The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 33,001-34,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
35465EP4CLONEDHUMAN3H-PGE2AH-6809>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35466EP4CLONEDHUMAN3H-PGE2Butaprost (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35467EP4CLONEDHUMAN3H-PGE2Butaprost (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35468EP4CLONEDHUMAN3H-PGE2SULPROSTONE7740Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35469EP4CLONEDHUMAN3H-PGE2M&B-2876710Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35470EP4CLONEDHUMAN3H-PGE2GR 63799149Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35471EP4CLONEDHUMAN3H-PGE2ENPROSTIL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35472EP4CLONEDHUMAN3H-PGE2MISOPROSTOL (Free Acid)23Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35473EP4CLONEDHUMAN3H-PGE2MISOPROSTOL (Methyl Ester)5499Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35474EP4CLONEDHUMAN3H-PGE2PGD21483Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35475EP4CLONEDHUMAN3H-PGE2BW245C132Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35476EP4CLONEDHUMAN3H-PGE2ZK11084141Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35477EP4CLONEDHUMAN3H-PGE2PGF2Alpha288Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35478EP4CLONEDHUMAN3H-PGE2FLUPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35479EP4CLONEDHUMAN3H-PGE2CLOPROSTENOL9137Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35480EP4CLONEDHUMAN3H-PGE2LATANOPROST (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35481EP4CLONEDHUMAN3H-PGE2Latanoprost (Isopropyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35482EP4CLONEDHUMAN3H-PGE2ILOPROST284Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35483EP4CLONEDHUMAN3H-PGE2CICAPROST44Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35484EP4CLONEDHUMAN3H-PGE2CARBACYCLIN352Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35485EP4CLONEDHUMAN3H-PGE2SQ 29548>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35486EP4CLONEDHUMAN3H-PGE2U466192013Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35487EP4CLONEDHUMAN3H-PGE2AH-23848>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35488EP4CLONEDHUMAN3H-PGE2AH-23848,(-)9287Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35489DP1CLONEDHUMAN3H-PGD2PGE2307Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35490DP1CLONEDHUMAN3H-PGD2SC-51322>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35491DP1CLONEDHUMAN3H-PGD2SC-51089>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35492DP1CLONEDHUMAN3H-PGD2AH-68091415Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35493DP1CLONEDHUMAN3H-PGD2Butaprost (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35494DP1CLONEDHUMAN3H-PGD2Butaprost (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35495DP1CLONEDHUMAN3H-PGD2SULPROSTONE>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35496DP1CLONEDHUMAN3H-PGD2M&B-28767>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35497DP1CLONEDHUMAN3H-PGD2GR 63799>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35498DP1CLONEDHUMAN3H-PGD2ENPROSTIL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35499DP1CLONEDHUMAN3H-PGD2MISOPROSTOL (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35500DP1CLONEDHUMAN3H-PGD2MISOPROSTOL (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35501DP1CLONEDHUMAN3H-PGD2PGD21.7Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35502DP1CLONEDHUMAN3H-PGD2BW245C0.4Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35503DP1CLONEDHUMAN3H-PGD2ZK1108410.3Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35504DP1CLONEDHUMAN3H-PGD2PGF2Alpha861Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35505DP1CLONEDHUMAN3H-PGD2FLUPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35506DP1CLONEDHUMAN3H-PGD2CLOPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35507DP1CLONEDHUMAN3H-PGD2LATANOPROST (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35508DP1CLONEDHUMAN3H-PGD2Latanoprost (Isopropyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35509DP1CLONEDHUMAN3H-PGD2ILOPROST1035Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35510DP1CLONEDHUMAN3H-PGD2CICAPROST1340Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35511DP1CLONEDHUMAN3H-PGD2CARBACYCLIN132Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35512DP1CLONEDHUMAN3H-PGD2SQ 29548>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35513DP1CLONEDHUMAN3H-PGD2U466193970Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35514DP1CLONEDHUMAN3H-PGD2AH-238481380Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35515DP1CLONEDHUMAN3H-PGD2AH-23848,(-)697Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35516PTGFRCLONEDHUMAN3H-PGF2AlphaPGE2119Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35517PTGFRCLONEDHUMAN3H-PGF2AlphaSC-51322>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35518PTGFRCLONEDHUMAN3H-PGF2AlphaSC-51089>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35519PTGFRCLONEDHUMAN3H-PGF2AlphaAH-6809>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35520PTGFRCLONEDHUMAN3H-PGF2AlphaButaprost (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35521PTGFRCLONEDHUMAN3H-PGF2AlphaButaprost (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35522PTGFRCLONEDHUMAN3H-PGF2AlphaSULPROSTONE198Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35523PTGFRCLONEDHUMAN3H-PGF2AlphaM&B-28767510Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35524PTGFRCLONEDHUMAN3H-PGF2AlphaGR 637991241Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35525PTGFRCLONEDHUMAN3H-PGF2AlphaENPROSTIL88Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35526PTGFRCLONEDHUMAN3H-PGF2AlphaMISOPROSTOL (Free Acid)9382Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35527PTGFRCLONEDHUMAN3H-PGF2AlphaMISOPROSTOL (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35528PTGFRCLONEDHUMAN3H-PGF2AlphaPGD26.7Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35529PTGFRCLONEDHUMAN3H-PGF2AlphaBW245C>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35530PTGFRCLONEDHUMAN3H-PGF2AlphaZK1108411670Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35531PTGFRCLONEDHUMAN3H-PGF2AlphaPGF2Alpha3.2Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35532PTGFRCLONEDHUMAN3H-PGF2AlphaFLUPROSTENOL2.3Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35533PTGFRCLONEDHUMAN3H-PGF2AlphaCLOPROSTENOL0.47Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35534PTGFRCLONEDHUMAN3H-PGF2AlphaLATANOPROST (Free Acid)2.8Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35535PTGFRCLONEDHUMAN3H-PGF2AlphaLatanoprost (Isopropyl Ester)555Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35536PTGFRCLONEDHUMAN3H-PGF2AlphaILOPROST619Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35537PTGFRCLONEDHUMAN3H-PGF2AlphaCICAPROST1340Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35538PTGFRCLONEDHUMAN3H-PGF2AlphaCARBACYCLIN427Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35539PTGFRCLONEDHUMAN3H-PGF2AlphaSQ 29548>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35540PTGFRCLONEDHUMAN3H-PGF2AlphaU46619241Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35541PTGFRCLONEDHUMAN3H-PGF2AlphaAH-23848>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35542PTGFRCLONEDHUMAN3H-PGF2AlphaAH-23848,(-)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35543IPCLONEDHUMAN3H-ILOPROSTPGE2>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35544IPCLONEDHUMAN3H-ILOPROSTSC-51322>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35545IPCLONEDHUMAN3H-ILOPROSTSC-51089>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35546IPCLONEDHUMAN3H-ILOPROSTAH-6809>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35547IPCLONEDHUMAN3H-ILOPROSTButaprost (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35548IPCLONEDHUMAN3H-ILOPROSTButaprost (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35549IPCLONEDHUMAN3H-ILOPROSTSULPROSTONE>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35550IPCLONEDHUMAN3H-ILOPROSTM&B-28767>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35551IPCLONEDHUMAN3H-ILOPROSTGR 63799>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35552IPCLONEDHUMAN3H-ILOPROSTENPROSTIL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35553IPCLONEDHUMAN3H-ILOPROSTMISOPROSTOL (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35554IPCLONEDHUMAN3H-ILOPROSTMISOPROSTOL (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35555IPCLONEDHUMAN3H-ILOPROSTPGD2>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35556IPCLONEDHUMAN3H-ILOPROSTBW245C>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35557IPCLONEDHUMAN3H-ILOPROSTZK1108412138Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35558IPCLONEDHUMAN3H-ILOPROSTPGF2Alpha>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35559IPCLONEDHUMAN3H-ILOPROSTFLUPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35560IPCLONEDHUMAN3H-ILOPROSTCLOPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35561IPCLONEDHUMAN3H-ILOPROSTLATANOPROST (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35562IPCLONEDHUMAN3H-ILOPROSTLatanoprost (Isopropyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35563IPCLONEDHUMAN3H-ILOPROSTILOPROST11Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35564IPCLONEDHUMAN3H-ILOPROSTCICAPROST17Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35565IPCLONEDHUMAN3H-ILOPROSTCARBACYCLIN275Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35566IPCLONEDHUMAN3H-ILOPROSTSQ 29548>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35567IPCLONEDHUMAN3H-ILOPROSTU46619>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35568IPCLONEDHUMAN3H-ILOPROSTAH-23848>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35569IPCLONEDHUMAN3H-ILOPROSTAH-23848,(-)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35570CLONEDHUMAN3H-SQ 29548PGE2>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35571CLONEDHUMAN3H-SQ 29548SC-51322507Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35572CLONEDHUMAN3H-SQ 29548SC-51089>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35573CLONEDHUMAN3H-SQ 29548AH-68094325Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35574CLONEDHUMAN3H-SQ 29548Butaprost (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35575CLONEDHUMAN3H-SQ 29548Butaprost (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35576CLONEDHUMAN3H-SQ 29548SULPROSTONE>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35577CLONEDHUMAN3H-SQ 29548M&B-28767343Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35578CLONEDHUMAN3H-SQ 29548GR 63799>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35579CLONEDHUMAN3H-SQ 29548ENPROSTIL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35580CLONEDHUMAN3H-SQ 29548MISOPROSTOL (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35581CLONEDHUMAN3H-SQ 29548MISOPROSTOL (Methyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35582CLONEDHUMAN3H-SQ 29548PGD26602Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35583CLONEDHUMAN3H-SQ 29548BW245C>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35584CLONEDHUMAN3H-SQ 29548ZK1108411121Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35585CLONEDHUMAN3H-SQ 29548PGF2Alpha8700Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35586CLONEDHUMAN3H-SQ 29548FLUPROSTENOL>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35587CLONEDHUMAN3H-SQ 29548CLOPROSTENOL6123Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35588CLONEDHUMAN3H-SQ 29548LATANOPROST (Free Acid)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35589CLONEDHUMAN3H-SQ 29548Latanoprost (Isopropyl Ester)>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35590CLONEDHUMAN3H-SQ 29548ILOPROST6487Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35591CLONEDHUMAN3H-SQ 29548CICAPROST1340Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35592CLONEDHUMAN3H-SQ 29548CARBACYCLIN>10000Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35593CLONEDHUMAN3H-SQ 29548SQ 295484.1Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35594CLONEDHUMAN3H-SQ 29548U4661935Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35595CLONEDHUMAN3H-SQ 29548AH-23848592Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35596CLONEDHUMAN3H-SQ 29548AH-23848,(-)330Abramovitz M, et al., 2000Jan 15, 2025Jan 15, 2025
35597D2CLONEDHUMAN3H-SPIPERONE10-(4-methylpiperazino)-5H-dibenz[b,f]oxepin21Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35598D2CLONEDHUMAN3H-SPIPERONELOXAPINE21Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35599D2CLONEDHUMAN3H-SPIPERONE10-[1-methyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin230Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35600D2CLONEDHUMAN3H-SPIPERONE1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin61Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35601D2CLONEDHUMAN3H-SPIPERONE1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin110Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35602D2CLONEDHUMAN3H-SPIPERONE10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin82Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35603D2CLONEDHUMAN3H-SPIPERONERISPERIDONE1.4Phillips ST, et. al., 1995Jan 15, 2025Jan 27, 2025
35604D4CLONEDHUMAN3H-SPIROPERIDOL10-(4-methylpiperazino)-5H-dibenz[b,f]oxepin2Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35605D4CLONEDHUMAN3H-SPIROPERIDOLLOXAPINE4.9Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35606D4CLONEDHUMAN3H-SPIROPERIDOL10-[1-methyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin29Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35607D4CLONEDHUMAN3H-SPIROPERIDOL1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin26Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35608D4CLONEDHUMAN3H-SPIROPERIDOL1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin37Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35609D4CLONEDHUMAN3H-SPIROPERIDOL10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin9.5Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35610D4CLONEDHUMAN3H-SPIROPERIDOLRISPERIDONE7Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356115-HT2ACLONEDRAT125I-LSD10-(4-methylpiperazino)-5H-dibenz[b,f]oxepin4Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356125-HT2ACLONEDRAT125I-LSD10-[1-methyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin6Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356135-HT2ACLONEDRAT125I-LSD1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin6Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356145-HT2ACLONEDRAT125I-LSD1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin22Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356155-HT2ACLONEDRAT125I-LSD10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin3Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356165-HT2ACLONEDRAT125I-LSDRISPERIDONE0.16Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356175-HT2CCLONEDRAT125I-LSD10-(4-methylpiperazino)-5H-dibenz[b,f]oxepin6Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356185-HT2CCLONEDRAT125I-LSD10-[1-methyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin20Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356195-HT2CCLONEDRAT125I-LSD1-ethyl-1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin14Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356205-HT2CCLONEDRAT125I-LSD1-(2-propenyl)-1,2,3,6-tetrahydro-4-pyridinyl]dibenz[b,f]oxepin51Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
356215-HT2CCLONEDRAT125I-LSD10-(1-methyl-4-piperidinyl)dibenz[b,f]oxepin8Phillips ST, et. al., 1995Jan 15, 2025Jan 15, 2025
35622STRIATUMRAT3H-SPIPERONEtrans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinone4.2Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35623D2STRIATUMRAT3H-SPIPERONEtrans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinone930Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35624STRIATUMRAT3H-PRAZOSINtrans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinone33Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35625STRIATUMRAT3H-SPIPERONEirindalone3.4Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35626D2STRIATUMRAT3H-SPIPERONEirindalone400Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35627STRIATUMRAT3H-PRAZOSINirindalone26Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35628STRIATUMRAT3H-SPIPERONEtrans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione4.9Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35629STRIATUMRAT3H-SPIPERONEtrans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2(lH)-pyrimidinone11Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35630STRIATUMRAT3H-SPIPERONEtrans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine30Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35631D2STRIATUMRAT3H-SPIPERONEtrans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine1900Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35632STRIATUMRAT3H-PRAZOSINtrans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine100Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35633STRIATUMRAT3H-SPIPERONEKETANSERIN1.7Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35634D2STRIATUMRAT3H-SPIPERONEKETANSERIN1800Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35635STRIATUMRAT3H-PRAZOSINKETANSERIN15Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35636STRIATUMRAT3H-SPIPERONEPRAZOSIN>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35637D2STRIATUMRAT3H-SPIPERONEPRAZOSIN>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35638STRIATUMRAT3H-PRAZOSINPRAZOSIN0.36Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35639STRIATUMRAT3H-SPIPERONEtefludazine8.4Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35640D2STRIATUMRAT3H-SPIPERONEtefludazine16Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35641STRIATUMRAT3H-PRAZOSINtefludazine17Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35642STRIATUMRAT3H-SPIPERONERITANSERIN4.4Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35643D2STRIATUMRAT3H-SPIPERONERITANSERIN12Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35644STRIATUMRAT3H-PRAZOSINRITANSERIN47Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35645NETBRAINRAT3H-Norepinephrineirindalone>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35646NETBRAINRAT3H-Norepinephrine(-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone69Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35647NETBRAINRAT3H-Norepinephrine(+)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine450Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35648NETBRAINRAT3H-Norepinephrine(-)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine140Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35649SLC6A3BRAINRAT3H-dopamineirindalone>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35650SLC6A3BRAINRAT3H-dopamine(-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone140Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35651SLC6A3BRAINRAT3H-dopamine(+)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine280Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35652SLC6A3BRAINRAT3H-dopamine(-)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine220Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35653SLC6A4BRAINRAT3H-5HTirindalone>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35654SLC6A4BRAINRAT3H-5HT(-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone9700Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35655SLC6A4BRAINRAT3H-5HT(+)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine42Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35656SLC6A4BRAINRAT3H-5HT(-)-trans - 1-[ 3-(4-Fluorophenyl)indan-l-yl]piperazine400Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35657BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexa-hydropyrazino[1,2-a]quinolin-3-yl)butyl]amide1710Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35658D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexa-hydropyrazino[1,2-a]quinolin-3-yl)butyl]amide585Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35659D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexa-hydropyrazino[1,2-a]quinolin-3-yl)butyl]amide19Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35660BRAINRAT3H-SCH23390BP-897636Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35661D2BRAINRAT3H-SPIPERONEBP-897162Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35662D3BRAINRAT3H-PD 128,907BP-8971.1Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35663BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)-butyl]amide258Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35664D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)-butyl]amide180Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35665D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid [4-(1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)-butyl]amide16Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35666BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide2710Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35667D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide644Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35668D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide8.3Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35669BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide6860Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35670D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide659Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35671D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid [4-(7-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide9.3Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35672BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35673D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide>10000Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35674D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide67Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35675BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35676D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide>10000Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35677D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid [4-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide126Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35678BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35679D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide1720Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35680D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide44Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35681BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide4330Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35682D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide990Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35683D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid [4-(9-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide96Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35684BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide7590Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35685D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide312Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35686D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide4.1Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35687BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide1960Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35688D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide88Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35689D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid [4-(10-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)butyl]-amide3.3Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35690BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35691D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35692D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide5.7Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35693BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35694D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35695D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid {4-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]cyclohexyl}amide10Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35696BRAINRAT3H-SCH23390(R)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35697D2BRAINRAT3H-SPIPERONE(R)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35698D3BRAINRAT3H-PD 128,907(R)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}amide4642Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35699BRAINRAT3H-SCH23390(S)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35700D2BRAINRAT3H-SPIPERONE(S)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}amide>10000Ding K, et al., 2005Jan 15, 2025Jan 27, 2025
35701D3BRAINRAT3H-PD 128,907(S)-Naphthalene-2-carboxylic acid {1-[2-(8-methoxy-1,2,4,4a,5,6-hexahydropyrazino[1,2-a]quinolin-3-yl)ethyl]piperidin-4-yl}amide7156Ding K, et al., 2005Jan 15, 2025Jan 15, 2025
35702CXCR4CLONEDUNDEFINED125I-SDF-1C29H41N11O5S2690Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35703CXCR4CLONEDUNDEFINED125I-SDF-1C37H49N11O6S2530Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35704CXCR4CLONEDUNDEFINED125I-SDF-1C30H43N11O5S2>10000Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35705CXCR4CLONEDUNDEFINED125I-SDF-1C38H51N11O6S2>10000Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35706CXCR4CLONEDUNDEFINED125I-SDF-1C31H43N11O5>10000Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35707CXCR4CLONEDUNDEFINED125I-SDF-1C32H46N11O5>10000Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35708CXCR4CLONEDUNDEFINED125I-SDF-1C33H47N11O5>10000Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35709CXCR4CLONEDUNDEFINED125I-SDF-1C39H51N11O6>10000Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35710CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-GLy-D-Tyr-D-Pro-Arg-)1600Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35711CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Pro-Arg-)420Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35712CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-D-Ala-Arg-)230Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35713CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-D-MeAla-Arg-)42Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35714CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Ala-Arg-)63Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35715CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-MeAla-Arg-)490Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35716CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Dab-Arg-)16Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35717CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Orn-Arg-)19Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35718CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Lys-Arg-)97Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35719CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-g-Dab-Arg-)24Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35720CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-g-Lys-Arg-)33Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35721CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Asn-Arg-)270Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35722CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Gln-Arg-)170Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35723CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-Glu-Arg-)610Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35724CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-trans-4-guanadino-Pro-Arg-)10Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35725CXCR4CLONEDUNDEFINED125I-SDF-1cyclo(-Nal-Gly-D-Tyr-cis-4-guanidino-Pro-Arg-)9.9Tamamura H, et al., 2005Jan 15, 2025Jan 15, 2025
35726UNDEFINEDHUMANUNDEFINEDmethyl-3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H--1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoate acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35727UNDEFINEDHUMANUNDEFINEDethyl-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoyl}amino)acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35728UNDEFINEDHUMANUNDEFINED(2S)-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)amino]-2-benzyl-3-oxopropanoyl}amino)pentanedioic acid acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35729UNDEFINEDHUMANUNDEFINED(3S)-3-({[2-({4-[amino(imino)methyl]benzyl}oxy)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}carbonyl}amino)-3-phenylpropanoate acetate3700Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35730UNDEFINEDHUMANUNDEFINEDmethyl-3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H--1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoate acetate5300Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35731UNDEFINEDHUMANUNDEFINEDethyl-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoyl}amino)acetate8400Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35732UNDEFINEDHUMANUNDEFINED(2S)-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)amino]-2-benzyl-3-oxopropanoyl}amino)pentanedioic acid acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35733UNDEFINEDHUMANUNDEFINED(3S)-3-({[2-({4-[amino(imino)methyl]benzyl}oxy)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}carbonyl}amino)-3-phenylpropanoate acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35734UNDEFINEDHUMANUNDEFINEDmethyl-3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H--1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoate acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35735UNDEFINEDHUMANUNDEFINEDethyl-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}amino]-2-benzyl-3-oxopropanoyl}amino)acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35736UNDEFINEDHUMANUNDEFINED(2S)-2-({3-[(4-{4-[amino(imino)methyl]benzyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)amino]-2-benzyl-3-oxopropanoyl}amino)pentanedioic acid acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35737UNDEFINEDHUMANUNDEFINED(3S)-3-({[2-({4-[amino(imino)methyl]benzyl}oxy)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl}carbonyl}amino)-3-phenylpropanoate acetate>10000Stefanic Anderluh P, et al., 2005Jan 15, 2025Jan 15, 2025
35738Alpha2ACLONEDHUMAN3H-RAUWOLSCINEA-804262.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35739Alpha2ACLONEDHUMAN3H-RAUWOLSCINES-343245.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35740Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole2.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35741Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35742Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35743Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35744Alpha2BCLONEDHUMAN3H-RAUWOLSCINEA-8042611Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35745Alpha2BCLONEDHUMAN3H-RAUWOLSCINES-3432423Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35746Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole14Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35747Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35748Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole14Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35749Alpha2BCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole14Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35750Alpha2CCLONEDHUMAN3H-RAUWOLSCINEA-804262.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35751Alpha2CCLONEDHUMAN3H-RAUWOLSCINES-3432419Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35752Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35753Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35754Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35755Alpha2CCLONEDHUMAN3H-RAUWOLSCINE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35756SLC6A4CLONEDHUMAN3H-PAROXETINEA-804264Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35757SLC6A4CLONEDHUMAN3H-PAROXETINES-3432477Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35758SLC6A4CLONEDHUMAN3H-PAROXETINE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35759SLC6A4CLONEDHUMAN3H-PAROXETINE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole5.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35760SLC6A4CLONEDHUMAN3H-PAROXETINE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole4.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35761SLC6A4CLONEDHUMAN3H-PAROXETINE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35762CLONEDHUMAN3H-PRAZOSINA-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35763CLONEDHUMAN3H-PRAZOSINS-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35764CLONEDHUMAN3H-PRAZOSIN(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35765CLONEDHUMAN3H-PRAZOSIN(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole380Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35766CLONEDHUMAN3H-PRAZOSIN(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35767CLONEDHUMAN3H-PRAZOSIN(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357685-HT2ACLONEDHUMAN125I-R091150A-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357695-HT2ACLONEDHUMAN125I-R091150S-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357705-HT2ACLONEDHUMAN125I-R091150(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357715-HT2ACLONEDHUMAN125I-R091150(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357725-HT2ACLONEDHUMAN125I-R091150(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357735-HT2ACLONEDHUMAN125I-R091150(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357745-HT2CCLONEDHUMAN3H-MESULERGINEA-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357755-HT2CCLONEDHUMAN3H-MESULERGINES-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357765-HT2CCLONEDHUMAN3H-MESULERGINE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357775-HT2CCLONEDHUMAN3H-MESULERGINE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357785-HT2CCLONEDHUMAN3H-MESULERGINE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357795-HT2CCLONEDHUMAN3H-MESULERGINE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357805-HT1ACLONEDHUMAN3H-8-OH-DPATA-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357815-HT1ACLONEDHUMAN3H-8-OH-DPATS-34324770Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357825-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357835-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole475Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357845-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357855-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357865-HT7CLONEDHUMAN3H-5HTS-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357875-HT7CLONEDHUMAN3H-5HT(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357885-HT7CLONEDHUMAN3H-5HT(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357895-HT7CLONEDHUMAN3H-5HT(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
357905-HT7CLONEDHUMAN3H-5HT(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35791H1CLONEDHUMAN3H-PYRILAMINEA-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35792H1CLONEDHUMAN3H-PYRILAMINES-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35793H1CLONEDHUMAN3H-PYRILAMINE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35794H1CLONEDHUMAN3H-PYRILAMINE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole113Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35795H1CLONEDHUMAN3H-PYRILAMINE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35796H1CLONEDHUMAN3H-PYRILAMINE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole460Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35797D2CLONEDHUMAN3H-SPIPERONEA-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35798D2CLONEDHUMAN3H-SPIPERONES-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35799D2CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole959Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35800D2CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole230Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35801D2CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35802D2CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35803D3CLONEDHUMAN125I-IODOSULPRIDE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole270Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35804D3CLONEDHUMAN125I-IODOSULPRIDE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole433Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35805D3CLONEDHUMAN125I-IODOSULPRIDE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole611Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35806D3CLONEDHUMAN125I-IODOSULPRIDE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole107Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35807D4CLONEDHUMAN3H-SPIPERONEA-80426234Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35808D4CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35809D4CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35810D4CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35811D4CLONEDHUMAN3H-SPIPERONE(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35812SLC6A3FR. CORTEXRAT3H-WIN 35,428A-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35813SLC6A3FR. CORTEXRAT3H-WIN 35,428S-343241000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35814SLC6A3FR. CORTEXRAT3H-WIN 35,428(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole515Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35815SLC6A3FR. CORTEXRAT3H-WIN 35,428(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35816SLC6A3FR. CORTEXRAT3H-WIN 35,428(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole368Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35817SLC6A3FR. CORTEXRAT3H-WIN 35,428(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole246Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35818NETFR. CORTEXRAT3H-NisoxetineA-804261000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35819NETFR. CORTEXRAT3H-NisoxetineS-34324365Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35820NETFR. CORTEXRAT3H-Nisoxetine(+)-7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole132Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35821NETFR. CORTEXRAT3H-Nisoxetine(+)-7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole177Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35822NETFR. CORTEXRAT3H-Nisoxetine(+)-7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole220Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35823NETFR. CORTEXRAT3H-Nisoxetine(+)-7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole33Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35824Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole8.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35825Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole6.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35826SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole8.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35827Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35828Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35829SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole2.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35830Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35831Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35832SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole10Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35833Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35834Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole3.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35835SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)-piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35836Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole20Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35837Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole15Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35838SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole84Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35839Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole2.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35840Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole9.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35841SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(Naphthalen-2-ylmethyl-piperazin-1-ylmethyl)]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole0.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35842Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35843Alpha2CCLONEDHUMAN3H-RAUWOLSCINE5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole4.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35844SLC6A4CLONEDHUMAN3H-PAROXETINE5-Methyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole16Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35845Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide20Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35846Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide2.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35847SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid Ethylamide23Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35848Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester33Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35849Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester9.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35850SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole-5-carboxylic Acid ethyl Ester2.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35851Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole47Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35852Alpha2CCLONEDHUMAN3H-RAUWOLSCINE5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole11Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35853SLC6A4CLONEDHUMAN3H-PAROXETINE5-Acetyl-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole61Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35854Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-(2,2,2-Trifluoroacetyl)-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole26Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35855Alpha2CCLONEDHUMAN3H-RAUWOLSCINE5-(2,2,2-Trifluoroacetyl)-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole6.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35856SLC6A4CLONEDHUMAN3H-PAROXETINE5-(2,2,2-Trifluoroacetyl)-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole15Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35857Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole7.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35858Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole5.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35859SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole9.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35860Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole2.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35861Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole0.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35862SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole8.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35863Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole6.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35864Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole3.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35865SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(3-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole15Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35866Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35867Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole23Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35868SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(4-Chlorobenzyl)piperazin-1-ylmethyl]-7,8-dimethoxy-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole141Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35869Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole74Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35870Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole12Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35871SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35872Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(quinolin-6-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35873Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(quinolin-6-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1000Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35874SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(quinolin-6-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole22Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35875Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(2-phenoxyethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole9.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35876Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-3-[4-(2-phenoxyethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole1.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35877SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-3-[4-(2-phenoxyethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole154Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35878Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-5-methyl-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole11Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35879Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7,8-Dimethoxy-5-methyl-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35880SLC6A4CLONEDHUMAN3H-PAROXETINE7,8-Dimethoxy-5-methyl-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydroquinolino[4,3-c]isoxazole104Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35881Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole43Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35882Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole112Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35883SLC6A4CLONEDHUMAN3H-PAROXETINE3-[4-(3-Phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole106Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35884Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-Methoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole1.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35885Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-Methoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole3.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35886SLC6A4CLONEDHUMAN3H-PAROXETINE7-Methoxy-3-[4-(3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole7.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35887Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-Methoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole1.8Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35888Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-Methoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole6.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35889SLC6A4CLONEDHUMAN3H-PAROXETINE7-Methoxy-3-[4-(naphthalen-2-ylmethyl)piperazin-1-ylmethyl]-3,3a,4,5-tetrahydronaphtho[4,3-c]isoxazole1.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35890Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-Hydroxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35891Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-Hydroxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35892SLC6A4CLONEDHUMAN3H-PAROXETINE7-Hydroxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole3.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35893Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-(2-Methoxyethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ymethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35894Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-(2-Methoxyethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ymethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.03Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35895SLC6A4CLONEDHUMAN3H-PAROXETINE7-(2-Methoxyethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ymethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole4.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35896Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-[2-(2-Ethoxyethoxy)ethoxy]-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35897Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-[2-(2-Ethoxyethoxy)ethoxy]-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35898SLC6A4CLONEDHUMAN3H-PAROXETINE7-[2-(2-Ethoxyethoxy)ethoxy]-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole17Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35899Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-Cyclopentyloxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole1.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35900Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-Cyclopentyloxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35901SLC6A4CLONEDHUMAN3H-PAROXETINE7-Cyclopentyloxy-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole56Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35902Alpha2ACLONEDHUMAN3H-RAUWOLSCINE7-(2-Dimethylaminoethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35903Alpha2CCLONEDHUMAN3H-RAUWOLSCINE7-(2-Dimethylaminoethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole0.1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35904SLC6A4CLONEDHUMAN3H-PAROXETINE7-(2-Dimethylaminoethoxy)-3-[4-(2-methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazole3.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35905Alpha2ACLONEDHUMAN3H-RAUWOLSCINEAcetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.4Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35906Alpha2CCLONEDHUMAN3H-RAUWOLSCINEAcetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35907SLC6A4CLONEDHUMAN3H-PAROXETINEAcetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester7.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35908Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPropionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35909Alpha2CCLONEDHUMAN3H-RAUWOLSCINEPropionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35910SLC6A4CLONEDHUMAN3H-PAROXETINEPropionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester21Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35911Alpha2ACLONEDHUMAN3H-RAUWOLSCINEMethoxyacetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35912Alpha2CCLONEDHUMAN3H-RAUWOLSCINEMethoxyacetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.2Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35913SLC6A4CLONEDHUMAN3H-PAROXETINEMethoxyacetic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester5.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35914Alpha2ACLONEDHUMAN3H-RAUWOLSCINECyclopropanecarboxylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35915Alpha2CCLONEDHUMAN3H-RAUWOLSCINECyclopropanecarboxylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.3Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35916SLC6A4CLONEDHUMAN3H-PAROXETINECyclopropanecarboxylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester26Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35917Alpha2ACLONEDHUMAN3H-RAUWOLSCINEAcrylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.9Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35918Alpha2CCLONEDHUMAN3H-RAUWOLSCINEAcrylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester0.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35919SLC6A4CLONEDHUMAN3H-PAROXETINEAcrylic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester41Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35920Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,2-Dimethyl-propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester4.7Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35921Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2,2-Dimethyl-propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester1.6Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35922SLC6A4CLONEDHUMAN3H-PAROXETINE2,2-Dimethyl-propionic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester12Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35923Alpha2ACLONEDHUMAN3H-RAUWOLSCINEIsonicotinic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 1Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35924Alpha2CCLONEDHUMAN3H-RAUWOLSCINEIsonicotinic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 0.5Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35925SLC6A4CLONEDHUMAN3H-PAROXETINEIsonicotinic Acid 3-[4-(2-Methyl-3-phenyl-2(E)-propen-1-yl)piperazin-1-ylmethyl]-3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazol-7-yl Ester 13Andres JI, et al., 2005Jan 15, 2025Jan 15, 2025
35926STRIATUMRAT3H-SPIPERONE(-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone570Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35927D2STRIATUMRAT3H-SPIPERONE(-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35928STRIATUMRAT3H-PRAZOSIN(-)-trans-1-[2-[4-[3-(4-Fluorophenyl)-l-indanyll-l-piperazinyl]ethyl]-2-imidazolidinone540Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35929STRIATUMRAT3H-SPIPERONE(+)-trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione2.2Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35930D2STRIATUMRAT3H-SPIPERONE(+)-trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione29Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35931STRIATUMRAT3H-PRAZOSIN(+)-trans-1-[2-[4-[3-(4-Fluorophenyl)-6-fluoro-l-indanyl]-l-piperazinyl]ethyl]-2-imidazolidinethione13Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35932STRIATUMRAT3H-SPIPERONE(+)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine18Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35933D2STRIATUMRAT3H-SPIPERONE(+)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine580Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35934STRIATUMRAT3H-PRAZOSIN(+)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine37Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35935STRIATUMRAT3H-SPIPERONE(-)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine180Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35936D2STRIATUMRAT3H-SPIPERONE(-)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine8500Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35937STRIATUMRAT3H-PRAZOSIN(-)-trans-1-[3-(4-Fluorophenyl)indan-1-yl]piperazine540Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35938STRIATUMRAT3H-KETANSERIN1-[2-(4-Benzyl-1-piperazinyl)ethyl]-2-imidazolidinone1000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35939D2STRIATUMRAT3H-SPIPERONE1-[2-(4-Benzyl-1-piperazinyl)ethyl]-2-imidazolidinone1000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35940STRIATUMRAT3H-PRAZOSIN1-[2-(4-Benzyl-1-piperazinyl)ethyl]-2-imidazolidinone>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35941STRIATUMRAT3H-KETANSERIN1-[2-(4-Benzoyl-1-piperazinyl)ethyl]-2-imidazolidinone4800Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35942D2STRIATUMRAT3H-SPIPERONE1-[2-(4-Benzoyl-1-piperazinyl)ethyl]-2-imidazolidinone1000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35943STRIATUMRAT3H-KETANSERIN1-[2-[4-(1-Indanyl)-1-piperazinyl]ethyl]-2-imidazolidinone5100Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
35944D2STRIATUMRAT3H-SPIPERONE1-[2-[4-(1-Indanyl)-1-piperazinyl]ethyl]-2-imidazolidinone>10000Bogeso KP, et al., 1988Jan 15, 2025Jan 15, 2025
359455-HT2ABRAIN CORTEXRAT3H-KETANSERIN4-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine2.15Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359465-HT2ABRAIN CORTEXRAT3H-KETANSERIN11-(4-Methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine7.25Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359475-HT2ABRAIN CORTEXRAT3H-KETANSERIN8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine1.35Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359485-HT2ABRAIN CORTEXRAT3H-KETANSERIN3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine4.99Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359495-HT2ABRAIN CORTEXRAT3H-KETANSERINOLANZAPINE4Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359505-HT2ABRAIN CORTEXRAT3H-KETANSERINST18990.65Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359515-HT2ABRAIN CORTEXRAT3H-KETANSERINHALOPERIDOL164Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35952D1STRIATUMRAT3H-SCH233904-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine4.91Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35953D1STRIATUMRAT3H-SCH2339011-(4-Methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine125Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35954D1STRIATUMRAT3H-SCH233908-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine47.4Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35955D1STRIATUMRAT3H-SCH233903-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine230Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359565-HT2ABRAIN CORTEXRAT3H-KETANSERINCLOZAPINE10Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35957D1STRIATUMRAT3H-SCH23390OLANZAPINE85Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35958D1STRIATUMRAT3H-SCH23390CLOZAPINE353Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35959D1STRIATUMRAT3H-SCH23390ST189919.7Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35960D1STRIATUMRAT3H-SCH23390HALOPERIDOL318Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35961D2STRIATUMRAT3H-SPIPERONE4-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine8.4Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35962D2STRIATUMRAT3H-SPIPERONE11-(4-Methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine578Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35963D2STRIATUMRAT3H-SPIPERONE8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine71.1Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35964D2STRIATUMRAT3H-SPIPERONE3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine923Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35965D2STRIATUMRAT3H-SPIPERONEOLANZAPINE69Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35966D2STRIATUMRAT3H-SPIPERONECLOZAPINE250Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35967D2STRIATUMRAT3H-SPIPERONEST189917.2Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35968D2STRIATUMRAT3H-SPIPERONEHALOPERIDOL4.8Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35969D3Sf9RAT3H-7-OH-DPAT4-(4-Methyipiperazino)pyrrolo[2,1-b]thieno[3,2-f][1,3]thiazepine25Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35970D3Sf9RAT3H-7-OH-DPAT11-(4-Methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine224Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35971D3Sf9RAT3H-7-OH-DPAT8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine24.2Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35972D3Sf9RAT3H-7-OH-DPAT3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine88.6Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35973D3Sf9RAT3H-7-OH-DPATOLANZAPINE39Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35974D3Sf9RAT3H-7-OH-DPATCLOZAPINE319Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35975D3Sf9RAT3H-7-OH-DPATST18998.3Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35976D3Sf9RAT3H-7-OH-DPATHALOPERIDOL18Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359775-HT2CBRAIN CORTEXGUINEA PIG3H-MESULERGINE8-Chloro-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine3.8Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
359785-HT2CBRAIN CORTEXGUINEA PIG3H-MESULERGINE3-Methyl-11-(4-methylpiperazin-1-yl)-5H-pyrrolo[2,1-b][2]benzazepine15Campiani G, et al., 2005Jan 15, 2025Jan 15, 2025
35979FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(4-chlorobenzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline31van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35980FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(tert-butoxymethylcarbonyl)aminophenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline76van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35981FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(2-furoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline27van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35982FSHCLONEDHUMAN3H-hFSH1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(4-[trifluoromethyl]-benzoyl)amino-2,2,4-trimethylquinoline7van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35983FSHCLONEDHUMAN3H-hFSH1-Acetyl-4-phenyl-6-(4-n-propylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline5van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35984FSHCLONEDHUMAN3H-hFSH1-Acetyl-4-phenyl-6-(4-phenylbenzoyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline28van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35985FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(4-[4-tert-butylphenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline74van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35986FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(4-[3-phenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline9van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35987FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(4-[2-phenyl]benzoyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline25van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35988FSHCLONEDHUMAN3H-hFSH1-Acetyl-4-phenyl-1,2,3,4-tetrahydro-6-(alpha-toluenesulfonyl)amino-2,2,4-trimethylquinoline2800van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35989FSHCLONEDHUMAN3H-hFSH1-Acetyl-4-phenyl-6-(phenylaminocarbonyl)amino-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline580van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35990FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(4-tert-butylbenzyl)amino-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline930van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35991FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-phenylethoxy-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline80van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35992FSHCLONEDHUMAN3H-hFSH1-Acetyl-6-(2-[4-methoxyphenyl]ethylamino)carbonyl-4-phenyl-1,2,3,4-tetrahydro-2,2,4-trimethylquinoline1880van Straten NC, et al., 2005Jan 15, 2025Jan 15, 2025
35993A1BRAINRAT3H-CCPA8-Cyclopentyl-3-(1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-ylmethyl)-1-propylxanthine5.47Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
35994A1BRAINRAT3H-CCPA8-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)-1,3-dipropylxanthine8.23Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
35995A1BRAINRAT3H-CCPA8-(1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)-1,3-dipropylxanthine160Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
35996A1BRAINRAT3H-CCPA3-benzyl-5-cyclopentyl-1-propylxanthine8.7Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
35997A1BRAINRAT3H-CCPADPCPX0.9Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
35998A2ABRAINRAT3H-MSX-28-Cyclopentyl-3-(1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-ylmethyl)-1-propylxanthine8780Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
35999A2ABRAINRAT3H-MSX-28-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)-1,3-dipropylxanthine3800Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36000A2ABRAINRAT3H-MSX-28-(1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)-1,3-dipropylxanthine6750Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36001A2ABRAINRAT3H-MSX-23-benzyl-5-cyclopentyl-1-propylxanthine511Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36002A2ABRAINRAT3H-MSX-2DPCPX470Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36003A2BCLONEDHUMAN3H-PSB-2988-Cyclopentyl-3-(1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-ylmethyl)-1-propylxanthine1000Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36004A2BCLONEDHUMAN3H-PSB-2988-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)-1,3-dipropylxanthine3100Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36005A2BCLONEDHUMAN3H-PSB-2988-(1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)-1,3-dipropylxanthine>10000Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36006A2BCLONEDHUMAN3H-PSB-298DPCPX51Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36007A3CLONEDHUMAN3H-PSB-118-Cyclopentyl-3-(1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-ylmethyl)-1-propylxanthine1700Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36008A3CLONEDHUMAN3H-PSB-118-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)-1,3-dipropylxanthine>10000Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36009A3CLONEDHUMAN3H-PSB-118-(1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)-1,3-dipropylxanthine>10000Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36010A3CLONEDHUMAN3H-PSB-113-benzyl-5-cyclopentyl-1-propylxanthine54.6Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36011A3CLONEDHUMAN3H-PSB-11DPCPX795Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36012A1BRAINRAT3H-CCPA8-[4-(((1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)amino)-2-oxoethoxy)phenyl]-1-propylxanthine15.7Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36013A2ABRAINRAT3H-MSX-28-[4-(((1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)amino)-2-oxoethoxy)phenyl]-1-propylxanthine1270Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36014A2BCLONEDHUMAN3H-PSB-2988-[4-(((1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)amino)-2-oxoethoxy)phenyl]-1-propylxanthine48Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36015A3CLONEDHUMAN3H-PSB-118-[4-(((1-Oxyl-2,2,6,6-tetramethylpiperidin-4-yl)amino)-2-oxoethoxy)phenyl]-1-propylxanthine350Ilas J, et al., 2005Jan 15, 2025Jan 15, 2025
36016BRAINRAT3H-3-PPP,(+)3PPP,(+)30Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36017BRAINRAT3H-3-PPP,(+)3PPP,(-)155Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36018BRAINRAT3H-3-PPP,(+)HALOPERIDOL2.4Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36019BRAINRAT3H-3-PPP,(+)BUTACLAMOL,(+)1800Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36020BRAINRAT3H-3-PPP,(+)BUTACLAMOL, (-)157Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36021BRAINRAT3H-3-PPP,(+)PERPHENAZINE24Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36022BRAINRAT3H-3-PPP,(+)FLUPHENAZINE62Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36023BRAINRAT3H-3-PPP,(+)SPIPERONE632Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36024BRAINRAT3H-3-PPP,(+)PIMOZIDE508Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36025BRAINRAT3H-3-PPP,(+)SKF 10047 (+/-)373Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36026BRAINRAT3H-3-PPP,(+)SKF 10,047 (+)343Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36027BRAINRAT3H-3-PPP,(+)SKF 10,047 (-)1350Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36028BRAINRAT3H-3-PPP,(+)Cyclazocine96Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36029BRAINRAT3H-3-PPP,(+)Cyclazocine (+)111Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36030BRAINRAT3H-3-PPP,(+)CYCLAZOCINE (-)408Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36031BRAINRAT3H-3-PPP,(+)Pentazocine,(+/-)23Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36032BRAINRAT3H-3-PPP,(+)PENTAZOCINE (-)29Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36033BRAINRAT3H-3-PPP,(+)Dextrallorphan154Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36034BRAINRAT3H-3-PPP,(+)Levallorphan1780Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36035BRAINRAT3H-3-PPP,(+)Dextromethorphan768Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36036BRAINRAT3H-3-PPP,(+)PHENCYCLIDINE711Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36037BRAINRAT3H-3-PPP,(+)Dexoxadrol1880Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36038BRAINRAT3H-3-PPP,(+)Levoxadrol2080Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36039BRAINRAT3H-Haloperidol3PPP,(+)58Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36040BRAINRAT3H-Haloperidol3PPP,(-)162Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36041BRAINRAT3H-HaloperidolHALOPERIDOL2Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36042BRAINRAT3H-HaloperidolBUTACLAMOL,(+)955Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36043BRAINRAT3H-HaloperidolBUTACLAMOL, (-)85Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36044BRAINRAT3H-HaloperidolPERPHENAZINE13Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36045BRAINRAT3H-HaloperidolSKF 10047 (+/-)516Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36046BRAINRAT3H-HaloperidolSKF 10,047 (+)319Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36047BRAINRAT3H-HaloperidolSKF 10,047 (-)1860Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36048BRAINRAT3H-HaloperidolCyclazocine180Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36049BRAINRAT3H-HaloperidolCyclazocine (+)149Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36050BRAINRAT3H-HaloperidolCYCLAZOCINE (-)504Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36051BRAINRAT3H-HaloperidolPentazocine,(+/-)43Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36052BRAINRAT3H-HaloperidolDextrallorphan78Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36053BRAINRAT3H-HaloperidolLevallorphan1060Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36054BRAINRAT3H-HaloperidolPHENCYCLIDINE956Largent BL, et al., 1984Jan 15, 2025Jan 15, 2025
36055MORMembranesRAT3H-DAMGO14-O-Allyloxymorphone0.61Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36056MORMembranesRAT3H-DAMGO14-O-Benzyloxymorphone0.12Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36057MORMembranesRAT3H-DAMGO14-Benzyloxymetopon0.18Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36058MORMembranesRAT3H-DAMGO14-O-(1-naphthylmethyl)oxymorphone0.18Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36059MORMembranesRAT3H-DAMGO14-O-(2,6-dichlorobenzyloxy)oxymorphone10.3Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36060MORMembranesRAT3H-DAMGO14-ethoxy-3-hydroxy-5-methyl- 17-(2-phenylethyl)morphinan-6-one0.16Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36061MORMembranesRAT3H-DAMGO14-O-methyloxymorphone0.1Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36062MORMembranesRAT3H-DAMGO14-methoxymetopon0.15Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36063MORMembranesRAT3H-DAMGOOxymorphone0.97Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36064MORMembranesRAT3H-DAMGOMorphine6.55Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36065DORMembranesRAT3H-[Ile5,6]deltorphin II14-O-Allyloxymorphone36Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36066DORMembranesRAT3H-[Ile5,6]deltorphin II14-O-Benzyloxymorphone2.14Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36067DORMembranesRAT3H-[Ile5,6]deltorphin II14-Benzyloxymetopon3.67Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36068DORMembranesRAT3H-[Ile5,6]deltorphin II14-O-(1-naphthylmethyl)oxymorphone2.92Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36069DORMembranesRAT3H-[Ile5,6]deltorphin II14-O-(2,6-dichlorobenzyloxy)oxymorphone152Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36070DORMembranesRAT3H-[Ile5,6]deltorphin II14-ethoxy-3-hydroxy-5-methyl- 17-(2-phenylethyl)morphinan-6-one3.14Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36071DORMembranesRAT3H-[Ile5,6]deltorphin II14-O-methyloxymorphone4.8Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36072DORMembranesRAT3H-[Ile5,6]deltorphin II14-methoxymetopon13.3Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36073DORMembranesRAT3H-[Ile5,6]deltorphin IIOxymorphone80.5Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36074DORMembranesRAT3H-[Ile5,6]deltorphin IIMorphine217Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36075KORMembranesRAT3H-U69,59314-O-Allyloxymorphone33.8Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36076KORMembranesRAT3H-U69,59314-O-Benzyloxymorphone1.18Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36077KORMembranesRAT3H-U69,59314-Benzyloxymetopon2.46Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36078KORMembranesRAT3H-U69,59314-O-(1-naphthylmethyl)oxymorphone0.92Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36079KORMembranesRAT3H-U69,59314-O-(2,6-dichlorobenzyloxy)oxymorphone33.2Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36080KORMembranesRAT3H-U69,59314-ethoxy-3-hydroxy-5-methyl- 17-(2-phenylethyl)morphinan-6-one83.2Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36081KORMembranesRAT3H-U69,59314-O-methyloxymorphone10.2Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36082KORMembranesRAT3H-U69,59314-methoxymetopon25.2Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36083KORMembranesRAT3H-U69,593Oxymorphone61.6Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36084KORMembranesRAT3H-U69,593Morphine113Lattanzi R, et al., 2005Jan 15, 2025Jan 15, 2025
36085COS-1whole blood assay (WBA)HUMANFunctionalAcetylsalicylic acid1700Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36086COS-1whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt75Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36087COS-1whole blood assay (WBA)HUMANFunctionalibuprofen7600Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36088COS-1whole blood assay (WBA)HUMANFunctionalKetorolac tris salt0.19Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36089COS-1whole blood assay (WBA)HUMANFunctionalNaproxen9300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36090COS-1whole blood assay (WBA)HUMANFunctionalPiroxicam2400Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36091COS-1whole blood assay (WBA)HUMANFunctionalMeloxicam sodium5700Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36092COS-1whole blood assay (WBA)HUMANFunctionalnimesulide>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36093COS-1whole blood assay (WBA)HUMANFunctionalvaleryl salicylate>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36094COX-2whole blood assay (WBA)HUMANFunctionalAcetylsalicylic acid>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36095COX-2whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt38Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36096COX-2whole blood assay (WBA)HUMANFunctionalibuprofen7200Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36097COX-2whole blood assay (WBA)HUMANFunctionalKetorolac tris salt86Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36098COX-2whole blood assay (WBA)HUMANFunctionalNaproxen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36099COX-2whole blood assay (WBA)HUMANFunctionalPiroxicam7900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36100COX-2whole blood assay (WBA)HUMANFunctionalMeloxicam sodium2100Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36101COX-2whole blood assay (WBA)HUMANFunctionalnimesulide1900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36102COX-2whole blood assay (WBA)HUMANFunctionalROFECOXIB840Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36103COX-2whole blood assay (WBA)HUMANFunctionalvaleryl salicylate2300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36104COS-1whole blood assay (WBA)HUMANFunctionalROFECOXIB>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36105COX-2WHMAHUMANFunctionalAcetylsalicylic acid7500Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36106COX-2WHMAHUMANFunctionalDiclofenac sodium salt20Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36107COX-2WHMAHUMANFunctionalibuprofen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36108COX-2WHMAHUMANFunctionalKetorolac tris salt75Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36109COX-2WHMAHUMANFunctionalNaproxen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36110COX-2WHMAHUMANFunctionalPiroxicam170Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36111COX-2WHMAHUMANFunctionalMeloxicam sodium230Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36112COX-2WHMAHUMANFunctionalnimesulide390Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36113COX-2WHMAHUMANFunctionalROFECOXIB310Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36114EP2CHO (COX-2)cellsHUMANFunctionalETORICOXIB79Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36115EP2CHO (COX-1)cellsHUMANFunctionalETORICOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36116CA2+ plateletsHUMANFunctionalETORICOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36117COX-2purifiedHUMANFunctionalETORICOXIB5000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36118COX-2purified w/detergentHUMANFunctionalETORICOXIB4100Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36119COS-1purified low substrateHUMANFunctionalETORICOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36120EP2U937HUMANFunctionalETORICOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36121COX-2whole blood assay (WBA)HUMANFunctionalETORICOXIB1100Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36122COS-1whole blood assay (WBA)HUMANFunctionalETORICOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36123EP2CHO (COX-2)cellsHUMANFunctionalIndomethacin27Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36124EP2CHO (COX-1)cellsHUMANFunctionalIndomethacin18Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36125CA2+ plateletsHUMANFunctionalIndomethacin2Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36126COX-2purifiedHUMANFunctionalIndomethacin600Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36127COX-2purified w/detergentHUMANFunctionalIndomethacin400Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36128EP2U937HUMANFunctionalIndomethacin19.8Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36129COX-2whole blood assay (WBA)HUMANFunctionalIndomethacin440Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36130COS-1whole blood assay (WBA)HUMANFunctionalIndomethacin190Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36131COS-1recombinantHUMANFunctionalCELECOXIB>10000Talley JJ, et. al., 2000Jan 15, 2025Jan 15, 2025
36132COX-2recombinantHUMANFunctionalCELECOXIB40Talley JJ, et. al., 2000Jan 15, 2025Jan 15, 2025
36133COS-1recombinantHUMANFunctionalVALDECOXIB>10000Talley JJ, et. al., 2000Jan 15, 2025Jan 15, 2025
36134COX-2recombinantHUMANFunctionalVALDECOXIB5Talley JJ, et. al., 2000Jan 15, 2025Jan 15, 2025
36135COS-1recombinantHUMANFunctionalPARECOXIB>10000Talley JJ, et. al., 2000aJan 15, 2025Jan 15, 2025
36136COX-2recombinantHUMANFunctionalPARECOXIB>10000Talley JJ, et. al., 2000aJan 15, 2025Jan 15, 2025
36137COS-1whole blood assay (WBA)HUMANFunctionalETORICOXIB>10000Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36138COS-1whole blood assay (WBA)HUMANFunctionalCELECOXIB>10000Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36139COS-1whole blood assay (WBA)HUMANFunctionalROFECOXIB>10000Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36140COS-1whole blood assay (WBA)HUMANFunctional3-[4-(methylsulfonyl)phenyl]-5-(trifluoromethyl)(2-pyridyl) phenyl ketone>10000Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36141COX-2whole blood assay (WBA)HUMANFunctional3-[4-(methylsulfonyl)phenyl]-5-(trifluoromethyl)(2-pyridyl) phenyl ketone250Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36142COX-2whole blood assay (WBA)HUMANFunctionalETORICOXIB2000Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36143COX-2whole blood assay (WBA)HUMANFunctionalCELECOXIB1200Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36144COX-2whole blood assay (WBA)HUMANFunctionalROFECOXIB500Khanapure SP, et al., 2005Jan 15, 2025Jan 15, 2025
36145COS-1whole blood assay (WBA)HUMANFunctionalROFECOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36146COS-1whole blood assay (WBA)HUMANFunctionalVALDECOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36147COS-1whole blood assay (WBA)HUMANFunctionalCELECOXIB6700Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36148COS-1whole blood assay (WBA)HUMANFunctionalnimesulide4100Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36149COS-1whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt150Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36150COS-1whole blood assay (WBA)HUMANFunctionalEtodolac9000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36151COS-1whole blood assay (WBA)HUMANFunctionalMeloxicam sodium1400Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36152COS-1whole blood assay (WBA)HUMANFunctionalibuprofen4800Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36153COS-1whole blood assay (WBA)HUMANFunctional6MNA>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36154COS-1whole blood assay (WBA)HUMANFunctionalPiroxicam760Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36155COS-1whole blood assay (WBA)HUMANFunctionalJTE-522>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36156COX-2whole blood assay (WBA)HUMANFunctionalROFECOXIB530Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36157COX-2whole blood assay (WBA)HUMANFunctionalVALDECOXIB870Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36158COX-2whole blood assay (WBA)HUMANFunctionalCELECOXIB870Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36159COX-2whole blood assay (WBA)HUMANFunctionalnimesulide560Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36160COX-2whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt50Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36161COX-2whole blood assay (WBA)HUMANFunctionalEtodolac3700Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36162COX-2whole blood assay (WBA)HUMANFunctionalMeloxicam sodium700Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36163COX-2whole blood assay (WBA)HUMANFunctionalibuprofen>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36164COX-2whole blood assay (WBA)HUMANFunctional6MNA>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36165COX-2whole blood assay (WBA)HUMANFunctionalPiroxicam9000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36166COX-2whole blood assay (WBA)HUMANFunctionalJTE-522>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36167COS-1U937HUMANFunctionalETORICOXIB>10000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36168COS-1U937HUMANFunctionalROFECOXIB2000Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36169COS-1U937HUMANFunctionalEtodolac1200Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36170COS-1U937HUMANFunctionalVALDECOXIB250Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36171COS-1U937HUMANFunctionalMeloxicam sodium140Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36172COS-1U937HUMANFunctionalnimesulide120Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36173COS-1U937HUMANFunctionalCELECOXIB52Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36174COS-1U937HUMANFunctionalDiclofenac sodium salt7Riendeau D, et.al., 2001Jan 15, 2025Jan 15, 2025
36175COS-1whole blood assay (WBA)HUMANFunctional6MNA>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36176COS-1whole blood assay (WBA)HUMANFunctionalCarprofen87Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36177COS-1whole blood assay (WBA)HUMANFunctionalFenoprofen3400Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36178COS-1whole blood assay (WBA)HUMANFunctionalFlufenamate3000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36179COS-1whole blood assay (WBA)HUMANFunctionalFlubiprofen75Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36180COS-1whole blood assay (WBA)HUMANFunctionalIndomethacin13Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36181COS-1whole blood assay (WBA)HUMANFunctionalKetoprofen47Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36182COS-1whole blood assay (WBA)HUMANFunctionalMeclofenamate220Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36183COS-1whole blood assay (WBA)HUMANFunctionalMefenamic acid>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36184COS-1whole blood assay (WBA)HUMANFunctionalNiflumic acid>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36185COS-1whole blood assay (WBA)HUMANFunctionalSulindac sulphide1900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36186COS-1whole blood assay (WBA)HUMANFunctionalSuprofen1100Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36187COS-1whole blood assay (WBA)HUMANFunctionalTenidap81Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36188COS-1whole blood assay (WBA)HUMANFunctionalTolmetin350Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36189COS-1whole blood assay (WBA)HUMANFunctionalTomoxiprol7600Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36190COS-1whole blood assay (WBA)HUMANFunctionalZomepirac430Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36191COS-1whole blood assay (WBA)HUMANFunctionalCELECOXIB1200Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36192COS-1whole blood assay (WBA)HUMANFunctionalEtodolac>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36193COS-1whole blood assay (WBA)HUMANFunctionalDiisopropyl fluorophosphate>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36194COS-1whole blood assay (WBA)HUMANFunctionalL745,337>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36195COS-1whole blood assay (WBA)HUMANFunctionalNS3986900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36196COS-1whole blood assay (WBA)HUMANFunctionalSC58125>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36197COS-1whole blood assay (WBA)HUMANFunctional5-Aminosalicylic acid>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36198COS-1whole blood assay (WBA)HUMANFunctionalAmpyrone>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36199COS-1whole blood assay (WBA)HUMANFunctionalDiflunisal>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36200COS-1whole blood assay (WBA)HUMANFunctionalNabumetone>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36201COS-1whole blood assay (WBA)HUMANFunctionalParacetamol>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36202COS-1whole blood assay (WBA)HUMANFunctionalResveratrol>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36203COS-1whole blood assay (WBA)HUMANFunctionalSalicin>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36204COS-1whole blood assay (WBA)HUMANFunctionalSalicylaldehyde>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36205COS-1whole blood assay (WBA)HUMANFunctionalSodium salicylate>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36206COS-1whole blood assay (WBA)HUMANFunctionalSulfasalazine>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36207COS-1whole blood assay (WBA)HUMANFunctionalSulindac>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36208COS-1whole blood assay (WBA)HUMANFunctionalTamoxifen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36209COS-1whole blood assay (WBA)HUMANFunctionalTiclopidine>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36210COX-2whole blood assay (WBA)HUMANFunctional6MNA>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36211COX-2whole blood assay (WBA)HUMANFunctionalCarprofen4300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36212COX-2whole blood assay (WBA)HUMANFunctionalFenoprofen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36213COX-2whole blood assay (WBA)HUMANFunctionalFlufenamate9300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36214COX-2whole blood assay (WBA)HUMANFunctionalFlubiprofen5500Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36215COX-2whole blood assay (WBA)HUMANFunctionalIndomethacin1000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36216COX-2whole blood assay (WBA)HUMANFunctionalKetoprofen2900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36217COX-2whole blood assay (WBA)HUMANFunctionalMeclofenamate700Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36218COX-2whole blood assay (WBA)HUMANFunctionalMefenamic acid2900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36219COX-2whole blood assay (WBA)HUMANFunctionalNiflumic acid5400Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36220COX-2whole blood assay (WBA)HUMANFunctionalSulindac sulphide>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36221COX-2whole blood assay (WBA)HUMANFunctionalSuprofen8700Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36222COX-2whole blood assay (WBA)HUMANFunctionalTenidap2900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36223COX-2whole blood assay (WBA)HUMANFunctionalTolmetin820Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36224COX-2whole blood assay (WBA)HUMANFunctionalTomoxiprol>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36225COX-2whole blood assay (WBA)HUMANFunctionalZomepirac810Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36226COX-2whole blood assay (WBA)HUMANFunctionalCELECOXIB830Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36227COX-2whole blood assay (WBA)HUMANFunctionalEtodolac2200Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36228COX-2whole blood assay (WBA)HUMANFunctionalDiisopropyl fluorophosphate760Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36229COX-2whole blood assay (WBA)HUMANFunctionalL745,3378600Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36230COX-2whole blood assay (WBA)HUMANFunctionalNS398350Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36231COX-2whole blood assay (WBA)HUMANFunctionalSC581252000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36232COX-2whole blood assay (WBA)HUMANFunctional5-Aminosalicylic acid>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36233COX-2whole blood assay (WBA)HUMANFunctionalAmpyrone>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36234COX-2whole blood assay (WBA)HUMANFunctionalDiflunisal8200Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36235COX-2whole blood assay (WBA)HUMANFunctionalNabumetone>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36236COX-2whole blood assay (WBA)HUMANFunctionalParacetamol>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36237COX-2whole blood assay (WBA)HUMANFunctionalResveratrol>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36238COX-2whole blood assay (WBA)HUMANFunctionalSalicin>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36239COX-2whole blood assay (WBA)HUMANFunctionalSalicylaldehyde>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36240COX-2whole blood assay (WBA)HUMANFunctionalSodium salicylate>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36241COX-2whole blood assay (WBA)HUMANFunctionalSulfasalazine>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36242COX-2whole blood assay (WBA)HUMANFunctionalSulindac>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36243COX-2whole blood assay (WBA)HUMANFunctionalTamoxifen>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36244COX-2whole blood assay (WBA)HUMANFunctionalTiclopidine>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36245COX-2WHMAHUMANFunctionalFenoprofen5900Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36246COX-2WHMAHUMANFunctionalFlubiprofen770Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36247COX-2WHMAHUMANFunctionalIndomethacin130Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36248COX-2WHMAHUMANFunctionalKetoprofen240Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36249COX-2WHMAHUMANFunctionalMeclofenamate200Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36250COX-2WHMAHUMANFunctionalMefenamic acid1300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36251COX-2WHMAHUMANFunctionalNiflumic acid>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36252COX-2WHMAHUMANFunctionalSulindac sulphide1210Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36253COX-2WHMAHUMANFunctionalSuprofen8300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36254COX-2WHMAHUMANFunctionalTolmetin1300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36255COX-2WHMAHUMANFunctionalTomoxiprol320Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36256COX-2WHMAHUMANFunctionalZomepirac96Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36257COX-2WHMAHUMANFunctionalCELECOXIB340Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36258COX-2WHMAHUMANFunctionalEtodolac940Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36259COX-2WHMAHUMANFunctionalDiisopropyl fluorophosphate170Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36260COX-2WHMAHUMANFunctionalL745,3371300Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36261COX-2WHMAHUMANFunctionalNS39842Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36262COX-2WHMAHUMANFunctionalAmpyrone>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36263COX-2WHMAHUMANFunctionalDiflunisal>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36264COX-2WHMAHUMANFunctionalNabumetone>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36265COX-2WHMAHUMANFunctionalParacetamol>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36266COX-2WHMAHUMANFunctionalSodium salicylate>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36267COX-2WHMAHUMANFunctionalSulindac>10000Warner TD, et al., 1999Jan 15, 2025Jan 15, 2025
36268COS-1whole blood assay (WBA)HUMANFunctionalKetoprofen110Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36269COS-1whole blood assay (WBA)HUMANFunctionalIndomethacin210Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36270COS-1whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt260Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36271COS-1whole blood assay (WBA)HUMANFunctionalKetorolac tris salt270Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36272COS-1whole blood assay (WBA)HUMANFunctionalFlubiprofen410Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36273COS-1whole blood assay (WBA)HUMANFunctionalTolmetin1080Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36274COS-1whole blood assay (WBA)HUMANFunctionalMefenamic acid1940Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36275COS-1whole blood assay (WBA)HUMANFunctionalPiroxicam2680Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36276COS-1whole blood assay (WBA)HUMANFunctionalFenoprofen2730Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36277COS-1whole blood assay (WBA)HUMANFunctionalAcetylsalicylic acid4450Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36278COS-1whole blood assay (WBA)HUMANFunctionalibuprofen5900Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36279COS-1whole blood assay (WBA)HUMANFunctionalnimesulide>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36280COS-1whole blood assay (WBA)HUMANFunctionaloxaprosin>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36281COS-1whole blood assay (WBA)HUMANFunctionalEtodolac>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36282COS-1whole blood assay (WBA)HUMANFunctionalNS398>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36283COS-1whole blood assay (WBA)HUMANFunctional6MNA>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36284COS-1whole blood assay (WBA)HUMANFunctionalNaproxen>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36285COS-1whole blood assay (WBA)HUMANFunctionalvaleryl salicylate>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36286COS-1whole blood assay (WBA)HUMANFunctionalNabumetone>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36287COS-1whole blood assay (WBA)HUMANFunctionalSulindac>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36288COS-1whole blood assay (WBA)HUMANFunctionalacetaminophen>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36289COS-1whole blood assay (WBA)HUMANFunctionaldexamethasone>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36290COS-1whole blood assay (WBA)HUMANFunctionalBismuth subsalicylate>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36291COS-1whole blood assay (WBA)HUMANFunctionalsalicylic acid>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36292COS-1whole blood assay (WBA)HUMANFunctionalsalsalate>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36293COX-2whole blood assay (WBA)HUMANFunctionalKetoprofen880Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36294COX-2whole blood assay (WBA)HUMANFunctionalIndomethacin370Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36295COX-2whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt10Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36296COX-2whole blood assay (WBA)HUMANFunctionalKetorolac tris salt180Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36297COX-2whole blood assay (WBA)HUMANFunctionalFlubiprofen4230Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36298COX-2whole blood assay (WBA)HUMANFunctionalTolmetin2250Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36299COX-2whole blood assay (WBA)HUMANFunctionalMefenamic acid160Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36300COX-2whole blood assay (WBA)HUMANFunctionalPiroxicam2110Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36301COX-2whole blood assay (WBA)HUMANFunctionalFenoprofen>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36302COX-2whole blood assay (WBA)HUMANFunctionalAcetylsalicylic acid>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36303COX-2whole blood assay (WBA)HUMANFunctionalibuprofen9900Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36304COX-2whole blood assay (WBA)HUMANFunctionalnimesulide180Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36305COX-2whole blood assay (WBA)HUMANFunctionaloxaprosin>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36306COX-2whole blood assay (WBA)HUMANFunctionalEtodolac2470Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36307COX-2whole blood assay (WBA)HUMANFunctionalNS398920Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36308COX-2whole blood assay (WBA)HUMANFunctional6MNA>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36309COX-2whole blood assay (WBA)HUMANFunctionalNaproxen>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36310COX-2whole blood assay (WBA)HUMANFunctionalvaleryl salicylate40Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36311COX-2whole blood assay (WBA)HUMANFunctionalNabumetone>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36312COX-2whole blood assay (WBA)HUMANFunctionalSulindac>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36313COX-2whole blood assay (WBA)HUMANFunctionalacetaminophen>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36314COX-2whole blood assay (WBA)HUMANFunctionaldexamethasone130Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36315COX-2whole blood assay (WBA)HUMANFunctionalBismuth subsalicylate>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36316COX-2whole blood assay (WBA)HUMANFunctionalsalicylic acid>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36317COX-2whole blood assay (WBA)HUMANFunctionalsalsalate>10000Cryer B, et al., 1998Jan 15, 2025Jan 15, 2025
36318NMDACORTEXRAT3H-MK-801MK-801,(+)2.5Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36319NMDACORTEXRAT3H-MK-801MK-801,(-)13.7Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36320NMDACORTEXRAT3H-MK-801PCP42.2Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36321NMDACORTEXRAT3H-MK-801Ketamine1190Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36322NMDACORTEXRAT3H-MK-801Memantine690Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36323NMDACORTEXRAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36324NMDACEREBELLUMRAT3H-MK-801MK-801,(+)9.4Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36325NMDACEREBELLUMRAT3H-MK-801MK-801,(-)53.7Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36326NMDACEREBELLUMRAT3H-MK-801PCP180Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36327NMDACEREBELLUMRAT3H-MK-801Ketamine2507Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36328NMDACEREBELLUMRAT3H-MK-801Memantine700Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36329NMDACEREBELLUMRAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36330NMDASTRIATUMRAT3H-MK-801MK-801,(+)6.5Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36331NMDASTRIATUMRAT3H-MK-801MK-801,(-)24.9Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36332NMDASTRIATUMRAT3H-MK-801Memantine433Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36333NMDASTRIATUMRAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36334NMDAparietal cortexRAT3H-MK-801MK-801,(+)8.9Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36335NMDAHIPPOCAMPUS CA1RAT3H-MK-801MK-801,(+)8.4Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36336NMDAHIPPOCAMPUS CA3RAT3H-MK-801MK-801,(+)10.8Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36337NMDAHIPPOCAMPUS DGRAT3H-MK-801MK-801,(+)27.2Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36338NMDASTRIATUMRAT3H-MK-801MK-801,(+)20.4Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36339NMDAparietal cortexRAT3H-MK-801Memantine1730Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36340NMDAHIPPOCAMPUS CA1RAT3H-MK-801Memantine1370Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36341NMDAHIPPOCAMPUS CA3RAT3H-MK-801Memantine1320Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36342NMDAHIPPOCAMPUS DGRAT3H-MK-801Memantine2420Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36343NMDASTRIATUMRAT3H-MK-801Memantine1780Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36344NMDAparietal cortexRAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36345NMDAHIPPOCAMPUS CA1RAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36346NMDAHIPPOCAMPUS CA3RAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36347NMDAHIPPOCAMPUS DGRAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36348NMDASTRIATUMRAT3H-MK-801Amantadine>10000Bresink I, et al., 1995Jan 15, 2025Jan 28, 2025
36349MORBRAINRAT3H-DAMGOMorphine6.55Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36350MORBRAINRAT3H-DAMGO14-O-methyloxymorphone0.1Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36351MORBRAINRAT3H-DAMGO14-methoxymetopon0.15Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36352MORBRAINRAT3H-DAMGOHS378340Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36353DORBRAINRAT3H-[Ile5,6]deltorphin IIMorphine217Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36354DORBRAINRAT3H-[Ile5,6]deltorphin II14-O-methyloxymorphone4.8Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36355DORBRAINRAT3H-[Ile5,6]deltorphin II14-methoxymetopon13.3Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36356DORBRAINRAT3H-[Ile5,6]deltorphin IIHS3780.78Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36357KORBRAINRAT3H-U69,593Morphine113Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36358DORBRAINRAT3H-U69,59314-O-methyloxymorphone10.2Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36359KORBRAINRAT3H-U69,59314-methoxymetopon25.2Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36360KORBRAINRAT3H-U69,593HS378134Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36361MORBRAINRAT3H-DAMGO2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]acetic acid bis(tetrafluoroborate)0.89Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36362MORBRAINRAT3H-DAMGO2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]acetic acid bis(tetrafluoroborate)0.83Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36363MORBRAINRAT3H-DAMGO(2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]propanoic acid bis(tetrafluoroborate)0.77Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36364MORBRAINRAT3H-DAMGO(2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]propanoic acid bis(tetrafluoroborate)1.9Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36365MORBRAINRAT3H-DAMGO(2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]-3-phenylpropanoic acid bis(tetrafluroborate)0.95Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36366MORBRAINRAT3H-DAMGO(2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]-3-phenylpropanoic acid bis(tetrafluoroborate)2.58Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36367DORBRAINRAT3H-[Ile5,6]deltorphin II2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]acetic acid bis(tetrafluoroborate)15.4Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36368DORBRAINRAT3H-[Ile5,6]deltorphin II2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]acetic acid bis(tetrafluoroborate)7.86Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36369DORBRAINRAT3H-[Ile5,6]deltorphin II(2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]propanoic acid bis(tetrafluoroborate)26.9Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36370DORBRAINRAT3H-[Ile5,6]deltorphin II(2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]propanoic acid bis(tetrafluoroborate)7.71Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36371DORBRAINRAT3H-[Ile5,6]deltorphin II(2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]-3-phenylpropanoic acid bis(tetrafluroborate)3.67Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36372DORBRAINRAT3H-[Ile5,6]deltorphin II(2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]-3-phenylpropanoic acid bis(tetrafluoroborate)1.03Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36373KORBRAINRAT3H-U69,5932-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]acetic acid bis(tetrafluoroborate)43.2Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36374KORBRAINRAT3H-U69,5932-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]acetic acid bis(tetrafluoroborate)44.8Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36375KORBRAINRAT3H-U69,593(2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]propanoic acid bis(tetrafluoroborate)142Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36376KORBRAINRAT3H-U69,593(2S)-2-[4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]propanoic acid bis(tetrafluoroborate)63.7Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36377KORBRAINRAT3H-U69,593(2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6beta-yl)amino]-3-phenylpropanoic acid bis(tetrafluoroborate)151Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36378KORBRAINRAT3H-U69,593(2S)-2-[(4,5alpha-epoxy-3-hydroxy-14beta-methoxy-17-methylmorphinan-6alpha-yl)amino]-3-phenylpropanoic acid bis(tetrafluroborate)28.5Spetea M, et al., 2004Jan 15, 2025Jan 15, 2025
36379PlateletsHUMAN3H-SQ 29548SQ 2954821Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36380PlateletsHUMAN3H-SQ 29548BM 5731.3Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36381PlateletsHUMAN3H-SQ 29548BM 6131.4Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36382CLONEDHUMAN3H-SQ 29548BM 5731.1Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36383CLONEDHUMAN3H-SQ 29548BM 6132.1Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36384CLONEDHUMAN3H-SQ 29548BM 5730.8Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36385CLONEDHUMAN3H-SQ 29548BM 6133.1Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36386Coronary arteryHUMAN3H-SQ 29548BM 573>10000Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36387Coronary arteryHUMAN3H-SQ 29548BM 613>10000Hanson J, et al., 2005Jan 15, 2025Jan 15, 2025
36388COS-1U937HUMANFunctionalETORICOXIB>10000Cochrane DJ, et al., 2002Jan 15, 2025Jan 15, 2025
36389COS-1U937HUMANFunctionalROFECOXIB2000Cochrane DJ, et al., 2002Jan 15, 2025Jan 15, 2025
36390COS-1U937HUMANFunctionalVALDECOXIB250Cochrane DJ, et al., 2002Jan 15, 2025Jan 15, 2025
36391COS-1U937HUMANFunctionalCELECOXIB52Cochrane DJ, et al., 2002Jan 15, 2025Jan 15, 2025
36392COS-1PlateletsHUMANFunctionalibuprofen48Weir MR, et al., 2003Jan 15, 2025Jan 15, 2025
36393COS-1PlateletsHUMANFunctionalCELECOXIB210Weir MR, et al., 2003Jan 15, 2025Jan 15, 2025
36394COS-1PlateletsHUMANFunctionalVALDECOXIB700Weir MR, et al., 2003Jan 15, 2025Jan 15, 2025
36395COS-1PlateletsHUMANFunctionalROFECOXIB5300Weir MR, et al., 2003Jan 15, 2025Jan 15, 2025
36396COS-1PlateletsHUMANFunctionalETORICOXIB>10000Weir MR, et al., 2003Jan 15, 2025Jan 15, 2025
36397EP2osteosarcoma cellsHUMANFunctionalROFECOXIB26Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36398EP2U937HUMANFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36399EP2CHO (COX-2)cellsHUMANFunctionalROFECOXIB18Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36400EP2CHO (COX-1)cellsHUMANFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36401EP2CELLSHUMANFunctionalROFECOXIB45Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36402EP2CELLSRATFunctionalROFECOXIB41Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36403EP2Sf9RATFunctionalROFECOXIB46Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36404EP2KIDNEYHUMANFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36405EP2KIDNEYRATFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36406EP2KIDNEYDogFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36407EP2U937HUMANFunctionalROFECOXIB2000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36408COX-2purifiedHUMANFunctionalROFECOXIB340Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36409COX-2purified w/detergentHUMANFunctionalROFECOXIB400Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36410COS-1purified low substrateHUMANFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36411PMNLHUMANFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36412EP2osteosarcoma cellsHUMANFunctionalIndomethacin21Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36413EP2U937HUMANFunctionalIndomethacin7Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36414EP2CHO (COX-2)cellsHUMANFunctionalIndomethacin27Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36415EP2CHO (COX-1)cellsHUMANFunctionalIndomethacin18Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36416EP2CELLSHUMANFunctionalIndomethacin57Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36417EP2Sf9RATFunctionalIndomethacin18Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36418EP2KIDNEYHUMANFunctionalIndomethacin100Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36419EP2KIDNEYRATFunctionalIndomethacin300Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36420EP2KIDNEYDogFunctionalIndomethacin300Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36421EP2U937HUMANFunctionalIndomethacin19.8Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36422COX-2purifiedHUMANFunctionalIndomethacin600Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36423COX-2purified w/detergentHUMANFunctionalIndomethacin400Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36424COS-1whole blood assay (WBA)HUMANFunctionalROFECOXIB>10000Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36425COS-1whole blood assay (WBA)HUMANFunctionalCELECOXIB6300Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36426COS-1whole blood assay (WBA)HUMANFunctionalMeloxicam sodium1400Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36427COS-1whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt150Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36428COS-1whole blood assay (WBA)HUMANFunctionalIndomethacin190Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36429COX-2whole blood assay (WBA)HUMANFunctionalROFECOXIB530Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36430COX-2whole blood assay (WBA)HUMANFunctionalCELECOXIB960Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36431COX-2whole blood assay (WBA)HUMANFunctionalMeloxicam sodium700Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36432COX-2whole blood assay (WBA)HUMANFunctionalDiclofenac sodium salt50Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36433COX-2whole blood assay (WBA)HUMANFunctionalIndomethacin440Chan CC, et al., 1999Jan 15, 2025Jan 15, 2025
36434CLONEDHUMANFunctionalacetazolamide250Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36435CLONEDHUMANFunctionalmethazolamide50Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36436CLONEDHUMANFunctionalethoxzolamide25Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36437CLONEDHUMANFunctionalDichlorphenamide1200Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36438CLONEDHUMANFunctionaldorzolamide>10000Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36439CLONEDHUMANFunctionalindisulam31Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36440CLONEDHUMANFunctional4-carboxybenzenesulfonamide3400Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36441CLONEDHUMANFunctional4-Sulfamoylbenzoic acid hydrazide2950Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36442CLONEDHUMANFunctional4-(N-(3,4-dichlorophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1150Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36443CLONEDHUMANFunctional4-(N-(4-acetylphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1450Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36444CLONEDHUMANFunctional4-(N-(4-ethyloxycarbonylphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfona mide1200Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36445CLONEDHUMANFunctional4-(N-(4-nitrophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide760Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36446CLONEDHUMANFunctional4-(N-(4-bromophenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide865Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36447CLONEDHUMANFunctional4-(N-(4-biphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1160Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36448CLONEDHUMANFunctional4-(N-(4-phenoxyphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1450Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36449CLONEDHUMANFunctional4-(N-(4-benzyloxyphenyl)aminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1300Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36450CLONEDHUMANFunctional4-(N-fluorenylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1360Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36451CLONEDHUMANFunctional4-(N-phenylsulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide1250Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36452CLONEDHUMANFunctional4-(N-(2-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide800Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36453CLONEDHUMANFunctional4-(N-(4-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide700Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36454CLONEDHUMANFunctional4-(N-(4-chlorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide600Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36455CLONEDHUMANFunctional2-carboxymethylbenzenesfulfonamide>10000Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36456CLONEDHUMANFunctional2-Sulfamoylbenzoic acid hydrazide>10000Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36457CLONEDHUMANFunctional2-(N-(2-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide4700Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36458CLONEDHUMANFunctional2-(N-(4-methylphenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide3400Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36459CLONEDHUMANFunctional2-(N-(4-fluorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide4900Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36460CLONEDHUMANFunctional2-(N-(4-chlorophenyl)sulfonylaminocarbonyl-hydrazinocarbonyl)-benzenesulfonamide3600Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36461CLONEDHUMANFunctional4-Hydrazino-3-fluorobenzenesulfonamide3300Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36462CLONEDHUMANFunctional4-Hydrazino-3-chlorobenzenesulfonamide2800Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36463CLONEDHUMANFunctional2-Hydrazinobenzenesulfonamide>10000Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025
36464CLONEDHUMANFunctionalN-Acetyl-2-hydrazinobenzenesulfonamide>10000Winum JY, et al., 2005Jan 15, 2025Jan 15, 2025