96749 CORTEX RAT [3H]rauwolscine N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 16.3 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96750 CORTEX RAT [3H]rauwolscine RISPERIDONE 28.2 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96751 CORTEX RAT [3H]rauwolscine N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide 193 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96752 H1 CEREBELLUM GUINEA PIG [3H]mepyramine N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 2143 Huang L et al 2020 Jan 15, 2025 Jan 28, 2025
96753 H1 CEREBELLUM GUINEA PIG [3H]mepyramine RISPERIDONE 49.3 Huang L et al 2020 Jan 15, 2025 Jan 28, 2025
96754 5-HT2C CORTEX RAT [3H]mesulergine N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 1987 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96755 5-HT2C CORTEX RAT [3H]mesulergine RISPERIDONE 39.1 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96756 5-HT2C CORTEX RAT [3H]mesulergine N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide 186 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96757 CORTEX RAT [3H]prazosin N-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide 3296 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96758 CORTEX RAT [3H]prazosin RISPERIDONE 21.9 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96759 CORTEX RAT [3H]prazosin N-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide 195 Huang L et al 2020 Jan 15, 2025 Jan 15, 2025
96760 D1 CLONED HUMAN [3H]SCH23390 ARIPIPRAZOLE 310 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96761 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96762 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96763 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96764 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96765 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96766 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 4800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96767 D1 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 3800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96768 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96769 D1 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96770 D1 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96771 D1 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96772 D1 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96773 D1 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96774 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96775 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96776 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96777 D1 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 7700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96778 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96779 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 8800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96780 D1 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96781 D2 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 0.52 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96782 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 1 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96783 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 1.1 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96784 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 5.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96785 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 3.4 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96786 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.6 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96787 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 0.91 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96788 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.98 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96789 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 29 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96790 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96791 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 5300 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96792 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 8300 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96793 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96794 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96795 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 780 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96796 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 630 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96797 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 6400 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96798 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 3200 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96799 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96800 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 120 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96801 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 360 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96802 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96803 D2 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 0.38 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96804 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 0.58 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96805 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 0.73 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96806 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96807 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 1.3 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96808 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.54 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96809 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 0.67 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96810 D2 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.95 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96811 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 16 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96812 D2 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 1.1 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96813 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1200 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96814 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1800 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96815 D2 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 8900 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96816 D2 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 6000 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96817 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 250 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96818 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 200 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96819 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 3400 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96820 D2 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 1500 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96821 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 480 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96822 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 35 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96823 D2 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 5700 Mannel B et al 2017 Jan 15, 2025 Jan 29, 2025
96824 D3 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96825 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 2.3 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96826 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 1.2 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96827 D3 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 24 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96828 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96829 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96830 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 0.35 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96831 D3 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 0.39 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96832 D3 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 30 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96833 D3 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 35 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96834 D3 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96835 D3 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 160 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96836 D3 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 510 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96837 D3 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 110 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96838 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 380 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96839 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 48 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96840 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 42 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96841 D3 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 790 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96842 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 420 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96843 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 5.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96844 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 3.7 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96845 D3 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 2800 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96846 D4 CLONED HUMAN [3H]spiperone ARIPIPRAZOLE 63 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96847 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 41 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96848 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 10 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96849 D4 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 130 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96850 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 11 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96851 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 31 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96852 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2.3 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96853 D4 CLONED HUMAN [3H]spiperone 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 2.9 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96854 D4 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 140 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96855 D4 CLONED HUMAN [3H]spiperone 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 62 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96856 D4 CLONED HUMAN [3H]spiperone 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 6100 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96857 D4 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 440 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96858 D4 CLONED HUMAN [3H]spiperone 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96859 D4 CLONED HUMAN [3H]spiperone 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96860 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 560 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96861 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 59 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96862 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 4900 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96863 D4 CLONED HUMAN [3H]spiperone 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 2600 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96864 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 7600 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96865 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 880 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96866 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 210 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96867 D4 CLONED HUMAN [3H]spiperone 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96868 D5 CLONED HUMAN [3H]SCH23390 ARIPIPRAZOLE 1600 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96869 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96870 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 7700 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96871 D5 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96872 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96873 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96874 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96875 D5 CLONED HUMAN [3H]SCH23390 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96876 D5 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96877 D5 CLONED HUMAN [3H]SCH23390 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96878 D5 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96879 D5 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96880 D5 CLONED HUMAN [3H]SCH23390 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96881 D5 CLONED HUMAN [3H]SCH23390 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96882 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96883 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96884 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96885 D5 CLONED HUMAN [3H]SCH23390 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96886 D5 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96887 D5 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96888 D5 CLONED HUMAN [3H]SCH23390 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 28, 2025
96889 5-HT1A CLONED PIG [3H]WAY100635 ARIPIPRAZOLE 88 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96890 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 14 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96891 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 21 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96892 5-HT1A CLONED PIG [3H]WAY100635 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 4.7 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96893 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 13 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96894 5-HT1A CLONED HUMAN [3H]WAY100635 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 33 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96895 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 12 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96896 5-HT1A CLONED PIG [3H]WAY100635 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 19 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96897 5-HT1A CLONED PIG [3H]WAY100635 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 23 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96898 5-HT1A CLONED PIG [3H]WAY100635 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 16 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96899 5-HT1A CLONED PIG [3H]WAY100635 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96900 5-HT1A CLONED PIG [3H]WAY100635 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 4500 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96901 5-HT1A CLONED PIG [3H]WAY100635 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96902 5-HT1A CLONED PIG [3H]WAY100635 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96903 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 620 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96904 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1700 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96905 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96906 5-HT1A CLONED PIG [3H]WAY100635 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 1600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96907 5-HT1A CLONED PIG [3H]WAY100635 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96908 5-HT1A CLONED HUMAN [3H]WAY100635 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 180 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96909 5-HT1A CLONED PIG [3H]WAY100635 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96910 5-HT1A CLONED PIG [3H]WAY100635 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 5800 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96911 5-HT2A CLONED HUMAN [3H]ketanserin ARIPIPRAZOLE 3.6 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96912 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96913 5-HT2A CLONED HUMAN [3H]ketanserin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 1000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96914 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96915 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 5400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96916 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 2400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96917 5-HT2A CLONED HUMAN [3H]ketanserin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 880 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96918 5-HT2A CLONED HUMAN [3H]ketanserin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96919 5-HT2A CLONED HUMAN [3H]ketanserin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 980 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96920 5-HT2A CLONED HUMAN [3H]ketanserin 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96921 5-HT2A CLONED HUMAN [3H]ketanserin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96922 5-HT2A CLONED HUMAN [3H]ketanserin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96923 5-HT2A CLONED HUMAN [3H]ketanserin 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 3600 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96924 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96925 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96926 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 6400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96927 5-HT2A CLONED HUMAN [3H]ketanserin 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 2100 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96928 5-HT2A CLONED HUMAN [3H]ketanserin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96929 5-HT2A CLONED HUMAN [3H]ketanserin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 3700 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96930 5-HT2A CLONED HUMAN [3H]ketanserin 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96931 CLONED PIG [3H]prazosin ARIPIPRAZOLE 17 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96932 CLONED PIG [3H]prazosin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 49 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96933 CLONED PIG [3H]prazosin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde 11 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96934 CLONED PIG [3H]prazosin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde 160 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96935 CLONED PIG [3H]prazosin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 29 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96936 CLONED PIG [3H]prazosin 5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 39 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96937 CLONED PIG [3H]prazosin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 13 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96938 CLONED PIG [3H]prazosin 5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 17 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96939 CLONED PIG [3H]prazosin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form) 120 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96940 CLONED PIG [3H]prazosin 5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form) 89 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96941 CLONED PIG [3H]prazosin 4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96942 CLONED PIG [3H]prazosin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 4200 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96943 CLONED PIG [3H]prazosin 4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96944 CLONED PIG [3H]prazosin 4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA 4200 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96945 CLONED PIG [3H]prazosin 1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA 1500 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96946 CLONED PIG [3H]prazosin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 1500 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96947 CLONED PIG [3H]prazosin 1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96948 CLONED PIG [3H]prazosin 1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine 2400 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96949 CLONED PIG [3H]prazosin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96950 CLONED PIG [3H]prazosin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA 160 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96951 CLONED PIG [3H]prazosin 1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA 900 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96952 CLONED PIG [3H]prazosin 1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA >10000 Mannel B et al 2017 Jan 15, 2025 Jan 15, 2025
96953 M2 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96954 M3 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96955 M4 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96956 M5 CLONED HUMAN [3H]QNB 3′′-F-DPPy 913 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96957 MOR CLONED HUMAN [3H]DAMGO 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96958 NET CLONED HUMAN [3H]Nisoxetine 3′′-F-DPPy 189 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96959 PBR CLONED HUMAN [3H]PK11195 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96960 SERT CLONED HUMAN [3H]Citalopram 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96961 Sigma 1 CLONED HUMAN [3H]Pentazocine 3′′-F-DPPy 124 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96962 Sigma 2 CLONED HUMAN [3H]DTG 3′′-F-DPPy 741 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96963 NMDA FOREBRAIN RAT [3H]MK-801 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96964 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96965 5-HT1B CLONED HUMAN [3H]GR127543 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96966 5-HT1D CLONED HUMAN [3H]GR127543 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96967 5-HT1E CLONED HUMAN [3H]5-HT 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96968 5-HT2A CLONED HUMAN [3H]ketanserin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96969 5-HT2C CLONED HUMAN [3H]mesulergine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96970 5-HT3 CLONED HUMAN [3H]LY278584 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96971 Alpha1A CLONED HUMAN [3H]prazosin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96972 Alpha1B CLONED HUMAN [3H]prazosin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96973 Alpha1D CLONED HUMAN [3H]prazosin 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96974 Alpha2A CLONED HUMAN [3H]Clonidine 4′′-F-DPPy 86 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96975 Alpha2C CLONED HUMAN [3H]Clonidine 4′′-F-DPPy 101 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96976 Beta1 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96977 Beta2 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96978 Beta3 CLONED HUMAN [125I]Iodopindolol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96979 D1 CLONED HUMAN [3H]SCH23390 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96980 D2 CLONED HUMAN [3H]N-methylspiperone 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96981 D3 CLONED HUMAN [3H]N-methylspiperone 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96982 D4 CLONED HUMAN [3H]N-methylspiperone 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96983 D5 CLONED HUMAN [3H]SCH23390 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96984 DAT CLONED HUMAN [3H]WIN35428 4′′-F-DPPy 231 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96985 DOR CLONED HUMAN [3H]DADLE 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96986 GABAA BRAIN RAT [3H]-Muscimol 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
96987 H1 CLONED HUMAN [3H]Pyrilamine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96988 5-HT1D CLONED HUMAN [3H]Tiotidine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96989 H3 CLONED HUMAN [3H]-alpha-methylhistamine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96990 H4 CLONED HUMAN [3H]Histamine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96991 KOR CLONED HUMAN [3H]U69593 4′′-F-DPPy 4460 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96992 M1 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96993 M2 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96994 M4 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96995 M5 CLONED HUMAN [3H]QNB 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96996 MOR CLONED HUMAN [3H]DAMGO 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
96997 NET CLONED HUMAN [3H]Nisoxetine 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96998 PBR CLONED HUMAN [3H]PK11195 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
96999 SERT CLONED HUMAN [3H]Citalopram 4′′-F-DPPy 352 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97000 Sigma 1 CLONED HUMAN [3H]Pentazocine 4′′-F-DPPy 139 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97001 Sigma 2 CLONED HUMAN [3H]DTG 4′′-F-DPPy 321 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97002 NMDA FOREBRAIN RAT [3H]MK-801 PCP 57.9 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97003 NMDA FOREBRAIN RAT [3H]MK-801 PCP 22.1 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97004 NMDA FOREBRAIN RAT [3H]MK-801 Diphenidine 18.2 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97005 NMDA FOREBRAIN RAT [3H]MK-801 Ketamine 323.9 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97006 NMDA FOREBRAIN RAT [3H]MK-801 (+)-MK-801 2.5 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97007 NMDA FOREBRAIN RAT [3H]MK-801 Memantine 378.4 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97008 NMDA FOREBRAIN RAT [3H]MK-801 DPPy 280 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97009 NMDA FOREBRAIN RAT [3H]MK-801 Fluorolintane (2-F-DPPy) 87.92 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97010 NMDA FOREBRAIN RAT [3H]MK-801 3-F-DPPy 632.64 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97011 NMDA FOREBRAIN RAT [3H]MK-801 4-F-DPPy 953.37 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97012 NMDA FOREBRAIN RAT [3H]MK-801 2′′-F-DPPy 609.74 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97013 NMDA FOREBRAIN RAT [3H]MK-801 3′′-F-DPPy 261.84 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97014 NMDA FOREBRAIN RAT [3H]MK-801 4′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97015 NMDA FOREBRAIN RAT [3H]MK-801 Fluorolintane (2-F-DPPy) 88 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97016 5-HT1A CLONED HUMAN [3H]8-OH-DPAT Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97017 5-HT1B CLONED HUMAN [3H]GR127543 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97018 5-HT1D CLONED HUMAN [3H]GR127543 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97019 5-HT1E CLONED HUMAN [3H]5-HT Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97020 5-HT2A CLONED HUMAN [3H]ketanserin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97021 5-HT2C CLONED HUMAN [3H]mesulergine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97022 5-HT3 CLONED HUMAN [3H]LY278584 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97023 Alpha1A CLONED HUMAN [3H]prazosin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97024 Alpha1B CLONED HUMAN [3H]prazosin Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97025 Alpha2A CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) 829 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97026 Alpha2B CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) 388 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97027 Alpha2C CLONED HUMAN [3H]Clonidine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97028 Beta1 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97029 Beta2 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97030 Beta3 CLONED HUMAN [125I]Iodopindolol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97031 D1 CLONED HUMAN [3H]SCH23390 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97032 D2 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97033 D3 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97034 D4 CLONED HUMAN [3H]N-methylspiperone Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97035 D5 CLONED HUMAN [3H]SCH23390 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97036 DAT CLONED HUMAN [3H]WIN35428 Fluorolintane (2-F-DPPy) 327 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97037 DOR CLONED HUMAN [3H]DADLE Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97038 GABAA BRAIN RAT [3H]-Muscimol Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97039 H1 CLONED HUMAN [3H]Pyrilamine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97040 5-HT1D CLONED HUMAN [3H]Tiotidine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97041 H4 CLONED HUMAN [3H]Histamine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97042 KOR CLONED HUMAN [3H]U69593 Fluorolintane (2-F-DPPy) 1278 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97043 M1 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) 1597 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97044 M2 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97045 M3 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97046 M4 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97047 M5 CLONED HUMAN [3H]QNB Fluorolintane (2-F-DPPy) 556 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97048 MOR CLONED HUMAN [3H]DAMGO Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97049 NET CLONED HUMAN [3H]Nisoxetine Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97050 PBR CLONED HUMAN [3H]PK11195 Fluorolintane (2-F-DPPy) >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97051 SERT CLONED HUMAN [3H]Citalopram Fluorolintane (2-F-DPPy) 4115 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97052 Sigma 1 CLONED HUMAN [3H]Pentazocine Fluorolintane (2-F-DPPy) 110 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97053 NMDA FOREBRAIN RAT [3H]MK-801 3-F-DPPy 633 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97054 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97055 5-HT1B CLONED HUMAN [3H]GR127543 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97056 5-HT1D CLONED HUMAN [3H]GR127543 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97057 5-HT1E CLONED HUMAN [3H]5-HT 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97058 5-HT2A CLONED HUMAN [3H]ketanserin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97059 5-HT2C CLONED HUMAN [3H]mesulergine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97060 5-HT3 CLONED HUMAN [3H]LY278584 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97061 Alpha1A CLONED HUMAN [3H]prazosin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97062 Alpha1B CLONED HUMAN [3H]prazosin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97063 Alpha1D CLONED HUMAN [3H]prazosin 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97064 Alpha2A CLONED HUMAN [3H]Clonidine 3-F-DPPy 732 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97065 Alpha2B CLONED HUMAN [3H]Clonidine 3-F-DPPy 129 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97066 Alpha2C CLONED HUMAN [3H]Clonidine 3-F-DPPy 333 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97067 Beta1 CLONED HUMAN [125I]Iodopindolol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97068 Beta2 CLONED HUMAN 3-F-DPPy [125I]Iodopindolol >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97069 Beta3 CLONED HUMAN [125I]Iodopindolol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97070 D1 CLONED HUMAN [3H]SCH23390 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97071 D2 CLONED HUMAN [3H]N-methylspiperone 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97072 D3 CLONED HUMAN [3H]N-methylspiperone 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97073 D4 CLONED HUMAN [3H]N-methylspiperone 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97074 D5 CLONED HUMAN [3H]SCH23390 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97075 DAT CLONED HUMAN [3H]WIN35428 3-F-DPPy 12 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97076 DOR CLONED HUMAN [3H]DADLE 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97077 GABAA BRAIN RAT [3H]-Muscimol 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97078 H1 CLONED HUMAN [3H]Pyrilamine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97079 5-HT1D CLONED HUMAN [3H]Tiotidine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97080 H3 CLONED HUMAN [3H]-alpha-methylhistamine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97081 H4 CLONED HUMAN [3H]Histamine 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97082 KOR CLONED HUMAN [3H]U69593 3-F-DPPy 1583 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97083 M1 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97084 M2 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97085 M3 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97086 M5 CLONED HUMAN [3H]QNB 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97087 MOR CLONED HUMAN [3H]DAMGO 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97088 NET CLONED HUMAN [3H]Nisoxetine 3-F-DPPy 192 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97089 PBR CLONED HUMAN [3H]PK11195 3-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97090 SERT CLONED HUMAN [3H]Citalopram 3-F-DPPy 1202 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97091 Sigma 1 CLONED HUMAN [3H]Pentazocine 3-F-DPPy 193 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97092 Sigma 2 CLONED HUMAN [3H]DTG 3-F-DPPy 1934 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97093 NMDA FOREBRAIN RAT [3H]MK-801 4-F-DPPy 953 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97094 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97095 5-HT1B CLONED HUMAN [3H]GR127543 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97096 5-HT1D CLONED HUMAN [3H]GR127543 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97097 5-HT1E CLONED HUMAN [3H]5-HT 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97098 5-HT2C CLONED HUMAN [3H]mesulergine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97099 5-HT3 CLONED HUMAN [3H]LY278584 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97100 Alpha1A CLONED HUMAN [3H]prazosin 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97101 Alpha1B CLONED HUMAN [3H]prazosin 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97102 Alpha1D CLONED HUMAN [3H]prazosin 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97103 Alpha2A CLONED HUMAN [3H]Clonidine 4-F-DPPy 1401 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97104 Alpha2B CLONED HUMAN [3H]Clonidine 4-F-DPPy 1242 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97105 Beta2 CLONED HUMAN [125I]Iodopindolol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97106 Beta3 CLONED HUMAN [125I]Iodopindolol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97107 D1 CLONED HUMAN [3H]SCH23390 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97108 D2 CLONED HUMAN [3H]N-methylspiperone 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97109 D3 CLONED HUMAN [3H]N-methylspiperone 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97110 D4 CLONED HUMAN [3H]N-methylspiperone 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97111 D5 CLONED HUMAN [3H]SCH23390 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97112 DAT CLONED HUMAN [3H]WIN35428 4-F-DPPy 140 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97113 DOR CLONED HUMAN [3H]DADLE 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97114 GABAA BRAIN RAT [3H]-Muscimol 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97115 H1 CLONED HUMAN [3H]Pyrilamine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97116 5-HT1D CLONED HUMAN [3H]Tiotidine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97117 H3 CLONED HUMAN [3H]-alpha-methylhistamine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97118 H4 CLONED HUMAN [3H]Histamine 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97119 KOR CLONED HUMAN [3H]U69593 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97120 M1 CLONED HUMAN [3H]QNB 4-F-DPPy 1900 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97121 M2 CLONED HUMAN [3H]QNB 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97122 M3 CLONED HUMAN [3H]QNB 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97123 M5 CLONED HUMAN [3H]QNB 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97124 MOR CLONED HUMAN [3H]DAMGO 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97125 NET CLONED HUMAN [3H]Nisoxetine 4-F-DPPy 249 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97126 PBR CLONED HUMAN [3H]PK11195 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97127 SERT CLONED HUMAN [3H]Citalopram 4-F-DPPy 681 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97128 Sigma 1 CLONED HUMAN [3H]Pentazocine 4-F-DPPy 386 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97129 Sigma 2 CLONED HUMAN [3H]DTG 4-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97130 NMDA FOREBRAIN RAT [3H]MK-801 2′′-F-DPPy 610 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97131 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97132 5-HT1B CLONED HUMAN [3H]GR127543 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97133 5-HT1D CLONED HUMAN [3H]GR127543 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97134 5-HT1E CLONED HUMAN [3H]5-HT 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97135 5-HT2A CLONED HUMAN [3H]ketanserin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97136 5-HT2C CLONED HUMAN [3H]mesulergine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97137 5-HT3 CLONED HUMAN [3H]LY278584 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97138 Alpha1A CLONED HUMAN [3H]prazosin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97139 Alpha1B CLONED HUMAN [3H]prazosin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97140 Alpha1D CLONED HUMAN [3H]prazosin 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97141 Alpha2A CLONED HUMAN [3H]Clonidine 2′′-F-DPPy 307 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97142 Alpha2B CLONED HUMAN [3H]Clonidine 2′′-F-DPPy 89 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97143 Alpha2C CLONED HUMAN [3H]Clonidine 2′′-F-DPPy 214 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97144 Beta1 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97145 Beta2 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97146 Beta3 CLONED HUMAN [125I]Iodopindolol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97147 D1 CLONED HUMAN [3H]SCH23390 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97148 D2 CLONED HUMAN [3H]N-methylspiperone 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97149 D3 CLONED HUMAN [3H]N-methylspiperone 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97150 D4 CLONED HUMAN [3H]N-methylspiperone 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97151 D5 CLONED HUMAN [3H]SCH23390 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97152 DAT CLONED HUMAN [3H]WIN35428 2′′-F-DPPy 85 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97153 DOR CLONED HUMAN [3H]DADLE 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97154 GABAA BRAIN RAT [3H]-Muscimol 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97155 H1 CLONED HUMAN [3H]Pyrilamine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97156 5-HT1D CLONED HUMAN [3H]Tiotidine 2′′-F-DPPy 2194 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97157 H3 CLONED HUMAN [3H]-alpha-methylhistamine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97158 H4 CLONED HUMAN [3H]Histamine 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97159 KOR CLONED HUMAN [3H]U69593 2′′-F-DPPy 642 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97160 M1 CLONED HUMAN [3H]QNB 2′′-F-DPPy 1660 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97161 M2 CLONED HUMAN [3H]QNB 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97162 M4 CLONED HUMAN [3H]QNB 2′′-F-DPPy 576 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97163 M5 CLONED HUMAN [3H]QNB 2′′-F-DPPy 489 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97164 MOR CLONED HUMAN [3H]DAMGO 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97165 NET CLONED HUMAN [3H]Nisoxetine 2′′-F-DPPy 215 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97166 PBR CLONED HUMAN [3H]PK11195 2′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97167 SERT CLONED HUMAN [3H]Citalopram 2′′-F-DPPy 661 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97168 Sigma 1 CLONED HUMAN [3H]Pentazocine 2′′-F-DPPy 146 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97169 Sigma 2 CLONED HUMAN [3H]DTG 2′′-F-DPPy 712 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97170 NMDA CLONED HUMAN [3H]MK-801 3′′-F-DPPy 262 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97171 5-HT1A CLONED HUMAN [3H]8-OH-DPAT 3′′-F-DPPy 534 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97172 5-HT1B CLONED HUMAN [3H]GR127543 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97173 5-HT1D CLONED HUMAN [3H]GR127543 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97174 5-HT1E CLONED HUMAN [3H]5-HT 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97175 5-HT2A CLONED HUMAN [3H]ketanserin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97176 5-HT2C CLONED HUMAN [3H]mesulergine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97177 5-HT3 CLONED HUMAN [3H]LY278584 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97178 Alpha1A CLONED HUMAN [3H]prazosin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97179 Alpha1B CLONED HUMAN [3H]prazosin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97180 Alpha1D CLONED HUMAN [3H]prazosin 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97181 Alpha2A CLONED HUMAN [3H]Clonidine 3′′-F-DPPy 915 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97182 Alpha2B CLONED HUMAN [3H]Clonidine 3′′-F-DPPy 307 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97183 Alpha2C CLONED HUMAN [3H]Clonidine 3′′-F-DPPy 1159 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97184 Beta1 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97185 Beta2 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97186 Beta3 CLONED HUMAN [125I]Iodopindolol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97187 D1 CLONED HUMAN [3H]SCH23390 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97188 D2 CLONED HUMAN 3′′-F-DPPy [3H]N-methylspiperone >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97189 D3 CLONED HUMAN [3H]N-methylspiperone 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97190 D4 CLONED HUMAN [3H]N-methylspiperone 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97191 D5 CLONED HUMAN [3H]SCH23390 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97192 DAT CLONED HUMAN [3H]WIN35428 3′′-F-DPPy 103 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97193 DOR CLONED HUMAN [3H]DADLE 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97194 GABAA BRAIN RAT [3H]-Muscimol 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 29, 2025
97195 H1 CLONED HUMAN [3H]Pyrilamine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97196 5-HT1D CLONED HUMAN [3H]Tiotidine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97197 H3 CLONED HUMAN [3H]-alpha-methylhistamine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97198 H4 CLONED HUMAN [3H]Histamine 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97199 KOR CLONED HUMAN [3H]U69593 3′′-F-DPPy 1435 Wallach J et al 2019 Jan 15, 2025 Jan 28, 2025
97200 M1 CLONED HUMAN [3H]QNB 3′′-F-DPPy >10000 Wallach J et al 2019 Jan 15, 2025 Jan 15, 2025
97201 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5200 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97202 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 9.5 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97203 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 740 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97204 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97205 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 4.2 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97206 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97207 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 18 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97208 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 26 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97209 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine  63 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97210 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-methoxyphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine  28 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97211 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 117 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97212 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 84 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97213 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 160 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97214 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl 16 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97215 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 180 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97216 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 400 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97217 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl >10000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97218 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 910 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97219 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 22 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97220 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 5.2 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97221 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 97 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97222 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 450 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97223 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 240 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97224 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 600 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97225 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 33 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97226 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 2600 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97227 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 71 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97228 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 180 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97229 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 17 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97230 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 390 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97231 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 5.9 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97232 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 190 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97233 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 34 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97234 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 740 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97235 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 5.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97236 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine 1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl 51 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97237 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine AS-19 12 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97238 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (R)-8-OH-DPAT 48 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97239 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine (S)-8-OH-DPAT 1000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97240 5-HT7 CLONED HUMAN [3H]-5-carboxamidotryptamine BUSPIRONE 840 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97241 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1100 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97242 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 6.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97243 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97244 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 4 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97245 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 14 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97246 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 7.5 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97247 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 23 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97248 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 82 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97249 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine  180 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97250 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 73 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97251 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 30 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97252 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 19 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97253 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 190 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97254 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl 33 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97255 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 230 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97256 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 2200 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97257 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl >10000 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97258 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 2230 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97259 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 130 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97260 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine 64 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97261 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 650 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97262 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 1400 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97263 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine 98 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97264 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 550 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97265 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 24 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97266 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5600 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97267 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 33 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97268 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 150 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97269 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine 4.5 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97270 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 130 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97271 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 0.64 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97272 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 210 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97273 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl 5.9 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97274 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 92 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97275 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine 1.8 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97276 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine 1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl 1.3 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97277 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine AS-19 240 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97278 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (R)-8-OH-DPAT 7.1 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97279 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine (S)-8-OH-DPAT 7.6 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97280 5-HT1A CLONED HUMAN [3H]-5-carboxamidotryptamine BUSPIRONE 50 Perry CK et al 2020 Jan 15, 2025 Jan 15, 2025
97281 MOR CLONED HUMAN [3H]diprenorphine SRI-22138 7.55 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97282 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 23.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97283 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 138 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97284 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 2.33 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97285 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 171 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97286 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 370 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97287 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 235 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97288 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 24.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97289 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 191 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97290 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97291 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 135 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97292 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 249 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97293 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 61.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97294 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 91.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97295 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 148 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97296 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 12.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97297 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.97 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97298 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 15.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97299 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 4.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97300 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol 56.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97301 MOR CLONED HUMAN [3H]diprenorphine N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 141 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97302 MOR CLONED HUMAN [3H]diprenorphine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 337 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97303 MOR CLONED HUMAN [3H]diprenorphine N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 159 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97304 MOR CLONED HUMAN [3H]diprenorphine NALOXONE 59.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97305 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 14.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97306 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 105 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97307 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 82.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97308 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 47.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97309 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 1.05 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97310 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 10.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97311 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 66.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97312 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 47.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97313 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 88.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97314 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 121 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97315 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 3.79 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97316 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 99.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97317 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.18 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97318 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.37 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97319 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 819 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97320 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 799 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97321 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.96 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97322 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.82 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97323 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 70.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97324 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 95.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97325 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.99 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97326 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 92.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97327 MOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol 499 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97328 DOR CLONED HUMAN [3H]diprenorphine SRI-22138 2.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97329 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 19.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97330 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 20.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97331 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.42 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97332 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 53.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97333 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 7.52 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97334 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 97.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97335 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 26.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97336 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 34.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97337 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.78 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97338 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 64.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97339 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 93.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97340 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97341 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 48 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97342 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 30.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97343 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 8.37 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97344 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 69.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97345 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 68.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97346 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 53.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97347 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol 14 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97348 DOR CLONED HUMAN [3H]diprenorphine N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 3333 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97349 DOR CLONED HUMAN [3H]diprenorphine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 3333 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97350 DOR CLONED HUMAN [3H]diprenorphine N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 394 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97351 DOR CLONED HUMAN [3H]diprenorphine NALOXONE 98.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97352 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 0.169 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97353 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 6.52 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97354 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 30.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97355 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.43 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97356 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 63.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97357 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 3.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97358 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 22.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97359 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.18 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97360 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 40.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97361 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 257 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97362 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 7.96 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97363 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 64.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97364 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 8.12 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97365 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.24 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97366 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 172 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97367 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 32.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97368 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.89 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97369 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97370 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 11 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97371 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 12.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97372 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 64.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97373 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 14.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97374 DOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol 7.48 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97375 KOR CLONED HUMAN [3H]diprenorphine SRI-22138 60.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97376 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 132 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97377 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 75.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97378 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.69 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97379 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 35.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97380 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 71.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97381 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 152 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97382 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 17.6 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97383 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 102 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97384 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 129 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97385 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 175 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97386 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 134 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97387 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 126 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97388 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 103 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97389 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 140 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97390 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 18.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97391 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 7.96 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97392 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 11.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97393 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.18 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97394 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol 22.7 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97395 KOR CLONED HUMAN [3H]diprenorphine N-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 13.5 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97396 KOR CLONED HUMAN [3H]diprenorphine N-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 608 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97397 KOR CLONED HUMAN [3H]diprenorphine N-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide 15.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97398 KOR CLONED HUMAN [3H]diprenorphine U50,488 31.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97399 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 13.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97400 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 19.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97401 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 27.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97402 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 15.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97403 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 0.51 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97404 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 6.62 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97405 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 30.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97406 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 24.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97407 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 19.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97408 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 29.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97409 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 8.4 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97410 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 23.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97411 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 14.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97412 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 10.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97413 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o 21.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97414 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 31 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97415 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 5.3 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97416 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 21.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97417 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 60.2 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97418 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 57.9 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97419 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol 24.8 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97420 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol 57.1 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97421 KOR CLONED HUMAN [3H]diprenorphine (4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol 252 Vekariya RH et al 2020 Jan 15, 2025 Jan 28, 2025
97422 A1 CLONED HUMAN [3H]DPCPX ISAM-141 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97423 A1 CLONED HUMAN [3H]DPCPX ISAM-142 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97424 A1 CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97425 A1 CLONED HUMAN [3H]DPCPX propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97426 A1 CLONED HUMAN [3H]DPCPX ISAM-134 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97427 A1 CLONED HUMAN [3H]DPCPX ISAM-140 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97428 A1 CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97429 A1 CLONED HUMAN [3H]DPCPX DPCPX 2.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97430 A1 CLONED HUMAN [3H]DPCPX ZM241385 683 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97431 A1 CLONED HUMAN [3H]DPCPX Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97432 A1 CLONED HUMAN [3H]DPCPX Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97433 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97434 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97435 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97436 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97437 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97438 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97439 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97440 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97441 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97442 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97443 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97444 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97445 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97446 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97447 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97448 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97449 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97450 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97451 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 14.8 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97452 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 8.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97453 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97454 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97455 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 20.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97456 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97457 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97458 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97459 A1 CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97460 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97461 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97462 A1 CLONED HUMAN [3H]DPCPX (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97463 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97464 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97465 A1 CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97466 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97467 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97468 A1 CLONED HUMAN [3H]DPCPX ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97469 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 233 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97470 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 301 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97471 A1 CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97472 A1 CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97473 A2A CLONED HUMAN [3H]ZM-241385 ISAM-141 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97474 A2A CLONED HUMAN [3H]ZM-241385 ISAM-142 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97475 A2A CLONED HUMAN [3H]ZM-241385 ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97476 A2A CLONED HUMAN [3H]ZM-241385 propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97477 A2A CLONED HUMAN [3H]ZM-241385 ISAM-134 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97478 A2A CLONED HUMAN [3H]ZM-241385 ISAM-140 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97479 A2A CLONED HUMAN [3H]ZM-241385 ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97480 A2A CLONED HUMAN Leucyl-3H-NC DPCPX 157 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97481 A2A CLONED HUMAN [3H]ZM-241385 ZM241385 1.9 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97482 A2A CLONED HUMAN [3H]ZM-241385 Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97483 A2A CLONED HUMAN [3H]ZM-241385 Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97484 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97485 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97486 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97487 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97488 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97489 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97490 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97491 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97492 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97493 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97494 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97495 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97496 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97497 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97498 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97499 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97500 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97501 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97502 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97503 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97504 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97505 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97506 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97507 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97508 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97509 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97510 A2A CLONED HUMAN [3H]ZM-241385 ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97511 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97512 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 5 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97513 A2A CLONED HUMAN [3H]ZM-241385 (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97514 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97515 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97516 A2A CLONED HUMAN [3H]ZM-241385 ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97517 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97518 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97519 A2A CLONED HUMAN [3H]ZM-241385 ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97520 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 282 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97521 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97522 A2A CLONED HUMAN [3H]ZM-241385 (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97523 A2A CLONED HUMAN [3H]ZM-241385 (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97524 A2B CLONED HUMAN [3H]DPCPX ISAM-141 20.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97525 A2B CLONED HUMAN [3H]DPCPX ISAM-142 11.4 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97526 A2B CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 29.71 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97527 A2B CLONED HUMAN [3H]DPCPX propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  29.34 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97528 A2B CLONED HUMAN [3H]DPCPX ISAM-134 12.03 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97529 A2B CLONED HUMAN [3H]DPCPX ISAM-140 3.49 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97530 A2B CLONED HUMAN [3H]DPCPX ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 484.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97531 A2B CLONED HUMAN [3H]DPCPX propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  371.2 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97532 A2B CLONED HUMAN [3H]DPCPX DPCPX 73.24 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97533 A2B CLONED HUMAN [3H]DPCPX ZM241385 65.7 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97534 A2B CLONED HUMAN [3H]DPCPX Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97535 A2B CLONED HUMAN [3H]DPCPX Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97536 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97537 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97538 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97539 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97540 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 449.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97541 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 517.1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97542 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 49.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97543 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 31.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97544 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97545 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97546 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 789 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97547 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 721 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97548 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 707 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97549 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1104 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97550 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 23.4 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97551 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 29.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97552 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97553 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 278 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97554 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 92.6 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97555 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 340 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97556 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 714 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97557 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1031 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97558 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 98.7 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97559 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 175 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97560 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 769 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97561 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 708 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97562 A2B CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 388 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97563 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 753 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97564 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 402 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97565 A2B CLONED HUMAN [3H]DPCPX (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97566 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 8.1 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97567 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 43.41 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97568 A2B CLONED HUMAN [3H]DPCPX ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97569 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97570 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97571 A2B CLONED HUMAN [3H]DPCPX ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97572 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 508 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97573 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97574 A2B CLONED HUMAN [3H]DPCPX (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 215 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97575 A2B CLONED HUMAN [3H]DPCPX (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 68.3 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97576 A3 CLONED HUMAN [3H]NECA ISAM-141 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97577 A3 CLONED HUMAN [3H]NECA ISAM-142 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97578 A3 CLONED HUMAN [3H]NECA ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97579 A3 CLONED HUMAN [3H]NECA propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97580 A3 CLONED HUMAN [3H]NECA ISAM-134 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97581 A3 CLONED HUMAN [3H]NECA ISAM-140 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97582 A3 CLONED HUMAN [3H]NECA ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97583 A3 CLONED HUMAN [3H]NECA DPCPX 1722 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97584 A3 CLONED HUMAN [3H]NECA ZM241385 863 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97585 A3 CLONED HUMAN [3H]NECA Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97586 A3 CLONED HUMAN [3H]NECA Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97587 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97588 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97589 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97590 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97591 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97592 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97593 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97594 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97595 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97596 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97597 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate ( 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97598 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97599 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97600 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97601 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97602 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97603 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97604 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97605 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97606 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97607 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97608 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97609 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97610 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97611 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97612 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97613 A3 CLONED HUMAN [3H]NECA ±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97614 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97615 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97616 A3 CLONED HUMAN [3H]NECA (±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97617 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97618 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97619 A3 CLONED HUMAN [3H]NECA ±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97620 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97621 A3 CLONED HUMAN [3H]NECA (±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97622 A3 CLONED HUMAN [3H]NECA ±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97623 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 418 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97624 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97625 A3 CLONED HUMAN [3H]NECA (±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97626 A3 CLONED HUMAN [3H]NECA (±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate 1000 Mallo-Abreu A et al 2020 Jan 15, 2025 Jan 15, 2025
97627 SST1 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97628 SST2 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.04 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97629 SST3 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 0.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97630 SST4 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 1.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97631 SST5 CLONED HUMAN 125I-LTT-SST-28 Somatostatin-14 2.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97632 SST1 CLONED HUMAN 125I-LTT-SST-28 L-363,377 5664 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97633 SST2 CLONED HUMAN 125I-LTT-SST-28 L-363,377 0.5 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97634 SST3 CLONED HUMAN 125I-LTT-SST-28 L-363,377 3072 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97635 SST4 CLONED HUMAN 125I-LTT-SST-28 L-363,377 >10000 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97636 SST5 CLONED HUMAN 125I-LTT-SST-28 L-363,377 2009 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97637 SST1 CLONED HUMAN 125I-LTT-SST-28 L-797,591 1.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97638 SST2 CLONED HUMAN 125I-LTT-SST-28 L-797,591 1875 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97639 SST3 CLONED HUMAN 125I-LTT-SST-28 L-797,591 2240 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97640 SST4 CLONED HUMAN 125I-LTT-SST-28 L-797,591 170 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97641 SST5 CLONED HUMAN 125I-LTT-SST-28 L-797,591 3600 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97642 SST1 CLONED HUMAN 125I-LTT-SST-28 L-779,976 2760 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97643 SST2 CLONED HUMAN 125I-LTT-SST-28 L-779,976 0.05 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97644 SST3 CLONED HUMAN 125I-LTT-SST-28 L-779,976 729 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97645 SST4 CLONED HUMAN 125I-LTT-SST-28 L-779,976 310 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97646 SST5 CLONED HUMAN 125I-LTT-SST-28 L-779,976 4260 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97647 SST1 CLONED HUMAN 125I-LTT-SST-28 L-796,778 1255 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97648 SST2 CLONED HUMAN 125I-LTT-SST-28 L-796,778 >10000 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97649 SST3 CLONED HUMAN 125I-LTT-SST-28 L-796,778 24 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97650 SST4 CLONED HUMAN 125I-LTT-SST-28 L-796,778 8650 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97651 SST5 CLONED HUMAN 125I-LTT-SST-28 L-796,778 1200 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97652 SST1 CLONED HUMAN 125I-LTT-SST-28 L-803,087 199 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97653 SST2 CLONED HUMAN 125I-LTT-SST-28 L-803,087 4720 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97654 SST3 CLONED HUMAN 125I-LTT-SST-28 L-803,087 1280 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97655 SST4 CLONED HUMAN 125I-LTT-SST-28 L-803,087 0.7 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97656 SST5 CLONED HUMAN 125I-LTT-SST-28 L-803,087 3880 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97657 SST1 CLONED HUMAN 125I-LTT-SST-28 L-817,818 3.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97658 SST2 CLONED HUMAN 125I-LTT-SST-28 L-817,818 52 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97659 SST3 CLONED HUMAN 125I-LTT-SST-28 L-817,818 64 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97660 SST4 CLONED HUMAN 125I-LTT-SST-28 L-817,818 82 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97661 SST5 CLONED HUMAN 125I-LTT-SST-28 L-817,818 0.4 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97662 SST1 CLONED HUMAN Functional L-797,591 3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97663 SST2 CLONED HUMAN Functional L-779,976 0.05 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97664 SST4 CLONED HUMAN Functional L-803,087 0.2 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97665 SST5 CLONED HUMAN Functional L-817,818 1.3 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97666 SST3 CLONED HUMAN Functional L-796,778 18 Rohrer SP, et.al., 1998 Jan 15, 2025 Jan 15, 2025
97667 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 4-quinolone 122 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97668 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-ethyl-4-quinolone 20 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97669 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-propoxycarbonyl-4-quinolone 1.8 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97670 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Butoxycarbonyl-6-ethyl-4-quinolone 13 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97671 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 28 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97672 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone 28 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97673 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-pentoxycarbonyl-4-quinolone 35 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97674 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone 92 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97675 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Cyclopentoxycarbonyl-6-ethyl-4-quinolone 19 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97676 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-i-propoxycarbonyl-4-quinolone 214 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97677 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(4-methyl-2-pentoxycarbonyl)-4-quinolone 295 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97678 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-pentoxycarbonyl)-4-quinolone 2600 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97679 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Carboxy-6-ethyl-4-quinolone 208 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97680 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-4-quinolone 78 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97681 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Butoxycarbonyl-4-quinolone 54 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97682 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-4-quinolone 16 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97683 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-propyl-4-quinolone 17 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97684 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-i-propyl-4-quinolone 15 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97685 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 1.4 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97686 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-propoxycarbonyl-4-quinolone 0.17 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97687 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone 6850 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97688 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-2-methyl-4-quinolone 4200 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97689 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-propylaminocarbonyl-4-quinolone 0.26 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97690 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 3-Butylaminocarbonyl-6-ethyl-4-quinolone 0.54 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97691 KOR CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-propylaminocarbonyl-4-quinolone 0.048 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97692 KOR CORTICAL MEMBRANES RAT 3H-flumazenil Propyl 2-methyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate 870 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97693 KOR CORTICAL MEMBRANES RAT 3H-flumazenil Ethyl 7-Oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate >10000 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97694 KOR CORTICAL MEMBRANES RAT 3H-flumazenil Propyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate 7130 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97695 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 4.1 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97696 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone 89 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97697 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-4-quinolone 26 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97698 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Bromo-3-ethoxycarbonyl-4-quinolone 14 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97699 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 0.27 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97700 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil 6-Benzyl-3-ethoxycarbonyl-4-quinolone 7.2 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97701 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil DIAZEPAM 12 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97702 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil DIAZEPAM 14 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97703 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil Zolpidem 1850 Lager, E. et al., 2006 Jan 15, 2025 Jan 28, 2025
97704 GABAA CORTICAL MEMBRANES RAT 3H-flumazenil Zolpidem 53 Lager, E. et al., 2006 Jan 15, 2025 Jan 27, 2025
97705 L1210 cells MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 1800 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97706 L1210 cells MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 700 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97707 L1210 cells MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97708 L1210 cells MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97709 L1210 cells MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 1300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97710 L1210 cells MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97711 L1210 cells MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97712 L1210 + DFMO MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97713 L1210 + DFMO MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97714 L1210 + DFMO MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 700 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97715 L1210 + DFMO MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 150 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97716 L1210 + DFMO MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 200 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97717 L1210 + DFMO MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 300 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97718 L1210 + DFMO MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 1400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97719 L1210 cells MOUSE 14C-spermidine N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97720 L1210 cells MOUSE 14C-spermidine N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 2500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97721 L1210 cells MOUSE 14C-spermidine N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 6200 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97722 L1210 cells MOUSE 14C-spermidine N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 1800 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97723 L1210 cells MOUSE 14C-spermidine N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 5000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97724 L1210 cells MOUSE 14C-spermidine N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 1700 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97725 L1210 cells MOUSE 14C-spermidine N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97726 CHO-MG MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97727 C.H.O. MOUSE Functional N-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97728 CHO-MG MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97729 C.H.O. MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 1500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97730 C.H.O. MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt 4100 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97731 CHO-MG MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97732 CHO-MG MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt >10000 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97733 C.H.O. MOUSE Functional N-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 450 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97734 C.H.O. MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97735 CHO-MG MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt 9500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97736 CHO-MG MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 8800 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97737 C.H.O. MOUSE Functional N1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt 2500 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97738 C.H.O. MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 1900 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97739 CHO-MG MOUSE Functional N-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt 3400 Wang C, et al., 2003 Jan 15, 2025 Jan 15, 2025
97740 Y5 CLONED HUMAN 125I-PYY FMS586 4.3 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97741 Y5 CLONED HUMAN 125I-PYY L-152,804 25 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97742 Y5 CLONED HUMAN 125I-PYY PYY 1 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97743 Y1 CLONED HUMAN 125I-PYY PYY 2 Kakui, N. et al., 2006 Jan 15, 2025 Jan 15, 2025
97744 Y1 CLONED HUMAN 125I-PYY L-152,804 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 15, 2025
97745 Y1 CLONED HUMAN 125I-PYY FMS586 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 15, 2025
97746 Y2 CLONED HUMAN 125I-PYY FMS586 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97747 Y2 CLONED HUMAN 125I-PYY L-152,804 >10000 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025
97748 Y2 CLONED HUMAN 125I-PYY PYY 2.1 Kakui, N. et al., 2006 Jan 15, 2025 Jan 29, 2025