47615 ADK recombinant HUMAN Functional 4-N-Benzylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 30 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47616 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47617 ADK recombinant HUMAN Functional 4-N-(4-Methoxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 6 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47618 ADK recombinant HUMAN Functional 4-N-(4-Hydroxyphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47619 ADK recombinant HUMAN Functional 4-N-Cyclohexylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 250 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47620 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-beta-D-ribofuranosylpyrrolo[2,3-d]pyrimidine 0.8 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47621 ADK recombinant HUMAN Functional 4-N-(4-Fluorophenyl)amino-5-(4-fluorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 26 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47622 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.2 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47623 ADK recombinant HUMAN Functional 4-N-(4-Chlorophenyl)amino-5-(4-chlorophenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2.7 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47624 ADK recombinant HUMAN Functional 4-N-(4-Cyanophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 14 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47625 ADK recombinant HUMAN Functional 4-N-(4-Cyanophenyl)amino-5-(4-methoxyphenyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47626 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 3.6 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47627 ADK recombinant HUMAN Functional 4-N-(4-Methoxyphenyl)amino-5-(2-furanyl)-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 9 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47628 ADK recombinant HUMAN Functional 4-N-(3-Pyridyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 25 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47629 ADK recombinant HUMAN Functional 4-N-(4-Chlorophenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 2.3 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47630 ADK recombinant HUMAN Functional 4-N-(4-Methylphenyl)amino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47631 ADK recombinant HUMAN Functional 2-Methyl-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 47 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47632 ADK recombinant HUMAN Functional 6-Bromo-4-N-phenylamino-5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47633 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(5-azido-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 1.5 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47634 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(5-amino-5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 6.3 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47635 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(2-deoxy-beta-D-erythropentofuranosyl)pyrrolo[2,3-d]pyrimidine 300 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47636 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(2,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 100 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47637 ADK recombinant HUMAN Functional 4-N-Phenylamino-5-phenyl-7-(3,5-dideoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidine 44 Ugarkar BG, et al., 2000 Jan 15, 2025 Jan 15, 2025
47638 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 13 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47639 GABAA CLONED HUMAN 3H-RO-15-1788 NS-2710 2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47640 GABAA CLONED HUMAN 3H-RO-15-1788 7-trifluoromethyl-3-(2'-cyano-2,4'-difluorobiphenyl-5-yl) analogue 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47641 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1-hydroxy-1-methylethyl)-3-[4-fluoro-3-(pyridine-3-yl)phenyl derivative 0.85 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47642 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(7-Methyl-imidazo[1,2-b]pyridazin-3-yl)-biphenyl-2-carbonitrile 13 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47643 GABAA CLONED HUMAN 3H-RO-15-1788 7-Methyl-3-[3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]imidazo-[1,2-a]pyridine 0.4 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47644 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 1.5 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47645 GABAA CLONED HUMAN 3H-RO-15-1788 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.25 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47646 GABAA CLONED HUMAN 3H-RO-15-1788 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47647 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.73 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47648 GABAA CLONED HUMAN 3H-RO-15-1788 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.15 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47649 GABAA CLONED HUMAN 3H-RO-15-1788 DIAZEPAM 33 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47650 GABAA CLONED HUMAN 3H-RO-15-1788 NS-2710 14 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47651 GABAA CLONED HUMAN 3H-RO-15-1788 7-trifluoromethyl-3-(2'-cyano-2,4'-difluorobiphenyl-5-yl) analogue 0.73 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47652 GABAA CLONED HUMAN 3H-RO-15-1788 7-(1-hydroxy-1-methylethyl)-3-[4-fluoro-3-(pyridine-3-yl)phenyl derivative 4 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47653 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(7-Methyl-imidazo[1,2-b]pyridazin-3-yl)-biphenyl-2-carbonitrile 19 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47654 GABAA CLONED HUMAN 3H-RO-15-1788 7-Methyl-3-[3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]imidazo-[1,2-a]pyridine 0.4 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47655 GABAA CLONED HUMAN 3H-RO-15-1788 3'-(3-Methyl-imidazo[1,2-b][1,2,4]triazin-7-yl)biphenyl-2-carbonitrile 1.2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47656 GABAA CLONED HUMAN 3H-RO-15-1788 2',4-Difluoro-5'-[3-(trifluoromethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 0.8 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47657 GABAA CLONED HUMAN 3H-RO-15-1788 4,2'-Difluoro-5'-[3-(1-hydroxy-1-methyl-ethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]-biphenyl-2-carbonitrile 2.1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47658 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 1.8 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47659 GABAA CLONED HUMAN 3H-RO-15-1788 2',4,6-Trifluoro-5'-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47660 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 2 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47661 GABAA CLONED HUMAN 3H-RO-15-1788 6,2’-Difluoro-5’-[3-(1-hydroxy-1-methylethyl)imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile 1.1 Russell MG, et al., 2006 Jan 15, 2025 Jan 27, 2025
47662 OT CLONED HUMAN 3H-Oxytocin (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 28 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47663 OT CLONED HEK293 3H-Oxytocin (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 17 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47664 V1A CLONED HUMAN 3H-AVP (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 170 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47665 V1B CLONED HUMAN 3H-AVP (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide >10000 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47666 V2 CLONED HUMAN 3H-AVP (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide >10000 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47667 OT CLONED RAT 3H-Oxytocin (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino)-1-[(2'-methyl[1,1'-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide 135 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47668 OT CLONED HUMAN 3H-Oxytocin Atosiban 81 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47669 OT CLONED HEK293 3H-Oxytocin Atosiban 27 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47670 V1A CLONED HUMAN 3H-AVP Atosiban 3.5 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47671 V1B CLONED HUMAN 3H-AVP Atosiban 657 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47672 V2 CLONED HUMAN 3H-AVP Atosiban 954 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47673 OT CLONED RAT 3H-Oxytocin Atosiban 76 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47674 OT CLONED HUMAN 3H-Oxytocin Oxytocin 0.5 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47675 OT CLONED HEK293 3H-Oxytocin Oxytocin 0.71 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47676 V1A CLONED HUMAN 3H-AVP Oxytocin 123 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47677 V1B CLONED HUMAN 3H-AVP Oxytocin 1782 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47678 V2 CLONED HUMAN 3H-AVP Oxytocin 1544 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47679 OT CLONED RAT 3H-Oxytocin Oxytocin 1.9 Cirillo R, et al., 2003 Jan 15, 2025 Jan 15, 2025
47680 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE PAROXETINE 0.019 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47681 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE SERTRALINE 0.047 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47682 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Indatraline 0.13 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47683 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE CLOMIPRAMINE 0.14 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47684 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE CITALOPRAM 0.65 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47685 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE FLUOXETINE 1.96 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47686 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Desmethylsertraline 2.29 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47687 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE NORFLUOXETINE 3.15 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47688 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE IMIPRAMINE 14.2 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47689 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE AMITRIPTYLINE 17.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47690 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Dothiepin 31.3 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47691 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Zimeldine 67.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47692 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE NORTRYPTYLINE 60.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47693 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE DOXEPIN 126 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47694 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE northiaden 130 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47695 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE DESIPRAMINE 152 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47696 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE AMOXAPINE 290 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47697 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Fenfluramine (+) 855 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47698 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Fenfluramine (-) 2784 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47699 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE sibutramine 2135 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47700 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake PAROXETINE 0.48 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47701 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake SERTRALINE 2.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47702 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Indatraline 1.5 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47703 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake CLOMIPRAMINE 5.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47704 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake CITALOPRAM 3.51 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47705 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake FLUOXETINE 10.9 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47706 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Desmethylsertraline 53.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47707 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake NORFLUOXETINE 13.9 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47708 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Fluvoxamine 3.57 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47709 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake AMITRIPTYLINE 48.6 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47710 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake BTS 54 505 26.2 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47711 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake BTS 54 354 18.2 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47712 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Dothiepin 77.8 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47713 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Zimeldine 56.7 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47714 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake NORTRYPTYLINE 197 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47715 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake DOXEPIN 201 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47716 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake northiaden 192 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47717 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake DESIPRAMINE 200 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47718 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake AMOXAPINE 409 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47719 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Fenfluramine (+) 279 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47720 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake Fenfluramine (-) 809 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47721 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake sibutramine 3131 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47722 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE Fluvoxamine 4.17 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47723 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE BTS 54 505 18 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47724 SLC6A4 FR. CORTEX RAT 3H-PAROXETINE BTS 54 354 19.3 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47725 SLC6A4 FR. CORTEX RAT 3H-5-HT Uptake IMIPRAMINE 30.9 Cheetham SC, et.al., 1993 Jan 15, 2025 Jan 15, 2025
47726 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY, porcine 0.043 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47727 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY, porcine 0.048 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47728 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY, zebrafish 0.066 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47729 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY, zebrafish 0.11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47730 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.035 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47731 Y1 CLONED GUINEA PIG [125I] - Peptide YY PYY,[leu31,Pro34], human 0.035 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47732 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY2-36, porcine 0.26 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47733 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY 3-36, porcine 2 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47734 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY18-36 260 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47735 Y1 CLONED GUINEA PIG [125I] - Peptide YY PP, guinea pig 3.2 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47736 Y1 CLONED GUINEA PIG [125I] - Peptide YY SR 120819A 0.8 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47737 Y1 CLONED GUINEA PIG [125I] - Peptide YY BIBP3226 4.9 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47738 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY 28-36, [P30, Y32, L34] 2.4 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47739 Y1 CLONED GUINEA PIG [125I] - Peptide YY NPY D-Trp32, porcine 1000 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47740 Y1 CLONED RAT [125I] - Peptide YY NPY, porcine 0.06 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47741 Y1 CLONED RAT [125I] - Peptide YY PYY, porcine 0.13 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47742 Y1 CLONED RAT [125I] - Peptide YY NPY, zebrafish 0.1 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47743 Y1 CLONED RAT [125I] - Peptide YY PYY, zebrafish 0.18 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47744 Y1 CLONED RAT [125I] - Peptide YY NPY,[leu31,Pro34], porcine 0.061 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47745 Y1 CLONED RAT [125I] - Peptide YY PYY,[leu31,Pro34], human 0.11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47746 Y1 CLONED RAT [125I] - Peptide YY NPY2-36, porcine 0.38 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47747 Y1 CLONED RAT [125I] - Peptide YY NPY 3-36, porcine 4.1 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47748 Y1 CLONED RAT [125I] - Peptide YY NPY18-36 100 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47749 Y1 CLONED RAT [125I] - Peptide YY PP, guinea pig 11 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47750 Y1 CLONED RAT [125I] - Peptide YY SR 120819A 1.3 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47751 Y1 CLONED RAT [125I] - Peptide YY BIBP3226 3.2 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47752 Y1 CLONED RAT [125I] - Peptide YY NPY 28-36, [P30, Y32, L34] 1.4 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47753 Y1 CLONED RAT [125I] - Peptide YY NPY D-Trp32, porcine 1000 Berglund MM, et al., 1999 Jan 15, 2025 Jan 15, 2025
47754 CEREBRAL CORTEX RAT Functional Val-D-Pro-NHBu >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47755 CEREBRAL CORTEX RAT Functional L-Valyl-L-Proline hexylamide hydrogen oxalate 900 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47756 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline benzylamide hydrogen oxalate 3300 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47757 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline cyclohexylmethylamide hydrogen oxalate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47758 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline-N- β-naphthylamide trifluroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47759 CEREBRAL CORTEX RAT Functional L-Valyl-L-proline piperidinylamide hydrogen oxalate hemihydrate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47760 CEREBRAL CORTEX RAT Functional L-Valyl-L-prolinamide trifluoroacetate 6000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47761 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-prolinamide trifluoroacetate hemihydrate 570 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47762 CEREBRAL CORTEX RAT Functional L-Norvalyl-L-prolinamide trifluoroacetate hemihydrate 1600 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47763 CEREBRAL CORTEX RAT Functional L-Norleucyl-L-prolinamide hydrogen oxalate hemihydrate 2000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47764 CEREBRAL CORTEX RAT Functional L-Leucyl-L-prolinamide trifluoroacetate 2100 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47765 CEREBRAL CORTEX RAT Functional L-Isoleucyl-L-prolinamide trifluoroacetate 4300 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47766 CEREBRAL CORTEX RAT Functional L-Phenylalanyl-L-prolinamide trifluoroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47767 CEREBRAL CORTEX RAT Functional α-Methylalanyl-L-proline butylamide hydrochloride hemihydrate 5000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47768 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline n-propylamide trifluoroacetate 80 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47769 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline n-butylamide hydrogen oxalate 80 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47770 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline n-pentylamide hydrogen oxalate 270 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47771 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline isobutylamide trifluoroacetate 320 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47772 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline (R)-sec-butylamide hydrogen oxalate 4500 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47773 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline-(2S)-methylbutylamide hydrogen oxalate hemihydrate 500 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47774 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-proline 3-methylthiopropylamide hydrogen oxalate hemihydrate 300 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47775 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-azetidine carboxamide trifluoroacetate hydrate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47776 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(R)-pipecolinic acid amide trifluoroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47777 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-L-pipecolinic acid n-butylamide trifluoroacetate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47778 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(S)-nipecotamide hydrogen oxalate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47779 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-4-thia-L-prolinamide trifluoroacetate hemihydrate >10000 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47780 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(4S)-fluoro-L-proline n-Butylamide Trifluoroacetate 320 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47781 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-4-cis-benzyl-L-proline n-butylamide Hydrogen Oxalate 140 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47782 CEREBRAL CORTEX RAT Functional butabindide 7 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47783 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-indoline carboxylic acid methylamide hydrogen oxalate hydrate 340 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47784 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-indoline carboxylic acid ethylamide hydrogen oxalate hydrate 12 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47785 CEREBRAL CORTEX RAT Functional (2S)-Aminobutyryl-(2S)-indoline carboxylic acid propylamide hydrogen oxalate hydrate 6 Ganellin CR, et al., 2005 Jan 15, 2025 Jan 15, 2025
47786 MOR CLONED HUMAN 3H-DAMGO Enadoline 22 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47787 MOR CLONED HUMAN 3H-DAMGO Cyclorphan 0.062 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47788 MOR CLONED HUMAN 3H-DAMGO MCL-101 0.23 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47789 MOR CLONED HUMAN 3H-DAMGO Levorphanol 0.21 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47790 MOR CLONED HUMAN 3H-DAMGO MCL-133 48 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47791 MOR CLONED HUMAN 3H-DAMGO MCL-134 52 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47792 MOR CLONED HUMAN 3H-DAMGO MCL-153 29 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47793 MOR CLONED HUMAN 3H-DAMGO MCL-154 66 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47794 MOR CLONED HUMAN 3H-DAMGO MCL-135 0.14 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47795 MOR CLONED HUMAN 3H-DAMGO MCL-136 0.93 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47796 MOR CLONED HUMAN 3H-DAMGO MCL-176 0.23 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47797 MOR CLONED HUMAN 3H-DAMGO MCL-139 0.16 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47798 MOR CLONED HUMAN 3H-DAMGO MCL-140 3.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47799 MOR CLONED HUMAN 3H-DAMGO MCL-177 0.89 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47800 MOR CLONED HUMAN 3H-DAMGO MCL-179 0.97 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47801 MOR CLONED HUMAN 3H-DAMGO MCL-144 0.09 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47802 MOR CLONED HUMAN 3H-DAMGO MCL-178 1.8 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47803 MOR CLONED HUMAN 3H-DAMGO MCL-145 0.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47804 MOR CLONED HUMAN 3H-DAMGO MCL-141 4.7 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47805 MOR CLONED HUMAN 3H-DAMGO MCL-142 3.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47806 MOR CLONED HUMAN 3H-DAMGO MCL-143 0.28 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47807 DOR CLONED HUMAN 3H-Naltrindole Enadoline 1000 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47808 DOR CLONED HUMAN 3H-Naltrindole Cyclorphan 1.9 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47809 DOR CLONED HUMAN 3H-Naltrindole MCL-101 5.9 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47810 DOR CLONED HUMAN 3H-Naltrindole Levorphanol 4.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47811 DOR CLONED HUMAN 3H-Naltrindole MCL-133 600 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47812 DOR CLONED HUMAN 3H-Naltrindole MCL-134 370 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47813 DOR CLONED HUMAN 3H-Naltrindole MCL-153 730 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47814 DOR CLONED HUMAN 3H-Naltrindole MCL-154 2500 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47815 DOR CLONED HUMAN 3H-Naltrindole MCL-135 3.8 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47816 DOR CLONED HUMAN 3H-Naltrindole MCL-136 32 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47817 DOR CLONED HUMAN 3H-Naltrindole MCL-176 44 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47818 DOR CLONED HUMAN 3H-Naltrindole MCL-139 9.4 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47819 DOR CLONED HUMAN 3H-Naltrindole MCL-140 80 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47820 DOR CLONED HUMAN 3H-Naltrindole MCL-177 24 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47821 DOR CLONED HUMAN 3H-Naltrindole MCL-179 21 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47822 DOR CLONED HUMAN 3H-Naltrindole MCL-144 4.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47823 DOR CLONED HUMAN 3H-Naltrindole MCL-178 82 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47824 DOR CLONED HUMAN 3H-Naltrindole MCL-145 9.4 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47825 DOR CLONED HUMAN 3H-Naltrindole MCL-141 400 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47826 DOR CLONED HUMAN 3H-Naltrindole MCL-142 920 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47827 DOR CLONED HUMAN 3H-Naltrindole MCL-143 16 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47828 KOR CLONED HUMAN 3H-U69,593 Enadoline 0.27 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47829 KOR CLONED HUMAN 3H-U69,593 Cyclorphan 0.034 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47830 KOR CLONED HUMAN 3H-U69,593 MCL-101 0.079 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47831 KOR CLONED HUMAN 3H-U69,593 Levorphanol 2.3 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47832 KOR CLONED HUMAN 3H-U69,593 MCL-133 24 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47833 KOR CLONED HUMAN 3H-U69,593 MCL-134 50 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47834 KOR CLONED HUMAN 3H-U69,593 MCL-153 18 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47835 KOR CLONED HUMAN 3H-U69,593 MCL-154 120 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47836 KOR CLONED HUMAN 3H-U69,593 MCL-135 0.1 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47837 KOR CLONED HUMAN 3H-U69,593 MCL-136 0.41 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47838 KOR CLONED HUMAN 3H-U69,593 MCL-176 0.07 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47839 KOR CLONED HUMAN 3H-U69,593 MCL-139 0.076 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47840 KOR CLONED HUMAN 3H-U69,593 MCL-140 1.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47841 KOR CLONED HUMAN 3H-U69,593 MCL-177 0.65 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47842 KOR CLONED HUMAN 3H-U69,593 MCL-179 0.59 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47843 KOR CLONED HUMAN 3H-U69,593 MCL-144 0.049 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47844 KOR CLONED HUMAN 3H-U69,593 MCL-178 1.1 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47845 KOR CLONED HUMAN 3H-U69,593 MCL-145 0.078 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47846 KOR CLONED HUMAN 3H-U69,593 MCL-141 4.2 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47847 KOR CLONED HUMAN 3H-U69,593 MCL-142 3.4 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47848 KOR CLONED HUMAN 3H-U69,593 MCL-143 0.17 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47849 BRAIN RAT 3H-MK912 MCL-202 3000 Neumeyer JL, et al., 2003 Jan 15, 2025 Jan 15, 2025
47850 CLONED HUMAN 1251-CGRP h-alpha-CGRP 8-37 1.3 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47851 CLONED HUMAN 1251-CGRP h-alpha-CGRP 0.18 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47852 CLONED HUMAN 1251-CGRP [D31,p34,F35]-h-alpha-CGRP 27-37 14 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47853 CLONED HUMAN 1251-CGRP [D31,Tic34,F35]-h-alpha-CGRP 27-37 70.5 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47854 CLONED HUMAN 1251-CGRP [D31,A34,F35]-h-alpha-CGRP 27-37 76.8 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47855 CLONED HUMAN 3H-CGRP 8-37 [propionyl-K24]-h-alpha-CGRP 8-37 0.6 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47856 CLONED HUMAN 3H-CGRP 8-37 h-alpha-CGRP 8-37 0.06 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47857 CLONED HUMAN 3H-CGRP 8-37 h-alpha-CGRP 0.29 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47858 CLONED HUMAN 3H-CGRP 8-37 [D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47859 CLONED HUMAN 3H-CGRP 8-37 [D31,Tic34,F35]-h-alpha-CGRP 27-37 1.8 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47860 CLONED HUMAN 3H-CGRP 8-37 [D31,A34,F35]-h-alpha-CGRP 27-37 13.6 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47861 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 h-alpha-CGRP 0.29 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47862 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 h-alpha-CGRP (reduced) 10.2 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47863 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47864 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47865 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47866 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47867 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 34,F35]-h-alpha-CGRP 8-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47868 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 (1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47869 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1S,2S,3S)-beta-aminocyclopropane carboxylic acid, F35]-h-alpha-CGRP 8-37 31 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47870 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [D31,(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 34, F35]-h-alpha-CGRP 8-37 65.3 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47871 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Hop29,D31,p34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47872 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Tic29,D31,p34,F35]-h-alpha-CGRP 27-37 0.02 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47873 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Hyp29,D31,p34,F35]-h-alpha-CGRP 27-37 0.006 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47874 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [Aib29,D31,p34,F35]-h-alpha-CGRP 27-37 0.002 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47875 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [A29,D31,p34,F35]-h-alpha-CGRP 27-37 8.4 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47876 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1S,2S,3S)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 >10000 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47877 CLONED HUMAN 3H-propionyl-K24-CGRP 8-37 [(1R,2R,3R)-beta-aminocyclopropane carboxylic acid 29,D31,p34,F35]-h-alpha-CGRP 27-37 0.7 Lang M, et al., 2006 Jan 15, 2025 Jan 15, 2025
47878 PDE5 AORTA RAT Functional sildenafil 7.94328 Teixeira CE, et al., 2006 Jan 15, 2025 Jan 15, 2025
47879 PDE5 AORTA RAT Functional vardenafil 2.95121 Teixeira CE, et al., 2006 Jan 15, 2025 Jan 15, 2025
47880 PDE5 AORTA RAT Functional tadalafil 9.77237 Teixeira CE, et al., 2006 Jan 15, 2025 Jan 15, 2025
47881 SST1 CLONED HUMAN 3H-thymidine BIM-23926 3.6 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47882 SST2 CLONED HUMAN 3H-thymidine BIM-23926 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47883 SST3 CLONED HUMAN 3H-thymidine BIM-23926 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47884 SST4 CLONED HUMAN 3H-thymidine BIM-23926 833 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47885 SST5 CLONED HUMAN 3H-thymidine BIM-23926 788 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47886 SST1 CLONED HUMAN 3H-thymidine BIM-23745 42 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47887 SST2 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47888 SST3 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47889 SST4 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47890 SST5 CLONED HUMAN 3H-thymidine BIM-23745 1000 Zatelli MC, et.al., 2002 Jan 15, 2025 Jan 15, 2025
47891 P2X1 CLONED Xenopus Functional NF279 19 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025
47892 P2X2 CLONED Xenopus Functional NF279 770 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025
47893 P2X3 CLONED Xenopus Functional NF279 1620 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025
47894 P2X4 CLONED Xenopus Functional NF279 >10000 Rettinger J, et.al., 2000 Jan 15, 2025 Jan 15, 2025
47895 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 2.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47896 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 10 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47897 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 13 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47898 GABAA CLONED HUMAN 3H-RO-15-1788 DMCM 7.5 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47899 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47900 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 66 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47901 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 56 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47902 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 21 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47903 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47904 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 12 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47905 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 16 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47906 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 16 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47907 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 4.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47908 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 22 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47909 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 28 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47910 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-propylthio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 41 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47911 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 18 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47912 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 57 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47913 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 184 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47914 GABAA CLONED HUMAN 3H-RO-15-1788 3-Butylthio-6,6-dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 182 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47915 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47916 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47917 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 12 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47918 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1-methylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47919 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 170 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47920 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47921 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47922 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(1,1-dimethylethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47923 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2.9 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47924 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 31 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47925 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 21 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47926 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 24 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47927 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 4.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47928 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 60 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47929 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 46 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47930 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 50 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47931 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 1.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47932 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 4.3 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47933 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 19 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47934 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 48 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47935 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 2.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47936 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 10 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47937 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 7.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47938 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-3-(thien-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 18 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47939 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 67 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47940 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47941 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47942 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47943 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 15 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47944 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 119 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47945 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 182 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47946 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropoxy-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 69 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47947 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 132 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47948 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47949 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47950 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47951 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 3.9 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47952 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 72 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47953 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 44 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47954 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-isopropylamino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 87 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47955 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 78 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47956 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47957 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47958 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)amino-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47959 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 11 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47960 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 211 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47961 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 162 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47962 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-ethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 240 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47963 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47964 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47965 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47966 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(pyrazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47967 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 1.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47968 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 45 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47969 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 26 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47970 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 25 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47971 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5.8 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47972 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 165 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47973 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 31 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47974 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 33 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47975 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 9.1 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47976 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 172 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47977 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 43 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47978 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyridin-4-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 35 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47979 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 15 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47980 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 175 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47981 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 161 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47982 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 159 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47983 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47984 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47985 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47986 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-phenyl-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47987 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 85 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47988 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47989 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47990 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(pyrrol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47991 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 0.5 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47992 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 3.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47993 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 5.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47994 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(pyridin-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 10 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47995 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 37 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47996 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47997 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 300 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47998 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(3-methyl-1,2,4-oxadiazol-5-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 185 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
47999 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 2.2 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48000 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 61 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48001 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 44 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48002 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 47 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48003 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 19 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48004 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 267 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48005 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 49 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48006 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-methylthio-1-(1-methyl-1,2,4-triazol-3-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 102 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48007 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 1.6 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48008 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 20 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48009 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 16 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48010 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(2-hydroxyethyl)thio-1-(thiazol-2-yl)6,7-dihydro-2-benzothiophen-4(5H)-one- 20 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48011 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 4.7 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48012 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 79 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48013 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 48 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48014 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-3-(3-hydroxypropyl)thio-1-(thiazol-2-yl)-6,7-dihydro-2-benzothiophen-4(5H)-one 48 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48015 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 1.4 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48016 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 24 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48017 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 39 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48018 GABAA CLONED HUMAN 3H-RO-15-1788 6,6-Dimethyl-1-(thiazol-2-yl)-3-(thiazol-2-yl)thio-6,7-dihydro-2-benzothiophen-4(5H)-one 28 Chambers, MS et al., 2003 Jan 15, 2025 Jan 27, 2025
48019 AORTA RAT 3H-PRAZOSIN N-(1-Benzylpiperidin-4-yl)-1-isopropylindazole-3-carboxamide Hydrochloride >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
48020 AORTA RAT 3H-PRAZOSIN N-(1-(2-((N-Methylsulfonyl)amino)ethyl)piperidin-4-yl)-1-isopropylindazole-3-carboxamide Maleate >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
48021 AORTA RAT 3H-PRAZOSIN CISAPRIDE 199.526 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
48022 AORTA RAT 3H-PRAZOSIN N-(2-(4-((Benzyloxycarbonyl)amino)-1-piperidinyl)-ethyl)-1-isopropylindazole-3-carboxamide Oxalate >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
48023 AORTA RAT 3H-PRAZOSIN N-(2-(4-(1-Adamantylcarboxamido)-1-piperidinyl)ethyl)-1-isopropylindazole-3-carboxamide Oxalate >10000 SCHAUS JM, ET AL., 1997 Jan 15, 2025 Jan 15, 2025
48024 AMPA CORTEX RAT 3H-AMPA AMPA 40 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48025 AMPA CORTEX RAT 3H-AMPA Br-HIBO,(RS) 650 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48026 AMPA CORTEX RAT 3H-AMPA C1-HIBO 220 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48027 KA CORTEX RAT 3H-Kainic acid C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48028 KA CORTEX RAT 3H-Kainic acid Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48029 KA CORTEX RAT 3H-Kainic acid AMPA >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48030 NMDA CORTEX RAT 3H-CGP39653 AMPA >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 27, 2025
48031 NMDA CORTEX RAT 3H-CGP39653 Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 27, 2025
48032 NMDA CORTEX RAT 3H-CGP39653 C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 27, 2025
48033 GRIA1 CLONED RAT 3H-AMPA AMPA 22 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48034 GRIA1 CLONED RAT 3H-AMPA Br-HIBO,(RS) 170 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48035 GRIA2 CLONED RAT 3H-AMPA AMPA 17 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48036 GRIA1 CLONED RAT 3H-AMPA C1-HIBO 130 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48037 GRIA2 CLONED RAT 3H-AMPA Br-HIBO,(RS) 250 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48038 GRIA2 CLONED RAT 3H-AMPA C1-HIBO 370 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48039 AMPA CLONED RAT 3H-AMPA AMPA 21 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48040 AMPA CLONED RAT 3H-AMPA Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48041 AMPA CLONED RAT 3H-AMPA C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48042 GRIA4 CLONED RAT 3H-AMPA C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48043 GRIA4 CLONED RAT 3H-AMPA Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48044 GRIA4 CLONED RAT 3H-AMPA AMPA 40 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48045 CLONED RAT 3H-AMPA AMPA 740 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48046 CLONED RAT 3H-AMPA Br-HIBO,(RS) 4800 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48047 CLONED RAT 3H-AMPA C1-HIBO 6800 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48048 CLONED RAT 3H-AMPA C1-HIBO >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48049 CLONED RAT 3H-AMPA Br-HIBO,(RS) >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48050 CLONED RAT 3H-AMPA AMPA >10000 Bjerrum, EJ et al 2003 Jan 15, 2025 Jan 15, 2025
48051 CLONED HUMAN 3H-25-OHC paxilline 660 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025
48052 CLONED HUMAN 3H-25-OHC paxilline 1100 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025
48053 CLONED HUMAN 3H-25-OHC [22(R)-hydroxycholesterol 250 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025
48054 CLONED HUMAN 3H-25-OHC [22(R)-hydroxycholesterol 490 Bramlett KS, et al., 2003 Jan 15, 2025 Jan 15, 2025
48055 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 1 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48056 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 7 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48057 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 7 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48058 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48059 SST1 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48060 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.05 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48061 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48062 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.8 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48063 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.3 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48064 SST2 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.09 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48065 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.1 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48066 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48067 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.9 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48068 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.7 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48069 SST3 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.3 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48070 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48071 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48072 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48073 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48074 SST4 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48075 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 Somatostatin-14 0.2 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48076 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 17 0.4 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48077 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 15 0.6 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48078 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 hCS 13 0.5 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48079 SST5 CLONED HUMAN 125I-Tyr11-somatostatin-14 CST14 0.3 Fukusumi S, et al., 1997 Jan 15, 2025 Jan 15, 2025
48080 CLONED RAT Functional (S)-Glu >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48081 mGluR2 CLONED RAT Functional (S)-Glu 4400 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48082 mGluR4 CLONED RAT Functional (S)-Glu >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48083 mGluR5 CLONED RAT Functional (S)-Glu 7400 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48084 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48085 mGluR2 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48086 mGluR4 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48087 mGluR5 CLONED RAT Functional (S)-2-Aminoadipic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48088 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48089 mGluR2 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48090 mGluR4 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48091 mGluR5 CLONED RAT Functional Ibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48092 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48093 mGluR2 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48094 mGluR4 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48095 mGluR5 CLONED RAT Functional (S)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48096 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48097 mGluR2 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48098 mGluR4 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48099 mGluR5 CLONED RAT Functional (R)-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48100 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48101 mGluR2 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48102 mGluR4 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48103 mGluR5 CLONED RAT Functional (S)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48104 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48105 mGluR2 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48106 mGluR4 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48107 mGluR5 CLONED RAT Functional (R)-4-Methylhomoibotenic acid >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48108 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48109 mGluR2 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48110 mGluR4 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48111 mGluR5 CLONED RAT Functional Br-HIBO,(S) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48112 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48113 mGluR2 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48114 mGluR4 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48115 mGluR5 CLONED RAT Functional Br-HIBO,(R) >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48116 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48117 mGluR2 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48118 mGluR4 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48119 mGluR5 CLONED RAT Functional (S)-(+)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48120 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48121 mGluR2 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48122 mGluR4 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48123 mGluR5 CLONED RAT Functional (R)-Bu-HIBO >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48124 CLONED RAT Functional (S)-4-Carboxyphenylglycine >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 15, 2025
48125 mGluR5 CLONED RAT Functional (S)-4-Carboxyphenylglycine >10000 Brauner-Osborne H, et.al., 1998 Jan 15, 2025 Jan 28, 2025
48126 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.23 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48127 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 700 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48128 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48129 Y1 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 530 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48130 Y1 CLONED HUMAN 3H-Propionyl-NPY PP, human 170 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48131 Y1 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 760 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48132 Y1 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48133 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 29 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48134 Y2 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 0.03 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48135 Y2 CLONED HUMAN 3H-Propionyl-NPY PP, human 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48136 Y2 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48137 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48138 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 500 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48139 Y2 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.04 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48140 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY, human 5.8 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48141 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48142 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 170 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48143 Y4 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 51 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48144 Y4 CLONED HUMAN 3H-Propionyl-NPY PP, human 0.06 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48145 Y4 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 15 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48146 Y4 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 1000 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48147 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY D-Trp32, human, rat 35 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48148 Y5 CLONED HUMAN 3H-Propionyl-NPY PYY 3-36 17 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48149 Y5 CLONED HUMAN 3H-Propionyl-NPY PP, human 1.4 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48150 Y5 CLONED HUMAN 3H-Propionyl-NPY PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], human 0.24 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48151 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY [hPP(1-17), Ala31,Aib32], human 0.92 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48152 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY [Ala31, Aib32], porcine 6 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48153 Y5 CLONED HUMAN 3H-Propionyl-NPY NPY, human 0.6 Cabrele C, et al., 2000 Jan 15, 2025 Jan 15, 2025
48154 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(Pyrrol-1-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 61.5 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025
48155 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(Thien-2-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 10.3 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025
48156 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(Thien-3-yl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 36.3 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025
48157 GABAA BRAIN BOVINE 3H-RO-15-1788 3-(N-Formylcarbamoyl)-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxide 844.2 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025
48158 GABAA BRAIN BOVINE 3H-RO-15-1788 DIAZEPAM 10 Costanzo A, et al., 1999 Jan 15, 2025 Jan 15, 2025
48159 A1 BRAIN RAT 3H-cyclohexyladenosine BS-DMPX 1200 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48160 A1 BRAIN RAT 3H-cyclohexyladenosine MS-DMPX 1280 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48161 A1 BRAIN RAT 3H-cyclohexyladenosine 3-(2-Hydroxyethyl)-8-(m-methoxystyryl)-7-methyl-1-propargylxanthine 1040 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48162 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(m-Bromostyryl)-3-(2-hydroxyethyl)-7-methyl-1-propargylxanthine 1280 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48163 A1 CLONED HUMAN 3H-CCPA MSX-2 2500 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48164 A1 BRAIN RAT 3H-cyclohexyladenosine MSX-2 900 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48165 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(m-Bromostyryl)-3-(3-hydroxypropyl)-7-methyl-1-propargylxanthine 625 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48166 A1 BRAIN RAT 3H-cyclohexyladenosine 8-(m-Aminostyryl)-3,7-dimethyl-1-propargylxanthine 1070 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48167 A1 BRAIN RAT 3H-cyclohexyladenosine 3,7-Dimethyl-8-(m-hydroxystyryl)-1-propargylxanthine 940 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48168 A2A BRAIN RAT 3H-CGS-21680 BS-DMPX 8.2 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48169 A2A BRAIN RAT 3H-CGS-21680 MS-DMPX 12 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48170 A2A BRAIN RAT 3H-CGS-21680 3-(2-Hydroxyethyl)-8-(m-methoxystyryl)-7-methyl-1-propargylxanthine 39 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48171 A2A BRAIN RAT 3H-CGS-21680 8-(m-Bromostyryl)-3-(2-hydroxyethyl)-7-methyl-1-propargylxanthine 25 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48172 A2A CLONED HUMAN 3H-CGS-21680 MSX-2 5 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48173 A2A BRAIN HUMAN 3H-CGS-21680 MSX-2 15 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48174 A2A BRAIN RAT 3H-CGS-21680 MSX-2 8 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48175 A2A BRAIN RAT 3H-CGS-21680 8-(m-Bromostyryl)-3-(3-hydroxypropyl)-7-methyl-1-propargylxanthine 13 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48176 A2A BRAIN RAT 3H-CGS-21680 8-(m-Aminostyryl)-3,7-dimethyl-1-propargylxanthine 42 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48177 A2A BRAIN RAT 3H-CGS-21680 3,7-Dimethyl-8-(m-hydroxystyryl)-1-propargylxanthine 21 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48178 A3 CLONED HUMAN 3H-NECA BS-DMPX >10000 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48179 A3 CLONED HUMAN 3H-NECA MSX-2 >10000 Sauer, R et. al. 2000 Jan 15, 2025 Jan 15, 2025
48180 Y4 CLONED GUINEA PIG 125I-hPP PP, guinea pig 0.046 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48181 Y4 CLONED GUINEA PIG 125I-hPP PP, human 0.031 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48182 Y4 CLONED GUINEA PIG 125I-hPP PP, rat 0.044 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48183 Y4 CLONED GUINEA PIG 125I-hPP PP, BOVINE 0.013 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48184 Y4 CLONED HUMAN 125I-hPP PP, guinea pig 0.06 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48185 Y4 CLONED HUMAN 125I-hPP PP, human 0.039 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48186 Y4 CLONED HUMAN 125I-hPP PP, rat 0.071 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48187 Y4 CLONED HUMAN 125I-hPP PP, BOVINE 0.031 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48188 Y4 CLONED RAT 125I-hPP PP, guinea pig 0.007 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48189 Y4 CLONED RAT 125I-hPP PP, human 0.003 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48190 Y4 CLONED RAT 125I-hPP PP, rat 0.0027 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48191 Y4 CLONED RAT 125I-hPP PP, BOVINE 0.006 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48192 Y4 CLONED GUINEA PIG 125I-hPP NPY, porcine 25 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48193 Y4 CLONED GUINEA PIG 125I-hPP PYY, porcine 26 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48194 Y4 CLONED GUINEA PIG 125I-hPP NPY,[leu31,Pro34], porcine 20 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48195 Y4 CLONED GUINEA PIG 125I-hPP PYY,[leu31,Pro34], human 16 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48196 Y4 CLONED GUINEA PIG 125I-hPP NPY2-36, porcine 130 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48197 Y4 CLONED GUINEA PIG 125I-hPP NPY13-36, porcine 29 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48198 Y4 CLONED GUINEA PIG 125I-hPP NPY D-Trp32, porcine 1000 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48199 Y4 CLONED HUMAN 125I-hPP NPY, porcine 6 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48200 Y4 CLONED HUMAN 125I-hPP PYY, porcine 4 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48201 Y4 CLONED HUMAN 125I-hPP NPY,[leu31,Pro34], porcine 6.6 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48202 Y4 CLONED HUMAN 125I-hPP PYY,[leu31,Pro34], human 11 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48203 Y4 CLONED HUMAN 125I-hPP NPY2-36, porcine 17 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48204 Y4 CLONED HUMAN 125I-hPP NPY13-36, porcine 9 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48205 Y4 CLONED HUMAN 125I-hPP NPY D-Trp32, porcine 1000 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48206 Y4 CLONED RAT 125I-hPP NPY, porcine 18 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48207 Y4 CLONED RAT 125I-hPP PYY, porcine 11 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48208 Y4 CLONED RAT 125I-hPP PYY,[leu31,Pro34], human 0.62 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48209 Y4 CLONED RAT 125I-hPP NPY2-36, porcine 29 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48210 Y4 CLONED RAT 125I-hPP NPY13-36, porcine 2.2 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48211 Y4 CLONED RAT 125I-hPP NPY D-Trp32, porcine 60 Eriksson H, et al., 1998 Jan 15, 2025 Jan 15, 2025
48212 nAChR BRAIN RAT 3H-NICOTINE Nicotine 1.26 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48213 nAChR BRAIN RAT 3H-NICOTINE 6-Bromonicotine 0.45 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48214 nAChR BRAIN RAT 3H-NICOTINE 6-Fluoro-3-( l-methyl-2-pyrrohdinyl )pyridme maleate 1.03 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48215 nAChR BRAIN RAT 3H-NICOTINE 6-Methyl-3-(1 -methyl-2-pyrrohdmyl)pyridme dthydrochlortde 1.8 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48216 nAChR BRAIN RAT 3H-NICOTINE 6-methoxynicotine 22 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48217 nAChR BRAIN RAT 3H-NICOTINE 5-(N-Ethyl)amino-5,0,7,8-tetrahydroquinoline maleate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48218 nAChR BRAIN RAT 3H-NICOTINE 1,2,3.4-Tetrahydro[2,7]naphthyrldine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48219 nAChR BRAIN RAT 3H-NICOTINE 2-Methyl-l,2,3.4-tetrahydro[2,7]naphthyridine oxalate 18 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48220 nAChR BRAIN RAT 3H-NICOTINE 2-Ethyl-l,2,3,4-tetrahydro[2,7]naphthyrtdme oxalate 52 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48221 nAChR BRAIN RAT 3H-NICOTINE 2-Propyl-l,2,3,4-tetrahydro[2,7]naphthyrMme oxalate 1640 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48222 nAChR BRAIN RAT 3H-NICOTINE 2-1sopropyl-l.2,3,4-tetrahydro[2.7]naphthyridine oxalate 123 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48223 nAChR BRAIN RAT 3H-NICOTINE 5,6,7,9-Tetrahydro-8H-pyrldo[3,4-c]azepine oxalate 1100 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48224 nAChR BRAIN RAT 3H-NICOTINE 8-Methyl-5.6,7,9-tetrahydro-8H-pyrido[3,4-c]azepine oxalate 780 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48225 nAChR BRAIN RAT 3H-NICOTINE 2-Methyl- 2.3-dihydro-l H-pyrrolo[3,4-c]pyrMine oxalate 85 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48226 nAChR BRAIN RAT 3H-NICOTINE 6-Chloro-3-(N-ethyl-N-methyl)aminomethylpyridine oxalat 41 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48227 nAChR BRAIN RAT 3H-NICOTINE 6-Methyl-3-(N-ethyl-N-methylammomethyl)pyridme oxalate 66 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48228 nAChR BRAIN RAT 3H-NICOTINE 6-Metho,D'-3-(N-ethyl-N-methylamtnomethyl)pyndine oxalate 640 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48229 nAChR BRAIN RAT 3H-NICOTINE 6-Fluoro-3-(N-ethyl-N-methyl)aminomethylpyridine oxalate 93 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48230 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Methyl-N-n-propylammomethyl)-2-methylpyridine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48231 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Methyl-N-n-propylaminomethyl)pyridine oxalate 1140 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48232 nAChR BRAIN RAT 3H-NICOTINE 3-(N-n-Butyl-N-methylaminornethyl)pyridine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48233 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Methyl-N-n-peno, laminomethyl)pyrtdine oxalate >10000 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48234 nAChR BRAIN RAT 3H-NICOTINE 3-(N-Cyclopropyl-N-methylaminornethyl)pyrMine oxalate 840 Dukat, M et al, 1999 Jan 15, 2025 Jan 15, 2025
48235 SLC6A4 CLONED HUMAN 3H-CITALOPRAM stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48236 5-HT1A CLONED HUMAN 3H-8-OH-DPAT stepholidine 143.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48237 5-HT1B CLONED HUMAN 3H-GR-125743 stepholidine 6984 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48238 5-HT1D CLONED HUMAN 3H-GR-125743 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48239 5-HT1E CLONED HUMAN 3H-5HT stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48240 5-HT2A CLONED HUMAN 3H-KETANSERIN stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48241 5-HT2C CLONED RAT 3H-MESULERGINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48242 5-HT3 CLONED HUMAN 3H-LY 278584 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48243 CB1 CLONED HUMAN 3H-LSD stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
48244 5-HT6 CLONED HUMAN 3H-LSD stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48245 5-HT7 CLONED HUMAN 3H-LSD stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48246 5-HT2B CLONED HUMAN 3H-LSD stepholidine 226 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48247 SLC6A4 CLONED HUMAN 3H-CITALOPRAM PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48248 5-HT1A CLONED HUMAN 3H-8-OH-DPAT PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48249 5-HT1B CLONED HUMAN 3H-GR-125743 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48250 5-HT1D CLONED HUMAN 3H-GR-125743 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48251 5-HT1E CLONED HUMAN 3H-5HT PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48252 5-HT2A CLONED HUMAN 3H-KETANSERIN PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48253 5-HT2C CLONED RAT 3H-MESULERGINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48254 5-HT3 CLONED HUMAN 3H-ZACOPRIDE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48255 CB1 CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
48256 5-HT6 CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48257 5-HT7 CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48258 5-HT2B CLONED HUMAN 3H-LSD PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48259 Alpha1A CLONED HUMAN 3H-PRAZOSIN PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48260 Alpha1B CLONED HUMAN 3H-PRAZOSIN PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48261 Alpha2A CLONED HUMAN 3H-CLONIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48262 Alpha2B CLONED HUMAN 3H-CLONIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48263 Alpha2C CLONED HUMAN 3H-CLONIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48264 Beta1 CLONED HUMAN 125I-Pindolol PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48265 Beta2 CLONED HUMAN 125I-Pindolol PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
48266 H1 CLONED HUMAN 3H-PYRILAMINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48267 H2 CLONED HUMAN 3H-TIOTIDINE PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48268 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48269 H4 CLONED HUMAN 3H-Histamine PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48270 D1 CLONED HUMAN 3H-SCH23390 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48271 D2 CLONED HUMAN 3H-NMSP PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48272 D3 CLONED RAT 3H-NMSP PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48273 D4 CLONED HUMAN 3H-NMSP PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48274 SLC6A3 CLONED HUMAN 3H-WIN 35,428 PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48275 NET CLONED HUMAN 3H-Nisoxetine PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48276 M2 CLONED HUMAN 3H-QNB PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48277 M5 CLONED HUMAN 3H-QNB PBR28 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48278 KOR CLONED HUMAN 3H-Diprenorphine PBR28 2.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48279 Alpha1A CLONED HUMAN 3H-PRAZOSIN stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48280 Alpha1B CLONED HUMAN 3H-PRAZOSIN stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48281 Alpha2A CLONED HUMAN 3H-CLONIDINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48282 Alpha2B CLONED HUMAN 3H-CLONIDINE stepholidine 6884 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48283 Alpha2C CLONED HUMAN 3H-CLONIDINE stepholidine 214.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48284 Beta1 CLONED HUMAN 125I-Pindolol stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48285 Beta2 CLONED HUMAN 125I-Pindolol stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
48286 H1 CLONED HUMAN 3H-PYRILAMINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48287 H2 CLONED HUMAN 3H-TIOTIDINE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48288 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48289 H4 CLONED HUMAN 3H-Histamine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48290 D1 CLONED HUMAN 3H-SCH23390 stepholidine 5.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48291 D2 CLONED HUMAN 3H-NMSP stepholidine 974.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48292 D3 CLONED RAT 3H-NMSP stepholidine 30.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48293 D4 CLONED HUMAN 3H-NMSP stepholidine 3748 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48294 D5 CLONED HUMAN 3H-SCH23390 stepholidine 4.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48295 SLC6A3 CLONED HUMAN 3H-WIN 35,428 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48296 NET CLONED HUMAN 3H-Nisoxetine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48297 MOR CLONED HUMAN 3H-Diprenorphine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48298 M2 CLONED HUMAN 3H-QNB stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48299 DOR CLONED HUMAN 3H-DADLE stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48300 KOR CLONED HUMAN 3H-Diprenorphine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48301 M5 CLONED HUMAN 3H-QNB stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48302 KOR FOREBRAIN RAT 3H-MUSCIMOL stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
48303 HEART RAT 3H-Nitrendipine stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48304 CB2 CLONED HUMAN 3H-CP-55940 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48305 CB1 CLONED HUMAN 3H-CP-55940 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48306 I1 PC12 RAT 125I-Pindolol stepholidine 8909 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48307 Sigma 1 BRAIN RAT 3H-Pentazocine(+) stepholidine 1600 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48308 Sigma 2 PC12 RAT 3H-DTG stepholidine 53.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48309 NMDA FOREBRAIN RAT 3H-MK-801 stepholidine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48310 mGluR5 LLC-PK1 cells PORCINE Functional Glutamate 9750 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48311 LLC-PK1 cells PORCINE Functional Glutamate 7670 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48312 LLC-PK1 cells PORCINE Functional Quisqualate 260 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48313 mGluR5 LLC-PK1 cells PORCINE Functional Quisqualate 22 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48314 LLC-PK1 cells PORCINE Functional Quisqualate 47 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48315 LLC-PK1 cells PORCINE Functional Ibotenate >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48316 mGluR5 LLC-PK1 cells PORCINE Functional Ibotenate 2870 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48317 LLC-PK1 cells PORCINE Functional Ibotenate 1930 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48318 LLC-PK1 cells PORCINE Functional (+/-)-trans-ACPD 2880 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48319 mGluR5 LLC-PK1 cells PORCINE Functional (+/-)-trans-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48320 LLC-PK1 cells PORCINE Functional (+/-)-trans-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48321 LLC-PK1 cells PORCINE Functional 1S, 3R-ACPD 9300 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48322 mGluR5 LLC-PK1 cells PORCINE Functional 1S, 3R-ACPD 6700 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48323 LLC-PK1 cells PORCINE Functional 1S, 3R-ACPD 5300 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48324 LLC-PK1 cells PORCINE Functional 1R,3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48325 mGluR5 LLC-PK1 cells PORCINE Functional 1R,3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48326 LLC-PK1 cells PORCINE Functional 1R,3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48327 LLC-PK1 cells PORCINE Functional 1S, 3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48328 mGluR5 LLC-PK1 cells PORCINE Functional 1S, 3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48329 LLC-PK1 cells PORCINE Functional 1S, 3S-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48330 LLC-PK1 cells PORCINE Functional 1R,3R-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48331 mGluR5 LLC-PK1 cells PORCINE Functional 1R,3R-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 28, 2025
48332 LLC-PK1 cells PORCINE Functional 1R,3R-ACPD >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48333 LLC-PK1 cells PORCINE Functional Glutamate >10000 Joly C, et.al., 1995 Jan 15, 2025 Jan 15, 2025
48334 5-HT2A CLONED RAT 3H-KETANSERIN 1-(Aminomethyl)dibenzo[b,e]bicyclo[2.2.2]octadiene Hydrochloride 770 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48335 5-HT2A CLONED RAT 3H-KETANSERIN 9-Aminomethyl-9,10-dihydro-9,10-methanoanthracene Hydrochloride 6780 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48336 5-HT2A CLONED RAT 3H-KETANSERIN 9-Methyl-9-aminomethyl-9,10-dihydroanthracene Oxalate 65 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48337 5-HT2A CLONED RAT 3H-KETANSERIN 9-Aminomethyl-10,10-dimethyl-9,10-dihydroanthracene Oxalate 330 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48338 5-HT2A CLONED RAT 3H-KETANSERIN 11-Amino-9,10-dihydro-9,10-ethanoanthracene Oxalate >10000 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48339 5-HT2A CLONED RAT 3H-KETANSERIN 9-(1-Aminoethyl)-9,10-dihydroanthracene Hydrochloride 193 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48340 5-HT2A CLONED RAT 3H-KETANSERIN 2,3,7,11b-Tetrahydrodibenzo[d,e,h]isoquinoline Oxalate 296 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48341 5-HT2A CLONED RAT 3H-KETANSERIN AMDA 20 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48342 5-HT2A CLONED RAT 3H-KETANSERIN 2,2-diphenylethylamine 4610 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48343 5-HT2A CLONED RAT 3H-KETANSERIN tetrahydronaphthalene >10000 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48344 5-HT2A CLONED RAT 3H-KETANSERIN 2-(2-benzylphenyl)-ethylamine 1810 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48345 5-HT2A CLONED RAT 3H-KETANSERIN [a,d]dibenz-fused cycloheptane 112 Runyon SP et al., 2002 Jan 15, 2025 Jan 15, 2025
48346 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PERGOLIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48347 Sigma 2 PC12 RAT 3H-DTG PERGOLIDE 922.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48348 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Memantine 4131 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48349 Sigma 2 PC12 RAT 3H-DTG Memantine 9450 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48350 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Chloroquine 108.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48351 Sigma 2 PC12 RAT 3H-DTG Chloroquine 1129 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48352 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PPP, S(-)-3 774.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48353 Sigma 2 PC12 RAT 3H-DTG PPP, S(-)-3 1415 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48354 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PPP, R(+)-3 192.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48355 Sigma 2 PC12 RAT 3H-DTG PPP, R(+)-3 181.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48356 Sigma 1 BRAIN RAT 3H-Pentazocine(+) FLUOXETINE 1911 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48357 Sigma 2 PC12 RAT 3H-DTG FLUOXETINE 1121 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48358 Sigma 2 PC12 RAT 3H-DTG DESIPRAMINE 1611 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48359 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Amiodarone 791.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48360 Sigma 1 BRAIN RAT 3H-Pentazocine(+) SKF 82957 1444 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48361 Sigma 2 PC12 RAT 3H-DTG PHENYLEPHRINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48363 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 6-(((6-chloro-4H-1,3-benzodioxin-8-yl)methyl)thio)-3-(cyclopropylmethyl)-1,2,3,4-tetrahydro-1,3,5-triazine 410.83 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48364 Sigma 2 PC12 RAT 3H-DTG R-(+) staurosine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48365 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Lofepramine 2520 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48366 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Rimonabant 4350 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48367 Sigma 2 PC12 RAT 3H-DTG CLOZAPINE-N-OXIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48368 Sigma 1 BRAIN RAT 3H-Pentazocine(+) CLOZAPINE-N-OXIDE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48369 Sigma 1 BRAIN RAT 3H-Pentazocine(+) L-DOPA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48370 Sigma 2 PC12 RAT 3H-DTG L-DOPA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48371 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Picrotoxin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48372 Sigma 2 PC12 RAT 3H-DTG Picrotoxin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48373 Sigma 1 BRAIN RAT 3H-Pentazocine(+) YOHIMBINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48374 Sigma 2 PC12 RAT 3H-DTG YOHIMBINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48375 Sigma 1 BRAIN RAT 3H-Pentazocine(+) SKF 75670 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48376 Sigma 2 PC12 RAT 3H-DTG SKF 75670 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48377 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Arecoline >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48378 Sigma 2 PC12 RAT 3H-DTG Arecoline >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48379 Sigma 1 BRAIN RAT 3H-Pentazocine(+) DESIPRAMINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48380 Sigma 2 PC12 RAT 3H-DTG Amiodarone >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48381 Sigma 2 PC12 RAT 3H-DTG SKF 82957 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48382 Sigma 2 PC12 RAT 3H-DTG Tramadol(+-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48383 Sigma 2 PC12 RAT 3H-DTG Pramipexole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48384 Sigma 2 PC12 RAT 3H-DTG Amantadine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48385 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Agomelatine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48386 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Tramadol(+-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48387 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Amantadine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48388 Sigma 1 BRAIN RAT 3H-Pentazocine(+) topiramate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48389 Sigma 2 PC12 RAT 3H-DTG topiramate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48390 Sigma 1 BRAIN RAT 3H-Pentazocine(+) PHENYLEPHRINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48391 Sigma 1 BRAIN RAT 3H-Pentazocine(+) DDMV >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48392 Sigma 2 PC12 RAT 3H-DTG Menthol-(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48393 Sigma 2 PC12 RAT 3H-DTG Menthol-(-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48394 Sigma 2 PC12 RAT 3H-DTG Neomenthol-(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48395 Sigma 2 PC12 RAT 3H-DTG Neomenthol-(-) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48396 Sigma 2 PC12 RAT 3H-DTG Isomenthol-(+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48397 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Thujone >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48398 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Acetyl-L-Carnitine HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48399 Sigma 1 BRAIN RAT 3H-Pentazocine(+) L-Carnitine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48400 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Triamcinolone (Fluoxyprednisolone) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48401 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Phenobarbitol sodium salt >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48402 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Dieldrin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48403 Sigma 1 BRAIN RAT 3H-Pentazocine(+) D,L Kavain >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48404 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Myristicin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48405 Sigma 1 BRAIN RAT 3H-Pentazocine(+) alpha-Estradiol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48406 Sigma 1 BRAIN RAT 3H-Pentazocine(+) MTEP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48407 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Indinavir sulphate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48408 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Efavirenz >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48409 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Stavudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48410 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Ritonavir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48411 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Nelfinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48412 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Nevirapine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48413 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Zalcitabine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48414 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Saquinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48415 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Zidovudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48416 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Tenofovir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48417 Sigma 1 BRAIN RAT 3H-Pentazocine(+) DHL >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48418 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4OHBA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48419 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4OHMNA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48420 Sigma 1 BRAIN RAT 3H-Pentazocine(+) securinine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48421 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 3-(2,4-dithioxo-1,3-thiazolidin-3-yl)propanoic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48422 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4-methyl[1]benzofuro[3,2-g]quinolin-2-ol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48423 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Gitoxigenin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48424 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Triciribine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48425 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 6-Benzylthioinosine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48426 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Hoodia Extract >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48427 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Galnon >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48428 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Glaucine HBr >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48429 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Glaucium fl. extract >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48430 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Acamprosate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48431 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Oseltamivir PO4 - Tamiflu >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48432 Sigma 1 BRAIN RAT 3H-Pentazocine(+) Oseltamivir Acid - tamiflu metabolite >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48444 Sigma 2 PC12 RAT 3H-DTG Thujone >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48445 Sigma 2 PC12 RAT 3H-DTG Acetyl-L-Carnitine HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48446 Sigma 2 PC12 RAT 3H-DTG L-Carnitine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48447 Sigma 2 PC12 RAT 3H-DTG Triamcinolone (Fluoxyprednisolone) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48448 Sigma 2 PC12 RAT 3H-DTG Phenobarbitol sodium salt >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48449 Sigma 2 PC12 RAT 3H-DTG Dieldrin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48450 Sigma 2 PC12 RAT 3H-DTG D,L Kavain >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48451 Sigma 2 PC12 RAT 3H-DTG 1-phenlsemicarbazide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48452 Sigma 2 PC12 RAT 3H-DTG Myristicin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48453 Sigma 2 PC12 RAT 3H-DTG alpha-Estradiol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48454 Sigma 2 PC12 RAT 3H-DTG Indinavir sulphate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48455 Sigma 2 PC12 RAT 3H-DTG Efavirenz >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48456 Sigma 2 PC12 RAT 3H-DTG Stavudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48457 Sigma 2 PC12 RAT 3H-DTG Ritonavir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48458 Sigma 2 PC12 RAT 3H-DTG Nelfinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48459 Sigma 2 PC12 RAT 3H-DTG Nevirapine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48460 Sigma 2 PC12 RAT 3H-DTG Zalcitabine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48461 Sigma 2 PC12 RAT 3H-DTG Saquinavir mesylate >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48462 Sigma 2 PC12 RAT 3H-DTG Zidovudine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48463 Sigma 2 PC12 RAT 3H-DTG Tenofovir >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48464 Sigma 2 PC12 RAT 3H-DTG DHL >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48465 Sigma 2 PC12 RAT 3H-DTG 4OHBA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48466 Sigma 2 PC12 RAT 3H-DTG 4OHMNA >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48467 Sigma 2 PC12 RAT 3H-DTG securinine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48468 Sigma 2 PC12 RAT 3H-DTG 3-(2,4-dithioxo-1,3-thiazolidin-3-yl)propanoic acid >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48469 Sigma 2 PC12 RAT 3H-DTG 4-methyl[1]benzofuro[3,2-g]quinolin-2-ol >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48470 Sigma 2 PC12 RAT 3H-DTG Gitoxigenin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48471 Sigma 2 PC12 RAT 3H-DTG Triciribine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48472 Sigma 2 PC12 RAT 3H-DTG 6-Benzylthioinosine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48473 Sigma 2 PC12 RAT 3H-DTG Hoodia Extract >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48474 Sigma 2 PC12 RAT 3H-DTG Galnon >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48475 Sigma 2 PC12 RAT 3H-DTG MTEP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48476 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 1-phenlsemicarbazide >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48555 5-HT2B CLONED HUMAN 3H-LSD METHAMPHETAMINE (+) >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48556 NET CLONED HUMAN 3H-Nisoxetine METHAMPHETAMINE (+) 965.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48557 Alpha2A CLONED HUMAN 3H-CLONIDINE METHAMPHETAMINE (+) 4142 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48558 Alpha2B CLONED HUMAN 3H-CLONIDINE METHAMPHETAMINE (+) 744.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48559 Alpha2C CLONED HUMAN 3H-CLONIDINE METHAMPHETAMINE (+) 813.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48560 5-HT1A CLONED HUMAN 3H-8-OH-DPAT mCPP 43.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48561 5-HT1B CLONED HUMAN 3H-5CT mCPP 163.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48562 5-HT2A CLONED HUMAN 3H-KETANSERIN mCPP 196.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48563 5-HT2B CLONED HUMAN 3H-LSD mCPP 19.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48564 5-HT2C CLONED RAT 3H-MESULERGINE mCPP 108 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48565 5-HT3 CLONED HUMAN 3H-LY 278584 mCPP 427 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48566 5-HT5A CLONED HUMAN 3H-LSD mCPP 1354 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48567 5-HT6 CLONED HUMAN 3H-LSD mCPP 1748 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48568 5-HT7 CLONED HUMAN 3H-LSD mCPP 162.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48569 Alpha1A CLONED HUMAN 3H-PRAZOSIN mCPP 1386 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48570 Alpha1B CLONED HUMAN 3H-PRAZOSIN mCPP 914.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48571 Alpha2A CLONED HUMAN 3H-CLONIDINE mCPP 145.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48572 Alpha2B CLONED HUMAN 3H-CLONIDINE mCPP 105.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48573 Alpha2C CLONED HUMAN 3H-CLONIDINE mCPP 123.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48574 Beta1 CLONED HUMAN 125I-Pindolol mCPP 2359 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48575 Beta2 CLONED HUMAN 125I-Pindolol mCPP 3474 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
48576 HEART RAT 3H-Nitrendipine mCPP 6043 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48577 D3 CLONED RAT 3H-NMSP mCPP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48578 D5 CLONED HUMAN 3H-SCH23390 mCPP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48579 H1 CLONED HUMAN 3H-PYRILAMINE mCPP 326.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48580 I1 PC12 RAT 125I-Pindolol mCPP 758.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48581 NET CLONED HUMAN 3H-Nisoxetine mCPP >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48582 SLC6A4 CLONED HUMAN 3H-CITALOPRAM mCPP 328.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48583 Sigma 2 PC12 RAT 3H-DTG mCPP 8350 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
48585 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 800 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48586 CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 475 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48587 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2400 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48588 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 330 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48589 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 700 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48590 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 417 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48591 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 7700 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48592 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48593 CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48594 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48595 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48596 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48597 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.25 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48598 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.9 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48599 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 17.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48600 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 158 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48601 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 18.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48602 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 42.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48603 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 35 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48604 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 18.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48605 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 1.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48606 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 2.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48607 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48608 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48609 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48610 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48611 CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48612 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 30 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48613 CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 1.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48614 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 9 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48615 CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 4.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48616 CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48617 GNRHR CLONED HUMAN Functional alpha-tetrahydropyran-beta-sulfone 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48618 GNRHR CLONED HUMAN Functional tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48619 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48620 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(3-methoxybenzyl)-4-{[(4-phenoxyphenyl)sulfonyl]methyl}piperidine-4-carboxamide Hydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48621 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-(2-phenylethyl)piperidine-4-carboxamide Hydrochloride 1.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48622 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[(4-phenoxyphenyl)sulfonyl]methyl}-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.55 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48623 GNRHR CLONED HUMAN Functional 4-({[4-(3,4-Dimethylphenoxy)phenyl]sulfonyl}methyl)-N-hydroxy-1-prop-2-ynylpiperidine-4-carboxamide Hydrochloride 0.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48624 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 435 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48625 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48626 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 18.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48627 CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48628 GNRHR CLONED HUMAN Functional 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxytetrahydro-2H-pyran-4-carboxamide 0.15 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48629 CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 1140 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48630 CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48631 GNRHR CLONED HUMAN Functional 1-tert-Butyl 4-[(Hydroxyamino)carbonyl]-4-[(4-phenoxyphenyl)sulfonyl]piperidine-1-carboxylate 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48632 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 1060 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48633 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 0.22 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48634 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 59 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48635 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 3.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48636 CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48637 GNRHR CLONED HUMAN Functional 1-N-Hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide 0.37 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48638 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 464 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48639 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48640 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.29 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48641 GNRHR CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48642 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 350 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48643 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48644 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48645 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 9.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48646 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.7 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48647 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48648 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 400 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48649 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48650 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48651 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 12.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48652 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48653 GNRHR CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48654 CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 770 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48655 CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48656 GNRHR CLONED HUMAN Functional 1-(Cyclopropylmethyl)-N-hydroxy-4-[(4-phenoxyphenyl)sulfonyl]piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48657 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 274 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48658 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.13 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48659 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 12.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48660 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.85 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48661 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48662 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}-1- (2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.22 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48663 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 464 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48664 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48665 GNRHR CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48666 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 800 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48667 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48668 CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48669 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(methylsulfonyl)-4-{[4-(phenoxyphenyl]sulfonyl}piperidine-4-carboxamide 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48670 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48671 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48672 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 39.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48673 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 11.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48674 CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 9.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48675 GNRHR CLONED HUMAN Functional N-Hydroxy-1-methyl-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.68 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48676 CLONED HUMAN Functional 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48677 CLONED HUMAN Functional 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48678 GNRHR CLONED HUMAN Functional 1-Ethyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48679 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48680 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48681 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 20 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48682 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48683 CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48684 GNRHR CLONED HUMAN Functional N-Hydroxy-1-(2-methoxyethyl)-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48685 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48686 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.1 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48687 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 23.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48688 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 3.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48689 CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 2.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48690 GNRHR CLONED HUMAN Functional 1-Cyclopropyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide Hydrochloride 0.2 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48691 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride >10000 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48692 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride 0.15 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48693 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(vinylmethyl)piperidine-4-carboxamide Hydrochloride 0.3 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48694 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 8660 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48695 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.33 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48696 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 13 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48697 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 1.8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48698 CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 1.5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48699 GNRHR CLONED HUMAN Functional N-Hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}-1-(2-propynyl)-4-piperidinecarboxamide, Monohydrochloride 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48700 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 7300 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48701 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 0.4 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48702 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 23 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48703 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 5 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48704 CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 8 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025
48705 GNRHR CLONED HUMAN Functional 1-Acetyl-N-hydroxy-4-{[4-(phenylthio)phenyl]sulfonyl}piperidine-4-carboxamide 0.6 Becker DP, et al., 2005 Jan 15, 2025 Jan 15, 2025