The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 84,001-85,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
867495-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(furoyl)piperazin-1-yl)ethyl)isonicotinamide331Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867505-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) isonicotinamide55Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867515-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) isonicotinamide6.9Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867525-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) isonicotinamide0.658Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867535-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide10Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867545-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide0.00956Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867555-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide28.7Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867565-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl) isonicotinamide385Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867575-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl) isonicotinamide41.8Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867585-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl) isonicotinamide5.23Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867595-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-OH-DPAT0.8Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867605-HT2AFR. CORTEXRAT3H-KETANSERINKETANSERIN0.85Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867615-HT2CFR. CORTEXRAT3H-MESULERGINEMESULERGINE1.9Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867625-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-phenylpiperazin-1-yl)propyl)isonicotinamide29.8Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867635-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-phenylpiperazin-1-yl)propyl)isonicotinamide112Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867645-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-phenylpiperazin-1-yl)propyl)isonicotinamide56.7Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867655-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide13.9Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867665-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide0.254Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867675-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867685-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867695-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide1260Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867705-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) isonicotinamide24.7Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867715-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl) isonicotinamide9.59Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867725-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl) isonicotinamide207Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867735-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867745-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl) isonicotinamide191Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867755-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl) isonicotinamide182Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867765-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl) isonicotinamide122Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867775-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(o-tolyl)piperazin-1-yl)propyl)isonicotinamide3310Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867785-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(o-tolyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867795-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(o-tolyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867805-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867815-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide770Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867825-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide8.42Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867835-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide124Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867845-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide92.6Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867855-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867865-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867875-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide1380Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867885-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide590Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867895-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide325Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867905-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide3.53Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867915-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-chlorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867925-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867935-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide1.07Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867945-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(3,4-dichlorophenyl)piperazin-1-yl)propyl) isonicotinamide219Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867955-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide331Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867965-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide0.039Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867975-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide21.2Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867985-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
867995-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide0.228Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868005-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide99.1Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868015-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide100Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868025-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide792Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868035-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(pyridin-2-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868045-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868055-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide0.00985Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868065-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide9.19Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868075-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide0.0113Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868085-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868095-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide2.19Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868105-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(furoyl)piperazin-1-yl)propyl)isonicotinamide3080Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868115-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(furoyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868125-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(furoyl)piperazin-1-yl)propyl)isonicotinamide779Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868135-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868145-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868155-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-chlorobenzhydryl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868165-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868175-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868185-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide0.13Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868195-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide1060Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868205-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
868215-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(naphthalen-1-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86822BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide53Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86823BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide828Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86824D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86825D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl) isonicotinamide537Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86826D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86827D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86828BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1120Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86829BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide78.8Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86830BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide299Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86831BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86832D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86833D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86834D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86835D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86836BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide221Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86837BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide123Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86838BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide918Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86839BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86840D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86841D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86842D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86843D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86844BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86845BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)isonicotinamide1880Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86846BRAIN CORTEXRAT3H-PRAZOSINN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86847BRAIN CORTEXRAT3H-YohimbineN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86848D1Corpus StriatumRAT3H-SCH23390N-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86849D2Corpus StriatumRAT3H-SPIPERONEN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) isonicotinamide1680Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86850D2Corpus StriatumRAT3H-SPIPERONEN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86851D1Corpus StriatumRAT3H-SCH23390N-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86852BRAIN CORTEXRAT3H-YohimbineN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide170Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86853BRAIN CORTEXRAT3H-PRAZOSINN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) isonicotinamide67.6Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86854BRAIN CORTEXRAT3H-PRAZOSINN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide2350Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86855BRAIN CORTEXRAT3H-YohimbineN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide604Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86856D1Corpus StriatumRAT3H-SCH23390N-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86857D2Corpus StriatumRAT3H-SPIPERONEN-(3-(4-(2-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide1420Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86858D2Corpus StriatumRAT3H-SPIPERONEN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86859D1Corpus StriatumRAT3H-SCH23390N-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide451Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86860BRAIN CORTEXRAT3H-YohimbineN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide1310Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86861BRAIN CORTEXRAT3H-PRAZOSINN-(3-(4-(4-fluorophenyl)piperazin-1-yl)propyl) isonicotinamide976Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86862BRAIN CORTEXRAT3H-PRAZOSINN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86863BRAIN CORTEXRAT3H-YohimbineN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86864D1Corpus StriatumRAT3H-SCH23390N-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86865D2Corpus StriatumRAT3H-SPIPERONEN-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propyl) isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86866D2Corpus StriatumRAT3H-SPIPERONEN-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86867D1Corpus StriatumRAT3H-SCH23390N-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide127Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86868BRAIN CORTEXRAT3H-YohimbineN-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86869BRAIN CORTEXRAT3H-PRAZOSINN-(3-(4-(piperonyl)piperazin-1-yl)propyl)isonicotinamide1000Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86870BRAIN CORTEXRAT3H-PRAZOSINN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide2220Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86871BRAIN CORTEXRAT3H-YohimbineN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide2220Fiorino F et al 2016Jan 15, 2025Jan 15, 2025
86872D1Corpus StriatumRAT3H-SCH23390N-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide0.0983Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86873D2Corpus StriatumRAT3H-SPIPERONEN-(3-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)propyl) isonicotinamide26.6Fiorino F et al 2016Jan 15, 2025Jan 28, 2025
86874D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione1Zareba P et al 2020Jan 15, 2025Jan 28, 2025
868755-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione27Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868765-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione4Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868775-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione486Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868785-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione9Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86879D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione35Zareba P et al 2020Jan 15, 2025Jan 28, 2025
868805-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione12Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868815-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione541Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868825-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione1641Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868835-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)hexa hydro-1H-4,7-methanoisoindole-1,3(2H)-dione198Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868845-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione39Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868855-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione1142Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868865-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione81Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868875-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione18Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86888D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl) hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione225Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86889D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione370Zareba P et al 2020Jan 15, 2025Jan 28, 2025
868905-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione55Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868915-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione73Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868925-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione3028Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868935-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl) qhexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione202Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868945-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione117Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868955-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione536Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868965-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione161Zareba P et al 2020Jan 15, 2025Jan 15, 2025
868975-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione32Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86898D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione55Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86899D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(3-trifluoromethylphenyl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione168Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869005-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(3-trifluoromethylphenyl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione22Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869015-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(3-trifluoromethylphenyl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione189Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869025-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(3-trifluoromethylphenyl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione2205Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869035-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(3-trifluoromethylphenyl)piperazin-1- yl)hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione53Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869045-HT7CLONEDHUMAN3H-5-CT(3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione146Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869055-HT6CLONEDHUMAN3H-LSD(3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione4874Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869065-HT2ACLONEDHUMAN3H-KETANSERIN(3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione785Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869075-HT1ACLONEDHUMAN3H-8-OH-DPAT(3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione4Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86908D2CLONEDHUMAN3H-RACLOPRIDE(3aR,4S,7R,7aS)-2-(6-(4-(2-methoxyphenyl)piperazin-1-yl) hexyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione41Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86909D2CLONEDHUMAN3H-RACLOPRIDE2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)isoindoline1,3-dione10Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869105-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)isoindoline1,3-dione18Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869115-HT2ACLONEDHUMAN3H-KETANSERIN2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)isoindoline1,3-dione24Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869125-HT6CLONEDHUMAN3H-LSD2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)isoindoline1,3-dione160Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869135-HT7CLONEDHUMAN3H-5-CT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)isoindoline1,3-dione114Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869145-HT7CLONEDHUMAN3H-5-CT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-[1,2,4] triazolo[4,3-a]pyridin-3(2H)-one747Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869155-HT6CLONEDHUMAN3H-LSD2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-[1,2,4] triazolo[4,3-a]pyridin-3(2H)-one252Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869165-HT2ACLONEDHUMAN3H-KETANSERIN2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-[1,2,4] triazolo[4,3-a]pyridin-3(2H)-one5Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869175-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-[1,2,4] triazolo[4,3-a]pyridin-3(2H)-one11Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86918D2CLONEDHUMAN3H-RACLOPRIDE2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-[1,2,4] triazolo[4,3-a]pyridin-3(2H)-one9Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86919D2CLONEDHUMAN3H-RACLOPRIDE3-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d] oxazol-2(3H)-one16Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869205-HT1ACLONEDHUMAN3H-8-OH-DPAT3-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d] oxazol-2(3H)-one5Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869215-HT2ACLONEDHUMAN3H-KETANSERIN3-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d] oxazol-2(3H)-one6Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869225-HT6CLONEDHUMAN3H-LSD3-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d] oxazol-2(3H)-one189Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869235-HT7CLONEDHUMAN3H-5-CT3-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d] oxazol-2(3H)-one7Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869245-HT7CLONEDHUMAN3H-5-CT2-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)thio) benzo[d]oxazole72Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869255-HT6CLONEDHUMAN3H-LSD2-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)thio) benzo[d]oxazole302Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869265-HT2ACLONEDHUMAN3H-KETANSERIN2-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)thio) benzo[d]oxazole13Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869275-HT1ACLONEDHUMAN3H-8-OH-DPAT2-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)thio) benzo[d]oxazole10Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86928D2CLONEDHUMAN3H-RACLOPRIDE2-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)thio) benzo[d]oxazole33Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86929D2CLONEDHUMAN3H-RACLOPRIDE6-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)oxy)- 3,4-dihydroquinolin-2(1H)-one39Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869305-HT1ACLONEDHUMAN3H-8-OH-DPAT6-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)oxy)- 3,4-dihydroquinolin-2(1H)-one20Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869315-HT2ACLONEDHUMAN3H-KETANSERIN6-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)oxy)- 3,4-dihydroquinolin-2(1H)-one20Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869325-HT6CLONEDHUMAN3H-LSD6-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)oxy)- 3,4-dihydroquinolin-2(1H)-one805Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869335-HT7CLONEDHUMAN3H-5-CT6-((6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)oxy)- 3,4-dihydroquinolin-2(1H)-one387Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869345-HT7CLONEDHUMAN3H-5-CT1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[cd] indol-2(1H)-one36Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869355-HT6CLONEDHUMAN3H-LSD1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[cd] indol-2(1H)-one568Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869365-HT2ACLONEDHUMAN3H-KETANSERIN1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[cd] indol-2(1H)-one55Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869375-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[cd] indol-2(1H)-one71Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86938D2CLONEDHUMAN3H-RACLOPRIDE1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[cd] indol-2(1H)-one56Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86939D2CLONEDHUMAN3H-RACLOPRIDE2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)–2H-naphtho [1,8-cd]isothiazole 1,1-dioxide18Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869405-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)–2H-naphtho [1,8-cd]isothiazole 1,1-dioxide63Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869415-HT2ACLONEDHUMAN3H-KETANSERIN2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)–2H-naphtho [1,8-cd]isothiazole 1,1-dioxide32Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869425-HT6CLONEDHUMAN3H-LSD2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)–2H-naphtho [1,8-cd]isothiazole 1,1-dioxide158Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869435-HT7CLONEDHUMAN3H-5-CT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)–2H-naphtho [1,8-cd]isothiazole 1,1-dioxide105Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869445-HT7CLONEDHUMAN3H-5-CT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo[de] isoquinoline-1,3(2H)-dione118Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869455-HT6CLONEDHUMAN3H-LSD2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo[de] isoquinoline-1,3(2H)-dione110Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869465-HT2ACLONEDHUMAN3H-KETANSERIN2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo[de] isoquinoline-1,3(2H)-dione53Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869475-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo[de] isoquinoline-1,3(2H)-dione86Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86948D2CLONEDHUMAN3H-RACLOPRIDE2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo[de] isoquinoline-1,3(2H)-dione59Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86949D2CLONEDHUMAN3H-RACLOPRIDE1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-5,6- dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one1Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869505-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-5,6- dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one44Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869515-HT2ACLONEDHUMAN3H-KETANSERIN1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-5,6- dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one12Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869525-HT6CLONEDHUMAN3H-LSD1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-5,6- dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one379Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869535-HT7CLONEDHUMAN3H-5-CT1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-5,6- dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one16Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869545-HT7CLONEDHUMAN3H-5-CTN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-N-(3- (trifluoromethyl)phenyl)benzenesulfonamide193Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869555-HT6CLONEDHUMAN3H-LSDN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-N-(3- (trifluoromethyl)phenyl)benzenesulfonamide1103Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869565-HT2ACLONEDHUMAN3H-KETANSERINN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-N-(3- (trifluoromethyl)phenyl)benzenesulfonamide65Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869575-HT1ACLONEDHUMAN3H-8-OH-DPATN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-N-(3- (trifluoromethyl)phenyl)benzenesulfonamide42Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86958D2CLONEDHUMAN3H-RACLOPRIDEN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-N-(3- (trifluoromethyl)phenyl)benzenesulfonamide164Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86959D2CLONEDHUMAN3H-RACLOPRIDEN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-4- methyl-N-phenylbenzenesulfonamide106Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869605-HT1ACLONEDHUMAN3H-8-OH-DPATN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-4- methyl-N-phenylbenzenesulfonamide32Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869615-HT2ACLONEDHUMAN3H-KETANSERINN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-4- methyl-N-phenylbenzenesulfonamide26Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869625-HT6CLONEDHUMAN3H-LSDN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-4- methyl-N-phenylbenzenesulfonamide772Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869635-HT7CLONEDHUMAN3H-5-CTN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-4- methyl-N-phenylbenzenesulfonamide54Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869645-HT7CLONEDHUMAN3H-5-CT1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo [d]imidazol-2(3H)-one7Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869655-HT6CLONEDHUMAN3H-LSD1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo [d]imidazol-2(3H)-one189Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869665-HT2ACLONEDHUMAN3H-KETANSERIN1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo [d]imidazol-2(3H)-one6Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869675-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo [d]imidazol-2(3H)-one16Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86968D2CLONEDHUMAN3H-RACLOPRIDE1-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)-1H-benzo [d]imidazol-2(3H)-one16Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86969D2CLONEDHUMAN3H-RACLOPRIDEN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzamide14Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869705-HT1ACLONEDHUMAN3H-8-OH-DPATN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzamide22Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869715-HT2ACLONEDHUMAN3H-KETANSERINN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzamide4Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869725-HT6CLONEDHUMAN3H-LSDN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzamide221Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869735-HT7CLONEDHUMAN3H-5-CTN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzamide99Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869745-HT7CLONEDHUMAN3H-5-CTN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) benzenesulfonamide37Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869755-HT6CLONEDHUMAN3H-LSDN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) benzenesulfonamide317Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869765-HT2ACLONEDHUMAN3H-KETANSERINN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) benzenesulfonamide15Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869775-HT1ACLONEDHUMAN3H-8-OH-DPATN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) benzenesulfonamide8Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86978D2CLONEDHUMAN3H-RACLOPRIDEN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) benzenesulfonamide31Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86979D2CLONEDHUMAN3H-RACLOPRIDEN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-1-sulfonamide31Zareba P et al 2020Jan 15, 2025Jan 28, 2025
869805-HT1ACLONEDHUMAN3H-8-OH-DPATN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-1-sulfonamide39Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869815-HT2ACLONEDHUMAN3H-KETANSERINN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-1-sulfonamide63Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869825-HT6CLONEDHUMAN3H-LSDN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-1-sulfonamide52Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869835-HT7CLONEDHUMAN3H-5-CTN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-1-sulfonamide30Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869845-HT7CLONEDHUMAN3H-5-CTN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-2-sulfonamide31Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869855-HT6CLONEDHUMAN3H-LSDN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-2-sulfonamide57Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869865-HT2ACLONEDHUMAN3H-KETANSERINN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-2-sulfonamide44Zareba P et al 2020Jan 15, 2025Jan 15, 2025
869875-HT1ACLONEDHUMAN3H-8-OH-DPATN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-2-sulfonamide73Zareba P et al 2020Jan 15, 2025Jan 15, 2025
86988D2CLONEDHUMAN3H-RACLOPRIDEN-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl) naphthalene-2-sulfonamide27Zareba P et al 2020Jan 15, 2025Jan 28, 2025
86989D2STRIATUMRAT3H-SPIPERONE9-(3-(4-Phenylpiperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1764.8Cao X et al 2018Jan 15, 2025Jan 28, 2025
869905-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-Phenylpiperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1856.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
869915-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-Phenylpiperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one752.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
869925-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(Pyridin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one675.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
869935-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(Pyridin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1656.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
86994D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(Pyridin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1660.8Cao X et al 2018Jan 15, 2025Jan 28, 2025
86995D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(Pyrimidin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one2000Cao X et al 2018Jan 15, 2025Jan 28, 2025
869965-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(Pyrimidin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1965Cao X et al 2018Jan 15, 2025Jan 15, 2025
869975-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(Pyrimidin-2-yl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one557.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
869985-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one178.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
869995-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one964.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
87000D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(2-Methoxyphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one2000Cao X et al 2018Jan 15, 2025Jan 28, 2025
87001D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1852.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
870025-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one196.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
870035-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one207.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
870045-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one720.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
870055-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1628.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
87006D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one2000Cao X et al 2018Jan 15, 2025Jan 28, 2025
87007D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one1217.6Cao X et al 2018Jan 15, 2025Jan 28, 2025
870085-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one268.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
870095-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one207.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
870105-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one72Cao X et al 2018Jan 15, 2025Jan 15, 2025
870115-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one128.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
87012D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one182.1Cao X et al 2018Jan 15, 2025Jan 28, 2025
87013D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(Benzo[d]thiazol-2-yl)piperidin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one861.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
870145-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(Benzo[d]thiazol-2-yl)piperidin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one392Cao X et al 2018Jan 15, 2025Jan 15, 2025
870155-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(Benzo[d]thiazol-2-yl)piperidin-1-yl)propanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one173Cao X et al 2018Jan 15, 2025Jan 15, 2025
870165-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- propanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one52.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
870175-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- propanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one62.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
87018D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- propanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one58.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
87019D2STRIATUMRAT3H-SPIPERONERISPERIDONE3.7Cao X et al 2018Jan 15, 2025Jan 28, 2025
870205-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATRISPERIDONE181.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870215-HT2ACEREBRAL CORTEXRAT3H-KETANSERINRISPERIDONE0.18Cao X et al 2018Jan 15, 2025Jan 15, 2025
870225-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(2,3-Dimethylphenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one58.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870235-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(2,3-Dimethylphenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one169.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
87024D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(2,3-Dimethylphenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one185.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
87025D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one282.5Cao X et al 2018Jan 15, 2025Jan 28, 2025
870265-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one149.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
870275-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one79.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
870285-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one87.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870295-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one152.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
87030D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one91.4Cao X et al 2018Jan 15, 2025Jan 28, 2025
87031D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one18.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
870325-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one32.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870335-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one22.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
870345-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl)butanoyl)-1-methyl-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one32.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
870355-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl)butanoyl)-1-methyl-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one42.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
87036D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl)butanoyl)-1-methyl-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one62.1Cao X et al 2018Jan 15, 2025Jan 28, 2025
87037D2STRIATUMRAT3H-SPIPERONE9-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one31.8Cao X et al 2018Jan 15, 2025Jan 28, 2025
870385-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one32.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
870395-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one19.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
870405-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one765.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
870415-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one2000Cao X et al 2018Jan 15, 2025Jan 15, 2025
87042D2STRIATUMRAT3H-SPIPERONE9-(2-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)acetyl)- 1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one900.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
87043D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one44.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
870445-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one58.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
870455-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one73.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870465-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one186.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
870475-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one196.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
87048D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)piperidin-1-yl) propyl)-1,2,6,7-tetrahydropyrido[3,2,1- ij]quinolin-3(5H)-one582.1Cao X et al 2018Jan 15, 2025Jan 28, 2025
87049D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one394.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
870505-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one193.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870515-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one97.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
870525-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on83.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870535-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on98Cao X et al 2018Jan 15, 2025Jan 15, 2025
87054D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)-1,2,6,7- tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-on154.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
87055D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one74.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
870565-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one69.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
870575-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)- 1,2,6,7-tetrahydro pyrido[3,2,1-ij]quinolin-3(5H)-one59.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
870585-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one83.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
870595-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one82.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
87060D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-1- methyl-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one85.8Cao X et al 2018Jan 15, 2025Jan 28, 2025
87061D2STRIATUMRAT3H-SPIPERONE9-(3-(4-(6-fluoro benzo[d]isoxazol-3-yl)piperidin-1-yl)- 1-hydroxypropyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one28.4Cao X et al 2018Jan 15, 2025Jan 28, 2025
870625-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(3-(4-(6-fluoro benzo[d]isoxazol-3-yl)piperidin-1-yl)- 1-hydroxypropyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one19.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
870635-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(3-(4-(6-fluoro benzo[d]isoxazol-3-yl)piperidin-1-yl)- 1-hydroxypropyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one19.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870645-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one24.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
870655-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one79.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
87066D2STRIATUMRAT3H-SPIPERONE9-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-1,2,6,7-tetrahydropyrido[3,2,1-ij]quinolin-3(5H)-one29.7Cao X et al 2018Jan 15, 2025Jan 28, 2025
87067D2STRIATUMRAT3H-SPIPERONE8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one188.8Cao X et al 2018Jan 15, 2025Jan 28, 2025
870685-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one84.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
870695-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one174.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870705-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one92.5Cao X et al 2018Jan 15, 2025Jan 15, 2025
870715-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one81.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
87072D2STRIATUMRAT3H-SPIPERONE8-(3-(4-(2,3-Dichlorophenyl)piperazin-1-yl)propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one187.6Cao X et al 2018Jan 15, 2025Jan 28, 2025
87073D2STRIATUMRAT3H-SPIPERONE3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile574.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
870745-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile473.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870755-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN3-Fluoro-4-(4-(3-oxo-3-(4-oxo-2,4,5,6-tetrahydro-1H-pyrrolo- [3,2,1-ij]quinolin-8-yl)propyl)piperazin-1-yl)benzonitrile387.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
870765-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one68.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
870775-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one54.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
87078D2STRIATUMRAT3H-SPIPERONE8-(3-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)propanoyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one88.8Cao X et al 2018Jan 15, 2025Jan 28, 2025
87079D2STRIATUMRAT3H-SPIPERONE8-(3-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- propanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one19.7Cao X et al 2018Jan 15, 2025Jan 28, 2025
87080D2STRIATUMRAT3H-SPIPERONE8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one104.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
870815-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one53.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870825-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one37.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
870835-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one50.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
870845-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one31.8Cao X et al 2018Jan 15, 2025Jan 15, 2025
87085D2STRIATUMRAT3H-SPIPERONE8-(4-(4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one49.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
87086D2STRIATUMRAT3H-SPIPERONE8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one10.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
870875-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one12Cao X et al 2018Jan 15, 2025Jan 15, 2025
870885-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one9.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870895-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN7-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one17.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870905-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT7-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one25.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
87091D2STRIATUMRAT3H-SPIPERONE7-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one19.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
87092D2STRIATUMRAT3H-SPIPERONE9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one18.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
870935-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one19.1Cao X et al 2018Jan 15, 2025Jan 15, 2025
870945-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN9-Fluoro-8-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- butanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one21.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
870955-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one0.72Cao X et al 2018Jan 15, 2025Jan 15, 2025
870965-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one8.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
87097D2STRIATUMRAT3H-SPIPERONE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one2.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
87098D2STRIATUMRAT3H-SPIPERONE8-(6-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)hexanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one89.1Cao X et al 2018Jan 15, 2025Jan 28, 2025
870995-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(6-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)hexanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one168.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
871005-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(6-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)hexanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one34.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
871015-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(3-(4-(6-Fuorobenzo[d]isoxazol-3-yl)- piperidin-1-yl) propyl)-5,6-dihydro-1H-pyrrolo [3,2,1-ij]quinolin4(2H)-one29.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
871025-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(6-Fuorobenzo[d]isoxazol-3-yl)- piperidin-1-yl) propyl)-5,6-dihydro-1H-pyrrolo [3,2,1-ij]quinolin4(2H)-one38.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
87103D2STRIATUMRAT3H-SPIPERONE8-(3-(4-(6-Fuorobenzo[d]isoxazol-3-yl)- piperidin-1-yl) propyl)-5,6-dihydro-1H-pyrrolo [3,2,1-ij]quinolin4(2H)-one46.5Cao X et al 2018Jan 15, 2025Jan 28, 2025
87104D2STRIATUMRAT3H-SPIPERONE8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one9.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
871055-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one11.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
871065-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one19.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
871075-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(5-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)pentyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one58.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
871085-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(5-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)pentyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one54Cao X et al 2018Jan 15, 2025Jan 15, 2025
87109D2STRIATUMRAT3H-SPIPERONE8-(5-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)pentyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one43.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
87110D2STRIATUMRAT3H-SPIPERONE8-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)pperidin-1-yl)-1-hydroxypropyl)-5,6-dihydro-1Hpyrrolo[3,2,1-ij]quinolin-4(2H)-one19.6Cao X et al 2018Jan 15, 2025Jan 28, 2025
871115-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)pperidin-1-yl)-1-hydroxypropyl)-5,6-dihydro-1Hpyrrolo[3,2,1-ij]quinolin-4(2H)-one29.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
871125-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(3-(4-(6-fluorobenzo[d]- isoxazol-3-yl)pperidin-1-yl)-1-hydroxypropyl)-5,6-dihydro-1Hpyrrolo[3,2,1-ij]quinolin-4(2H)-one59.6Cao X et al 2018Jan 15, 2025Jan 15, 2025
871135-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one69.5Cao X et al 2018Jan 15, 2025Jan 15, 2025
871145-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one22.5Cao X et al 2018Jan 15, 2025Jan 15, 2025
87115D2STRIATUMRAT3H-SPIPERONE8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one13.4Cao X et al 2018Jan 15, 2025Jan 28, 2025
87116D2STRIATUMRAT3H-SPIPERONE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one8.4Cao X et al 2018Jan 15, 2025Jan 28, 2025
871175-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPAT8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one12Cao X et al 2018Jan 15, 2025Jan 15, 2025
871185-HT2ACEREBRAL CORTEXRAT3H-KETANSERIN8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one0.4Cao X et al 2018Jan 15, 2025Jan 15, 2025
871195-HT2CCEREBRAL CORTEXRAT3H-MESULERGINE8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one610.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
87120H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one421Cao X et al 2018Jan 15, 2025Jan 28, 2025
87121CEREBRAL CORTEXRAT3H-PRAZOSIN8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one491.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
871225-HT6CLONEDHUMAN3H-LSD8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one241Cao X et al 2018Jan 15, 2025Jan 15, 2025
87123D3olfactory tubercleRAT3H-7-OH-DPAT8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butanoyl)- 5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one61.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
87124D3olfactory tubercleRAT3H-7-OH-DPAT8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1.66Cao X et al 2018Jan 15, 2025Jan 28, 2025
871255-HT6CLONEDHUMAN3H-LSD8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one5.55Cao X et al 2018Jan 15, 2025Jan 15, 2025
87126CEREBRAL CORTEXRAT3H-PRAZOSIN8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one431Cao X et al 2018Jan 15, 2025Jan 15, 2025
87127H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one630.3Cao X et al 2018Jan 15, 2025Jan 28, 2025
871285-HT2CCEREBRAL CORTEXRAT3H-MESULERGINE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one616Cao X et al 2018Jan 15, 2025Jan 15, 2025
871295-HT2CCEREBRAL CORTEXRAT3H-MESULERGINE8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one539.9Cao X et al 2018Jan 15, 2025Jan 15, 2025
87130H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one711.7Cao X et al 2018Jan 15, 2025Jan 28, 2025
87131CEREBRAL CORTEXRAT3H-PRAZOSIN8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one99.3Cao X et al 2018Jan 15, 2025Jan 15, 2025
871325-HT6CLONEDHUMAN3H-LSD8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one17.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
87133D3olfactory tubercleRAT3H-7-OH-DPAT8-(4-(4-(6-Fuorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butyl)-5,6- dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one54.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
87134D3olfactory tubercleRAT3H-7-OH-DPAT8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one45.37Cao X et al 2018Jan 15, 2025Jan 28, 2025
871355-HT6CLONEDHUMAN3H-LSD8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one6.36Cao X et al 2018Jan 15, 2025Jan 15, 2025
87136CEREBRAL CORTEXRAT3H-PRAZOSIN8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one339Cao X et al 2018Jan 15, 2025Jan 15, 2025
87137H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one339Cao X et al 2018Jan 15, 2025Jan 28, 2025
871385-HT2CCEREBRAL CORTEXRAT3H-MESULERGINE8-(4-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxybutyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one742Cao X et al 2018Jan 15, 2025Jan 15, 2025
871395-HT2CCEREBRAL CORTEXRAT3H-MESULERGINE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one33.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
87140H1CEREBELLUMGUINEA PIG3H-MEPYRAMINE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one43.5Cao X et al 2018Jan 15, 2025Jan 28, 2025
87141CEREBRAL CORTEXRAT3H-PRAZOSIN8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one596Cao X et al 2018Jan 15, 2025Jan 15, 2025
871425-HT6CLONEDHUMAN3H-LSD8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one29.46Cao X et al 2018Jan 15, 2025Jan 15, 2025
87143D3olfactory tubercleRAT3H-7-OH-DPAT8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-1-hydroxypentyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one116.32Cao X et al 2018Jan 15, 2025Jan 28, 2025
87144D3olfactory tubercleRAT3H-7-OH-DPATRISPERIDONE31.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
871455-HT6CLONEDHUMAN3H-LSDRISPERIDONE1260Cao X et al 2018Jan 15, 2025Jan 15, 2025
87146CEREBRAL CORTEXRAT3H-PRAZOSINRISPERIDONE54.7Cao X et al 2018Jan 15, 2025Jan 15, 2025
87147H1CEREBELLUMGUINEA PIG3H-MEPYRAMINERISPERIDONE46.2Cao X et al 2018Jan 15, 2025Jan 28, 2025
871485-HT2CCEREBRAL CORTEXRAT3H-MESULERGINERISPERIDONE28.2Cao X et al 2018Jan 15, 2025Jan 15, 2025
87149D1STRIATUMRAT3H-SCH233908-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one76.9Cao X et al 2018Jan 15, 2025Jan 28, 2025
871505-HT7CEREBRAL CORTEXRAT3H-5-CT8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one226Cao X et al 2018Jan 15, 2025Jan 15, 2025
87151H3CEREBRAL CORTEXRAT3H-methylhistamine8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 28, 2025
87152CEREBRAL CORTEXRAT3H-RAUWOLSCINE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 15, 2025
87153SERTCEREBRAL CORTEXRAT3H-PAROXETINE8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 28, 2025
87154NETHIPPOCAMPUSRAT3H-Nisoxetine8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 15, 2025
87155DATSTRIATUMRAT3H-WIN354288-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 15, 2025
87156Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 15, 2025
87157Sigma 2BRAINGUINEA PIG3H-DTG8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 15, 2025
87158NMDAHIPPOCAMPUSRAT3H-Glycine8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 28, 2025
87159M1CLONEDHUMAN3H-QNB8-(5-(4-(6-Fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)- pentanoyl)-5,6-dihydro-1H-pyrrolo[3,2,1-ij]quinolin-4(2H)-one1000Cao X et al 2018Jan 15, 2025Jan 15, 2025
871605-HT2AHippocampalRAT3H-KETANSERIN[2-(4-Phenylpiperazin-1-yl)ethyl]pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871615-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871625-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one78Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871635-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one55Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871645-HT2AHippocampalRAT3H-KETANSERIN3-{2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871655-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871665-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871675-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one42Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871685-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871695-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(3-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871705-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871715-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871725-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871735-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(2-Fluorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871745-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871755-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(4-Fluorophenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871765-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Methylphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one514Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871775-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(2-Methylphenyl)piperazin-1-yl]ethyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871785-HT1AHippocampalRAT3H-8-OH-DPAT3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)pyr-imido[5,4-c]equinolin-4(3H)-one160Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871795-HT2AHippocampalRAT3H- Ketanserin3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)pyr-imido[5,4-c]equinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871805-HT1AHippocampalRAT3H-8-OH-DPAT3-[2-(4-Pyrimidin-2-ylpiperazin-1-yl)ethyl]pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871815-HT2AHippocampalRAT3H- Ketanserin3-[2-(4-Pyrimidin-2-ylpiperazin-1-yl)ethyl]pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871825-HT1AHippocampalRAT3H-8-OH-DPAT3-[3-(4-Phenylpiperazin-1-yl)propyl]pyrimido[5,4-c]quino-lin-4(3H)-one47Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871835-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(2-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one93Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871845-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(2-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871855-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one80Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871865-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(4-Chlorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871875-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one20Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871885-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871895-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(3-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one120Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871905-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(3-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871915-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(4-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871925-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(4-Methoxyphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871935-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one55Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871945-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871955-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(4-Fluorophenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one129Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871965-HT2AHippocampalRAT3H-KETANSERIN3-{3-[4-(2-Methylphenyl)piperazin-1-yl]propyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871975-HT1AHippocampalRAT3H-8-OH-DPAT3-(3-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}propyl)pyrimido[5,4-c]quinolin-4(3H)-one243Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871985-HT2AHippocampalRAT3H- Ketanserin3-(3-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}propyl)pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
871995-HT1AHippocampalRAT3H-8-OH-DPAT3-[3-(4-Pyrimidin-2-ylpiperazin-1-yl)propyl]pyrimido[5,4-c]quinolin-4(3H)-one48Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872005-HT2AHippocampalRAT3H- Ketanserin3-[3-(4-Pyrimidin-2-ylpiperazin-1-yl)propyl]pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872015-HT1AHippocampalRAT3H-8-OH-DPAT3-[4-(4-Phenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quino-lin-4(3H)-one28Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872025-HT7HEK293 cellsHUMAN3H-5CT3-[4-(4-Phenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quino-lin-4(3H)-one612Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872035-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one17Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872045-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(2-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one153Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872055-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one34Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872065-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one184Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872075-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(4-Chlorophenylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one328Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872085-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one6Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872095-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one276Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872105-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one31Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872115-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one484Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872125-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(4-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872135-HT2AHippocampalRAT3H- Ketanserin3-{4-[4-(4-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872145-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(4-Methoxyphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one>10000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872155-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one63Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872165-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one739Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872175-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one404Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872185-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Methylphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one52Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872195-HT7HEK293 cellsHUMAN3H-5CT3-{4-[4-(2-Methylphenyl)piperazin-1-yl]butyl}pyrimido[5,4-c]quinolin-4(3H)-one296Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872205-HT1AHippocampalRAT3H-8-OH-DPAT3-(4-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}butyl)pyrimido[5,4-c]quinolin-4(3H)-one127Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872215-HT7HEK293 cellsHUMAN3H-5CT3-(4-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}butyl)pyrimido[5,4-c]quinolin-4(3H)-one418Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872225-HT2AHippocampalRAT3H- Ketanserin3-[4-(4-Pyrimidin-2-ylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872235-HT7HEK293 cellsHUMAN3H-5CT3-[4-(4-Pyrimidin-2-ylpiperazin-1-yl)butyl]pyrimido[5,4-c]quinolin-4(3H)-one5800Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872245-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one14Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872255-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872265-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}-8-methylpyr-imido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872275-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}-8-methylpyr-imido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872285-HT1AHippocampalRAT3H-8-OH-DPAT3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)-8-methylpyrimido[5,4-c]quinolin-4(3H)-one241Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872295-HT2AHippocampalRAT3H- Ketanserin3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)-8-methylpyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872305-HT1AHippocampalRAT3H-8-OH-DPAT3-[3-(4-Phenylpiperazin-1-yl)propyl]-8-methylpyrimido[5,4-c]quinolin-4(3H)-one125Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872315-HT2AHippocampalRAT3H- Ketanserin3-[3-(4-Phenylpiperazin-1-yl)propyl]-8-methylpyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872325-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872335-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8-meth-ylpyrimido[5,4-c]-quinolin-4(3H)-one31Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872345-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8-meth-ylpyrimido[5,4-c]-quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872355-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(4-Fluorophenyl)piperazin-1-yl]propyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872365-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]-8-methylpyr-imido[5,4-c]quinolin-4(3H)-one172Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872375-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one20Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872385-HT2AHippocampalRAT3H- Ketanserin3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872395-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one83Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872405-HT2AHippocampalRAT3H- Ketanserin3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}-8-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872415-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one82Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872425-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(2-Methoxyphenyl)piperazin-1-yl]ethyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872435-HT1AHippocampalRAT3H-8-OH-DPAT3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872445-HT2AHippocampalRAT3H- Ketanserin3-{2-[4-(4-Methoxyphenyl)piperazin-1-yl]ethyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872455-HT2AHippocampalRAT3H- Ketanserin3-(2-{4-[3-(Trifluoromethyl)phenyl]piperazin-1-yl}ethyl)-9-methylpyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872465-HT1AHippocampalRAT3H-8-OH-DPAT3-[3-(4-Phenylpiperazin-1-yl)propyl]-9-methylpyrimido[5,4-c]quinolin-4(3H)-one128Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872475-HT2AHippocampalRAT3H- Ketanserin3-[3-(4-Phenylpiperazin-1-yl)propyl]-9-methylpyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872485-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872495-HT1AHippocampalRAT3H-8-OH-DPAT3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-9-meth-ylpyrimido[5,4-c]-quinolin-4(3H)-one26Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872505-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-9-meth-ylpyrimido[5,4-c]-quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872515-HT2AHippocampalRAT3H- Ketanserin3-{3-[4-(4-Fluorophenyl)piperazin-1-yl]propyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872525-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(3-Chlorophenylpiperazin-1-yl)butyl]-9-methylpyr-imido[5,4-c]quinolin-4(3H)-one67Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872535-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one8Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872545-HT2AHippocampalRAT3H- Ketanserin3-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872555-HT1AHippocampalRAT3H-8-OH-DPAT3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one97Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
872565-HT2AHippocampalRAT3H- Ketanserin3-{4-[4-(2-Fluorophenyl)piperazin-1-yl]butyl}-9-methyl-pyrimido[5,4-c]quinolin-4(3H)-one1000Lewgowd W et al 2011Jan 15, 2025Jan 15, 2025
87257CEREBRAL CORTEXRAT3H-PRAZOSIN(R)-3-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide241Rak A et al 2016Jan 15, 2025Jan 15, 2025
87258CEREBRAL CORTEXRAT3H-CLONIDINE(R)-3-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide1944Rak A et al 2016Jan 15, 2025Jan 15, 2025
87259CEREBRAL CORTEXRAT3H-CLONIDINE(S)-3-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide>10000Rak A et al 2016Jan 15, 2025Jan 15, 2025
87260CEREBRAL CORTEXRAT3H-PRAZOSIN(S)-3-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide348Rak A et al 2016Jan 15, 2025Jan 15, 2025
87261CEREBRAL CORTEXRAT3H-PRAZOSIN(R)-5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide289Rak A et al 2016Jan 15, 2025Jan 15, 2025
87262CEREBRAL CORTEXRAT3H-CLONIDINE(R)-5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide2354Rak A et al 2016Jan 15, 2025Jan 15, 2025
87263CEREBRAL CORTEXRAT3H-CLONIDINE(S)-5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide>10000Rak A et al 2016Jan 15, 2025Jan 15, 2025
87264CEREBRAL CORTEXRAT3H-PRAZOSIN(S)-5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide214Rak A et al 2016Jan 15, 2025Jan 15, 2025
87265CEREBRAL CORTEXRAT3H-PRAZOSIN(R)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide176Rak A et al 2016Jan 15, 2025Jan 15, 2025
87266CEREBRAL CORTEXRAT3H-CLONIDINE(R)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide378Rak A et al 2016Jan 15, 2025Jan 15, 2025
87267CEREBRAL CORTEXRAT3H-CLONIDINE(S)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide>10000Rak A et al 2016Jan 15, 2025Jan 15, 2025
87268CEREBRAL CORTEXRAT3H-PRAZOSIN(R)-5-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide106Rak A et al 2016Jan 15, 2025Jan 15, 2025
87269CEREBRAL CORTEXRAT3H-CLONIDINE(R)-5-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide398Rak A et al 2016Jan 15, 2025Jan 15, 2025
87270CEREBRAL CORTEXRAT3H-PRAZOSIN(S)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide92Rak A et al 2016Jan 15, 2025Jan 15, 2025
87271CEREBRAL CORTEXRAT3H-PRAZOSIN(S)-3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]pyrrolidin-3-yl}benzenesulfonamide242Rak A et al 2016Jan 15, 2025Jan 15, 2025
87272CEREBRAL CORTEXRAT3H-CLONIDINE3-Chloro-N-{[1-(2-(2-methoxyphenoxy)ethyl)piperidin4-yl]methyl}benzenesulfonamide439Rak A et al 2016Jan 15, 2025Jan 15, 2025
87273CEREBRAL CORTEXRAT3H-PRAZOSIN3-Chloro-N-{[1-(2-(2-methoxyphenoxy)ethyl)piperidin4-yl]methyl}benzenesulfonamide46Rak A et al 2016Jan 15, 2025Jan 15, 2025
87274CEREBRAL CORTEXRAT3H-PRAZOSIN5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide34Rak A et al 2016Jan 15, 2025Jan 15, 2025
87275CEREBRAL CORTEXRAT3H-CLONIDINE5-Chloro-2-fluoro-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide129Rak A et al 2016Jan 15, 2025Jan 15, 2025
87276CEREBRAL CORTEXRAT3H-CLONIDINE3,4-Dimethoxy-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide2140Rak A et al 2016Jan 15, 2025Jan 15, 2025
87277CEREBRAL CORTEXRAT3H-PRAZOSIN3,4-Dimethoxy-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide99Rak A et al 2016Jan 15, 2025Jan 15, 2025
87278CEREBRAL CORTEXRAT3H-PRAZOSINN-(1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl) quinoline-8-sulfonamide93Rak A et al 2016Jan 15, 2025Jan 15, 2025
87279CEREBRAL CORTEXRAT3H-CLONIDINEN-(1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl) quinoline-8-sulfonamide131Rak A et al 2016Jan 15, 2025Jan 15, 2025
87280CEREBRAL CORTEXRAT3H-CLONIDINEN-{1-[2-(2-Methoxyphenoxy)ethyl]piperidin-4-yl}isoquinoline-4-sulfonamide297Rak A et al 2016Jan 15, 2025Jan 15, 2025
87281CEREBRAL CORTEXRAT3H-PRAZOSINN-{1-[2-(2-Methoxyphenoxy)ethyl]piperidin-4-yl}isoquinoline-4-sulfonamide52Rak A et al 2016Jan 15, 2025Jan 15, 2025
87282CEREBRAL CORTEXRAT3H-PRAZOSIN3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]piperidin-4-yl}benzenesulfonamide131Rak A et al 2016Jan 15, 2025Jan 15, 2025
87283CEREBRAL CORTEXRAT3H-CLONIDINE3-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]piperidin-4-yl}benzenesulfonamide188Rak A et al 2016Jan 15, 2025Jan 15, 2025
87284CEREBRAL CORTEXRAT3H-CLONIDINE5-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]piperidin-4-yl}benzenesulfonamide293Rak A et al 2016Jan 15, 2025Jan 15, 2025
87285CEREBRAL CORTEXRAT3H-PRAZOSIN5-Chloro-2-fluoro-N-{1-[2-(2-isopropoxyphenoxy) ethyl]piperidin-4-yl}benzenesulfonamide118Rak A et al 2016Jan 15, 2025Jan 15, 2025
87286CEREBRAL CORTEXRAT3H-PRAZOSINN-{1-[2-(2-Isopropoxyphenoxy)ethyl]piperidin-4-yl} quinoline-8-sulfonamide73Rak A et al 2016Jan 15, 2025Jan 15, 2025
87287CEREBRAL CORTEXRAT3H-CLONIDINEN-{1-[2-(2-Isopropoxyphenoxy)ethyl]piperidin-4-yl} quinoline-8-sulfonamide194Rak A et al 2016Jan 15, 2025Jan 15, 2025
87288CEREBRAL CORTEXRAT3H-CLONIDINE3-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide678Rak A et al 2016Jan 15, 2025Jan 15, 2025
87289CEREBRAL CORTEXRAT3H-PRAZOSIN3-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide48Rak A et al 2016Jan 15, 2025Jan 15, 2025
87290CEREBRAL CORTEXRAT3H-PRAZOSIN5-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide56Rak A et al 2016Jan 15, 2025Jan 15, 2025
87291CEREBRAL CORTEXRAT3H-CLONIDINE5-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide1345Rak A et al 2016Jan 15, 2025Jan 15, 2025
87292CEREBRAL CORTEXRAT3H-CLONIDINE3,4-Dimethoxy-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide644Rak A et al 2016Jan 15, 2025Jan 15, 2025
87293CEREBRAL CORTEXRAT3H-PRAZOSIN3,4-Dimethoxy-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide81Rak A et al 2016Jan 15, 2025Jan 15, 2025
87294CEREBRAL CORTEXRAT3H-PRAZOSINN-{[1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl] methyl}isoquinoline-4-sulfonamide90Rak A et al 2016Jan 15, 2025Jan 15, 2025
87295CEREBRAL CORTEXRAT3H-CLONIDINEN-{[1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl] methyl}isoquinoline-4-sulfonamide695Rak A et al 2016Jan 15, 2025Jan 15, 2025
87296CEREBRAL CORTEXRAT3H-CLONIDINE4-Fluoro-N-{[1-(2-(2-isopropoxyphenoxy)ethyl)piperidin-4-yl]methyl}benzenesulfonamide416Rak A et al 2016Jan 15, 2025Jan 15, 2025
87297CEREBRAL CORTEXRAT3H-PRAZOSIN4-Fluoro-N-{[1-(2-(2-isopropoxyphenoxy)ethyl)piperidin-4-yl]methyl}benzenesulfonamide77Rak A et al 2016Jan 15, 2025Jan 15, 2025
87298CEREBRAL CORTEXRAT3H-PRAZOSIN3-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide71Rak A et al 2016Jan 15, 2025Jan 15, 2025
87299CEREBRAL CORTEXRAT3H-CLONIDINE3-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide1212Rak A et al 2016Jan 15, 2025Jan 15, 2025
87300CEREBRAL CORTEXRAT3H-CLONIDINE5-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide870Rak A et al 2016Jan 15, 2025Jan 15, 2025
87301CEREBRAL CORTEXRAT3H-PRAZOSIN5-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide133Rak A et al 2016Jan 15, 2025Jan 15, 2025
87302CEREBRAL CORTEXRAT3H-PRAZOSINN-{[1-(2-(2-Isopropoxyphenoxy)ethyl)piperidin-4-yl] methyl}quinoline-8-sulfonamide95Rak A et al 2016Jan 15, 2025Jan 15, 2025
87303CEREBRAL CORTEXRAT3H-CLONIDINEN-{[1-(2-(2-Isopropoxyphenoxy)ethyl)piperidin-4-yl] methyl}quinoline-8-sulfonamide947Rak A et al 2016Jan 15, 2025Jan 15, 2025
87304CEREBRAL CORTEXRAT3H-CLONIDINEN-{1-[2-(2-Isopropoxyphenoxy)ethyl]pyrrolidin-3-yl} isoquinoline-4-sulfonamide578Rak A et al 2016Jan 15, 2025Jan 15, 2025
87305CEREBRAL CORTEXRAT3H-PRAZOSINN-{1-[2-(2-Isopropoxyphenoxy)ethyl]pyrrolidin-3-yl} isoquinoline-4-sulfonamide67Rak A et al 2016Jan 15, 2025Jan 15, 2025
87306Alpha1AplaceholderHUMANPlaceholder3-Chloro-N-{[1-(2-(2-methoxyphenoxy)ethyl)piperidin4-yl]methyl}benzenesulfonamide120.6Rak A et al 2016Jan 15, 2025Jan 28, 2025
87307Alpha1AplaceholderHUMANPlaceholder3,4-Dimethoxy-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide191.6Rak A et al 2016Jan 15, 2025Jan 28, 2025
87308Alpha1BplaceholderHUMANPlaceholder3,4-Dimethoxy-N-{1-[2-(2-methoxyphenoxy)ethyl] piperidin-4-yl}benzenesulfonamide461.1Rak A et al 2016Jan 15, 2025Jan 28, 2025
87309Alpha1BplaceholderHUMANPlaceholderN-{1-[2-(2-Methoxyphenoxy)ethyl]piperidin-4-yl}isoquinoline-4-sulfonamide608.4Rak A et al 2016Jan 15, 2025Jan 28, 2025
87310Alpha1AplaceholderHUMANPlaceholderN-{1-[2-(2-Methoxyphenoxy)ethyl]piperidin-4-yl}isoquinoline-4-sulfonamide99.7Rak A et al 2016Jan 15, 2025Jan 28, 2025
87311Alpha1AplaceholderHUMANPlaceholder3-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide84.2Rak A et al 2016Jan 15, 2025Jan 28, 2025
87312Alpha1BplaceholderHUMANPlaceholder3-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide14.15Rak A et al 2016Jan 15, 2025Jan 28, 2025
87313Alpha1BplaceholderHUMANPlaceholder5-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide12.65Rak A et al 2016Jan 15, 2025Jan 28, 2025
87314Alpha1AplaceholderHUMANPlaceholder5-Chloro-2-fluoro-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide148.2Rak A et al 2016Jan 15, 2025Jan 28, 2025
87315Alpha1AplaceholderHUMANPlaceholder3,4-Dimethoxy-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide160.7Rak A et al 2016Jan 15, 2025Jan 28, 2025
87316Alpha1BplaceholderHUMANPlaceholder3,4-Dimethoxy-N-{[1-(2-(2-methoxyphenoxy)ethyl) piperidin-4-yl]methyl}benzenesulfonamide598.6Rak A et al 2016Jan 15, 2025Jan 28, 2025
87317Alpha1BplaceholderHUMANPlaceholderN-{[1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl] methyl}isoquinoline-4-sulfonamide514.8Rak A et al 2016Jan 15, 2025Jan 28, 2025
87318Alpha1AplaceholderHUMANPlaceholderN-{[1-(2-(2-Methoxyphenoxy)ethyl)piperidin-4-yl] methyl}isoquinoline-4-sulfonamide140.1Rak A et al 2016Jan 15, 2025Jan 28, 2025
87319Alpha1AplaceholderHUMANPlaceholder3-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide11.1Rak A et al 2016Jan 15, 2025Jan 28, 2025
87320Alpha1BplaceholderHUMANPlaceholder3-Chloro-2-fluoro-N-{[1-(2-(2-isopropoxyphenoxy) ethyl)piperidin-4-yl]methyl}benzenesulfonamide42.1Rak A et al 2016Jan 15, 2025Jan 28, 2025
87321Alpha1BplaceholderHUMANPlaceholderN-{[1-(2-(2-Isopropoxyphenoxy)ethyl)piperidin-4-yl] methyl}quinoline-8-sulfonamide104.8Rak A et al 2016Jan 15, 2025Jan 28, 2025
87322Alpha1AplaceholderHUMANPlaceholderN-{[1-(2-(2-Isopropoxyphenoxy)ethyl)piperidin-4-yl] methyl}quinoline-8-sulfonamide34.1Rak A et al 2016Jan 15, 2025Jan 28, 2025
87323Alpha1AplaceholderHUMANPlaceholderTamsulosin0.07Rak A et al 2016Jan 15, 2025Jan 28, 2025
87324Alpha1BplaceholderHUMANPlaceholderTamsulosin0.13Rak A et al 2016Jan 15, 2025Jan 28, 2025
87325Alpha1BplaceholderHUMANPlaceholderTerazosin1.73Rak A et al 2016Jan 15, 2025Jan 28, 2025
87326Alpha1AplaceholderHUMANPlaceholderTerazosin51.89Rak A et al 2016Jan 15, 2025Jan 28, 2025
87327Alpha1AplaceholderHUMANPlaceholderPhenylephrine,(+/-)55.99Rak A et al 2016Jan 15, 2025Jan 28, 2025
87328Alpha1BplaceholderHUMANPlaceholderPhenylephrine,(+/-)0.86Rak A et al 2016Jan 15, 2025Jan 28, 2025
87329Alpha1BplaceholderHUMANPlaceholder3-Chloro-N-{[1-(2-(2-methoxyphenoxy)ethyl)piperidin4-yl]methyl}benzenesulfonamide15.5Rak A et al 2016Jan 15, 2025Jan 28, 2025
87330Calcium channelUNDEFINEDUNDEFINEDUNDEFINEDxanomeline1660Thorn CA et al 2019Jan 15, 2025Jan 28, 2025
87331Calcium channelUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
87332Calcium channelUNDEFINEDUNDEFINEDUNDEFINEDxanomeline3180Thorn CA et al 2019Jan 15, 2025Jan 28, 2025
87333GABAAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
87334GABAAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
87335GABAAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87336AMPAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
87337NMDAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 28, 2025
87338NMDAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87339nAChRUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
87340nAChRUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
873415-HT3UNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87342UNDEFINEDUNDEFINEDUNDEFINEDxanomeline2710Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87343NETUNDEFINEDUNDEFINEDUNDEFINEDxanomeline1630Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87344DATUNDEFINEDUNDEFINEDUNDEFINEDxanomeline457Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87345SERTUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 28, 2025
87346UNDEFINEDUNDEFINEDUNDEFINEDxanomeline1390Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
87347GABAAUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 29, 2025
87348ARUNDEFINEDUNDEFINEDUNDEFINEDxanomeline>10000Thorn CA et al 2019Jan 15, 2025Jan 15, 2025
873495-HT2ACLONEDHUMAN3H-KETANSERIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide109Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873505-HT2BCLONEDHUMAN3H-LSD4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide380Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873515-HT2CCLONEDHUMAN3H-KETANSERIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide52Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873525-HT6CLONEDHUMAN3H-LSD4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide123Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87353BZPCORTICAL MEMBRANESRATFNZ4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide933Huang XP et al 2016Jan 15, 2025Jan 29, 2025
87354PBRKidney membranesRAT3H-PK111954-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide70Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87355A1CLONEDHUMAN3H-CCPA4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide3846Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87356Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide2818Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87357CB2CLONEDHUMAN3H-CP559404-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide8511Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87358V1ACLONEDHUMAN3H-VASOPRESSIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide3575Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87359hERGCLONEDHUMAN3H-Dofetilide4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide2042Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87360hERGCLONEDHUMAN3H-Dofetilide1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide1806Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87361V1ACLONEDHUMAN3H-VASOPRESSIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide3311Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87362CB2CLONEDHUMAN3H-CP559401-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide7470Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87363Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide2138Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87364A1CLONEDHUMAN3H-CCPA1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide5129Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87365PBRKidney membranesRAT3H-PK111951-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide77Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87366BZPCEREBRAL CORTEXRATFNZ1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide1023Huang XP et al 2016Jan 15, 2025Jan 29, 2025
873675-HT6CLONEDHUMAN3H-LSD1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide1008Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873685-HT2CCLONEDHUMAN3H-MESULERGINE1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide878Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873695-HT2BCLONEDHUMAN3H-LSD1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide2171Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873705-HT2ACLONEDHUMAN3H-KETANSERIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide1751Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873715-HT1ACLONEDHUMAN3H-WAY1006351-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873725-HT1BCLONEDHUMAN3H-5-CT1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873735-HT1DCLONEDHUMAN3H-5-CT1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873745-HT1ECLONEDHUMAN3H-5-HT1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873755-HT3CLONEDHUMAN3H-GR-656301-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873765-HT5ACLONEDHUMAN3H-LSD1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
873775-HT7CLONEDHUMAN3H-LSD1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87378A2ACLONEDHUMAN3H-NECA1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87379Alpha1ACLONEDHUMAN3H-PRAZOSIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87380Alpha1BCLONEDHUMAN3H-PRAZOSIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87381Alpha1DCLONEDHUMAN3H-PRAZOSIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87382Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87383Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87384Beta 1CLONEDHUMAN125I-Pindolol1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87385Beta3CLONEDHUMAN125I-Pindolol1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87386Beta 2CLONEDHUMAN3H-CGP121771-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87387D1CLONEDHUMAN3H-SCH233901-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87388D5CLONEDHUMAN3H-SCH233901-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87389D2CLONEDHUMAN3H-N-Methylspiperone1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87390D3CLONEDHUMAN3H-N-Methylspiperone1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87391D4CLONEDHUMAN3H-N-Methylspiperone1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87392DATCLONEDHUMAN3H-WIN 35,4281-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87393NETCLONEDHUMAN3H-Nisoxetine1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87394SERTCLONEDHUMAN3H-CITALOPRAM1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87395DORCLONEDHUMAN3H-DADLE1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87396MORCLONEDHUMAN3H-DAMGO1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87397KORCLONEDHUMAN3H-U695931-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87398KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 27, 2025
87399H1CLONEDHUMAN3H-PYRILAMINE1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
874005-HT1DCLONEDHUMAN125I-aminopotentidine1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87401H3CLONEDHUMAN3H-Alpha-methylhistamine1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87402H4CLONEDHUMAN3H-Histamine1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87403M1CLONEDHUMAN3H-QNB1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87404M2CLONEDHUMAN3H-QNB1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87405M3CLONEDHUMAN3H-QNB1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87406M4CLONEDHUMAN3H-QNB1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87407M5CLONEDHUMAN3H-QNB1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87408mGluR5CLONEDHUMAN3H-MPEP1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87409Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87410Sigma 2PC12RAT3H-DTG1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87411V1BCLONEDHUMAN3H-VASOPRESSIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87412V2CLONEDHUMAN3H-VASOPRESSIN1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87413OTCLONEDHUMAN3H-Oxytocin1-(4-Nitrophenylethyl)piperidylidene-2-(4-chlorophenyl)sulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87414OTCLONEDHUMAN3H-Oxytocin4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87415V2CLONEDHUMAN3H-VASOPRESSIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87416V1BCLONEDHUMAN3H-VASOPRESSIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87417Sigma 2PC12RAT3H-DTG4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87418Sigma 1CEREBRAL CORTEXGUINEA PIG3H-Pentazocine(+)4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87419mGluR5CLONEDHUMAN3H-MPEP4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87420M1CLONEDHUMAN3H-QNB4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87421M2CLONEDHUMAN3H-QNB4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87422M3CLONEDHUMAN3H-QNB4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87423M4CLONEDHUMAN3H-QNB4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87424M5CLONEDHUMAN3H-QNB4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87425H4CLONEDHUMAN3H-Histamine4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87426H3CLONEDHUMAN3H-Alpha-methylhistamine4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
874275-HT1DCLONEDHUMAN125I-aminopotentidine4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87428H1CLONEDHUMAN3H-PYRILAMINE4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87429KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 27, 2025
87430MORCLONEDHUMAN3H-DAMGO4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87431KORCLONEDHUMAN3H-U695934-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87432DORCLONEDHUMAN3H-DADLE4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87433SERTCLONEDHUMAN3H-CITALOPRAM4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87434NETCLONEDHUMAN3H-Nisoxetine4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87435DATCLONEDHUMAN3H-WIN 35,4284-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87436D5CLONEDHUMAN3H-SCH233904-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87437D1CLONEDHUMAN3H-SCH233904-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87438D2CLONEDHUMAN3H-N-Methylspiperone4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87439D3CLONEDHUMAN3H-N-Methylspiperone4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87440D4CLONEDHUMAN3H-N-Methylspiperone4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87441Beta3CLONEDHUMAN125I-Pindolol4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87442Beta 1CLONEDHUMAN125I-Pindolol4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87443Beta 2CLONEDHUMAN3H-CGP121774-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
87444Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87445Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87446Alpha1DCLONEDHUMAN3H-PRAZOSIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87447Alpha1BCLONEDHUMAN3H-PRAZOSIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87448Alpha1ACLONEDHUMAN3H-PRAZOSIN4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 28, 2025
87449Alpha2ACLONEDHUMAN3H-NECA4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 29, 2025
874505-HT7CLONEDHUMAN3H-LSD4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874515-HT5ACLONEDHUMAN3H-LSD4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874525-HT3CLONEDHUMAN3H-GR-656304-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874535-HT1ECLONEDHUMAN3H-5-HT4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874545-HT1DCLONEDHUMAN3H-5-CT4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874555-HT1BCLONEDHUMAN3H-5-CT4-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874565-HT1ACLONEDHUMAN3H-WAY1006354-chloro-N-[1-(2-phenylethyl)-2-piperidinylidene]-benzenesulfonamide>10000Huang XP et al 2016Jan 15, 2025Jan 15, 2025
874575-HT1ACLONEDHUMAN3H-WAY100635FK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874585-HT1BCLONEDHUMAN3H-5-CTFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874595-HT1DCLONEDHUMAN3H-5-CTFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874605-HT1ECLONEDHUMAN3H-5-HTFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874615-HT2ACLONEDHUMAN3H-KETANSERINFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874625-HT2BCLONEDHUMAN3H-LSDFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874635-HT2CCLONEDHUMAN3H-MESULERGINEFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874645-HT3CLONEDHUMAN3H-GR-65630FK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874655-HT5ACLONEDHUMAN3H-LSDFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874665-HT6CLONEDHUMAN3H-LSDFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
874675-HT7CLONEDHUMAN3H-LSDFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87468Alpha1ACLONEDHUMAN3H-PRAZOSINFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87469Alpha1BCLONEDHUMAN3H-PRAZOSINFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87470Alpha1DCLONEDHUMAN3H-PRAZOSINFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87471Alpha2ACLONEDHUMAN3H-RAUWOLSCINEFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87472Alpha2BCLONEDHUMAN3H-RAUWOLSCINEFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87473Beta 1CLONEDHUMAN125I-PindololFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87474Beta3CLONEDHUMAN125I-PindololFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87475Beta 2CLONEDHUMAN3H-CGP12177FK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87476D1CLONEDHUMAN3H-SCH23390FK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87477D5CLONEDHUMAN3H-SCH23390FK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87478D2CLONEDHUMAN3H-N-MethylspiperoneFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87479D3CLONEDHUMAN3H-N-MethylspiperoneFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87480D4CLONEDHUMAN3H-N-MethylspiperoneFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87481DATCLONEDHUMAN3H-WIN 35,428FK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87482DORCLONEDHUMAN3H-DADLEFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87483KORCORTICAL MEMBRANESRAT3H-MUSCIMOLFK881>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
87484H1CLONEDHUMAN3H-PYRILAMINEFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
874855-HT1DCLONEDHUMAN125I-aminopotentidineFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87486H3CLONEDHUMAN3H-Alpha-methylhistamineFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87487H4CLONEDHUMAN3H-HistamineFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87488KORCLONEDHUMAN3H-U69593FK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87489M1CLONEDHUMAN3H-QNBFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87490M2CLONEDHUMAN3H-QNBFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87491M4CLONEDHUMAN3H-QNBFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87492M5CLONEDHUMAN3H-QNBFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87493MORCLONEDHUMAN3H-DAMGOFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87494NETCLONEDHUMAN3H-NisoxetineFK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87495PBRKidney membranesRAT3H-PK11195FK881>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87496SERTCLONEDHUMAN3H-CITALOPRAMFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87497Sigma 1CLONEDHUMAN3H-Pentazocine(+)FK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87498Sigma 2CLONEDHUMAN3H-DTGFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87499Sigma 2PC12RAT3H-DTGFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87500BZPCEREBRAL CORTEXRATFNZFK881>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87501BZPCEREBRAL CORTEXRATFNZ1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
875025-HT1ACLONEDHUMAN3H-WAY1006351,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875035-HT1BCLONEDHUMAN3H-5-CT1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875045-HT1DCLONEDHUMAN3H-5-CT1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875055-HT1ECLONEDHUMAN3H-5-HT1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875065-HT2ACLONEDHUMAN3H-KETANSERIN1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875075-HT2BCLONEDHUMAN3H-LSD1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875085-HT2CCLONEDHUMAN3H-MESULERGINE1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875095-HT3CLONEDHUMAN3H-GR-656301,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875105-HT5ACLONEDHUMAN3H-LSD1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875115-HT6CLONEDHUMAN3H-LSD1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875125-HT7CLONEDHUMAN3H-LSD1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87513Alpha1ACLONEDHUMAN3H-PRAZOSIN1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87514Alpha1BCLONEDHUMAN3H-PRAZOSIN1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87515Alpha1DCLONEDHUMAN3H-PRAZOSIN1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87516Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87517Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87518Beta 1CLONEDHUMAN125I-Pindolol1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87519Beta3CLONEDHUMAN125I-Pindolol1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87520Beta 2CLONEDHUMAN3H-CGP121771,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87521D1CLONEDHUMAN3H-SCH233901,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87522D5CLONEDHUMAN3H-SCH233901,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87523D2CLONEDHUMAN3H-N-Methylspiperone1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87524D3CLONEDHUMAN3H-N-Methylspiperone1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87525D4CLONEDHUMAN3H-N-Methylspiperone1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87526DATCLONEDHUMAN3H-WIN 35,4281,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87527DORCLONEDHUMAN3H-DADLE1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87528KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
87529H1CLONEDHUMAN3H-PYRILAMINE1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
875305-HT1DCLONEDHUMAN125I-aminopotentidine1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87531H3CLONEDHUMAN3H-Alpha-methylhistamine1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87532H4CLONEDHUMAN3H-Histamine1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87533KORCLONEDHUMAN3H-U695931,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87534M1CLONEDHUMAN3H-QNB1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87535M2CLONEDHUMAN3H-QNB1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87536M4CLONEDHUMAN3H-QNB1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87537M5CLONEDHUMAN3H-QNB1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87538MORCLONEDHUMAN3H-DAMGO1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87539NETCLONEDHUMAN3H-Nisoxetine1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87540PBRKidney membranesRAT3H-PK111951,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87541SERTCLONEDHUMAN3H-CITALOPRAM1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87542Sigma 1CLONEDHUMAN3H-Pentazocine(+)1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87543Sigma 2CLONEDHUMAN3H-DTG1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87544Sigma 2PC12RAT3H-DTG1,5-Bis(4-methoxyphenyl)-3-(2,2,2-trifluoroethoxy)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
875455-HT1ACLONEDHUMAN3H-WAY1006352-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875465-HT1BCLONEDHUMAN3H-5-CT2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875475-HT1DCLONEDHUMAN3H-5-CT2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875485-HT1ECLONEDHUMAN3H-5-HT2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875495-HT2ACLONEDHUMAN3H-KETANSERIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875505-HT2BCLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875515-HT2CCLONEDHUMAN3H-MESULERGINE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875525-HT3CLONEDHUMAN3H-GR-656302-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875535-HT5ACLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875545-HT6CLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875555-HT7CLONEDHUMAN3H-LSD2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87556Alpha1ACLONEDHUMAN3H-PRAZOSIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87557Alpha1BCLONEDHUMAN3H-PRAZOSIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87558Alpha1DCLONEDHUMAN3H-PRAZOSIN2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87559Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87560Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87561Beta 1CLONEDHUMAN125I-Pindolol2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87562Beta3CLONEDHUMAN125I-Pindolol2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87563Beta 2CLONEDHUMAN3H-CGP121772-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87564D1CLONEDHUMAN3H-SCH233902-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87565D5CLONEDHUMAN3H-SCH233902-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87566D2CLONEDHUMAN3H-N-Methylspiperone2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87567D3CLONEDHUMAN3H-N-Methylspiperone2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87568D4CLONEDHUMAN3H-N-Methylspiperone2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87569DATCLONEDHUMAN3H-WIN 35,4282-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87570DORCLONEDHUMAN3H-DADLE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87571KORCORTICAL MEMBRANESRAT3H-MUSCIMOL2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
87572H1CLONEDHUMAN3H-PYRILAMINE2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
875735-HT1DCLONEDHUMAN125I-aminopotentidine2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87574H3CLONEDHUMAN3H-Alpha-methylhistamine2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87575H4CLONEDHUMAN3H-Histamine2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87576KORCLONEDHUMAN3H-U695932-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87577M1CLONEDHUMAN3H-QNB2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87578M2CLONEDHUMAN3H-QNB2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87579M4CLONEDHUMAN3H-QNB2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87580M5CLONEDHUMAN3H-QNB2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87581MORCLONEDHUMAN3H-DAMGO2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87582NETCLONEDHUMAN3H-Nisoxetine2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87583PBRKidney membranesRAT3H-PK111952-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87584SERTCLONEDHUMAN3H-CITALOPRAM2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87585Sigma 1CLONEDHUMAN3H-Pentazocine(+)2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87586Sigma 2CLONEDHUMAN3H-DTG2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87587Sigma 2PC12RAT3H-DTG2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87588BZPCORTICAL MEMBRANESRATFNZ2-Fluoro-5-(1-(4-methoxyphenyl)-3-(trifluoromethyl)-1H-1,2,4-triazol-5- yl)pyridine>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87589BZPCORTICAL MEMBRANESRATFNZ3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
875905-HT1ACLONEDHUMAN3H-WAY1006353-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875915-HT1BCLONEDHUMAN3H-5-CT3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875925-HT1DCLONEDHUMAN3H-5-CT3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875935-HT1ECLONEDHUMAN3H-5-HT3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875945-HT2ACLONEDHUMAN3H-KETANSERIN3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875955-HT2BCLONEDHUMAN3H-LSD3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875965-HT2CCLONEDHUMAN3H-MESULERGINE3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875975-HT3CLONEDHUMAN3H-GR656303-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875985-HT5ACLONEDHUMAN3H-LSD3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
875995-HT6CLONEDHUMAN3H-LSD3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876005-HT7CLONEDHUMAN3H-LSD3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87601Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87602Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87603Alpha1DCLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87604Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87605Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87606Beta 1CLONEDHUMAN125I-Pindolol3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87607Beta3CLONEDHUMAN125I-Pindolol3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87608Beta 2CLONEDHUMAN3H-CGP121773-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87609D1CLONEDHUMAN3H-SCH233903-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87610D5CLONEDHUMAN3H-SCH233903-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87611D2CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87612D3CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87613D4CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87614DATCLONEDHUMAN3H-WIN 35,4283-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87615DORCLONEDHUMAN3H-DADLE3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87616KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
87617H1CLONEDHUMAN3H-PYRILAMINE3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
876185-HT1DCLONEDHUMAN125I-aminopotentidine3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87619H3CLONEDHUMAN3H-Alpha-methylhistamine3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87620H4CLONEDHUMAN3H-Histamine3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87621KORCLONEDHUMAN3H-U695933-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87622M1CLONEDHUMAN3H-QNB3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87623M2CLONEDHUMAN3H-QNB3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87624M4CLONEDHUMAN3H-QNB3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87625M5CLONEDHUMAN3H-QNB3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87626MORCLONEDHUMAN3H-DAMGO3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87627NETCLONEDHUMAN3H-Nisoxetine3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87628PBRKidney membranesRAT3H-PK111953-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87629SERTCLONEDHUMAN3H-CITALOPRAM3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87630Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87631Sigma 2CLONEDHUMAN3H-DTG3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87632Sigma 2PC12RAT3H-DTG3-(Fluoromethylthio)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
876335-HT1ACLONEDHUMAN3H-WAY1006353-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876345-HT1BCLONEDHUMAN3H-5-CT3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876355-HT1DCLONEDHUMAN3H-5-CT3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876365-HT1ECLONEDHUMAN3H-5-HT3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876375-HT2ACLONEDHUMAN3H-KETANSERIN3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876385-HT2BCLONEDHUMAN3H-LSD3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876395-HT2CCLONEDHUMAN3H-MESULERGINE3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876405-HT3CLONEDHUMAN3H-GR656303-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876415-HT5ACLONEDHUMAN3H-LSD3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876425-HT6CLONEDHUMAN3H-LSD3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876435-HT7CLONEDHUMAN3H-LSD3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87644Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87645Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87646Alpha1DCLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87647Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87648Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87649Beta 1CLONEDHUMAN125I-Pindolol3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87650Beta3CLONEDHUMAN125I-Pindolol3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87651Beta 2CLONEDHUMAN3H-CGP121773-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87652D1CLONEDHUMAN3H-SCH233903-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87653D5CLONEDHUMAN3H-SCH233903-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87654D2CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87655D3CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87656D4CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87657DATCLONEDHUMAN3H-WIN 35,4283-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87658DORCLONEDHUMAN3H-DADLE3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87659KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
87660H1CLONEDHUMAN3H-PYRILAMINE3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
876615-HT1DCLONEDHUMAN125I-aminopotentidine3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87662H3CLONEDHUMAN3H-CGP121773-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87663H4CLONEDHUMAN3H-Histamine3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87664KORCLONEDHUMAN3H-U695933-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87665M1CLONEDHUMAN3H-QNB3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87666M2CLONEDHUMAN3H-QNB3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87667M4CLONEDHUMAN3H-QNB3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87668M5CLONEDHUMAN3H-QNB3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87669MORCLONEDHUMAN3H-DAMGO3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87670NETCLONEDHUMAN3H-Nisoxetine3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87671PBRKidney membranesRAT3H-PK111953-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87672SERTCLONEDHUMAN3H-CITALOPRAM3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87673Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87674Sigma 2CLONEDHUMAN3H-DTG3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87675Sigma 2PC12RAT3H-DTG3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87676BZPCORTICAL MEMBRANESRATFNZ3-(Fluoromethylsulfinyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87677BZPCORTICAL MEMBRANESRATFNZ3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
876785-HT1ACLONEDHUMAN3H-WAY1006353-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876795-HT1BCLONEDHUMAN3H-5-CT3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876805-HT1DCLONEDHUMAN3H-5-CT3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876815-HT1ECLONEDHUMAN3H-5-HT3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876825-HT2ACLONEDHUMAN3H-KETANSERIN3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876835-HT2BCLONEDHUMAN3H-LSD3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876845-HT2CCLONEDHUMAN3H-MESULERGINE3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876855-HT3CLONEDHUMAN3H-GR656303-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876865-HT5ACLONEDHUMAN3H-LSD3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876875-HT6CLONEDHUMAN3H-LSD3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
876885-HT7CLONEDHUMAN3H-LSD3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87689Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87690Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87691Alpha1DCLONEDHUMAN3H-PRAZOSIN3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87692Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87693Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87694Beta 1CLONEDHUMAN125I-Pindolol3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87695Beta3CLONEDHUMAN125I-Pindolol3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87696Beta 2CLONEDHUMAN3H-CGP121773-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87697D1CLONEDHUMAN3H-SCH233903-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87698D5CLONEDHUMAN3H-SCH233903-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87699D2CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87700D3CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87701D4CLONEDHUMAN3H-N-Methylspiperone3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87702DATCLONEDHUMAN3H-WIN 35,4283-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87703DORCLONEDHUMAN3H-DADLE3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87704KORCORTICAL MEMBRANESRAT3H-MUSCIMOL3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 27, 2025
87705H1CLONEDHUMAN3H-PYRILAMINE3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
877065-HT1DCLONEDHUMAN125I-aminopotentidine3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87707H3CLONEDHUMAN3H-Alpha-methylhistamine3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87708H4CLONEDHUMAN3H-Histamine3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87709KORCLONEDHUMAN3H-U695933-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87710M1CLONEDHUMAN3H-QNB3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87711M2CLONEDHUMAN3H-QNB3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87712M4CLONEDHUMAN3H-QNB3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87713M5CLONEDHUMAN3H-QNB3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87714MORCLONEDHUMAN3H-DAMGO3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87715NETCLONEDHUMAN3H-Nisoxetine3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87716PBRKidney membranesRAT3H-PK111953-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 15, 2025
87717SERTCLONEDHUMAN3H-CITALOPRAM3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87718Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87719Sigma 2CLONEDHUMAN3H-DTG3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
87720Sigma 2PC12RAT3H-DTG3-(Fluoromethylsulfonyl)-1,5-bis(4-methoxyphenyl)-1H-1,2,4-triazole>10000Singh P et al 2018Jan 15, 2025Jan 28, 2025
877215-HT6CLONEDHUMAN3H-LSD2‐methyl‐5‐(2‐phenylethyl)‐1H,2H,3H,4H,5H‐pyrido[4,3‐b]indole22Staron J et al 2016Jan 15, 2025Jan 15, 2025
87722D2CLONEDHUMAN3H-RACLOPRIDE2‐methyl‐5‐(2‐phenylethyl)‐1H,2H,3H,4H,5H‐pyrido[4,3‐b]indole77Staron J et al 2016Jan 15, 2025Jan 28, 2025
877235-HT7CLONEDHUMAN3H-5-CT2‐methyl‐5‐(2‐phenylethyl)‐1H,2H,3H,4H,5H‐pyrido[4,3‐b]indole8Staron J et al 2016Jan 15, 2025Jan 15, 2025
877245-HT1ACLONEDHUMAN3H-8-OH-DPAT2‐methyl‐5‐(2‐phenylethyl)‐1H,2H,3H,4H,5H‐pyrido[4,3‐b]indole217Staron J et al 2016Jan 15, 2025Jan 15, 2025
877255-HT2ACLONEDHUMAN3H-KETANSERIN2‐methyl‐5‐(2‐phenylethyl)‐1H,2H,3H,4H,5H‐pyrido[4,3‐b]indole29Staron J et al 2016Jan 15, 2025Jan 15, 2025
877265-HT1ACLONEDHUMAN3H-8-OH-DPAT(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(1‐phenylpiperidin‐4‐yl)methyl]amine10Staron J et al 2016Jan 15, 2025Jan 15, 2025
877275-HT7CLONEDHUMAN3H-5-CT(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(1‐phenylpiperidin‐4‐yl)methyl]amine430Staron J et al 2016Jan 15, 2025Jan 15, 2025
87728D2CLONEDHUMAN3H-RACLOPRIDE(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(1‐phenylpiperidin‐4‐yl)methyl]amine210Staron J et al 2016Jan 15, 2025Jan 28, 2025
877295-HT6CLONEDHUMAN3H-LSD(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(1‐phenylpiperidin‐4‐yl)methyl]amine2280Staron J et al 2016Jan 15, 2025Jan 15, 2025
877305-HT6CLONEDHUMAN3H-LSDN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline63Staron J et al 2016Jan 15, 2025Jan 15, 2025
87731D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline476Staron J et al 2016Jan 15, 2025Jan 28, 2025
877325-HT7CLONEDHUMAN3H-5-CTN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline121Staron J et al 2016Jan 15, 2025Jan 15, 2025
877335-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline1682Staron J et al 2016Jan 15, 2025Jan 15, 2025
877345-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(dimethylamino)ethyl]‐N‐(2‐phenylethyl)aniline233Staron J et al 2016Jan 15, 2025Jan 15, 2025
877355-HT1ACLONEDHUMAN3H-8-OH-DPAT[(1‐cyclohexylpiperidin‐4‐yl)methyl](2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)amine22Staron J et al 2016Jan 15, 2025Jan 15, 2025
877365-HT7CLONEDHUMAN3H-5-CT[(1‐cyclohexylpiperidin‐4‐yl)methyl](2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)amine3428Staron J et al 2016Jan 15, 2025Jan 15, 2025
87737D2CLONEDHUMAN3H-RACLOPRIDE[(1‐cyclohexylpiperidin‐4‐yl)methyl](2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)amine1609Staron J et al 2016Jan 15, 2025Jan 28, 2025
877385-HT6CLONEDHUMAN3H-LSD[(1‐cyclohexylpiperidin‐4‐yl)methyl](2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)amine2675Staron J et al 2016Jan 15, 2025Jan 15, 2025
877395-HT6CLONEDHUMAN3H-LSD(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(4‐phenylphenyl)methyl]amine3760Staron J et al 2016Jan 15, 2025Jan 15, 2025
87740D2CLONEDHUMAN3H-RACLOPRIDE(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(4‐phenylphenyl)methyl]amine110Staron J et al 2016Jan 15, 2025Jan 28, 2025
877415-HT7CLONEDHUMAN3H-5-CT(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(4‐phenylphenyl)methyl]amine857Staron J et al 2016Jan 15, 2025Jan 15, 2025
877425-HT1ACLONEDHUMAN3H-8-OH-DPAT(2,3‐dihydro‐1,4‐benzodioxin‐2‐ylmethyl)[(4‐phenylphenyl)methyl]amine101Staron J et al 2016Jan 15, 2025Jan 15, 2025
877435-HT2ACLONEDHUMAN3H-KETANSERINN‐[2‐(diethylamino)ethyl]‐N‐(2‐phenylethyl)aniline128Staron J et al 2016Jan 15, 2025Jan 15, 2025
877445-HT1ACLONEDHUMAN3H-8-OH-DPATN‐[2‐(diethylamino)ethyl]‐N‐(2‐phenylethyl)aniline7614Staron J et al 2016Jan 15, 2025Jan 15, 2025
877455-HT7CLONEDHUMAN3H-5-CTN‐[2‐(diethylamino)ethyl]‐N‐(2‐phenylethyl)aniline205Staron J et al 2016Jan 15, 2025Jan 15, 2025
87746D2CLONEDHUMAN3H-RACLOPRIDEN‐[2‐(diethylamino)ethyl]‐N‐(2‐phenylethyl)aniline266Staron J et al 2016Jan 15, 2025Jan 28, 2025
877475-HT6CLONEDHUMAN3H-LSDN‐[2‐(diethylamino)ethyl]‐N‐(2‐phenylethyl)aniline51Staron J et al 2016Jan 15, 2025Jan 15, 2025
877485-HT6CLONEDHUMAN3H-LSDN‐[3‐(dimethylamino)propyl]‐N‐(2‐phenylethyl)aniline67Staron J et al 2016Jan 15, 2025Jan 15, 2025