dihydro-2H-naphthlalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40417 MCF7 RAT Functional 2-[1-(2-Bromophenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 9000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40418 MCF7 RAT Functional 2-[1-(4-Hydroxyphenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one 7000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40419 MCF7 RAT Functional 6-Hydroxy-2-[1-(4-hydroxyphenyl)methylidene]-3,4-dihydro-2H-naphthalen-1-one 9000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40420 MCF7 RAT Functional 2-{1-[4-(Dimethylamino)phenyl]methylidene}-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40421 MCF7 RAT Functional 2-[1-(2-Bromophenyl)methylidene]-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40422 MCF7 RAT Functional 2-Biphenyl-2-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40423 MCF7 RAT Functional 2-Biphenyl-4-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40424 MCF7 RAT Functional Ketoconazole >10000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40425 MCF7 RAT Functional Liarozole 7000 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40426 MCF7 RAT Functional R 115866 5 Yee WS, et al., 2005 Jan 15, 2025 Jan 15, 2025
40427 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid 370 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40428 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40429 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40430 mGluR5 CLONED RAT Functional (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40431 mGluR4 CLONED RAT Functional (+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40432 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid 233 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40433 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40434 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40435 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid 210 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40436 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid 1900 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40437 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid 100 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40438 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid 960 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40439 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid 510 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40440 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid 2500 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40441 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40442 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40443 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40444 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40445 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40446 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40447 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40448 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40449 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40450 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40451 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40452 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40453 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40454 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40455 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40456 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40457 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40458 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40459 mGluR5 CLONED RAT Functional (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40460 mGluR5 CLONED RAT Functional (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40461 mGluR5 CLONED RAT Functional (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40462 mGluR5 CLONED RAT Functional (3aR,5R,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40463 mGluR5 CLONED RAT Functional (3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40464 mGluR5 CLONED RAT Functional (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40465 mGluR5 CLONED RAT Functional (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 15, 2025
40466 mGluR2 CLONED RAT Functional (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40467 mGluR2 CLONED RAT Functional (3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40468 mGluR2 CLONED RAT Functional (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40469 mGluR2 CLONED RAT Functional (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40470 mGluR4 CLONED RAT Functional (3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40471 mGluR4 CLONED RAT Functional (3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40472 mGluR4 CLONED RAT Functional (+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40473 mGluR4 CLONED RAT Functional (3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40474 mGluR4 CLONED RAT Functional (5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40475 mGluR4 CLONED RAT Functional (5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000 Conti P, et al., 2005 Jan 15, 2025 Jan 28, 2025
40476 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln-Thr-NH2 739 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40477 STAT3 CLONED HUMAN Functional Ac-pTyr-Val-Pro-Gln-Thr-NH2 1540 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40478 STAT3 CLONED HUMAN Functional Ac-pTyr-Ile-Pro-Gln-Thr-NH2 1070 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40479 STAT3 CLONED HUMAN Functional Ac-pTyr-Phe-Pro-Gln-Thr-NH2 1890 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40480 STAT3 CLONED HUMAN Functional Ac-pTyr-Cha-Pro-Gln-Thr-NH2 910 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40481 STAT3 CLONED HUMAN Functional Ac-pTyr-Nle-Pro-Gln-Thr-NH2 717 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40482 STAT3 CLONED HUMAN Functional Ac-pTyr-Phe2Ala-Pro-Gln-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40483 STAT3 CLONED HUMAN Functional Ac-pTyr-N-MeLeu-Pro-Gln-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40484 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Glu(Me)-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40485 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln(Me2)-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40486 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Met(O)-Thr-NH2 9870 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40487 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Met(O2)-Thr-NH2 >10000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40488 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln-NH2 856 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40489 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–NHMe 882 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40490 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–NHBn 409 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40491 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–NH(S)CHMePh 596 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40492 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–NH(R)CHMePh 801 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40493 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln-OH 748 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40494 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–NMe2 1850 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40495 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–NEt2 4220 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40496 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–pyrrolidine 2110 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40497 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln–piperidine 7000 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40498 STAT3 CLONED HUMAN Functional Ac-pTyr-Leu-Pro-Gln-N-MeThr-NH2 1220 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40499 STAT3 CLONED HUMAN Functional Benzoyl-pTyr-Leu -Pro-Gln-Thr-NH2 814 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40500 STAT3 CLONED HUMAN Functional Propionyl-pTyr-Leu -Pro-Gln-Thr-NH2 497 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40501 STAT3 CLONED HUMAN Functional Cbz-pTyr-Leu -Pro-Gln-Thr-NH2 750 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40502 STAT3 CLONED HUMAN Functional Dihydrocinnamoyl-pTyr-Leu-Pro-Gln-Thr-NH2 276 Coleman DR, et al., 2005 Jan 15, 2025 Jan 15, 2025
40503 5-HT2B CLONED HUMAN Functional BW-723C86 63.0957 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40504 5-HT2B CLONED RAT Functional BW-723C86 12.5893 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40505 5-HT2C CLONED HUMAN Functional BW-723C86 501.187 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40506 5-HT2C CLONED RAT UNDEFINED BW-723C86 125.893 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40507 5-HT2A CLONED HUMAN Functional BW-723C86 100 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40508 5-HT2A CLONED RAT UNDEFINED BW-723C86 251.189 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40509 5-HT1A CORTEX RAT UNDEFINED BW-723C86 1258.93 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40510 5-HT1B CLONED HUMAN UNDEFINED BW-723C86 125.893 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40511 5-HT1D CLONED HUMAN UNDEFINED BW-723C86 630.957 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40512 5-HT1E CLONED HUMAN UNDEFINED BW-723C86 3162.28 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40513 5-HT1F CLONED HUMAN 3H-5HT BW-723C86 7943.28 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40514 5-HT3 CORTEX RAT UNDEFINED BW-723C86 316.228 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40515 5-HT4 esophagus RAT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40516 5-HT6 CLONED HUMAN UNDEFINED BW-723C86 398.107 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40517 5-HT7 CLONED HUMAN 3H-5CT BW-723C86 3162.28 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40518 5-HT7 UNDEFINED RAT UNDEFINED BW-723C86 1000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40519 D1 STRIATUM RAT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40520 D2 STRIATUM RAT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40521 D4 CLONED HUMAN 3H-SPIPERONE BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40522 AORTA RABBIT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40523 vas deferens RAT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40524 Beta1 Right atrium GUINEA PIG UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40525 Beta2 jugular vein RABBIT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 28, 2025
40526 H1 trachea GUINEA PIG UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40527 H2 Saphenous vein RABBIT UNDEFINED BW-723C86 >10000 Kennett GA, et al., 1997a Jan 15, 2025 Jan 15, 2025
40528 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 14 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40529 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 20 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40530 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 15 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40531 GABAA CLONED HUMAN 3H-RO-15-1788 Zolpidem 27 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40532 GABAA CLONED HUMAN 3H-RO-15-1788 Zolpidem 160 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40533 GABAA CLONED HUMAN 3H-RO-15-1788 Zolpidem 380 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40534 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine 1.1 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40535 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine 2.9 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40536 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine 1.8 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40537 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine 0.78 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40538 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine 2.6 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40539 GABAA CLONED HUMAN 3H-RO-15-1788 3,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine 1.2 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40540 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 6.2 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40541 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 14 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40542 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 4.8 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40543 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.38 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40544 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.73 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40545 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.34 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40546 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.23 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40547 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.25 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40548 GABAA CLONED HUMAN 3H-RO-15-1788 7-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.17 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40549 GABAA CLONED HUMAN 3H-RO-15-1788 7-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.36 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40550 GABAA CLONED HUMAN 3H-RO-15-1788 7-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine 0.14 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40551 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine 0.27 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40552 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine 0.31 Carling RW, et al., 2005 Jan 15, 2025 Jan 27, 2025
40553 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine 0.2 Carling RW, et al., 2005 Jan 15, 2025 Jan 28, 2025
40554 UNDEFINED UNDEFINED Functional Phosphinothricin 600 Berlicki L, et al., 2005 Jan 15, 2025 Jan 15, 2025
40555 UNDEFINED UNDEFINED Functional (2S)-2-Amino-4-[(aminomethyl)(hydroxy)phosphinyl]butyric Acid 590 Berlicki L, et al., 2005 Jan 15, 2025 Jan 15, 2025
40556 UNDEFINED UNDEFINED Functional (2S)-2-Amino-4-[(hydroxymethyl)(hydroxy)phosphinyl]butyric Acid 2100 Berlicki L, et al., 2005 Jan 15, 2025 Jan 15, 2025