41605 SLC6A3 CLONED RAT 3H-WIN 35,428 4,4'-DifluoroBZT 8 Ukairo UT, et al., 2005 Jan 15, 2025 Jan 15, 2025
41606 SLC6A3 CLONED RAT 3H-WIN 35,428 4-TrifluoromethylBZT 541 Ukairo UT, et al., 2005 Jan 15, 2025 Jan 15, 2025
41607 SLC6A3 CLONED RAT 3H-WIN 35,428 N-CHO-4,4'-diFBZT >10000 Ukairo UT, et al., 2005 Jan 15, 2025 Jan 15, 2025
41608 DOR CLONED HUMAN 3H-DADLE N-DESMETHYLCLOZAPINE 127.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41609 KOR CLONED HUMAN 3H-Diprenorphine N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41610 5-HT1A CLONED HUMAN 3H-8-OH-DPAT N-DESMETHYLCLOZAPINE 13.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41611 5-HT1B CLONED HUMAN 3H-GR-125743 N-DESMETHYLCLOZAPINE 406.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41612 5-HT1D CLONED HUMAN 3H-GR-125743 N-DESMETHYLCLOZAPINE 476.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41613 5-HT1E CLONED HUMAN 3H-5HT N-DESMETHYLCLOZAPINE 393.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41614 5-HT2A CLONED HUMAN 3H-KETANSERIN N-DESMETHYLCLOZAPINE 10.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41615 5-HT2C CLONED RAT 3H-MESULERGINE N-DESMETHYLCLOZAPINE 11.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41616 5-HT3 CLONED HUMAN 3H-ZACOPRIDE N-DESMETHYLCLOZAPINE 272.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41617 CB1 CLONED HUMAN 3H-LSD N-DESMETHYLCLOZAPINE 350.6 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
41618 5-HT6 CLONED HUMAN 3H-LSD N-DESMETHYLCLOZAPINE 11.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41619 5-HT7 CLONED HUMAN 3H-LSD N-DESMETHYLCLOZAPINE 60.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41620 5-HT2B CLONED HUMAN 3H-LSD N-DESMETHYLCLOZAPINE 2.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41621 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-DESMETHYLCLOZAPINE 104.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41622 Alpha1B CLONED HUMAN 3H-PRAZOSIN N-DESMETHYLCLOZAPINE 85.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41623 Alpha2A CLONED HUMAN 3H-CLONIDINE N-DESMETHYLCLOZAPINE 137.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41624 Alpha2B CLONED HUMAN 3H-CLONIDINE N-DESMETHYLCLOZAPINE 95.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41625 Alpha2C CLONED HUMAN 3H-CLONIDINE N-DESMETHYLCLOZAPINE 117.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41626 Beta1 CLONED HUMAN 125I-Pindolol N-DESMETHYLCLOZAPINE 6239.04 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41627 Beta2 CLONED HUMAN 125I-Pindolol N-DESMETHYLCLOZAPINE 4725 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
41628 H1 CLONED HUMAN 3H-PYRILAMINE N-DESMETHYLCLOZAPINE 3.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41629 H2 CLONED HUMAN 3H-TIOTIDINE N-DESMETHYLCLOZAPINE 345.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41630 H3 CLONED GUINEA PIG 3H-Alpha-Me-histamine N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41631 H4 CLONED HUMAN 3H-Histamine N-DESMETHYLCLOZAPINE 1028 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41632 D1 CLONED HUMAN 3H-SCH23390 N-DESMETHYLCLOZAPINE 14.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41633 D2 CLONED HUMAN 3H-NMSP N-DESMETHYLCLOZAPINE 115.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41634 D3 CLONED RAT 3H-NMSP N-DESMETHYLCLOZAPINE 234 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41635 D4 CLONED HUMAN 3H-NMSP N-DESMETHYLCLOZAPINE 101.82 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41636 D5 CLONED HUMAN 3H-SCH23390 N-DESMETHYLCLOZAPINE 283.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41637 SLC6A3 CLONED HUMAN 3H-WIN 35,428 N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41638 NET CLONED HUMAN 3H-Nisoxetine N-DESMETHYLCLOZAPINE 493.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41639 M1 CLONED HUMAN 3H-QNB N-DESMETHYLCLOZAPINE 67.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41640 M2 CLONED HUMAN 3H-QNB N-DESMETHYLCLOZAPINE 414.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41641 M3 CLONED HUMAN 3H-QNB N-DESMETHYLCLOZAPINE 95.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41642 M4 CLONED HUMAN 3H-QNB N-DESMETHYLCLOZAPINE 169.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41643 M5 CLONED HUMAN 3H-QNB N-DESMETHYLCLOZAPINE 35.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41645 HEART RAT 3H-Nitrendipine N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41646 CB1 BRAIN RAT 3H-CP-55940 N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41647 CB2 CLONED HUMAN 3H-CP-55940 N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41648 EP3 CLONED HUMAN 3H-PGE2 N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41649 KOR FOREBRAIN RAT 3H-MUSCIMOL N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
41650 I1 PC12 RAT 125I-Pindolol N-DESMETHYLCLOZAPINE 757.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41651 MOR CLONED HUMAN 3H-Diprenorphine N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41652 NMDA FOREBRAIN RAT 3H-MK-801 N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41653 SLC6A4 CLONED HUMAN 3H-CITALOPRAM N-DESMETHYLCLOZAPINE 316.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41654 Sigma 1 BRAIN RAT 3H-Pentazocine(+) N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41655 CLONED HUMAN 3H-VASOPRESSIN N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41656 Sigma 2 PC12 RAT 3H-DTG N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41657 CLONED HUMAN 3H-VASOPRESSIN N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41658 V2 CLONED HUMAN 3H-VASOPRESSIN N-DESMETHYLCLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41668 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ORG-5222 53.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41669 5-HT1B CLONED HUMAN 3H-GR-125743 ORG-5222 5.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41670 5-HT1E CLONED HUMAN 3H-5HT ORG-5222 37.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41671 5-HT2A CLONED HUMAN 3H-KETANSERIN ORG-5222 0.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41672 5-HT2C CLONED RAT 3H-MESULERGINE ORG-5222 0.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41673 5-HT3 CLONED HUMAN 3H-ZACOPRIDE ORG-5222 447.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41674 CB1 CLONED HUMAN 3H-LSD ORG-5222 4 PDSP Certified Data Jan 15, 2025 Jan 27, 2025
41675 5-HT6 CLONED HUMAN 3H-LSD ORG-5222 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41676 5-HT7 CLONED HUMAN 3H-LSD ORG-5222 0.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41677 H2 CLONED HUMAN 3H-TIOTIDINE ORG-5222 2.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41678 H4 CLONED HUMAN 3H-Histamine ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41679 D1 CLONED HUMAN 3H-SCH23390 ORG-5222 2.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41680 D2 CLONED HUMAN 3H-NMSP ORG-5222 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41681 D3 CLONED RAT 3H-NMSP ORG-5222 46.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41682 D4 CLONED HUMAN 3H-NMSP ORG-5222 1.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41683 D5 CLONED HUMAN 3H-SCH23390 ORG-5222 22.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41684 SLC6A3 CLONED HUMAN 3H-WIN 35,428 ORG-5222 3136 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41685 M1 CLONED HUMAN 3H-NMS ORG-5222 782 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41686 M2 CLONED HUMAN 3H-NMS ORG-5222 915 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41687 M3 CLONED HUMAN 3H-NMS ORG-5222 3232 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41688 M4 CLONED HUMAN 3H-QNB ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41689 M5 CLONED HUMAN 3H-NMS ORG-5222 272 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41690 HEART RAT 3H-Nitrendipine ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41691 CB1 BRAIN RAT 3H-CP-55940 ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41692 EP3 CLONED HUMAN 3H-PGE2 ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41693 I1 PC12 RAT 125I-Pindolol ORG-5222 2371 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41694 MOR CLONED HUMAN 3H-Diprenorphine ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41695 NMDA FOREBRAIN RAT 3H-MK-801 ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41696 SLC6A4 CLONED HUMAN 3H-CITALOPRAM ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41697 Sigma 1 BRAIN RAT 3H-Pentazocine(+) ORG-5222 2069 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41698 NET CLONED HUMAN 3H-Nisoxetine ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41699 KOR CLONED HUMAN 3H-Diprenorphine ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41700 Sigma 2 PC12 RAT 3H-DTG ORG-5222 497.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41701 EP4 CLONED HUMAN 3H-PGE2 ORG-5222 >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41702 Alpha1A CLONED HUMAN 3H-PRAZOSIN ORG-5222 4.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41703 Alpha1B CLONED HUMAN 3H-PRAZOSIN ORG-5222 3.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41704 Alpha2A CLONED HUMAN 3H-CLONIDINE ORG-5222 10.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41705 Alpha2B CLONED HUMAN 3H-CLONIDINE ORG-5222 10.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41706 Alpha2C CLONED HUMAN 3H-CLONIDINE ORG-5222 17.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
41707 UNDEFINED UNDEFINED Functional Thiabendazole 472 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41708 UNDEFINED UNDEFINED Functional Carbendazim >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41709 UNDEFINED UNDEFINED Functional 2-Pyridin-3-yl-1H-benzoimidazol >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41710 UNDEFINED UNDEFINED Functional 2-Thiophen-2-yl-1H-benzoimidazol >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41711 UNDEFINED UNDEFINED Functional Fuberidazole >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41712 UNDEFINED UNDEFINED Functional 2-(1H-Benzoimidazol-2-yl)-phenol >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41713 UNDEFINED UNDEFINED Functional 1H-Benzimidazol-2-yl-thiourea 8956 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41714 UNDEFINED UNDEFINED Functional (1H-Benzimidazol-2-yl)-thiazol-2-yl-amin 540 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41715 UNDEFINED UNDEFINED Functional 2-Pyridin-2-yl-1H-benzoimidazol 574 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41716 UNDEFINED UNDEFINED Functional 6-(1H-Benzoimidazol-2-yl)-pyridin-2-ol 1343 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41717 UNDEFINED UNDEFINED Functional 2-(1H-Benzoimidazol-2-yl)-pyridin-3-ol 777 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41718 UNDEFINED UNDEFINED Functional 2-Pyrazin-2-yl-1H-benzoimidazol 4591 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41719 UNDEFINED UNDEFINED Functional 1-Methyl-2-thiazol-4-yl-1H-benzoimidazol 497 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41720 UNDEFINED UNDEFINED Functional 1-Benzyl-2-thiazol-4-yl-1H-benzoimidazole 461 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41721 UNDEFINED UNDEFINED Functional 1-Benzyl-2-pyridin-2-yl-1H-benzoimidazole 992 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41722 UNDEFINED UNDEFINED Functional 5-Methyl-2-thiazol-4-yl-1(3)H-benzoimidazole 7157 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41723 UNDEFINED UNDEFINED Functional 5-Methyl-2-pyridin-2-yl-1(3)H-benzoimidazol 2086 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41724 UNDEFINED UNDEFINED Functional 5,6-Dimethyl-2-thiazol-4-yl-1H-benzoimidazole >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41725 UNDEFINED UNDEFINED Functional 5,6-Dimethyl-2-pyridin-2-yl-1H-benzoimidazole 2433 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41726 UNDEFINED UNDEFINED Functional 5-tert-Butyl-2-thiazol-4-yl-1H-benzimidazol 3906 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41727 UNDEFINED UNDEFINED Functional 5-tert-Butyl-2-pyridin-2-yl-1H-Benzoimidazole 2598 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41728 UNDEFINED UNDEFINED Functional 5-Nitro-2-thiazol-4-yl-1(3)H-benzoimidazole 1218 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41729 UNDEFINED UNDEFINED Functional 5-Nitro-2-pyridin-2-yl-1(3)H-benzoimidazol 162 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41730 UNDEFINED UNDEFINED Functional 5-Amino-2-thiazol-4-yl-1H-benzimidazol 3390 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41731 UNDEFINED UNDEFINED Functional 2-Pyridin-2-yl-3H-benzoimidazol-5-ylamine 967 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41732 UNDEFINED UNDEFINED Functional 5-Fluor-2-thiazol-4-yl-1H-benzimidazol 4307 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41733 UNDEFINED UNDEFINED Functional 6-Fluoro-2-pyridin-2-yl-1H-benzoimidazole 1511 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41734 UNDEFINED UNDEFINED Functional 5-Chlor-2-thiazol-4-yl-1H-benzimidazol 5153 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41735 UNDEFINED UNDEFINED Functional 5-Chloro-2-pyridin-2-yl-1(3)H-benzoimidazole 1695 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41736 UNDEFINED UNDEFINED Functional Phenyl-(2-thiazol-4-yl-1H-benzoimidazol-5-yl)-methanone 2397 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41737 UNDEFINED UNDEFINED Functional Phenyl-(2-pyridin-2-yl-3H-benzoimidazol-5-yl)-methanone 403 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41738 UNDEFINED UNDEFINED Functional 2-Pyridin-2-yl-3H-benzoimidazole-5-carbonitrile 431 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41739 UNDEFINED UNDEFINED Functional Mebendazole >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41740 UNDEFINED UNDEFINED Functional Albendazole >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41741 UNDEFINED UNDEFINED Functional Fenbendazole >10000 Schiffmann R, et al., 2006 Jan 15, 2025 Jan 15, 2025
41742 AMPA CORTICAL MEMBRANES RAT 3H-AMPA AMPA 23 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41743 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate 94 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41744 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41745 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41746 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate 1500 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41747 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate 5800 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41748 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate 700 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41749 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41750 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41751 AMPA CORTICAL MEMBRANES RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate 30 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41752 KA CORTICAL MEMBRANES RAT 3H-Kainic acid AMPA >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41753 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate 4900 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41754 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41755 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41756 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41757 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41758 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41759 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41760 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41761 KA CORTICAL MEMBRANES RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 15, 2025
41762 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 AMPA >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41763 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41764 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41765 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41766 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41767 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41768 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41769 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41770 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41771 NMDA CORTICAL MEMBRANES RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate >10000 Bang-Andersen B, et al., 1997 Jan 15, 2025 Jan 28, 2025
41772 CLONED HUMAN Functional 17beta-Estradiol 0.019 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41773 CLONED HUMAN Functional (+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.059 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41774 CLONED HUMAN Functional 1-ethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.31 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41775 CLONED HUMAN Functional (+/-)-3-Ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxylic Acid 158 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41776 CLONED HUMAN Functional (+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride 100 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41777 CLONED HUMAN Functional (+/-)-N-(4-(2-(Dimethylamino)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide monohydrochloride 152 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41778 CLONED HUMAN Functional (+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide 427 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41779 CLONED HUMAN Functional 2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol 4.3 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41780 CLONED HUMAN Functional 1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol 7 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41781 CLONED HUMAN Functional 1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 3.9 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41782 CLONED HUMAN Functional 1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 17 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41783 CLONED HUMAN Functional 2-(4-Hydroxyphenyl)-1-p-tolyl-3H-inden-5-ol 17 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41784 CLONED HUMAN Functional 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-olol 15 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41785 CLONED HUMAN Functional 1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 6.7 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41786 CLONED HUMAN Functional 1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 109 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41787 CLONED HUMAN Functional 1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 14 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41788 CLONED HUMAN Functional 17beta-Estradiol 0.098 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41789 CLONED HUMAN Functional (+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.3 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41790 CLONED HUMAN Functional 1-ethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.3 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41791 CLONED HUMAN Functional (+/-)-3-Ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxylic Acid 52 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41792 CLONED HUMAN Functional (+/-)-N-(4-(2-(Dimethylamino)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide monohydrochloride 512 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41793 CLONED HUMAN Functional 2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol 54 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41794 CLONED HUMAN Functional 1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 10 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41795 CLONED HUMAN Functional 1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol 37 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41796 CLONED HUMAN 3H-Estradiol OHT 0.04 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41797 CLONED HUMAN 3H-Estradiol raloxifene 0.03 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41798 CLONED HUMAN 3H-Estradiol (+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride 184 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41799 CLONED HUMAN 3H-Estradiol 1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol 8.5 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41800 CLONED HUMAN 3H-Estradiol 1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 1.7 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41801 CLONED HUMAN 3H-Estradiol 1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 24 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41802 CLONED HUMAN 3H-Estradiol 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 2.1 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41803 CLONED HUMAN 3H-Estradiol 1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.67 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41804 CLONED HUMAN 3H-Estradiol 1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 59 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41805 CLONED HUMAN 3H-Estradiol 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzamide 4.2 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41806 CLONED HUMAN 3H-Estradiol Methyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate 7.3 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41807 CLONED HUMAN 3H-Estradiol Tamoxifen, 4-hydroxy 0.014 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41808 CLONED HUMAN 3H-Estradiol raloxifene 4.5 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41809 CLONED HUMAN 3H-Estradiol (+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride 147 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41810 CLONED HUMAN 3H-Estradiol 1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol 1.3 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41811 CLONED HUMAN 3H-Estradiol 1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.19 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41812 CLONED HUMAN 3H-Estradiol 1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 2.8 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41813 CLONED HUMAN 3H-Estradiol 1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.49 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41814 CLONED HUMAN 3H-Estradiol 2-(4-Hydroxyphenyl)-1-p-tolyl-3H-inden-5-ol 1.3 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41815 CLONED HUMAN 3H-Estradiol 1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 0.91 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41816 CLONED HUMAN 3H-Estradiol 1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 2.2 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41817 CLONED HUMAN 3H-Estradiol 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoic Acid 421 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41818 CLONED HUMAN 3H-Estradiol 1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol 15 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41819 CLONED HUMAN 3H-Estradiol 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzamide 0.46 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41820 CLONED HUMAN 3H-Estradiol Methyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate 3.8 Clegg NJ, et al., 2005 Jan 15, 2025 Jan 15, 2025
41821 H3 CLONED HUMAN 3H-Alpha-Me-histamine ABT-239 0.45 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41822 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(2-nitrophenyl)amine 0.31 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41823 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(4-nitrophenyl)amine 0.74 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41824 H3 CLONED HUMAN 3H-Alpha-Me-histamine 2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone 0.74 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41825 H3 CLONED HUMAN 3H-Alpha-Me-histamine 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)benzonitrile 0.4 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41826 H3 CLONED HUMAN 3H-Alpha-Me-histamine (6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 0.31 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41827 H3 CLONED HUMAN 3H-Alpha-Me-histamine 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyrazine-2-carbonitrile 1.04 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41828 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrazin-2-ylamine 0.29 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41829 H3 CLONED HUMAN 3H-Alpha-Me-histamine (5-Bromopyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 1.22 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41830 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-5-ylamine 0.69 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41831 H3 CLONED HUMAN 3H-Alpha-Me-histamine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 0.33 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41832 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-2-ylamine 0.84 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41833 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitrothiazol-2-yl)amine 0.19 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41834 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(3-nitropyridin-2-yl)amine 0.43 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41835 H3 CLONED HUMAN 3H-Alpha-Me-histamine (3,5-Dinitropyridin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 0.71 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41836 H3 CLONED HUMAN 3H-Alpha-Me-histamine 4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile 0.13 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41837 H3 CLONED HUMAN 3H-Alpha-Me-histamine 2-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 0.74 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41838 H3 CLONED HUMAN 3H-Alpha-Me-histamine 6-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 0.34 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41839 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitropyridin-2-yl)amine 0.3 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41840 H3 CLONED RAT 3H-Alpha-Me-histamine ABT-239 1.23 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41841 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(2-nitrophenyl)amine 0.87 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41842 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(4-nitrophenyl)amine 2.12 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41843 H3 CLONED RAT 3H-Alpha-Me-histamine 2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone 2.36 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41844 H3 CLONED RAT 3H-Alpha-Me-histamine 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)benzonitrile 1.18 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41845 H3 CLONED RAT 3H-Alpha-Me-histamine (6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 1.58 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41846 H3 CLONED RAT 3H-Alpha-Me-histamine 3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyrazine-2-carbonitrile 3.96 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41847 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrazin-2-ylamine 0.8 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41848 H3 CLONED RAT 3H-Alpha-Me-histamine (5-Bromopyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 4.02 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41849 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-5-ylamine 2.51 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41850 H3 CLONED RAT 3H-Alpha-Me-histamine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 0.58 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41851 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-2-ylamine 3.27 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41852 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitrothiazol-2-yl)amine 0.68 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41853 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(3-nitropyridin-2-yl)amine 2.71 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41854 H3 CLONED RAT 3H-Alpha-Me-histamine (3,5-Dinitropyridin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine 2.88 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41855 H3 CLONED RAT 3H-Alpha-Me-histamine 4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile 0.4 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41856 H3 CLONED RAT 3H-Alpha-Me-histamine 2-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 1.92 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41857 H3 CLONED RAT 3H-Alpha-Me-histamine 6-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile 1.42 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41858 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitropyridin-2-yl)amine 1.19 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41859 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(2-nitrophenyl)amine 0.22 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41860 H3 CLONED HUMAN 3H-Alpha-Me-histamine 4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 0.27 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41861 H3 CLONED HUMAN 3H-Alpha-Me-histamine 3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 0.29 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41862 H3 CLONED HUMAN 3H-Alpha-Me-histamine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine 0.62 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41863 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-2-ylamine 0.31 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41864 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-5-ylamine 0.08 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41865 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrazin-2-ylamine 0.11 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41866 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine 0.05 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41867 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(3-nitropyridin-2-yl)amine 0.14 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41868 H3 CLONED HUMAN 3H-Alpha-Me-histamine 6-Methyl-2-{2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}nicotinonitrile 2.98 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41869 H3 CLONED HUMAN 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-trifluoromethylpyridin-2-yl)amine 0.54 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41870 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(2-nitrophenyl)amine 0.87 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41871 H3 CLONED RAT 3H-Alpha-Me-histamine 4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 1.35 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41872 H3 CLONED RAT 3H-Alpha-Me-histamine 3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile 1.47 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41873 H3 CLONED RAT 3H-Alpha-Me-histamine (5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine 2.51 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41874 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-2-ylamine 2.01 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41875 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-5-ylamine 0.27 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41876 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrazin-2-ylamine 0.38 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41877 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine 0.11 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41878 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(3-nitropyridin-2-yl)amine 0.35 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41879 H3 CLONED RAT 3H-Alpha-Me-histamine 6-Methyl-2-{2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}nicotinonitrile 17.9 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41880 H3 CLONED RAT 3H-Alpha-Me-histamine {2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-trifluoromethylpyridin-2-yl)amine 2.76 Sun M, et al., 2005 Jan 15, 2025 Jan 15, 2025
41881 AMPA CORTICAL RAT 3H-AMPA (S)-AMPA 21 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41882 AMPA CORTICAL RAT 3H-AMPA 1-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41883 AMPA CORTICAL RAT 3H-AMPA 2-Me-Tet-AMPA 27 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41884 AMPA CORTICAL RAT 3H-AMPA (S)-(2)-Me-Tet-AMPA 9 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41885 AMPA CORTICAL RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41886 AMPA CORTICAL RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41887 AMPA CORTICAL RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41888 AMPA CORTICAL RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid 134 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41889 AMPA CORTICAL RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid 2500 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41890 AMPA CORTICAL RAT 3H-AMPA (RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid 6200 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41891 KA CORTICAL RAT 3H-Kainic acid (S)-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41892 KA CORTICAL RAT 3H-Kainic acid 1-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41893 KA CORTICAL RAT 3H-Kainic acid 2-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41894 KA CORTICAL RAT 3H-Kainic acid (S)-(2)-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41895 KA CORTICAL RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41896 KA CORTICAL RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41897 KA CORTICAL RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41898 KA CORTICAL RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41899 KA CORTICAL RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41900 KA CORTICAL RAT 3H-Kainic acid (RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 15, 2025
41901 NMDA CORTICAL RAT 3H-CGP39653 (S)-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41902 NMDA CORTICAL RAT 3H-CGP39653 1-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41903 NMDA CORTICAL RAT 3H-CGP39653 2-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41904 NMDA CORTICAL RAT 3H-CGP39653 (S)-(2)-Me-Tet-AMPA >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41905 NMDA CORTICAL RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41906 NMDA CORTICAL RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41907 NMDA CORTICAL RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41908 NMDA CORTICAL RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41909 NMDA CORTICAL RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41910 NMDA CORTICAL RAT 3H-CGP39653 (RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid >10000 Vogensen SB, et al., 2005 Jan 15, 2025 Jan 28, 2025
41911 GABAA CLONED HUMAN 3H-RO-15-1788 3,5-diphenylpyridazine 36 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41912 GABAA CLONED HUMAN 3H-RO-15-1788 4-(6-Phenylpyridazin-4-yl)benzonitrile 27 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41913 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenylpyridazin-4-yl)benzonitrile 7 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41914 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-phenyl pyridazine 7.5 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41915 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 12 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41916 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester 88 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41917 GABAA CLONED HUMAN 3H-RO-15-1788 5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine 8.5 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41918 GABAA CLONED HUMAN 3H-RO-15-1788 3-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine 1.3 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41919 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-ethoxy pyridazine 8.6 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41920 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-isopropoxypyridazine 26 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41921 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine 49 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41922 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine 55 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41923 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine 3.5 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41924 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine 7.3 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41925 GABAA CLONED HUMAN 3H-RO-15-1788 3-(5-Phenylpyridazin-3-yl)benzonitrile 666 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41926 GABAA CLONED HUMAN 3H-RO-15-1788 3,5-diphenylpyridazine 45 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41927 GABAA CLONED HUMAN 3H-RO-15-1788 2-(6-Phenylpyridazin-4-yl)benzonitrile 440 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41928 GABAA CLONED HUMAN 3H-RO-15-1788 4-(6-Phenylpyridazin-4-yl)benzonitrile 81 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41929 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenylpyridazin-4-yl)benzonitrile 14 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41930 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-phenyl pyridazine 15 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41931 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 27 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41932 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenyl-pyridazine-4-yl)-benzoic acid methyl ester 29 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41933 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester 45 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41934 GABAA CLONED HUMAN 3H-RO-15-1788 3-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine 41 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41935 GABAA CLONED HUMAN 3H-RO-15-1788 5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine 10.4 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41936 GABAA CLONED HUMAN 3H-RO-15-1788 3-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine 3.1 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41937 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(2-Fluorophenyl)-pyridazin-4-yl]benzonitrile 7.9 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41938 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 7.2 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41939 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(4-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 26 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41940 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(2,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 23 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41941 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 41 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41942 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-methoxypyridazine 205 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41943 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-ethoxy pyridazine 19 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41944 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-isopropoxypyridazine 60 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41945 GABAA CLONED HUMAN 3H-RO-15-1788 3-(Benzyloxy)-5-(3-bromophenyl)pyridazine 302 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41946 GABAA CLONED HUMAN 3H-RO-15-1788 3-(Benzyloxy)-5-(3-cyanophenyl)pyridazine 60 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41947 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Ethoxypyridazin-4-yl)benzonitrile 72 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41948 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine 113 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41949 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine 120 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41950 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine 7.3 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41951 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine 22 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41952 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-ethylaminopyridazin-4-yl)-benzonitrile 79 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41953 GABAA CLONED HUMAN 3H-RO-15-1788 N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine 51 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41954 GABAA CLONED HUMAN 3H-RO-15-1788 N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine 15 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41955 GABAA CLONED HUMAN 3H-RO-15-1788 3-(5-Phenylpyridazin-3-yl)benzonitrile 666 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41956 GABAA CLONED HUMAN 3H-RO-15-1788 3,5-diphenylpyridazine 29 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41957 GABAA CLONED HUMAN 3H-RO-15-1788 2-(6-Phenylpyridazin-4-yl)benzonitrile 323 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41958 GABAA CLONED HUMAN 3H-RO-15-1788 4-(6-Phenylpyridazin-4-yl)benzonitrile 56 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41959 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenylpyridazin-4-yl)benzonitrile 5.2 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41960 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-phenyl pyridazine 7.9 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41961 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 8.4 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41962 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenyl-pyridazine-4-yl)-benzoic acid methyl ester 11 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41963 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester 12 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41964 GABAA CLONED HUMAN 3H-RO-15-1788 3-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine 12 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41965 GABAA CLONED HUMAN 3H-RO-15-1788 5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine 8.8 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41966 GABAA CLONED HUMAN 3H-RO-15-1788 3-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine 1.6 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41967 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(2-Fluorophenyl)-pyridazin-4-yl]benzonitrile 3.4 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41968 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 4 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41969 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(4-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 14 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41970 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(2,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 17 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41971 GABAA CLONED HUMAN 3H-RO-15-1788 3-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 13 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41972 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-methoxypyridazine 54 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41973 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-ethoxy pyridazine 5.7 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41974 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-3-isopropoxypyridazine 36 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41975 GABAA CLONED HUMAN 3H-RO-15-1788 3-(Benzyloxy)-5-(3-bromophenyl)pyridazine 63 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41976 GABAA CLONED HUMAN 3H-RO-15-1788 3-(Benzyloxy)-5-(3-cyanophenyl)pyridazine 17 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41977 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-Ethoxypyridazin-4-yl)benzonitrile 36 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41978 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine 27 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41979 GABAA CLONED HUMAN 3H-RO-15-1788 5-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine 51 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41980 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine 3.8 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41981 GABAA CLONED HUMAN 3H-RO-15-1788 [5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine 7.2 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41982 GABAA CLONED HUMAN 3H-RO-15-1788 3-(6-ethylaminopyridazin-4-yl)-benzonitrile 33 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41983 GABAA CLONED HUMAN 3H-RO-15-1788 N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine 19 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41984 GABAA CLONED HUMAN 3H-RO-15-1788 N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine 6.1 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41985 GABAA CLONED HUMAN 3H-RO-15-1788 3-(5-Phenylpyridazin-3-yl)benzonitrile 666 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
41986 M1 CLONED HUMAN 3H-QNB Adinazolam >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41987 M1 CLONED HUMAN 3H-QNB AMITRIPTYLINE 14.7 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41988 M1 CLONED HUMAN 3H-QNB BUPROPION >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41989 M1 CLONED HUMAN 3H-QNB DESIPRAMINE 110 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41990 M1 CLONED HUMAN 3H-QNB Desmethylsertraline 1650 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41991 M1 CLONED HUMAN 3H-QNB Dothiepin 18 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41992 M1 CLONED HUMAN 3H-QNB DOXEPIN 38 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41993 M1 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41994 M1 CLONED HUMAN 3H-QNB Femoxetine 92 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41995 M1 CLONED HUMAN 3H-QNB FLUOXETINE 1030 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41996 M1 CLONED HUMAN 3H-QNB IMIPRAMINE 42 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41997 M1 CLONED HUMAN 3H-QNB Lofepramine 67 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41998 M1 CLONED HUMAN 3H-QNB NORFLUOXETINE 1200 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
41999 M1 CLONED HUMAN 3H-QNB NORTRYPTYLINE 40 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42000 M1 CLONED HUMAN 3H-QNB PAROXETINE 300 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42001 M1 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.044 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42002 M1 CLONED HUMAN 3H-QNB SERTRALINE 1300 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42003 M1 CLONED HUMAN 3H-QNB TRAZODONE >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42004 M1 CLONED HUMAN 3H-QNB Venlafaxine >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42005 M2 CLONED HUMAN 3H-QNB Adinazolam >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42006 M2 CLONED HUMAN 3H-QNB AMITRIPTYLINE 11.8 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42007 M2 CLONED HUMAN 3H-QNB BUPROPION >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42008 M2 CLONED HUMAN 3H-QNB DESIPRAMINE 540 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42009 M2 CLONED HUMAN 3H-QNB Desmethylsertraline 3300 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42010 M2 CLONED HUMAN 3H-QNB Dothiepin 109 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42011 M2 CLONED HUMAN 3H-QNB DOXEPIN 160 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42012 M2 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42013 M2 CLONED HUMAN 3H-QNB Femoxetine 150 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42014 M2 CLONED HUMAN 3H-QNB FLUOXETINE 2700 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42015 M2 CLONED HUMAN 3H-QNB IMIPRAMINE 88 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42016 M2 CLONED HUMAN 3H-QNB Lofepramine 330 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42017 M2 CLONED HUMAN 3H-QNB NORFLUOXETINE 4600 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42018 M2 CLONED HUMAN 3H-QNB NORTRYPTYLINE 110 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42019 M2 CLONED HUMAN 3H-QNB PAROXETINE 340 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42020 M2 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.03 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42021 M2 CLONED HUMAN 3H-QNB SERTRALINE 2100 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42022 M2 CLONED HUMAN 3H-QNB TRAZODONE >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42023 M2 CLONED HUMAN 3H-QNB Venlafaxine >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42024 M3 CLONED HUMAN 3H-QNB Adinazolam >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42025 M3 CLONED HUMAN 3H-QNB AMITRIPTYLINE 12.8 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42026 M3 CLONED HUMAN 3H-QNB BUPROPION >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42027 M3 CLONED HUMAN 3H-QNB DESIPRAMINE 210 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42028 M3 CLONED HUMAN 3H-QNB Desmethylsertraline 3500 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42029 M3 CLONED HUMAN 3H-QNB Dothiepin 38 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42030 M3 CLONED HUMAN 3H-QNB DOXEPIN 52 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42031 M3 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42032 M3 CLONED HUMAN 3H-QNB Femoxetine 220 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42033 M3 CLONED HUMAN 3H-QNB FLUOXETINE 1000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42034 M3 CLONED HUMAN 3H-QNB IMIPRAMINE 60 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42035 M3 CLONED HUMAN 3H-QNB Lofepramine 130 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42036 M3 CLONED HUMAN 3H-QNB NORFLUOXETINE 760 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42037 M3 CLONED HUMAN 3H-QNB NORTRYPTYLINE 50 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42038 M3 CLONED HUMAN 3H-QNB PAROXETINE 80 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42039 M3 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.08 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42040 M3 CLONED HUMAN 3H-QNB SERTRALINE 1300 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42041 M3 CLONED HUMAN 3H-QNB TRAZODONE >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42042 M3 CLONED HUMAN 3H-QNB Venlafaxine >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42043 M4 CLONED HUMAN 3H-QNB Adinazolam >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42044 M4 CLONED HUMAN 3H-QNB AMITRIPTYLINE 7.2 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42045 M4 CLONED HUMAN 3H-QNB BUPROPION >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42046 M4 CLONED HUMAN 3H-QNB DESIPRAMINE 160 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42047 M4 CLONED HUMAN 3H-QNB Desmethylsertraline 3100 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42048 M4 CLONED HUMAN 3H-QNB Dothiepin 61 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42049 M4 CLONED HUMAN 3H-QNB DOXEPIN 82 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42050 M4 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42051 M4 CLONED HUMAN 3H-QNB Femoxetine 470 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42052 M4 CLONED HUMAN 3H-QNB FLUOXETINE 2900 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42053 M4 CLONED HUMAN 3H-QNB IMIPRAMINE 112 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42054 M4 CLONED HUMAN 3H-QNB Lofepramine 340 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42055 M4 CLONED HUMAN 3H-QNB NORFLUOXETINE 2600 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42056 M4 CLONED HUMAN 3H-QNB NORTRYPTYLINE 84 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42057 M4 CLONED HUMAN 3H-QNB PAROXETINE 320 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42058 M4 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.037 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42059 M4 CLONED HUMAN 3H-QNB SERTRALINE 1400 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42060 M4 CLONED HUMAN 3H-QNB TRAZODONE >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42061 M4 CLONED HUMAN 3H-QNB Venlafaxine >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42062 M5 CLONED HUMAN 3H-QNB Adinazolam >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42063 M5 CLONED HUMAN 3H-QNB AMITRIPTYLINE 15.7 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42064 M5 CLONED HUMAN 3H-QNB BUPROPION >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42065 M5 CLONED HUMAN 3H-QNB DESIPRAMINE 143 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42066 M5 CLONED HUMAN 3H-QNB Desmethylsertraline 3800 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42067 M5 CLONED HUMAN 3H-QNB Dothiepin 92 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42068 M5 CLONED HUMAN 3H-QNB DOXEPIN 75 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42069 M5 CLONED HUMAN 3H-QNB Etoperidone >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42070 M5 CLONED HUMAN 3H-QNB Femoxetine 400 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42071 M5 CLONED HUMAN 3H-QNB FLUOXETINE 2700 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42072 M5 CLONED HUMAN 3H-QNB IMIPRAMINE 83 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42073 M5 CLONED HUMAN 3H-QNB Lofepramine 460 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42074 M5 CLONED HUMAN 3H-QNB NORFLUOXETINE 2200 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42075 M5 CLONED HUMAN 3H-QNB NORTRYPTYLINE 97 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42076 M5 CLONED HUMAN 3H-QNB PAROXETINE 650 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42077 M5 CLONED HUMAN 3H-QNB Quinuclidinyl benzilate 0.065 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42078 M5 CLONED HUMAN 3H-QNB SERTRALINE 1900 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42079 M5 CLONED HUMAN 3H-QNB TRAZODONE >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42080 M5 CLONED HUMAN 3H-QNB Venlafaxine >10000 Stanton T, et al., 1993 Jan 15, 2025 Jan 15, 2025
42081 Alpha2B CLONED HUMAN 35S-GTPGammaS A-54741 912.011 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42082 Alpha2B CLONED HUMAN 35S-GTPGammaS alpha-Methyl-(+/-)norepinephrine,(+/-) 2630.27 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42083 Alpha2B CLONED HUMAN 35S-GTPGammaS CLONIDINE 69.1831 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42084 Alpha2B CLONED HUMAN 35S-GTPGammaS Dexmedetomidine 33.8844 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42085 Alpha2B CLONED HUMAN 35S-GTPGammaS EPINEPHRINE 6309.57 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42086 Alpha2B CLONED HUMAN 35S-GTPGammaS Guanabenz 281.838 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42087 Alpha2B CLONED HUMAN 35S-GTPGammaS Guanfacine 1380.38 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42088 Alpha2B CLONED HUMAN 35S-GTPGammaS Levlofexidine 125.893 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42089 Alpha2B CLONED HUMAN 35S-GTPGammaS Naphazoline 407.38 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42090 Alpha2B CLONED HUMAN 35S-GTPGammaS Naphthalene 16.9824 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42091 Alpha2B CLONED HUMAN 35S-GTPGammaS NOREPINEPHRINE 2754.23 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42092 Alpha2B CLONED HUMAN 35S-GTPGammaS OXYMETAZOLINE 1778.28 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42093 Alpha2B CLONED HUMAN 35S-GTPGammaS p-AMINOCLONIDINE 29.5121 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42094 Alpha2B CLONED HUMAN 35S-GTPGammaS ST-91 794.328 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42095 Alpha2B CLONED HUMAN 35S-GTPGammaS Tramazoline 138.038 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42096 Alpha2B CLONED HUMAN 35S-GTPGammaS UK-14,304 954.993 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42097 Alpha2B CLONED HUMAN 35S-GTPGammaS Xylazine 3467.37 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42098 Alpha2B CLONED HUMAN 35S-GTPGammaS Xylometazoline 1047.13 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42099 Alpha2B CLONED HUMAN 35S-GTPGammaS Alinidine 6456.54 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42100 Alpha2B CLONED HUMAN 35S-GTPGammaS B-HT 920 512.861 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42101 Alpha2B CLONED HUMAN 35S-GTPGammaS IDAZOXAN 37.1535 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42102 Alpha2B CLONED HUMAN 35S-GTPGammaS ICI 106270 67.6083 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42103 Alpha2B CLONED HUMAN 35S-GTPGammaS IMILOXAN 67.6083 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42104 Alpha2B CLONED HUMAN 35S-GTPGammaS MK-912 0.891251 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42105 Alpha2B CLONED HUMAN 35S-GTPGammaS PHENTOLAMINE 33.1131 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42106 Alpha2B CLONED HUMAN 35S-GTPGammaS PRAZOSIN 89.1251 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42107 Alpha2B CLONED HUMAN 35S-GTPGammaS RAUWOLSCINE 1.20226 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42108 Alpha2B CLONED HUMAN 35S-GTPGammaS Rilmenidine 1737.8 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42109 Alpha2B CLONED HUMAN 35S-GTPGammaS RX821002 1.62181 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42110 Alpha2B CLONED HUMAN 35S-GTPGammaS TOLAZOLINE 3162.28 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42111 Alpha2C CLONED HUMAN 35S-GTPGammaS A-54741 776.247 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42112 Alpha2C CLONED HUMAN 35S-GTPGammaS alpha-Methyl-(+/-)norepinephrine,(+/-) 2884.03 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42113 Alpha2C CLONED HUMAN 35S-GTPGammaS CLONIDINE 134.896 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42114 Alpha2C CLONED HUMAN 35S-GTPGammaS Dexmedetomidine 95.4993 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42115 Alpha2C CLONED HUMAN 35S-GTPGammaS EPINEPHRINE 1698.24 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42116 Alpha2C CLONED HUMAN 35S-GTPGammaS Guanabenz 446.684 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42117 Alpha2C CLONED HUMAN 35S-GTPGammaS Guanfacine 3890.45 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42118 Alpha2C CLONED HUMAN 35S-GTPGammaS Levlofexidine 173.78 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42119 Alpha2C CLONED HUMAN 35S-GTPGammaS Naphazoline 407.38 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42120 Alpha2C CLONED HUMAN 35S-GTPGammaS Naphthalene 3.31131 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42121 Alpha2C CLONED HUMAN 35S-GTPGammaS NOREPINEPHRINE 1348.96 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42122 Alpha2C CLONED HUMAN 35S-GTPGammaS OXYMETAZOLINE 239.883 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42123 Alpha2C CLONED HUMAN 35S-GTPGammaS p-AMINOCLONIDINE 21.3796 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42124 Alpha2C CLONED HUMAN 35S-GTPGammaS ST-91 616.595 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42125 Alpha2C CLONED HUMAN 35S-GTPGammaS Tramazoline 275.423 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42126 Alpha2C CLONED HUMAN 35S-GTPGammaS UK-14,304 1949.84 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42127 Alpha2C CLONED HUMAN 35S-GTPGammaS Xylazine >10000 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42128 Alpha2C CLONED HUMAN 35S-GTPGammaS Xylometazoline 128.825 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42129 Alpha2C CLONED HUMAN 35S-GTPGammaS Alinidine >10000 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42130 Alpha2C CLONED HUMAN 35S-GTPGammaS B-HT 920 954.993 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42131 Alpha2C CLONED HUMAN 35S-GTPGammaS IDAZOXAN 19.9526 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42132 Alpha2C CLONED HUMAN 35S-GTPGammaS ICI 106270 281.838 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42133 Alpha2C CLONED HUMAN 35S-GTPGammaS IMILOXAN 151.356 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42134 Alpha2C CLONED HUMAN 35S-GTPGammaS MK-912 0.0676083 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42135 Alpha2C CLONED HUMAN 35S-GTPGammaS PHENTOLAMINE 257.04 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42136 Alpha2C CLONED HUMAN 35S-GTPGammaS PRAZOSIN 30.903 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42137 Alpha2C CLONED HUMAN 35S-GTPGammaS RAUWOLSCINE 0.549541 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42138 Alpha2C CLONED HUMAN 35S-GTPGammaS Rilmenidine 4677.35 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42139 Alpha2C CLONED HUMAN 35S-GTPGammaS RX821002 0.794328 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42140 Alpha2C CLONED HUMAN 35S-GTPGammaS TOLAZOLINE 3715.35 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42141 GABAA CLONED HUMAN Functional 4-(6-Phenylpyridazin-4-yl)benzonitrile 49 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42142 GABAA CLONED HUMAN Functional 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 22 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42143 GABAA CLONED HUMAN Functional 3-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine 13 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42144 GABAA CLONED HUMAN Functional 5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine 43 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42145 GABAA CLONED HUMAN Functional 3-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile 3.6 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42146 GABAA CLONED HUMAN Functional 3-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile 32 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42147 GABAA CLONED HUMAN Functional 5-(3-Bromophenyl)-3-methoxypyridazine 42 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42148 GABAA CLONED HUMAN Functional 5-(3-Bromophenyl)-3-ethoxy pyridazine 39 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42149 GABAA CLONED HUMAN Functional 5-(3-Bromophenyl)-3-isopropoxypyridazine 28 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42150 GABAA CLONED HUMAN Functional 3-(Benzyloxy)-5-(3-bromophenyl)pyridazine 32 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42151 GABAA CLONED HUMAN Functional 3-(Benzyloxy)-5-(3-cyanophenyl)pyridazine 60 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42152 GABAA CLONED HUMAN Functional 3-(6-Ethoxypyridazin-4-yl)benzonitrile 19 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42153 GABAA CLONED HUMAN Functional [5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine 3 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42154 GABAA CLONED HUMAN Functional [5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine 2 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42155 GABAA CLONED HUMAN Functional [5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine 25 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42156 GABAA CLONED HUMAN Functional 3-(6-ethylaminopyridazin-4-yl)-benzonitrile 8 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42157 GABAA CLONED HUMAN Functional N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine 66 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42158 GABAA CLONED HUMAN Functional N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine 59 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42159 GABAA CLONED HUMAN Functional 4-(6-Phenylpyridazin-4-yl)benzonitrile 45 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42160 GABAA CLONED HUMAN Functional 5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine 18 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42161 GABAA CLONED HUMAN Functional 5-(3-Bromophenyl)-3-ethoxy pyridazine 4 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42162 GABAA CLONED HUMAN Functional 5-(3-Bromophenyl)-3-isopropoxypyridazine 12 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42163 GABAA CLONED HUMAN Functional [5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine 14 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42164 GABAA CLONED HUMAN Functional N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine 14 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42165 GABAA CLONED HUMAN Functional N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine 17 van Niel MB, et al., 2005 Jan 15, 2025 Jan 27, 2025
42166 CLONED HUMAN Functional 1-Isopropyl-1H-benzotriazole-5-carboxylic acid 398.107 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42167 CLONED HUMAN Functional 1-(2’-Methoxy-1’-methyl-ethyl)-1H-benzotriazole-5-carboxylic acid 199.526 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42168 CLONED HUMAN Functional 1-(2’-Ethoxy-ethyl)-1H-benzotriazole-5-carboxylic acid 257.04 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42169 CLONED HUMAN Functional 1-t-Butyl-1H-benzotriazole-5-carboxylic acid 257.04 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42170 CLONED HUMAN Functional 1-Pentyl-1H-benzotriazole-5-carboxylic acid 288.403 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42171 CLONED HUMAN Functional 1-(2’-Ethylsulfanyl-ethyl)-1H-benzotriazole-5-carboxylic acid 301.995 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42172 CLONED HUMAN Functional 1-(2-Methoxy-ethyl)-1H-benzotriazole-5-carboxylic acid 316.228 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42173 CLONED HUMAN Functional 1-(2’-Butyl)-1H-benzotriazole-5-carboxylic acid 331.131 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42174 CLONED HUMAN Functional 1-Butyl-1H-benzotriazole-5-carboxylic acid 691.831 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42175 CLONED HUMAN Functional 1-Ethyl-1H-benzotriazole-5-carboxylic acid 891.251 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42176 CLONED HUMAN Functional 1-(3’-Pentyl)-1H-benzotriazole-5-carboxylic acid 3019.95 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42177 CLONED HUMAN Functional 1-Propyl-1H-benzotriazole-5-carboxylic acid 7413.1 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42178 CLONED HUMAN Functional 1-Cyclopropyl-1H-benzotriazole-5-carboxylic acid 2344.23 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42179 CLONED HUMAN Functional 4-Ethyl-5-(4-piperidyl)-3-isoxazolol 6626 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42180 CLONED HUMAN Functional 3-Phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 4337 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42181 CLONED HUMAN Functional N-Methyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 773 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42182 CLONED HUMAN Functional N-Ethyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 175 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42183 CLONED HUMAN Functional N-Isopropyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 199 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42184 CLONED HUMAN Functional N-Butyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 79 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42185 CLONED HUMAN Functional {(3-Phenylpropionyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester 105 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42186 CLONED HUMAN Functional {(3-Phenylpropionyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid 376 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42187 CLONED HUMAN Functional N-Benzyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 580 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42188 CLONED HUMAN Functional N-Cyclohexyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide 150 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42189 CLONED HUMAN Functional N-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 178 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42190 CLONED HUMAN Functional N-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]nicotinamide 1015 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42191 CLONED HUMAN Functional N-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isonicotinamide 394 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42192 CLONED HUMAN Functional N-Ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 41 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42193 CLONED HUMAN Functional N-Propyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 28 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42194 CLONED HUMAN Functional N-Butyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 20 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42195 CLONED HUMAN Functional N-(2-Dimethylaminoethyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 1147 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42196 CLONED HUMAN Functional N-(2-Hydroxyethyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 106 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42197 CLONED HUMAN Functional {Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester 34 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42198 CLONED HUMAN Functional {Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid 627 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42199 CLONED HUMAN Functional 5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester 26 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42200 CLONED HUMAN Functional 5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid 8 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42201 CLONED HUMAN Functional N-[4-(1H-Tetrazol-5-yl)butyl]-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 8 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42202 CLONED HUMAN Functional N-(4-Cyanobutyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide 20 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42203 CLONED HUMAN Functional 4-Cyano-N-ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]benzamide 37 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42204 CLONED HUMAN Functional N-Ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isonicotinamide 95 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42205 CLONED HUMAN Functional 1-Methyl-3-phenyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 1564 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42206 CLONED HUMAN Functional 1-Ethyl-3,3-dimethyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 59 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42207 CLONED HUMAN Functional 1,3-Diethyl-3-(4-hydroxybutyl)-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea 60 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42208 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Methyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 321 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42209 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Ethyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 74 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42210 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Propyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 34 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42211 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Butyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 30 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42212 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Pentyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 19 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42213 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Hexyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 31 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42214 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Heptyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 73 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42215 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Octyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 269 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42216 CLONED HUMAN Functional Morpholine-4-carboxylic Acid Phenethyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 43 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42217 CLONED HUMAN Functional Morpholine-4-carboxylic Acid (2-Hydroxyethyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 166 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42218 CLONED HUMAN Functional {(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester 80 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42219 CLONED HUMAN Functional 3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid Methyl Ester 99 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42220 CLONED HUMAN Functional 3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid 247 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42221 CLONED HUMAN Functional 4-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}butyric Acid Methyl Ester 75 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42222 CLONED HUMAN Functional Morpholine-4-carboxylic Acid (3-Cyanopropyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide 40 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42223 CLONED HUMAN Functional 5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester 42 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42224 CLONED HUMAN Functional 5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid 14 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42225 CLONED HUMAN Functional N-Phenethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide 2650 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42226 CLONED HUMAN Functional N-Methyl-N-phenethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide 1990 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42227 CLONED HUMAN Functional N-Benzyl-N-methyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide 1000 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42228 CLONED HUMAN Functional N-Methoxy-N-methyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide 1450 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42229 CLONED HUMAN Functional Pyrrolidin-1-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone 850 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42230 CLONED HUMAN Functional Morpholin-4-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone 1140 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42231 CLONED HUMAN Functional Piperidin-1-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone 980 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42232 CLONED HUMAN Functional N-(2-Cyanoethyl)-N-ethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide 290 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42233 CLONED HUMAN Functional N,N-Diisobutyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide 70 Cheng JF, et al., 2006 Jan 15, 2025 Jan 15, 2025
42234 KOR BRAIN RAT 3H-MUSCIMOL SR 95531 74 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42235 KOR BRAIN RAT 3H-MUSCIMOL 4-PIOL 9100 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42236 KOR BRAIN RAT 3H-MUSCIMOL Thio-4-PIOL 1870 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42237 KOR BRAIN RAT 3H-MUSCIMOL 4-Methyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 2200 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42238 KOR BRAIN RAT 3H-MUSCIMOL 5-(4-Piperidyl)-4-propylisothiazol-3-ol Hydrobromide 440 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42239 KOR BRAIN RAT 3H-MUSCIMOL 4-Benzyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 331 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42240 KOR BRAIN RAT 3H-MUSCIMOL 4-(2-Naphthylmethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 5.2 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42241 KOR BRAIN RAT 3H-MUSCIMOL 4-((1-Bromo-2-naphthyl)methyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 1.8 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42242 KOR BRAIN RAT 3H-MUSCIMOL 4-(2,2-Diphenyl-1-ethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 388 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42243 KOR BRAIN RAT 3H-MUSCIMOL 4-(3,3-Diphenyl-1-propyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide 9.6 Krehan D, et al., 2006 Jan 15, 2025 Jan 27, 2025
42244 CLONED HUMAN 125I-[Ile]Motilin [Bpa5,Ile13]Motilin 50 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42245 CLONED HUMAN 125I-[Ile]Motilin Motilin 2.3 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42246 CLONED HUMAN 125I-[Ile]Motilin [D-Bpa5,Ile13]Motilin 420 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42247 CLONED HUMAN 125I-[Ile]Motilin [L-Bpa5,Ile13]Motilin 50 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42248 CLONED HUMAN 125I-[Ile]Motilin cyanogen bromide, CNBr 0.85 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42249 CLONED HUMAN Functional cyanogen bromide, CNBr 8.4 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42250 CLONED HUMAN 125I-[Ile]Motilin K368,374C 0.6 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42251 CLONED HUMAN Functional K368,374C 0.3 Matsuura B, et al., 2005 Jan 15, 2025 Jan 15, 2025
42252 CLONED HUMAN Functional 1-Cyclobutyl-1H-benzotriazole-5-carboxylic acid 3090.3 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42253 CLONED HUMAN Functional 1-Cyclopentyl-1H-benzotriazole-5-carboxylic acid 1096.48 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42254 CLONED HUMAN Functional 1-Cyclohexyl-1H-benzotriazole-5-carboxylic acid 5888.44 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42255 CLONED HUMAN Functional 1-Benzyl-1H-benzotriazole-5-carboxylic acid 9120.11 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42256 CLONED HUMAN Functional 1-Benzhydryl-1H-benzotriazole-5-carboxylic acid >10000 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42257 CLONED HUMAN Functional 1-(3’-Methoxybenzyl)-1H-benzotriazole-5-carboxylic acid 5011.87 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42258 CLONED HUMAN Functional 1-(3’,5’-Difluorobenzyl)-1H-benzotriazole-5-carboxylic acid >10000 Semple G, et al., 2006 Jan 15, 2025 Jan 15, 2025
42259 CLONED HUMAN 125I-Motilin Delta 2-4 2.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42260 CLONED HUMAN 125I-Motilin Delta 5-8 1.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42261 CLONED HUMAN 125I-Motilin Delta 9-12 3.8 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42262 CLONED HUMAN 125I-Motilin Delta 13-16 2.6 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42263 CLONED HUMAN 125I-Motilin Delta 17-20 1.4 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42264 CLONED HUMAN 125I-Motilin Delta 21-24 2.3 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42265 CLONED HUMAN 125I-Motilin Delta 25C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42266 CLONED HUMAN 125I-Motilin Delta 26-28 1.6 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42267 CLONED HUMAN 125I-Motilin Delta 29 8.1 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42268 CLONED HUMAN 125I-Motilin Delta 30C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42269 CLONED HUMAN 125I-Motilin Delta 31-32 2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42270 CLONED HUMAN 125I-Motilin Delta 33-36 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42271 CLONED HUMAN 125I-Motilin Delta 103-104 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42272 CLONED HUMAN 125I-Motilin Delta 105-110 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42273 CLONED HUMAN 125I-Motilin Delta 111C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42274 CLONED HUMAN 125I-Motilin Delta 328-330 6.3 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42275 CLONED HUMAN 125I-Motilin Delta 331-332 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42276 CLONED HUMAN 125I-Motilin F33A 7.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42277 CLONED HUMAN 125I-Motilin P34A 4.2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42278 CLONED HUMAN 125I-Motilin L35A 3.7 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42279 CLONED HUMAN 125I-Motilin G36A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42280 CLONED HUMAN 125I-Motilin P103A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42281 CLONED HUMAN 125I-Motilin W104A 12.2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42282 CLONED HUMAN 125I-Motilin V105A 1.8 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42283 CLONED HUMAN 125I-Motilin F106A 1.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42284 CLONED HUMAN 125I-Motilin G107A 1 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42285 CLONED HUMAN 125I-Motilin P108A 2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42286 CLONED HUMAN 125I-Motilin L109A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42287 CLONED HUMAN 125I-Motilin L110A 2.3 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42288 CLONED HUMAN 125I-Motilin Y331A 2.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42289 CLONED HUMAN 125I-Motilin F332A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42290 CLONED HUMAN Functional Delta 2-4 4.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42291 CLONED HUMAN Functional Delta 5-8 5.1 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42292 CLONED HUMAN Functional Delta 9-12 4.2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42293 CLONED HUMAN Functional Delta 13-16 4.5 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42294 CLONED HUMAN Functional Delta 17-20 4.5 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42295 CLONED HUMAN Functional Delta 21-24 4 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42296 CLONED HUMAN Functional Delta 25C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42297 CLONED HUMAN Functional Delta 26-28 5.1 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42298 CLONED HUMAN Functional Delta 29 4.2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42299 CLONED HUMAN Functional Delta 30C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42300 CLONED HUMAN Functional Delta 31-32 3.7 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42301 CLONED HUMAN Functional Delta 33-36 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42302 CLONED HUMAN Functional Delta 103-104 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42303 CLONED HUMAN Functional Delta 105-110 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42304 CLONED HUMAN Functional Delta 111C 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42305 CLONED HUMAN Functional Delta 328-330 5.1 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42306 CLONED HUMAN Functional Delta 331-332 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42307 CLONED HUMAN Functional F33A 5.4 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42308 CLONED HUMAN Functional P34A 4.8 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42309 CLONED HUMAN Functional L35A 3.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42310 CLONED HUMAN Functional G36A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42311 CLONED HUMAN Functional P103A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42312 CLONED HUMAN Functional W104A 4.8 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42313 CLONED HUMAN Functional V105A 4.6 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42314 CLONED HUMAN Functional F106A 4.5 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42315 CLONED HUMAN Functional G107A 4.2 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42316 CLONED HUMAN Functional P108A 4.1 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42317 CLONED HUMAN Functional L109A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42318 CLONED HUMAN Functional L110A 4.5 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42319 CLONED HUMAN Functional Y331A 4.9 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42320 CLONED HUMAN Functional F332A 1000 Matsuura B, et al., 2006 Jan 15, 2025 Jan 15, 2025
42321 SLC6A3 Striatal Membranes RAT 3H-LBT-999 GBR-12935 2.4 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42322 SLC6A3 Striatal Membranes RAT 3H-LBT-999 PE2I 18 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42323 SLC6A3 Striatal Membranes RAT 3H-LBT-999 PAROXETINE 1000 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42324 SLC6A3 Striatal Membranes RAT 3H-LBT-999 CITALOPRAM 1000 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42325 SLC6A3 Striatal Membranes RAT 3H-LBT-999 MADAM 1000 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42326 SLC6A3 Striatal Membranes RAT 3H-LBT-999 Nisoxetine 1000 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42327 SLC6A3 Striatal Membranes RAT 3H-LBT-999 DESIPRAMINE 1000 Chalon S, et al., 2006 Jan 15, 2025 Jan 15, 2025
42328 CLONED HUMAN 125I-Motilin Motilin 2.81838 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42329 CLONED HUMAN 125I-Motilin ABT-229 58.8844 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42330 CLONED HUMAN 125I-Motilin erythromycin-A 3090.3 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42331 CLONED HUMAN 125I-Motilin ME36 >10000 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42332 CLONED HUMAN 125I-Motilin ME4 537.032 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42333 CLONED HUMAN 125I-Motilin EM-B enolether 323.594 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42334 CLONED HUMAN 125I-Motilin ME523 257.04 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42335 CLONED HUMAN 125I-Motilin 4'deoxy EM-A enolether 69.1831 Thielemans L, et al., 2005 Jan 15, 2025 Jan 15, 2025
42336 Alpha2A CLONED HUMAN 35S-GTPGammaS A-54741 245.471 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42337 Alpha2A CLONED HUMAN 35S-GTPGammaS alpha-Methyl-(+/-)norepinephrine,(+/-) 3630.78 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42338 Alpha2A CLONED HUMAN 35S-GTPGammaS CLONIDINE 61.6595 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42339 Alpha2A CLONED HUMAN 35S-GTPGammaS Dexmedetomidine 13.1826 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42340 Alpha2A CLONED HUMAN 35S-GTPGammaS EPINEPHRINE 1479.11 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42341 Alpha2A CLONED HUMAN 35S-GTPGammaS Guanabenz 21.8776 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42342 Alpha2A CLONED HUMAN 35S-GTPGammaS Guanfacine 93.3254 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42343 Alpha2A CLONED HUMAN 35S-GTPGammaS Levlofexidine 14.4544 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42344 Alpha2A CLONED HUMAN 35S-GTPGammaS Naphazoline 20.893 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42345 Alpha2A CLONED HUMAN 35S-GTPGammaS Naphthalene 4.57088 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42346 Alpha2A CLONED HUMAN 35S-GTPGammaS NOREPINEPHRINE 1995.26 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42347 Alpha2A CLONED HUMAN 35S-GTPGammaS OXYMETAZOLINE 7.24436 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42348 Alpha2A CLONED HUMAN 35S-GTPGammaS p-AMINOCLONIDINE 7.94328 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42349 Alpha2A CLONED HUMAN 35S-GTPGammaS ST-91 575.44 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42350 Alpha2A CLONED HUMAN 35S-GTPGammaS Tramazoline 31.6228 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42351 Alpha2A CLONED HUMAN 35S-GTPGammaS UK-14,304 213.796 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42352 Alpha2A CLONED HUMAN 35S-GTPGammaS Xylazine 5754.4 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42353 Alpha2A CLONED HUMAN 35S-GTPGammaS Xylometazoline 15.1356 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42354 Alpha2A CLONED HUMAN 35S-GTPGammaS Alinidine 6025.6 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42355 Alpha2A CLONED HUMAN 35S-GTPGammaS B-HT 920 398.107 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42356 Alpha2A CLONED HUMAN 35S-GTPGammaS IDAZOXAN 9.77237 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42357 Alpha2A CLONED HUMAN 35S-GTPGammaS ICI 106270 7.94328 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42358 Alpha2A CLONED HUMAN 35S-GTPGammaS IMILOXAN 316.228 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42359 Alpha2A CLONED HUMAN 35S-GTPGammaS MK-912 0.851138 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42360 Alpha2A CLONED HUMAN 35S-GTPGammaS PHENTOLAMINE 20.4174 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42361 Alpha2A CLONED HUMAN 35S-GTPGammaS PRAZOSIN 794.328 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42362 Alpha2A CLONED HUMAN 35S-GTPGammaS RAUWOLSCINE 1.20226 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42363 Alpha2A CLONED HUMAN 35S-GTPGammaS Rilmenidine 1584.89 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42364 Alpha2A CLONED HUMAN 35S-GTPGammaS RX821002 0.363078 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42365 Alpha2A CLONED HUMAN 35S-GTPGammaS TOLAZOLINE 229.087 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42366 Alpha2A CLONED MOUSE 35S-GTPGammaS EPINEPHRINE 389.045 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42367 Alpha2A CLONED MOUSE 35S-GTPGammaS NOREPINEPHRINE 1412.54 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42368 Alpha2A CLONED MOUSE 35S-GTPGammaS Isoproterenol >10000 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42369 Alpha2A CLONED MOUSE 35S-GTPGammaS A-54741 9.77237 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42370 Alpha2A CLONED MOUSE 35S-GTPGammaS UK-14,304 43.6516 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42371 Alpha2A CLONED MOUSE 35S-GTPGammaS Dexmedetomidine 3.38844 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42372 Alpha2A CLONED MOUSE 35S-GTPGammaS ST-91 537.032 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42373 Alpha2A CLONED MOUSE 35S-GTPGammaS Guanfacine 20.4174 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42374 Alpha2A CLONED MOUSE 35S-GTPGammaS Xylazine 2398.83 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42375 Alpha2A CLONED MOUSE 35S-GTPGammaS Rilmenidine 724.436 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42376 Alpha2A CLONED MOUSE 35S-GTPGammaS CLONIDINE 40.738 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42377 Alpha2A CLONED MOUSE 35S-GTPGammaS OXYMETAZOLINE 15.4882 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42378 Alpha2A CLONED MOUSE 35S-GTPGammaS Tramazoline 15.4882 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42379 Alpha2A CLONED MOUSE 35S-GTPGammaS Naphthalene 7.76247 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42380 Alpha2A CLONED MOUSE 35S-GTPGammaS Naphazoline 11.4815 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42381 Alpha2A CLONED MOUSE 35S-GTPGammaS Xylometazoline 25.704 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42382 Alpha2A CLONED MOUSE 35S-GTPGammaS RX821002 0.616595 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42383 Alpha2A CLONED MOUSE 35S-GTPGammaS Naphthalene 9.33254 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42384 Alpha2A CLONED MOUSE 35S-GTPGammaS Naphazoline 16.9824 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42385 Alpha2A CLONED MOUSE 35S-GTPGammaS Xylometazoline 23.9883 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42386 Alpha2A CLONED MOUSE 35S-GTPGammaS OXYMETAZOLINE 25.704 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42387 Alpha2A CLONED MOUSE 35S-GTPGammaS RAUWOLSCINE 36.3078 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42388 Alpha2A CLONED MOUSE 35S-GTPGammaS YOHIMBINE 61.6595 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42389 Alpha2A CLONED MOUSE 35S-GTPGammaS CLONIDINE 61.6595 Jasper JR, et al., 1998 Jan 15, 2025 Jan 15, 2025
42390 ß-Amyloid BRAIN HUMAN 125I-IMPY 4-Amino-4'-hydroxystilbene 95 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42391 ß-Amyloid BRAIN HUMAN 125I-IMPY 3-{4-[2-(4-Aminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol 15 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42392 ß-Amyloid BRAIN HUMAN 125I-IMPY 4-N,N'-Dimethylamino-4'-hydroxystilbene 1.1 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42393 ß-Amyloid BRAIN HUMAN 125I-IMPY (4-{2-[4-(2,2-Dimethyl-[1,3]dioxan-5-ylmethoxy)phenyl]vinyl}phenyl)dimethylamine 59 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42394 ß-Amyloid BRAIN HUMAN 125I-IMPY 2-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol 38 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42395 ß-Amyloid BRAIN HUMAN 125I-IMPY Toluene-4-sulfonic Acid 3-{4-[2-(4-(Dimethylamino)phenyl)vinyl]phenoxy}-2-hydroxymethylpropyl Ester 150 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42396 ß-Amyloid BRAIN HUMAN 125I-IMPY 3-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol 15 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42397 ß-Amyloid BRAIN HUMAN 125I-IMPY 2-(4-Bromobenzyl)-3-{4-[2-(4-(dimethylamino)phenyl)vinyl]phenoxy}propan-1-ol 80 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42398 ß-Amyloid BRAIN HUMAN 125I-IMPY 4-N-Methylamino-4'-hydroxystilbene, SB-13 1.2 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42399 ß-Amyloid BRAIN HUMAN 125I-IMPY 2-{4-[2-(4-Methylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol 32.5 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42400 ß-Amyloid BRAIN HUMAN 125I-IMPY 2-Fluoromethyl-3-{4-[2-(4-methylaminophenyl)vinyl]phenoxy}propan-1-ol 5 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42401 ß-Amyloid BRAIN HUMAN 125I-IMPY PIB 2.8 Zhang W, et al., 2005 Jan 15, 2025 Jan 15, 2025
42402 PLC bladder RAT Functional ET-18-OCH3 5000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42403 PLC bladder RAT Functional Neomycin 5000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42404 PLC bladder RAT Functional D609 >10000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 28, 2025
42405 PLC bladder RAT Functional Neomycin 5000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 28, 2025
42406 PAK bladder RAT Functional (R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride >10000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42407 PAK bladder RAT Functional HA-1077 1600 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42408 PAK bladder RAT Functional H7 3000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42409 PAK bladder RAT Functional H89 50 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42410 PKG bladder RAT Functional HA-1077 1600 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42411 PKG bladder RAT Functional H7 5800 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42412 PKG bladder RAT Functional H89 500 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42413 PKC bladder RAT Functional (R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride >10000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42414 PKC bladder RAT Functional Chelerytherine 660 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42415 PKC bladder RAT Functional H7 6000 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42416 Rho Kinase bladder RAT Functional (R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride 100 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42417 Rho Kinase bladder RAT Functional HA-1077 330 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42418 Rho Kinase bladder RAT Functional H7 450 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42419 Rho Kinase bladder RAT Functional H89 270 Braverman AS, et al., 2006 Jan 15, 2025 Jan 15, 2025
42420 GABAA WHOLE BRAIN RAT FNZ 1-Phenyl-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 6280 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42421 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 4350 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42422 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one 1040 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42423 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-1,5-dihydro-imidazol-2-one 4290 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42424 GABAA WHOLE BRAIN RAT FNZ 1-(4-Bromophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 3060 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42425 GABAA WHOLE BRAIN RAT FNZ 1-(4-Iodophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 3320 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42426 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-azepan-1-yl-1,5-dihydro-imidazol-2-one >10000 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42427 GABAA WHOLE BRAIN RAT FNZ 1-(4-Methoxyphenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one 938 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42428 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 141 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42429 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-2,4-dihydro-pyrrol-2-one 67 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42430 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-azepan-1-yl-2,4-dihydro-pyrrol-2-one 440 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42431 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-4-piperidin-1-yl-2,4-dihydro-pyrrol-2-one 90 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42432 GABAA WHOLE BRAIN RAT FNZ 1-(4-Fluorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 494 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42433 GABAA WHOLE BRAIN RAT FNZ 1-(3-Methylphenyl)-4-morpholin-1-yl-2,4-dihydro-pyrrol-2-one 4450 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42434 GABAA WHOLE BRAIN RAT FNZ 1-(4-Methylphenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one 344 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42435 GABAA WHOLE BRAIN RAT FNZ 1-(3-Chloro-4-fluorophenyl)-4-(morpholin-4-yl)-1,5-dihydro-pyrrole-2-one 2050 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42436 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione 4340 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42437 GABAA WHOLE BRAIN RAT FNZ 1-(4-Chlorophenyl)-3-pyrrolidin-1-yl-pyrrole-2,5-dione 3260 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42438 GABAA WHOLE BRAIN RAT FNZ 1-(4-Fluorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione 5410 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42439 GABAA WHOLE BRAIN RAT FNZ 4-(4-Chlorophenyl)-1-pyrid-2-yl-pyrazole 4480 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42440 GABAA WHOLE BRAIN RAT FNZ 3-(4-Chlorophenyl)-5-morpholin-4-yl-1,2,4-oxadiazole >10000 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42441 GABAA WHOLE BRAIN RAT FNZ 2-(4-Chlorophenyl)-5-phenyl-4-isoxazolin-3-one 1120 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42442 GABAA WHOLE BRAIN RAT FNZ CGS 9896 2.4 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42443 GABAA WHOLE BRAIN RAT FNZ DIAZEPAM 6.8 Grunwald C, et al., 2006 Jan 15, 2025 Jan 15, 2025
42444 D1 CLONED HUMAN 3H-SCH23390 LE300 1.9 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42445 D2 CLONED HUMAN 3H-SPIPERONE LE300 44.7 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42446 D5 CLONED HUMAN 3H-SCH23390 LE300 7.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42447 D1 CLONED HUMAN 3H-SCH23390 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 0.39 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42448 D2 CLONED HUMAN 3H-SPIPERONE 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 17.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42449 D3 CLONED HUMAN 3H-SPIPERONE 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 47.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42450 D5 CLONED HUMAN 3H-SCH23390 3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42451 D1 CLONED HUMAN 3H-SCH23390 3-methoxy-dibenz[d,g]azecine 28.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42452 D2 CLONED HUMAN 3H-SPIPERONE 3-methoxy-dibenz[d,g]azecine 13 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42453 D3 CLONED HUMAN 3H-SPIPERONE 3-methoxy-dibenz[d,g]azecine 75.7 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42454 D1 CLONED HUMAN 3H-SCH23390 4-chloro-3-hydroxy-dibenz[d,g]azecine 0.83 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42455 D2 CLONED HUMAN 3H-SPIPERONE 4-chloro-3-hydroxy-dibenz[d,g]azecine 4 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42456 D3 CLONED HUMAN 3H-SPIPERONE 4-chloro-3-hydroxy-dibenz[d,g]azecine 24.6 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42457 D5 CLONED HUMAN 3H-SCH23390 4-chloro-3-hydroxy-dibenz[d,g]azecine 0.057 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42458 D1 CLONED HUMAN 3H-SCH23390 2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine 3.2 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42459 D2 CLONED HUMAN 3H-SPIPERONE 2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine 88 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42460 D1 CLONED HUMAN 3H-SCH23390 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 9.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42461 D2 CLONED HUMAN 3H-SPIPERONE 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 37.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42462 D5 CLONED HUMAN 3H-SCH23390 2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 226.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42463 D1 CLONED HUMAN 3H-SCH23390 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 8.9 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42464 D2 CLONED HUMAN 3H-SPIPERONE 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 36.9 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42465 D3 CLONED HUMAN 3H-SPIPERONE 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 296 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42466 D5 CLONED HUMAN 3H-SCH23390 2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 42.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42467 D1 CLONED HUMAN 3H-SCH23390 2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 82 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42468 D2 CLONED HUMAN 3H-SPIPERONE 2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 62 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42469 D3 CLONED HUMAN 3H-SPIPERONE 2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine 150.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42470 D1 CLONED HUMAN 3H-SCH23390 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 25.3 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42471 D2 CLONED HUMAN 3H-SPIPERONE 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 210 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42472 D3 CLONED HUMAN 3H-SPIPERONE 1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 415 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42473 D1 CLONED HUMAN 3H-SCH23390 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 0.46 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42474 D2 CLONED HUMAN 3H-SPIPERONE 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 0.99 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42475 D3 CLONED HUMAN 3H-SPIPERONE 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1.88 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42476 D5 CLONED HUMAN 3H-SCH23390 1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 0.98 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42477 D1 CLONED HUMAN 3H-SCH23390 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 3.1 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42478 D2 CLONED HUMAN 3H-SPIPERONE 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 2 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42479 D3 CLONED HUMAN 3H-SPIPERONE 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 27.7 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42480 D5 CLONED HUMAN 3H-SCH23390 3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 4.9 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42481 D1 CLONED HUMAN 3H-SCH23390 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 8.7 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42482 D2 CLONED HUMAN 3H-SPIPERONE 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 84 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42483 D3 CLONED HUMAN 3H-SPIPERONE 1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 215 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42484 D1 CLONED HUMAN 3H-SCH23390 4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 7.6 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42485 D2 CLONED HUMAN 3H-SPIPERONE 4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 164 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42486 D3 CLONED HUMAN 3H-SPIPERONE 4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1833 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42487 D1 CLONED HUMAN 3H-SCH23390 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 2 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42488 D2 CLONED HUMAN 3H-SPIPERONE 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 58.7 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42489 D3 CLONED HUMAN 3H-SPIPERONE 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 342 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42490 D5 CLONED HUMAN 3H-SCH23390 3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 1.68 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42491 D1 CLONED HUMAN 3H-SCH23390 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 9.4 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42492 D2 CLONED HUMAN 3H-SPIPERONE 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 6.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 27, 2025
42493 D3 CLONED HUMAN 3H-SPIPERONE 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 101.5 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42494 D5 CLONED HUMAN 3H-SCH23390 3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine 12.6 Mohr P, et al., 2006 Jan 15, 2025 Jan 15, 2025
42495 MEK UNDEFINED UNDEFINED Functional 4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 39 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42496 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 124 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42497 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 6.8 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42498 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 40 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42499 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 30 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42500 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 45 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42501 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-5-fluoro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide 9.3 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42502 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide 18 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42503 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-chlorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-6-methoxynicotinamide 6786 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42504 MEK UNDEFINED UNDEFINED Functional 4-(4-Bromo-2-chlorophenylamino)-5,6-dichloro-N-(2-hydroxyethoxy)nicotinamide 4496 Wallace EM, et al., 2006 Jan 15, 2025 Jan 15, 2025
42505 CLONED RABBIT UNDEFINED Motilin 0.977237 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42506 CLONED RABBIT UNDEFINED [Nle13]-Motilin 0.851138 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42507 CLONED RABBIT UNDEFINED erythromycin-A 190.546 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42508 CLONED RABBIT 35S-GTPGammaS Motilin 1.34896 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42509 CLONED RABBIT 35S-GTPGammaS [Nle13]-Motilin 1.69824 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42510 CLONED RABBIT 35S-GTPGammaS erythromycin-A 741.31 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42511 CLONED HUMAN UNDEFINED Motilin 0.162181 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42512 CLONED HUMAN UNDEFINED [Nle13]-Motilin 0.436516 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42513 CLONED HUMAN UNDEFINED erythromycin-A 512.861 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42514 CLONED HUMAN 35S-GTPGammaS Motilin 1.28825 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42515 CLONED HUMAN 35S-GTPGammaS [Nle13]-Motilin 1.94984 Dass NB, et al., 2003 Jan 15, 2025 Jan 15, 2025
42516 CLONED HUMAN Functional [leu13]pMOT(1-5) 8912.51 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42517 CLONED HUMAN Functional [leu13]pMOT(1-7) 6918.31 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42518 CLONED HUMAN Functional [leu13]pMOT(1-9) 4073.8 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42519 CLONED HUMAN Functional [leu13]pMOT(1-11) 89.1251 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42520 CLONED HUMAN Functional [leu13]pMOT(1-14) 3.16228 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42521 CLONED HUMAN Functional [leu13]pMOT(1-16) 2.13796 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42522 CLONED HUMAN Functional [leu13]pMOT(1-19) 0.977237 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42523 CLONED HUMAN Functional [leu13]pMOT(1-22) 1 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42524 CLONED HUMAN Functional [ala1,leu13]pMOT(1-14) 588.844 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42525 CLONED HUMAN Functional [ala3,leu13]pMOT(1-14) 1.31826 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42526 CLONED HUMAN Functional [ala4,leu13]pMOT(1-14) 2570.4 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42527 CLONED HUMAN Functional [ala5,leu13]pMOT(1-14) 28.8403 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42528 CLONED HUMAN Functional [ala6,leu13]pMOT(1-14) 46.7735 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42529 CLONED HUMAN Functional [ala7,leu13]pMOT(1-14) 1445.44 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42530 CLONED HUMAN Functional [ala8,leu13]pMOT(1-14) 36.3078 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42531 CLONED HUMAN Functional [ala9,leu13]pMOT(1-14) 75.8578 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42532 CLONED HUMAN Functional [ala10,leu13]pMOT(1-14) 5.01187 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42533 CLONED HUMAN Functional [ala11,leu13]pMOT(1-14) 4.57088 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42534 CLONED HUMAN Functional [ala12,leu13]pMOT(1-14) 6.30957 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42535 CLONED HUMAN Functional [ala13,leu13]pMOT(1-14) 7.24436 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42536 CLONED HUMAN Functional [ala14,leu13]pMOT(1-14) 7.07946 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42537 CLONED HUMAN Functional erythromycin-A 77.6247 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42538 CLONED HUMAN Functional N-ethyl, N-Methyl Erythromycin-A 239.883 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42539 CLONED HUMAN Functional Erythromycin-A enol ether 8.31764 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42540 CLONED HUMAN Functional Erythromycin-B 144.544 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42541 CLONED HUMAN Functional Erythromycin-B enol ether 7.58578 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42542 CLONED HUMAN Functional N-ethyl, N-methyl Erythromycin-A enol ether 6.0256 Thielemans L, et al., 2002 Jan 15, 2025 Jan 15, 2025
42543 UNDEFINED UNDEFINED Functional LY-364947 59 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42544 UNDEFINED UNDEFINED Functional 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42545 UNDEFINED UNDEFINED Functional 1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole 4100 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42546 UNDEFINED UNDEFINED Functional 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42547 UNDEFINED UNDEFINED Functional 6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole 47 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42548 UNDEFINED UNDEFINED Functional 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 68 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42549 UNDEFINED UNDEFINED Functional LY-364947 400 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42550 UNDEFINED UNDEFINED Functional 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42551 UNDEFINED UNDEFINED Functional 1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42552 UNDEFINED UNDEFINED Functional 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42553 UNDEFINED UNDEFINED Functional 6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole 1300 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42554 UNDEFINED UNDEFINED Functional 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 409 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42555 UNDEFINED UNDEFINED Functional LY-364947 1400 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42556 UNDEFINED UNDEFINED Functional 5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42557 UNDEFINED UNDEFINED Functional 1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42558 UNDEFINED UNDEFINED Functional 1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42559 UNDEFINED UNDEFINED Functional 6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole >10000 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42560 UNDEFINED UNDEFINED Functional 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 9450 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42561 UNDEFINED UNDEFINED Functional LY-364947 40 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42562 UNDEFINED UNDEFINED Functional 6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole 15 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42563 UNDEFINED UNDEFINED Functional 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 57 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42564 UNDEFINED UNDEFINED Functional LY-364947 81 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42565 UNDEFINED UNDEFINED Functional 6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole 42 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42566 UNDEFINED UNDEFINED Functional 6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole 118 Li HY, et al., 2006 Jan 15, 2025 Jan 15, 2025
42567 Alpha1A CLONED UNDEFINED UNDEFINED PRAZOSIN 0.2 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42568 Alpha1A CLONED UNDEFINED UNDEFINED Terazosin 6.3 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42569 Alpha1A CLONED UNDEFINED UNDEFINED Doxazosin 3.16 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42570 Alpha1A CLONED UNDEFINED UNDEFINED Alfuzosin 10 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42571 Alpha1A CLONED UNDEFINED UNDEFINED Urapidil-5-methyl 0.63 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42572 Alpha1A CLONED UNDEFINED UNDEFINED RS-100975 1 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42573 Alpha1A CLONED UNDEFINED UNDEFINED WB 4101 0.16 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42574 Alpha1A CLONED UNDEFINED UNDEFINED RS-17053 0.6 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42575 Alpha1B CLONED UNDEFINED UNDEFINED PRAZOSIN 0.25 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42576 Alpha1B CLONED UNDEFINED UNDEFINED Terazosin 2 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42577 Alpha1B CLONED UNDEFINED UNDEFINED Doxazosin 1 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42578 Alpha1B CLONED UNDEFINED UNDEFINED Alfuzosin 10 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42579 Alpha1B CLONED UNDEFINED UNDEFINED Urapidil-5-methyl 40 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42580 Alpha1B CLONED UNDEFINED UNDEFINED RS-100975 79 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42581 Alpha1B CLONED UNDEFINED UNDEFINED WB 4101 2.5 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42582 Alpha1B CLONED UNDEFINED UNDEFINED RS-17053 16 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42583 Alpha1C CLONED UNDEFINED UNDEFINED PRAZOSIN 0.32 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42584 Alpha1C CLONED UNDEFINED UNDEFINED Terazosin 2.5 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42585 Alpha1C CLONED UNDEFINED UNDEFINED Doxazosin 4 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42586 Alpha1C CLONED UNDEFINED UNDEFINED Alfuzosin 3.16 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42587 Alpha1C CLONED UNDEFINED UNDEFINED Urapidil-5-methyl 10 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42588 Alpha1C CLONED UNDEFINED UNDEFINED RS-100975 100 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42589 Alpha1C CLONED UNDEFINED UNDEFINED WB 4101 0.25 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42590 Alpha1C CLONED UNDEFINED UNDEFINED RS-17053 16 Kinsella GK, et al., 2006 Jan 15, 2025 Jan 15, 2025
42591 CLONED HUMAN Functional 2-amino-4-oxo-6-methyl-5-substituted pyrrolo[2,3-d]pyrimidine 54 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42592 CLONED HUMAN Functional 2-Amino-6-methyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 150 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42593 CLONED HUMAN Functional N-[4-[(2-amino-6-ethyl-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidin-5-yl)thio]benzoyl]-L-glutamic acid 90 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42594 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3',4'-dichlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 230 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42595 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 240 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42596 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-fluorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2700 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42597 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 3.1E-5 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42598 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 1000 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42599 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine >10000 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42600 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2600 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42601 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]p-yrimidine 1100 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42602 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 3.2E-5 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42603 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3',5'-trifluoromethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 2.2E-5 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42604 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(2',6'-dimethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine >10000 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42605 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(1'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 5600 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42606 CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(2'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine 5600 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42607 CLONED HUMAN Functional PDDF 72 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42608 CLONED HUMAN Functional raltitrexed 380 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42609 CLONED HUMAN Functional Pemetrexed 9500 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42610 DHFR CLONED HUMAN Functional 2-amino-4-oxo-6-methyl-5-substituted pyrrolo[2,3-d]pyrimidine 2100 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42611 DHFR CLONED HUMAN Functional N-[4-[(2-amino-6-ethyl-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidin-5-yl)thio]benzoyl]-L-glutamic acid 420 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42612 DHFR CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(3',4'-dichlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine >10000 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42613 DHFR CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine >10000 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025
42614 DHFR CLONED HUMAN Functional 2-Amino-6-ethyl-5-[(4'-fluorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine >10000 Gangjee A, et al., 2006 Jan 15, 2025 Jan 15, 2025