The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 96,001-97,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
98749D3CLONEDHUMAN125I-IABN1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperidine1098Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98750D2CLONEDHUMAN125I-IABN1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperidine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98751D2CLONEDHUMAN125I-IABN4,4-Dimethyl-1-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)- thio)propyl)piperidine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98752D3CLONEDHUMAN125I-IABN4,4-Dimethyl-1-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)- thio)propyl)piperidine631Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98753D3CLONEDHUMAN125I-IABN3-(2-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9- diazaspiro[5.5]undecane1145Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98754D2CLONEDHUMAN125I-IABN3-(2-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9- diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98755D2CLONEDHUMAN125I-IABN1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98756D3CLONEDHUMAN125I-IABN1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98757D1CLONEDHUMAN3H-SCH233903-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98758D5CLONEDHUMAN3H-SCH233903-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98759D2CLONEDHUMAN3H-N-Methylspiperone3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98760D3CLONEDHUMAN3H-N-Methylspiperone3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane94Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98761D4CLONEDHUMAN3H-N-Methylspiperone3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
987625-HT1ACLONEDHUMAN3H-WAY1006353-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane1297Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987635-HT1BCLONEDHUMAN3H-GR-1257433-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987645-HT1DCLONEDHUMAN3H-GR-1257433-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987655-HT1ECLONEDHUMAN3H-5-HT3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987665-HT2ACLONEDHUMAN3H-KETANSERIN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987675-HT2BCLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane2144Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987685-HT2CCLONEDHUMAN3H-MESULERGINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987695-HT3CLONEDHUMAN3H-GR656303-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987705-HT5ACLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987715-HT6CLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
987725-HT7CLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98773H1CLONEDHUMAN3H-PYRILAMINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane8Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
987745-HT1DCLONEDHUMAN125I-aminopotentidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane596Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98775H3CLONEDHUMAN3H-Alpha-methylhistamine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane509Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98776H4CLONEDHUMAN3H-Histamine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98777MORCLONEDHUMAN3H-DAMGO3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98778DORCLONEDHUMAN3H-DADLE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98779KORCLONEDHUMAN3H-U695933-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98780M1CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98781M2CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane52Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98782M3CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane514Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98783M4CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane590Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98784M5CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98785Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane2178Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98786Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane2173Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98787Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98788Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98789Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane1557Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98790nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98791nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98792nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98793nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane8523Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98794nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98795nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98796Beta 1CLONEDHUMAN125I-Pindolol3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98797Beta3CLONEDHUMAN125I-Pindolol3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98798Beta 2CLONEDHUMAN3H-CGP-121773-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98799DATCLONEDHUMAN3H-WIN 35,4283-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98800NETCLONEDHUMAN3H-Nisoxetine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane931Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98801SERTCLONEDHUMAN3H-CITALOPRAM3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane295Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98802KORCLONEDHUMAN3H-MUSCIMOL3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 27, 2025
98803D1CLONEDHUMAN3H-SCH233901-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98804D5CLONEDHUMAN3H-SCH233901-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine3016Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98805D2CLONEDHUMAN3H-N-Methylspiperone1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine577Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98806D3CLONEDHUMAN3H-N-Methylspiperone1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine6Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98807D4CLONEDHUMAN3H-N-Methylspiperone1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine721Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
988085-HT1ACLONEDHUMAN3H-WAY1006351-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine0.9Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988095-HT1BCLONEDHUMAN3H-GR-1257431-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine2032Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988105-HT1DCLONEDHUMAN3H-GR-1257431-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988115-HT1ECLONEDHUMAN3H-5HT1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988125-HT2ACLONEDHUMAN3H-KETANSERIN1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine1415Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988135-HT2BCLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine42Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988145-HT2CCLONEDHUMAN3H-MESULERGINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine159Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988155-HT3CLONEDHUMAN3H-GR-656301-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988165-HT5ACLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988175-HT7CLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988185-HT6CLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98819H1CLONEDHUMAN3H-PYRILAMINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine40Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
988205-HT1DCLONEDHUMAN125I-aminopotentidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine871Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98821H3CLONEDHUMAN3H-Alpha-methylhistamine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98822H4CLONEDHUMAN3H-Histamine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98823MORCLONEDHUMAN3H-DAMGO1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98824DORCLONEDHUMAN3H-DADLE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98825KORCLONEDHUMAN3H-U695931-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98826M1CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98827M2CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98828M3CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98829M4CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98830M5CLONEDHUMAN3H-QNB1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98831Alpha1ACLONEDHUMAN3H-PRAZOSIN1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine49Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98832Alpha1BCLONEDHUMAN3H-PRAZOSIN1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine94Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98833Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine221Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98834Alpha2BCLONEDHUMAN3H-RAUWOLSCINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine241Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98835Alpha2CCLONEDHUMAN3H-RAUWOLSCINE1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine433Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98836nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98837nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98838nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98839nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98840nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98841nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98842Beta 1CLONEDHUMAN125I-Pindolol1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98843Beta3CLONEDHUMAN125I-Pindolol1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98844Beta 2CLONEDHUMAN3H-CGP-121771-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98845DATCLONEDHUMAN3H-WIN 35,4281-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98846NETCLONEDHUMAN3H-Nisoxetine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98847SERTCLONEDHUMAN3H-Cimetidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98848GABAACLONEDHUMAN3H-MUSCIMOL1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98849D3CLONEDHUMAN125I-IABN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane12Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98850D3CLONEDHUMAN125I-IABN3-(2-Methoxyphenyl)-9-(3-((5-phenyl-4H-1,2,4-triazol-3-yl)thio)- propyl)-3,9-diazaspiro[5.5]undecane32.5Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98851D3CLONEDHUMAN125I-IABN3-(2,4-Dimethoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane112Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98852D3CLONEDHUMAN125I-IABNtert-Butyl 9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undec-7-ene3-carboxylate>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98853D2CLONEDHUMAN125I-IABNtert-Butyl 9-(2-methoxyphenyl)-3,9-diazaspiro[5.5]undec-7-ene3-carboxylate>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98854D3CLONEDHUMAN125I-IABN4-Methyl-3-phenyl-5-(propylthio)-4H-1,2,4-triazole>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98855D2CLONEDHUMAN125I-IABN4,4-Dimethyl-1-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)- thio)propyl)piperidine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98856D2CLONEDHUMAN125I-IABN3-(2-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9- diazaspiro[5.5]undecane225.74Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98857D2CLONEDHUMAN125I-IABN1-(3-((4-Methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)- piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98858D1CLONEDHUMAN3H-SCH233903-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98859D5CLONEDHUMAN3H-SCH233903-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98860D2CLONEDHUMAN3H-N-Methylspiperone3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98861D4CLONEDHUMAN3H-N-Methylspiperone3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98862D3CLONEDHUMAN3H-N-Methylspiperone3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane94Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
988635-HT1ACLONEDHUMAN3H-WAY1006353-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane1297Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988645-HT1BCLONEDHUMAN3H-GR-1257433-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988655-HT1DCLONEDHUMAN3H-GR-1257433-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988665-HT1ECLONEDHUMAN3H-5-HT3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988675-HT2ACLONEDHUMAN3H-KETANSERIN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988685-HT2BCLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane2144Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988695-HT2CCLONEDHUMAN3H-MESULERGINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988705-HT3CLONEDHUMAN3H-GR-656303-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988715-HT5ACLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988725-HT6CLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
988735-HT7CLONEDHUMAN3H-LSD3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98874H1CLONEDHUMAN3H-PYRILAMINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane8Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
988755-HT1DCLONEDHUMAN125I-iodoaminopotentidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane596Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98876H3CLONEDHUMAN3H-Alpha-methylhistamine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane509Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98877H4CLONEDHUMAN3H-Histamine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98878MORCLONEDHUMAN3H-DAMGO3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98879DORCLONEDHUMAN3H-DADLE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98880KORCLONEDHUMAN3H-U695933-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98881M1CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98882M5CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98883M2CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane52Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98884M3CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane514Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98885M4CLONEDHUMAN3H-QNB3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane590Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98886Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane2178Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98887Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane2173Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98888Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98889Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98890Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane1557Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98891nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98892nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98893nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98894nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane8523Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98895nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98896nAChRCLONEDHUMAN3H-Epibatidine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98897Beta 1CLONEDHUMAN125I-Pindolol3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98898Beta3CLONEDHUMAN125I-Pindolol3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98899Beta 2CLONEDHUMAN3H-CGP121773-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98900DATCLONEDHUMAN3H-WIN 35,4283-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98901NETCLONEDHUMAN3H-Nisoxetine3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane931Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98902SERTCLONEDHUMAN3H-CITALOPRAM3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane295Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98903KORCortical MembrainsRAT3H-MUSCIMOL3-(2-methoxyphenyl)-9-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)-3,9-diazaspiro[5.5]undecane>10000Reilly SW et al 2019Jan 15, 2025Jan 27, 2025
989045-HT1BCLONEDHUMAN3H-GR1257431-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine2032Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
989055-HT1DCLONEDHUMAN3H-GR1257431-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
989065-HT7CLONEDHUMAN3H-LSD1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine128Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
989075-HT1DCLONEDHUMAN125I-iodoaminopotentidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine871Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98908nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98909nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98910nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98911nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98912nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98913nAChRCLONEDHUMAN3H-Epibatidine1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 29, 2025
98914Beta 1CLONEDHUMAN125I-Iodopindolol1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 15, 2025
98915Beta3CLONEDHUMAN125I-Iodopindolol1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98916SERTCLONEDHUMAN3H-CITALOPRAM1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 28, 2025
98917KORCORTICAL MEMBRANESRAT3H-MUSCIMOL1-(2-methoxyphenyl)-4-(3-((4-methyl-5-phenyl-4H-1,2,4-triazol-3-yl)thio)propyl)piperazine>10000Reilly SW et al 2019Jan 15, 2025Jan 27, 2025
98918A1HEK293 cells? HUMAN[3H]N6-R-phenylisopropyladenosine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide432Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98919A1HEK293 cells? HUMAN[3H]N6-R-phenylisopropyladenosine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide369Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98920A1HEK293 cellsMOUSE[3H]N6-R-phenylisopropyladenosine(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide3260Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98921A1HEK293 cells? HUMAN[3H]N6-R-phenylisopropyladenosine(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide3980Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98922A2AHEK293 cells? HUMAN[3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide2460Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98923A2AHEK293 cells? HUMAN[3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide4620Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98924A2AHEK293 cells? HUMAN[3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5′-N-ethylcarboxamidoadenosine(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide838Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98925A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide2.3Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98926A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide1510Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98927A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide8.51Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98928A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4dihydroxy-N-methyltetrahydrofuran-2-carboxamide435Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98929A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide26.6Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98930A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide1200Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98931A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide0.28Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98932A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide85Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98933A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide10.6Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98934A3HEK293 cellsHUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide1.13Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98935A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5b]pyridin-3-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide0.896Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98936A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5b]pyridin-3-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide37Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98937A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(7-(Ethylamino)-5-((5-fluorothiophen-2-yl)ethynyl)-3H-imidazo[4,5b]pyridin-3-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide2.78Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98938A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-Nmethyluronamide(1S,2R,3S,4R,5S)-4-(7-(Ethylamino)-5-((5-fluorothiophen-2-yl)ethynyl)-3H-imidazo[4,5b]pyridin-3-yl)-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamide25Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98939A3HEK293 cells? HUMAN[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-NmethyluronamideEthyl (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate10.4Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98940A3HEK293 cellsMOUSE[125I]N6 -(4-amino-3-iodobenzyl)adenosine-5′-NmethyluronamideEthyl (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate625Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98941A1HEK293 cells? HUMAN[3 H]N6 -R-phenylisopropyladenosineEthyl (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate1670Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98942A1HEK293 cellsMOUSE[3 H]N6 -R-phenylisopropyladenosineEthyl (1S,2R,3S,4R,5S)-4-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9yl)-2,3-dihydroxybicyclo[3.1.0]hexane-1-carboxylate864Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989435-HT1ACLONEDHUMAN[3H]WAY100635C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989445-HT1BCLONEDHUMAN3H-GR-125743C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989455-HT1DCLONEDHUMAN3H-GR-125743C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989465-HT1ECLONEDHUMAN3H-GR-125743C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989475-HT1ECLONEDHUMAN3H-5HTC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989485-HT2ACLONEDHUMAN3H-KETANSERINC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989495-HT2BCLONEDHUMAN3H-LSDC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989505-HT2CCLONEDHUMAN3H-MESULERGINEC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989515-HT3CLONEDHUMAN3H-GR-65630C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989525-HT5ACLONEDHUMAN3H-LSDC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989535-HT6CLONEDHUMAN3H-LSDC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989545-HT7CLONEDHUMAN3H-LSDC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 29, 2025
98955Alpha1ACLONEDHUMAN3H-PRAZOSINC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98956Alpha1BCLONEDHUMAN3H-PRAZOSINC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98957Alpha1DCLONEDHUMAN3H-PRAZOSINC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98958Alpha2ACLONEDHUMAN3H-RAUWOLSCINEC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98959Alpha2BCLONEDHUMAN3H-RAUWOLSCINEC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98960Alpha2CCLONEDHUMAN3H-RAUWOLSCINEC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98961Beta 1CLONEDHUMAN125I-PindololC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98962Beta3CLONEDHUMAN125I-PindololC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98963Beta 2CLONEDHUMAN3H-CGP12177C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98964BZPbrain membranesRATFNZC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98965D1CLONEDHUMAN3H-SCH233930C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98966D5CLONEDHUMAN3H-SCH233930C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98967D2CLONEDHUMAN3H-N-MethylspiperoneC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98968D3CLONEDHUMAN3H-N-MethylspiperoneC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98969D4CLONEDHUMAN3H-N-MethylspiperoneC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98970DORCLONEDHUMAN3H-DADLEC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98971KORbrain membranesRAT3H-MUSCIMOLC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 27, 2025
98972H1CLONEDHUMAN3H-PYRILAMINEC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
989735-HT1DCLONEDHUMAN125I-iodoaminopotentidineC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98974H3CLONEDHUMAN3H-Alpha-methylhistamineC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98975H4CLONEDHUMAN3H-HistamineC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98976M2CLONEDHUMAN3H-QNBC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98977M5CLONEDHUMAN3H-QNBC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98978MORCLONEDHUMAN3H-DAMGOC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98979Sigma 1CLONEDHUMAN3H-Pentazocine(+)C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98980Sigma 2CLONEDHUMAN3H-DTGC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98981DATCLONEDHUMAN3H-WIN 35,428C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98982NETCLONEDHUMAN3H-NisoxetineC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
98983SERTCLONEDHUMAN3H-CITALOPRAMC2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98984KORCLONEDHUMAN3H-U69593C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98985PBRKidney membranesRAT3H-PK11195C2- (5-Halothien-2-yl)-ethynyl 5′-methy ester>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989865-HT1ACLONEDHUMAN3H-WAY100635[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989875-HT1BCLONEDHUMAN3H-GR125743[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989885-HT1DCLONEDHUMAN3H-GR125743[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989895-HT1ECLONEDHUMAN3H-5-HT[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989905-HT2ACLONEDHUMAN3H-KETANSERIN[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989915-HT2BCLONEDHUMAN3H-LSD[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989925-HT2CCLONEDHUMAN3H-MESULERGINE[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989935-HT3CLONEDHUMAN3H-GR-65630[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989945-HT5ACLONEDHUMAN3H-LSD[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989955-HT6CLONEDHUMAN3H-LSD[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
989965-HT7CLONEDHUMAN3H-LSD[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 29, 2025
98997Alpha1ACLONEDHUMAN3H-PRAZOSIN[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98998Alpha1BCLONEDHUMAN3H-PRAZOSIN[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
98999Alpha1DCLONEDHUMAN3H-PRAZOSIN[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99000Alpha2ACLONEDHUMAN3H-RAUWOLSCINE[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99001Alpha2BCLONEDHUMAN3H-RAUWOLSCINE[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99002Alpha2CCLONEDHUMAN3H-RAUWOLSCINE[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99003Beta 1CLONEDHUMAN125I-Pindolol[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99004Beta3CLONEDHUMAN125I-Pindolol[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99005Beta 2CLONEDHUMAN3H-CGP12177[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99006BZPbrain membranesRATFNZ[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99007D1CLONEDHUMAN3H-SCH23390[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99008D5CLONEDHUMAN3H-SCH23390[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99009D2CLONEDHUMAN3H-N-Methylspiperone[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99010D3CLONEDHUMAN3H-N-Methylspiperone[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99011D4CLONEDHUMAN3H-N-Methylspiperone[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99012DORCLONEDHUMAN3H-DADLE[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99013KORbrain membranesRAT3H-MUSCIMOL[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 27, 2025
99014H1CLONEDHUMAN3H-PYRILAMINE[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
990155-HT1DCLONEDHUMAN125I-aminopotentidine[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99016H3CLONEDHUMAN3H-Alpha-methylhistamine[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99017H4CLONEDHUMAN3H-Histamine[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99018M2CLONEDHUMAN3H-QNB[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99019M5CLONEDHUMAN3H-QNB[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99020MORCLONEDHUMAN3H-DAMGO[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99021Sigma 1CLONEDHUMAN3H-Pentazocine(+)[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99022Sigma 2CLONEDHUMAN3H-DTG[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99023DATCLONEDHUMAN3H-WIN 35,428[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99024NETCLONEDHUMAN3H-Nisoxetine[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99025SERTCLONEDHUMAN3H-CITALOPRAM[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99026KORCLONEDHUMAN3H-U69593[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99027PBRKidney membranesRAT3H-PK11195[[(2R,3R,4S,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3R,4S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990285-HT1ACLONEDHUMAN3H-WAY100635(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990295-HT1ACLONEDHUMAN3H-WAY100635(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990305-HT1ACLONEDHUMAN3H-WAY100635(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990315-HT1BCLONEDHUMAN3H-GR125743(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990325-HT1BCLONEDHUMAN3H-GR125743(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990335-HT1BCLONEDHUMAN3H-GR125743(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990345-HT1DCLONEDHUMAN3H-GR125743(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990355-HT1DCLONEDHUMAN3H-GR125743(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990365-HT1DCLONEDHUMAN3H-GR125743(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990375-HT1ECLONEDHUMAN3H-5-HT(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990385-HT1ECLONEDHUMAN3H-5-HT(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990395-HT1ECLONEDHUMAN3H-5-HT(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990405-HT2ACLONEDHUMAN3H-Ketaserin(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990415-HT2ACLONEDHUMAN3H-Ketaserin(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990425-HT2ACLONEDHUMAN3H-Ketaserin(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990435-HT2BCLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990445-HT2BCLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990455-HT2BCLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990465-HT2CCLONEDHUMAN3H-MESULERGINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990475-HT2CCLONEDHUMAN3H-MESULERGINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990485-HT2CCLONEDHUMAN3H-MESULERGINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990495-HT3CLONEDHUMAN3H-GR-65630(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990505-HT3CLONEDHUMAN3H-GR-65630(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990515-HT3CLONEDHUMAN3H-GR-65630(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990525-HT5ACLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990535-HT5ACLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990545-HT5ACLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990555-HT6CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990565-HT6CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990575-HT6CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
990585-HT7CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 29, 2025
990595-HT7CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 29, 2025
990605-HT7CLONEDHUMAN3H-LSD(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 29, 2025
99061Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99062Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99063Alpha1ACLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99064Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99065Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99066Alpha1BCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99067Alpha1DCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99068Alpha1DCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99069Alpha1DCLONEDHUMAN3H-PRAZOSIN(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99070Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99071Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99072Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99073Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99074Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99075Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99076Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99077Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99078Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99079Beta1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99080Beta1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99081Beta1CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99082Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99083Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99084Beta3CLONEDHUMAN125I-Pindolol(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99085Beta 2CLONEDHUMAN3H-CGP12177(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99086Beta 2CLONEDHUMAN3H-CGP12177(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99087Beta 2CLONEDHUMAN3H-CGP12177(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99088BZPbrain membranesRATFNZ(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99089BZPbrain membranesRATFNZ(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99090BZPbrain membranesRATFNZ(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99091D1CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99092D1CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99093D1CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99094D5CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99095D5CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99096D5CLONEDHUMAN3H-SCH23390(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99097D2CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99098D2CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99099D2CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99100D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99101D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99102D3CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99103D4CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99104D4CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99105D4CLONEDHUMAN3H-N-Methylspiperone(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99106DORCLONEDHUMAN3H-DADLE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99107DORCLONEDHUMAN3H-DADLE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99108DORCLONEDHUMAN3H-DADLE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99109KORbrain membranesRAT3H-MUSCIMOL(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 27, 2025
99110KORbrain membranesRAT3H-MUSCIMOL(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 27, 2025
99111KORbrain membranesRAT3H-MUSCIMOL(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 27, 2025
99112H1CLONEDHUMAN3H-PYRILAMINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99113H1CLONEDHUMAN3H-PYRILAMINE(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99114H1CLONEDHUMAN3H-PYRILAMINE(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
991155-HT1DCLONEDHUMAN125I-aminopotentidine(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
991165-HT1DCLONEDHUMAN125I-aminopotentidine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
991175-HT1DCLONEDHUMAN125I-aminopotentidine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99118H3CLONEDHUMAN3H-Alpha-methylhistamine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99119H3CLONEDHUMAN3H-Alpha-methylhistamine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99120H3CLONEDHUMAN3H-Alpha-methylhistamine(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99121H4CLONEDHUMAN3H-Histamine(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99122H4CLONEDHUMAN3H-Histamine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99123H4CLONEDHUMAN3H-Histamine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99124M2CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99125M2CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99126M2CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99127M5CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99128M5CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99129M5CLONEDHUMAN3H-QNB(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99130MORCLONEDHUMAN3H-DAMGO(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99131MORCLONEDHUMAN3H-DAMGO(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99132MORCLONEDHUMAN3H-DAMGO(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99133Sigma 1CLONEDHUMAN3H-Pentazocine(+)(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99134Sigma 1CLONEDHUMAN3H-Pentazocine(+)(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide3260Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99135Sigma 1CLONEDHUMAN3H-Pentazocine(+)(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99136Sigma 2CLONEDHUMAN3H-DTG(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide1830Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99137Sigma 2CLONEDHUMAN3H-DTG(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide980Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99138Sigma 2CLONEDHUMAN3H-DTG(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide2220Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99139DATCLONEDHUMAN3H-WIN 35,428(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99140DATCLONEDHUMAN3H-WIN 35,428(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99141DATCLONEDHUMAN3H-WIN 35,428(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99142NETCLONEDHUMAN3H-Nisoxetine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99143NETCLONEDHUMAN3H-Nisoxetine(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99144NETCLONEDHUMAN3H-Nisoxetine(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99145SERTCLONEDHUMAN3H-CITALOPRAM(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99146SERTCLONEDHUMAN3H-CITALOPRAM(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99147SERTCLONEDHUMAN3H-CITALOPRAM(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99148KORCLONEDHUMAN3H-U69593(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99149KORCLONEDHUMAN3H-U69593(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99150KORCLONEDHUMAN3H-U69593(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 28, 2025
99151PBRKidney membranesRAT3H-PK11195(2S,3S,4R,5R)-5-(5-((5-Fluorothiophen-2-yl)ethynyl)-7-(methylamino)-3H-imidazo[4,5-b]pyridin-3-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99152PBRKidney membranesRAT3H-PK11195(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(propylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99153PBRKidney membranesRAT3H-PK11195(2S,3S,4R,5R)-5-(2-((5-Fluorothiophen-2-yl)ethynyl)-6-(methylamino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide>10000Tosh DK et al 2020Jan 15, 2025Jan 15, 2025
99154A1CLONEDHUMAN[3H]CCPAcaffeine>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99155A1CLONEDHUMAN[3H]CCPACn4c(=O)c3c(nc2CN(Cc1ccccc1)CCn23)n(C)c4=O265Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99156A1CLONEDHUMAN[3H]CCPACn4c(=O)c3c(nc2CN(Cc1ccc(Cl)c(Cl)c1)CCn23)n(C)c4=O791Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99157A1CLONEDHUMAN[3H]CCPA8-(3-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99158A1CLONEDHUMAN[3H]CCPA8-(2,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione3520Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99159A1CLONEDHUMAN[3H]CCPA8-(4-Chloro-2-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione0.553Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99160A1CLONEDHUMAN[3H]CCPA8-(3-(4-Chlorophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione65.5Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99161A1CLONEDHUMAN[3H]CCPA8-(3-(3-Bromophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione3880Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99162A1CLONEDHUMAN[3H]CCPA(R)-1,3-Dimethyl-8-(2,1,3,4-tetrahydronaphthalen-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione393Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99163A1CLONEDHUMAN[3H]CCPA1,3-Dimethyl-8-((2-(thiophen-2-yl)thiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione642Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99164A1CLONEDHUMAN[3H]CCPA1,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)thia-zol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione236Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99165A1CLONEDHUMAN[3H]CCPA8-((2-(3-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione73Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99166A1CLONEDHUMAN[3H]CCPA8-((2-(4-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione492Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99167A1CLONEDRAT[3H]CCPAcaffeine>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99168A1CLONEDRAT[3H]CCPACn4c(=O)c3c(nc2CN(Cc1ccccc1)CCn23)n(C)c4=O79.3Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99169A1CLONEDRAT[3H]CCPACn4c(=O)c3c(nc2CN(Cc1ccc(Cl)c(Cl)c1)CCn23)n(C)c4=O351Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99170A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-phenyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1.5Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99171A1CLONEDRAT[3H]CCPA8-(3-Fluorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99172A1CLONEDRAT[3H]CCPA8-(4-Fluorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99173A1CLONEDRAT[3H]CCPA8-(3-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione159Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99174A1CLONEDRAT[3H]CCPA8-(4-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99175A1CLONEDRAT[3H]CCPA8-(4-Bromophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99176A1CLONEDRAT[3H]CCPA8-(3-Methoxyphenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99177A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(naphtha-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99178A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-phenethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99179A1CLONEDRAT[3H]CCPA8-(2-Fluorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99180A1CLONEDRAT[3H]CCPA8-(3-Fluorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99181A1CLONEDRAT[3H]CCPA8-(2-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99182A1CLONEDRAT[3H]CCPA8-(3-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99183A1CLONEDRAT[3H]CCPA8-(4-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99184A1CLONEDRAT[3H]CCPA8-(2-Bromophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99185A1CLONEDRAT[3H]CCPA8-(3-Bromophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99186A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99187A1CLONEDRAT[3H]CCPA8-(4-Hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99188A1CLONEDRAT[3H]CCPA8-(2-Methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99189A1CLONEDRAT[3H]CCPA8-(3-Methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99190A1CLONEDRAT[3H]CCPA8-(3,4-Difluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99191A1CLONEDRAT[3H]CCPA8-(2-Fluoro-5-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99192A1CLONEDRAT[3H]CCPA8-(2,6-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99193A1CLONEDRAT[3H]CCPA8-(3,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99194A1CLONEDRAT[3H]CCPA8-(2,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione416Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99195A1CLONEDRAT[3H]CCPA8-(4-Chloro-2-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione138Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99196A1CLONEDRAT[3H]CCPA8-(2-(5-Bromo-2-methoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99197A1CLONEDRAT[3H]CCPA8-(2-(2,3-Dimethoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99198A1CLONEDRAT[3H]CCPA8-(2-(3,4-Dimethoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99199A1CLONEDRAT[3H]CCPA8-(2-(Benzo[d][1,3]dioxol-5-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99200A1CLONEDRAT[3H]CCPA8-(2-Hydroxy-2-phenylethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99201A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(2-methyl-2-phenylethyl)-6,7,8,9-tetrahy-dropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99202A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(2-(thiophen-2-yl)ethyl)-6,7,8,9-tetra-hydropyrazino[2,1-f]purine2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99203A1CLONEDRAT[3H]CCPA8-(2-(1H-Pyrrol-1-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99204A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(3-phenylpropyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99205A1CLONEDRAT[3H]CCPA8-(3-(4-Chlorophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione352Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99206A1CLONEDRAT[3H]CCPA8-(3-(3-Bromophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99207A1CLONEDRAT[3H]CCPA8-(3-(1H-Pyrrol-1-yl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99208A1CLONEDRAT[3H]CCPA8-(3-(1H-Imidazol-1-yl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99209A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(2-phenoxyethyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99210A1CLONEDRAT[3H]CCPA8-(2-(2-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99211A1CLONEDRAT[3H]CCPA8-(2-(3-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99212A1CLONEDRAT[3H]CCPA8-(2-(3-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1250Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99213A1CLONEDRAT[3H]CCPA(R)-1,3-Dimethyl-8-(2,1,3,4-tetrahydronaphthalen-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione100Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99214A1CLONEDRAT[3H]CCPA(S)-8-(5-Methoxy-2,1,3,4-tetrahydronaphth-2-yl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99215A1CLONEDRAT[3H]CCPA8-(2,3-Dihydro-1H-inden-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99216A1CLONEDRAT[3H]CCPA(R,S)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99217A1CLONEDRAT[3H]CCPA(S)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7, 8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99218A1CLONEDRAT[3H]CCPA(R)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7, 8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99219A1CLONEDRAT[3H]CCPA8-(1-Benzylpiperidin-4-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99220A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-((4-phenylisoxazol-3-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99221A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-((2-(thiophen-2-yl)thiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione166Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99222A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)thia-zol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione157Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99223A1CLONEDRAT[3H]CCPA8-((2-(3-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione437Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99224A1CLONEDRAT[3H]CCPA8-((2-(4-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione76Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99225A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)-5-methylthiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99226A1CLONEDRAT[3H]CCPA8-((1,3-Dimethyl-1H-pyrazol-5-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99227A1CLONEDRAT[3H]CCPA8-(1-((4-Chlorophenyl)-1H-2,1,3-triazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]pur-ine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99228A1CLONEDRAT[3H]CCPA1,3-Dimethyl-8-(propyn-2-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99229A1CLONEDRAT[3H]CCPA8-(3-(3-Chlorophenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99230A1CLONEDRAT[3H]CCPA8-(3-(3,4-Dichlorophenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99231A1CLONEDRAT[3H]CCPA8-(3-(3-Methoxyphenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99232A2ACLONEDHUMAN[3H]MSX-2caffeine>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99233A2ACLONEDHUMAN[3H]MSX-2Cn4c(=O)c3c(nc2CN(Cc1ccccc1)CCn23)n(C)c4=O1060Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99234A2ACLONEDHUMAN[3H]MSX-2Cn4c(=O)c3c(nc2CN(Cc1ccc(Cl)c(Cl)c1)CCn23)n(C)c4=O1510Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99235A2ACLONEDHUMAN[3H]MSX-28-(3-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione8860Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99236A2ACLONEDHUMAN[3H]MSX-28-(3-(4-Chlorophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione230Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99237A2ACLONEDHUMAN[3H]MSX-28-(3-(3-Bromophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione512Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99238A2ACLONEDHUMAN[3H]MSX-2(R)-1,3-Dimethyl-8-(2,1,3,4-tetrahydronaphthalen-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione595Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99239A2ACLONEDHUMAN[3H]MSX-21,3-Dimethyl-8-((2-(thiophen-2-yl)thiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione203Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99240A2ACLONEDHUMAN[3H]MSX-21,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)thia-zol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione217Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99241A2ACLONEDHUMAN[3H]MSX-28-((2-(3-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione363Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99242A2ACLONEDHUMAN[3H]MSX-28-((2-(4-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione346Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99243A2ACLONEDRAT[3H]MSX-2caffeine>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99244A2ACLONEDRAT[3H]MSX-2Cn4c(=O)c3c(nc2CN(Cc1ccccc1)CCn23)n(C)c4=O598Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99245A2ACLONEDRAT[3H]MSX-2Cn4c(=O)c3c(nc2CN(Cc1ccc(Cl)c(Cl)c1)CCn23)n(C)c4=O322Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99246A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-phenyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione3830Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99247A2ACLONEDRAT[3H]MSX-28-(3-Fluorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2920Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99248A2ACLONEDRAT[3H]MSX-28-(4-Fluorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2130Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99249A2ACLONEDRAT[3H]MSX-28-(3-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione557Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99250A2ACLONEDRAT[3H]MSX-28-(4-Chlorophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99251A2ACLONEDRAT[3H]MSX-28-(4-Bromophenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione3900Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99252A2ACLONEDRAT[3H]MSX-28-(3-Methoxyphenyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1010Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99253A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(naphtha-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2940Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99254A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-phenethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione9610Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99255A2ACLONEDRAT[3H]MSX-28-(2-Fluorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione5630Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99256A2ACLONEDRAT[3H]MSX-28-(3-Fluorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1500Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99257A2ACLONEDRAT[3H]MSX-28-(2-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2730Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99258A2ACLONEDRAT[3H]MSX-28-(3-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1310Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99259A2ACLONEDRAT[3H]MSX-28-(4-Chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione4960Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99260A2ACLONEDRAT[3H]MSX-28-(2-Bromophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99261A2ACLONEDRAT[3H]MSX-28-(3-Bromophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2120Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99262A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(3-(trifluoromethyl)phenethyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione2580Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99263A2ACLONEDRAT[3H]MSX-28-(4-Hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione6040Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99264A2ACLONEDRAT[3H]MSX-28-(2-Methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99265A2ACLONEDRAT[3H]MSX-28-(3-Methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99266A2ACLONEDRAT[3H]MSX-28-(3,4-Difluorophenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99267A2ACLONEDRAT[3H]MSX-28-(2-Fluoro-5-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99268A2ACLONEDRAT[3H]MSX-28-(2,6-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione3050Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99269A2ACLONEDRAT[3H]MSX-28-(3,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2850Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99270A2ACLONEDRAT[3H]MSX-28-(2,4-Dichlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione2250Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99271A2ACLONEDRAT[3H]MSX-28-(4-Chloro-2-(trifluoromethyl)phenethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione2910Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99272A2ACLONEDRAT[3H]MSX-28-(2-(5-Bromo-2-methoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99273A2ACLONEDRAT[3H]MSX-28-(2-(2,3-Dimethoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99274A2ACLONEDRAT[3H]MSX-28-(2-(3,4-Dimethoxyphenyl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99275A2ACLONEDRAT[3H]MSX-28-(2-(Benzo[d][1,3]dioxol-5-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione6170Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99276A2ACLONEDRAT[3H]MSX-28-(2-Hydroxy-2-phenylethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione7110Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99277A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(2-methyl-2-phenylethyl)-6,7,8,9-tetrahy-dropyrazino[2,1-f]purine-2,4-(1H,3H)-dione4520Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99278A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(2-(thiophen-2-yl)ethyl)-6,7,8,9-tetra-hydropyrazino[2,1-f]purine2,4-(1H,3H)-dione1590Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99279A2ACLONEDRAT[3H]MSX-28-(2-(1H-Pyrrol-1-yl)ethyl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99280A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(3-phenylpropyl)-6,7,8,9-tetrahydro-pyrazino[2,1-f]purine-2,4(1H,3H)-dione1840Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99281A2ACLONEDRAT[3H]MSX-28-(3-(4-Chlorophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione316Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99282A2ACLONEDRAT[3H]MSX-28-(3-(3-Bromophenyl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione450Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99283A2ACLONEDRAT[3H]MSX-28-(3-(1H-Pyrrol-1-yl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99284A2ACLONEDRAT[3H]MSX-28-(3-(1H-Imidazol-1-yl)propyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99285A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(2-phenoxyethyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99286A2ACLONEDRAT[3H]MSX-28-(2-(2-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99287A2ACLONEDRAT[3H]MSX-28-(2-(3-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99288A2ACLONEDRAT[3H]MSX-28-(2-(3-Fluorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione2420Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99289A2ACLONEDRAT[3H]MSX-2(R)-1,3-Dimethyl-8-(2,1,3,4-tetrahydronaphthalen-1-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione510Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99290A2ACLONEDRAT[3H]MSX-2(S)-8-(5-Methoxy-2,1,3,4-tetrahydronaphth-2-yl)-1,3-dimethyl-6,7,8,9-tetra-hydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99291A2ACLONEDRAT[3H]MSX-28-(2,3-Dihydro-1H-inden-2-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione>10000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99292A2ACLONEDRAT[3H]MSX-2(R,S)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione4210Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99293A2ACLONEDRAT[3H]MSX-2(S)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7, 8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione2480Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99294A2ACLONEDRAT[3H]MSX-2(R)-8-(2,3-Dihydro-1H-inden-1-yl)-1,3-dimethyl-6,7, 8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione5080Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99295A2ACLONEDRAT[3H]MSX-28-(1-Benzylpiperidin-4-yl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4-(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99296A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-((4-phenylisoxazol-3-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99297A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-((2-(thiophen-2-yl)thiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione121Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99298A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)thia-zol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione355Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99299A2ACLONEDRAT[3H]MSX-28-((2-(3-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione160Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99300A2ACLONEDRAT[3H]MSX-28-((2-(4-Chlorophenyl)thiazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione62Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99301A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-((2-(4-(trifluoromethyl)phenyl)-5-methylthiazol-4-yl)methyl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99302A2ACLONEDRAT[3H]MSX-28-((1,3-Dimethyl-1H-pyrazol-5-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99303A2ACLONEDRAT[3H]MSX-28-(1-((4-Chlorophenyl)-1H-2,1,3-triazol-4-yl)methyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]pur-ine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99304A2ACLONEDRAT[3H]MSX-21,3-Dimethyl-8-(propyn-2-yl)-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99305A2ACLONEDRAT[3H]MSX-28-(3-(3-Chlorophenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99306A2ACLONEDRAT[3H]MSX-28-(3-(3,4-Dichlorophenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99307A2ACLONEDRAT[3H]MSX-28-(3-(3-Methoxyphenyl)prop-2-ynyl)-1,3-dimethyl-6,7,8,9-tetrahydropyrazino-[2,1-f]purine-2,4(1H,3H)-dione1000Brunschweiger A et al 2016Jan 15, 2025Jan 15, 2025
99308D2CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine31.5Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99309D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2-methoxyphenyl)piperazine57.2Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99310D2CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole51.8Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99311D2CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline83.4Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99312D2CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-phenyl-1H-1,2,3-triazol-4-yl)butyl)piperazine53.6Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99313D2CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine80.8Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99314D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2,3-dichlorophenyl)piperazine424Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99315D2CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole46.4Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99316D2CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine23.3Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99317D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine50.1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99318D2CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole43.7Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99319D2CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline42.5Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99320D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine69Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99321D2CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(4-phenyl-1H-1,2,3-triazol-1-yl)butyl)piperazine137Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99322D2CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine103Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99323D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2,3-dichlorophenyl)piperazine885Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99324D2CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole56.1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99325D2CLONEDHUMAN[3H]N-methylspiperone6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline53.9Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99326D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine2590Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99327D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol189Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99328D2CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol819Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99329D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)butan-2-ol1210Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99330D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(2-Methoxyphenyl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol1020Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99331D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol607Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99332D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(quinolin-6-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol424Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99333D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(naphtha-len-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99334D2CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,1’-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99335D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol789Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99336D2CLONEDHUMAN[3H]N-methylspiperone4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol963Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99337D2CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(quinolin-3-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol244Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99338D2CLONEDHUMAN[3H]N-methylspiperonePG648746Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99339D2CLONEDHUMAN[3H]N-methylspiperoneOMO5-057321Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99340D2CLONEDHUMAN[3H]N-methylspiperoneNGB290454.7Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99341D3CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine2.93Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99342D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2-methoxyphenyl)piperazine1.59Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99343D3CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole3.1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99344D3CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline13.1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99345D3CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-phenyl-1H-1,2,3-triazol-4-yl)butyl)piperazine5.42Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99346D3CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine3.8Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99347D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2,3-dichlorophenyl)piperazine5.05Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99348D3CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99349D3CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine11.1Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99350D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine5.55Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99351D3CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole5.48Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99352D3CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline6.72Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99353D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine5.88Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99354D3CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(4-phenyl-1H-1,2,3-triazol-1-yl)butyl)piperazine22.9Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99355D3CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine7.7Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99356D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2,3-dichlorophenyl)piperazine14Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99357D3CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole1.47Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99358D3CLONEDHUMAN[3H]N-methylspiperone6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline1.35Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99359D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine8.32Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99360D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol40.7Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99361D3CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol30.5Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99362D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)butan-2-ol173Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99363D3CLONEDHUMAN[3H]N-methylspiperone4-(4-(2-Methoxyphenyl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol493Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99364D3CLONEDHUMAN[3H]N-methylspiperone4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol18.5Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99365D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(quinolin-6-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol68.2Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99366D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(naphtha-len-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol25.2Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99367D3CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,1’-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol55.8Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99368D3CLONEDHUMAN[3H]N-methylspiperone4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol33.6Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99369D3CLONEDHUMAN[3H]N-methylspiperone4-(4-(1H-Indol-5-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol5.85Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99370D3CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(quinolin-3-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol18Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99371D3CLONEDHUMAN[3H]N-methylspiperonePG6481.88Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99372D3CLONEDHUMAN[3H]N-methylspiperoneOMO5-0572.91Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99373D3CLONEDHUMAN[3H]N-methylspiperoneNGB29040.233Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99374D4CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine299Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99375D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2-methoxyphenyl)piperazine329Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99376D4CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole353Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99377D4CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline1000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99378D4CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(1-phenyl-1H-1,2,3-triazol-4-yl)butyl)piperazine486Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99379D4CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(1-(naphthalen-2-yl)-1H-1,2,3-triazol-4-yl)butyl)piperazine2000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99380D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(1-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-4-yl)butyl)-4-(2,3-dichlorophenyl)piperazine4450Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99381D4CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)-1H-indole510Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99382D4CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine232Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99383D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine588Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99384D4CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole222Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99385D4CLONEDHUMAN[3H]N-methylspiperone5-(4-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)quinoline269Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99386D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2-methoxyphenyl)piperazine425Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99387D4CLONEDHUMAN[3H]N-methylspiperone1-(2-Methoxyphenyl)-4-(4-(4-phenyl-1H-1,2,3-triazol-1-yl)butyl)piperazine480Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99388D4CLONEDHUMAN[3H]N-methylspiperone1-(2,3-Dichlorophenyl)-4-(4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butyl)piperazine1000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99389D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)butyl)-4-(2,3-dichlorophenyl)piperazine>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99390D4CLONEDHUMAN[3H]N-methylspiperone5-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)-1H-indole2000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99391D4CLONEDHUMAN[3H]N-methylspiperone6-(1-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)-1H-1,2,3-triazol-4-yl)quinoline1000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99392D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-butyl)-4-(2,3-dichlorophenyl)piperazine>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99393D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(naphthalen-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol2000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99394D4CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,10-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol2000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99395D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)butan-2-ol3000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99396D4CLONEDHUMAN[3H]N-methylspiperone4-(4-(2-Methoxyphenyl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol3000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99397D4CLONEDHUMAN[3H]N-methylspiperone4-(4-(9H-Fluoren-2-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2-methoxyphenyl)piperazin-1-yl)butan-2-ol1000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99398D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(2-Methoxyphenyl)piperazin-1-yl)-4-(4-(quinolin-6-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol3000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99399D4CLONEDHUMAN[3H]N-methylspiperone1-(4-(2,3-Dichlorophenyl)piperazin-1-yl)-4-(4-(naphtha-len-2-yl)-1H-1,2,3-triazol-1-yl)butan-2-ol>10000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99400D4CLONEDHUMAN[3H]N-methylspiperone4-(4-([1,1’-Biphenyl]-4-yl)-1H-1,2,3-triazol-1-yl)-1-(4-(2,3-dichlorophenyl)piperazin-1-yl)butan-2-ol7000Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99401D4CLONEDHUMAN[3H]N-methylspiperonePG6482600Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99402D4CLONEDHUMAN[3H]N-methylspiperoneNGB29043670Keck TM et al 2015Jan 15, 2025Jan 28, 2025
99403D2CLONEDHUMANUNDEFINED2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide45Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99404D2CLONEDHUMANUNDEFINED2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide24Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99405D2CLONEDHUMANUNDEFINED2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide39Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99406D2CLONEDHUMANUNDEFINED2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide29Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99407D2CLONEDHUMANUNDEFINED2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide132Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99408D2CLONEDHUMANUNDEFINED2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide105Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99409D2CLONEDHUMANUNDEFINED2-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide61Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99410D2CLONEDHUMANUNDEFINED2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide113Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99411D2CLONEDHUMANUNDEFINED2-(6-(4-(4-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide950Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99412D2CLONEDHUMANUNDEFINED2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide27Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99413D2CLONEDHUMANUNDEFINED2-(6-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide7Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99414D2CLONEDHUMANUNDEFINED2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide48Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99415D2CLONEDHUMANUNDEFINED2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide8Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99416D2CLONEDHUMANUNDEFINED2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide15Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99417D2CLONEDHUMANUNDEFINED2-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide230Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99418D2CLONEDHUMANUNDEFINED2-(6-(4-(pyrimidin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide51Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
99419D2CLONEDHUMANUNDEFINED2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide9Kulaga D et al 2019Jan 15, 2025Jan 28, 2025
994205-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide26Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994215-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide12Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994225-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide21Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994235-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(4-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide84Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994245-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide58Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994255-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide54Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994265-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide91Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994275-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide19Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994285-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(4-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide327Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994295-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide156Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994305-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide25Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994315-HT1ACLONEDHUMANUNDEFINED2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide20Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994325-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide9Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994335-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide4Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994345-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide13Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994355-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(pyrimidin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide24Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994365-HT1ACLONEDHUMANUNDEFINED2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide23Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994375-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide266Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994385-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide307Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994395-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide361Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994405-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide209Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994415-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide283Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994425-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide342Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994435-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide922Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994445-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide167Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994455-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide321Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994465-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide91Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994475-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide205Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994485-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide1290Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994495-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(pyrimidin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide183Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994505-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide23Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994515-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide459Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994525-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide1619Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994535-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide372Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994545-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide920Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994555-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide132Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994565-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide921Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994575-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide1272Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994585-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide52Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994595-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide971Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994605-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide157Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994615-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide1718Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994625-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide2352Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994635-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(pyrimidin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide104Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994645-HT6UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide59Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994655-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide120Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994665-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-fluorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide322Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994675-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-chlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide233Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994685-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2,3-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide119Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994695-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3,4-dichlorophenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide258Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994705-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-methoxyphenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide305Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994715-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(2-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide195Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994725-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide58Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994735-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-phenylpiperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide192Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994745-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(naphthalen-1-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide20Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994755-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(quinolin-8-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide21Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994765-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide552Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994775-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(pyrimidin-2-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide35Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
994785-HT7UNDEFINEDUNDEFINEDUNDEFINED2-(6-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)hexyl)benzo[d]isothiazol-3(2H)-one 1,1-dioxide45Kulaga D et al 2019Jan 15, 2025Jan 15, 2025
99479A1CHO cellsHUMAN3H-CCPA4-Methoxy-N-[4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-benzamide688Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99480A2ACHO cellsHUMAN3H-NECA4-Methoxy-N-[4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-benzamide128Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99481A3CHO cellsHUMAN3H-HEMADO4-Methoxy-N-[4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-benzamide201Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99482A1CHO cellsHUMAN3H-CCPA4-Methoxy-N-[4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99483A2ACHO cellsHUMAN3H-NECA4-Methoxy-N-[4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99484A3CHO cellsHUMAN3H-HEMADO4-Methoxy-N-[4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99485A1CHO cellsHUMAN3H-CCPAN-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methoxybenzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99486A2ACHO cellsHUMAN3H-NECAN-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methoxybenzamide2010Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99487A3CHO cellsHUMAN3H-HEMADON-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methoxybenzamide2640Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99488A1CHO cellsHUMAN3H-CCPAN-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methylbenzamide3630Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99489A2ACHO cellsHUMAN3H-NECAN-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methylbenzamide562Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99490A3CHO cellsHUMAN3H-HEMADON-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)-4-methylbenzamide816Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99491A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-6-dimethylamino-[1,3,5]triazin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide801Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99492A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-6-dimethylamino-[1,3,5]triazin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide327Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99493A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-6-dimethylamino-[1,3,5]triazin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide567Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99494A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99495A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99496A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide2470Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99497A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99498A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99499A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide1380Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99500A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide7240Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99501A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide4870Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99502A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide676Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99503A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99504A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99505A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methoxy-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99506A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99507A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99508A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-4-methyl-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99509A1CHO cellsHUMAN3H-CCPAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99510A2ACHO cellsHUMAN3H-NECAN-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99511A3CHO cellsHUMAN3H-HEMADON-[5-(4-Amino-5,6,7,8-tetrahydro-benzo[4,5]-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-benzamide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99512A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic-acid [4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-amide406Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99513A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic-acid [4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-amide74.7Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99514A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic-acid [4-phenyl-5-(pyridine-2-carbonyl)-thiazol-2-yl]-amide951Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99515A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid [4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-amide177Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99516A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid [4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-amide552Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99517A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid [4-phenyl-5-(pyridine-3-carbonyl)-thiazol-2-yl]-amide1870Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99518A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid (4-phenyl-5-pyridin-2-yl-thiazol-2-yl)-amide276Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99519A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid (4-phenyl-5-pyridin-2-yl-thiazol-2-yl)-amide193Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99520A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid (4-phenyl-5-pyridin-2-yl-thiazol-2-yl)-amide2040Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99521A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid (4-phenyl-5-pyridin-4-yl-thiazol-2-yl)-amide0.58Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99522A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid (4-phenyl-5-pyridin-4-yl-thiazol-2-yl)-amide6.65Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99523A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid (4-phenyl-5-pyridin-4-yl-thiazol-2-yl)-amide9.36Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99524A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid [5-(4-amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99525A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid [5-(4-amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide5950Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99526A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid [5-(4-amino-5,6-dimethyl-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide746Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99527A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid [5-(4-amino-5,6,7,8-tetrahydro-benzo[4,5]thieno[2,3-d]pyrim-idin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99528A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid [5-(4-amino-5,6,7,8-tetrahydro-benzo[4,5]thieno[2,3-d]pyrim-idin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99529A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid [5-(4-amino-5,6,7,8-tetrahydro-benzo[4,5]thieno[2,3-d]pyrim-idin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99530A1CHO cellsHUMAN3H-CCPAN-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide536Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99531A2ACHO cellsHUMAN3H-NECAN-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide179Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99532A3CHO cellsHUMAN3H-HEMADON-(5-(4-Amino-6-(dimethylamino)-1,3,5-triazin-2-yl)-4-phenylthiazol-2-yl)furan-2-carboxamide918Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99533A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid [5-(5,6-dimethyl-4-oxo-3,4-dihydro-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99534A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid [5-(5,6-dimethyl-4-oxo-3,4-dihydro-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99535A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid [5-(5,6-dimethyl-4-oxo-3,4-dihydro-thieno[2,3-d]pyrimidin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99536A1CHO cellsHUMAN3H-CCPAFuran-2-carboxylic acid [5-(4-oxo-3,4-dihydro-quinazolin-2-yl)-4-phenyl-thiazol-2-yl]-amide>10000Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99537A2ACHO cellsHUMAN3H-NECAFuran-2-carboxylic acid [5-(4-oxo-3,4-dihydro-quinazolin-2-yl)-4-phenyl-thiazol-2-yl]-amide8780Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99538A3CHO cellsHUMAN3H-HEMADOFuran-2-carboxylic acid [5-(4-oxo-3,4-dihydro-quinazolin-2-yl)-4-phenyl-thiazol-2-yl]-amide3930Inamdar GS et al 2013Jan 15, 2025Jan 15, 2025
99539A1CLONEDHUMAN3H-CCPA8-[4-(2-Dimethylaminoethoxy)phenyl]-1,3-dimethylxanthine1820Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99540A1CLONEDHUMAN3H-CCPA8-[4-(2-Diethylaminoethoxy)phenyl]-1,3-dimethylxanthine1590Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99541A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-(2-piperidin-4-ylethoxy)phenyl]xanthine1330Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99542A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-(2-morpholin-4-ylethoxy)phenyl]xanthine2580Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99543A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-(2-pyrrolidin-1-ylethoxy)phenyl]xanthine1200Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99544A1CLONEDHUMAN3H-CCPA8-[4-(3-Chloropropoxy)phenyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99545A1CLONEDHUMAN3H-CCPA8-[4-(Cyclopentyloxy)phenyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99546A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-(3-imidazol-1-ylpropoxy)phenyl]xanthine890Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99547A1CLONEDHUMAN3H-CCPA8-[4-{3-(4-(2-Chlorobenzyl)piperazin-1-yl)propoxy}phenyl]- 1,3-dimethylxanthine1850Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99548A1CLONEDHUMAN3H-CCPA8-[4-(3-Chloropropoxy)benzyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99549A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-(3-morpholinopropoxy)benzyl]xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99550A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{3-(1H-imidazol-1-yl)propoxy}benzyl] xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99551A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{3-(1,4-dioxa-8-azaspiro[4.5]decan-1-yl)- propoxy}benzyl]-xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99552A2ACLONEDHUMAN3H-NECA8-[4-(2-Dimethylaminoethoxy)phenyl]-1,3-dimethylxanthine400Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99553A2ACLONEDHUMAN3H-NECA8-[4-(2-Diethylaminoethoxy)phenyl]-1,3-dimethylxanthine250Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99554A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-(2-piperidin-4-ylethoxy)phenyl]xanthine290Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99555A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-(2-morpholin-4-ylethoxy)phenyl]xanthine310Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99556A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-(2-pyrrolidin-1-ylethoxy)phenyl]xanthine200Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99557A2ACLONEDHUMAN3H-NECA8-[4-(3-Chloropropoxy)phenyl]-1,3-dimethylxanthine45Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99558A2ACLONEDHUMAN3H-NECA8-[4-(Cyclopentyloxy)phenyl]-1,3-dimethylxanthine72Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99559A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-(3-imidazol-1-ylpropoxy)phenyl]xanthine42Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99560A2ACLONEDHUMAN3H-NECA8-[4-{3-(4-(2-Chlorobenzyl)piperazin-1-yl)propoxy}phenyl]- 1,3-dimethylxanthine120Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99561A2ACLONEDHUMAN3H-NECA8-[4-(3-Chloropropoxy)benzyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99562A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-(3-morpholinopropoxy)benzyl]xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99563A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{3-(1H-imidazol-1-yl)propoxy}benzyl] xanthine3170Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99564A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{3-(1,4-dioxa-8-azaspiro[4.5]decan-1-yl)- propoxy}benzyl]-xanthine8090Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99565A3CLONEDHUMAN3H-HEMADO8-[4-(2-Dimethylaminoethoxy)phenyl]-1,3-dimethylxanthine9380Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99566A3CLONEDHUMAN3H-HEMADO8-[4-(2-Diethylaminoethoxy)phenyl]-1,3-dimethylxanthine6820Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99567A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-(2-piperidin-4-ylethoxy)phenyl]xanthine6510Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99568A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-(2-morpholin-4-ylethoxy)phenyl]xanthine2740Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99569A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-(2-pyrrolidin-1-ylethoxy)phenyl]xanthine4600Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99570A3CLONEDHUMAN3H-HEMADO8-[4-(3-Chloropropoxy)phenyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99571A3CLONEDHUMAN3H-HEMADO8-[4-(Cyclopentyloxy)phenyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99572A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-(3-imidazol-1-ylpropoxy)phenyl]xanthine2270Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99573A3CLONEDHUMAN3H-HEMADO8-[4-{3-(4-(2-Chlorobenzyl)piperazin-1-yl)propoxy}phenyl]- 1,3-dimethylxanthine6890Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99574A3CLONEDHUMAN3H-HEMADO8-[4-(3-Chloropropoxy)benzyl]-1,3-dimethylxanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99575A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-(3-morpholinopropoxy)benzyl]xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99576A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{3-(1H-imidazol-1-yl)propoxy}benzyl] xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99577A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{3-(1,4-dioxa-8-azaspiro[4.5]decan-1-yl)- propoxy}benzyl]-xanthine>10000Yadav R et al 2014Jan 15, 2025Jan 15, 2025
99578A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]xanthine0.319Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99579A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-(2-methoxy-2-oxoethoxy)-phenyl]xanthine3.95Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99580A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{4-(2-methoxy-2-oxoethoxy)-3-methoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99581A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{3-(2-methoxy-2-oxoethoxy)-4-methoxy}-phenyl]xanthine11.8Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99582A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine0.22Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99583A1CLONEDHUMAN3H-CCPA8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine0.298Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99584A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phenyl]xanthine0.796Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99585A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthine0.419Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99586A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine0.609Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99587A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine1.25Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99588A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthin0.499Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99589A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine3.99Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99590A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine1.68Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99591A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine0.683Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99592A1CLONEDHUMAN3H-CCPA8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine1.22Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99593A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine3.29Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99594A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine1.52Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99595A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine2.43Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99596A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(morpholin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine5.37Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99597A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine1.9Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99598A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99599A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine5.98Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99600A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine9.25Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99601A1CLONEDHUMAN3H-CCPA8-[{4-(2-(Diethylaminoethylamino)-2-oxoethoxy)-3-meth-oxy}-phenyl]-1,3-dimethyl-xanthine10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99602A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-methoxy-4-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99603A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99604A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-3-methoxy}-phenyl]-xanthin10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99605A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-methoxy-4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99606A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[3-methoxy-4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]-xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99607A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{4-(2-(imidazol-1-yl)-2-oxoethoxy)-3-methoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99608A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{4-(2-(homoveratrylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99609A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-oxo-ethoxy)-4-methoxy}-phenyl]-xanthine0.847Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99610A1CLONEDHUMAN3H-CCPA8-[{3-(2-(Diethylaminoethylamino)-2-oxoethoxy)-4-meth-oxy}phenyl]-1,3-dimethylxanthine1.97Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99611A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine5.94Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99612A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine1.62Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99613A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine1.91Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99614A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2-oxo-ethoxy}-phenyl]-xanthine3.51Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99615A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine3.64Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99616A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{3-(2-(imidazol-1-yl)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99617A1CLONEDHUMAN3H-CCPA1,3-Dimethyl-8-[{3-(2-(homoveratrylamino)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99618A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]xanthine0.17Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99619A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-(2-methoxy-2-oxoethoxy)-phenyl]xanthine0.375Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99620A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{4-(2-methoxy-2-oxoethoxy)-3-methoxy}-phenyl]xanthine4.38Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99621A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{3-(2-methoxy-2-oxoethoxy)-4-methoxy}-phenyl]xanthine0.717Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99622A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine0.1Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99623A2ACLONEDHUMAN3H-NECA8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine0.063Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99624A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phenyl]xanthine1.22Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99625A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthin0.178Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99626A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine0.273Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99627A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine0.283Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99628A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthine0.193Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99629A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine2.69Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99630A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine0.128Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99631A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine0.163Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99632A2ACLONEDHUMAN3H-NECA8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine0.179Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99633A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine0.237Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99634A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine0.209Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99635A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine0.226Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99636A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(morpholin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine0.679Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99637A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine0.561Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99638A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine0.509Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99639A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine1.39Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99640A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine0.821Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99641A2ACLONEDHUMAN3H-NECA8-[{4-(2-(Diethylaminoethylamino)-2-oxoethoxy)-3-meth-oxy}-phenyl]-1,3-dimethyl-xanthine0.692Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99642A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-methoxy-4-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine4.57Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99643A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine3.35Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99644A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-3-methoxy}-phenyl]-xanthine2.41Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99645A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-methoxy-4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine2.74Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99646A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[3-methoxy-4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]-xanthine4.21Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99647A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{4-(2-(imidazol-1-yl)-2-oxoethoxy)-3-methoxy}-phenyl]xanthine7.74Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99648A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{4-(2-(homoveratrylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine0.843Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99649A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-oxo-ethoxy)-4-methoxy}-phenyl]-xanthine0.075Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99650A2ACLONEDHUMAN3H-NECA8-[{3-(2-(Diethylaminoethylamino)-2-oxoethoxy)-4-meth-oxy}phenyl]-1,3-dimethylxanthine0.126Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99651A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-methoxy-3-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine0.259Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99652A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine0.076Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99653A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine0.094Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99654A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2-oxo-ethoxy}-phenyl]-xanthine0.466Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99655A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine0.685Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99656A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{3-(2-(imidazol-1-yl)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine1.12Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99657A2ACLONEDHUMAN3H-NECA1,3-Dimethyl-8-[{3-(2-(homoveratrylamino)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine0.772Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99658A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-(2-methoxy-2-oxoethoxy)-phenyl]xanthine5.86Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99659A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-(2-methoxy-2-oxoethoxy)-phenyl]xanthine3.81Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99660A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{4-(2-methoxy-2-oxoethoxy)-3-methoxy}-phenyl]xanthine10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99661A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{3-(2-methoxy-2-oxoethoxy)-4-methoxy}-phenyl]xanthine10.7Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99662A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine10.5Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99663A3CLONEDHUMAN3H-HEMADO8-[4-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine8.35Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99664A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phenyl]xanthine5.68Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99665A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(piperidin-1-yl)-2-oxoethoxy}-phenyl]xanthine13Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99666A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine4.15Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99667A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine7.11Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99668A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]xanthine10.1Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99669A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99670A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine6Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99671A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(dimethylaminoethylamino)-2-oxo-ethoxy}-phenyl]xanthine8.97Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99672A3CLONEDHUMAN3H-HEMADO8-[3-{2-(Diethylaminoethylamino)-2-oxoethoxy}-phenyl]-1,3-dimethylxanthine8.39Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99673A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(pyrrolidin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine4.64Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99674A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(piperidin-1-yl)]-2-oxoethoxy}-phe-nyl]xanthine4.16Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99675A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine3.69Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99676A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(morpholin-1-yl)-2-oxoethoxy}-phe-nyl]xanthine7.9Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99677A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine5.67Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99678A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(imidazol-1-yl)-2-oxoethoxy}-phenyl]xanthine4.89Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99679A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-{2-(homoveratrylamino)-2-oxoethoxy}-phenyl]xanthine9.25Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99680A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{4-(2-(dimethylaminoethylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99681A3CLONEDHUMAN3H-HEMADO8-[{4-(2-(Diethylaminoethylamino)-2-oxoethoxy)-3-meth-oxy}-phenyl]-1,3-dimethyl-xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99682A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-methoxy-4-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99683A3CLONEDHUMAN3H-HEMADO3-Dimethyl-8-[3-methoxy-4-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99684A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{4-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-3-methoxy}-phenyl]-xanthine9.01Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99685A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-methoxy-4-{2-(morpholin-1-yl)-2-oxoethoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99686A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[3-methoxy-4-{2-(1-methylpiperazin-4-yl)-2-oxoethoxy}-phenyl]-xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99687A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{4-(2-(imidazol-1-yl)-2-oxoethoxy)-3-methoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99688A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{4-(2-(homoveratrylamino)-2-oxoethoxy)-3-methoxy}-phenyl]-xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99689A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{3-(2-(dimethylaminoethylamino)-2-oxo-ethoxy)-4-methoxy}-phenyl]-xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99690A3CLONEDHUMAN3H-HEMADO8-[{3-(2-(Diethylaminoethylamino)-2-oxoethoxy)-4-meth-oxy}phenyl]-1,3-dimethylxanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99691A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-methoxy-3-{2-(pyrrolidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine8.98Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99692A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-methoxy-3-{2-(piperidin-1-yl)-2-oxo-ethoxy}-phenyl]xanthine1.97Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99693A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{3-(2-(hexamethyleneimin-1-yl)-2-oxo-ethoxy)-4-methoxy}-phenyl]xanthine0.797Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99694A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-methoxy-3-{(2-(morpholin-1-yl)-2-oxo-ethoxy}-phenyl]-xanthine14.3Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99695A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[4-methoxy-3-{2-(1-methylpiperazin-4-yl)-2-oxo-ethoxy}-phenyl]xanthine10Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99696A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{3-(2-(imidazol-1-yl)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine4.1Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99697A3CLONEDHUMAN3H-HEMADO1,3-Dimethyl-8-[{3-(2-(homoveratrylamino)-2-oxoethoxy)-4-methoxy}-phenyl]xanthine30Yasdav R et al 2016Jan 15, 2025Jan 15, 2025
99698D2CLONEDRAT[3H]spiperoneDOPAMINE990Luo D et al 2016Jan 15, 2025Jan 28, 2025
99699D2CLONEDRAT[3H]spiperone(-)-5-OH-DPAT153Luo D et al 2016Jan 15, 2025Jan 28, 2025
99700D2CLONEDRAT[3H]spiperone(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol175Luo D et al 2016Jan 15, 2025Jan 28, 2025
99701D2CLONEDRAT[3H]spiperone(S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol68.3Luo D et al 2016Jan 15, 2025Jan 28, 2025
99702D2CLONEDRAT[3H]spiperone4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol116Luo D et al 2016Jan 15, 2025Jan 28, 2025
99703D2CLONEDRAT[3H]spiperone(S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol65.7Luo D et al 2016Jan 15, 2025Jan 28, 2025
99704D2CLONEDHUMAN[3H]spiperone2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,4-diol117Luo D et al 2016Jan 15, 2025Jan 28, 2025
99705D2CLONEDRAT[3H]spiperone(S)-2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,4-diol112Luo D et al 2016Jan 15, 2025Jan 28, 2025
99706D2CLONEDHUMAN[3H]spiperone(Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol233Luo D et al 2016Jan 15, 2025Jan 28, 2025
99707D2CLONEDRAT[3H]spiperone(S)-4-(5-((5-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)pentyl)benzene-1,2-diol4.67Luo D et al 2016Jan 15, 2025Jan 28, 2025
99708D2CLONEDRAT[3H]spiperone(E)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol150Luo D et al 2016Jan 15, 2025Jan 28, 2025
99709D2CLONEDRAT[3H]spiperone(S,E)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol123Luo D et al 2016Jan 15, 2025Jan 28, 2025
99710D2CLONEDRAT[3H]spiperone4-(6-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)hexyl)-2-methoxyphenol58.5Luo D et al 2016Jan 15, 2025Jan 28, 2025
99711D2CLONEDRAT[3H]spiperone4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)propyl)-2-methoxyphenol2404Luo D et al 2016Jan 15, 2025Jan 28, 2025
99712D2CLONEDRAT[3H]spiperone4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)propyl)benzene-1,2-diol499Luo D et al 2016Jan 15, 2025Jan 28, 2025
99713D2CLONEDRAT[3H]spiperone(E)-4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)prop-1-en-1-yl)-2-methoxyphenol4634Luo D et al 2016Jan 15, 2025Jan 28, 2025
99714D2CLONEDRAT[3H]spiperone(Z)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)benzene-1,2-diol and (Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)cyclohexa-3,5-diene-1,2-dione121Luo D et al 2016Jan 15, 2025Jan 28, 2025
99715D3CLONEDRAT[3H]spiperoneDOPAMINE101Luo D et al 2016Jan 15, 2025Jan 28, 2025
99716D3CLONEDRAT[3H]spiperone(-)-5-OH-DPAT2.07Luo D et al 2016Jan 15, 2025Jan 28, 2025
99717D3CLONEDRAT[3H]spiperone(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol3.62Luo D et al 2016Jan 15, 2025Jan 28, 2025
99718D3CLONEDRAT[3H]spiperone(S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)-2-methoxyphenol1.57Luo D et al 2016Jan 15, 2025Jan 28, 2025
99719D3CLONEDRAT[3H]spiperone4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol2.59Luo D et al 2016Jan 15, 2025Jan 28, 2025
99720D3CLONEDHUMAN[3H]spiperone(S)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,2-diol1.42Luo D et al 2016Jan 15, 2025Jan 28, 2025
99721D3CLONEDHUMAN[3H]spiperone2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,4-diol1.01Luo D et al 2016Jan 15, 2025Jan 28, 2025
99722D3CLONEDHUMAN[3H]spiperone(S)-2-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pentyl)benzene-1,4-diol0.78Luo D et al 2016Jan 15, 2025Jan 28, 2025
99723D3CLONEDRAT[3H]spiperone(Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol23.3Luo D et al 2016Jan 15, 2025Jan 28, 2025
99724D3CLONEDHUMAN[3H]spiperone(S)-4-(5-((5-Hydroxy-1,2,3,4-tetrahydronaphthalen-2-yl)(propyl)amino)pentyl)benzene-1,2-diol0.493Luo D et al 2016Jan 15, 2025Jan 28, 2025
99725D3CLONEDRAT[3H]spiperone(E)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol4.24Luo D et al 2016Jan 15, 2025Jan 28, 2025
99726D3CLONEDRAT[3H]spiperone(S,E)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)-2-methoxyphenol22.3Luo D et al 2016Jan 15, 2025Jan 28, 2025
99727D3CLONEDRAT[3H]spiperone4-(6-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)hexyl)-2-methoxyphenol0.675Luo D et al 2016Jan 15, 2025Jan 28, 2025
99728D3CLONEDHUMAN[3H]spiperone4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)propyl)-2-methoxyphenol15.8Luo D et al 2016Jan 15, 2025Jan 28, 2025
99729D3CLONEDRAT[3H]spiperone4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)propyl)benzene-1,2-diol11.9Luo D et al 2016Jan 15, 2025Jan 28, 2025
99730D3CLONEDRAT[3H]spiperone(E)-4-(3-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)prop-1-en-1-yl)-2-methoxyphenol39.1Luo D et al 2016Jan 15, 2025Jan 28, 2025
99731D3CLONEDRAT[3H]spiperone(Z)-4-(5-((2-Amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)benzene-1,2-diol and (Z)-4-(5-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)pent-1-en-1-yl)cyclohexa-3,5-diene-1,2-dione25Luo D et al 2016Jan 15, 2025Jan 28, 2025
99732MORCLONEDRAT3H-DAMGO(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide88Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99733MORCLONEDRAT3H-DAMGO(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl] propyl}-Nmethylpropanamide7Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99734MORCLONEDRAT3H-DAMGO(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide16Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99735MORCLONEDRAT3H-DAMGO(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide12Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99736MORCLONEDRAT3H-DAMGO(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide1Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99737MORCLONEDRAT3H-DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4- chloroph enyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4- tetrahydroisoquinoline-335Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99738MORCLONEDRAT3H-DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4- chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3- carboxamide10Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99739MORCLONEDRAT3H-DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car7Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99740MORCLONEDRAT3H-DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide0.4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99741MORCLONEDRAT3H-DAMGOYaGF-NH22.8Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99742MORCLONEDRAT3H-DAMGO[D-Ala2, Leu5] enkephalin amide7.7Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99743DORCLONEDHUMAN3H-DPDPE[D-Ala2, Leu5] enkephalin amide2.4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99744DORCLONEDHUMAN3H-DPDPEYaGF-NH2300Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99745DORCLONEDHUMAN3H-DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide13Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99746DORCLONEDHUMAN3H-DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car0.91Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99747DORCLONEDHUMAN3H-DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4- chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3- carboxamide0.88Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99748DORCLONEDHUMAN3H-DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4- chloroph enyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4- tetrahydroisoquinoline-320Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025