The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

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Showing 37,001-38,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
394865-HT2CCLONEDRAT3H-MESULERGINE4-Hydroxy-3-(2-[N-1,2,3,4 tetrahydroquinolino]ethyl)indole1446Sard H, et al., 2005Jan 15, 2025Jan 15, 2025
394875-HT2CCLONEDRAT3H-MESULERGINE4-Hydroxygramine49Sard H, et al., 2005Jan 15, 2025Jan 15, 2025
394885-HT2CCLONEDRAT3H-MESULERGINE1-(2-Dimethylaminoethyl)-4-hydroxyindole9351Sard H, et al., 2005Jan 15, 2025Jan 15, 2025
394895-HT4CLONEDHUMAN3H-GR-113808ML103025Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394905-HT4CLONEDHUMAN3H-GR-113808C36H50Cl2N6O9•0.75H2O), C, H, N19Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394915-HT4CLONEDHUMAN3H-GR-113808(C38H54Cl2N6O10•H2O), C, H, N3Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394925-HT4CLONEDHUMAN3H-GR-113808(C34H46Cl2N6O8•1.5H2O), C, H, N24Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394935-HT4CLONEDHUMAN3H-GR-113808(C35H48Cl2N6O8•2.5H2O), C, H, N31Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394945-HT4CLONEDHUMAN3H-GR-113808(C37H52Cl2N6O8), C, H, N7Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394955-HT4CLONEDHUMAN3H-GR-113808C42H62Cl2N6O8•0.75H2O), C, H, N20Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394965-HT4CLONEDHUMAN3H-GR-113808(C34H46Cl2N6O8•H2O), C, H, N21Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394975-HT4CLONEDHUMAN3H-GR-113808(C35H48Cl2N6O8), C, H, N5Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394985-HT4CLONEDHUMAN3H-GR-113808(C37H52Cl2N6O8•1.5H2O), C, H, N9Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
394995-HT4CLONEDHUMAN3H-GR-113808(C42H62Cl2N6O8•0.5H2O), C, H, N16Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
395005-HT4CLONEDHUMAN3H-GR-113808(C34H46Cl2N6O8•3H2O), C, H, N37Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
395015-HT4CLONEDHUMAN3H-GR-113808(C35H48Cl2N6O8•H2O), C, H, N13Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
395025-HT4CLONEDHUMAN3H-GR-113808(C37H52Cl2N6O8•2.5H2O), C, H, N5Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
395035-HT4CLONEDHUMAN3H-GR-113808(C42H62Cl2N6O8•1.5H2O), C, H, N8Soulier JL, et al., 2005Jan 15, 2025Jan 15, 2025
395045-HT6CLONEDHUMAN3H-LSD3-benzyl-N1-(N,N-dimethylaminoethyl)indole32Kolanos R, et al., 2005Jan 15, 2025Jan 15, 2025
395055-HT6CLONEDHUMAN3H-LSD1-benzyl-3-(N,N-dimethylaminoethyl)indene3Kolanos R, et al., 2005Jan 15, 2025Jan 15, 2025
395065-HT6CLONEDHUMAN3H-LSD3-(4-aminobenzyl)indene>10000Kolanos R, et al., 2005Jan 15, 2025Jan 15, 2025
395075-HT6CLONEDHUMAN3H-LSD1-(4-aminobenzyl)indene4470Kolanos R, et al., 2005Jan 15, 2025Jan 15, 2025
395085-HT6CLONEDHUMAN3H-LSD3-(4-aminobenzyl)indole2530Kolanos R, et al., 2005Jan 15, 2025Jan 15, 2025
39509S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid3.8Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39510S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid1.3Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39511S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid1.3Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39512S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid2.9Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39513S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid29Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39514S1P1CLONEDHUMAN35S-GTPGammaS1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid0.6Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39515S1P1CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid3.8Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39516S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid1.8Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39517S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid4.5Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39518S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid2.2Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39519S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid0.4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39520S1P1CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid1.4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39521S1P1CLONEDHUMAN35S-GTPGammaS1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid1.7Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39522S1P1CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid0.4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39523S1P1CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid0.9Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39524S1P1CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid0.8Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39525S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39526S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid3086Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39527S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39528S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39529S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39530S1P3CLONEDHUMAN35S-GTPGammaS1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39531S1P3CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39532S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39533S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39534S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39535S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39536S1P3CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39537S1P3CLONEDHUMAN35S-GTPGammaS1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39538S1P3CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39539S1P3CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid4282Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39540S1P3CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid4018Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39541SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid370Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39542SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid75Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39543SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid150Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39544SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid350Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39545SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid>10000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39546SIP4CLONEDHUMAN35S-GTPGammaS1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid70Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39547SIP4CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid90Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39548SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid370Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39549SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid1000Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39550SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid520Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39551SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid49Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39552SIP4CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid40Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39553SIP4CLONEDHUMAN35S-GTPGammaS1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid240Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39554SIP4CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid430Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39555SIP4CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid68Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39556SIP4CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid89Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39557S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid5.2Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39558S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-tert-butylphenyl)-1,3,4-oxadiazol-2-yl]benzyl}azetidine-3-carboxylic acid1.8Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39559S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-propylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid1.6Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39560S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-butyllphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid2.4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39561S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-hexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid6.4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39562S1P5CLONEDHUMAN35S-GTPGammaS1-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylic acid1Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39563S1P5CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(2,2-dimethylpropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid6.6Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39564S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid12Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39565S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopropylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid12Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39566S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclobutylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39567S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclopentylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid0.5Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39568S1P5CLONEDHUMAN35S-GTPGammaS1-{4-[5-(4-cyclohexylphenyl)-1,2,4-oxadiazol-3-yl]benzyl}azetidine-3-carboxylic acid0.8Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39569S1P5CLONEDHUMAN35S-GTPGammaS1-[[4-(5-[1,1'-biphenyl]-4-yl-1,2,4-oxadiazol-3-yl)phenyl]methyl]-3-azetidine-carboxylic acid11Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39570S1P5CLONEDHUMAN35S-GTPGammaS1-(4-{5-[4-(3,3,3-trifluoropropyl)phenyl]-1,2,4-oxadiazol-3-yl}benzyl)azetidine-3-carboxylic acid0.3Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39571S1P5CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1S)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid0.5Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
39572S1P5CLONEDHUMAN35S-GTPGammaS1-[4-(5-{4-[(1R)-3,3-difluorocyclopentyl]phenyl}-1,2,4-oxadiazol-3-yl)benzyl]-azetidine-3-carboxylic acid0.4Li Z, et al., 2005Jan 15, 2025Jan 15, 2025
395735-HT2ACLONEDHUMANFunctionalBW-723C86218.776Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395745-HT2BCLONEDHUMANFunctionalBW-723C861.07152Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395755-HT2CCLONEDHUMANFunctionalBW-723C8693.3254Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395765-HT2ACLONEDHUMANFunctional5-Hydroxy Tryptamine30.903Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395775-HT2ACLONEDHUMANFunctional5-HT,a-Me40.738Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395785-HT2ACLONEDHUMANFunctionalTRYPTAMINE257.04Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395795-HT2ACLONEDHUMANFunctional5-CT549.541Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395805-HT2ACLONEDHUMANFunctional5-HT,20Me2398.83Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395815-HT2ACLONEDHUMANFunctionalmCPP223.872Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395825-HT2ACLONEDHUMANFunctionalTFMPP162.181Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395835-HT2ACLONEDHUMANFunctionalORG-12962416.869Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395845-HT2ACLONEDHUMANFunctionalRo 60-0175446.684Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395855-HT2ACLONEDHUMANFunctional5,6-difluoroindol-methylethylamine758.578Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395865-HT2ACLONEDHUMANFunctionalNor-d-fenfluramine1047.13Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395875-HT2ACLONEDHUMANFunctionalORG-3768477.6247Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395885-HT2ACLONEDHUMANFunctionalDOI0.891251Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395895-HT2ACLONEDHUMANFunctionalDOB1.51356Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395905-HT2ACLONEDHUMANFunctionalLSD21.3796Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395915-HT2ACLONEDHUMANFunctionallisuride, (S)6918.31Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395925-HT2ACLONEDHUMANFunctionallisuride, R1096.48Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395935-HT2ACLONEDHUMANFunctionalQUIPAZINE309.03Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395945-HT2ACLONEDHUMANFunctional8-OH-DPAT,(-)>10000Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395955-HT2ACLONEDHUMANFunctionalRU 2496981.2831Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395965-HT2ACLONEDHUMANFunctionalSCH 2339013.1826Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395975-HT2BCLONEDHUMANFunctional5-Hydroxy Tryptamine2.0893Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395985-HT2BCLONEDHUMANFunctional5-HT,a-Me1.99526Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
395995-HT2BCLONEDHUMANFunctionalTRYPTAMINE29.5121Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396005-HT2BCLONEDHUMANFunctional5-CT15.4882Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396015-HT2BCLONEDHUMANFunctional5-HT,20Me169.824Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396025-HT2BCLONEDHUMANFunctionalmCPP63.0957Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396035-HT2BCLONEDHUMANFunctionalTFMPP288.403Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396045-HT2BCLONEDHUMANFunctionalORG-12962524.807Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396055-HT2BCLONEDHUMANFunctionalMK 212295.121Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396065-HT2BCLONEDHUMANFunctionalRo 60-01750.891251Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396075-HT2BCLONEDHUMANFunctional5,6-difluoroindol-methylethylamine0.977237Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396085-HT2BCLONEDHUMANFunctionalNor-d-fenfluramine8.70964Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396095-HT2BCLONEDHUMANFunctionalORG-3768410.9648Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396105-HT2BCLONEDHUMANFunctionalDOI1.41254Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396115-HT2BCLONEDHUMANFunctionalDOB2.88403Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396125-HT2BCLONEDHUMANFunctionalLSD8.91251Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396135-HT2BCLONEDHUMANFunctionalQUIPAZINE177.828Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396145-HT2BCLONEDHUMANFunctional8-OH-DPAT,(-)891.251Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396155-HT2BCLONEDHUMANFunctionalRU 2496926.3027Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396165-HT2BCLONEDHUMANFunctionalSCH 2339070.7946Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396175-HT2CCLONEDHUMANFunctional5-Hydroxy Tryptamine5.7544Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396185-HT2CCLONEDHUMANFunctional5-HT,a-Me11.4815Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396195-HT2CCLONEDHUMANFunctionalTRYPTAMINE45.7088Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396205-HT2CCLONEDHUMANFunctional5-CT407.38Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396215-HT2CCLONEDHUMANFunctional5-HT,20Me1202.26Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396225-HT2CCLONEDHUMANFunctionalmCPP81.2831Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396235-HT2CCLONEDHUMANFunctionalTFMPP74.131Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396245-HT2CCLONEDHUMANFunctionalORG-1296297.7237Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396255-HT2CCLONEDHUMANFunctionalMK 212213.796Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396265-HT2CCLONEDHUMANFunctionalRo 60-017532.3594Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396275-HT2CCLONEDHUMANFunctional5,6-difluoroindol-methylethylamine37.1535Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396285-HT2CCLONEDHUMANFunctionalNor-d-fenfluramine169.824Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396295-HT2CCLONEDHUMANFunctionalORG-376846.76083Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396305-HT2CCLONEDHUMANFunctionalDOI7.94328Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396315-HT2CCLONEDHUMANFunctionalDOB7.76247Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396325-HT2CCLONEDHUMANFunctionalLSD45.7088Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396335-HT2CCLONEDHUMANFunctionalQUIPAZINE338.844Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396345-HT2CCLONEDHUMANFunctionalRU 24969281.838Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
396355-HT2CCLONEDHUMANFunctionalSCH 2339040.738Porter RH, et.al., 1999Jan 15, 2025Jan 15, 2025
39636D1STRIATUMRAT3H-SCH23390SCH 391663.6Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39637D1STRIATUMRAT3H-SCH23390SCH 233900.4Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39638D1STRIATUMRAT3H-SCH23390HALOPERIDOL781Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39639D2STRIATUMRAT3H-SPIPERONESCH 391664268Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39640D2STRIATUMRAT3H-SPIPERONESCH 23390359Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39641D2STRIATUMRAT3H-SPIPERONEHALOPERIDOL3.6Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39642FR. CORTEXRAT3H-KETANSERINSCH 39166320.8Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39643FR. CORTEXRAT3H-KETANSERINSCH 2339013.1Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
39644FR. CORTEXRAT3H-KETANSERINHALOPERIDOL160.6Chipkin RE, et al., 1988Jan 15, 2025Jan 15, 2025
396455-HT2Bjugular veinRATFunctionalBW-723C8612.5893Ellis ES, et al., 1995Jan 15, 2025Jan 15, 2025
396465-HT2Acaudal arteryRATFunctionalBW-723C865011.87Ellis ES, et al., 1995Jan 15, 2025Jan 15, 2025
396475-HT2CCLONEDHUMANFunctionalBW-723C86316.228Ellis ES, et al., 1995Jan 15, 2025Jan 15, 2025
396485-HT2CCLONEDRATUNDEFINEDYOHIMBINE5011.87Ellis ES, et al., 1995Jan 15, 2025Jan 15, 2025
396495-HT2ACLONEDHUMAN125I-DOI5-CT316.228Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396505-HT2ACLONEDHUMAN125I-DOI5-Hydroxy Tryptamine16.2181Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396515-HT2ACLONEDHUMAN125I-DOI8-OH-DPAT2691.53Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396525-HT2ACLONEDHUMAN125I-DOI5-HT,a-Me15.8489Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396535-HT2ACLONEDHUMAN125I-DOIBW-723C8663.0957Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396545-HT2ACLONEDHUMAN125I-DOICGS 12066B4265.8Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396555-HT2ACLONEDHUMAN125I-DOILSD0.758578Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396565-HT2ACLONEDHUMAN125I-DOIDOB1.1749Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396575-HT2ACLONEDHUMAN125I-DOIDOI,(+)0.933254Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396585-HT2ACLONEDHUMAN125I-DOIDOI,(-)0.645654Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396595-HT2ACLONEDHUMAN125I-DOIERGOTAMINE0.977237Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396605-HT2ACLONEDHUMAN125I-DOImCPP54.9541Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396615-HT2ACLONEDHUMAN125I-DOIMETHYLERGONOVINE0.354813Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396625-HT2ACLONEDHUMAN125I-DOIMK 2121023.29Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396635-HT2ACLONEDHUMAN125I-DOIORG-1296230.1995Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396645-HT2ACLONEDHUMAN125I-DOIORG-3768432.3594Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396655-HT2ACLONEDHUMAN125I-DOIPINDOLOL,(+/-)9332.54Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396665-HT2ACLONEDHUMAN125I-DOIQUINPIROLE3311.31Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396675-HT2ACLONEDHUMAN125I-DOIQUIPAZINE128.825Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396685-HT2ACLONEDHUMAN125I-DOIRo 60-017536.3078Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396695-HT2ACLONEDHUMAN125I-DOIRU 24969125.893Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396705-HT2ACLONEDHUMAN125I-DOITFMPP31.6228Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396715-HT2ACLONEDHUMAN125I-DOITRYPTAMINE218.776Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396725-HT2ACLONEDHUMAN125I-DOIVER-3323354.813Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396735-HT2BCLONEDHUMAN3H-5HT5-CT186.209Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396745-HT2BCLONEDHUMAN3H-5HT5-Hydroxy Tryptamine13.4896Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396755-HT2BCLONEDHUMAN3H-5HT8-OH-DPAT4073.8Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396765-HT2BCLONEDHUMAN3H-5HT5-HT,a-Me6.91831Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396775-HT2BCLONEDHUMAN3H-5HTBW-723C8646.7735Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396785-HT2BCLONEDHUMAN3H-5HTCGS 12066B870.964Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396795-HT2BCLONEDHUMAN3H-5HTLSD0.977237Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396805-HT2BCLONEDHUMAN3H-5HTDOB43.6516Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396815-HT2BCLONEDHUMAN3H-5HTDOI,(+)28.1838Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396825-HT2BCLONEDHUMAN3H-5HTDOI,(-)53.7032Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396835-HT2BCLONEDHUMAN3H-5HTERGOTAMINE1.28825Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396845-HT2BCLONEDHUMAN3H-5HTmCPP40.738Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396855-HT2BCLONEDHUMAN3H-5HTMETHYLERGONOVINE0.457088Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396865-HT2BCLONEDHUMAN3H-5HTMK 212616.595Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396875-HT2BCLONEDHUMAN3H-5HTORG-1296291.2011Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396885-HT2BCLONEDHUMAN3H-5HTORG-3768442.658Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396895-HT2BCLONEDHUMAN3H-5HTPINDOLOL,(+/-)2187.76Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396905-HT2BCLONEDHUMAN3H-5HTQUINPIROLE301.995Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396915-HT2BCLONEDHUMAN3H-5HTQUIPAZINE85.1138Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396925-HT2BCLONEDHUMAN3H-5HTRo 60-01755.37032Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396935-HT2BCLONEDHUMAN3H-5HTRU 24969134.896Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396945-HT2BCLONEDHUMAN3H-5HTTFMPP58.8844Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396955-HT2BCLONEDHUMAN3H-5HTTRYPTAMINE102.329Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396965-HT2BCLONEDHUMAN3H-5HTVER-332330.1995Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396975-HT2CCLONEDHUMAN3H-5HT5-CT204.174Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396985-HT2CCLONEDHUMAN3H-5HT5-Hydroxy Tryptamine5.7544Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
396995-HT2CCLONEDHUMAN3H-5HT8-OH-DPAT2511.89Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397005-HT2CCLONEDHUMAN3H-5HT5-HT,a-Me2.69153Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397015-HT2CCLONEDHUMAN3H-5HTBW-723C8677.6247Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397025-HT2CCLONEDHUMAN3H-5HTCGS 12066B2511.89Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397035-HT2CCLONEDHUMAN3H-5HTLSD1.09648Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397045-HT2CCLONEDHUMAN3H-5HTDOB6.30957Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397055-HT2CCLONEDHUMAN3H-5HTDOI,(+)8.31764Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397065-HT2CCLONEDHUMAN3H-5HTDOI,(-)5.37032Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397075-HT2CCLONEDHUMAN3H-5HTERGOTAMINE1.90546Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397085-HT2CCLONEDHUMAN3H-5HTmCPP14.1254Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397095-HT2CCLONEDHUMAN3H-5HTMETHYLERGONOVINE4.57088Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397105-HT2CCLONEDHUMAN3H-5HTMK 21297.7237Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397115-HT2CCLONEDHUMAN3H-5HTORG-1296214.7911Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397125-HT2CCLONEDHUMAN3H-5HTORG-376847.58578Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397135-HT2CCLONEDHUMAN3H-5HTPINDOLOL,(+/-)>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397145-HT2CCLONEDHUMAN3H-5HTQUINPIROLE3311.31Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397155-HT2CCLONEDHUMAN3H-5HTQUIPAZINE53.7032Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397165-HT2CCLONEDHUMAN3H-5HTRo 60-01756.0256Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397175-HT2CCLONEDHUMAN3H-5HTRU 24969173.78Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397185-HT2CCLONEDHUMAN3H-5HTTFMPP14.4544Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397195-HT2CCLONEDHUMAN3H-5HTTRYPTAMINE2344.23Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397205-HT2CCLONEDHUMAN3H-5HTVER-33235.62341Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397215-HT2ACLONEDHUMAN125I-DOId-Fenfluramine3801.89Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397225-HT2ACLONEDHUMAN125I-DOId-Norfenfluramine151.356Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397235-HT2ACLONEDHUMAN125I-DOIFLUOXETINE245.471Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397245-HT2ACLONEDHUMAN125I-DOIsibutramine>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397255-HT2ACLONEDHUMAN125I-DOIBTS 54 505>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397265-HT2BCLONEDHUMAN3H-5HTd-Fenfluramine5495.41Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397275-HT2BCLONEDHUMAN3H-5HTd-Norfenfluramine100Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397285-HT2BCLONEDHUMAN3H-5HTFLUOXETINE>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397295-HT2BCLONEDHUMAN3H-5HTsibutramine>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397305-HT2BCLONEDHUMAN3H-5HTBTS 54 505>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397315-HT2CCLONEDHUMAN3H-5HTd-Fenfluramine1412.54Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397325-HT2CCLONEDHUMAN3H-5HTd-Norfenfluramine51.2861Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397335-HT2CCLONEDHUMAN3H-5HTFLUOXETINE398.107Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397345-HT2CCLONEDHUMAN3H-5HTsibutramine>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397355-HT2CCLONEDHUMAN3H-5HTBTS 54 505>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397365-HT2ACLONEDHUMAN125I-DOIAMI-19322.3872Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397375-HT2ACLONEDHUMAN125I-DOICLOZAPINE25.1189Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397385-HT2ACLONEDHUMAN125I-DOIKETANSERIN8.12831Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397395-HT2ACLONEDHUMAN125I-DOIMDL 1009071.86209Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397405-HT2ACLONEDHUMAN125I-DOIMDL 11,93926.3027Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397415-HT2ACLONEDHUMAN125I-DOIMESULERGINE45.7088Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397425-HT2ACLONEDHUMAN125I-DOIMETERGOLINE2.29087Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397435-HT2ACLONEDHUMAN125I-DOIMETHIOTHEPIN3.16228Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397445-HT2ACLONEDHUMAN125I-DOIMETHYSERGIDE3.98107Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397455-HT2ACLONEDHUMAN125I-DOIMIANSERIN18.197Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397465-HT2ACLONEDHUMAN125I-DOIRITANSERIN4.57088Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397475-HT2ACLONEDHUMAN125I-DOIRS-1022212884.03Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397485-HT2ACLONEDHUMAN125I-DOIRS-127445933.254Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397495-HT2ACLONEDHUMAN125I-DOISB204741>10000Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397505-HT2ACLONEDHUMAN125I-DOISB 2065532290.87Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397515-HT2ACLONEDHUMAN125I-DOISB 221284549.541Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397525-HT2ACLONEDHUMAN125I-DOISB-2242895011.87Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397535-HT2ACLONEDHUMAN125I-DOISB 242084851.138Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397545-HT2ACLONEDHUMAN125I-DOISDZ SER-082512.861Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397555-HT2ACLONEDHUMAN125I-DOISPIPERONE15.4882Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397565-HT2ACLONEDHUMAN125I-DOITRAZODONE44.6684Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397575-HT2BCLONEDHUMAN3H-5HTAMI-193977.237Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397585-HT2BCLONEDHUMAN3H-5HTCLOZAPINE10.2329Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397595-HT2BCLONEDHUMAN3H-5HTKETANSERIN741.31Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397605-HT2BCLONEDHUMAN3H-5HTMDL 1009071023.29Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397615-HT2BCLONEDHUMAN3H-5HTMDL 11,9393311.31Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397625-HT2BCLONEDHUMAN3H-5HTMESULERGINE3.46737Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397635-HT2BCLONEDHUMAN3H-5HTMETERGOLINE1.77828Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397645-HT2BCLONEDHUMAN3H-5HTMETHIOTHEPIN2.0893Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397655-HT2BCLONEDHUMAN3H-5HTMETHYSERGIDE0.363078Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397665-HT2BCLONEDHUMAN3H-5HTMIANSERIN12.0226Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397675-HT2BCLONEDHUMAN3H-5HTRITANSERIN2.13796Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397685-HT2BCLONEDHUMAN3H-5HTRS-1022212884.03Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397695-HT2BCLONEDHUMAN3H-5HTRS-1274451.07152Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397705-HT2BCLONEDHUMAN3H-5HTSB204741125.893Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397715-HT2BCLONEDHUMAN3H-5HTSB 20655322.3872Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397725-HT2BCLONEDHUMAN3H-5HTSB 2212842.45471Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397735-HT2BCLONEDHUMAN3H-5HTSB-2242891348.96Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397745-HT2BCLONEDHUMAN3H-5HTSB 242084144.544Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397755-HT2BCLONEDHUMAN3H-5HTSDZ SER-082204.174Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397765-HT2BCLONEDHUMAN3H-5HTSPIPERONE1318.26Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397775-HT2BCLONEDHUMAN3H-5HTTRAZODONE83.1764Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397785-HT2CCLONEDHUMAN3H-5HTAMI-1931548.82Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397795-HT2CCLONEDHUMAN3H-5HTCLOZAPINE13.4896Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397805-HT2CCLONEDHUMAN3H-5HTKETANSERIN61.6595Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397815-HT2CCLONEDHUMAN3H-5HTMDL 10090730.1995Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397825-HT2CCLONEDHUMAN3H-5HTMDL 11,939263.027Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397835-HT2CCLONEDHUMAN3H-5HTMESULERGINE1.8197Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397845-HT2CCLONEDHUMAN3H-5HTMETERGOLINE1.77828Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397855-HT2CCLONEDHUMAN3H-5HTMETHIOTHEPIN4.46684Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397865-HT2CCLONEDHUMAN3H-5HTMETHYSERGIDE4.46684Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397875-HT2CCLONEDHUMAN3H-5HTMIANSERIN5.49541Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397885-HT2CCLONEDHUMAN3H-5HTRITANSERIN6.60693Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397895-HT2CCLONEDHUMAN3H-5HTRS-1022215.01187Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397905-HT2CCLONEDHUMAN3H-5HTRS-127445467.735Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397915-HT2CCLONEDHUMAN3H-5HTSB2047412754.23Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397925-HT2CCLONEDHUMAN3H-5HTSB 20655316.2181Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397935-HT2CCLONEDHUMAN3H-5HTSB 2212842.18776Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397945-HT2CCLONEDHUMAN3H-5HTSB-2242891995.26Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397955-HT2CCLONEDHUMAN3H-5HTSB 2420847.07946Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397965-HT2CCLONEDHUMAN3H-5HTSDZ SER-0827.58578Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397975-HT2CCLONEDHUMAN3H-5HTSPIPERONE602.56Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
397985-HT2CCLONEDHUMAN3H-5HTTRAZODONE223.872Knight AR, et al., 2004Jan 15, 2025Jan 15, 2025
39799CLONEDHUMAN3H-CCK8Cyclosporin A1200Letschert K, et al., 2005Jan 15, 2025Jan 15, 2025
39800CLONEDHUMAN3H-CCK8Cyclosporin A>10000Letschert K, et al., 2005Jan 15, 2025Jan 15, 2025
39801CLONEDHUMAN3H-CCK8MK 571600Letschert K, et al., 2005Jan 15, 2025Jan 15, 2025
39802CLONEDHUMAN3H-CCK8MK 5718500Letschert K, et al., 2005Jan 15, 2025Jan 15, 2025
398035-HT2CCLONEDHUMAN3H-MESULERGINE5-Hydroxy Tryptamine18.197Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398045-HT2CCLONEDHUMAN3H-MESULERGINEmCPP85.1138Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398055-HT2CCLONEDHUMAN3H-MESULERGINEMK 212891.251Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398065-HT2CCLONEDHUMAN3H-MESULERGINERo 60033213.8038Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398075-HT2CCLONEDHUMAN3H-MESULERGINEDOI18.6209Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398085-HT2CCLONEDHUMAN3H-MESULERGINEBW-723C86114.815Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398095-HT2CCLONEDHUMAN3H-MESULERGINERo 60-017526.9153Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398105-HT2CCLONEDHUMAN3H-MESULERGINELISURIDE6.45654Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398115-HT2CCLONEDHUMAN3H-MESULERGINERo 6008692.75423Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398125-HT2BCLONEDHUMAN3H-MESULERGINE5-Hydroxy Tryptamine2.81838Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398135-HT2BCLONEDHUMAN3H-MESULERGINEmCPP12.0226Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398145-HT2BCLONEDHUMAN3H-MESULERGINEMK 212151.356Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398155-HT2BCLONEDHUMAN3H-MESULERGINERo 60033215.8489Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398165-HT2BCLONEDHUMAN3H-MESULERGINEDOI7.07946Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398175-HT2BCLONEDHUMAN3H-MESULERGINEBW-723C863.16228Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398185-HT2BCLONEDHUMAN3H-MESULERGINERo 60-01750.549541Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398195-HT2BCLONEDHUMAN3H-MESULERGINELISURIDE1.38038Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398205-HT2BCLONEDHUMAN3H-MESULERGINERo 6008697.94328Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398215-HT2CCLONEDHUMAN3H-MESULERGINERS-1022211.47911Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398225-HT2CCLONEDHUMAN3H-MESULERGINESB 2420840.47863Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398235-HT2CCLONEDHUMAN3H-MESULERGINEKETANSERIN16.9824Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398245-HT2CCLONEDHUMAN3H-MESULERGINEMESULERGINE1.12202Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398255-HT2CCLONEDHUMAN3H-MESULERGINEMETERGOLINE0.467735Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398265-HT2CCLONEDHUMAN3H-MESULERGINESB 2065533.16228Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398275-HT2CCLONEDHUMAN3H-MESULERGINEMIANSERIN1.51356Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398285-HT2CCLONEDHUMAN3H-MESULERGINERITANSERIN1.62181Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398295-HT2CCLONEDHUMAN3H-MESULERGINESB-21550511.2202Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398305-HT2CCLONEDHUMAN3H-MESULERGINESB2047412137.96Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398315-HT2CCLONEDHUMAN3H-MESULERGINES33526457.088Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398325-HT2CCLONEDHUMAN3H-MESULERGINELY 26609767.6083Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398335-HT2BCLONEDHUMAN3H-MESULERGINERS-102221234.423Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398345-HT2BCLONEDHUMAN3H-MESULERGINESB 24208445.7088Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398355-HT2BCLONEDHUMAN3H-MESULERGINEKETANSERIN234.423Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398365-HT2BCLONEDHUMAN3H-MESULERGINEMESULERGINE1.94984Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398375-HT2BCLONEDHUMAN3H-MESULERGINEMETERGOLINE0.707946Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398385-HT2BCLONEDHUMAN3H-MESULERGINESB 2065535.49541Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398395-HT2BCLONEDHUMAN3H-MESULERGINEMIANSERIN5.49541Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398405-HT2BCLONEDHUMAN3H-MESULERGINERITANSERIN1.25893Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398415-HT2BCLONEDHUMAN3H-MESULERGINESB-2155051.47911Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398425-HT2BCLONEDHUMAN3H-MESULERGINESB20474151.2861Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398435-HT2BCLONEDHUMAN3H-MESULERGINES335264.0738Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
398445-HT2BCLONEDHUMAN3H-MESULERGINELY 2660970.199526Cussac D, et al., 2002Jan 15, 2025Jan 15, 2025
39845MORCLONEDHUMAN3H-DAMGOMCL-145200Mathews JL, et al., 2005Jan 15, 2025Jan 15, 2025
39846MORCLONEDHUMAN3H-DAMGOMCL-101230Mathews JL, et al., 2005Jan 15, 2025Jan 15, 2025
39847DORCLONEDHUMAN3H-NaltrindoleMCL-1459400Mathews JL, et al., 2005Jan 15, 2025Jan 15, 2025
39848DORCLONEDHUMAN3H-NaltrindoleMCL-1015900Mathews JL, et al., 2005Jan 15, 2025Jan 15, 2025
39849KORCLONEDHUMAN3H-U69,593MCL-14578Mathews JL, et al., 2005Jan 15, 2025Jan 15, 2025
39850KORCLONEDHUMAN3H-U69,593MCL-10179Mathews JL, et al., 2005Jan 15, 2025Jan 15, 2025
39851AT1LIVERRAT125I-Angiotensin IIAngiotensin II0.95Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39852AT1LIVERRAT125I-Angiotensin IIAng II Sar10.16Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39853AT1LIVERRAT125I-Angiotensin IIAng II 4-NH2-Phe6>10000Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39854AT1LIVERRAT125I-Angiotensin IIC45H56N11O10>10000Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39855AT1LIVERRAT125I-Angiotensin IIC51H67N12O11>10000Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39856AT1LIVERRAT125I-Angiotensin IIC50H65N12O11>10000Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39857AT1LIVERRAT125I-Angiotensin IIC44H54N11O10>10000Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39858AT1LIVERRAT125I-Angiotensin IIC49H63N12O1130.3Georgsson J, et al., 2005Jan 15, 2025Jan 15, 2025
39859AT2UterusPIG125I-Angiotensin IIAngiotensin II0.2Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39860AT2UterusPIG125I-Angiotensin IIAng II Sar10.18Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39861AT2UterusPIG125I-Angiotensin IIAng II 4-NH2-Phe60.7Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39862AT2UterusPIG125I-Angiotensin IIC45H56N11O1010.1Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39863AT2UterusPIG125I-Angiotensin IIC51H67N12O11463.7Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39864AT2UterusPIG125I-Angiotensin IIC50H65N12O111.85Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39865AT2UterusPIG125I-Angiotensin IIC44H54N11O1041.3Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
39866AT2UterusPIG125I-Angiotensin IIC49H63N12O119.8Georgsson J, et al., 2005Jan 15, 2025Jan 28, 2025
399385-HT2BCLONEDHUMANUNDEFINEDBW-723C8679.4328Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399395-HT2BStomachRATFunctionalBW-723C8612.5893Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399405-HT2CCLONEDHUMANFunctionalBW-723C86501.187Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399415-HT2CUNDEFINEDRATUNDEFINEDBW-723C86125.893Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399425-HT2ACLONEDHUMANFunctionalBW-723C86100Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399435-HT2AUNDEFINEDRATFunctionalBW-723C86251.189Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399445-HT1AUNDEFINEDRATUNDEFINEDBW-723C861258.93Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399455-HT1BUNDEFINEDHUMANUNDEFINEDBW-723C86125.893Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399465-HT1DUNDEFINEDHUMANUNDEFINEDBW-723C86630.957Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399475-HT1EUNDEFINEDHUMANUNDEFINEDBW-723C863162.28Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399485-HT1FCLONEDHUMANUNDEFINEDBW-723C867943.28Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399495-HT3UNDEFINEDRATUNDEFINEDBW-723C86316.228Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399505-HT4UNDEFINEDRATFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399515-HT7CLONEDHUMANUNDEFINEDBW-723C863162.28Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
399525-HT7CLONEDRATFunctionalBW-723C861000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39953D1UNDEFINEDUNDEFINEDUNDEFINEDBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39954D2UNDEFINEDUNDEFINEDUNDEFINEDBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39955D4CLONEDHUMANUNDEFINEDBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39956UNDEFINEDUNDEFINEDFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39957UNDEFINEDUNDEFINEDFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39958Beta1UNDEFINEDUNDEFINEDFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39959Beta2UNDEFINEDUNDEFINEDFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 28, 2025
39960H1UNDEFINEDUNDEFINEDFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39961H2UNDEFINEDUNDEFINEDFunctionalBW-723C86>10000Kennett GA, et al., 1996aJan 15, 2025Jan 15, 2025
39962CEREBRAL CORTEXRAT3H-PRAZOSINFLUOXETINE3981.07Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39963CEREBRAL CORTEXRAT3H-RX821002FLUOXETINE5011.87Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39964SLC6A4FR. CORTEXRAT3H-PAROXETINEFLUOXETINE10Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39965NETFR. CORTEXRAT3H-NisoxetineFLUOXETINE794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39966CEREBRAL CORTEXRAT3H-PRAZOSINNapamezole100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39967CEREBRAL CORTEXRAT3H-RX821002Napamezole3.16228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39968SLC6A4FR. CORTEXRAT3H-PAROXETINENapamezole199.526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39969NETFR. CORTEXRAT3H-NisoxetineNapamezole1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39970CEREBRAL CORTEXRAT3H-PRAZOSINATIPAMEZOLE1995.26Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39971CEREBRAL CORTEXRAT3H-RX821002ATIPAMEZOLE0.125893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39972SLC6A4FR. CORTEXRAT3H-PAROXETINEATIPAMEZOLE3162.28Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39973NETFR. CORTEXRAT3H-NisoxetineATIPAMEZOLE>10000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39974CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39975CEREBRAL CORTEXRAT3H-RX8210024(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39976SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate39.8107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39977NETFR. CORTEXRAT3H-Nisoxetine4(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39978CEREBRAL CORTEXRAT3H-PRAZOSINC14H15ClN2·C4H4O4 398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39979CEREBRAL CORTEXRAT3H-RX821002C14H15ClN2·C4H4O4 25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39980SLC6A4FR. CORTEXRAT3H-PAROXETINEC14H15ClN2·C4H4O4 19.9526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39981NETFR. CORTEXRAT3H-NisoxetineC14H15ClN2·C4H4O4 50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39982CEREBRAL CORTEXRAT3H-PRAZOSINC14H15FN2·C4H4O4 501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39983CEREBRAL CORTEXRAT3H-RX821002C14H15FN2·C4H4O4 39.8107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39984SLC6A4FR. CORTEXRAT3H-PAROXETINEC14H15FN2·C4H4O4 79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39985NETFR. CORTEXRAT3H-NisoxetineC14H15FN2·C4H4O4 125.893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39986CEREBRAL CORTEXRAT3H-PRAZOSINC15H16N2O·C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39987CEREBRAL CORTEXRAT3H-RX821002C15H16N2O·C4H4O4 25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39988SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H16N2O·C4H4O4 15.8489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39989NETFR. CORTEXRAT3H-NisoxetineC15H16N2O·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39990CEREBRAL CORTEXRAT3H-PRAZOSINC15H16N2·C4H4O4 630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39991CEREBRAL CORTEXRAT3H-RX821002C15H16N2·C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39992SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H16N2·C4H4O4 12.5893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39993NETFR. CORTEXRAT3H-NisoxetineC15H16N2·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39994CEREBRAL CORTEXRAT3H-PRAZOSINC14H15FN2·C4H4O4 251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39995CEREBRAL CORTEXRAT3H-RX821002C14H15FN2·C4H4O4 199.526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39996SLC6A4FR. CORTEXRAT3H-PAROXETINEC14H15FN2·C4H4O4 1.58489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39997NETFR. CORTEXRAT3H-NisoxetineC14H15FN2·C4H4O4 50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39998CEREBRAL CORTEXRAT3H-PRAZOSINC15H15F3N2·C4H4O4 1258.93Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
39999CEREBRAL CORTEXRAT3H-RX821002C15H15F3N2·C4H4O4 398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40000SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H15F3N2·C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40001NETFR. CORTEXRAT3H-NisoxetineC15H15F3N2·C4H4O4 >10000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40002CEREBRAL CORTEXRAT3H-PRAZOSINC15H18N2O·C4H4O4 2511.89Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40003CEREBRAL CORTEXRAT3H-RX821002C15H18N2O·C4H4O4 501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40004SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H18N2O·C4H4O4 199.526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40005NETFR. CORTEXRAT3H-NisoxetineC15H18N2O·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40006CEREBRAL CORTEXRAT3H-PRAZOSINC15H18N2·C4H4O4 398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40007CEREBRAL CORTEXRAT3H-RX821002C15H18N2·C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40008SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H18N2·C4H4O4 63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40009NETFR. CORTEXRAT3H-NisoxetineC15H18N2·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40010CEREBRAL CORTEXRAT3H-RX821002C15H18N2·C4H4O4 398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40011SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H18N2·C4H4O4 15.8489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40012NETFR. CORTEXRAT3H-NisoxetineC15H18N2·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40013CEREBRAL CORTEXRAT3H-PRAZOSIN2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40014CEREBRAL CORTEXRAT3H-RX8210022-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate316.228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40015SLC6A4FR. CORTEXRAT3H-PAROXETINE2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate39.8107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40016NETFR. CORTEXRAT3H-Nisoxetine2-Amino-4(5)-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Bromhydrate79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40017CEREBRAL CORTEXRAT3H-RX8210022-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40018SLC6A4FR. CORTEXRAT3H-PAROXETINE2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40019NETFR. CORTEXRAT3H-Nisoxetine2-Amino-4-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hydrochloride501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40020CEREBRAL CORTEXRAT3H-RX8210022-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40021SLC6A4FR. CORTEXRAT3H-PAROXETINE2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40022NETFR. CORTEXRAT3H-Nisoxetine2-Amino-5-[(3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40023CEREBRAL CORTEXRAT3H-PRAZOSIN2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate316.228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40024CEREBRAL CORTEXRAT3H-RX8210022-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40025NETFR. CORTEXRAT3H-Nisoxetine2-Amino-5-[(8-chloro-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40026CEREBRAL CORTEXRAT3H-PRAZOSIN2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40027CEREBRAL CORTEXRAT3H-RX8210022-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate1584.89Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40028SLC6A4FR. CORTEXRAT3H-PAROXETINE2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40029NETFR. CORTEXRAT3H-Nisoxetine2-Amino-5-[(7-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40030CEREBRAL CORTEXRAT3H-RX8210022-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate1584.89Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40031SLC6A4FR. CORTEXRAT3H-PAROXETINE2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40032NETFR. CORTEXRAT3H-Nisoxetine2-Amino-5-[(6-methyl-3,4-dihydronaphthalen-2-yl)methyl]-4,5-dihydrooxazole, Hemifumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40033CEREBRAL CORTEXRAT3H-PRAZOSINC14H14N2·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40034CEREBRAL CORTEXRAT3H-RX821002C14H14N2·C4H4O4 125.893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40035SLC6A4FR. CORTEXRAT3H-PAROXETINEC14H14N2·C4H4O4 50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40036NETFR. CORTEXRAT3H-NisoxetineC14H14N2·C4H4O4 15.8489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40037CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40038CEREBRAL CORTEXRAT3H-RX8210024(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40039SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40040NETFR. CORTEXRAT3H-Nisoxetine4(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate19.9526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40041CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40042CEREBRAL CORTEXRAT3H-RX8210024(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate15.8489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40043SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate10Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40044NETFR. CORTEXRAT3H-Nisoxetine4(5)-[(1,2,3,4-Tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Succinate100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40045CEREBRAL CORTEXRAT3H-PRAZOSINC13H14N2O·C4H4O4 1584.89Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40046CEREBRAL CORTEXRAT3H-RX821002C13H14N2O·C4H4O4 125.893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40047SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H14N2O·C4H4O4 251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40048NETFR. CORTEXRAT3H-NisoxetineC13H14N2O·C4H4O4 63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40049CEREBRAL CORTEXRAT3H-PRAZOSINC12H14N2O2·C4H4O4 630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40050CEREBRAL CORTEXRAT3H-RX821002C12H14N2O2·C4H4O4 31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40051SLC6A4FR. CORTEXRAT3H-PAROXETINEC12H14N2O2·C4H4O4 1258.93Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40052NETFR. CORTEXRAT3H-NisoxetineC12H14N2O2·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40053CEREBRAL CORTEXRAT3H-PRAZOSINC13H16N2O·C4H4O4 316.228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40054CEREBRAL CORTEXRAT3H-RX821002C13H16N2O·C4H4O4 50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40055SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H16N2O·C4H4O4 501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40056NETFR. CORTEXRAT3H-NisoxetineC13H16N2O·C4H4O4 794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40057CEREBRAL CORTEXRAT3H-PRAZOSINC16H20N2·0.5C4H4O4 794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40058CEREBRAL CORTEXRAT3H-RX821002C16H20N2·0.5C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40059SLC6A4FR. CORTEXRAT3H-PAROXETINEC16H20N2·0.5C4H4O4 >10000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40060NETFR. CORTEXRAT3H-NisoxetineC16H20N2·0.5C4H4O4 39.8107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40061CEREBRAL CORTEXRAT3H-PRAZOSINC13H14N2·C4H4O4 1258.93Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40062CEREBRAL CORTEXRAT3H-RX821002C13H14N2·C4H4O4 15.8489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40063SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H14N2·C4H4O4 79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40064NETFR. CORTEXRAT3H-NisoxetineC13H14N2·C4H4O4 31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40065CEREBRAL CORTEXRAT3H-PRAZOSINC13H16N2·0.5C4H4O4 501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40066CEREBRAL CORTEXRAT3H-RX821002C13H16N2·0.5C4H4O4 1.99526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40067SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H16N2·0.5C4H4O4 63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40068NETFR. CORTEXRAT3H-NisoxetineC13H16N2·0.5C4H4O4 39.8107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40069CEREBRAL CORTEXRAT3H-PRAZOSINC12H12N2O·C4H4O4 2511.89Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40070CEREBRAL CORTEXRAT3H-RX821002C12H12N2O·C4H4O4 12.5893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40071SLC6A4FR. CORTEXRAT3H-PAROXETINEC12H12N2O·C4H4O4 1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40072NETFR. CORTEXRAT3H-NisoxetineC12H12N2O·C4H4O4 63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40073CEREBRAL CORTEXRAT3H-RX821002C12H11FN2O·C4H4O4100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40074SLC6A4FR. CORTEXRAT3H-PAROXETINEC12H11FN2O·C4H4O4158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40075NETFR. CORTEXRAT3H-NisoxetineC12H11FN2O·C4H4O4794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40076CEREBRAL CORTEXRAT3H-PRAZOSINC18H16N2O·C4H4O4 3162.28Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40077CEREBRAL CORTEXRAT3H-RX821002C18H16N2O·C4H4O4 >10000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40078SLC6A4FR. CORTEXRAT3H-PAROXETINEC18H16N2O·C4H4O4 >10000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40079NETFR. CORTEXRAT3H-NisoxetineC18H16N2O·C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40080CEREBRAL CORTEXRAT3H-PRAZOSINC13H15FN2·0.5C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40081CEREBRAL CORTEXRAT3H-RX821002C13H15FN2·0.5C4H4O4 1.25893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40082SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H15FN2·0.5C4H4O4 100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40083NETFR. CORTEXRAT3H-NisoxetineC13H15FN2·0.5C4H4O4 100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40084CEREBRAL CORTEXRAT3H-PRAZOSINC13H15FN2·0.5C4H4O4 630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40085CEREBRAL CORTEXRAT3H-RX821002C13H15FN2·0.5C4H4O4 7.94328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40086SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H15FN2·0.5C4H4O4 25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40087NETFR. CORTEXRAT3H-NisoxetineC13H15FN2·0.5C4H4O4 316.228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40088CEREBRAL CORTEXRAT3H-PRAZOSINC13H14F2N2·0.5C4H4O4794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40089CEREBRAL CORTEXRAT3H-RX821002C13H14F2N2·0.5C4H4O450.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40090SLC6A4FR. CORTEXRAT3H-PAROXETINEC13H14F2N2·0.5C4H4O412.5893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40091NETFR. CORTEXRAT3H-NisoxetineC13H14F2N2·0.5C4H4O4100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40092CEREBRAL CORTEXRAT3H-PRAZOSINC15H20N2·C4H4O4 199.526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40093CEREBRAL CORTEXRAT3H-RX821002C15H20N2·C4H4O4 25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40094SLC6A4FR. CORTEXRAT3H-PAROXETINEC15H20N2·C4H4O4 19.9526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40095NETFR. CORTEXRAT3H-NisoxetineC15H20N2·C4H4O4 25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40096CEREBRAL CORTEXRAT3H-PRAZOSINSpiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40097CEREBRAL CORTEXRAT3H-RX821002Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate10Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40098SLC6A4FR. CORTEXRAT3H-PAROXETINESpiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate15.8489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40099NETFR. CORTEXRAT3H-NisoxetineSpiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate199.526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40100CEREBRAL CORTEXRAT3H-PRAZOSINSpiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40101CEREBRAL CORTEXRAT3H-RX821002Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40102SLC6A4FR. CORTEXRAT3H-PAROXETINESpiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40103NETFR. CORTEXRAT3H-NisoxetineSpiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40104CEREBRAL CORTEXRAT3H-PRAZOSINSpiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate5011.87Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40105CEREBRAL CORTEXRAT3H-RX821002Spiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40106SLC6A4FR. CORTEXRAT3H-PAROXETINESpiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate6309.57Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40107NETFR. CORTEXRAT3H-NisoxetineSpiro{(1,3-diazacyclopent-1-ene)-5:3'-[spiro(cyclobutane-1':2-indan)]}, Fumarate>10000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40108CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate1258.93Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40109CEREBRAL CORTEXRAT3H-RX8210024(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40110SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40111NETFR. CORTEXRAT3H-Nisoxetine4(5)-[(3,4-Dihydronaphthalen-2-yl)methyl]-4(5)-methyl-4,5-dihydroimidazole, Fumarate316.228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40112CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40113CEREBRAL CORTEXRAT3H-RX8210024(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40114SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate10Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40115NETFR. CORTEXRAT3H-Nisoxetine4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate199.526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40116CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate1995.26Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40117CEREBRAL CORTEXRAT3H-RX8210024(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40118SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40119NETFR. CORTEXRAT3H-Nisoxetine4(5)-[(2-Methyl-1,2,3,4-tetrahydronaphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40120CLONEDHUMAN3H-RX821002Napamezole6.30957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40121CLONEDHUMAN3H-RX821002ATIPAMEZOLE3.16228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40122CLONEDHUMAN3H-RX8210024(5)-[(3,4-dihydro-2-naphthalen-2-yl)methyl]-4,5-dihydroimidazole, Fumarate100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40123CLONEDHUMAN3H-RX821002C14H15ClN2·C4H4O4 31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40124CLONEDHUMAN3H-RX821002C14H15FN2·C4H4O4 39.8107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40125CLONEDHUMAN3H-RX821002C14H15FN2·C4H4O4 158.489Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40126CLONEDHUMAN3H-RX821002C14H14N2·C4H4O4 50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40127CLONEDHUMAN3H-RX8210024(5)-(8-Chloro-2-naphthylmethyl)-4,5-dihydroimidazole, Fumarate25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40128CLONEDHUMAN3H-RX821002C13H16N2·0.5C4H4O4 3.98107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40129CLONEDHUMAN3H-RX821002C12H12N2O·C4H4O4 19.9526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40130CLONEDHUMAN3H-RX8210024(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate63.0957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40131CLONEDHUMAN3H-RX8210024(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate3.16228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40132CLONEDHUMAN3H-RX821002Spiro[(1,3-diazacyclopent-1-ene)-5:2'-(trans-1',2',3',4',4'a,9',9'a,10'-octahydroanthracene)], Fumarate1.25893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40133NMDACORTICAL MEMBRANESRAT3H-CPP(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40134AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40135KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40136NMDACORTICAL MEMBRANESRAT3H-CPP(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid490Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40137AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40138KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40139NMDACORTICAL MEMBRANESRAT3H-CPP(+/-)-AP5290Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40140NMDACORTICAL MEMBRANESRAT3H-CPP(R)-AP5880Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40141NMDACORTICAL MEMBRANESRAT3H-CPP(S)-AP5>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40142NMDACORTICAL MEMBRANESRAT3H-CPP(R)-CPPene40Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40143mGluR5CLONEDRATUNDEFINED(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40144mGluR5CLONEDRATUNDEFINED(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40145mGluR2CLONEDRATFunctional(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40146mGluR4CLONEDRATUNDEFINED(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40147mGluR5CLONEDRATUNDEFINED(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40148mGluR5CLONEDRATUNDEFINED(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40149mGluR4CLONEDRATUNDEFINED(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40150mGluR5CLONEDRATFunctional(+/-)-trans-ACPD>10000Conti P, et al., 2003Jan 15, 2025Jan 15, 2025
40151mGluR5CLONEDRATFunctional(+/-)-trans-ACPD>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40152mGluR2CLONEDRATFunctional(+/-)-trans-ACPD2000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40153mGluR4CLONEDRATFunctional(+/-)-trans-ACPD>10000Conti P, et al., 2003Jan 15, 2025Jan 28, 2025
40154MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluoroacetic Acid Salt0.057Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40155TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(4-methyl-1,4-diazepan-1-yl)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide Trifluoroacetic Acid Salt3.3Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40156MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide0.047Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40157TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(methyl(neopentyl)amino)-2-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide64Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40158MAPK14CLONEDHUMANFunctional3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide0.05Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40159TNFαwhole blood assay (WBA)HUMANFunctional3-(2-Amino-5-cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide17Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40160MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide0.15Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40161TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(methyl(neopentyl)amino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide42Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40162MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide16Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40163TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(methylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide250Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40164MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(propylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide0.97Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40165TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(propylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide158Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40166MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide0.61Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40167TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide4.6Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40168MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide0.42Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40169TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-methoxy-4-methylbenzamide4.1Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40170MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide0.41Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40171TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide8.7Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40172MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide1.6Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40173TNFαwhole blood assay (WBA)HUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide3.5Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40174MAPK14CLONEDHUMANFunctional3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide0.057Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40175TNFαwhole blood assay (WBA)HUMANFunctional3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methybenzamide18Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40176MAPK14CLONEDHUMANFunctional3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide0.16Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40177TNFαwhole blood assay (WBA)HUMANFunctional3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide1.5Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40178MAPK14CLONEDHUMANFunctional3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide1.5Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40179TNFαwhole blood assay (WBA)HUMANFunctional3-(2-Amino-5-cyano-6-(isopropylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide67Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40180MAPK14CLONEDHUMANFunctional3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide1.9Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40181TNFαwhole blood assay (WBA)HUMANFunctional3-(2-Amino-5-cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(1-ethyl-1H-pyrazol-5-yl)-4-methylbenzamide21Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
401825-HT1AUNDEFINEDRATUNDEFINEDmCPP316.228Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401835-HT1BUNDEFINEDRATUNDEFINEDmCPP251.189Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401845-HT1DUNDEFINEDRATUNDEFINEDmCPP1584.89Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401855-HT2AUNDEFINEDRATUNDEFINEDmCPP199.526Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401865-HT2BUNDEFINEDRATUNDEFINEDmCPP25.1189Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401875-HT2CUNDEFINEDRATUNDEFINEDmCPP19.9526Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401885-HT3UNDEFINEDRATUNDEFINEDmCPP100Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401895-HT6UNDEFINEDRATUNDEFINEDmCPP2511.89Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
401905-HT7UNDEFINEDRATUNDEFINEDmCPP251.189Martin RS, et al., 2001Jan 15, 2025Jan 15, 2025
40191DP2BRAINRAT3H-PGD2PGD219Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40192DP2BRAINRAT3H-PGD2PGD2-methyl ester27Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40193DP2BRAINRAT3H-PGD2PGD1523Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40194DP2BRAINRAT3H-PGD2PGF2Alpha693Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40195DP2BRAINRAT3H-PGD2PGE13758Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40196DP2BRAINRAT3H-PGD2PGE22948Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40197DP2BRAINRAT3H-PGD2PGI23537Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40198DP2BRAINRAT3H-PGD2PG Thromboxane B24200Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40199DP2BRAINRAT3H-PGD2PG 13,14-dihydro-15-keto-D2>10000Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40200DP2BRAINRAT3H-PGD2PGF1 alpha 6-keto>10000Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40201DP2BRAINRAT3H-PGD2PGA2>10000Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40202DP2BRAINRAT3H-PGD2PGB2>10000Shimizu T, et al., 1982Jan 15, 2025Jan 15, 2025
40203IPNCB-20MOUSE3H-PGI2PGI216.6MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40204IPNCB-20MOUSE3H-PGI2PGE1137MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40205IPNCB-20MOUSE3H-PGI2PGE1, 13,14-dihydro315MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40206IPNCB-20MOUSE3H-PGI2PGE1, 8-iso735MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40207IPNCB-20MOUSE3H-PGI2PGE2, 5,6-trans735MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40208IPNCB-20MOUSE3H-PGI2PGE2,17-Phenyl4370MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40209IPNCB-20MOUSE3H-PGI2PGI1, 6beta7350MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40210IPNCB-20MOUSE3H-PGI2PGE2>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40211IPNCB-20MOUSE3H-PGI2PGE2, 13,14-dihydro15-oxo>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40212IPNCB-20MOUSE3H-PGI2PGE2, 15-epi>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40213IPNCB-20MOUSE3H-PGI2PGF1alpha>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40214IPNCB-20MOUSE3H-PGI2PGF1alpha, 6-oxo>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40215IPNCB-20MOUSE3H-PGI2PGF2Alpha>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40216IPNCB-20MOUSE3H-PGI2PGD1>10000MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40217IPNCB-20MOUSE3H-PGI2PGE2 13,14-dihydro8410MacDermot J, et al., 1981Jan 15, 2025Jan 28, 2025
40218CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate1258.93Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40219CEREBRAL CORTEXRAT3H-RX8210024(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40220SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40221NETFR. CORTEXRAT3H-Nisoxetine4(5)-(1,2,3,7b-Tetrahydrocyclopropa[a]naphthalen-1a-ylmethyl)-4,5-dihydroimidazole, Fumarate794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40222CEREBRAL CORTEXRAT3H-RX8210024(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40223SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate3162.28Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40224NETFR. CORTEXRAT3H-Nisoxetine4(5)-(1a,2,3,7b-tetrahydro-1H-cyclopropal[a]napthalen-1-yl)-4,5-dihydroimidazole, Fumarate251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40225CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40226CEREBRAL CORTEXRAT3H-RX8210024(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40227SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole630.957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40228CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole794.328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40229CEREBRAL CORTEXRAT3H-RX8210024(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole3162.28Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40230SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40231NETFR. CORTEXRAT3H-Nisoxetine4(5)-(1a,2,7,7a-Tetrahydro-1H-cyclopropal[b]naphthalen-1-yl)-4,5-dihydroimidazole50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40232CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate501.187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40233CEREBRAL CORTEXRAT3H-RX8210024(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate6.30957Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40234SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate1.99526Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40235NETFR. CORTEXRAT3H-Nisoxetine4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate100Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40236CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate1000Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40237CEREBRAL CORTEXRAT3H-RX8210024(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate251.189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40238SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate25.1189Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40239NETFR. CORTEXRAT3H-Nisoxetine4(5)-{Spiro[cyclopropane-2':2-(1,2,3,4-tetrahydronaphthalene)]-1-yl}-4,5-dihydroimidazole, Fumarate398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40240CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate6309.57Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40241CEREBRAL CORTEXRAT3H-RX8210024(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate79.4328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40242SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate398.107Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40243NETFR. CORTEXRAT3H-Nisoxetine4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate316.228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40244CEREBRAL CORTEXRAT3H-PRAZOSIN4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate125.893Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40245CEREBRAL CORTEXRAT3H-RX8210024(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate0.794328Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40246SLC6A4FR. CORTEXRAT3H-PAROXETINE4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate50.1187Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40247NETFR. CORTEXRAT3H-Nisoxetine4(5)-[Spiro(cyclopropane-2':2-indan)-1'-yl]-4,5-dihydroimidazole, Fumarate31.6228Cordi AA, et al., 2001Jan 15, 2025Jan 15, 2025
40248NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid210Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40249AMPACORTICAL MEMBRANESRAT3H-AMPA(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
40250KACORTICAL MEMBRANESRAT3H-Kainic acid(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
40251NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2'S*)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid960Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40252NMDACORTICAL MEMBRANESRAT3H-CGP39653(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40253AMPACORTICAL MEMBRANESRAT3H-AMPA(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
40254KACORTICAL MEMBRANESRAT3H-Kainic acid(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
40255NMDACORTICAL MEMBRANESRAT3H-CGP39653(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40256AMPACORTICAL MEMBRANESRAT3H-AMPA(4R*,2'R*)-4-(2-Amino-2-carboxyethyl)-5,5-dimethyl-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
40257NMDACORTICAL MEMBRANESRAT3H-CGP39653(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid370Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40258NMDACORTICAL MEMBRANESRAT3H-D-APV(-)-2-aminoadipic acid>10000Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40259NMDACORTICAL MEMBRANESRAT3H-CPPCGS 1975595Conti P, et al., 2004Jan 15, 2025Jan 28, 2025
40260AMPACORTICAL MEMBRANESRAT3H-AMPA(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
40261KACORTICAL MEMBRANESRAT3H-Kainic acid(3aS*,5R*,6aS*)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2004Jan 15, 2025Jan 15, 2025
402625-HT2BCLONEDHUMAN3H-5HTMETHYSERGIDE7.94328Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402635-HT2BCLONEDHUMAN3H-5HTYOHIMBINE398.107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402645-HT2BCLONEDHUMAN3H-5HTMIANSERIN19.9526Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402655-HT2BCLONEDHUMAN3H-5HTSPIPERONE1584.89Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402665-HT2BCLONEDHUMAN3H-5HTKETANSERIN630.957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402675-HT2BCLONEDHUMAN3H-5HTRITANSERIN5.01187Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402685-HT2BCLONEDHUMAN3H-5HTSB20474179.4328Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402695-HT2BCLONEDRAT3H-5HTLY 538576.30957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402705-HT2BCLONEDRAT3H-5HTMESULERGINE39.8107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402715-HT2BCLONEDRAT3H-5HTMETHYSERGIDE6.30957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402725-HT2BCLONEDRAT3H-5HTRAUWOLSCINE39.8107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402735-HT2BCLONEDRAT3H-5HTYOHIMBINE50.1187Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402745-HT2BCLONEDRAT3H-5HTMIANSERIN50.1187Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402755-HT2BCLONEDRAT3H-5HTSPIPERONE3162.28Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402765-HT2BCLONEDRAT3H-5HTKETANSERIN3162.28Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402775-HT2BCLONEDRAT3H-5HTRITANSERIN5.01187Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402785-HT2CChoroid PlexusPIG3H-MESULERGINELY 538577.94328Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402795-HT2CChoroid PlexusPIG3H-MESULERGINEMESULERGINE1.58489Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402805-HT2CChoroid PlexusPIG3H-MESULERGINEMETHYSERGIDE2.51189Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402815-HT2CChoroid PlexusPIG3H-MESULERGINEMETERGOLINE0.630957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402825-HT2CChoroid PlexusPIG3H-MESULERGINERAUWOLSCINE1584.89Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402835-HT2CChoroid PlexusPIG3H-MESULERGINEYOHIMBINE>10000Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402845-HT2CChoroid PlexusPIG3H-MESULERGINECHLORPROMAZINE15.8489Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402855-HT2CChoroid PlexusPIG3H-MESULERGINEMIANSERIN10Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402865-HT2CChoroid PlexusPIG3H-MESULERGINESPIPERONE1258.93Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402875-HT2CChoroid PlexusPIG3H-MESULERGINEKETANSERIN100Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402885-HT2CChoroid PlexusPIG3H-MESULERGINEMETHIOTHEPIN25.1189Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402895-HT2CChoroid PlexusPIG3H-MESULERGINEPIZOTIFEN7.94328Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402905-HT2CChoroid PlexusPIG3H-KETANSERINRITANSERIN2.51189Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402915-HT2CChoroid PlexusPIG3H-MESULERGINESB2047411000Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402925-HT6CLONEDRAT3H-LSDMESULERGINE1584.89Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402935-HT6CLONEDRAT3H-LSDMETHYSERGIDE398.107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402945-HT6CLONEDRAT3H-LSDMETERGOLINE31.6228Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402955-HT6CLONEDRAT3H-LSDAMITRIPTYLINE63.0957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402965-HT6CLONEDRAT3H-LSDAMOXAPINE6.30957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402975-HT6CLONEDRAT3H-LSDCHLORPROMAZINE3.98107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402985-HT6CLONEDRAT3H-LSDCHLORPROTHIXENE3.16228Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
402995-HT6CLONEDRAT3H-LSDFLUPHENAZINE15.8489Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403005-HT6CLONEDRAT3H-LSDLOXAPINE15.8489Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403015-HT6CLONEDRAT3H-LSDMIANSERIN50.1187Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403025-HT6CLONEDRAT3H-LSDPERPHENAZINE15.8489Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403035-HT6CLONEDRAT3H-LSDSPIPERONE1584.89Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403045-HT6CLONEDRAT3H-LSDTHIORIDAZINE6.30957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403055-HT6CLONEDRAT3H-LSDKETANSERIN>10000Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403065-HT6CLONEDRAT3H-LSDMETHIOTHEPIN1.99526Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403075-HT6CLONEDRAT3H-LSDRITANSERIN39.8107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403085-HT7CLONEDRAT3H-LSDMESULERGINE6.30957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403095-HT7CLONEDRAT3H-LSDMETHYSERGIDE12.5893Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403105-HT7CLONEDRAT3H-LSDMETERGOLINE1.99526Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403115-HT7CLONEDRAT3H-LSDAMITRIPTYLINE125.893Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403125-HT7CLONEDRAT3H-LSDAMOXAPINE39.8107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403135-HT7CLONEDRAT3H-LSDCHLORPROMAZINE19.9526Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403145-HT7CLONEDRAT3H-LSDCHLORPROTHIXENE5.01187Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403155-HT7CLONEDRAT3H-LSDFLUPHENAZINE7.94328Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403165-HT7CLONEDRAT3H-LSDLOXAPINE39.8107Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403175-HT7CLONEDRAT3H-LSDMIANSERIN100Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403185-HT7CLONEDRAT3H-LSDPERPHENAZINE25.1189Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403195-HT7CLONEDRAT3H-LSDSPIPERONE10Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403205-HT7CLONEDRAT3H-LSDTHIORIDAZINE63.0957Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403215-HT7CLONEDRAT3H-LSDKETANSERIN199.526Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403225-HT7CLONEDRAT3H-LSDMETHIOTHEPIN1Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
403235-HT7CLONEDRAT3H-LSDRITANSERIN19.9526Glusa E, et al., 2000Jan 15, 2025Jan 15, 2025
40324recombinantHUMANFunctional6-phenylsulfonylpyridazin-2H-3-one600Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40325recombinantHUMANFunctional6-(2-Bromobenzenesulfonyl)-2H-pyridazin-3-one210Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40326recombinantHUMANFunctional6-(4-Bromobenzenesulfonyl)-2H-pyridazin-3-one350Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40327recombinantHUMANFunctional6-(2-Chlorobenzenesulfonyl)-2H-pyridazin-3-one170Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40328recombinantHUMANFunctional6-(3-Chlorobenzenesulfonyl)-2H-pyridazin-3-one240Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40329recombinantHUMANFunctional6-(4-Chlorobenzenesulfonyl)-2H-pyridazin-3-one380Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40330recombinantHUMANFunctional6-(2-Fluorobenzenesulfonyl)-2H-pyridazin-3-one540Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40331recombinantHUMANFunctional6-(4-Fluorobenzenesulfonyl)-2H-pyridazin-3-one474Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40332recombinantHUMANFunctional6-(4-Methoxybenzenesulfonyl)-2H-pyridazin-3-one2000Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40333recombinantHUMANFunctional6-(Biphenylyl-2-sulfonyl)-2H-pyridazin-3-one2200Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40334recombinantHUMANFunctional6-(2,3-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one55Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40335recombinantHUMANFunctional6-(2,4-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one190Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40336recombinantHUMANFunctional6-(2,5-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one73Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40337recombinantHUMANFunctional6-(2,6-Dichlorobenzenesulfonyl)-2H-pyridazin-3-one50Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40338recombinantHUMANFunctional6-(2,3-Difluorobenzenesulfonyl)-2H-pyridazin-3-one390Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40339recombinantHUMANFunctional6-(2,4-Difluorobenzenesulfonyl)-2H-pyridazin-3-one870Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40340recombinantHUMANFunctional6-(2-Chloro-4-fluorobenzenesulfonyl)-2H-pyridazin-3-one280Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40341recombinantHUMANFunctional6-(4-Bromo-2-fluorobenzenesulfonyl)-2H-pyridazin-3-one140Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40342recombinantHUMANFunctional6-(3-Trifluoromethylbenzenesulfonyl)-2H-pyridazin-3-one175Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40343recombinantHUMANFunctional6-(4-Trifluoromethylbenzenesulfonyl)-2H-pyridazin-3-one360Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40344recombinantHUMANFunctional6-(alpha-Naphthylmethylbenzenesulfonyl)-2H-pyridazin-3-one150Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40345recombinantHUMANFunctional6-(beta-Naphthylmethylbenzenesulfonyl)-2H-pyridazin-3-one360Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40346recombinantHUMANFunctionalsorbinil140Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40347recombinantHUMANFunctionalzopolrestat4Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40348recombinantHUMANFunctional6-(2-Cl-phenylmethanesulfonyl)-2H-pyridazin-3-one118Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40349recombinantHUMANFunctional6-(2-F-phenylmethanesulfonyl)-2H-pyridazin-3-one422Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40350recombinantHUMANFunctional6-(2-CF3-phenylmethanesulfonyl)-2H-pyridazin-3-one500Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40351recombinantHUMANFunctional6-(3-CF3-phenylmethanesulfonyl-2H-pyridazin-3-one72Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40352recombinantHUMANFunctional6-(2,3-Cl2-phenylmethanesulfonyl)-2H-pyridazin-3-one35Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40353recombinantHUMANFunctional6-(2,6-Cl2-phenylmethanesulfonyl)-2H-pyridazin-3-one52Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40354recombinantHUMANFunctional6-(2,3-F2-phenylmethanesulfonyl)-2H-pyridazin-3-one257Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40355recombinantHUMANFunctional6-(2F,4Br-phenylmethanesulfonyl)-2H-pyridazin-3-one667Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40356recombinantHUMANFunctional6-(2Cl,6F-phenylmethanesulfonyl)-2H-pyridazin-3-one26Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40357recombinantHUMANFunctional6-(2F,3-Cl-phenylmethanesulfonyl)-2H-pyridazin-3-one54Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40358recombinantHUMANFunctional6-(2F,3-CF3-phenylmethanesulfonyl)-2H-pyridazin-3-one44Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40359recombinantHUMANFunctional6-(Indole-2-sulfonyl)-2H-pyridazin-3-one590Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40360recombinantHUMANFunctional6-(5-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one1100Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40361recombinantHUMANFunctional6-(6-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one645Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40362recombinantHUMANFunctional6-(7-Chloroindole-2-sulfonyl)-2H-pyridazin-3-one450Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40363recombinantHUMANFunctional6-(6-Fluoroindole-2-sulfonyl)-2H-pyridazin-3-one1400Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40364recombinantHUMANFunctional6-(5,6-Methylenedioxyindole-2-sulfonyl)-2H-pyridazin-3-one3800Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40365recombinantHUMANFunctional6-(5,7-Dichloroindole-2-sulfonyl)-2H-pyridazin-3-one200Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40366recombinantHUMANFunctional6-(Benzofuran-2-sulfonyl)-2H-pyridazin-3-one150Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40367recombinantHUMANFunctional6-(5-Chlorobenzofuran-2-sulfonyl)-2H-pyridazin-3-one25Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40368recombinantHUMANFunctional6-(3-Methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one140Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40369recombinantHUMANFunctional6-(5-Methoxybenzofuran-2-sulfonyl)-2H-pyridazin-3-one230Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40370recombinantHUMANFunctional6-(5,7-Dichlorobenzofuran-2-sulfonyl)-2H-pyridazin-3-one87Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40371recombinantHUMANFunctional6-(5-Chloro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one1Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40372recombinantHUMANFunctional6-(6-Chloro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one190Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40373recombinantHUMANFunctional6-(5-Fluoro-3-methylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one3Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40374recombinantHUMANFunctional6-(3,5-Dimethylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one13Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40375recombinantHUMANFunctional6-(5-Chloro-3-ethylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one6Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40376recombinantHUMANFunctional6-(5-Chloro-3-isopropylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one92Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40377recombinantHUMANFunctional6-(3-Phenylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one23Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40378recombinantHUMANFunctional6-(3-[4-Fluorophenyl]benzofuran-2-methylsulfonyl)-2H-pyridazin-3-one49Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40379recombinantHUMANFunctional6-(5-Chloro-3-phenylbenzofuran-2-sulfonyl)-2H-pyridazin-3-one34Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40380recombinantHUMANFunctional6-(Benzothiophene-2-sulfonyl)-2H-pyridazin-3-one180Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40381recombinantHUMANFunctional6-(5-Methylbenzothiophene-2-sulfonyl)-2H-pyridazin-3-one160Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40382recombinantHUMANFunctional6-(Benzothiazole-2-sulfonyl)-2H-pyridazin-3-one450Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40383recombinantHUMANFunctional6-(5-Chloro-3-methylbenzothiophene-2-sulfonyl)-2H-pyridazin-3-one 55Mylari BL, et al., 2005Jan 15, 2025Jan 15, 2025
40384STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-D-Pro-Gln-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40385STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-alphaMe-Pro-Gln-Thr-NH1870Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40386STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-4-hydroxy-Pro-Gln-Thr-NH2484Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40387STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-cis-3,4-methanoPro-Gln-Thr-NH2–1265Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40388STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-cis-3,4-methanoPro-Gln-Thr-NH2–23110Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40389STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Azt-Gln-Thr-NH21660Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40390STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pip-Gln-Thr-NH21240Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40391STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Nip-Gln-Thr-NH2-1>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40392STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Nip-Gln-Thr-NH2-2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40393STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Inp-Gln-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40394STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Cmpi-Gln-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40395STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-1Ac6c-Gln-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40396STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gaba1780Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40397STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Ahx9780Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40398STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-3-carboxamidoanilide>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40399STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-3Ac6c-NH29810Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40400STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Nip-NH23020Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40401STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Inp-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40402STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Cmpi-NH21400Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40403STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-PyA-NH21690Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40404LIVERRATFunctional2-{1-[2,5-Di(trifluoromethyl)phenyl]methylidene}-6-methoxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40405LIVERRATFunctional6-Methoxy-2-[1-(2-methylphenyl)methylidene]-3,4-dihydro-2H-naphthlalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40406LIVERRATFunctional2-[1-(2-Bromophenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40407LIVERRATFunctional2-[1-(4-Hydroxyphenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40408LIVERRATFunctional6-Hydroxy-2-[1-(4-hydroxyphenyl)methylidene]-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40409LIVERRATFunctional2-{1-[4-(Dimethylamino)phenyl]methylidene}-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40410LIVERRATFunctional2-[1-(2-Bromophenyl)methylidene]-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one2400Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40411LIVERRATFunctional2-Biphenyl-2-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40412LIVERRATFunctional2-Biphenyl-4-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40413LIVERRATFunctionalKetoconazole>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40414LIVERRATFunctionalR 1158669000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40415MCF7RATFunctional2-{1-[2,5-Di(trifluoromethyl)phenyl]methylidene}-6-methoxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40416MCF7RATFunctional6-Methoxy-2-[1-(2-methylphenyl)methylidene]-3,4-dihydro-2H-naphthlalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40417MCF7RATFunctional2-[1-(2-Bromophenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one9000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40418MCF7RATFunctional2-[1-(4-Hydroxyphenyl)methylidene]-6-methoxy-3,4-dihydro-2H-naphthalen-1-one7000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40419MCF7RATFunctional6-Hydroxy-2-[1-(4-hydroxyphenyl)methylidene]-3,4-dihydro-2H-naphthalen-1-one9000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40420MCF7RATFunctional2-{1-[4-(Dimethylamino)phenyl]methylidene}-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40421MCF7RATFunctional2-[1-(2-Bromophenyl)methylidene]-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40422MCF7RATFunctional2-Biphenyl-2-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40423MCF7RATFunctional2-Biphenyl-4-ylmethylene-6-hydroxy-3,4-dihydro-2H-naphthalen-1-one>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40424MCF7RATFunctionalKetoconazole>10000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40425MCF7RATFunctionalLiarozole7000Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40426MCF7RATFunctionalR 1158665Yee WS, et al., 2005Jan 15, 2025Jan 15, 2025
40427NMDACORTICAL MEMBRANESRAT3H-CGP39653(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid370Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40428AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40429KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40430mGluR5CLONEDRATFunctional(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40431mGluR4CLONEDRATFunctional(+/-)-(3aS,5R,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40432NMDACORTICAL MEMBRANESRAT3H-CGP39653(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid233Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40433NMDACORTICAL MEMBRANESRAT3H-CGP39653(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40434NMDACORTICAL MEMBRANESRAT3H-CGP39653(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40435NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid210Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40436NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid1900Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40437NMDACORTICAL MEMBRANESRAT3H-CGP39653(5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid100Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40438NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid 960Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40439NMDACORTICAL MEMBRANESRAT3H-CGP39653(5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid510Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40440NMDACORTICAL MEMBRANESRAT3H-CGP39653(5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid2500Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40441AMPACORTICAL MEMBRANESRAT3H-AMPA(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40442AMPACORTICAL MEMBRANESRAT3H-AMPA(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40443AMPACORTICAL MEMBRANESRAT3H-AMPA(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40444AMPACORTICAL MEMBRANESRAT3H-AMPA(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40445AMPACORTICAL MEMBRANESRAT3H-AMPA(5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40446AMPACORTICAL MEMBRANESRAT3H-AMPA(5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40447AMPACORTICAL MEMBRANESRAT3H-AMPA(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40448AMPACORTICAL MEMBRANESRAT3H-AMPA(5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40449AMPACORTICAL MEMBRANESRAT3H-AMPA(5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40450KACORTICAL MEMBRANESRAT3H-Kainic acid(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40451KACORTICAL MEMBRANESRAT3H-Kainic acid(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40452KACORTICAL MEMBRANESRAT3H-Kainic acid(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40453KACORTICAL MEMBRANESRAT3H-Kainic acid(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40454KACORTICAL MEMBRANESRAT3H-Kainic acid(5R,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40455KACORTICAL MEMBRANESRAT3H-Kainic acid(5S,2'R)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40456KACORTICAL MEMBRANESRAT3H-Kainic acid(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40457KACORTICAL MEMBRANESRAT3H-Kainic acid(5R,2'R)-5-(2-Amino-2-carboxy-ethyl)-4,5-dihydro-isoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40458KACORTICAL MEMBRANESRAT3H-Kainic acid(5S,2'S)-5-(2-Amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40459mGluR5CLONEDRATFunctional(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40460mGluR5CLONEDRATFunctional(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40461mGluR5CLONEDRATFunctional(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40462mGluR5CLONEDRATFunctional(3aR,5R,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40463mGluR5CLONEDRATFunctional(3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40464mGluR5CLONEDRATFunctional(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40465mGluR5CLONEDRATFunctional(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 15, 2025
40466mGluR2CLONEDRATFunctional(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40467mGluR2CLONEDRATFunctional(3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40468mGluR2CLONEDRATFunctional(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40469mGluR2CLONEDRATFunctional(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40470mGluR4CLONEDRATFunctional(3aR,5S,6aR)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40471mGluR4CLONEDRATFunctional(3aS,5R,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40472mGluR4CLONEDRATFunctional(+/-)-(3aS,5S,6aS)-5-Amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic Acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40473mGluR4CLONEDRATFunctional(3aS,5S,6aS)-5-amino-4,5,6,6a-tetrahydro-3aH-cyclopenta[d]isoxazole-3,5-dicarboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40474mGluR4CLONEDRATFunctional(5R*,2’S*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid>10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40475mGluR4CLONEDRATFunctional(5R*,2’R*)-5-(2-amino-2-carboxyethyl)-4,5-dihydroisoxazole-3-carboxylic acid >10000Conti P, et al., 2005Jan 15, 2025Jan 28, 2025
40476STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln-Thr-NH2739Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40477STAT3CLONEDHUMANFunctionalAc-pTyr-Val-Pro-Gln-Thr-NH21540Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40478STAT3CLONEDHUMANFunctionalAc-pTyr-Ile-Pro-Gln-Thr-NH21070Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40479STAT3CLONEDHUMANFunctionalAc-pTyr-Phe-Pro-Gln-Thr-NH21890Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40480STAT3CLONEDHUMANFunctionalAc-pTyr-Cha-Pro-Gln-Thr-NH2910Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40481STAT3CLONEDHUMANFunctionalAc-pTyr-Nle-Pro-Gln-Thr-NH2717Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40482STAT3CLONEDHUMANFunctionalAc-pTyr-Phe2Ala-Pro-Gln-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40483STAT3CLONEDHUMANFunctionalAc-pTyr-N-MeLeu-Pro-Gln-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40484STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Glu(Me)-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40485STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln(Me2)-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40486STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Met(O)-Thr-NH29870Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40487STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Met(O2)-Thr-NH2>10000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40488STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln-NH2856Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40489STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–NHMe882Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40490STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–NHBn409Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40491STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–NH(S)CHMePh596Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40492STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–NH(R)CHMePh801Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40493STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln-OH748Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40494STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–NMe21850Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40495STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–NEt24220Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40496STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–pyrrolidine2110Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40497STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln–piperidine7000Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40498STAT3CLONEDHUMANFunctionalAc-pTyr-Leu-Pro-Gln-N-MeThr-NH21220Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40499STAT3CLONEDHUMANFunctionalBenzoyl-pTyr-Leu -Pro-Gln-Thr-NH2814Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40500STAT3CLONEDHUMANFunctionalPropionyl-pTyr-Leu -Pro-Gln-Thr-NH2497Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40501STAT3CLONEDHUMANFunctionalCbz-pTyr-Leu -Pro-Gln-Thr-NH2750Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
40502STAT3CLONEDHUMANFunctionalDihydrocinnamoyl-pTyr-Leu-Pro-Gln-Thr-NH2276Coleman DR, et al., 2005Jan 15, 2025Jan 15, 2025
405035-HT2BCLONEDHUMANFunctionalBW-723C8663.0957Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405045-HT2BCLONEDRATFunctionalBW-723C8612.5893Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405055-HT2CCLONEDHUMANFunctionalBW-723C86501.187Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405065-HT2CCLONEDRATUNDEFINEDBW-723C86125.893Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405075-HT2ACLONEDHUMANFunctionalBW-723C86100Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405085-HT2ACLONEDRATUNDEFINEDBW-723C86251.189Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405095-HT1ACORTEXRATUNDEFINEDBW-723C861258.93Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405105-HT1BCLONEDHUMANUNDEFINEDBW-723C86125.893Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405115-HT1DCLONEDHUMANUNDEFINEDBW-723C86630.957Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405125-HT1ECLONEDHUMANUNDEFINEDBW-723C863162.28Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405135-HT1FCLONEDHUMAN3H-5HTBW-723C867943.28Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405145-HT3CORTEXRATUNDEFINEDBW-723C86316.228Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405155-HT4esophagusRATUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405165-HT6CLONEDHUMANUNDEFINEDBW-723C86398.107Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405175-HT7CLONEDHUMAN3H-5CTBW-723C863162.28Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
405185-HT7UNDEFINEDRATUNDEFINEDBW-723C861000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40519D1STRIATUMRATUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40520D2STRIATUMRATUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40521D4CLONEDHUMAN3H-SPIPERONEBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40522AORTARABBITUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40523vas deferensRATUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40524Beta1Right atriumGUINEA PIGUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40525Beta2jugular veinRABBITUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 28, 2025
40526H1tracheaGUINEA PIGUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40527H2Saphenous veinRABBITUNDEFINEDBW-723C86>10000Kennett GA, et al., 1997aJan 15, 2025Jan 15, 2025
40528GABAACLONEDHUMAN3H-RO-15-1788DIAZEPAM14Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40529GABAACLONEDHUMAN3H-RO-15-1788DIAZEPAM20Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40530GABAACLONEDHUMAN3H-RO-15-1788DIAZEPAM15Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40531GABAACLONEDHUMAN3H-RO-15-1788Zolpidem27Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40532GABAACLONEDHUMAN3H-RO-15-1788Zolpidem160Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40533GABAACLONEDHUMAN3H-RO-15-1788Zolpidem380Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40534GABAACLONEDHUMAN3H-RO-15-17883,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine1.1Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40535GABAACLONEDHUMAN3H-RO-15-17883,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine2.9Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40536GABAACLONEDHUMAN3H-RO-15-17883,7-Diphenyl-6-(2-pyridyl)methyloxy-1,2,4-triazolo[4,3-b]pyridazine1.8Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40537GABAACLONEDHUMAN3H-RO-15-17883,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine0.78Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40538GABAACLONEDHUMAN3H-RO-15-17883,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine2.6Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40539GABAACLONEDHUMAN3H-RO-15-17883,7-Diphenyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-1,2,4-triazolo[4,3-b]pyridazine1.2Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40540GABAACLONEDHUMAN3H-RO-15-17887-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine6.2Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40541GABAACLONEDHUMAN3H-RO-15-17887-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine14Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40542GABAACLONEDHUMAN3H-RO-15-17887-Cyclohexyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine4.8Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40543GABAACLONEDHUMAN3H-RO-15-17887-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.38Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40544GABAACLONEDHUMAN3H-RO-15-17887-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.73Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40545GABAACLONEDHUMAN3H-RO-15-17887-Cyclopentyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.34Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40546GABAACLONEDHUMAN3H-RO-15-17887-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.23Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40547GABAACLONEDHUMAN3H-RO-15-17887-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.25Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40548GABAACLONEDHUMAN3H-RO-15-17887-Cyclobutyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.17Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40549GABAACLONEDHUMAN3H-RO-15-17887-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.36Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40550GABAACLONEDHUMAN3H-RO-15-17887-tert-butyl-6-(2-methyl-2H-1,2,4-triazol-3-ylmethoxy)-3-phenyl-1,2,4-triazolo[4,3-b]pyridazine0.14Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40551GABAACLONEDHUMAN3H-RO-15-17887-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine0.27Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40552GABAACLONEDHUMAN3H-RO-15-17887-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine0.31Carling RW, et al., 2005Jan 15, 2025Jan 27, 2025
40553GABAACLONEDHUMAN3H-RO-15-17887-(1,1-Dimethyleth-1-yl)-3-(2-fluoro-phenyl)-6-(2-ethyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine0.2Carling RW, et al., 2005Jan 15, 2025Jan 28, 2025
40554UNDEFINEDUNDEFINEDFunctionalPhosphinothricin600Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025
40555UNDEFINEDUNDEFINEDFunctional(2S)-2-Amino-4-[(aminomethyl)(hydroxy)phosphinyl]butyric Acid590Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025
40556UNDEFINEDUNDEFINEDFunctional(2S)-2-Amino-4-[(hydroxymethyl)(hydroxy)phosphinyl]butyric Acid2100Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025