The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 94,001-95,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
96749CORTEXRAT[3H]rauwolscineN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide16.3Huang L et al 2020Jan 15, 2025Jan 15, 2025
96750CORTEXRAT[3H]rauwolscineRISPERIDONE28.2Huang L et al 2020Jan 15, 2025Jan 15, 2025
96751CORTEXRAT[3H]rauwolscineN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide193Huang L et al 2020Jan 15, 2025Jan 15, 2025
96752H1CEREBELLUMGUINEA PIG[3H]mepyramineN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide2143Huang L et al 2020Jan 15, 2025Jan 28, 2025
96753H1CEREBELLUMGUINEA PIG[3H]mepyramineRISPERIDONE49.3Huang L et al 2020Jan 15, 2025Jan 28, 2025
967545-HT2CCORTEXRAT[3H]mesulergineN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide1987Huang L et al 2020Jan 15, 2025Jan 15, 2025
967555-HT2CCORTEXRAT[3H]mesulergineRISPERIDONE39.1Huang L et al 2020Jan 15, 2025Jan 15, 2025
967565-HT2CCORTEXRAT[3H]mesulergineN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide186Huang L et al 2020Jan 15, 2025Jan 15, 2025
96757CORTEXRAT[3H]prazosinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide3296Huang L et al 2020Jan 15, 2025Jan 15, 2025
96758CORTEXRAT[3H]prazosinRISPERIDONE21.9Huang L et al 2020Jan 15, 2025Jan 15, 2025
96759CORTEXRAT[3H]prazosinN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide195Huang L et al 2020Jan 15, 2025Jan 15, 2025
96760D1CLONEDHUMAN[3H]SCH23390ARIPIPRAZOLE310Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96761D1CLONEDHUMAN[3H]SCH233905-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96762D1CLONEDHUMAN[3H]SCH233905-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96763D1CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96764D1CLONEDHUMAN[3H]SCH233905-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96765D1CLONEDHUMAN[3H]SCH233905-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96766D1CLONEDHUMAN[3H]SCH233905-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)4800Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96767D1CLONEDHUMAN[3H]SCH233905-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)3800Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96768D1CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96769D1CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96770D1CLONEDHUMAN[3H]SCH233904-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96771D1CLONEDHUMAN[3H]SCH233904-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96772D1CLONEDHUMAN[3H]SCH233904-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96773D1CLONEDHUMAN[3H]SCH233904-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA6000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96774D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96775D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96776D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96777D1CLONEDHUMAN[3H]SCH233901-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine7700Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96778D1CLONEDHUMAN[3H]SCH233901-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96779D1CLONEDHUMAN[3H]SCH233901-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA8800Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96780D1CLONEDHUMAN[3H]SCH233901-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96781D2CLONEDHUMAN[3H]spiperoneARIPIPRAZOLE0.52Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96782D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde1Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96783D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde1.1Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96784D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde5.7Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96785D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)3.4Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96786D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)1.6Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96787D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)0.91Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96788D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)0.98Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96789D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)29Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96790D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)1.7Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96791D2CLONEDHUMAN[3H]spiperone4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA5300Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96792D2CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA8300Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96793D2CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96794D2CLONEDHUMAN[3H]spiperone4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA6900Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96795D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA780Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96796D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA630Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96797D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA6400Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96798D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine3200Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96799D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA1900Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96800D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA120Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96801D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA360Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96802D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96803D2CLONEDHUMAN[3H]spiperoneARIPIPRAZOLE0.38Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96804D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde0.58Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96805D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde0.73Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96806D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde2.9Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96807D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)1.3Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96808D2CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)0.54Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96809D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)0.67Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96810D2CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)0.95Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96811D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)16Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96812D2CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)1.1Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96813D2CLONEDHUMAN[3H]spiperone4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA1200Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96814D2CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA1800Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96815D2CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA8900Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96816D2CLONEDHUMAN[3H]spiperone4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA6000Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96817D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA250Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96818D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA200Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96819D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA3400Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96820D2CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine1500Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96821D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA480Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96822D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA35Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96823D2CLONEDHUMAN[3H]spiperone1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA5700Mannel B et al 2017Jan 15, 2025Jan 29, 2025
96824D3CLONEDHUMAN[3H]spiperoneARIPIPRAZOLE2.9Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96825D3CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde2.3Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96826D3CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde1.2Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96827D3CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde24Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96828D3CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)2.7Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96829D3CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)2.9Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96830D3CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)0.35Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96831D3CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)0.39Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96832D3CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)30Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96833D3CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)35Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96834D3CLONEDHUMAN[3H]spiperone4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA1700Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96835D3CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA160Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96836D3CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA510Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96837D3CLONEDHUMAN[3H]spiperone4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA110Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96838D3CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA380Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96839D3CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA48Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96840D3CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA42Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96841D3CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine790Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96842D3CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA420Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96843D3CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA5.9Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96844D3CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA3.7Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96845D3CLONEDHUMAN[3H]spiperone1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA2800Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96846D4CLONEDHUMAN[3H]spiperoneARIPIPRAZOLE63Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96847D4CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde41Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96848D4CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde10Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96849D4CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde130Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96850D4CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)11Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96851D4CLONEDHUMAN[3H]spiperone5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)31Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96852D4CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)2.3Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96853D4CLONEDHUMAN[3H]spiperone5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)2.9Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96854D4CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)140Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96855D4CLONEDHUMAN[3H]spiperone5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)62Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96856D4CLONEDHUMAN[3H]spiperone4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA6100Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96857D4CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA440Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96858D4CLONEDHUMAN[3H]spiperone4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96859D4CLONEDHUMAN[3H]spiperone4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96860D4CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA560Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96861D4CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA59Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96862D4CLONEDHUMAN[3H]spiperone1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA4900Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96863D4CLONEDHUMAN[3H]spiperone1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine2600Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96864D4CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA7600Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96865D4CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA880Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96866D4CLONEDHUMAN[3H]spiperone1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA210Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96867D4CLONEDHUMAN[3H]spiperone1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96868D5CLONEDHUMAN[3H]SCH23390ARIPIPRAZOLE1600Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96869D5CLONEDHUMAN[3H]SCH233905-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96870D5CLONEDHUMAN[3H]SCH233905-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde7700Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96871D5CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96872D5CLONEDHUMAN[3H]SCH233905-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96873D5CLONEDHUMAN[3H]SCH233905-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96874D5CLONEDHUMAN[3H]SCH233905-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96875D5CLONEDHUMAN[3H]SCH233905-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96876D5CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96877D5CLONEDHUMAN[3H]SCH233905-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96878D5CLONEDHUMAN[3H]SCH233904-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96879D5CLONEDHUMAN[3H]SCH233904-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96880D5CLONEDHUMAN[3H]SCH233904-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96881D5CLONEDHUMAN[3H]SCH233904-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96882D5CLONEDHUMAN[3H]SCH233901-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96883D5CLONEDHUMAN[3H]SCH233901-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96884D5CLONEDHUMAN[3H]SCH233901-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96885D5CLONEDHUMAN[3H]SCH233901-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96886D5CLONEDHUMAN[3H]SCH233901-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96887D5CLONEDHUMAN[3H]SCH233901-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
96888D5CLONEDHUMAN[3H]SCH233901-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 28, 2025
968895-HT1ACLONEDPIG[3H]WAY100635ARIPIPRAZOLE88Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968905-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde14Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968915-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde21Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968925-HT1ACLONEDPIG[3H]WAY1006355-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde4.7Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968935-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)13Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968945-HT1ACLONEDHUMAN[3H]WAY1006355-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)33Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968955-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)12Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968965-HT1ACLONEDPIG[3H]WAY1006355-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)19Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968975-HT1ACLONEDPIG[3H]WAY1006355-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)23Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968985-HT1ACLONEDPIG[3H]WAY1006355-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)16Mannel B et al 2017Jan 15, 2025Jan 15, 2025
968995-HT1ACLONEDPIG[3H]WAY1006354-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA1600Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969005-HT1ACLONEDPIG[3H]WAY1006354-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA4500Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969015-HT1ACLONEDPIG[3H]WAY1006354-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969025-HT1ACLONEDPIG[3H]WAY1006354-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969035-HT1ACLONEDPIG[3H]WAY1006351-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA620Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969045-HT1ACLONEDPIG[3H]WAY1006351-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA1700Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969055-HT1ACLONEDPIG[3H]WAY1006351-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969065-HT1ACLONEDPIG[3H]WAY1006351-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine1600Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969075-HT1ACLONEDPIG[3H]WAY1006351-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969085-HT1ACLONEDHUMAN[3H]WAY1006351-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA180Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969095-HT1ACLONEDPIG[3H]WAY1006351-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969105-HT1ACLONEDPIG[3H]WAY1006351-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA5800Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969115-HT2ACLONEDHUMAN[3H]ketanserinARIPIPRAZOLE3.6Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969125-HT2ACLONEDHUMAN[3H]ketanserin5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969135-HT2ACLONEDHUMAN[3H]ketanserin5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde1000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969145-HT2ACLONEDHUMAN[3H]ketanserin5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969155-HT2ACLONEDHUMAN[3H]ketanserin5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)5400Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969165-HT2ACLONEDHUMAN[3H]ketanserin5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)2400Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969175-HT2ACLONEDHUMAN[3H]ketanserin5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)880Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969185-HT2ACLONEDHUMAN[3H]ketanserin5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)600Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969195-HT2ACLONEDHUMAN[3H]ketanserin5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)980Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969205-HT2ACLONEDHUMAN[3H]ketanserin4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969215-HT2ACLONEDHUMAN[3H]ketanserin4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969225-HT2ACLONEDHUMAN[3H]ketanserin4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969235-HT2ACLONEDHUMAN[3H]ketanserin4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA3600Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969245-HT2ACLONEDHUMAN[3H]ketanserin1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969255-HT2ACLONEDHUMAN[3H]ketanserin1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969265-HT2ACLONEDHUMAN[3H]ketanserin1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA6400Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969275-HT2ACLONEDHUMAN[3H]ketanserin1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine2100Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969285-HT2ACLONEDHUMAN[3H]ketanserin1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969295-HT2ACLONEDHUMAN[3H]ketanserin1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA3700Mannel B et al 2017Jan 15, 2025Jan 15, 2025
969305-HT2ACLONEDHUMAN[3H]ketanserin1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96931CLONEDPIG[3H]prazosinARIPIPRAZOLE17Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96932CLONEDPIG[3H]prazosin5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde49Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96933CLONEDPIG[3H]prazosin5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehyde11Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96934CLONEDPIG[3H]prazosin5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)pyrazolo[1,5-a]pyridine-3-carbaldehyde160Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96935CLONEDPIG[3H]prazosin5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)29Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96936CLONEDPIG[3H]prazosin5-{4-[4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)39Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96937CLONEDPIG[3H]prazosin5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)13Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96938CLONEDPIG[3H]prazosin5-{4-[4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazin-1-yl]butoxy}pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)17Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96939CLONEDPIG[3H]prazosin5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (trans form)120Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96940CLONEDPIG[3H]prazosin5-(4-[4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl]butoxy)-pyrazolo[1,5-a]pyridine-3-carbaldehydoxime (cis form)89Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96941CLONEDPIG[3H]prazosin4-(8-Hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96942CLONEDPIG[3H]prazosin4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA4200Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96943CLONEDPIG[3H]prazosin4-(5-Hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96944CLONEDPIG[3H]prazosin4-(8-Hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA4200Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96945CLONEDPIG[3H]prazosin1-Methyl-4-(8-hydroxyquinolin-2(1H)-one-5-yl)piperazineTFA1500Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96946CLONEDPIG[3H]prazosin1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA1500Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96947CLONEDPIG[3H]prazosin1-Methyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96948CLONEDPIG[3H]prazosin1-Methyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazine2400Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96949CLONEDPIG[3H]prazosin1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96950CLONEDPIG[3H]prazosin1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)piperazineTFA160Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96951CLONEDPIG[3H]prazosin1-Propyl-4-(5-hydroxy-2H-benzo[b][1,4]oxazin-3(4H)-one-8-yl)-1,4-diazepaneTFA900Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96952CLONEDPIG[3H]prazosin1-Propyl-4-(8-hydroxy-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)piperazineTFA>10000Mannel B et al 2017Jan 15, 2025Jan 15, 2025
96953M2CLONEDHUMAN[3H]QNB3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96954M3CLONEDHUMAN[3H]QNB3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96955M4CLONEDHUMAN[3H]QNB3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96956M5CLONEDHUMAN[3H]QNB3′′-F-DPPy913Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96957MORCLONEDHUMAN[3H]DAMGO3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96958NETCLONEDHUMAN[3H]Nisoxetine3′′-F-DPPy189Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96959PBRCLONEDHUMAN[3H]PK111953′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96960SERTCLONEDHUMAN[3H]Citalopram3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96961Sigma 1CLONEDHUMAN[3H]Pentazocine3′′-F-DPPy124Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96962Sigma 2CLONEDHUMAN[3H]DTG3′′-F-DPPy741Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96963NMDAFOREBRAINRAT[3H]MK-8014′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
969645-HT1ACLONEDHUMAN[3H]8-OH-DPAT4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
969655-HT1BCLONEDHUMAN[3H]GR1275434′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
969665-HT1DCLONEDHUMAN[3H]GR1275434′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
969675-HT1ECLONEDHUMAN[3H]5-HT4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
969685-HT2ACLONEDHUMAN[3H]ketanserin4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
969695-HT2CCLONEDHUMAN[3H]mesulergine4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
969705-HT3CLONEDHUMAN[3H]LY2785844′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96971Alpha1ACLONEDHUMAN[3H]prazosin4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96972Alpha1BCLONEDHUMAN[3H]prazosin4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96973Alpha1DCLONEDHUMAN[3H]prazosin4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96974Alpha2ACLONEDHUMAN[3H]Clonidine4′′-F-DPPy86Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96975Alpha2CCLONEDHUMAN[3H]Clonidine4′′-F-DPPy101Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96976Beta1CLONEDHUMAN[125I]Iodopindolol4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96977Beta2CLONEDHUMAN[125I]Iodopindolol4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96978Beta3CLONEDHUMAN[125I]Iodopindolol4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96979D1CLONEDHUMAN[3H]SCH233904′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96980D2CLONEDHUMAN[3H]N-methylspiperone4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96981D3CLONEDHUMAN[3H]N-methylspiperone4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96982D4CLONEDHUMAN[3H]N-methylspiperone4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96983D5CLONEDHUMAN[3H]SCH233904′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96984DATCLONEDHUMAN[3H]WIN354284′′-F-DPPy231Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96985DORCLONEDHUMAN[3H]DADLE4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96986GABAABRAINRAT[3H]-Muscimol4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 29, 2025
96987H1CLONEDHUMAN[3H]Pyrilamine4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
969885-HT1DCLONEDHUMAN[3H]Tiotidine4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96989H3CLONEDHUMAN[3H]-alpha-methylhistamine4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96990H4CLONEDHUMAN[3H]Histamine4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96991KORCLONEDHUMAN[3H]U695934′′-F-DPPy4460Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96992M1CLONEDHUMAN[3H]QNB4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96993M2CLONEDHUMAN[3H]QNB4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96994M4CLONEDHUMAN[3H]QNB4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96995M5CLONEDHUMAN[3H]QNB4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96996MORCLONEDHUMAN[3H]DAMGO4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
96997NETCLONEDHUMAN[3H]Nisoxetine4′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96998PBRCLONEDHUMAN[3H]PK111954′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
96999SERTCLONEDHUMAN[3H]Citalopram4′′-F-DPPy352Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97000Sigma 1CLONEDHUMAN[3H]Pentazocine4′′-F-DPPy139Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97001Sigma 2CLONEDHUMAN[3H]DTG4′′-F-DPPy321Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97002NMDAFOREBRAINRAT[3H]MK-801PCP57.9Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97003NMDAFOREBRAINRAT[3H]MK-801PCP22.1Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97004NMDAFOREBRAINRAT[3H]MK-801Diphenidine18.2Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97005NMDAFOREBRAINRAT[3H]MK-801Ketamine323.9Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97006NMDAFOREBRAINRAT[3H]MK-801(+)-MK-8012.5Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97007NMDAFOREBRAINRAT[3H]MK-801Memantine378.4Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97008NMDAFOREBRAINRAT[3H]MK-801DPPy280Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97009NMDAFOREBRAINRAT[3H]MK-801Fluorolintane (2-F-DPPy)87.92Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97010NMDAFOREBRAINRAT[3H]MK-8013-F-DPPy632.64Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97011NMDAFOREBRAINRAT[3H]MK-8014-F-DPPy953.37Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97012NMDAFOREBRAINRAT[3H]MK-8012′′-F-DPPy609.74Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97013NMDAFOREBRAINRAT[3H]MK-8013′′-F-DPPy261.84Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97014NMDAFOREBRAINRAT[3H]MK-8014′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97015NMDAFOREBRAINRAT[3H]MK-801Fluorolintane (2-F-DPPy)88Wallach J et al 2019Jan 15, 2025Jan 28, 2025
970165-HT1ACLONEDHUMAN[3H]8-OH-DPATFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970175-HT1BCLONEDHUMAN[3H]GR127543Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970185-HT1DCLONEDHUMAN[3H]GR127543Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970195-HT1ECLONEDHUMAN[3H]5-HTFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970205-HT2ACLONEDHUMAN[3H]ketanserinFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970215-HT2CCLONEDHUMAN[3H]mesulergineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970225-HT3CLONEDHUMAN[3H]LY278584Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97023Alpha1ACLONEDHUMAN[3H]prazosinFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97024Alpha1BCLONEDHUMAN[3H]prazosinFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97025Alpha2ACLONEDHUMAN[3H]ClonidineFluorolintane (2-F-DPPy)829Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97026Alpha2BCLONEDHUMAN[3H]ClonidineFluorolintane (2-F-DPPy)388Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97027Alpha2CCLONEDHUMAN[3H]ClonidineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97028Beta1CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97029Beta2CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97030Beta3CLONEDHUMAN[125I]IodopindololFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97031D1CLONEDHUMAN[3H]SCH23390Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97032D2CLONEDHUMAN[3H]N-methylspiperoneFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97033D3CLONEDHUMAN[3H]N-methylspiperoneFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97034D4CLONEDHUMAN[3H]N-methylspiperoneFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97035D5CLONEDHUMAN[3H]SCH23390Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97036DATCLONEDHUMAN[3H]WIN35428Fluorolintane (2-F-DPPy)327Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97037DORCLONEDHUMAN[3H]DADLEFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97038GABAABRAINRAT[3H]-MuscimolFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 29, 2025
97039H1CLONEDHUMAN[3H]PyrilamineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
970405-HT1DCLONEDHUMAN[3H]TiotidineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97041H4CLONEDHUMAN[3H]HistamineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97042KORCLONEDHUMAN[3H]U69593Fluorolintane (2-F-DPPy)1278Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97043M1CLONEDHUMAN[3H]QNBFluorolintane (2-F-DPPy)1597Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97044M2CLONEDHUMAN[3H]QNBFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97045M3CLONEDHUMAN[3H]QNBFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97046M4CLONEDHUMAN[3H]QNBFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97047M5CLONEDHUMAN[3H]QNBFluorolintane (2-F-DPPy)556Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97048MORCLONEDHUMAN[3H]DAMGOFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97049NETCLONEDHUMAN[3H]NisoxetineFluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97050PBRCLONEDHUMAN[3H]PK11195Fluorolintane (2-F-DPPy)>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97051SERTCLONEDHUMAN[3H]CitalopramFluorolintane (2-F-DPPy)4115Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97052Sigma 1CLONEDHUMAN[3H]PentazocineFluorolintane (2-F-DPPy)110Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97053NMDAFOREBRAINRAT[3H]MK-8013-F-DPPy633Wallach J et al 2019Jan 15, 2025Jan 28, 2025
970545-HT1ACLONEDHUMAN[3H]8-OH-DPAT3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970555-HT1BCLONEDHUMAN[3H]GR1275433-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970565-HT1DCLONEDHUMAN[3H]GR1275433-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970575-HT1ECLONEDHUMAN[3H]5-HT3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970585-HT2ACLONEDHUMAN[3H]ketanserin3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970595-HT2CCLONEDHUMAN[3H]mesulergine3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970605-HT3CLONEDHUMAN[3H]LY2785843-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97061Alpha1ACLONEDHUMAN[3H]prazosin3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97062Alpha1BCLONEDHUMAN[3H]prazosin3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97063Alpha1DCLONEDHUMAN[3H]prazosin3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97064Alpha2ACLONEDHUMAN[3H]Clonidine3-F-DPPy732Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97065Alpha2BCLONEDHUMAN[3H]Clonidine3-F-DPPy129Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97066Alpha2CCLONEDHUMAN[3H]Clonidine3-F-DPPy333Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97067Beta1CLONEDHUMAN[125I]Iodopindolol3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97068Beta2CLONEDHUMAN3-F-DPPy[125I]Iodopindolol>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97069Beta3CLONEDHUMAN[125I]Iodopindolol3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97070D1CLONEDHUMAN[3H]SCH233903-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97071D2CLONEDHUMAN[3H]N-methylspiperone3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97072D3CLONEDHUMAN[3H]N-methylspiperone3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97073D4CLONEDHUMAN[3H]N-methylspiperone3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97074D5CLONEDHUMAN[3H]SCH233903-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97075DATCLONEDHUMAN[3H]WIN354283-F-DPPy12Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97076DORCLONEDHUMAN[3H]DADLE3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97077GABAABRAINRAT[3H]-Muscimol3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 29, 2025
97078H1CLONEDHUMAN[3H]Pyrilamine3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
970795-HT1DCLONEDHUMAN[3H]Tiotidine3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97080H3CLONEDHUMAN[3H]-alpha-methylhistamine3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97081H4CLONEDHUMAN[3H]Histamine3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97082KORCLONEDHUMAN[3H]U695933-F-DPPy1583Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97083M1CLONEDHUMAN[3H]QNB3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97084M2CLONEDHUMAN[3H]QNB3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97085M3CLONEDHUMAN[3H]QNB3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97086M5CLONEDHUMAN[3H]QNB3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97087MORCLONEDHUMAN[3H]DAMGO3-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97088NETCLONEDHUMAN[3H]Nisoxetine3-F-DPPy192Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97089PBRCLONEDHUMAN[3H]PK111953-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97090SERTCLONEDHUMAN[3H]Citalopram3-F-DPPy1202Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97091Sigma 1CLONEDHUMAN[3H]Pentazocine3-F-DPPy193Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97092Sigma 2CLONEDHUMAN[3H]DTG3-F-DPPy1934Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97093NMDAFOREBRAINRAT[3H]MK-8014-F-DPPy953Wallach J et al 2019Jan 15, 2025Jan 28, 2025
970945-HT1ACLONEDHUMAN[3H]8-OH-DPAT4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970955-HT1BCLONEDHUMAN[3H]GR1275434-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970965-HT1DCLONEDHUMAN[3H]GR1275434-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970975-HT1ECLONEDHUMAN[3H]5-HT4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970985-HT2CCLONEDHUMAN[3H]mesulergine4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
970995-HT3CLONEDHUMAN[3H]LY2785844-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97100Alpha1ACLONEDHUMAN[3H]prazosin4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97101Alpha1BCLONEDHUMAN[3H]prazosin4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97102Alpha1DCLONEDHUMAN[3H]prazosin4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97103Alpha2ACLONEDHUMAN[3H]Clonidine4-F-DPPy1401Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97104Alpha2BCLONEDHUMAN[3H]Clonidine4-F-DPPy1242Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97105Beta2CLONEDHUMAN[125I]Iodopindolol4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97106Beta3CLONEDHUMAN[125I]Iodopindolol4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97107D1CLONEDHUMAN[3H]SCH233904-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97108D2CLONEDHUMAN[3H]N-methylspiperone4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97109D3CLONEDHUMAN[3H]N-methylspiperone4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97110D4CLONEDHUMAN[3H]N-methylspiperone4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97111D5CLONEDHUMAN[3H]SCH233904-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97112DATCLONEDHUMAN[3H]WIN354284-F-DPPy140Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97113DORCLONEDHUMAN[3H]DADLE4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97114GABAABRAINRAT[3H]-Muscimol4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 29, 2025
97115H1CLONEDHUMAN[3H]Pyrilamine4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
971165-HT1DCLONEDHUMAN[3H]Tiotidine4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97117H3CLONEDHUMAN[3H]-alpha-methylhistamine4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97118H4CLONEDHUMAN[3H]Histamine4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97119KORCLONEDHUMAN[3H]U695934-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97120M1CLONEDHUMAN[3H]QNB4-F-DPPy1900Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97121M2CLONEDHUMAN[3H]QNB4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97122M3CLONEDHUMAN[3H]QNB4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97123M5CLONEDHUMAN[3H]QNB4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97124MORCLONEDHUMAN[3H]DAMGO4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97125NETCLONEDHUMAN[3H]Nisoxetine4-F-DPPy249Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97126PBRCLONEDHUMAN[3H]PK111954-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97127SERTCLONEDHUMAN[3H]Citalopram4-F-DPPy681Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97128Sigma 1CLONEDHUMAN[3H]Pentazocine4-F-DPPy386Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97129Sigma 2CLONEDHUMAN[3H]DTG4-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97130NMDAFOREBRAINRAT[3H]MK-8012′′-F-DPPy610Wallach J et al 2019Jan 15, 2025Jan 28, 2025
971315-HT1ACLONEDHUMAN[3H]8-OH-DPAT2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971325-HT1BCLONEDHUMAN[3H]GR1275432′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971335-HT1DCLONEDHUMAN[3H]GR1275432′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971345-HT1ECLONEDHUMAN[3H]5-HT2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971355-HT2ACLONEDHUMAN[3H]ketanserin2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971365-HT2CCLONEDHUMAN[3H]mesulergine2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971375-HT3CLONEDHUMAN[3H]LY2785842′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97138Alpha1ACLONEDHUMAN[3H]prazosin2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97139Alpha1BCLONEDHUMAN[3H]prazosin2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97140Alpha1DCLONEDHUMAN[3H]prazosin2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97141Alpha2ACLONEDHUMAN[3H]Clonidine2′′-F-DPPy307Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97142Alpha2BCLONEDHUMAN[3H]Clonidine2′′-F-DPPy89Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97143Alpha2CCLONEDHUMAN[3H]Clonidine2′′-F-DPPy214Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97144Beta1CLONEDHUMAN[125I]Iodopindolol2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97145Beta2CLONEDHUMAN[125I]Iodopindolol2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97146Beta3CLONEDHUMAN[125I]Iodopindolol2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97147D1CLONEDHUMAN[3H]SCH233902′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97148D2CLONEDHUMAN[3H]N-methylspiperone2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97149D3CLONEDHUMAN[3H]N-methylspiperone2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97150D4CLONEDHUMAN[3H]N-methylspiperone2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97151D5CLONEDHUMAN[3H]SCH233902′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97152DATCLONEDHUMAN[3H]WIN354282′′-F-DPPy85Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97153DORCLONEDHUMAN[3H]DADLE2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97154GABAABRAINRAT[3H]-Muscimol2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 29, 2025
97155H1CLONEDHUMAN[3H]Pyrilamine2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
971565-HT1DCLONEDHUMAN[3H]Tiotidine2′′-F-DPPy2194Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97157H3CLONEDHUMAN[3H]-alpha-methylhistamine2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97158H4CLONEDHUMAN[3H]Histamine2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97159KORCLONEDHUMAN[3H]U695932′′-F-DPPy642Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97160M1CLONEDHUMAN[3H]QNB2′′-F-DPPy1660Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97161M2CLONEDHUMAN[3H]QNB2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97162M4CLONEDHUMAN[3H]QNB2′′-F-DPPy576Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97163M5CLONEDHUMAN[3H]QNB2′′-F-DPPy489Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97164MORCLONEDHUMAN[3H]DAMGO2′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97165NETCLONEDHUMAN[3H]Nisoxetine2′′-F-DPPy215Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97166PBRCLONEDHUMAN[3H]PK111952′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97167SERTCLONEDHUMAN[3H]Citalopram2′′-F-DPPy661Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97168Sigma 1CLONEDHUMAN[3H]Pentazocine2′′-F-DPPy146Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97169Sigma 2CLONEDHUMAN[3H]DTG2′′-F-DPPy712Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97170NMDACLONEDHUMAN[3H]MK-8013′′-F-DPPy262Wallach J et al 2019Jan 15, 2025Jan 28, 2025
971715-HT1ACLONEDHUMAN[3H]8-OH-DPAT3′′-F-DPPy534Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971725-HT1BCLONEDHUMAN[3H]GR1275433′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971735-HT1DCLONEDHUMAN[3H]GR1275433′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971745-HT1ECLONEDHUMAN[3H]5-HT3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971755-HT2ACLONEDHUMAN[3H]ketanserin3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971765-HT2CCLONEDHUMAN[3H]mesulergine3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
971775-HT3CLONEDHUMAN[3H]LY2785843′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97178Alpha1ACLONEDHUMAN[3H]prazosin3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97179Alpha1BCLONEDHUMAN[3H]prazosin3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97180Alpha1DCLONEDHUMAN[3H]prazosin3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97181Alpha2ACLONEDHUMAN[3H]Clonidine3′′-F-DPPy915Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97182Alpha2BCLONEDHUMAN[3H]Clonidine3′′-F-DPPy307Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97183Alpha2CCLONEDHUMAN[3H]Clonidine3′′-F-DPPy1159Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97184Beta1CLONEDHUMAN[125I]Iodopindolol3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97185Beta2CLONEDHUMAN[125I]Iodopindolol3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97186Beta3CLONEDHUMAN[125I]Iodopindolol3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97187D1CLONEDHUMAN[3H]SCH233903′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97188D2CLONEDHUMAN3′′-F-DPPy[3H]N-methylspiperone>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97189D3CLONEDHUMAN[3H]N-methylspiperone3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97190D4CLONEDHUMAN[3H]N-methylspiperone3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97191D5CLONEDHUMAN[3H]SCH233903′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97192DATCLONEDHUMAN[3H]WIN354283′′-F-DPPy103Wallach J et al 2019Jan 15, 2025Jan 15, 2025
97193DORCLONEDHUMAN[3H]DADLE3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97194GABAABRAINRAT[3H]-Muscimol3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 29, 2025
97195H1CLONEDHUMAN[3H]Pyrilamine3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
971965-HT1DCLONEDHUMAN[3H]Tiotidine3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97197H3CLONEDHUMAN[3H]-alpha-methylhistamine3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97198H4CLONEDHUMAN[3H]Histamine3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97199KORCLONEDHUMAN[3H]U695933′′-F-DPPy1435Wallach J et al 2019Jan 15, 2025Jan 28, 2025
97200M1CLONEDHUMAN[3H]QNB3′′-F-DPPy>10000Wallach J et al 2019Jan 15, 2025Jan 15, 2025
972015-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl5200Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972025-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl9.5Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972035-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl740Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972045-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl5.3Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972055-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl4.2Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972065-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl1Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972075-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine18Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972085-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine26Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972095-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamineN,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine  63Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972105-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3-methoxyphenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine  28Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972115-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl117Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972125-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl84Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972135-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl160Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972145-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl16Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972155-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine180Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972165-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl400Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972175-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl>10000Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972185-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl910Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972195-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamineN,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine22Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972205-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine5.2Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972215-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl97Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972225-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl450Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972235-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine240Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972245-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine600Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972255-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine33Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972265-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl2600Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972275-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl71Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972285-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine180Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972295-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine17Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972305-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl390Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972315-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine5.9Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972325-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine190Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972335-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl34Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972345-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine740Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972355-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine5.3Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972365-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl51Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972375-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamineAS-1912Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972385-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(R)-8-OH-DPAT48Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972395-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamine(S)-8-OH-DPAT1000Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972405-HT7CLONEDHUMAN[3H]-5-carboxamidotryptamineBUSPIRONE840Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972415-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl1100Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972425-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-N,N-dimethyl-5-phenyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl6.3Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972435-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl1000Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972445-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-(2-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl4Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972455-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl14Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972465-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-(2-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl7.5Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972475-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine23Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972485-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine82Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972495-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamineN,N-dimethyl-5-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydronaphthalen-2-amine  180Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972505-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl73Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972515-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl30Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972525-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl19Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972535-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(4-chlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl190Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972545-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(2-chloro-4-fluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amineHCl33Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972555-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3,5-difluorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine230Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972565-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(3,5-dichlorophenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl2200Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972575-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl>10000Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972585-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(3,5-bis(trifluoromethyl)phenyl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl2230Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972595-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamineN,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine130Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972605-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-N,N-dimethyl-5,6,7,8-tetrahydro-[1,1′-binaphthalen]-6-amine64Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972615-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(isoquinolin-4-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl650Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972625-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-(anthracen-9-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl1400Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972635-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine5-cyclopentyl-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine98Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972645-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine550Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972655-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-N,N-dimethyl-5-(1-methyl-1H-pyrrol-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine24Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972665-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl5600Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972675-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(furan-2-yl)-N,N-dimethyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl33Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972685-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine150Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972695-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-N,N-dimethyl-5-(thiophen-2-yl)-1,2,3,4-tetrahydronaphthalen-2-amine4.5Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972705-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2R)-5-(2-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl130Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972715-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine0.64Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972725-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2R)-5-(2′-chlorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine210Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972735-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(2S)-5-phenyl-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine HCl5.9Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972745-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(+)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine92Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972755-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(-)-5-(2-fluorophenyl)-N,N-dipropyl-1,2,3,4-tetrahydronaphthalen-2-amine1.8Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972765-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine1-(5-(2-fluorophenyl)-1,2,3,4-tetrahydronaphthalen-2-yl)pyrrolidine HCl1.3Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972775-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamineAS-19240Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972785-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(R)-8-OH-DPAT7.1Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972795-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamine(S)-8-OH-DPAT7.6Perry CK et al 2020Jan 15, 2025Jan 15, 2025
972805-HT1ACLONEDHUMAN[3H]-5-carboxamidotryptamineBUSPIRONE50Perry CK et al 2020Jan 15, 2025Jan 15, 2025
97281MORCLONEDHUMAN[3H]diprenorphineSRI-221387.55Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97282MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol23.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97283MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o138Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97284MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol2.33Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97285MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol171Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97286MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol370Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97287MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o235Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97288MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o24.4Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97289MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o191Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97290MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol29.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97291MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o135Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97292MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o249Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97293MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol61.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97294MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol91.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97295MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol148Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97296MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol12.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97297MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol6.97Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97298MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol15.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97299MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol4.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97300MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol56.4Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97301MORCLONEDHUMAN[3H]diprenorphineN-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide141Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97302MORCLONEDHUMAN[3H]diprenorphineN-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide337Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97303MORCLONEDHUMAN[3H]diprenorphineN-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide159Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97304MORCLONEDHUMAN[3H]diprenorphineNALOXONE59.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97305MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o14.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97306MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o105Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97307MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol82.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97308MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol47.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97309MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol1.05Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97310MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol10.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97311MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol66.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97312MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol47.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97313MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol88.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97314MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol121Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97315MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o3.79Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97316MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o99.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97317MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol3.18Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97318MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol5.37Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97319MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o819Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97320MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol799Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97321MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol3.96Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97322MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol3.82Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97323MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol70.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97324MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol95.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97325MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol5.99Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97326MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol92.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97327MORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol499Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97328DORCLONEDHUMAN[3H]diprenorphineSRI-221382.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97329DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol19.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97330DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o20.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97331DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol3.42Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97332DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol53.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97333DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol7.52Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97334DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o97.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97335DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o26.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97336DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o34.4Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97337DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol3.78Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97338DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o64.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97339DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o93.4Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97340DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol29.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97341DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol48Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97342DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol30.6Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97343DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol8.37Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97344DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol69.6Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97345DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol68.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97346DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol53.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97347DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol14Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97348DORCLONEDHUMAN[3H]diprenorphineN-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide3333Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97349DORCLONEDHUMAN[3H]diprenorphineN-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide3333Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97350DORCLONEDHUMAN[3H]diprenorphineN-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide394Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97351DORCLONEDHUMAN[3H]diprenorphineNALOXONE98.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97352DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o0.169Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97353DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o6.52Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97354DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol30.6Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97355DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol6.43Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97356DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol63.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97357DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol3.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97358DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol22.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97359DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol5.18Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97360DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol40.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97361DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol257Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97362DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o7.96Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97363DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o64.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97364DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol8.12Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97365DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol5.24Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97366DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o172Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97367DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol32.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97368DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol5.89Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97369DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol29.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97370DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol11Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97371DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol12.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97372DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol64.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97373DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol14.6Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97374DORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol7.48Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97375KORCLONEDHUMAN[3H]diprenorphineSRI-2213860.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97376KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol132Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97377KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Bromophenyl)-7-(cyclopropylmethyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o75.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97378KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol6.69Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97379KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol35.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97380KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3,4-difluorophenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol71.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97381KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(o-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o152Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97382KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(m-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o17.6Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97383KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(p-tolyl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o102Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97384KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-fluoro-2-methyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol129Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97385KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-cyclopropyl-phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o175Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97386KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2,6-dimethylphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o134Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97387KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol126Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97388KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol103Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97389KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-methoxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol140Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97390KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-hydroxyphenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol18.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97391KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol7.96Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97392KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol11.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97393KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(4-(dimethylamino)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol6.18Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97394KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-((dimethylamino)methyl)phenyl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido-[3,4-g]quinolin-1-ol22.7Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97395KORCLONEDHUMAN[3H]diprenorphineN-(2-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide13.5Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97396KORCLONEDHUMAN[3H]diprenorphineN-(3-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide608Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97397KORCLONEDHUMAN[3H]diprenorphineN-(4-((4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-1-hydroxy-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-11-yl)phenyl)-acetamide15.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97398KORCLONEDHUMAN[3H]diprenorphineU50,48831.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97399KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrrol-1-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o13.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97400KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o19.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97401KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-3-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol27.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97402KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyridin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol15.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97403KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methylpyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol0.51Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97404KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(2-methoxypyridin-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol6.62Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97405KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol30.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97406KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrimidin-5-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol24.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97407KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(pyrazin-2-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol19.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97408KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-phenylpropoxy)-11-(1H-pyrazol-4-yl)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol29.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97409KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(1-methyl-1H-pyrazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o8.4Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97410KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(3-methylisoxazol-4-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o23.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97411KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-(5-methyl-1,3,4-oxadiazol-2-yl)-8a-(3-phenylpropoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol14.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97412KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol10.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97413KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(2-phenoxyethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-o21.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97414KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-11-(4-Chlorophenyl)-7-(cyclopropylmethyl)-8a-(quinolin-2-ylmethoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol31Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97415KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-3-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol5.3Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97416KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(pyridin-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol21.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97417KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-8a-(3-(4-fluorophenyl)propoxy)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol60.2Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97418KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-8a-(3-Cyclohexylpropoxy)-7-(cyclopropylmethyl)-11-phenyl-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol57.9Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97419KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(3-(tetrahydro-2H-pyran-4-yl)propoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]pyrido[3,4-g]quinolin-1-ol24.8Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97420KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-(4-phenylbutoxy)-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro-[3,2-h]pyrido[3,4-g]quinolin-1-ol57.1Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97421KORCLONEDHUMAN[3H]diprenorphine(4bS,8R,8aS,13bR)-7-(Cyclopropylmethyl)-11-phenyl-8a-propoxy-6,7,8,8a,9,13b-hexahydro-5H-4,8-methanobenzofuro[3,2-h]-pyrido[3,4-g]quinolin-1-ol252Vekariya RH et al 2020Jan 15, 2025Jan 28, 2025
97422A1CLONEDHUMAN[3H]DPCPXISAM-1411000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97423A1CLONEDHUMAN[3H]DPCPXISAM-1421000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97424A1CLONEDHUMAN[3H]DPCPXethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97425A1CLONEDHUMAN[3H]DPCPXpropan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97426A1CLONEDHUMAN[3H]DPCPXISAM-1341000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97427A1CLONEDHUMAN[3H]DPCPXISAM-1401000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97428A1CLONEDHUMAN[3H]DPCPXethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97429A1CLONEDHUMAN[3H]DPCPXDPCPX2.2Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97430A1CLONEDHUMAN[3H]DPCPXZM241385683Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97431A1CLONEDHUMAN[3H]DPCPXEthyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97432A1CLONEDHUMAN[3H]DPCPXIsopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97433A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97434A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97435A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97436A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97437A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97438A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97439A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97440A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97441A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97442A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97443A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97444A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97445A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97446A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97447A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97448A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97449A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97450A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97451A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate14.8Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97452A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate8.3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97453A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97454A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97455A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate20.2Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97456A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97457A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97458A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97459A1CLONEDHUMAN[3H]DPCPX±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97460A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97461A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97462A1CLONEDHUMAN[3H]DPCPX(±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97463A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97464A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97465A1CLONEDHUMAN[3H]DPCPX±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97466A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97467A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97468A1CLONEDHUMAN[3H]DPCPX±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97469A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate233Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97470A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate301Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97471A1CLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97472A1CLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97473A2ACLONEDHUMAN[3H]ZM-241385ISAM-1411000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97474A2ACLONEDHUMAN[3H]ZM-241385ISAM-1421000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97475A2ACLONEDHUMAN[3H]ZM-241385ethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97476A2ACLONEDHUMAN[3H]ZM-241385propan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97477A2ACLONEDHUMAN[3H]ZM-241385ISAM-1341000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97478A2ACLONEDHUMAN[3H]ZM-241385ISAM-1401000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97479A2ACLONEDHUMAN[3H]ZM-241385ethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97480A2ACLONEDHUMANLeucyl-3H-NCDPCPX157Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97481A2ACLONEDHUMAN[3H]ZM-241385ZM2413851.9Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97482A2ACLONEDHUMAN[3H]ZM-241385Ethyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97483A2ACLONEDHUMAN[3H]ZM-241385Isopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97484A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97485A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97486A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97487A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97488A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97489A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97490A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97491A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97492A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97493A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97494A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97495A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97496A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97497A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97498A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97499A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97500A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97501A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97502A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97503A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97504A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97505A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97506A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97507A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97508A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate2Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97509A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97510A2ACLONEDHUMAN[3H]ZM-241385±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97511A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97512A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate5Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97513A2ACLONEDHUMAN[3H]ZM-241385(±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97514A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97515A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97516A2ACLONEDHUMAN[3H]ZM-241385±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97517A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97518A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97519A2ACLONEDHUMAN[3H]ZM-241385±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97520A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate282Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97521A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97522A2ACLONEDHUMAN[3H]ZM-241385(±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97523A2ACLONEDHUMAN[3H]ZM-241385(±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97524A2BCLONEDHUMAN[3H]DPCPXISAM-14120.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97525A2BCLONEDHUMAN[3H]DPCPXISAM-14211.4Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97526A2BCLONEDHUMAN[3H]DPCPXethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate29.71Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97527A2BCLONEDHUMAN[3H]DPCPXpropan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  29.34Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97528A2BCLONEDHUMAN[3H]DPCPXISAM-13412.03Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97529A2BCLONEDHUMAN[3H]DPCPXISAM-1403.49Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97530A2BCLONEDHUMAN[3H]DPCPXethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate484.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97531A2BCLONEDHUMAN[3H]DPCPXpropan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  371.2Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97532A2BCLONEDHUMAN[3H]DPCPXDPCPX73.24Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97533A2BCLONEDHUMAN[3H]DPCPXZM24138565.7Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97534A2BCLONEDHUMAN[3H]DPCPXEthyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97535A2BCLONEDHUMAN[3H]DPCPXIsopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97536A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97537A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97538A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97539A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97540A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate449.3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97541A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate517.1Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97542A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate49.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97543A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate31.3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97544A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97545A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97546A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (789Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97547A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate721Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97548A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate707Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97549A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1104Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97550A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate23.4Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97551A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate29.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97552A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97553A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate278Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97554A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate92.6Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97555A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate340Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97556A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate714Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97557A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1031Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97558A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate98.7Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97559A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate175Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97560A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate769Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97561A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate708Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97562A2BCLONEDHUMAN[3H]DPCPX±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate388Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97563A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate753Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97564A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate402Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97565A2BCLONEDHUMAN[3H]DPCPX(±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97566A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate8.1Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97567A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate43.41Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97568A2BCLONEDHUMAN[3H]DPCPX±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97569A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97570A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97571A2BCLONEDHUMAN[3H]DPCPX±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97572A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate508Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97573A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97574A2BCLONEDHUMAN[3H]DPCPX(±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate215Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97575A2BCLONEDHUMAN[3H]DPCPX(±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate68.3Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97576A3CLONEDHUMAN[3H]NECAISAM-1411000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97577A3CLONEDHUMAN[3H]NECAISAM-1421000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97578A3CLONEDHUMAN[3H]NECAethyl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97579A3CLONEDHUMAN[3H]NECApropan-2-yl 2-methyl-4-thiophen-3-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate  1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97580A3CLONEDHUMAN[3H]NECAISAM-1341000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97581A3CLONEDHUMAN[3H]NECAISAM-1401000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97582A3CLONEDHUMAN[3H]NECAethyl 2-methyl-4-thiophen-2-yl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97583A3CLONEDHUMAN[3H]NECADPCPX1722Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97584A3CLONEDHUMAN[3H]NECAZM241385863Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97585A3CLONEDHUMAN[3H]NECAEthyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97586A3CLONEDHUMAN[3H]NECAIsopropyl 2-Methyl-1,4-dihydrobenzo[4,5]imidazo[1,2-a]-pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97587A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97588A3CLONEDHUMAN[3H]NECA(±) Isopropyl 4-Cyclopentyl-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97589A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimi-dine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97590A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-phenyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97591A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97592A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(1H-pyrrol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97593A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97594A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(1H-pyrrol-2-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97595A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97596A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(5-methylfuran-2-yl)-1,4-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97597A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate (1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97598A3CLONEDHUMAN[3H]NECA(±) Isopropyl 4-(Isoxazol-3-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97599A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97600A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(1H-pyrazol-3-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97601A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97602A3CLONEDHUMAN[3H]NECA(±) Isopropyl 4-(Isoxazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97603A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97604A3CLONEDHUMAN[3H]NECA(±) Isopropyl 4-(Isothiazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97605A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97606A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(1H-pyrazol-4-yl)-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97607A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97608A3CLONEDHUMAN[3H]NECA(±) Isopropyl 4-(Isoxazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97609A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97610A3CLONEDHUMAN[3H]NECA(±) Isopropyl 4-(Isothiazol-5-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97611A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97612A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(oxazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97613A3CLONEDHUMAN[3H]NECA±) Ethyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97614A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(thiazol-2-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97615A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97616A3CLONEDHUMAN[3H]NECA(±)Isopropyl4-(1H-Imidazol-2-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97617A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97618A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(oxazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97619A3CLONEDHUMAN[3H]NECA±) Ethyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97620A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(thiazol-4-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97621A3CLONEDHUMAN[3H]NECA(±) Ethyl 4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97622A3CLONEDHUMAN[3H]NECA±)Isopropyl4-(1H-Imidazol-4-yl)-2-methyl-1,4-dihydrobenzo[4,5]imidazo [1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97623A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate418Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97624A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(oxazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97625A3CLONEDHUMAN[3H]NECA(±) Ethyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo[4,5]-imidazo[1,2-a]pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97626A3CLONEDHUMAN[3H]NECA(±) Isopropyl 2-Methyl-4-(thiazol-5-yl)-1,4-dihydrobenzo-[4,5]imidazo[1,2-a] pyrimidine-3-carboxylate1000Mallo-Abreu A et al 2020Jan 15, 2025Jan 15, 2025
97627SST1CLONEDHUMAN125I-LTT-SST-28Somatostatin-140.4Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97628SST2CLONEDHUMAN125I-LTT-SST-28Somatostatin-140.04Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97629SST3CLONEDHUMAN125I-LTT-SST-28Somatostatin-140.7Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97630SST4CLONEDHUMAN125I-LTT-SST-28Somatostatin-141.7Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97631SST5CLONEDHUMAN125I-LTT-SST-28Somatostatin-142.3Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97632SST1CLONEDHUMAN125I-LTT-SST-28L-363,3775664Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97633SST2CLONEDHUMAN125I-LTT-SST-28L-363,3770.5Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97634SST3CLONEDHUMAN125I-LTT-SST-28L-363,3773072Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97635SST4CLONEDHUMAN125I-LTT-SST-28L-363,377>10000Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97636SST5CLONEDHUMAN125I-LTT-SST-28L-363,3772009Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97637SST1CLONEDHUMAN125I-LTT-SST-28L-797,5911.4Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97638SST2CLONEDHUMAN125I-LTT-SST-28L-797,5911875Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97639SST3CLONEDHUMAN125I-LTT-SST-28L-797,5912240Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97640SST4CLONEDHUMAN125I-LTT-SST-28L-797,591170Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97641SST5CLONEDHUMAN125I-LTT-SST-28L-797,5913600Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97642SST1CLONEDHUMAN125I-LTT-SST-28L-779,9762760Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97643SST2CLONEDHUMAN125I-LTT-SST-28L-779,9760.05Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97644SST3CLONEDHUMAN125I-LTT-SST-28L-779,976729Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97645SST4CLONEDHUMAN125I-LTT-SST-28L-779,976310Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97646SST5CLONEDHUMAN125I-LTT-SST-28L-779,9764260Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97647SST1CLONEDHUMAN125I-LTT-SST-28L-796,7781255Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97648SST2CLONEDHUMAN125I-LTT-SST-28L-796,778>10000Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97649SST3CLONEDHUMAN125I-LTT-SST-28L-796,77824Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97650SST4CLONEDHUMAN125I-LTT-SST-28L-796,7788650Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97651SST5CLONEDHUMAN125I-LTT-SST-28L-796,7781200Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97652SST1CLONEDHUMAN125I-LTT-SST-28L-803,087199Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97653SST2CLONEDHUMAN125I-LTT-SST-28L-803,0874720Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97654SST3CLONEDHUMAN125I-LTT-SST-28L-803,0871280Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97655SST4CLONEDHUMAN125I-LTT-SST-28L-803,0870.7Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97656SST5CLONEDHUMAN125I-LTT-SST-28L-803,0873880Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97657SST1CLONEDHUMAN125I-LTT-SST-28L-817,8183.3Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97658SST2CLONEDHUMAN125I-LTT-SST-28L-817,81852Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97659SST3CLONEDHUMAN125I-LTT-SST-28L-817,81864Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97660SST4CLONEDHUMAN125I-LTT-SST-28L-817,81882Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97661SST5CLONEDHUMAN125I-LTT-SST-28L-817,8180.4Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97662SST1CLONEDHUMANFunctionalL-797,5913Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97663SST2CLONEDHUMANFunctionalL-779,9760.05Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97664SST4CLONEDHUMANFunctionalL-803,0870.2Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97665SST5CLONEDHUMANFunctionalL-817,8181.3Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97666SST3CLONEDHUMANFunctionalL-796,77818Rohrer SP, et.al., 1998Jan 15, 2025Jan 15, 2025
97667KORCORTICAL MEMBRANESRAT3H-flumazenil4-quinolone122Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97668KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-ethyl-4-quinolone20Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97669KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-propoxycarbonyl-4-quinolone1.8Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97670KORCORTICAL MEMBRANESRAT3H-flumazenil3-Butoxycarbonyl-6-ethyl-4-quinolone13Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97671KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone28Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97672KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(2-methylbutoxycarbonyl)-4-quinolone28Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97673KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-pentoxycarbonyl-4-quinolone35Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97674KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(2-ethylbutoxycarbonyl)-4-quinolone92Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97675KORCORTICAL MEMBRANESRAT3H-flumazenil3-Cyclopentoxycarbonyl-6-ethyl-4-quinolone19Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97676KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-i-propoxycarbonyl-4-quinolone214Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97677KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(4-methyl-2-pentoxycarbonyl)-4-quinolone295Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97678KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-pentoxycarbonyl)-4-quinolone2600Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97679KORCORTICAL MEMBRANESRAT3H-flumazenil3-Carboxy-6-ethyl-4-quinolone208Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97680KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-4-quinolone78Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97681KORCORTICAL MEMBRANESRAT3H-flumazenil3-Butoxycarbonyl-4-quinolone54Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97682KORCORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-4-quinolone16Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97683KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-propyl-4-quinolone17Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97684KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-i-propyl-4-quinolone15Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97685KORCORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-ethoxycarbonyl-4-quinolone1.4Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97686KORCORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-propoxycarbonyl-4-quinolone0.17Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97687KORCORTICAL MEMBRANESRAT3H-flumazenil3-Ethoxycarbonyl-6-ethyl-2-methyl-4-quinolone6850Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97688KORCORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-2-methyl-4-quinolone4200Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97689KORCORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-propylaminocarbonyl-4-quinolone0.26Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97690KORCORTICAL MEMBRANESRAT3H-flumazenil3-Butylaminocarbonyl-6-ethyl-4-quinolone0.54Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97691KORCORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-propylaminocarbonyl-4-quinolone0.048Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97692KORCORTICAL MEMBRANESRAT3H-flumazenilPropyl 2-methyl-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate870Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97693KORCORTICAL MEMBRANESRAT3H-flumazenilEthyl 7-Oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate>10000Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97694KORCORTICAL MEMBRANESRAT3H-flumazenilPropyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylate7130Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97695GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone4.1Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97696GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone89Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
97697GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-4-quinolone26Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
97698GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Bromo-3-ethoxycarbonyl-4-quinolone14Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97699GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-ethoxycarbonyl-4-quinolone0.27Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97700GABAACORTICAL MEMBRANESRAT3H-flumazenil6-Benzyl-3-ethoxycarbonyl-4-quinolone7.2Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
97701GABAACORTICAL MEMBRANESRAT3H-flumazenilDIAZEPAM12Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97702GABAACORTICAL MEMBRANESRAT3H-flumazenilDIAZEPAM14Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
97703GABAACORTICAL MEMBRANESRAT3H-flumazenilZolpidem1850Lager, E. et al., 2006Jan 15, 2025Jan 28, 2025
97704GABAACORTICAL MEMBRANESRAT3H-flumazenilZolpidem53Lager, E. et al., 2006Jan 15, 2025Jan 27, 2025
97705L1210 cellsMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt1800Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97706L1210 cellsMOUSEFunctionalN1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt700Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97707L1210 cellsMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt400Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97708L1210 cellsMOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt300Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97709L1210 cellsMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt1300Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97710L1210 cellsMOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt400Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97711L1210 cellsMOUSEFunctionalN-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97712L1210 + DFMOMOUSEFunctionalN-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97713L1210 + DFMOMOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt300Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97714L1210 + DFMOMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt700Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97715L1210 + DFMOMOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt150Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97716L1210 + DFMOMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt200Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97717L1210 + DFMOMOUSEFunctionalN1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt300Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97718L1210 + DFMOMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt1400Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97719L1210 cellsMOUSE14C-spermidineN-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97720L1210 cellsMOUSE14C-spermidineN1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt2500Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97721L1210 cellsMOUSE14C-spermidineN-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt6200Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97722L1210 cellsMOUSE14C-spermidineN-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt1800Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97723L1210 cellsMOUSE14C-spermidineN-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt5000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97724L1210 cellsMOUSE14C-spermidineN-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt1700Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97725L1210 cellsMOUSE14C-spermidineN-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97726CHO-MGMOUSEFunctionalN-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97727C.H.O.MOUSEFunctionalN-(Anthracen-9-ylmethyl)butylamine, Monohydrochloride>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97728CHO-MGMOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97729C.H.O.MOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt1500Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97730C.H.O.MOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt4100Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97731CHO-MGMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpentane-1,5-diamine trihydrochloride salt>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97732CHO-MGMOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt>10000Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97733C.H.O.MOUSEFunctionalN-(4-Aminobutyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt450Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97734C.H.O.MOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt400Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97735CHO-MGMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylbutane-1,4-diamine trihydrochloride salt9500Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97736CHO-MGMOUSEFunctionalN1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt8800Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97737C.H.O.MOUSEFunctionalN1-{3-[(Anthracen-9-ylmethyl)amino]propyl}butane-1,4-diamine trihydrochloride salt2500Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97738C.H.O.MOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt1900Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97739CHO-MGMOUSEFunctionalN-(3-Aminopropyl)-N-anthracen-9-ylmethylpropane-1,3-diamine trihydrochloride salt3400Wang C, et al., 2003Jan 15, 2025Jan 15, 2025
97740Y5CLONEDHUMAN125I-PYYFMS5864.3Kakui, N. et al., 2006Jan 15, 2025Jan 29, 2025
97741Y5CLONEDHUMAN125I-PYYL-152,80425Kakui, N. et al., 2006Jan 15, 2025Jan 29, 2025
97742Y5CLONEDHUMAN125I-PYYPYY1Kakui, N. et al., 2006Jan 15, 2025Jan 29, 2025
97743Y1CLONEDHUMAN125I-PYYPYY2Kakui, N. et al., 2006Jan 15, 2025Jan 15, 2025
97744Y1CLONEDHUMAN125I-PYYL-152,804>10000Kakui, N. et al., 2006Jan 15, 2025Jan 15, 2025
97745Y1CLONEDHUMAN125I-PYYFMS586>10000Kakui, N. et al., 2006Jan 15, 2025Jan 15, 2025
97746Y2CLONEDHUMAN125I-PYYFMS586>10000Kakui, N. et al., 2006Jan 15, 2025Jan 29, 2025
97747Y2CLONEDHUMAN125I-PYYL-152,804>10000Kakui, N. et al., 2006Jan 15, 2025Jan 29, 2025
97748Y2CLONEDHUMAN125I-PYYPYY2.1Kakui, N. et al., 2006Jan 15, 2025Jan 29, 2025