The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 38,001-39,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
40557UNDEFINEDUNDEFINEDFunctional(2S)-2-Amino-4-[(1'-aminoethyl)(hydroxy)phosphinyl]butyric Acid3400Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025
40558UNDEFINEDUNDEFINEDFunctional(1'RS)-(2S)-2-Amino-4-[(1'-aminoethyl)(hydroxy)phosphinyl]butyric Acid3700Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025
40559UNDEFINEDUNDEFINEDFunctional(2S)-2-Amino-4-[(2'-Aminoethyl)(hydroxy)phosphinyl]butyric Acid>10000Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025
40560UNDEFINEDUNDEFINEDFunctional(2S)-2-Amino-4-[(2'-Carboxyethyl)(hydroxy)phosphinyl]butyric Acid >10000Berlicki L, et al., 2005Jan 15, 2025Jan 15, 2025
40561MOABRAINBOVINEUNDEFINED1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole31Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40562MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3,5-di-(4-methylphenyl)-4,5-dihydropyrazole6Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40563MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-methylphenyl)-5-(furan-2-yl)-4,5-dihydropyrazole4Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40564MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole6Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40565MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydropyrazole7Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40566MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydropyrazole8Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40567MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-chlorophenyl)-4,5-dihydropyrazole41Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40568MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-methylphenyl)-4,5-dihydropyrazole50Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40569MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(furan-2-yl)-4,5-dihydropyrazole50Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40570MOABRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(thiopen-2-yl)-4,5-dihydropyrazole27Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40571MOBBRAINBOVINEUNDEFINED1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole1.5Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40572MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3,5-di-(4-methylphenyl)-4,5-dihydropyrazole10Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40573MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-methylphenyl)-5-(furan-2-yl)-4,5-dihydropyrazole170Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40574MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole1000Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40575MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydropyrazole50Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40576MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydropyrazole370Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40577MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-chlorophenyl)-4,5-dihydropyrazole6Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40578MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(4-methylphenyl)-4,5-dihydropyrazole10Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40579MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(furan-2-yl)-4,5-dihydropyrazole20Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40580MOBBRAINBOVINEUNDEFINED1-thiocarbamoyl-3-(thiopen-2-yl)-5-(thiopen-2-yl)-4,5-dihydropyrazole50Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40581MOABRAINBOVINEUNDEFINED(+/-)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole31Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40582MOABRAINBOVINEUNDEFINED(-)(S)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole50Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40583MOABRAINBOVINEUNDEFINED(+)(R)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole13Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40584MOABRAINBOVINEUNDEFINED(+/-)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole6Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40585MOABRAINBOVINEUNDEFINED(-)(S)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole5Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40586MOABRAINBOVINEUNDEFINED(+)(R)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole12Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40587MOBBRAINBOVINEUNDEFINED(+/-)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole1.5Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40588MOBBRAINBOVINEUNDEFINED(-)(S)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole1Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40589MOBBRAINBOVINEUNDEFINED(+)(R)-1-Thiocarbamoyl-3-(4-methylphenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole2.7Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40590MOBBRAINBOVINEUNDEFINED(+/-)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole1000Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40591MOBBRAINBOVINEUNDEFINED(-)(S)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole2400Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40592MOBBRAINBOVINEUNDEFINED(+)(R)-1-Thiocarbamoyl-3-(4-fluorophenyl)-5-(4-chlorophenyl)-4,5-dihydropyrazole1400Chimenti F, et al., 2005Jan 15, 2025Jan 15, 2025
40593nAChRCLONEDHUMAN3H-Epibatidine9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
40594CCR5CLONEDHUMAN3H-Epibatidine9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
40595nAChRCLONEDHUMAN3H-Epibatidine9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 27, 2025
40596nAChRCLONEDHUMAN3H-Epibatidine9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 27, 2025
40597nAChR7CLONEDHUMAN3H-Epibatidine9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
40598GABABFOREBRAINRAT3H-BACLOFEN9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
40599H1CLONEDHUMAN3H-PYRILAMINE9-OH-risperidone5.61PDSP Certified DataJan 15, 2025Jan 15, 2025
40600H3CLONEDGUINEA PIG3H-Alpha-Me-histamine9-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
40601H4CLONEDHUMAN3H-Histamine9-OH-risperidone8698PDSP Certified DataJan 15, 2025Jan 15, 2025
40602EP4CLONEDHUMAN3H-PGE29-OH-risperidone>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
406035-HT1DCLONEDHUMAN3H-GR-1257439-OH-risperidone15.01PDSP Certified DataJan 15, 2025Jan 15, 2025
406045-HT2BCLONEDHUMAN3H-LSDRISPERIDONE41.5833PDSP Certified DataJan 15, 2025Jan 15, 2025
40605Beta2C2C12 cellsHUMAN3H-CGP-12177ISOPRENALINE1258.93Carter AA, et al., 2005Jan 15, 2025Jan 28, 2025
40606Beta2C2C12 cellsHUMAN3H-CGP-12177EPINEPHRINE1995.26Carter AA, et al., 2005Jan 15, 2025Jan 28, 2025
40607Beta2C2C12 cellsHUMAN3H-CGP-12177NOREPINEPHRINE3162.28Carter AA, et al., 2005Jan 15, 2025Jan 28, 2025
40608Beta2C2C12 cellsHUMAN3H-CGP-12177Terbutaline2511.89Carter AA, et al., 2005Jan 15, 2025Jan 28, 2025
40609Beta2C2C12 cellsHUMAN3H-CGP-12177Salbutamol,(+/-)501.187Carter AA, et al., 2005Jan 15, 2025Jan 28, 2025
40610Beta2C2C12 cellsHUMAN3H-CGP-12177Salmeterol25.1189Carter AA, et al., 2005Jan 15, 2025Jan 28, 2025
40611mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-tolyl)-3H-5-thia-1,3,6-triazafluoren-4-one5Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40612mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-tolyl)-3H-5-thia-1,3,6-triazafluoren-4-one890Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40613mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(o-hydroxyphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one50Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40614mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(o-hydroxyphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40615mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-fluorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one23Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40616mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-fluorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40617mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-chlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one16Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40618mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-chlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one1810Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40619mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-bromophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one4Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40620mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-bromophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one1250Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40621mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-trifluoromethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one32Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40622mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(p-trifluoromethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40623mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2,4-dimethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one17Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40624mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2,4-dimethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40625mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2,4-dichlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one45Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40626mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2,4-dichlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40627mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2'-methoxy-5'-pyridyl)-3H-5-thia-1,3,6-triazafluoren-4-one39Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40628mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2'-methoxy-5'-pyridyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40629mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(1H-indazol-6-yl)-3H-5-thia-1,3,6-triazafluoren-4-one122Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40630mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(1H-indazol-6-yl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40631mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one251Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40632mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40633mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(3-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one9Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40634mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(3-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40635mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one3Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40636mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one442Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40637mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-benzyl-3H-5-thia-1,3,6-triazafluoren-4-one281Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40638mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-benzyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40639mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(p-tolyl)-3H-5-thia-1,3,6-triazafluoren-4-one2Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40640mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(p-tolyl)-3H-5-thia-1,3,6-triazafluoren-4-one500Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40641mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(o-hydroxyphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one99Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40642mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(o-hydroxyphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40643mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(p-fluorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one8Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40644mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(p-fluorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40645mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(p-chlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one4Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40646mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(p-chlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one1030Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40647mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(p-bromophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one1Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40648mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(p-bromophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40649mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(p-trifluoromethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one8Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40650mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(p-trifluoromethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40651mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(2,4-dimethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one4Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40652mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(2,4-dimethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one2440Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40653mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(2,4-dichlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one11Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40654mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(2,4-dichlorophenyl)-3H-5-thia-1,3,6-triazafluoren-4-one2300Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40655mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(2'-methoxy-5'-pyridyl)-3H-5-thia-1,3,6-triazafluoren-4-one261Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40656mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(2'-methoxy-5'-pyridyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40657mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(1H-indazol-6-yl)-3H-5-thia-1,3,6-triazafluoren-4-one62Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40658mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(1H-indazol-6-yl)-3H-5-thia-1,3,6-triazafluoren-4-one1180Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40659mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(2-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one142Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40660mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(2-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40661mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(3-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one6Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40662mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(3-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one613Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40663mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one5Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40664mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one194Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40665mGluR5CEREBELLUMRAT3H-R2141279-Dimethylamino-3-benzyl-3H-5-thia-1,3,6-triazafluoren-4-one87Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40666mGluR5CORTEXRAT3H-MPEP9-Dimethylamino-3-benzyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40667mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-hydrogen-3H-5-thia-1,3,6-triazafluoren-4-one20Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40668mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-hydrogen-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40669mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-n-propylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one180Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40670mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-n-propylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one2040Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40671mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-isopropylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one407Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40672mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-isopropylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one3540Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40673mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-tert-butylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one8500Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40674mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-tert-butylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40675mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-cyclopropylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one87Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40676mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-cyclopropylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one4620Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40677mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-cyclohexylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40678mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-cyclohexylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40679mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopropyl-3H-5-thia-1,3,6-triazafluoren-4-one632Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40680mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopropyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40681mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclobutyl-3H-5-thia-1,3,6-triazafluoren-4-one167Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40682mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclobutyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40683mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopentyl-3H-5-thia-1,3,6-triazafluoren-4-one5Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40684mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopentyl-3H-5-thia-1,3,6-triazafluoren-4-one1160Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40685mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclohexyl-3H-5-thia-1,3,6-triazafluoren-4-one50Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40686mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclohexyl-3H-5-thia-1,3,6-triazafluoren-4-one650Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40687mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one130Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40688mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40689mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one482Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40690mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(2-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one2160Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40691mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one140Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40692mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-methylcyclohexyl)-3H-5-thia-1,3,6-triazafluoren-4-one592Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40693mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cycoheptyl-3H-5-thia-1,3,6-triazafluoren-4-one1Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40694mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cycoheptyl-3H-5-thia-1,3,6-triazafluoren-4-one147Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40695mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(N-hexamethyleneiminyl)-3H-5-thia-1,3,6-triazafluoren-4-one10Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40696mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(N-hexamethyleneiminyl)-3H-5-thia-1,3,6-triazafluoren-4-one342Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40697mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclooctyl-3H-5-thia-1,3,6-triazafluoren-4-one13Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40698mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclooctyl-3H-5-thia-1,3,6-triazafluoren-4-one179Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40699mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(1-adamantyl)-3H-5-thia-1,3,6-triazafluoren-4-one76Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40700mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(1-adamantyl)-3H-5-thia-1,3,6-triazafluoren-4-one154Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40701mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(3-n-pentyl)-3H-5-thia-1,3,6-triazafluoren-4-one335Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40702mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(3-n-pentyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40703mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopentylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one26Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40704mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclopentylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40705mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one139Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40706mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-cyclohexylmethyl-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40707mGluR5CLONEDHUMANFunctional3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one19Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40708mGluR5CLONEDHUMANFunctional3-Cycloheptyl -9-dimethylamino-3H-5-thia-1,2,3,6-tetraazafluoren-4-one816Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40709mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one44Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40710mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-methyl-3H-5-thia-1,3,6-triazafluoren-4-one344Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40711mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one84Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40712mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-ethyl-3H-5-thia-1,3,6-triazafluoren-4-one4530Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40713mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one101Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40714mGluR5CLONEDHUMANFunctional9-Dimethylamino-2-n-butyl-3H-5-thia-1,3,6-triazafluoren-4-one901Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40715mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4'-ethylphenyl)-3H-1,3,6-triazafluoren-4-one1460Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40716mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4'-ethylphenyl)-3H-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40717mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4'-methyl-1'-cyclohexyl)-3H-1,3,6-triazafluoren-4-one82Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40718mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4'-methyl-1'-cyclohexyl)-3H-1,3,6-triazafluoren-4-one901Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40719mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3-diazafluoren-4-one949Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40720mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3-diazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40721mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one183Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40722mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-ethylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one2160Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40723mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-methylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one43Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40724mGluR5CLONEDHUMANFunctional9-Dimethylamino-3-(4-methylphenyl)-3H-5-thia-1,3,7-triazafluoren-4-one4040Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40725mGluR5CLONEDHUMANFunctional9-(N,N-Ethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one37Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40726mGluR5CLONEDHUMANFunctional9-(N,N-Ethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one2570Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40727mGluR5CLONEDHUMANFunctional9-(2'-Methoxyethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one71Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40728mGluR5CLONEDHUMANFunctional9-(2'-Methoxyethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40729mGluR5CLONEDHUMANFunctional9-N-Azetidinyl-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one113Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40730mGluR5CLONEDHUMANFunctional9-N-Azetidinyl-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40731mGluR5CLONEDHUMANFunctional9-Cyclopropylamino-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one41Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40732mGluR5CLONEDHUMANFunctional9-Cyclopropylamino-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40733mGluR5CLONEDHUMANFunctional9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one49Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40734mGluR5CLONEDHUMANFunctional9-(1'-Cyanomethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one2100Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40735mGluR5CLONEDHUMANFunctional9-(2',2',2'-Trifluoroethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one99Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40736mGluR5CLONEDHUMANFunctional9-(2',2',2'-Trifluoroethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40737mGluR5CLONEDHUMANFunctional9-(Methylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one98Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40738mGluR5CLONEDHUMANFunctional9-(Methylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one5960Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40739mGluR5CLONEDHUMANFunctional9-(N,N,-Dimethyl-N-oxyamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one306Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40740mGluR5CLONEDHUMANFunctional9-(N,N,-Dimethyl-N-oxyamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
40741mGluR5CLONEDHUMANFunctional9-(N,N-Dimethyl-N-oxyamino)-3-(N-hexamethyleneiminyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one167Zheng GZ, et al., 2005Jan 15, 2025Jan 15, 2025
40742mGluR5CLONEDHUMANFunctional9-(N,N-Dimethyl-N-oxyamino)-3-(N-hexamethyleneiminyl)-3H-5-thia-1,3,6-triaza-fluoren-4-one>10000Zheng GZ, et al., 2005Jan 15, 2025Jan 28, 2025
407435-HT1ACLONEDHUMAN3H-8-OH-DPATURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407445-HT1BCLONEDHUMAN3H-GR-125743URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407455-HT1DCLONEDHUMAN3H-GR-125743URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407465-HT1ECLONEDHUMAN3H-5HTURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407475-HT2ACLONEDHUMAN3H-KETANSERINURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407485-HT2CCLONEDRAT3H-MESULERGINEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407495-HT3CLONEDHUMAN3H-ZACOPRIDEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407505-HT6CLONEDHUMAN3H-LSDURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
407515-HT7CLONEDHUMAN3H-LSDURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40752Alpha1ACLONEDHUMAN3H-PRAZOSINURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40753Alpha1BCLONEDHUMAN3H-PRAZOSINURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40754Alpha2ACLONEDHUMAN3H-CLONIDINEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40755Alpha2BCLONEDHUMAN3H-CLONIDINEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40756Alpha2CCLONEDHUMAN3H-CLONIDINEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40757Beta1CLONEDRAT125I-PindololURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40758Beta2CLONEDRAT125I-PindololURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 28, 2025
40759D1CLONEDHUMAN3H-SCH23390URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40760D2CLONEDHUMAN3H-NMSPURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40761D3CLONEDRAT3H-NMSPURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40762D4CLONEDHUMAN3H-NMSPURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40763D5CLONEDHUMAN3H-SCH23390URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40764M1CLONEDHUMAN3H-QNBURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40765M2CLONEDHUMAN3H-QNBURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40766M3CLONEDHUMAN3H-QNBURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40767M4CLONEDHUMAN3H-QNBURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40768M5CLONEDHUMAN3H-QNBURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40769CCR5CLONEDHUMAN3H-EpibatidineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40770nAChRCLONEDHUMAN3H-EpibatidineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 27, 2025
40771nAChRCLONEDHUMAN3H-EpibatidineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 27, 2025
40772nAChRCLONEDHUMAN3H-EpibatidineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 28, 2025
40773nAChRCLONEDHUMAN3H-EpibatidineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40774nAChRCLONEDHUMAN3H-EpibatidineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 27, 2025
40775CB1BRAINRAT3H-CP-55940URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40776CB2CLONEDHUMAN3H-CP-55940URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40777H1CLONEDHUMAN3H-PYRILAMINEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40778H2CLONEDHUMAN3H-TIOTIDINEURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40779MORCLONEDHUMAN3H-DiprenorphineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40780KORCLONEDHUMAN3H-BremazocineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40781Sigma 1BRAINRAT3H-Pentazocine(+)URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40782Sigma 2PC12RAT3H-DTGURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40783SLC6A4CLONEDHUMAN3H-CITALOPRAMURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40784NETCLONEDHUMAN3H-NisoxetineURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40785SLC6A3CLONEDHUMAN3H-WIN 35,428URB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40786UNDEFINEDUNDEFINEDUNDEFINEDURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40787hERGCLONEDHUMAN3H-MethylspiperoneURB 597>10000Gobbi G, et al., 2005Jan 15, 2025Jan 15, 2025
40800SLC6A4CLONEDHUMAN3H-CITALOPRAMRWAY,(-)3269PDSP Certified DataJan 15, 2025Jan 15, 2025
408015-HT1ACLONEDHUMAN3H-8-OH-DPATRWAY,(-)0.6PDSP Certified DataJan 15, 2025Jan 15, 2025
408025-HT1BCLONEDHUMAN3H-GR-125743RWAY,(-)444.7PDSP Certified DataJan 15, 2025Jan 15, 2025
408035-HT1DCLONEDHUMAN3H-GR-125743RWAY,(-)9.487PDSP Certified DataJan 15, 2025Jan 15, 2025
408045-HT2ACLONEDHUMAN3H-KETANSERINRWAY,(-)147.5PDSP Certified DataJan 15, 2025Jan 15, 2025
408055-HT2CCLONEDRAT3H-MESULERGINERWAY,(-)1682PDSP Certified DataJan 15, 2025Jan 15, 2025
40806CB1CLONEDHUMAN3H-LSDRWAY,(-)306PDSP Certified DataJan 15, 2025Jan 27, 2025
408075-HT7CLONEDHUMAN3H-LSDRWAY,(-)65.4PDSP Certified DataJan 15, 2025Jan 15, 2025
408085-HT2BCLONEDHUMAN3H-LSDRWAY,(-)7.2PDSP Certified DataJan 15, 2025Jan 15, 2025
40809Alpha1ACLONEDHUMAN3H-PRAZOSINRWAY,(-)10.35PDSP Certified DataJan 15, 2025Jan 15, 2025
40810Alpha1BCLONEDHUMAN3H-PRAZOSINRWAY,(-)222PDSP Certified DataJan 15, 2025Jan 15, 2025
40811Alpha2ACLONEDHUMAN3H-CLONIDINERWAY,(-)1311PDSP Certified DataJan 15, 2025Jan 15, 2025
40812Alpha2BCLONEDHUMAN3H-CLONIDINERWAY,(-)1476PDSP Certified DataJan 15, 2025Jan 15, 2025
40813Alpha2CCLONEDHUMAN3H-CLONIDINERWAY,(-)92PDSP Certified DataJan 15, 2025Jan 15, 2025
40814Beta1CLONEDHUMAN125I-PindololRWAY,(-)770PDSP Certified DataJan 15, 2025Jan 15, 2025
40815Beta2CLONEDHUMAN125I-PindololRWAY,(-)>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
40816H1CLONEDHUMAN3H-PYRILAMINERWAY,(-)335.4PDSP Certified DataJan 15, 2025Jan 15, 2025
40817H2CLONEDHUMAN3H-TIOTIDINERWAY,(-)3296PDSP Certified DataJan 15, 2025Jan 15, 2025
40818D1CLONEDHUMAN3H-SCH23390RWAY,(-)732PDSP Certified DataJan 15, 2025Jan 15, 2025
40819D2CLONEDHUMAN3H-NMSPRWAY,(-)34.5PDSP Certified DataJan 15, 2025Jan 15, 2025
40820D3CLONEDRAT3H-NMSPRWAY,(-)5.1PDSP Certified DataJan 15, 2025Jan 15, 2025
40821D4CLONEDHUMAN3H-NMSPRWAY,(-)15.6PDSP Certified DataJan 15, 2025Jan 15, 2025
40822KORCLONEDHUMAN3H-DiprenorphineRWAY,(-)1609PDSP Certified DataJan 15, 2025Jan 15, 2025
40843MAPK14CLONEDHUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide4.1Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40844MAPK P38CLONEDHUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide100Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40845MAPK12CLONEDHUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40846CLONEDHUMANFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40847AKTUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40848CaMKUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40849CDK2UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40850UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40851ERKUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide5000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40852FGFUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40853GSK-3UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40854HER2UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40855IGF-IRUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40856IKKUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40857JAK3UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40858LckUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40859MEKUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40860MetUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40861UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40862PKCαUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40863RafUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40864SykUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40865KDRUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40866HER1UNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40867PAKUNDEFINEDUNDEFINEDFunctional3-(5-Cyano-6-(cyclopentylamino)pyrimidin-4-ylamino)-N-(isoxazol-3-yl)-4-methylbenzamide>10000Liu C, et al., 2005Jan 15, 2025Jan 15, 2025
40868MAPK14CLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine15Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40869MAPK14CLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-methylpyridine53Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40870MAPK14CLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-fluoropyridine94Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40871MAPK14CLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine20Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40872MAPK14CLONEDHUMANFunctional2-Chloro-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine240Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40873MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]acetamide26Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40874MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]propionamide8.8Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40875MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]butyramide13Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40876MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]cyclohexanecarboxamide7.9Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40877MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-2-phenylacetamide5.6Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40878MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-3-phenylpropionamide8.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40879MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide7.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40880MAPK14CLONEDHUMANFunctionalN-Benzyl-N-[4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]amine6.7Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40881MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(2-phenylethyl)amine5.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40882MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(3-phenylpropyl)amine8.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40883MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-methylbenzamide1000Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40884MAPK14CLONEDHUMANFunctionalN-Cyclopentyl-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine3Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40885MAPK14CLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-(1-pyrrolidinyl)pyridine160Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40886MAPK14CLONEDHUMANFunctionalN-[4-[4-(3-Chlorophenyl)-2-ethyl-1,3-thiazol-5-yl]-2-pyridyl]benzamide30Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40887MAPK14CLONEDHUMANFunctionalN-[4-(2-Ethyl-4-phenyl-1,3-thiazol-5-yl)-2-pyridyl]benzamide31Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40888MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(4-fluorophenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide31Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40889MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-pyridyl]benzamide91Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40890MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(2-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide110Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40891MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(4-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide 210Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40892MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methoxyphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide120Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40893MAPK14CLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(4-methoxyphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide130Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40894MAPK14CLONEDHUMANFunctionalN-[4-[2-Methyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide13Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40895MAPK14CLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-propyl-1,3-thiazol-5-yl]-2-pyridyl]benzamide13Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40896MAPK14CLONEDHUMANFunctional4-[4-(3-Methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine14Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40897MAPK14CLONEDHUMANFunctional2-Methyl-4-[4-(3-methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine26Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40898MAPK14CLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide37Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40899MAPK14CLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-2-phenylacetamide34Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40900MAPK14CLONEDHUMANFunctionalN-Benzyl-N-[4-[4-(3-methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]amine11Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40901MAPK14CLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(2-phenylethyl)amine9.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40902TNFαCLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine73Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40903TNFαCLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-methylpyridine450Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40904TNFαCLONEDHUMANFunctional4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine130Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40905TNFαCLONEDHUMANFunctional2-Chloro-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]pyridine890Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40906TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]propionamide6.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40907TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]cyclohexanecarboxamide77Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40908TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-2-phenylacetamide13Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40909TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-3-phenylpropionamide19Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40910TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide48Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40911TNFαCLONEDHUMANFunctionalN-Benzyl-N-[4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]amine28Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40912TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(2-phenylethyl)amine42Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40913TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(3-phenylpropyl)amine120Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40914TNFαCLONEDHUMANFunctionalN-Cyclopentyl-4-[2-ethyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridylamine5.1Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40915TNFαCLONEDHUMANFunctionalN-[4-[4-(3-Chlorophenyl)-2-ethyl-1,3-thiazol-5-yl]-2-pyridyl]benzamide130Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40916TNFαCLONEDHUMANFunctionalN-[4-(2-Ethyl-4-phenyl-1,3-thiazol-5-yl)-2-pyridyl]benzamide110Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40917TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(4-fluorophenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide93Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40918TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-2-pyridyl]benzamide690Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40919TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(2-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide220Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40920TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(4-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide 450Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40921TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(3-methoxyphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide110Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40922TNFαCLONEDHUMANFunctionalN-[4-[2-Ethyl-4-(4-methoxyphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide130Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40923TNFαCLONEDHUMANFunctionalN-[4-[2-Methyl-4-(3-methylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide33Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40924TNFαCLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-propyl-1,3-thiazol-5-yl]-2-pyridyl]benzamide37Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40925TNFαCLONEDHUMANFunctional4-[4-(3-Methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine49Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40926TNFαCLONEDHUMANFunctional2-Methyl-4-[4-(3-methylphenyl)-2-[4-(methylsulfonyl)phenyl]-1,3-thiazol-5-yl]pyridine440Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40927TNFαCLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]benzamide70Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40928TNFαCLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-2-phenylacetamide61Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40929TNFαCLONEDHUMANFunctionalN-Benzyl-N-[4-[4-(3-methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]amine130Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
40930TNFαCLONEDHUMANFunctionalN-[4-[4-(3-Methylphenyl)-2-(4-methylsulfonylphenyl)-1,3-thiazol-5-yl]-2-pyridyl]-N-(2-phenylethyl)amine43Miwatashi S, et al., 2005Jan 15, 2025Jan 15, 2025
409315-HT6CLONEDHUMAN3H-LSDpiperazinoindole2700Pullagurla M, et al., 2005Jan 15, 2025Jan 15, 2025
40932SLC6A3Striatal MembranesRAT3H-WIN 35,428WIN 35,065-223Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40933SLC6A3Striatal MembranesRAT3H-WIN 35,428WIN 35,42813.9Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40934SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-321.71Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40935SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-311.12Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40936SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-551.26Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40937SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-511.69Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40938SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-881.35Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40939SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1110.79Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40940SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1120.81Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40941NETCEREBRAL CORTEXRAT3H-NisoxetineWIN 35,065-2920Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40942NETCEREBRAL CORTEXRAT3H-NisoxetineWIN 35,428835Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40943NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-3260Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40944NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-3137Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40945NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-5536Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40946NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-5137.4Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40947NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-881329Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40948NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-11117.96Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40949NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-11236.2Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40950SLC6A4MidbrainRAT3H-PAROXETINEWIN 35,065-21962Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40951SLC6A4MidbrainRAT3H-PAROXETINEWIN 35,428692Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40952SLC6A4MidbrainRAT3H-PAROXETINERTI-32240Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40953SLC6A4MidbrainRAT3H-PAROXETINERTI-3144.5Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40954SLC6A4MidbrainRAT3H-PAROXETINERTI-554.21Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40955SLC6A4MidbrainRAT3H-PAROXETINERTI-5110.6Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40956SLC6A4MidbrainRAT3H-PAROXETINERTI-88120Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40957SLC6A4MidbrainRAT3H-PAROXETINERTI-1113.13Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40958SLC6A4MidbrainRAT3H-PAROXETINERTI-11210.5Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40959SLC6A3Striatal MembranesRAT3H-WIN 35,428COCAINE89Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40960SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-12195Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40961SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-13196Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40962SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-14219Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40963SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-15112Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40964SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-52257Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40965SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-53181Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40966SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-49147Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40967SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-74371Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40968NETCEREBRAL CORTEXRAT3H-NisoxetineCOCAINE3298Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40969NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-12>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40970NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-136124Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40971NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-14>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40972NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-15>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40973NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-52>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40974NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-53>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40975NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-494893Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40976NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-74>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40977SLC6A4MidbrainRAT3H-PAROXETINECOCAINE1045Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40978SLC6A4MidbrainRAT3H-PAROXETINERTI-125801Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40979SLC6A4MidbrainRAT3H-PAROXETINERTI-134517Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40980SLC6A4MidbrainRAT3H-PAROXETINERTI-14>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40981SLC6A4MidbrainRAT3H-PAROXETINERTI-15>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40982SLC6A4MidbrainRAT3H-PAROXETINERTI-52302Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40983SLC6A4MidbrainRAT3H-PAROXETINERTI-53615Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40984SLC6A4MidbrainRAT3H-PAROXETINERTI-49374Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40985SLC6A4MidbrainRAT3H-PAROXETINERTI-74368Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40986SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-13585.1Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40987SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-13476.7Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40988SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1176.45Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40989SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-12719.1Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40990SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-14917.8Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40991SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1503.74Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40992SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1931.68Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40993SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1203.26Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40994SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2058.19Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40995SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-20981.2Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40996SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-20723.2Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40997SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-211117Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40998SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-21395.6Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
40999SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1141.4Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41000SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1900.96Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41001SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1131.98Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41002SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-11632.6Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41003SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2039.37Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41004SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-20627.4Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41005SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2043.91Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41006SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-21255Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41007SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-21071Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41008SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1210.43Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41009SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1910.61Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41010SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1221.5Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41011NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-135>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41012NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-134>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41013NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1171926Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41014NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1273444Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41015NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1492628Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41016NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1504738Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41017NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-193644Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41018NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1205833Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41019NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2052136Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41020NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2094096Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41021NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-207>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41022NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2119519Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41023NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2133151Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41024NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-114778Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41025NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-190235Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41026NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1132955Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41027NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-116967.6Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41028NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2032744Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41029NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2061277Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41030NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2044783Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41031NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2124883Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41032NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2101522Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41033NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-121285Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41034NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-191102Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41035NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1223791Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41036SLC6A4MidbrainRAT3H-PAROXETINERTI-135>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41037SLC6A4MidbrainRAT3H-PAROXETINERTI-134>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41038SLC6A4MidbrainRAT3H-PAROXETINERTI-1176090Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41039SLC6A4MidbrainRAT3H-PAROXETINERTI-1274499Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41040SLC6A4MidbrainRAT3H-PAROXETINERTI-149485Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41041SLC6A4MidbrainRAT3H-PAROXETINERTI-1502019Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41042SLC6A4MidbrainRAT3H-PAROXETINERTI-1931066Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41043SLC6A4MidbrainRAT3H-PAROXETINERTI-120>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41044SLC6A4MidbrainRAT3H-PAROXETINERTI-2055237Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41045SLC6A4MidbrainRAT3H-PAROXETINERTI-209>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41046SLC6A4MidbrainRAT3H-PAROXETINERTI-207>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41047SLC6A4MidbrainRAT3H-PAROXETINERTI-211>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41048SLC6A4MidbrainRAT3H-PAROXETINERTI-213>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41049SLC6A4MidbrainRAT3H-PAROXETINERTI-1141404Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41050SLC6A4MidbrainRAT3H-PAROXETINERTI-190168Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41051SLC6A4MidbrainRAT3H-PAROXETINERTI-1132336Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41052SLC6A4MidbrainRAT3H-PAROXETINERTI-1161227Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41053SLC6A4MidbrainRAT3H-PAROXETINERTI-2032153Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41054SLC6A4MidbrainRAT3H-PAROXETINERTI-2061203Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41055SLC6A4MidbrainRAT3H-PAROXETINERTI-2043772Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41056SLC6A4MidbrainRAT3H-PAROXETINERTI-212>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41057SLC6A4MidbrainRAT3H-PAROXETINERTI-210>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41058SLC6A4MidbrainRAT3H-PAROXETINERTI-12166.8Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41059SLC6A4MidbrainRAT3H-PAROXETINERTI-19115.5Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41060SLC6A4MidbrainRAT3H-PAROXETINERTI-122184Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41061SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-11811.5Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41062SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-10612.4Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41063SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-19610.7Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41064SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1462.05Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41065SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1291.38Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41066SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2155.48Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41067SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1830.85Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41068SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1471.38Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41069SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1566.95Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41070SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1986.57Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41071SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2081.47Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41072SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2142.9Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41073SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-22645.5Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41074SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-13341.8Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41075SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-22124.7Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41076SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-1862.55Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41077SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-22211.7Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41078SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2290.37Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41079SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2281.08Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41080SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-2270.75Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41081SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-128753Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41082SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-160127Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41083SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-19260Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41084SLC6A3Striatal MembranesRAT3H-WIN 35,428RTI-662424Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41085NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1184270Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41086NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1061584Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41087NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1969907Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41088NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-146144Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41089NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-129942Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41090NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2155532Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41091NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-183549Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41092NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1473950Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41093NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1561752Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41094NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-198990Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41095NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2081083Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41096NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2148545Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41097NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2262202Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41098NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1334398Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41099NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-2216222Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41100NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-186442Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41101NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-222>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41102NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-229991Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41103NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-228103Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41104NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-227357Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41105NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1283981Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41106NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1607329Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41107NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-1923935Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41108NETCEREBRAL CORTEXRAT3H-NisoxetineRTI-664213Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41109SLC6A4MidbrainRAT3H-PAROXETINERTI-1181621Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41110SLC6A4MidbrainRAT3H-PAROXETINERTI-1061313Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41111SLC6A4MidbrainRAT3H-PAROXETINERTI-196>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41112SLC6A4MidbrainRAT3H-PAROXETINERTI-14697.8Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41113SLC6A4MidbrainRAT3H-PAROXETINERTI-1291079Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41114SLC6A4MidbrainRAT3H-PAROXETINERTI-2159433Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41115SLC6A4MidbrainRAT3H-PAROXETINERTI-183724Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41116SLC6A4MidbrainRAT3H-PAROXETINERTI-147>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41117SLC6A4MidbrainRAT3H-PAROXETINERTI-1563470Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41118SLC6A4MidbrainRAT3H-PAROXETINERTI-198814Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41119SLC6A4MidbrainRAT3H-PAROXETINERTI-2082470Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41120SLC6A4MidbrainRAT3H-PAROXETINERTI-214>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41121SLC6A4MidbrainRAT3H-PAROXETINERTI-226>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41122SLC6A4MidbrainRAT3H-PAROXETINERTI-1336371Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41123SLC6A4MidbrainRAT3H-PAROXETINERTI-221>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41124SLC6A4MidbrainRAT3H-PAROXETINERTI-1863402Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41125SLC6A4MidbrainRAT3H-PAROXETINERTI-222>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41126SLC6A4MidbrainRAT3H-PAROXETINERTI-2291728Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41127SLC6A4MidbrainRAT3H-PAROXETINERTI-22873.9Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41128SLC6A4MidbrainRAT3H-PAROXETINERTI-227130Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41129SLC6A4MidbrainRAT3H-PAROXETINERTI-128>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41130SLC6A4MidbrainRAT3H-PAROXETINERTI-160>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41131SLC6A4MidbrainRAT3H-PAROXETINERTI-192>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41132SLC6A4MidbrainRAT3H-PAROXETINERTI-66>10000Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41133SLC6A3Striatal MembranesRAT3H-dopamineCOCAINE241.3Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41134SLC6A3Striatal MembranesRAT3H-dopamineWIN 35,065-249.8Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41135SLC6A3Striatal MembranesRAT3H-dopamineWIN 35,42822.95Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41136SLC6A3Striatal MembranesRAT3H-dopamineRTI-327.02Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41137SLC6A3Striatal MembranesRAT3H-dopamineRTI-313.68Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41138SLC6A3Striatal MembranesRAT3H-dopamineRTI-551.96Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41139SLC6A3Striatal MembranesRAT3H-dopamineRTI-11715.31Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41140SLC6A3Striatal MembranesRAT3H-dopamineRTI-1209.13Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41141SLC6A3Striatal MembranesRAT3H-dopamineRTI-1146.04Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41142SLC6A3Striatal MembranesRAT3H-dopamineRTI-1135.25Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41143SLC6A3Striatal MembranesRAT3H-dopamineRTI-1212.79Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41144SLC6A3Striatal MembranesRAT3H-dopamineRTI-1226.85Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41145NETFR. CORTEXRAT3H-NorepinephrineCOCAINE160.55Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41146NETFR. CORTEXRAT3H-NorepinephrineWIN 35,065-237.2Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41147NETFR. CORTEXRAT3H-NorepinephrineWIN 35,42838.59Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41148NETFR. CORTEXRAT3H-NorepinephrineRTI-328.42Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41149NETFR. CORTEXRAT3H-NorepinephrineRTI-315.86Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41150NETFR. CORTEXRAT3H-NorepinephrineRTI-557.51Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41151NETFR. CORTEXRAT3H-NorepinephrineRTI-11773.43Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41152NETFR. CORTEXRAT3H-NorepinephrineRTI-120277.66Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41153NETFR. CORTEXRAT3H-NorepinephrineRTI-114250.32Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41154NETFR. CORTEXRAT3H-NorepinephrineRTI-113242.29Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41155NETFR. CORTEXRAT3H-NorepinephrineRTI-12141.22Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41156NETFR. CORTEXRAT3H-NorepinephrineRTI-12232.73Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41157SLC6A4MidbrainRAT3H-5HTCOCAINE112.11Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41158SLC6A4MidbrainRAT3H-5HTWIN 35,065-2172.79Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41159SLC6A4MidbrainRAT3H-5HTWIN 35,428100.56Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41160SLC6A4MidbrainRAT3H-5HTRTI-3219.38Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41161SLC6A4MidbrainRAT3H-5HTRTI-315Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41162SLC6A4MidbrainRAT3H-5HTRTI-551.74Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41163SLC6A4MidbrainRAT3H-5HTRTI-117917.11Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41164SLC6A4MidbrainRAT3H-5HTRTI-1201537.14Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41165SLC6A4MidbrainRAT3H-5HTRTI-114128.62Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41166SLC6A4MidbrainRAT3H-5HTRTI-113390.68Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41167SLC6A4MidbrainRAT3H-5HTRTI-12112.54Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41168SLC6A4MidbrainRAT3H-5HTRTI-12251.64Carroll FI, et al., 1995Jan 15, 2025Jan 15, 2025
41169CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-2-ylpiperazine-1-carboxamide Hydrochloride7800Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41170CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-3-ylpiperazine-1-carboxamide Hydrochloride120Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41171CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyridin-4-ylpiperazine-1-carboxamide Hydrochloride140Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41172CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-2-ylpiperazine-1-carboxamide>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41173CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-4-ylpiperazine-1-carboxamide4600Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41174CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-pyrimidin-5-ylpiperazine-1-carboxamide1000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41175CLONEDHUMANFunctionalbicalutamide890Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41176CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(1-oxidopyridin-3-yl)piperazine-1-carboxamide>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41177CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(2-methylpyridin-3-yl)piperazine-1-carboxamide 680Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41178CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(4-methylpyridin-3-yl)piperazine-1-carboxamide330Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41179CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(5-methylpyridin-3-yl)piperazine-1-carboxamide hydrochloride250Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41180CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-(6-methylpyridin-3-yl)piperazine-1-carboxamide130Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41181CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(2-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide190Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41182CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(4-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide Hydrochloride1200Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41183CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(5-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide440Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41184CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(6-methoxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide170Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41185CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(methylthio)pyridin-3-yl]piperazine-1-carboxamide220Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41186CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-N-(6-hydroxypyridin-3-yl)-2,5-dimethylpiperazine-1-carboxamide>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41187CLONEDHUMANFunctional(+/-)-trans-N-(6-Chloropyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide730Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41188CLONEDHUMANFunctional(+/-)-Methyl 5-[({trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazin-1-yl}carbonyl)amino]pyridine-2-carboxylate470Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41189CLONEDHUMANFunctional(+/-)-trans-N-(6-Acetylpyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide500Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41190CLONEDHUMANFunctional(+/-)-trans-N-(6-Cyanopyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide 200Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41191CLONEDHUMANFunctional(+/-)-trans-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]piperazine-1-carboxamide210Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41192CLONEDHUMANFunctionalYM580110Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41193CLONEDHUMANFunctional(-)-(2S,5R)-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3-yl]piperazine-1-carboxamide1300Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41194ADKrecombinantHUMANFunctional4-Amino-5-iodo-7-(4'-C-spirocyclopropyl-beta-D-erythro-pentofuranosyl)pyrrolo[2,3-d]pyrimidine600Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41195ADKrecombinantHUMANFunctional4-Amino-5-iodo-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine6Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41196ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-phenyl-7-(4'-C-spirocyclopropyl-beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine0.3Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41197ADKrecombinantHUMANFunctional4-N-Phenylamino-5-phenyl-7-(5'-deoxy-4'-C-methyl-beta-D-ribo-furanosyl)pyrrolo[2,3-d]pyrimidine4000Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41198ADKrecombinantHUMANFunctional4-N-Phenylamino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine4Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41199ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine6Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41200ADKrecombinantHUMANFunctional4-N-(4-Bromophenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine5Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41201ADKrecombinantHUMANFunctional4-N-(4-Ethoxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine3Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41202ADKrecombinantHUMANFunctional4-N-(3-Ethoxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine2Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41203ADKrecombinantHUMANFunctional4-N-(3,4-Ethylenedioxyphenyl)amino-5-phenyl-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine4Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41204ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-(3-aminophenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine10Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41205ADKrecombinantHUMANFunctional4-N-(4-Cyanophenyl)amino-5-(4-ethoxyphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine2Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41206ADKrecombinantHUMANFunctional4-N-(4-Cyanophenyl)amino-5-(4-chlorophenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine7Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41207ADKrecombinantHUMANFunctional4-N-(3,4-Ethylenedioxyphenyl)amino-5-(2-methylphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine1Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41208ADKrecombinantHUMANFunctional4-N-(2-Methoxyphenyl)amino-5-(4-ethoxyphenyl)-7-(beta-D-erythro-furanosyl)pyrrolo[2,3-d]pyrimidine5.3Boyer SH, et al., 2005Jan 15, 2025Jan 15, 2025
41209CB1BRAINRAT3H-CP-55940AM36771.3Li C, et al., 2005Jan 15, 2025Jan 15, 2025
41210CB1BRAINRAT3H-CP-55940AM36610.9Li C, et al., 2005Jan 15, 2025Jan 15, 2025
41211CB1BRAINRAT3H-CP-55940ACPA2.7Li C, et al., 2005Jan 15, 2025Jan 15, 2025
41212CB2SPLEENMOUSE3H-CP-55940AM367748.5Li C, et al., 2005Jan 15, 2025Jan 15, 2025
41213CB2SPLEENMOUSE3H-CP-55940AM366157.6Li C, et al., 2005Jan 15, 2025Jan 15, 2025
41214CB2SPLEENMOUSE3H-CP-55940ACPA157Li C, et al., 2005Jan 15, 2025Jan 15, 2025
41215CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile9300Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41216CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-phenylpiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41217CLONEDHUMAN125I-Chemokine5-(4-(3-Chloro-4-trifluoromethylphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41218CLONEDHUMAN125I-Chemokine5-(4-(4-Bromophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41219CLONEDHUMAN125I-Chemokine5-(4-(4-Methoxyphenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41220CLONEDHUMAN125I-Chemokine5-(4-(3,4-Dichlorophenyl)-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41221CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-p-tolylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41222CLONEDHUMAN125I-Chemokine5-(4-Benzyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41223CLONEDHUMAN125I-Chemokine5-(4-Hydroxy-4-methylpiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41224CLONEDHUMAN125I-Chemokine5-(4-Butyl-4-hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41225CLONEDHUMAN125I-Chemokine5-(4-Hydroxypiperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41226CLONEDHUMAN125I-Chemokine1-(4-Cyano-4,4-diphenylbutyl)-4-phenylpiperidine-4-carbonitrile >10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41227CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)piperidin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41228CLONEDHUMAN125I-Chemokine1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Amide>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41229CLONEDHUMAN125I-Chemokine1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Ethyl Ester Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41230CLONEDHUMAN125I-Chemokine1-(4-Cyano-4,4-diphenylbutyl)piperidine-4-carboxylic Acid Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41231CLONEDHUMAN125I-Chemokine5-(4-(Diphenylmethylene)piperidin-1-yl)-2,2-diphenylpentanenitrile Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41232CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-cyano-4,4-diphenylbutyl)-4-hydroxy-1-methylpiperidinium Iodide>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41233CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)piperazin-1-yl)-2,2-diphenypentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41234CLONEDHUMAN125I-Chemokine5-(4-(4-Chlorophenyl)-3,6-dihydro-2H-pyridin-1-yl)-2,2-diphenylpentanenitrile>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41235CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4,4-diphenylbutyl)piperidin-4-ol 6500Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41236CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(3-phenoxypropyl)piperidin-4-ol >10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41237CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-phenylbutyl)piperidin-4-ol>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41238CLONEDHUMAN125I-Chemokine4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-1-phenylbutan-1-one>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41239CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-hydroxy-4-phenylbutyl)piperidin-4-ol >10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41240CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-(4-methoxyphenyl)-4-phenylbutyl)piperidin-4-ol>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41241CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-(3,4-dichlorophenyl)-4-phenylbutyl)piperidin-4-ol Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41242CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-(4-chlorophenyl)-4-phenylbutyl)piperidin-4-ol >10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41243CLONEDHUMAN125I-Chemokine1-(4,4-Bis(4-chlorophenyl)butyl)-4-(4-chlorophenyl)piperidin-4-ol Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41244CLONEDHUMAN125I-ChemokineC28H32NClO5500Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41245CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-phenyl-4-m-tolylbutyl)piperidin-4-ol Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41246CLONEDHUMAN125I-Chemokine4-(4-Chlorophenyl)-1-(4-phenyl-4-p-tolylbutyl)piperidin-4-ol Hydrochloride>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41247CLONEDHUMAN125I-Chemokine1-(4-Biphenyl-4-y)-4-(4-chlorophenyl)butyl]-4-(4-chlorophenyl)piperidin-4-ol>10000Hulshof JW, et al., 2005Jan 15, 2025Jan 15, 2025
41248UNDEFINEDRATFunctionalYM5803300Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41249UNDEFINEDRATFunctionalbicalutamide7200Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41250CLONEDHUMANFunctionalYM580>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41251CLONEDHUMANFunctionalbicalutamide>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41252CLONEDHUMANFunctionalYM580>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41253CLONEDHUMANFunctionalbicalutamide>10000Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41254CLONEDHUMANFunctional(+/-)-trans-N-(6-Aminopyridin-3-yl)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethylpiperazine-1-carboxamide370Kinoyama I, et al., 2006Jan 15, 2025Jan 15, 2025
41255SLC6A4CLONEDHUMAN3H-PAROXETINECHLORIMIPRAMINE0.3Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41256SLC6A4CLONEDHUMAN3H-PAROXETINEDuloxetine0.8Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41257SLC6A4CLONEDHUMAN3H-PAROXETINEMilnacipran123Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41258SLC6A4CLONEDHUMAN3H-PAROXETINEVenlafaxine82Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41259SLC6A4CLONEDHUMAN3H-PAROXETINEDESIPRAMINE179Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41260SLC6A4CLONEDHUMAN3H-PAROXETINESERTRALINE0.9Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41261NETCLONEDHUMAN3H-NisoxetineCHLORIMIPRAMINE38Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41262NETCLONEDHUMAN3H-NisoxetineDuloxetine7.5Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41263NETCLONEDHUMAN3H-NisoxetineMilnacipran200Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41264NETCLONEDHUMAN3H-NisoxetineVenlafaxine2483Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41265NETCLONEDHUMAN3H-NisoxetineDESIPRAMINE3.8Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41266NETCLONEDHUMAN3H-NisoxetineSERTRALINE715Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41267SLC6A3CLONEDHUMAN3H-WIN 35,428CHLORIMIPRAMINE2190Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41268SLC6A3CLONEDHUMAN3H-WIN 35,428Duloxetine240Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41269SLC6A3CLONEDHUMAN3H-WIN 35,428Milnacipran>10000Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41270SLC6A3CLONEDHUMAN3H-WIN 35,428Venlafaxine7647Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41271SLC6A3CLONEDHUMAN3H-WIN 35,428DESIPRAMINE>10000Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41272SLC6A3CLONEDHUMAN3H-WIN 35,428SERTRALINE26Koch S, et al., 2003Jan 15, 2025Jan 15, 2025
41273D1CLONEDHUMANFunctionalLE30060.4Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41274D1CLONEDHUMANFunctional7-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine170Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41275D1CLONEDHUMANFunctional3-Methyl-6-phenyl-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole742Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41276D1CLONEDHUMANFunctional3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine1000Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41277D1CLONEDHUMANFunctional6-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine207Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41278D1CLONEDHUMANFunctional7-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine40.4Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41279D1CLONEDHUMANFunctional7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide20.7Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41280D1CLONEDHUMANFunctionalLE4006.93Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41281D2CLONEDHUMANFunctionalLE30019Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41282D2CLONEDHUMANFunctional7-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine82.6Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41283D2CLONEDHUMANFunctional3-Methyl-6-phenyl-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole943Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41284D2CLONEDHUMANFunctional3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine264Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41285D2CLONEDHUMANFunctional6-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine92Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41286D2CLONEDHUMANFunctional7-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine8.47Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41287D2CLONEDHUMANFunctional7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide65.7Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41288D2CLONEDHUMANFunctionalLE40033.5Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41289D5CLONEDHUMANFunctionalLE30012.7Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41290D5CLONEDHUMANFunctional7-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine22.3Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41291D5CLONEDHUMANFunctional3-Methyl-6-phenyl-1,2,3,4,5,6,7,8-octahydroazonino[5,4-b]indole112Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41292D5CLONEDHUMANFunctional3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine337Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41293D5CLONEDHUMANFunctional6-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine33.7Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41294D5CLONEDHUMANFunctional7-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine3.09Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41295D5CLONEDHUMANFunctional7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide2.32Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41296D5CLONEDHUMANFunctionalLE4001.69Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41297D1CLONEDHUMAN3H-SCH23390LE3001.9Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41298D1CLONEDHUMAN3H-SCH233907-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine16.4Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41299D1CLONEDHUMAN3H-SCH233907-Cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine767Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41300D1CLONEDHUMAN3H-SCH233903,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine61Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41301D1CLONEDHUMAN3H-SCH233906-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine10.7Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41302D1CLONEDHUMAN3H-SCH233907-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine4.5Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41303D1CLONEDHUMAN3H-SCH233902,3-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine509Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41304D1CLONEDHUMAN3H-SCH233907-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide341Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41305D1CLONEDHUMAN3H-SCH23390LE4000.39Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41306D2CLONEDHUMAN3H-SPIPERONELE30044.7Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41307D2CLONEDHUMAN3H-SPIPERONE7-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine253Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41308D2CLONEDHUMAN3H-SPIPERONE7-Cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine5000Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41309D2CLONEDHUMAN3H-SPIPERONE3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine712Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41310D2CLONEDHUMAN3H-SPIPERONE6-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine198Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41311D2CLONEDHUMAN3H-SPIPERONE7-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine56.5Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41312D2CLONEDHUMAN3H-SPIPERONE2,3-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine5000Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41313D2CLONEDHUMAN3H-SPIPERONE7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide5000Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41314D2CLONEDHUMAN3H-SPIPERONELE40017.5Hoefgen B, et al., 2006Jan 15, 2025Jan 27, 2025
41315D4CLONEDHUMAN3H-SPIPERONELE300109Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41316D4CLONEDHUMAN3H-SPIPERONE7-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine378.5Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41317D4CLONEDHUMAN3H-SPIPERONE7-Cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine5000Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41318D4CLONEDHUMAN3H-SPIPERONE3,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine1647Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41319D4CLONEDHUMAN3H-SPIPERONE6-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine299Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41320D4CLONEDHUMAN3H-SPIPERONE7-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine134Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41321D4CLONEDHUMAN3H-SPIPERONE2,3-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine2514Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41322D4CLONEDHUMAN3H-SPIPERONE7-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide165Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41323D4CLONEDHUMAN3H-SPIPERONELE40011.3Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41324D5CLONEDHUMAN3H-SCH23390LE3007.5Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41325D5CLONEDHUMAN3H-SCH233907-Ethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine14.7Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41326D5CLONEDHUMAN3H-SCH233907-Cyclopropylmethyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine893Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41327D5CLONEDHUMAN3H-SCH233903,6-dimethyl-4,5,6,7,8,13-hexahydro-3H-benzo[d]pyrrolo[3,2-g]azecine361Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41328D5CLONEDHUMAN3H-SCH233906-Methyl-4,5,6,7,8,13-hexahydrothieno[2,3-f][3]benzazecine79.1Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41329D5CLONEDHUMAN3H-SCH233907-Methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine11.2Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41330D5CLONEDHUMAN3H-SCH233902,3-Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine2610Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41331D5CLONEDHUMAN3H-SCH233907-Methyl-2,3-dihydroxy-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine hydrobromide1078Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41332D5CLONEDHUMAN3H-SCH23390LE4001.5Hoefgen B, et al., 2006Jan 15, 2025Jan 15, 2025
41333CLONEDHUMANFunctional2,3-dichloro-alpha-methyl benzylamine1330Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41334CLONEDHUMANFunctional3,4-dichloro amphetamine>10000Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41335CLONEDHUMANFunctionalSKF 296612840Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41336CLONEDHUMANFunctional7-nitro-THIQ2360Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41337CLONEDHUMANFunctional2,3-dichloro-alpha-methyl benzylamine72Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41338CLONEDHUMANFunctional3,4-dichloro amphetamine2270Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41339CLONEDHUMANFunctionalSKF 2966157Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41340CLONEDHUMANFunctional7-nitro-THIQ56Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41341CLONEDHUMANUNDEFINEDSKF 641391.55Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41342CLONEDHUMANUNDEFINEDSKF 296610.12Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41343CLONEDHUMANUNDEFINEDLY 1340464.4Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41344CLONEDHUMANUNDEFINED7-iodo-THIQ0.04Wu Q, et al., 2005Jan 15, 2025Jan 15, 2025
41345ADKrecombinantHUMANFunctional4-Amino-5-iodo-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine68Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41346ADKrecombinantHUMANFunctional4-Amino-5-bromo-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine280Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41347ADKrecombinantHUMANFunctional4-Amino-5-iodo-7-(5-O-methyl-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine2000Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41348ADKrecombinantHUMANFunctional4-Amino-5-iodo-7-(5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine400Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41349ADKrecombinantHUMANFunctional4-Amino-5-bromo-7-(5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine>10000Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41350ADKrecombinantHUMANFunctional5-Phenyl-4-N-phenylamino-7-alpha-L-lyxofuranosylpyrrolo[2,3-d]pyrimidine0.47Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41351ADKrecombinantHUMANFunctional4-N-(4-Fluorophenyl)amino-5-phenyl-7-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine1.5Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41352ADKrecombinantHUMANFunctional5-Phenyl-4-N-phenylamino-7-(5-O-methyl-alpha-L-lyxofuranosyl)pyrrolo[2,3- d]pyrimidine15Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41353ADKrecombinantHUMANFunctional5-Phenyl-4-N-phenylamino-7-(5-deoxy-alpha-L-lyxofuranosylpyrrolo[2,3- d]pyrimidine0.8Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41354ADKrecombinantHUMANFunctional4-Amino-3-bromo-1-alpha-L-lyxofuranosylpyrazolo[3,4-d]pyrimidine>10000Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41355ADKrecombinantHUMANFunctional3-Phenyl-4-N-phenylamino-1-alpha-L-lyxofuranosylpyrazolo[3,4-d]pyrimidine2.8Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41356ADKrecombinantHUMANFunctional9-alpha-L-Lyxofuranosyladenine1000Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41357ADKrecombinantHUMANFunctional4-Amino-5-iodo-7-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrrolo[2,3-d]pyrimidine16Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41358ADKrecombinantHUMANFunctional5-Phenyl-4-N-phenylamino-7-(5-amino-5-deoxy-alpha-L- lyxofuranosylpyrrolo[2,3-d]pyrimidine36Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41359ADKrecombinantHUMANFunctional9-(5-Amino-5-deoxy-alpha-L-lyxofuranosyl)adenine>10000Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41360ADKrecombinantHUMANFunctional4-Amino-3-bromo-1-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrazolo[3,4-d]pyrimidine170Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41361ADKrecombinantHUMANFunctional3-Phenyl-4-N-phenylamino-1-(5-amino-5-deoxy-alpha-L-lyxofuranosyl)pyrazolo[3,4-d]pyrimidine42Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41362ADKrecombinantHUMANFunctional5'-amino-5'-deoxy- 5-iodotubercidin5Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41363ADKrecombinantHUMANFunctional5'-deoxy-5-iodotubercidin26Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
41364ADKrecombinantHUMANFunctionalGP 5154Ugarkar BG, et al., 2003Jan 15, 2025Jan 15, 2025
413655-HT1ACLONEDHUMAN3H-8-OH-DPAT2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione1.36Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
413665-HT2ACLONEDHUMAN3H-KETANSERIN2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione41.5Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
413675-HT2CCLONEDRAT3H-MESULERGINE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione99.6Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
413685-HT3CLONEDHUMAN3H-ZACOPRIDE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
413695-HT5ACLONEDHUMAN3H-LSD2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione228.6Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
413705-HT6CLONEDHUMAN3H-LSD2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione120.3Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
413715-HT7CLONEDHUMAN3H-LSD2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione9.1Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41372UNDEFINEDUNDEFINED3H-NECA2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41373A3UNDEFINEDUNDEFINED3H-NMSP2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41374UNDEFINEDUNDEFINED3H-NMSP2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41375CLONEDHUMAN125I-HEAT2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione32.2Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41376Alpha2ACLONEDHUMAN3H-CLONIDINE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione1012Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41377Alpha2BCLONEDHUMAN3H-CLONIDINE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione316.2Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41378Alpha2CCLONEDHUMAN3H-CLONIDINE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione23.7Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41379Beta1CLONEDRAT125I-Pindolol2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione475.8Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41380Beta2CLONEDRAT125I-Pindolol2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione60.6Kumar JS, et al., 2006Jan 15, 2025Jan 28, 2025
41381Beta3CLONEDRAT125I-Pindolol2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41382GABAAUNDEFINEDRAT3H-RO-15-17882-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41383HEARTRAT3H-Nitrendipine2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41384NETCLONEDHUMAN3H-Nisoxetine2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione6980Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41385Sigma 1BRAINRAT3H-Pentazocine(+)2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione480Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41386CLONEDHUMAN3H-VASOPRESSIN2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41387V2CLONEDHUMAN3H-VASOPRESSIN2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41388BRAINRAT3H-Batrachotoxin2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41389CB1BRAINRAT3H-CP-559402-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41390CB2CLONEDHUMAN3H-CP-559402-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41391D1CLONEDHUMAN3H-SCH233902-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione7396Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41392D2CLONEDHUMAN3H-NMSP2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione22.01Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41393D3CLONEDRAT3H-NMSP2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione62.8Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41394D4CLONEDHUMAN3H-NMSP2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione8.5Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41395D5CLONEDHUMAN3H-NMSP2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41396SLC6A3CLONEDHUMAN3H-WIN 35,4282-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione407.4Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41397DORUNDEFINEDGUINEA PIG3H-DADLE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41398UNDEFINEDRAT3H-MUSCIMOL2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41399H1CLONEDHUMAN3H-PYRILAMINE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione150Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41400H2CLONEDHUMAN3H-TIOTIDINE2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione302Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41401H3CLONEDGUINEA PIG3H-Alpha-Me-histamine2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41402H4CLONEDHUMAN3H-Histamine2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41403hERGUNDEFINEDUNDEFINEDUNDEFINED2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41404KORCLONEDHUMAN3H-Bremazocine2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41405CLONEDHUMAN3H-QNB2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41406UNDEFINEDUNDEFINEDFunctional2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41407MORCLONEDHUMAN3H-Diprenorphine2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41408mGluR5CLONEDRATFunctional2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41409NMDAUNDEFINEDRAT3H-MK-8012-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 28, 2025
41410SLC6A4CLONEDHUMAN3H-CITALOPRAM2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione6144Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41411Sigma 2PC12RAT3H-DTG2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41412VMAT1UNDEFINEDUNDEFINEDUNDEFINED2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41413VMAT2UNDEFINEDUNDEFINEDUNDEFINED2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41414NTSR1UNDEFINEDUNDEFINED125I-Tyr3, NT2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41415I1PC12RAT125I-Pindolol2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41416AMPAFOREBRAINRAT3H-AMPA2-{4-[4-(7-Methoxy-naphthalen-1-yl)piperazin-1-yl]-butyl}-4-methyl-2H-[1,2,4]triazine-3,5-dione>10000Kumar JS, et al., 2006Jan 15, 2025Jan 15, 2025
41417IPCLONEDUNDEFINED3H-PGI2PGI216.6Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41418IPCLONEDUNDEFINED3H-PGI2PGE1137Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41419IPCLONEDUNDEFINED3H-PGI2PGE1, 13,14-dihydro315Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41420IPCLONEDUNDEFINED3H-PGI2PGE1, 8-iso735Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41421IPCLONEDUNDEFINED3H-PGI2PGE2, 5,6-trans735Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41422IPCLONEDUNDEFINED3H-PGI2PGE2,17-Phenyl4370Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41423IPCLONEDUNDEFINED3H-PGI2PGI1, 6beta7350Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41424IPCLONEDUNDEFINED3H-PGI2PGE2 13,14-dihydro8410Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41425IPCLONEDUNDEFINED3H-PGI2PGE2>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41426IPCLONEDUNDEFINED3H-PGI2PGE2, 13,14-dihydro15-oxo>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41427IPCLONEDUNDEFINED3H-PGI2PGE2, 15-epi>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41428IPCLONEDUNDEFINED3H-PGI2PGF1alpha>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41429IPCLONEDUNDEFINED3H-PGI2PGF1alpha, 6-oxo>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41430IPCLONEDUNDEFINED3H-PGI2PGF2Alpha>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41431IPCLONEDUNDEFINEDFunctionalPGD1>10000Blair IA, et al., 1981Jan 15, 2025Jan 28, 2025
41432CB1CEREBELLUMRAT3H-CP-55940CP 55,9400.55Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41433CB1CEREBELLUMRAT3H-CP-55940Noladin Ether, NE9.14Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41434CB1CEREBELLUMRAT3H-CP-559402-AG1750Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41435CB2CLONEDHUMAN3H-CP-55940CP 55,9400.58Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41436CB2CLONEDHUMAN3H-CP-55940Noladin Ether, NE480Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41437CB2CLONEDHUMAN3H-CP-559402-AG1016Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41438CB2CLONEDHUMAN35S-GTPGammaSCP 55,9400.39Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41439CB2CLONEDHUMAN35S-GTPGammaSNoladin Ether, NE35Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41440CB2CLONEDHUMAN35S-GTPGammaS2-AG230Shoemaker JL, et.al., 2005Jan 15, 2025Jan 15, 2025
41441recombinantHUMAN3H-TCAAtorvastatin9120Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41442recombinantHUMAN3H-TCACerivastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41443recombinantHUMAN3H-TCAFluvastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41444recombinantHUMAN3H-TCAPitavastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41445recombinantHUMAN3H-TCAPravastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41446recombinantHUMAN3H-TCARosuvastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41447recombinantHUMAN3H-TCASimvastatin acid>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41448recombinantHUMAN3H-TCAAtorvastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41449recombinantHUMAN3H-TCAPitavastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41450recombinantHUMAN3H-TCAPravastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41451recombinantHUMAN3H-TCASimvastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41452recombinantRAT3H-TCAAtorvastatin7570Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41453recombinantRAT3H-TCACerivastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41454recombinantRAT3H-TCAFluvastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41455recombinantRAT3H-TCAPitavastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41456recombinantRAT3H-TCAPravastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41457recombinantRAT3H-TCARosuvastatin>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41458recombinantRAT3H-TCASimvastatin acid>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41459recombinantRAT3H-TCAAtorvastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41460recombinantRAT3H-TCAPitavastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41461recombinantRAT3H-TCAPravastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41462recombinantRAT3H-TCASimvastatin lactone>10000Hirano M, et al., 2005Jan 15, 2025Jan 15, 2025
41463A1CEREBRAL CORTEXRAT3H-cyclohexyladenosine1,3-Diallylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41464A1CORTEXRAT3H-cyclohexyladenosinecaffeine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41465A1CORTEXRAT3H-cyclohexyladenosine3,7-dimethyl-1-n-propylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41466A1CORTEXRAT3H-cyclohexyladenosine1-allyl-3,7-dimethylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41467A1CORTEXRAT3H-cyclohexyladenosine3,7-dimethyl-1-proporgylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41468A1CORTEXRAT3H-cyclohexyladenosine1,7-dimethyl-3-n-propylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41469A1CORTEXRAT3H-cyclohexyladenosine1,7-dimethyl-3-isobutylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41470A1CORTEXRAT3H-cyclohexyladenosine7-(n-propyl)-theophylline>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41471A1CORTEXRAT3H-cyclohexyladenosine7-(allyl)-theophylline>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41472A1CORTEXRAT3H-cyclohexyladenosine7-(propargyl)-theophylline>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41473A1CORTEXRAT3H-cyclohexyladenosine7-(beta-chloroethyl)-theophylline8000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41474A1CORTEXRAT3H-cyclohexyladenosine7-(beta-hydroxyethyl)-theophylline>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41475A1CORTEXRAT3H-cyclohexyladenosine7-(beta-acetoxyethyl)-theophylline>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41476A1CORTEXRAT3H-cyclohexyladenosine7-(benzyl)-theophylline6000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41477A1CORTEXRAT3H-cyclohexyladenosine7-CH3-methyl-1,3-n-dipropyl-xantine7000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41478A1CORTEXRAT3H-cyclohexyladenosine1,3-diallyl-7-methylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41479A1CORTEXRAT3H-cyclohexyladenosine3-isobutyl-1-methyl-7-n-propylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41480A1CORTEXRAT3H-cyclohexyladenosine7-allyl-3-isobutyl-1-methylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41481A1CORTEXRAT3H-cyclohexyladenosine3-isobutyl-1-methyl-7-propargylxantine3100Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41482A1CORTEXRAT3H-cyclohexyladenosine7-benzyl-3-isobutyl-1-methylxantine9000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41483A1CORTEXRAT3H-cyclohexyladenosine1,3,7-n-tripropylxantine2600Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41484A1CORTEXRAT3H-cyclohexyladenosine7-allyl-1,3-n-dipropylxantine1900Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41485A1CORTEXRAT3H-cyclohexyladenosine1,3-n-dipropyl-7-propargyl600Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41486A1CORTEXRAT3H-cyclohexyladenosine7-benzyl-1,3-n-dipropylxantine1000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41487A1CORTEXRAT3H-cyclohexyladenosinetheophylline>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41488A1CORTEXRAT3H-cyclohexyladenosine1-ethyl-3-methylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41489A1CORTEXRAT3H-cyclohexyladenosine1-beta-hydroxyethyl-3-methylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41490A1CORTEXRAT3H-cyclohexyladenosine3-isopropyl-1-methyl>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41491A1CORTEXRAT3H-cyclohexyladenosine3-isobutyl-1-methylxantine7000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41492A1CORTEXRAT3H-cyclohexyladenosine3-beta-hydroxyethyl-1-methylxantine>10000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41493A1CORTEXRAT3H-cyclohexyladenosine1,3-diethylxantine3300Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41494A1CORTEXRAT3H-cyclohexyladenosine1,3-n-dipropylxantine700Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41495A1CORTEXRAT3H-cyclohexyladenosine1,3-diisobutylxantine500Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41496A1CORTEXRAT3H-cyclohexyladenosine1,3-dibenzylxantine2000Daly JW et al., 1986Jan 15, 2025Jan 15, 2025
41497CLONEDHUMAN3H-dexamethasoneciclesonide37Belvisi MG, et al., 2005Jan 15, 2025Jan 15, 2025
41498CLONEDHUMAN3H-dexamethasonedes-CIC0.31Belvisi MG, et al., 2005Jan 15, 2025Jan 15, 2025
41499CLONEDHUMAN3H-dexamethasoneFluticasone0.238Belvisi MG, et al., 2005Jan 15, 2025Jan 15, 2025
41500CLONEDHUMAN3H-dexamethasonedexamethasone6.7Belvisi MG, et al., 2005Jan 15, 2025Jan 15, 2025
41501mGluR5CLONEDRATFunctional4-(3-Fluorophenylethynyl)-2-methylthiazole23Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41502mGluR5CLONEDRATFunctional4-(4-Fluorophenylethynyl)-2-methylthiazole2966Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41503mGluR5CLONEDRATFunctional4-(2-Fluorophenylethynyl)-2-methylthiazole140Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41504mGluR5CLONEDRATFunctional4-(3,5-Difluorophenylethynyl)-2-methylthiazole25.3Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41505mGluR5CLONEDRATFunctional4-(3-Methoxyphenylethynyl)-2-methylthiazole49Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41506mGluR5CLONEDRATFunctional4-(2-Methoxyphenylethynyl)-2-methylthiazole36.3Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41507mGluR5CLONEDRATFunctional2-Methyl-4-(m-tolylethynyl)thiazole82.6Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41508mGluR5CLONEDRATFunctional4-(3-Chlorophenylethynyl)-2-methylthiazole129Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41509mGluR5CLONEDRATFunctional2-Methyl-4-[[3-(trifluoromethyl)phenyl]ethynyl]thiazole413Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41510mGluR5CLONEDRATFunctional2-Methyl-4-[[3-(trifluoromethoxy)phenyl]ethynyl]thiazole266Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41511mGluR5CLONEDRATFunctional3-[(2-Methyl-4-thiazolyl)ethynyl]benzonitrile0.94Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41512mGluR5CLONEDRATFunctionalN-[3-[(2-Methyl-4-thiazolyl)ethynyl]phenyl]acetamide2020Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41513mGluR5CLONEDRATFunctional3-[(2-Methyl-4-thiazolyl)ethynyl]phenol654Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41514mGluR5CLONEDRATFunctional3-[(2-Methyl-4-thiazolyl)ethynyl]benzamide1000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41515mGluR5CLONEDRATFunctionalMPEP39Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41516mGluR5CLONEDRATFunctionalMTEP462Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41517mGluR5CLONEDRATFunctional5-Fluoro-2-[(2-methyl-4-thiazolyl)ethynyl]pyridine1093Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41518mGluR5CLONEDRATFunctional5-[(2-Methyl-4-thiazolyl)ethynyl]pyrimidine946Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41519mGluR5CLONEDRATFunctional2-[(2-Methyl-4-thiazolyl)ethynyl]pyrazine1830Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41520mGluR5CLONEDRATFunctional2-Methyl-4-(2-thienylethynyl)thiazole475Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41521mGluR5CLONEDRATFunctional2-Methyl-4-(3-thienylethynyl)thiazole337Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41522mGluR5CLONEDRATFunctional3-[(2-Methyl-4-thiazolyl)ethynyl]quinoline>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41523mGluR5CLONEDRATFunctional6-[(2-Methyl-4-thiazolyl)ethynyl]quinoxaline>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41524mGluR5CLONEDRATFunctional5-[(2-Methyl-4-thiazolyl)ethynyl]-1H-indole>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41525mGluR5CLONEDRATFunctional3-[(2,5-Dimethyl-4-thiazolyl)ethynyl]pyridine698Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41526mGluR5CLONEDRATFunctional3-[(5-Ethyl-2-methyl-4-thiazolyl)ethynyl]pyridine1243Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41527mGluR5CLONEDRATFunctional3-[(2-Methyl-5-phenyl-4-thiazolyl)ethynyl]pyridine>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41528mGluR5CLONEDRATFunctional4-(3-Pyridylethynyl)-2-thiazolylamine789Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41529mGluR5CLONEDRATFunctionalN-[4-(3-Pyridylethynyl)-2-thiazolyl]acetamide1920Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41530mGluR5CLONEDRATFunctionalN-[4-(3-Pyridylethynyl)-2-thiazolyl]benzamide>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41531mGluR5CLONEDRATFunctional1-(2,4-Difluorophenyl)-3-[4-(3-pyridylethynyl)-2-thiazolyl]urea>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41532mGluR5CLONEDRATFunctional[4-(3-Pyridylethynyl)-2-thiazolyl]carbamic Acid Methyl Ester>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41533mGluR5CLONEDRATFunctional4-(3-Fluorophenylethynyl)-2-thiazolylamine78.6Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41534mGluR5CLONEDRATFunctional2-Bromo-4-(3-fluorophenylethynyl)thiazole526Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41535mGluR5CLONEDRATFunctional2-(3,5-Difluorophenyl)-4-(3-fluorophenylethynyl)thiazole>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41536mGluR5CLONEDRATFunctional3-[4-(3-Fluorophenylethynyl)-2-thiazolyl]-2-propyn-1-ol >10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41537mGluR5CLONEDRATFunctional2-Ethynyl-4-(3-fluorophenylethynyl)thiazole2920Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41538mGluR5CLONEDRATFunctional3-Bromo-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine60Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41539mGluR5CLONEDRATFunctional3-(4-Fluorophenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine162Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41540mGluR5CLONEDRATFunctional3-(4-Methoxyphenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine225Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41541mGluR5CLONEDRATFunctional3-[5-[(2-Methyl-4-thiazolyl)ethynyl]-3-pyridyl]-2-propyn-1-ol68.6Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41542mGluR5CLONEDRATFunctional3-Ethynyl-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine19.2Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41543mGluR5CLONEDRATFunctional3-[(2-Methyl-4-thiazolyl)ethynyl]-5-vinylpyridine2.01Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41544mGluR5CLONEDRATFunctional2-Methoxy-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine426Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41545mGluR5CLONEDRATFunctional2-Fluoro-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine833Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41546mGluR5CLONEDRATFunctionalMethanesulfonic Acid 5-[(2-Methyl-4-thiazolyl)ethynyl]-2-pyridyl Ester2340Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41547mGluR5CLONEDRATFunctional2-Chloro-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41548mGluR5CLONEDRATFunctional2-(4-Fluorophenyl)-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine10.2Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41549mGluR5CLONEDRATFunctional3-Ethynyl-5-[(2-methyl-4-thiazolyl)ethynyl]pyridine2950Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41550mGluR5CLONEDRATFunctional5-[(2-Methyl-4-thiazolyl)ethynyl]-2-vinylpyridine>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41551mGluR5CLONEDRATFunctional2-Methoxy-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine228Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41552mGluR5CLONEDRATFunctionalMethanesulfonic Acid 3-[(2-Methyl-4-thiazolyl)ethynyl]-2-pyridyl Ester>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41553mGluR5CLONEDRATFunctional2-Chloro-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine45.5Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41554mGluR5CLONEDRATFunctional2-Ethynyl-3-[(2-methyl-4-thiazolyl)ethynyl]pyridine192Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41555mGluR5CLONEDRATFunctional(E)-3-[2-(2-Methyl-4-thiazolyl)vinyl]pyridine3090Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41556mGluR5CLONEDRATFunctional2-Methylthiazole-4-carboxylic Acid 3-Pyridylamide>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41557mGluR5CLONEDRATFunctional2-Methylthiazole-4-carboxylic Acid 3-Fluorophenylamide>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41558mGluR5CLONEDRATFunctional3-[(2-Methyl-4-oxazolyl)ethynyl]pyridine>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41559mGluR5CLONEDRATFunctional4-[(3-Fluorophenyl)ethynyl]-2-methyloxazole>10000Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41560mGluR5CLONEDRAT3H-MPEP3-[(2-Methyl-4-thiazolyl)ethynyl]benzonitrile0.37Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41561mGluR5CLONEDRAT3H-MPEP3-[(2-Methyl-4-thiazolyl)ethynyl]-5-vinylpyridine1.003Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41562mGluR5BRAINRAT3H-MPEP3-[(2-Methyl-4-thiazolyl)ethynyl]benzonitrile0.25Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41563mGluR5BRAINRAT3H-MPEP3-[(2-Methyl-4-thiazolyl)ethynyl]-5-vinylpyridine0.71Iso Y, et al., 2006Jan 15, 2025Jan 28, 2025
41580SLC6A3CLONEDRAT3H-DA UPTAKEWIN 35,42874Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41581SLC6A3CLONEDRAT3H-DA UPTAKE4-ARA-1271630Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41582SLC6A3CLONEDRAT3H-DA UPTAKECOCAINE555Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41583SLC6A3CLONEDRAT3H-DA UPTAKE8-Oxa-norcocaine9777Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41584SLC6A3CLONEDRAT3H-DA UPTAKEMAZINDOL31Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41585SLC6A3CLONEDRAT3H-DA UPTAKEMETHYLPHENIDATE152Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41586SLC6A3CLONEDRAT3H-DA UPTAKEBENZTROPINE160Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41587SLC6A3CLONEDRAT3H-DA UPTAKEGBR-1290915Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41588SLC6A3CLONEDRAT3H-DA UPTAKERIMCAZOLE643Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41589SLC6A3CLONEDRAT3H-WIN 35,428WIN 35,42820Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41590SLC6A3CLONEDRAT3H-WIN 35,4284-ARA-1273300Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41591SLC6A3CLONEDRAT3H-WIN 35,428COCAINE128Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41592SLC6A3CLONEDRAT3H-WIN 35,4288-Oxa-norcocaine1564Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41593SLC6A3CLONEDRAT3H-WIN 35,428MAZINDOL13Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41594SLC6A3CLONEDRAT3H-WIN 35,428METHYLPHENIDATE57Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41595SLC6A3CLONEDRAT3H-WIN 35,428BENZTROPINE127Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41596SLC6A3CLONEDRAT3H-WIN 35,428GBR-1290931Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41597SLC6A3CLONEDRAT3H-WIN 35,428RIMCAZOLE180Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41598SLC6A3CLONEDRAT3H-DA UPTAKE4-ChloroBZT83Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41599SLC6A3CLONEDRAT3H-DA UPTAKE3beta-4-ChloroBZT964Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41600SLC6A3CLONEDRAT3H-DA UPTAKE4,4'-DifluoroBZT22Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41601SLC6A3CLONEDRAT3H-DA UPTAKE4-TrifluoromethylBZT1282Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41602SLC6A3CLONEDRAT3H-DA UPTAKEN-CHO-4,4'-diFBZT>10000Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41603SLC6A3CLONEDRAT3H-WIN 35,4284-ChloroBZT45Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41604SLC6A3CLONEDRAT3H-WIN 35,4283beta-4-ChloroBZT680Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025