The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 39,001-40,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
41605SLC6A3CLONEDRAT3H-WIN 35,4284,4'-DifluoroBZT8Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41606SLC6A3CLONEDRAT3H-WIN 35,4284-TrifluoromethylBZT541Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41607SLC6A3CLONEDRAT3H-WIN 35,428N-CHO-4,4'-diFBZT>10000Ukairo UT, et al., 2005Jan 15, 2025Jan 15, 2025
41608DORCLONEDHUMAN3H-DADLEN-DESMETHYLCLOZAPINE127.9PDSP Certified DataJan 15, 2025Jan 15, 2025
41609KORCLONEDHUMAN3H-DiprenorphineN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
416105-HT1ACLONEDHUMAN3H-8-OH-DPATN-DESMETHYLCLOZAPINE13.9PDSP Certified DataJan 15, 2025Jan 15, 2025
416115-HT1BCLONEDHUMAN3H-GR-125743N-DESMETHYLCLOZAPINE406.8PDSP Certified DataJan 15, 2025Jan 15, 2025
416125-HT1DCLONEDHUMAN3H-GR-125743N-DESMETHYLCLOZAPINE476.2PDSP Certified DataJan 15, 2025Jan 15, 2025
416135-HT1ECLONEDHUMAN3H-5HTN-DESMETHYLCLOZAPINE393.4PDSP Certified DataJan 15, 2025Jan 15, 2025
416145-HT2ACLONEDHUMAN3H-KETANSERINN-DESMETHYLCLOZAPINE10.9PDSP Certified DataJan 15, 2025Jan 15, 2025
416155-HT2CCLONEDRAT3H-MESULERGINEN-DESMETHYLCLOZAPINE11.9PDSP Certified DataJan 15, 2025Jan 15, 2025
416165-HT3CLONEDHUMAN3H-ZACOPRIDEN-DESMETHYLCLOZAPINE272.2PDSP Certified DataJan 15, 2025Jan 15, 2025
41617CB1CLONEDHUMAN3H-LSDN-DESMETHYLCLOZAPINE350.6PDSP Certified DataJan 15, 2025Jan 27, 2025
416185-HT6CLONEDHUMAN3H-LSDN-DESMETHYLCLOZAPINE11.6PDSP Certified DataJan 15, 2025Jan 15, 2025
416195-HT7CLONEDHUMAN3H-LSDN-DESMETHYLCLOZAPINE60.1PDSP Certified DataJan 15, 2025Jan 15, 2025
416205-HT2BCLONEDHUMAN3H-LSDN-DESMETHYLCLOZAPINE2.8PDSP Certified DataJan 15, 2025Jan 15, 2025
41621Alpha1ACLONEDHUMAN3H-PRAZOSINN-DESMETHYLCLOZAPINE104.8PDSP Certified DataJan 15, 2025Jan 15, 2025
41622Alpha1BCLONEDHUMAN3H-PRAZOSINN-DESMETHYLCLOZAPINE85.2PDSP Certified DataJan 15, 2025Jan 15, 2025
41623Alpha2ACLONEDHUMAN3H-CLONIDINEN-DESMETHYLCLOZAPINE137.6PDSP Certified DataJan 15, 2025Jan 15, 2025
41624Alpha2BCLONEDHUMAN3H-CLONIDINEN-DESMETHYLCLOZAPINE95.1PDSP Certified DataJan 15, 2025Jan 15, 2025
41625Alpha2CCLONEDHUMAN3H-CLONIDINEN-DESMETHYLCLOZAPINE117.7PDSP Certified DataJan 15, 2025Jan 15, 2025
41626Beta1CLONEDHUMAN125I-PindololN-DESMETHYLCLOZAPINE6239.04PDSP Certified DataJan 15, 2025Jan 15, 2025
41627Beta2CLONEDHUMAN125I-PindololN-DESMETHYLCLOZAPINE4725PDSP Certified DataJan 15, 2025Jan 28, 2025
41628H1CLONEDHUMAN3H-PYRILAMINEN-DESMETHYLCLOZAPINE3.4PDSP Certified DataJan 15, 2025Jan 15, 2025
41629H2CLONEDHUMAN3H-TIOTIDINEN-DESMETHYLCLOZAPINE345.1PDSP Certified DataJan 15, 2025Jan 15, 2025
41630H3CLONEDGUINEA PIG3H-Alpha-Me-histamineN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41631H4CLONEDHUMAN3H-HistamineN-DESMETHYLCLOZAPINE1028PDSP Certified DataJan 15, 2025Jan 15, 2025
41632D1CLONEDHUMAN3H-SCH23390N-DESMETHYLCLOZAPINE14.3PDSP Certified DataJan 15, 2025Jan 15, 2025
41633D2CLONEDHUMAN3H-NMSPN-DESMETHYLCLOZAPINE115.2PDSP Certified DataJan 15, 2025Jan 15, 2025
41634D3CLONEDRAT3H-NMSPN-DESMETHYLCLOZAPINE234PDSP Certified DataJan 15, 2025Jan 15, 2025
41635D4CLONEDHUMAN3H-NMSPN-DESMETHYLCLOZAPINE101.82PDSP Certified DataJan 15, 2025Jan 15, 2025
41636D5CLONEDHUMAN3H-SCH23390N-DESMETHYLCLOZAPINE283.6PDSP Certified DataJan 15, 2025Jan 15, 2025
41637SLC6A3CLONEDHUMAN3H-WIN 35,428N-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41638NETCLONEDHUMAN3H-NisoxetineN-DESMETHYLCLOZAPINE493.9PDSP Certified DataJan 15, 2025Jan 15, 2025
41639M1CLONEDHUMAN3H-QNBN-DESMETHYLCLOZAPINE67.6PDSP Certified DataJan 15, 2025Jan 15, 2025
41640M2CLONEDHUMAN3H-QNBN-DESMETHYLCLOZAPINE414.5PDSP Certified DataJan 15, 2025Jan 15, 2025
41641M3CLONEDHUMAN3H-QNBN-DESMETHYLCLOZAPINE95.7PDSP Certified DataJan 15, 2025Jan 15, 2025
41642M4CLONEDHUMAN3H-QNBN-DESMETHYLCLOZAPINE169.9PDSP Certified DataJan 15, 2025Jan 15, 2025
41643M5CLONEDHUMAN3H-QNBN-DESMETHYLCLOZAPINE35.4PDSP Certified DataJan 15, 2025Jan 15, 2025
41645HEARTRAT3H-NitrendipineN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41646CB1BRAINRAT3H-CP-55940N-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41647CB2CLONEDHUMAN3H-CP-55940N-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41648EP3CLONEDHUMAN3H-PGE2N-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41649KORFOREBRAINRAT3H-MUSCIMOLN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 27, 2025
41650I1PC12RAT125I-PindololN-DESMETHYLCLOZAPINE757.3PDSP Certified DataJan 15, 2025Jan 15, 2025
41651MORCLONEDHUMAN3H-DiprenorphineN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41652NMDAFOREBRAINRAT3H-MK-801N-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41653SLC6A4CLONEDHUMAN3H-CITALOPRAMN-DESMETHYLCLOZAPINE316.6PDSP Certified DataJan 15, 2025Jan 15, 2025
41654Sigma 1BRAINRAT3H-Pentazocine(+)N-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41655CLONEDHUMAN3H-VASOPRESSINN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41656Sigma 2PC12RAT3H-DTGN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41657CLONEDHUMAN3H-VASOPRESSINN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41658V2CLONEDHUMAN3H-VASOPRESSINN-DESMETHYLCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
416685-HT1ACLONEDHUMAN3H-8-OH-DPATORG-522253.6PDSP Certified DataJan 15, 2025Jan 15, 2025
416695-HT1BCLONEDHUMAN3H-GR-125743ORG-52225.2PDSP Certified DataJan 15, 2025Jan 15, 2025
416705-HT1ECLONEDHUMAN3H-5HTORG-522237.4PDSP Certified DataJan 15, 2025Jan 15, 2025
416715-HT2ACLONEDHUMAN3H-KETANSERINORG-52220.3PDSP Certified DataJan 15, 2025Jan 15, 2025
416725-HT2CCLONEDRAT3H-MESULERGINEORG-52220.8PDSP Certified DataJan 15, 2025Jan 15, 2025
416735-HT3CLONEDHUMAN3H-ZACOPRIDEORG-5222447.6PDSP Certified DataJan 15, 2025Jan 15, 2025
41674CB1CLONEDHUMAN3H-LSDORG-52224PDSP Certified DataJan 15, 2025Jan 27, 2025
416755-HT6CLONEDHUMAN3H-LSDORG-52221.4PDSP Certified DataJan 15, 2025Jan 15, 2025
416765-HT7CLONEDHUMAN3H-LSDORG-52220.9PDSP Certified DataJan 15, 2025Jan 15, 2025
41677H2CLONEDHUMAN3H-TIOTIDINEORG-52222.3PDSP Certified DataJan 15, 2025Jan 15, 2025
41678H4CLONEDHUMAN3H-HistamineORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41679D1CLONEDHUMAN3H-SCH23390ORG-52222.9PDSP Certified DataJan 15, 2025Jan 15, 2025
41680D2CLONEDHUMAN3H-NMSPORG-52221.4PDSP Certified DataJan 15, 2025Jan 15, 2025
41681D3CLONEDRAT3H-NMSPORG-522246.2PDSP Certified DataJan 15, 2025Jan 15, 2025
41682D4CLONEDHUMAN3H-NMSPORG-52221.8PDSP Certified DataJan 15, 2025Jan 15, 2025
41683D5CLONEDHUMAN3H-SCH23390ORG-522222.7PDSP Certified DataJan 15, 2025Jan 15, 2025
41684SLC6A3CLONEDHUMAN3H-WIN 35,428ORG-52223136PDSP Certified DataJan 15, 2025Jan 15, 2025
41685M1CLONEDHUMAN3H-NMSORG-5222782PDSP Certified DataJan 15, 2025Jan 15, 2025
41686M2CLONEDHUMAN3H-NMSORG-5222915PDSP Certified DataJan 15, 2025Jan 15, 2025
41687M3CLONEDHUMAN3H-NMSORG-52223232PDSP Certified DataJan 15, 2025Jan 15, 2025
41688M4CLONEDHUMAN3H-QNBORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41689M5CLONEDHUMAN3H-NMSORG-5222272PDSP Certified DataJan 15, 2025Jan 15, 2025
41690HEARTRAT3H-NitrendipineORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41691CB1BRAINRAT3H-CP-55940ORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41692EP3CLONEDHUMAN3H-PGE2ORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41693I1PC12RAT125I-PindololORG-52222371PDSP Certified DataJan 15, 2025Jan 15, 2025
41694MORCLONEDHUMAN3H-DiprenorphineORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41695NMDAFOREBRAINRAT3H-MK-801ORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41696SLC6A4CLONEDHUMAN3H-CITALOPRAMORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41697Sigma 1BRAINRAT3H-Pentazocine(+)ORG-52222069PDSP Certified DataJan 15, 2025Jan 15, 2025
41698NETCLONEDHUMAN3H-NisoxetineORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41699KORCLONEDHUMAN3H-DiprenorphineORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41700Sigma 2PC12RAT3H-DTGORG-5222497.5PDSP Certified DataJan 15, 2025Jan 15, 2025
41701EP4CLONEDHUMAN3H-PGE2ORG-5222>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
41702Alpha1ACLONEDHUMAN3H-PRAZOSINORG-52224.4PDSP Certified DataJan 15, 2025Jan 15, 2025
41703Alpha1BCLONEDHUMAN3H-PRAZOSINORG-52223.9PDSP Certified DataJan 15, 2025Jan 15, 2025
41704Alpha2ACLONEDHUMAN3H-CLONIDINEORG-522210.5PDSP Certified DataJan 15, 2025Jan 15, 2025
41705Alpha2BCLONEDHUMAN3H-CLONIDINEORG-522210.7PDSP Certified DataJan 15, 2025Jan 15, 2025
41706Alpha2CCLONEDHUMAN3H-CLONIDINEORG-522217.8PDSP Certified DataJan 15, 2025Jan 15, 2025
41707UNDEFINEDUNDEFINEDFunctionalThiabendazole472Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41708UNDEFINEDUNDEFINEDFunctionalCarbendazim>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41709UNDEFINEDUNDEFINEDFunctional2-Pyridin-3-yl-1H-benzoimidazol>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41710UNDEFINEDUNDEFINEDFunctional2-Thiophen-2-yl-1H-benzoimidazol>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41711UNDEFINEDUNDEFINEDFunctionalFuberidazole>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41712UNDEFINEDUNDEFINEDFunctional2-(1H-Benzoimidazol-2-yl)-phenol>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41713UNDEFINEDUNDEFINEDFunctional1H-Benzimidazol-2-yl-thiourea8956Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41714UNDEFINEDUNDEFINEDFunctional(1H-Benzimidazol-2-yl)-thiazol-2-yl-amin540Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41715UNDEFINEDUNDEFINEDFunctional2-Pyridin-2-yl-1H-benzoimidazol574Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41716UNDEFINEDUNDEFINEDFunctional6-(1H-Benzoimidazol-2-yl)-pyridin-2-ol1343Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41717UNDEFINEDUNDEFINEDFunctional2-(1H-Benzoimidazol-2-yl)-pyridin-3-ol777Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41718UNDEFINEDUNDEFINEDFunctional2-Pyrazin-2-yl-1H-benzoimidazol4591Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41719UNDEFINEDUNDEFINEDFunctional1-Methyl-2-thiazol-4-yl-1H-benzoimidazol497Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41720UNDEFINEDUNDEFINEDFunctional1-Benzyl-2-thiazol-4-yl-1H-benzoimidazole461Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41721UNDEFINEDUNDEFINEDFunctional1-Benzyl-2-pyridin-2-yl-1H-benzoimidazole992Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41722UNDEFINEDUNDEFINEDFunctional5-Methyl-2-thiazol-4-yl-1(3)H-benzoimidazole7157Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41723UNDEFINEDUNDEFINEDFunctional5-Methyl-2-pyridin-2-yl-1(3)H-benzoimidazol2086Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41724UNDEFINEDUNDEFINEDFunctional5,6-Dimethyl-2-thiazol-4-yl-1H-benzoimidazole>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41725UNDEFINEDUNDEFINEDFunctional5,6-Dimethyl-2-pyridin-2-yl-1H-benzoimidazole2433Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41726UNDEFINEDUNDEFINEDFunctional5-tert-Butyl-2-thiazol-4-yl-1H-benzimidazol3906Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41727UNDEFINEDUNDEFINEDFunctional5-tert-Butyl-2-pyridin-2-yl-1H-Benzoimidazole2598Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41728UNDEFINEDUNDEFINEDFunctional5-Nitro-2-thiazol-4-yl-1(3)H-benzoimidazole1218Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41729UNDEFINEDUNDEFINEDFunctional5-Nitro-2-pyridin-2-yl-1(3)H-benzoimidazol162Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41730UNDEFINEDUNDEFINEDFunctional5-Amino-2-thiazol-4-yl-1H-benzimidazol3390Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41731UNDEFINEDUNDEFINEDFunctional2-Pyridin-2-yl-3H-benzoimidazol-5-ylamine967Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41732UNDEFINEDUNDEFINEDFunctional5-Fluor-2-thiazol-4-yl-1H-benzimidazol4307Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41733UNDEFINEDUNDEFINEDFunctional6-Fluoro-2-pyridin-2-yl-1H-benzoimidazole1511Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41734UNDEFINEDUNDEFINEDFunctional5-Chlor-2-thiazol-4-yl-1H-benzimidazol5153Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41735UNDEFINEDUNDEFINEDFunctional5-Chloro-2-pyridin-2-yl-1(3)H-benzoimidazole1695Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41736UNDEFINEDUNDEFINEDFunctionalPhenyl-(2-thiazol-4-yl-1H-benzoimidazol-5-yl)-methanone2397Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41737UNDEFINEDUNDEFINEDFunctionalPhenyl-(2-pyridin-2-yl-3H-benzoimidazol-5-yl)-methanone403Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41738UNDEFINEDUNDEFINEDFunctional2-Pyridin-2-yl-3H-benzoimidazole-5-carbonitrile431Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41739UNDEFINEDUNDEFINEDFunctionalMebendazole>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41740UNDEFINEDUNDEFINEDFunctionalAlbendazole>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41741UNDEFINEDUNDEFINEDFunctionalFenbendazole>10000Schiffmann R, et al., 2006Jan 15, 2025Jan 15, 2025
41742AMPACORTICAL MEMBRANESRAT3H-AMPAAMPA23Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41743AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate94Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41744AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41745AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41746AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate1500Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41747AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate5800Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41748AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate700Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41749AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41750AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41751AMPACORTICAL MEMBRANESRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate30Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41752KACORTICAL MEMBRANESRAT3H-Kainic acidAMPA>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41753KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate4900Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41754KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41755KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41756KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41757KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41758KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41759KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41760KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41761KACORTICAL MEMBRANESRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 15, 2025
41762NMDACORTICAL MEMBRANESRAT3H-CGP39653AMPA>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41763NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(thiazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41764NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41765NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-imidazol-2-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41766NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41767NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Monohydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41768NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-1,2,4-triazol-3-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41769NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41770NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Dihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41771NMDACORTICAL MEMBRANESRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic Acid Hemihydrate>10000Bang-Andersen B, et al., 1997Jan 15, 2025Jan 28, 2025
41772CLONEDHUMANFunctional17beta-Estradiol0.019Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41773CLONEDHUMANFunctional(+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol0.059Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41774CLONEDHUMANFunctional1-ethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol0.31Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41775CLONEDHUMANFunctional(+/-)-3-Ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxylic Acid158Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41776CLONEDHUMANFunctional(+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride100Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41777CLONEDHUMANFunctional(+/-)-N-(4-(2-(Dimethylamino)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide monohydrochloride152Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41778CLONEDHUMANFunctional(+/-)-3-Ethyl-6-hydroxy-N,2-bis(4-hydroxyphenyl)-1H-indene-1-carboxamide427Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41779CLONEDHUMANFunctional2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol4.3Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41780CLONEDHUMANFunctional1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol7Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41781CLONEDHUMANFunctional1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol3.9Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41782CLONEDHUMANFunctional1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol17Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41783CLONEDHUMANFunctional2-(4-Hydroxyphenyl)-1-p-tolyl-3H-inden-5-ol17Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41784CLONEDHUMANFunctional1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-olol15Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41785CLONEDHUMANFunctional1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol6.7Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41786CLONEDHUMANFunctional1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol109Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41787CLONEDHUMANFunctional1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol14Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41788CLONEDHUMANFunctional17beta-Estradiol0.098Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41789CLONEDHUMANFunctional(+/-)-1,3-Diethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol0.3Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41790CLONEDHUMANFunctional1-ethyl-2-(4-hydroxyphenyl)-3H-inden-5-ol0.3Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41791CLONEDHUMANFunctional(+/-)-3-Ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxylic Acid52Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41792CLONEDHUMANFunctional(+/-)-N-(4-(2-(Dimethylamino)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide monohydrochloride512Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41793CLONEDHUMANFunctional2-(4-hydroxyphenyl)-1-phenyl-3H-inden-5-ol54Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41794CLONEDHUMANFunctional1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol10Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41795CLONEDHUMANFunctional1-Benzyl-2-(4-hydroxyphenyl)-3H-inden-5-ol37Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41796CLONEDHUMAN3H-EstradiolOHT0.04Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41797CLONEDHUMAN3H-Estradiolraloxifene0.03Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41798CLONEDHUMAN3H-Estradiol(+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride184Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41799CLONEDHUMAN3H-Estradiol1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol8.5Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41800CLONEDHUMAN3H-Estradiol1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol1.7Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41801CLONEDHUMAN3H-Estradiol1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol24Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41802CLONEDHUMAN3H-Estradiol1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol2.1Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41803CLONEDHUMAN3H-Estradiol1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol0.67Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41804CLONEDHUMAN3H-Estradiol1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol59Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41805CLONEDHUMAN3H-Estradiol4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzamide4.2Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41806CLONEDHUMAN3H-EstradiolMethyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate7.3Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41807CLONEDHUMAN3H-EstradiolTamoxifen, 4-hydroxy0.014Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41808CLONEDHUMAN3H-Estradiolraloxifene4.5Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41809CLONEDHUMAN3H-Estradiol(+/-)-N-(4-(2-(Piperidinyl)ethoxy)phenyl)-3-ethyl-6-hydroxy-2-(4-hydroxyphenyl)-1H-indene-1-carboxamide Monohydrochloride147Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41810CLONEDHUMAN3H-Estradiol1,2-Bis(4-hydroxyphenyl)-3H-inden-5-ol1.3Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41811CLONEDHUMAN3H-Estradiol1-(4-(2-(Piperidin-1-yl)ethoxy)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol0.19Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41812CLONEDHUMAN3H-Estradiol1-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol2.8Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41813CLONEDHUMAN3H-Estradiol1-(4-Chlorophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol0.49Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41814CLONEDHUMAN3H-Estradiol2-(4-Hydroxyphenyl)-1-p-tolyl-3H-inden-5-ol1.3Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41815CLONEDHUMAN3H-Estradiol1-(4-(Trifluoromethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol0.91Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41816CLONEDHUMAN3H-Estradiol1-(4-Aminophenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol2.2Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41817CLONEDHUMAN3H-Estradiol4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoic Acid421Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41818CLONEDHUMAN3H-Estradiol1-(4-(Bromomethyl)phenyl)-2-(4-hydroxyphenyl)-3H-inden-5-ol15Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41819CLONEDHUMAN3H-Estradiol4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzamide0.46Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41820CLONEDHUMAN3H-EstradiolMethyl 4-(6-Hydroxy-2-(4-hydroxyphenyl)-1H-inden-3-yl)benzoate3.8Clegg NJ, et al., 2005Jan 15, 2025Jan 15, 2025
41821H3CLONEDHUMAN3H-Alpha-Me-histamineABT-2390.45Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41822H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(2-nitrophenyl)amine0.31Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41823H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(4-nitrophenyl)amine0.74Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41824H3CLONEDHUMAN3H-Alpha-Me-histamine2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone0.74Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41825H3CLONEDHUMAN3H-Alpha-Me-histamine3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)benzonitrile0.4Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41826H3CLONEDHUMAN3H-Alpha-Me-histamine(6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine0.31Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41827H3CLONEDHUMAN3H-Alpha-Me-histamine3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyrazine-2-carbonitrile1.04Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41828H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrazin-2-ylamine0.29Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41829H3CLONEDHUMAN3H-Alpha-Me-histamine(5-Bromopyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine1.22Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41830H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-5-ylamine0.69Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41831H3CLONEDHUMAN3H-Alpha-Me-histamine(5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine0.33Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41832H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-2-ylamine0.84Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41833H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitrothiazol-2-yl)amine0.19Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41834H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(3-nitropyridin-2-yl)amine0.43Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41835H3CLONEDHUMAN3H-Alpha-Me-histamine(3,5-Dinitropyridin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine0.71Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41836H3CLONEDHUMAN3H-Alpha-Me-histamine4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile0.13Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41837H3CLONEDHUMAN3H-Alpha-Me-histamine2-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile0.74Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41838H3CLONEDHUMAN3H-Alpha-Me-histamine6-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile0.34Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41839H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitropyridin-2-yl)amine0.3Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41840H3CLONEDRAT3H-Alpha-Me-histamineABT-2391.23Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41841H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(2-nitrophenyl)amine0.87Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41842H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(4-nitrophenyl)amine2.12Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41843H3CLONEDRAT3H-Alpha-Me-histamine2,2,2-Trifluoro-1-[4-({2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)phenyl]ethanone2.36Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41844H3CLONEDRAT3H-Alpha-Me-histamine3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)benzonitrile1.18Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41845H3CLONEDRAT3H-Alpha-Me-histamine(6-Chloropyridazin-3-yl){2-[2-(2-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine1.58Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41846H3CLONEDRAT3H-Alpha-Me-histamine3-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyrazine-2-carbonitrile3.96Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41847H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrazin-2-ylamine0.8Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41848H3CLONEDRAT3H-Alpha-Me-histamine(5-Bromopyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine4.02Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41849H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-5-ylamine2.51Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41850H3CLONEDRAT3H-Alpha-Me-histamine(5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine0.58Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41851H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}pyrimidin-2-ylamine3.27Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41852H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitrothiazol-2-yl)amine0.68Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41853H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(3-nitropyridin-2-yl)amine2.71Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41854H3CLONEDRAT3H-Alpha-Me-histamine(3,5-Dinitropyridin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amine2.88Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41855H3CLONEDRAT3H-Alpha-Me-histamine4-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)pyridine-2,6-dicarbonitrile0.4Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41856H3CLONEDRAT3H-Alpha-Me-histamine2-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile1.92Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41857H3CLONEDRAT3H-Alpha-Me-histamine6-({2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}amino)nicotinonitrile1.42Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41858H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylmethyl}(5-nitropyridin-2-yl)amine1.19Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41859H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(2-nitrophenyl)amine0.22Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41860H3CLONEDHUMAN3H-Alpha-Me-histamine4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile0.27Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41861H3CLONEDHUMAN3H-Alpha-Me-histamine3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile0.29Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41862H3CLONEDHUMAN3H-Alpha-Me-histamine(5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine0.62Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41863H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-2-ylamine0.31Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41864H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-5-ylamine0.08Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41865H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrazin-2-ylamine0.11Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41866H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine0.05Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41867H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(3-nitropyridin-2-yl)amine0.14Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41868H3CLONEDHUMAN3H-Alpha-Me-histamine6-Methyl-2-{2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}nicotinonitrile2.98Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41869H3CLONEDHUMAN3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-trifluoromethylpyridin-2-yl)amine0.54Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41870H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(2-nitrophenyl)amine0.87Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41871H3CLONEDRAT3H-Alpha-Me-histamine4-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile1.35Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41872H3CLONEDRAT3H-Alpha-Me-histamine3-{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}benzonitrile1.47Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41873H3CLONEDRAT3H-Alpha-Me-histamine(5-Ethylpyrimidin-2-yl){2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}amine2.51Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41874H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-2-ylamine2.01Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41875H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrimidin-5-ylamine0.27Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41876H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}pyrazin-2-ylamine0.38Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41877H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-nitropyridin-2-yl)amine0.11Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41878H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(3-nitropyridin-2-yl)amine0.35Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41879H3CLONEDRAT3H-Alpha-Me-histamine6-Methyl-2-{2-[2-(2-(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-ylamino}nicotinonitrile17.9Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41880H3CLONEDRAT3H-Alpha-Me-histamine{2-[2-(2-(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl}(5-trifluoromethylpyridin-2-yl)amine2.76Sun M, et al., 2005Jan 15, 2025Jan 15, 2025
41881AMPACORTICALRAT3H-AMPA(S)-AMPA21Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41882AMPACORTICALRAT3H-AMPA1-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41883AMPACORTICALRAT3H-AMPA2-Me-Tet-AMPA27Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41884AMPACORTICALRAT3H-AMPA(S)-(2)-Me-Tet-AMPA9Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41885AMPACORTICALRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41886AMPACORTICALRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41887AMPACORTICALRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41888AMPACORTICALRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid134Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41889AMPACORTICALRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid2500Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41890AMPACORTICALRAT3H-AMPA(RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid6200Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41891KACORTICALRAT3H-Kainic acid(S)-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41892KACORTICALRAT3H-Kainic acid1-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41893KACORTICALRAT3H-Kainic acid2-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41894KACORTICALRAT3H-Kainic acid(S)-(2)-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41895KACORTICALRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41896KACORTICALRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41897KACORTICALRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41898KACORTICALRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41899KACORTICALRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41900KACORTICALRAT3H-Kainic acid(RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 15, 2025
41901NMDACORTICALRAT3H-CGP39653(S)-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41902NMDACORTICALRAT3H-CGP396531-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41903NMDACORTICALRAT3H-CGP396532-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41904NMDACORTICALRAT3H-CGP39653(S)-(2)-Me-Tet-AMPA>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41905NMDACORTICALRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-ethyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41906NMDACORTICALRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-propyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41907NMDACORTICALRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(1-isopropyl-1H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41908NMDACORTICALRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41909NMDACORTICALRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41910NMDACORTICALRAT3H-CGP39653(RS)-2-Amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid>10000Vogensen SB, et al., 2005Jan 15, 2025Jan 28, 2025
41911GABAACLONEDHUMAN3H-RO-15-17883,5-diphenylpyridazine36van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41912GABAACLONEDHUMAN3H-RO-15-17884-(6-Phenylpyridazin-4-yl)benzonitrile27van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41913GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenylpyridazin-4-yl)benzonitrile7van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41914GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-phenyl pyridazine7.5van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41915GABAACLONEDHUMAN3H-RO-15-17885-(3-Isopropoxy-phenyl)-3-phenyl pyridazine12van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41916GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester88van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41917GABAACLONEDHUMAN3H-RO-15-17885-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine8.5van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41918GABAACLONEDHUMAN3H-RO-15-17883-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine1.3van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41919GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-ethoxy pyridazine8.6van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41920GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-isopropoxypyridazine26van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41921GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine49van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41922GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine55van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41923GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine3.5van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41924GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine7.3van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41925GABAACLONEDHUMAN3H-RO-15-17883-(5-Phenylpyridazin-3-yl)benzonitrile666van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41926GABAACLONEDHUMAN3H-RO-15-17883,5-diphenylpyridazine45van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41927GABAACLONEDHUMAN3H-RO-15-17882-(6-Phenylpyridazin-4-yl)benzonitrile440van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41928GABAACLONEDHUMAN3H-RO-15-17884-(6-Phenylpyridazin-4-yl)benzonitrile81van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41929GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenylpyridazin-4-yl)benzonitrile14van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41930GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-phenyl pyridazine15van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41931GABAACLONEDHUMAN3H-RO-15-17885-(3-Isopropoxy-phenyl)-3-phenyl pyridazine27van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41932GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenyl-pyridazine-4-yl)-benzoic acid methyl ester29van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41933GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester45van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41934GABAACLONEDHUMAN3H-RO-15-17883-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine41van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41935GABAACLONEDHUMAN3H-RO-15-17885-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine10.4van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41936GABAACLONEDHUMAN3H-RO-15-17883-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine3.1van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41937GABAACLONEDHUMAN3H-RO-15-17883-[6-(2-Fluorophenyl)-pyridazin-4-yl]benzonitrile7.9van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41938GABAACLONEDHUMAN3H-RO-15-17883-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile7.2van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41939GABAACLONEDHUMAN3H-RO-15-17883-[6-(4-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile26van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41940GABAACLONEDHUMAN3H-RO-15-17883-[6-(2,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile23van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41941GABAACLONEDHUMAN3H-RO-15-17883-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile41van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41942GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-methoxypyridazine205van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41943GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-ethoxy pyridazine19van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41944GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-isopropoxypyridazine60van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41945GABAACLONEDHUMAN3H-RO-15-17883-(Benzyloxy)-5-(3-bromophenyl)pyridazine302van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41946GABAACLONEDHUMAN3H-RO-15-17883-(Benzyloxy)-5-(3-cyanophenyl)pyridazine60van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41947GABAACLONEDHUMAN3H-RO-15-17883-(6-Ethoxypyridazin-4-yl)benzonitrile72van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41948GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine113van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41949GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine120van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41950GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine7.3van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41951GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine22van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41952GABAACLONEDHUMAN3H-RO-15-17883-(6-ethylaminopyridazin-4-yl)-benzonitrile79van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41953GABAACLONEDHUMAN3H-RO-15-1788N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine51van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41954GABAACLONEDHUMAN3H-RO-15-1788N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine15van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41955GABAACLONEDHUMAN3H-RO-15-17883-(5-Phenylpyridazin-3-yl)benzonitrile666van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41956GABAACLONEDHUMAN3H-RO-15-17883,5-diphenylpyridazine29van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41957GABAACLONEDHUMAN3H-RO-15-17882-(6-Phenylpyridazin-4-yl)benzonitrile323van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41958GABAACLONEDHUMAN3H-RO-15-17884-(6-Phenylpyridazin-4-yl)benzonitrile56van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41959GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenylpyridazin-4-yl)benzonitrile5.2van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41960GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-phenyl pyridazine7.9van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41961GABAACLONEDHUMAN3H-RO-15-17885-(3-Isopropoxy-phenyl)-3-phenyl pyridazine8.4van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41962GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenyl-pyridazine-4-yl)-benzoic acid methyl ester11van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41963GABAACLONEDHUMAN3H-RO-15-17883-(6-Phenyl-pyridazin-4-yl)-thiophene-2-carboxylic acid methyl ester12van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41964GABAACLONEDHUMAN3H-RO-15-17883-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine12van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41965GABAACLONEDHUMAN3H-RO-15-17885-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine8.8van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41966GABAACLONEDHUMAN3H-RO-15-17883-Phenyl-5-(2-pyridin-4-yl-pyrimidin-4-yl)-pyridazine1.6van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41967GABAACLONEDHUMAN3H-RO-15-17883-[6-(2-Fluorophenyl)-pyridazin-4-yl]benzonitrile3.4van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41968GABAACLONEDHUMAN3H-RO-15-17883-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile4van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41969GABAACLONEDHUMAN3H-RO-15-17883-[6-(4-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile14van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41970GABAACLONEDHUMAN3H-RO-15-17883-[6-(2,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile17van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41971GABAACLONEDHUMAN3H-RO-15-17883-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile13van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41972GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-methoxypyridazine54van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41973GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-ethoxy pyridazine5.7van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41974GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-3-isopropoxypyridazine36van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41975GABAACLONEDHUMAN3H-RO-15-17883-(Benzyloxy)-5-(3-bromophenyl)pyridazine63van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41976GABAACLONEDHUMAN3H-RO-15-17883-(Benzyloxy)-5-(3-cyanophenyl)pyridazine17van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41977GABAACLONEDHUMAN3H-RO-15-17883-(6-Ethoxypyridazin-4-yl)benzonitrile36van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41978GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine27van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41979GABAACLONEDHUMAN3H-RO-15-17885-(3-Bromophenyl)-N,N-dimethylpyridazin-3-amine51van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41980GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine3.8van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41981GABAACLONEDHUMAN3H-RO-15-1788[5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine7.2van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41982GABAACLONEDHUMAN3H-RO-15-17883-(6-ethylaminopyridazin-4-yl)-benzonitrile33van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41983GABAACLONEDHUMAN3H-RO-15-1788N-Benzyl-5-(3-bromophenyl)pyridazin-3-amine19van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41984GABAACLONEDHUMAN3H-RO-15-1788N-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine6.1van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41985GABAACLONEDHUMAN3H-RO-15-17883-(5-Phenylpyridazin-3-yl)benzonitrile666van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
41986M1CLONEDHUMAN3H-QNBAdinazolam>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41987M1CLONEDHUMAN3H-QNBAMITRIPTYLINE14.7Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41988M1CLONEDHUMAN3H-QNBBUPROPION>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41989M1CLONEDHUMAN3H-QNBDESIPRAMINE110Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41990M1CLONEDHUMAN3H-QNBDesmethylsertraline1650Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41991M1CLONEDHUMAN3H-QNBDothiepin18Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41992M1CLONEDHUMAN3H-QNBDOXEPIN38Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41993M1CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41994M1CLONEDHUMAN3H-QNBFemoxetine92Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41995M1CLONEDHUMAN3H-QNBFLUOXETINE1030Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41996M1CLONEDHUMAN3H-QNBIMIPRAMINE42Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41997M1CLONEDHUMAN3H-QNBLofepramine67Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41998M1CLONEDHUMAN3H-QNBNORFLUOXETINE1200Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
41999M1CLONEDHUMAN3H-QNBNORTRYPTYLINE40Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42000M1CLONEDHUMAN3H-QNBPAROXETINE300Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42001M1CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.044Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42002M1CLONEDHUMAN3H-QNBSERTRALINE1300Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42003M1CLONEDHUMAN3H-QNBTRAZODONE>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42004M1CLONEDHUMAN3H-QNBVenlafaxine>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42005M2CLONEDHUMAN3H-QNBAdinazolam>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42006M2CLONEDHUMAN3H-QNBAMITRIPTYLINE11.8Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42007M2CLONEDHUMAN3H-QNBBUPROPION>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42008M2CLONEDHUMAN3H-QNBDESIPRAMINE540Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42009M2CLONEDHUMAN3H-QNBDesmethylsertraline3300Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42010M2CLONEDHUMAN3H-QNBDothiepin109Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42011M2CLONEDHUMAN3H-QNBDOXEPIN160Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42012M2CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42013M2CLONEDHUMAN3H-QNBFemoxetine150Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42014M2CLONEDHUMAN3H-QNBFLUOXETINE2700Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42015M2CLONEDHUMAN3H-QNBIMIPRAMINE88Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42016M2CLONEDHUMAN3H-QNBLofepramine330Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42017M2CLONEDHUMAN3H-QNBNORFLUOXETINE4600Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42018M2CLONEDHUMAN3H-QNBNORTRYPTYLINE110Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42019M2CLONEDHUMAN3H-QNBPAROXETINE340Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42020M2CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.03Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42021M2CLONEDHUMAN3H-QNBSERTRALINE2100Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42022M2CLONEDHUMAN3H-QNBTRAZODONE>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42023M2CLONEDHUMAN3H-QNBVenlafaxine>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42024M3CLONEDHUMAN3H-QNBAdinazolam>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42025M3CLONEDHUMAN3H-QNBAMITRIPTYLINE12.8Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42026M3CLONEDHUMAN3H-QNBBUPROPION>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42027M3CLONEDHUMAN3H-QNBDESIPRAMINE210Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42028M3CLONEDHUMAN3H-QNBDesmethylsertraline3500Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42029M3CLONEDHUMAN3H-QNBDothiepin38Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42030M3CLONEDHUMAN3H-QNBDOXEPIN52Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42031M3CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42032M3CLONEDHUMAN3H-QNBFemoxetine220Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42033M3CLONEDHUMAN3H-QNBFLUOXETINE1000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42034M3CLONEDHUMAN3H-QNBIMIPRAMINE60Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42035M3CLONEDHUMAN3H-QNBLofepramine130Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42036M3CLONEDHUMAN3H-QNBNORFLUOXETINE760Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42037M3CLONEDHUMAN3H-QNBNORTRYPTYLINE50Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42038M3CLONEDHUMAN3H-QNBPAROXETINE80Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42039M3CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.08Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42040M3CLONEDHUMAN3H-QNBSERTRALINE1300Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42041M3CLONEDHUMAN3H-QNBTRAZODONE>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42042M3CLONEDHUMAN3H-QNBVenlafaxine>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42043M4CLONEDHUMAN3H-QNBAdinazolam>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42044M4CLONEDHUMAN3H-QNBAMITRIPTYLINE7.2Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42045M4CLONEDHUMAN3H-QNBBUPROPION>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42046M4CLONEDHUMAN3H-QNBDESIPRAMINE160Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42047M4CLONEDHUMAN3H-QNBDesmethylsertraline3100Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42048M4CLONEDHUMAN3H-QNBDothiepin61Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42049M4CLONEDHUMAN3H-QNBDOXEPIN82Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42050M4CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42051M4CLONEDHUMAN3H-QNBFemoxetine470Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42052M4CLONEDHUMAN3H-QNBFLUOXETINE2900Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42053M4CLONEDHUMAN3H-QNBIMIPRAMINE112Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42054M4CLONEDHUMAN3H-QNBLofepramine340Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42055M4CLONEDHUMAN3H-QNBNORFLUOXETINE2600Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42056M4CLONEDHUMAN3H-QNBNORTRYPTYLINE84Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42057M4CLONEDHUMAN3H-QNBPAROXETINE320Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42058M4CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.037Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42059M4CLONEDHUMAN3H-QNBSERTRALINE1400Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42060M4CLONEDHUMAN3H-QNBTRAZODONE>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42061M4CLONEDHUMAN3H-QNBVenlafaxine>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42062M5CLONEDHUMAN3H-QNBAdinazolam>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42063M5CLONEDHUMAN3H-QNBAMITRIPTYLINE15.7Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42064M5CLONEDHUMAN3H-QNBBUPROPION>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42065M5CLONEDHUMAN3H-QNBDESIPRAMINE143Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42066M5CLONEDHUMAN3H-QNBDesmethylsertraline3800Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42067M5CLONEDHUMAN3H-QNBDothiepin92Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42068M5CLONEDHUMAN3H-QNBDOXEPIN75Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42069M5CLONEDHUMAN3H-QNBEtoperidone>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42070M5CLONEDHUMAN3H-QNBFemoxetine400Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42071M5CLONEDHUMAN3H-QNBFLUOXETINE2700Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42072M5CLONEDHUMAN3H-QNBIMIPRAMINE83Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42073M5CLONEDHUMAN3H-QNBLofepramine460Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42074M5CLONEDHUMAN3H-QNBNORFLUOXETINE2200Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42075M5CLONEDHUMAN3H-QNBNORTRYPTYLINE97Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42076M5CLONEDHUMAN3H-QNBPAROXETINE650Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42077M5CLONEDHUMAN3H-QNBQuinuclidinyl benzilate0.065Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42078M5CLONEDHUMAN3H-QNBSERTRALINE1900Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42079M5CLONEDHUMAN3H-QNBTRAZODONE>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42080M5CLONEDHUMAN3H-QNBVenlafaxine>10000Stanton T, et al., 1993Jan 15, 2025Jan 15, 2025
42081Alpha2BCLONEDHUMAN35S-GTPGammaSA-54741912.011Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42082Alpha2BCLONEDHUMAN35S-GTPGammaSalpha-Methyl-(+/-)norepinephrine,(+/-)2630.27Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42083Alpha2BCLONEDHUMAN35S-GTPGammaSCLONIDINE69.1831Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42084Alpha2BCLONEDHUMAN35S-GTPGammaSDexmedetomidine33.8844Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42085Alpha2BCLONEDHUMAN35S-GTPGammaSEPINEPHRINE6309.57Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42086Alpha2BCLONEDHUMAN35S-GTPGammaSGuanabenz281.838Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42087Alpha2BCLONEDHUMAN35S-GTPGammaSGuanfacine1380.38Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42088Alpha2BCLONEDHUMAN35S-GTPGammaSLevlofexidine125.893Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42089Alpha2BCLONEDHUMAN35S-GTPGammaSNaphazoline407.38Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42090Alpha2BCLONEDHUMAN35S-GTPGammaSNaphthalene16.9824Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42091Alpha2BCLONEDHUMAN35S-GTPGammaSNOREPINEPHRINE2754.23Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42092Alpha2BCLONEDHUMAN35S-GTPGammaSOXYMETAZOLINE1778.28Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42093Alpha2BCLONEDHUMAN35S-GTPGammaSp-AMINOCLONIDINE29.5121Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42094Alpha2BCLONEDHUMAN35S-GTPGammaSST-91794.328Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42095Alpha2BCLONEDHUMAN35S-GTPGammaSTramazoline138.038Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42096Alpha2BCLONEDHUMAN35S-GTPGammaSUK-14,304954.993Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42097Alpha2BCLONEDHUMAN35S-GTPGammaSXylazine3467.37Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42098Alpha2BCLONEDHUMAN35S-GTPGammaSXylometazoline1047.13Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42099Alpha2BCLONEDHUMAN35S-GTPGammaSAlinidine6456.54Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42100Alpha2BCLONEDHUMAN35S-GTPGammaSB-HT 920512.861Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42101Alpha2BCLONEDHUMAN35S-GTPGammaSIDAZOXAN37.1535Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42102Alpha2BCLONEDHUMAN35S-GTPGammaSICI 10627067.6083Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42103Alpha2BCLONEDHUMAN35S-GTPGammaSIMILOXAN67.6083Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42104Alpha2BCLONEDHUMAN35S-GTPGammaSMK-9120.891251Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42105Alpha2BCLONEDHUMAN35S-GTPGammaSPHENTOLAMINE33.1131Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42106Alpha2BCLONEDHUMAN35S-GTPGammaSPRAZOSIN89.1251Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42107Alpha2BCLONEDHUMAN35S-GTPGammaSRAUWOLSCINE1.20226Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42108Alpha2BCLONEDHUMAN35S-GTPGammaSRilmenidine1737.8Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42109Alpha2BCLONEDHUMAN35S-GTPGammaSRX8210021.62181Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42110Alpha2BCLONEDHUMAN35S-GTPGammaSTOLAZOLINE3162.28Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42111Alpha2CCLONEDHUMAN35S-GTPGammaSA-54741776.247Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42112Alpha2CCLONEDHUMAN35S-GTPGammaSalpha-Methyl-(+/-)norepinephrine,(+/-)2884.03Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42113Alpha2CCLONEDHUMAN35S-GTPGammaSCLONIDINE134.896Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42114Alpha2CCLONEDHUMAN35S-GTPGammaSDexmedetomidine95.4993Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42115Alpha2CCLONEDHUMAN35S-GTPGammaSEPINEPHRINE1698.24Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42116Alpha2CCLONEDHUMAN35S-GTPGammaSGuanabenz446.684Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42117Alpha2CCLONEDHUMAN35S-GTPGammaSGuanfacine3890.45Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42118Alpha2CCLONEDHUMAN35S-GTPGammaSLevlofexidine173.78Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42119Alpha2CCLONEDHUMAN35S-GTPGammaSNaphazoline407.38Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42120Alpha2CCLONEDHUMAN35S-GTPGammaSNaphthalene3.31131Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42121Alpha2CCLONEDHUMAN35S-GTPGammaSNOREPINEPHRINE1348.96Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42122Alpha2CCLONEDHUMAN35S-GTPGammaSOXYMETAZOLINE239.883Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42123Alpha2CCLONEDHUMAN35S-GTPGammaSp-AMINOCLONIDINE21.3796Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42124Alpha2CCLONEDHUMAN35S-GTPGammaSST-91616.595Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42125Alpha2CCLONEDHUMAN35S-GTPGammaSTramazoline275.423Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42126Alpha2CCLONEDHUMAN35S-GTPGammaSUK-14,3041949.84Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42127Alpha2CCLONEDHUMAN35S-GTPGammaSXylazine>10000Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42128Alpha2CCLONEDHUMAN35S-GTPGammaSXylometazoline128.825Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42129Alpha2CCLONEDHUMAN35S-GTPGammaSAlinidine>10000Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42130Alpha2CCLONEDHUMAN35S-GTPGammaSB-HT 920954.993Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42131Alpha2CCLONEDHUMAN35S-GTPGammaSIDAZOXAN19.9526Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42132Alpha2CCLONEDHUMAN35S-GTPGammaSICI 106270281.838Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42133Alpha2CCLONEDHUMAN35S-GTPGammaSIMILOXAN151.356Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42134Alpha2CCLONEDHUMAN35S-GTPGammaSMK-9120.0676083Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42135Alpha2CCLONEDHUMAN35S-GTPGammaSPHENTOLAMINE257.04Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42136Alpha2CCLONEDHUMAN35S-GTPGammaSPRAZOSIN30.903Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42137Alpha2CCLONEDHUMAN35S-GTPGammaSRAUWOLSCINE0.549541Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42138Alpha2CCLONEDHUMAN35S-GTPGammaSRilmenidine4677.35Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42139Alpha2CCLONEDHUMAN35S-GTPGammaSRX8210020.794328Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42140Alpha2CCLONEDHUMAN35S-GTPGammaSTOLAZOLINE3715.35Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42141GABAACLONEDHUMANFunctional4-(6-Phenylpyridazin-4-yl)benzonitrile49van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42142GABAACLONEDHUMANFunctional5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine22van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42143GABAACLONEDHUMANFunctional3-Phenyl-5-[1,2,4]triazol-4-ylphenyl)pyridazine13van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42144GABAACLONEDHUMANFunctional5-[3-(2-Methyl-2H-[1,2,4]triazol-3-ylmethoxy)-phenyl]-3-phenyl-pyridazine43van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42145GABAACLONEDHUMANFunctional3-[6-(3-Fluoro-phenyl)-pyridazin-4-yl]-benzonitrile3.6van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42146GABAACLONEDHUMANFunctional3-[6-(3,4-Difluoro-phenyl)-pyridazin-4-yl]-benzonitrile32van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42147GABAACLONEDHUMANFunctional5-(3-Bromophenyl)-3-methoxypyridazine42van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42148GABAACLONEDHUMANFunctional5-(3-Bromophenyl)-3-ethoxy pyridazine39van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42149GABAACLONEDHUMANFunctional5-(3-Bromophenyl)-3-isopropoxypyridazine28van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42150GABAACLONEDHUMANFunctional3-(Benzyloxy)-5-(3-bromophenyl)pyridazine32van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42151GABAACLONEDHUMANFunctional3-(Benzyloxy)-5-(3-cyanophenyl)pyridazine60van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42152GABAACLONEDHUMANFunctional3-(6-Ethoxypyridazin-4-yl)benzonitrile19van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42153GABAACLONEDHUMANFunctional[5-(3-Bromo-phenyl)-pyridazin-3-yl]-methyl-amine3van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42154GABAACLONEDHUMANFunctional[5-(3-Bromophenyl)-N-pyridazin-3-yl]ethylamine2van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42155GABAACLONEDHUMANFunctional[5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine25van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42156GABAACLONEDHUMANFunctional3-(6-ethylaminopyridazin-4-yl)-benzonitrile8van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42157GABAACLONEDHUMANFunctionalN-Benzyl-5-(3-bromophenyl)pyridazin-3-amine66van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42158GABAACLONEDHUMANFunctionalN-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine59van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42159GABAACLONEDHUMANFunctional4-(6-Phenylpyridazin-4-yl)benzonitrile45van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42160GABAACLONEDHUMANFunctional5-(3-Isopropoxy-phenyl)-3-phenyl pyridazine18van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42161GABAACLONEDHUMANFunctional5-(3-Bromophenyl)-3-ethoxy pyridazine4van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42162GABAACLONEDHUMANFunctional5-(3-Bromophenyl)-3-isopropoxypyridazine12van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42163GABAACLONEDHUMANFunctional[5-(3-Bromo-phenyl)-pyridazin-3-yl]-isopropyl-amine14van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42164GABAACLONEDHUMANFunctionalN-Benzyl-5-(3-bromophenyl)pyridazin-3-amine14van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42165GABAACLONEDHUMANFunctionalN-Benzyl-5-(3-cyanophenyl)pyridazin-3-amine17van Niel MB, et al., 2005Jan 15, 2025Jan 27, 2025
42166CLONEDHUMANFunctional1-Isopropyl-1H-benzotriazole-5-carboxylic acid398.107Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42167CLONEDHUMANFunctional1-(2’-Methoxy-1’-methyl-ethyl)-1H-benzotriazole-5-carboxylic acid199.526Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42168CLONEDHUMANFunctional1-(2’-Ethoxy-ethyl)-1H-benzotriazole-5-carboxylic acid257.04Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42169CLONEDHUMANFunctional1-t-Butyl-1H-benzotriazole-5-carboxylic acid257.04Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42170CLONEDHUMANFunctional1-Pentyl-1H-benzotriazole-5-carboxylic acid288.403Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42171CLONEDHUMANFunctional1-(2’-Ethylsulfanyl-ethyl)-1H-benzotriazole-5-carboxylic acid301.995Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42172CLONEDHUMANFunctional1-(2-Methoxy-ethyl)-1H-benzotriazole-5-carboxylic acid316.228Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42173CLONEDHUMANFunctional1-(2’-Butyl)-1H-benzotriazole-5-carboxylic acid331.131Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42174CLONEDHUMANFunctional1-Butyl-1H-benzotriazole-5-carboxylic acid691.831Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42175CLONEDHUMANFunctional1-Ethyl-1H-benzotriazole-5-carboxylic acid891.251Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42176CLONEDHUMANFunctional1-(3’-Pentyl)-1H-benzotriazole-5-carboxylic acid3019.95Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42177CLONEDHUMANFunctional1-Propyl-1H-benzotriazole-5-carboxylic acid7413.1Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42178CLONEDHUMANFunctional1-Cyclopropyl-1H-benzotriazole-5-carboxylic acid2344.23Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42179CLONEDHUMANFunctional4-Ethyl-5-(4-piperidyl)-3-isoxazolol6626Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42180CLONEDHUMANFunctional3-Phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide4337Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42181CLONEDHUMANFunctionalN-Methyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide773Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42182CLONEDHUMANFunctionalN-Ethyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide175Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42183CLONEDHUMANFunctionalN-Isopropyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide199Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42184CLONEDHUMANFunctionalN-Butyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide79Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42185CLONEDHUMANFunctional{(3-Phenylpropionyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester105Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42186CLONEDHUMANFunctional{(3-Phenylpropionyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid376Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42187CLONEDHUMANFunctionalN-Benzyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide580Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42188CLONEDHUMANFunctionalN-Cyclohexyl-3-phenyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]propionamide150Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42189CLONEDHUMANFunctionalN-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide178Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42190CLONEDHUMANFunctionalN-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]nicotinamide1015Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42191CLONEDHUMANFunctionalN-Methyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isonicotinamide394Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42192CLONEDHUMANFunctionalN-Ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide41Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42193CLONEDHUMANFunctionalN-Propyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide28Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42194CLONEDHUMANFunctionalN-Butyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide20Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42195CLONEDHUMANFunctionalN-(2-Dimethylaminoethyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide1147Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42196CLONEDHUMANFunctionalN-(2-Hydroxyethyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide106Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42197CLONEDHUMANFunctional{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester34Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42198CLONEDHUMANFunctional{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid627Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42199CLONEDHUMANFunctional5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester26Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42200CLONEDHUMANFunctional5-{Isobutyryl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid8Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42201CLONEDHUMANFunctionalN-[4-(1H-Tetrazol-5-yl)butyl]-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide8Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42202CLONEDHUMANFunctionalN-(4-Cyanobutyl)-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isobutyramide20Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42203CLONEDHUMANFunctional4-Cyano-N-ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]benzamide37Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42204CLONEDHUMANFunctionalN-Ethyl-N-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]isonicotinamide95Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42205CLONEDHUMANFunctional1-Methyl-3-phenyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea1564Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42206CLONEDHUMANFunctional1-Ethyl-3,3-dimethyl-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea59Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42207CLONEDHUMANFunctional1,3-Diethyl-3-(4-hydroxybutyl)-1-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]urea60Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42208CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Methyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide321Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42209CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Ethyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide74Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42210CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Propyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide34Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42211CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Butyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide30Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42212CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Pentyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide19Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42213CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Hexyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide31Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42214CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Heptyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide73Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42215CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Octyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide269Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42216CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid Phenethyl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide43Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42217CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid (2-Hydroxyethyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide166Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42218CLONEDHUMANFunctional{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}acetic Acid Methyl Ester80Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42219CLONEDHUMANFunctional3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid Methyl Ester99Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42220CLONEDHUMANFunctional3-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}propionic Acid247Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42221CLONEDHUMANFunctional4-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}butyric Acid Methyl Ester75Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42222CLONEDHUMANFunctionalMorpholine-4-carboxylic Acid (3-Cyanopropyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amide40Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42223CLONEDHUMANFunctional5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid Methyl Ester42Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42224CLONEDHUMANFunctional5-{(Morpholine-4-carbonyl)-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]amino}pentanoic Acid14Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42225CLONEDHUMANFunctionalN-Phenethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide2650Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42226CLONEDHUMANFunctionalN-Methyl-N-phenethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide1990Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42227CLONEDHUMANFunctionalN-Benzyl-N-methyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide1000Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42228CLONEDHUMANFunctionalN-Methoxy-N-methyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide1450Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42229CLONEDHUMANFunctionalPyrrolidin-1-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone850Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42230CLONEDHUMANFunctionalMorpholin-4-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone1140Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42231CLONEDHUMANFunctionalPiperidin-1-yl-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)phenyl]methanone980Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42232CLONEDHUMANFunctionalN-(2-Cyanoethyl)-N-ethyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide290Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42233CLONEDHUMANFunctionalN,N-Diisobutyl-4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl)benzamide70Cheng JF, et al., 2006Jan 15, 2025Jan 15, 2025
42234KORBRAINRAT3H-MUSCIMOLSR 9553174Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42235KORBRAINRAT3H-MUSCIMOL4-PIOL9100Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42236KORBRAINRAT3H-MUSCIMOLThio-4-PIOL1870Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42237KORBRAINRAT3H-MUSCIMOL4-Methyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide2200Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42238KORBRAINRAT3H-MUSCIMOL5-(4-Piperidyl)-4-propylisothiazol-3-ol Hydrobromide440Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42239KORBRAINRAT3H-MUSCIMOL4-Benzyl-5-(4-piperidyl)isothiazol-3-ol Hydrobromide331Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42240KORBRAINRAT3H-MUSCIMOL4-(2-Naphthylmethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide5.2Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42241KORBRAINRAT3H-MUSCIMOL4-((1-Bromo-2-naphthyl)methyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide1.8Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42242KORBRAINRAT3H-MUSCIMOL4-(2,2-Diphenyl-1-ethyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide388Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42243KORBRAINRAT3H-MUSCIMOL4-(3,3-Diphenyl-1-propyl)-5-(4-piperidyl)isothiazol-3-ol Hydrobromide9.6Krehan D, et al., 2006Jan 15, 2025Jan 27, 2025
42244CLONEDHUMAN125I-[Ile]Motilin[Bpa5,Ile13]Motilin50Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42245CLONEDHUMAN125I-[Ile]MotilinMotilin2.3Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42246CLONEDHUMAN125I-[Ile]Motilin[D-Bpa5,Ile13]Motilin420Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42247CLONEDHUMAN125I-[Ile]Motilin[L-Bpa5,Ile13]Motilin50Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42248CLONEDHUMAN125I-[Ile]Motilincyanogen bromide, CNBr0.85Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42249CLONEDHUMANFunctionalcyanogen bromide, CNBr8.4Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42250CLONEDHUMAN125I-[Ile]MotilinK368,374C0.6Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42251CLONEDHUMANFunctionalK368,374C0.3Matsuura B, et al., 2005Jan 15, 2025Jan 15, 2025
42252CLONEDHUMANFunctional1-Cyclobutyl-1H-benzotriazole-5-carboxylic acid3090.3Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42253CLONEDHUMANFunctional1-Cyclopentyl-1H-benzotriazole-5-carboxylic acid1096.48Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42254CLONEDHUMANFunctional1-Cyclohexyl-1H-benzotriazole-5-carboxylic acid5888.44Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42255CLONEDHUMANFunctional1-Benzyl-1H-benzotriazole-5-carboxylic acid9120.11Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42256CLONEDHUMANFunctional1-Benzhydryl-1H-benzotriazole-5-carboxylic acid>10000Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42257CLONEDHUMANFunctional1-(3’-Methoxybenzyl)-1H-benzotriazole-5-carboxylic acid5011.87Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42258CLONEDHUMANFunctional1-(3’,5’-Difluorobenzyl)-1H-benzotriazole-5-carboxylic acid>10000Semple G, et al., 2006Jan 15, 2025Jan 15, 2025
42259CLONEDHUMAN125I-MotilinDelta 2-42.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42260CLONEDHUMAN125I-MotilinDelta 5-81.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42261CLONEDHUMAN125I-MotilinDelta 9-123.8Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42262CLONEDHUMAN125I-MotilinDelta 13-162.6Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42263CLONEDHUMAN125I-MotilinDelta 17-201.4Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42264CLONEDHUMAN125I-MotilinDelta 21-242.3Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42265CLONEDHUMAN125I-MotilinDelta 25C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42266CLONEDHUMAN125I-MotilinDelta 26-281.6Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42267CLONEDHUMAN125I-MotilinDelta 298.1Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42268CLONEDHUMAN125I-MotilinDelta 30C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42269CLONEDHUMAN125I-MotilinDelta 31-322Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42270CLONEDHUMAN125I-MotilinDelta 33-361000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42271CLONEDHUMAN125I-MotilinDelta 103-1041000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42272CLONEDHUMAN125I-MotilinDelta 105-1101000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42273CLONEDHUMAN125I-MotilinDelta 111C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42274CLONEDHUMAN125I-MotilinDelta 328-3306.3Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42275CLONEDHUMAN125I-MotilinDelta 331-3321000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42276CLONEDHUMAN125I-MotilinF33A7.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42277CLONEDHUMAN125I-MotilinP34A4.2Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42278CLONEDHUMAN125I-MotilinL35A3.7Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42279CLONEDHUMAN125I-MotilinG36A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42280CLONEDHUMAN125I-MotilinP103A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42281CLONEDHUMAN125I-MotilinW104A12.2Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42282CLONEDHUMAN125I-MotilinV105A1.8Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42283CLONEDHUMAN125I-MotilinF106A1.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42284CLONEDHUMAN125I-MotilinG107A1Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42285CLONEDHUMAN125I-MotilinP108A2Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42286CLONEDHUMAN125I-MotilinL109A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42287CLONEDHUMAN125I-MotilinL110A2.3Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42288CLONEDHUMAN125I-MotilinY331A2.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42289CLONEDHUMAN125I-MotilinF332A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42290CLONEDHUMANFunctionalDelta 2-44.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42291CLONEDHUMANFunctionalDelta 5-85.1Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42292CLONEDHUMANFunctionalDelta 9-124.2Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42293CLONEDHUMANFunctionalDelta 13-164.5Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42294CLONEDHUMANFunctionalDelta 17-204.5Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42295CLONEDHUMANFunctionalDelta 21-244Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42296CLONEDHUMANFunctionalDelta 25C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42297CLONEDHUMANFunctionalDelta 26-285.1Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42298CLONEDHUMANFunctionalDelta 294.2Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42299CLONEDHUMANFunctionalDelta 30C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42300CLONEDHUMANFunctionalDelta 31-323.7Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42301CLONEDHUMANFunctionalDelta 33-361000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42302CLONEDHUMANFunctionalDelta 103-1041000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42303CLONEDHUMANFunctionalDelta 105-1101000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42304CLONEDHUMANFunctionalDelta 111C1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42305CLONEDHUMANFunctionalDelta 328-3305.1Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42306CLONEDHUMANFunctionalDelta 331-3321000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42307CLONEDHUMANFunctionalF33A5.4Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42308CLONEDHUMANFunctionalP34A4.8Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42309CLONEDHUMANFunctionalL35A3.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42310CLONEDHUMANFunctionalG36A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42311CLONEDHUMANFunctionalP103A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42312CLONEDHUMANFunctionalW104A4.8Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42313CLONEDHUMANFunctionalV105A4.6Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42314CLONEDHUMANFunctionalF106A4.5Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42315CLONEDHUMANFunctionalG107A4.2Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42316CLONEDHUMANFunctionalP108A4.1Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42317CLONEDHUMANFunctionalL109A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42318CLONEDHUMANFunctionalL110A4.5Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42319CLONEDHUMANFunctionalY331A4.9Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42320CLONEDHUMANFunctionalF332A1000Matsuura B, et al., 2006Jan 15, 2025Jan 15, 2025
42321SLC6A3Striatal MembranesRAT3H-LBT-999GBR-129352.4Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42322SLC6A3Striatal MembranesRAT3H-LBT-999PE2I18Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42323SLC6A3Striatal MembranesRAT3H-LBT-999PAROXETINE1000Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42324SLC6A3Striatal MembranesRAT3H-LBT-999CITALOPRAM1000Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42325SLC6A3Striatal MembranesRAT3H-LBT-999MADAM1000Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42326SLC6A3Striatal MembranesRAT3H-LBT-999Nisoxetine1000Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42327SLC6A3Striatal MembranesRAT3H-LBT-999DESIPRAMINE1000Chalon S, et al., 2006Jan 15, 2025Jan 15, 2025
42328CLONEDHUMAN125I-MotilinMotilin2.81838Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42329CLONEDHUMAN125I-MotilinABT-22958.8844Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42330CLONEDHUMAN125I-Motilinerythromycin-A3090.3Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42331CLONEDHUMAN125I-MotilinME36>10000Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42332CLONEDHUMAN125I-MotilinME4537.032Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42333CLONEDHUMAN125I-MotilinEM-B enolether323.594Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42334CLONEDHUMAN125I-MotilinME523257.04Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42335CLONEDHUMAN125I-Motilin4'deoxy EM-A enolether69.1831Thielemans L, et al., 2005Jan 15, 2025Jan 15, 2025
42336Alpha2ACLONEDHUMAN35S-GTPGammaSA-54741245.471Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42337Alpha2ACLONEDHUMAN35S-GTPGammaSalpha-Methyl-(+/-)norepinephrine,(+/-)3630.78Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42338Alpha2ACLONEDHUMAN35S-GTPGammaSCLONIDINE61.6595Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42339Alpha2ACLONEDHUMAN35S-GTPGammaSDexmedetomidine13.1826Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42340Alpha2ACLONEDHUMAN35S-GTPGammaSEPINEPHRINE1479.11Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42341Alpha2ACLONEDHUMAN35S-GTPGammaSGuanabenz21.8776Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42342Alpha2ACLONEDHUMAN35S-GTPGammaSGuanfacine93.3254Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42343Alpha2ACLONEDHUMAN35S-GTPGammaSLevlofexidine14.4544Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42344Alpha2ACLONEDHUMAN35S-GTPGammaSNaphazoline20.893Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42345Alpha2ACLONEDHUMAN35S-GTPGammaSNaphthalene4.57088Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42346Alpha2ACLONEDHUMAN35S-GTPGammaSNOREPINEPHRINE1995.26Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42347Alpha2ACLONEDHUMAN35S-GTPGammaSOXYMETAZOLINE7.24436Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42348Alpha2ACLONEDHUMAN35S-GTPGammaSp-AMINOCLONIDINE7.94328Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42349Alpha2ACLONEDHUMAN35S-GTPGammaSST-91575.44Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42350Alpha2ACLONEDHUMAN35S-GTPGammaSTramazoline31.6228Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42351Alpha2ACLONEDHUMAN35S-GTPGammaSUK-14,304213.796Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42352Alpha2ACLONEDHUMAN35S-GTPGammaSXylazine5754.4Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42353Alpha2ACLONEDHUMAN35S-GTPGammaSXylometazoline15.1356Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42354Alpha2ACLONEDHUMAN35S-GTPGammaSAlinidine6025.6Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42355Alpha2ACLONEDHUMAN35S-GTPGammaSB-HT 920398.107Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42356Alpha2ACLONEDHUMAN35S-GTPGammaSIDAZOXAN9.77237Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42357Alpha2ACLONEDHUMAN35S-GTPGammaSICI 1062707.94328Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42358Alpha2ACLONEDHUMAN35S-GTPGammaSIMILOXAN316.228Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42359Alpha2ACLONEDHUMAN35S-GTPGammaSMK-9120.851138Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42360Alpha2ACLONEDHUMAN35S-GTPGammaSPHENTOLAMINE20.4174Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42361Alpha2ACLONEDHUMAN35S-GTPGammaSPRAZOSIN794.328Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42362Alpha2ACLONEDHUMAN35S-GTPGammaSRAUWOLSCINE1.20226Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42363Alpha2ACLONEDHUMAN35S-GTPGammaSRilmenidine1584.89Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42364Alpha2ACLONEDHUMAN35S-GTPGammaSRX8210020.363078Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42365Alpha2ACLONEDHUMAN35S-GTPGammaSTOLAZOLINE229.087Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42366Alpha2ACLONEDMOUSE35S-GTPGammaSEPINEPHRINE389.045Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42367Alpha2ACLONEDMOUSE35S-GTPGammaSNOREPINEPHRINE1412.54Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42368Alpha2ACLONEDMOUSE35S-GTPGammaSIsoproterenol>10000Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42369Alpha2ACLONEDMOUSE35S-GTPGammaSA-547419.77237Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42370Alpha2ACLONEDMOUSE35S-GTPGammaSUK-14,30443.6516Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42371Alpha2ACLONEDMOUSE35S-GTPGammaSDexmedetomidine3.38844Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42372Alpha2ACLONEDMOUSE35S-GTPGammaSST-91537.032Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42373Alpha2ACLONEDMOUSE35S-GTPGammaSGuanfacine20.4174Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42374Alpha2ACLONEDMOUSE35S-GTPGammaSXylazine2398.83Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42375Alpha2ACLONEDMOUSE35S-GTPGammaSRilmenidine724.436Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42376Alpha2ACLONEDMOUSE35S-GTPGammaSCLONIDINE40.738Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42377Alpha2ACLONEDMOUSE35S-GTPGammaSOXYMETAZOLINE15.4882Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42378Alpha2ACLONEDMOUSE35S-GTPGammaSTramazoline15.4882Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42379Alpha2ACLONEDMOUSE35S-GTPGammaSNaphthalene7.76247Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42380Alpha2ACLONEDMOUSE35S-GTPGammaSNaphazoline11.4815Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42381Alpha2ACLONEDMOUSE35S-GTPGammaSXylometazoline25.704Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42382Alpha2ACLONEDMOUSE35S-GTPGammaSRX8210020.616595Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42383Alpha2ACLONEDMOUSE35S-GTPGammaSNaphthalene9.33254Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42384Alpha2ACLONEDMOUSE35S-GTPGammaSNaphazoline16.9824Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42385Alpha2ACLONEDMOUSE35S-GTPGammaSXylometazoline23.9883Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42386Alpha2ACLONEDMOUSE35S-GTPGammaSOXYMETAZOLINE25.704Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42387Alpha2ACLONEDMOUSE35S-GTPGammaSRAUWOLSCINE36.3078Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42388Alpha2ACLONEDMOUSE35S-GTPGammaSYOHIMBINE61.6595Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42389Alpha2ACLONEDMOUSE35S-GTPGammaSCLONIDINE61.6595Jasper JR, et al., 1998Jan 15, 2025Jan 15, 2025
42390ß-AmyloidBRAINHUMAN125I-IMPY4-Amino-4'-hydroxystilbene95Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42391ß-AmyloidBRAINHUMAN125I-IMPY3-{4-[2-(4-Aminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol15Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42392ß-AmyloidBRAINHUMAN125I-IMPY4-N,N'-Dimethylamino-4'-hydroxystilbene1.1Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42393ß-AmyloidBRAINHUMAN125I-IMPY(4-{2-[4-(2,2-Dimethyl-[1,3]dioxan-5-ylmethoxy)phenyl]vinyl}phenyl)dimethylamine59Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42394ß-AmyloidBRAINHUMAN125I-IMPY2-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol38Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42395ß-AmyloidBRAINHUMAN125I-IMPYToluene-4-sulfonic Acid 3-{4-[2-(4-(Dimethylamino)phenyl)vinyl]phenoxy}-2-hydroxymethylpropyl Ester150Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42396ß-AmyloidBRAINHUMAN125I-IMPY3-{4-[2-(4-Dimethylaminophenyl)vinyl]phenoxy}-2-fluoromethylpropan-1-ol15Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42397ß-AmyloidBRAINHUMAN125I-IMPY2-(4-Bromobenzyl)-3-{4-[2-(4-(dimethylamino)phenyl)vinyl]phenoxy}propan-1-ol80Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42398ß-AmyloidBRAINHUMAN125I-IMPY4-N-Methylamino-4'-hydroxystilbene, SB-131.2Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42399ß-AmyloidBRAINHUMAN125I-IMPY2-{4-[2-(4-Methylaminophenyl)vinyl]phenoxymethyl}propane-1,3-diol32.5Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42400ß-AmyloidBRAINHUMAN125I-IMPY2-Fluoromethyl-3-{4-[2-(4-methylaminophenyl)vinyl]phenoxy}propan-1-ol5Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42401ß-AmyloidBRAINHUMAN125I-IMPYPIB2.8Zhang W, et al., 2005Jan 15, 2025Jan 15, 2025
42402PLCbladderRATFunctionalET-18-OCH35000Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42403PLCbladderRATFunctionalNeomycin5000Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42404PLCbladderRATFunctionalD609>10000Braverman AS, et al., 2006Jan 15, 2025Jan 28, 2025
42405PLCbladderRATFunctionalNeomycin5000Braverman AS, et al., 2006Jan 15, 2025Jan 28, 2025
42406PAKbladderRATFunctional(R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride>10000Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42407PAKbladderRATFunctionalHA-10771600Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42408PAKbladderRATFunctionalH73000Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42409PAKbladderRATFunctionalH8950Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42410PKGbladderRATFunctionalHA-10771600Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42411PKGbladderRATFunctionalH75800Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42412PKGbladderRATFunctionalH89500Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42413PKCbladderRATFunctional(R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride>10000Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42414PKCbladderRATFunctionalChelerytherine660Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42415PKCbladderRATFunctionalH76000Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42416Rho KinasebladderRATFunctional(R)-(+)-trans-4-(1-aminoethyl)-N-(4-pyridyl)cyclohexanecarboxamide dihydrochloride100Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42417Rho KinasebladderRATFunctionalHA-1077330Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42418Rho KinasebladderRATFunctionalH7450Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42419Rho KinasebladderRATFunctionalH89270Braverman AS, et al., 2006Jan 15, 2025Jan 15, 2025
42420GABAAWHOLE BRAINRATFNZ1-Phenyl-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one6280Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42421GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one 4350Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42422GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one1040Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42423GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-1,5-dihydro-imidazol-2-one4290Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42424GABAAWHOLE BRAINRATFNZ1-(4-Bromophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one3060Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42425GABAAWHOLE BRAINRATFNZ1-(4-Iodophenyl)-4-morpholin-4-yl-1,5-dihydro-imidazol-2-one3320Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42426GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-azepan-1-yl-1,5-dihydro-imidazol-2-one>10000Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42427GABAAWHOLE BRAINRATFNZ1-(4-Methoxyphenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-one938Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42428GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one141Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42429GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-pyrrolidin-1-yl-2,4-dihydro-pyrrol-2-one67Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42430GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-azepan-1-yl-2,4-dihydro-pyrrol-2-one440Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42431GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-4-piperidin-1-yl-2,4-dihydro-pyrrol-2-one90Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42432GABAAWHOLE BRAINRATFNZ1-(4-Fluorophenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one494Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42433GABAAWHOLE BRAINRATFNZ1-(3-Methylphenyl)-4-morpholin-1-yl-2,4-dihydro-pyrrol-2-one4450Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42434GABAAWHOLE BRAINRATFNZ1-(4-Methylphenyl)-4-morpholin-4-yl-2,4-dihydro-pyrrol-2-one344Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42435GABAAWHOLE BRAINRATFNZ1-(3-Chloro-4-fluorophenyl)-4-(morpholin-4-yl)-1,5-dihydro-pyrrole-2-one2050Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42436GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione4340Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42437GABAAWHOLE BRAINRATFNZ1-(4-Chlorophenyl)-3-pyrrolidin-1-yl-pyrrole-2,5-dione3260Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42438GABAAWHOLE BRAINRATFNZ1-(4-Fluorophenyl)-3-piperidin-1-yl-pyrrole-2,5-dione5410Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42439GABAAWHOLE BRAINRATFNZ4-(4-Chlorophenyl)-1-pyrid-2-yl-pyrazole4480Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42440GABAAWHOLE BRAINRATFNZ3-(4-Chlorophenyl)-5-morpholin-4-yl-1,2,4-oxadiazole>10000Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42441GABAAWHOLE BRAINRATFNZ2-(4-Chlorophenyl)-5-phenyl-4-isoxazolin-3-one1120Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42442GABAAWHOLE BRAINRATFNZCGS 98962.4Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42443GABAAWHOLE BRAINRATFNZDIAZEPAM6.8Grunwald C, et al., 2006Jan 15, 2025Jan 15, 2025
42444D1CLONEDHUMAN3H-SCH23390LE3001.9Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42445D2CLONEDHUMAN3H-SPIPERONELE30044.7Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42446D5CLONEDHUMAN3H-SCH23390LE3007.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42447D1CLONEDHUMAN3H-SCH233903-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine0.39Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42448D2CLONEDHUMAN3H-SPIPERONE3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine17.5Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42449D3CLONEDHUMAN3H-SPIPERONE3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine47.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42450D5CLONEDHUMAN3H-SCH233903-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine1.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42451D1CLONEDHUMAN3H-SCH233903-methoxy-dibenz[d,g]azecine28.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42452D2CLONEDHUMAN3H-SPIPERONE3-methoxy-dibenz[d,g]azecine13Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42453D3CLONEDHUMAN3H-SPIPERONE3-methoxy-dibenz[d,g]azecine75.7Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42454D1CLONEDHUMAN3H-SCH233904-chloro-3-hydroxy-dibenz[d,g]azecine0.83Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42455D2CLONEDHUMAN3H-SPIPERONE4-chloro-3-hydroxy-dibenz[d,g]azecine4Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42456D3CLONEDHUMAN3H-SPIPERONE4-chloro-3-hydroxy-dibenz[d,g]azecine24.6Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42457D5CLONEDHUMAN3H-SCH233904-chloro-3-hydroxy-dibenz[d,g]azecine0.057Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42458D1CLONEDHUMAN3H-SCH233902,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine3.2Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42459D2CLONEDHUMAN3H-SPIPERONE2,4-dichloro-3-hydroxy-7-methyl-5,6,7,8,9,14-dibenz[d,g]azecine88Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42460D1CLONEDHUMAN3H-SCH233902-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine9.3Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42461D2CLONEDHUMAN3H-SPIPERONE2-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine37.3Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42462D5CLONEDHUMAN3H-SCH233902-Amino-3-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine226.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42463D1CLONEDHUMAN3H-SCH233902-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine8.9Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42464D2CLONEDHUMAN3H-SPIPERONE2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine36.9Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42465D3CLONEDHUMAN3H-SPIPERONE2-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine296Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42466D5CLONEDHUMAN3H-SCH233902-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine42.3Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42467D1CLONEDHUMAN3H-SCH233902-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine82Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42468D2CLONEDHUMAN3H-SPIPERONE2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine62Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42469D3CLONEDHUMAN3H-SPIPERONE2-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenz[d,g]azecine150.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42470D1CLONEDHUMAN3H-SCH233901,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine25.3Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42471D2CLONEDHUMAN3H-SPIPERONE1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine210Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42472D3CLONEDHUMAN3H-SPIPERONE1,3-Dichloro-2-methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine415Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42473D1CLONEDHUMAN3H-SCH233901-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine0.46Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42474D2CLONEDHUMAN3H-SPIPERONE1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine0.99Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42475D3CLONEDHUMAN3H-SPIPERONE1-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine1.88Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42476D5CLONEDHUMAN3H-SCH233901-Chloro-2-hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine0.98Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42477D1CLONEDHUMAN3H-SCH233903-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine3.1Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42478D2CLONEDHUMAN3H-SPIPERONE3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine2Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42479D3CLONEDHUMAN3H-SPIPERONE3-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine27.7Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42480D5CLONEDHUMAN3H-SCH233903-Chloro-2-hydroxy- 7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine4.9Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42481D1CLONEDHUMAN3H-SCH233901-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine8.7Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42482D2CLONEDHUMAN3H-SPIPERONE1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine84Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42483D3CLONEDHUMAN3H-SPIPERONE1-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine215Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42484D1CLONEDHUMAN3H-SCH233904-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine7.6Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42485D2CLONEDHUMAN3H-SPIPERONE4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine164Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42486D3CLONEDHUMAN3H-SPIPERONE4-Chloro-1-Methoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine1833Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42487D1CLONEDHUMAN3H-SCH233903,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine2Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42488D2CLONEDHUMAN3H-SPIPERONE3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine58.7Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42489D3CLONEDHUMAN3H-SPIPERONE3,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine342Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42490D5CLONEDHUMAN3H-SCH233903,11-Hydroxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine1.68Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42491D1CLONEDHUMAN3H-SCH233903,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine9.4Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42492D2CLONEDHUMAN3H-SPIPERONE3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine6.5Mohr P, et al., 2006Jan 15, 2025Jan 27, 2025
42493D3CLONEDHUMAN3H-SPIPERONE3,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine101.5Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42494D5CLONEDHUMAN3H-SCH233903,11- Dimethoxy-7-methyl-5,6,7,8,9,14-hexahydrodibenzo[d,g]azecine12.6Mohr P, et al., 2006Jan 15, 2025Jan 15, 2025
42495MEKUNDEFINEDUNDEFINEDFunctional4-(4-bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide39Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42496MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(cyclopropylmethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide124Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42497MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-5-fluoro-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide6.8Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42498MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-N-(cyclopropylmethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide40Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42499MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide30Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42500MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide45Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42501MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-5-fluoro-N-(2-hydroxyethoxy)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide9.3Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42502MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-fluorophenylamino)-N-(2-hydroxyethoxy)-1,5-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide18Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42503MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-chlorophenylamino)-5-chloro-N-(2-hydroxyethoxy)-6-methoxynicotinamide6786Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42504MEKUNDEFINEDUNDEFINEDFunctional4-(4-Bromo-2-chlorophenylamino)-5,6-dichloro-N-(2-hydroxyethoxy)nicotinamide4496Wallace EM, et al., 2006Jan 15, 2025Jan 15, 2025
42505CLONEDRABBITUNDEFINEDMotilin0.977237Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42506CLONEDRABBITUNDEFINED[Nle13]-Motilin0.851138Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42507CLONEDRABBITUNDEFINEDerythromycin-A190.546Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42508CLONEDRABBIT35S-GTPGammaSMotilin1.34896Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42509CLONEDRABBIT35S-GTPGammaS[Nle13]-Motilin1.69824Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42510CLONEDRABBIT35S-GTPGammaSerythromycin-A741.31Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42511CLONEDHUMANUNDEFINEDMotilin0.162181Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42512CLONEDHUMANUNDEFINED[Nle13]-Motilin0.436516Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42513CLONEDHUMANUNDEFINEDerythromycin-A512.861Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42514CLONEDHUMAN35S-GTPGammaSMotilin1.28825Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42515CLONEDHUMAN35S-GTPGammaS[Nle13]-Motilin1.94984Dass NB, et al., 2003Jan 15, 2025Jan 15, 2025
42516CLONEDHUMANFunctional[leu13]pMOT(1-5)8912.51Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42517CLONEDHUMANFunctional[leu13]pMOT(1-7)6918.31Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42518CLONEDHUMANFunctional[leu13]pMOT(1-9)4073.8Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42519CLONEDHUMANFunctional[leu13]pMOT(1-11)89.1251Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42520CLONEDHUMANFunctional[leu13]pMOT(1-14)3.16228Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42521CLONEDHUMANFunctional[leu13]pMOT(1-16)2.13796Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42522CLONEDHUMANFunctional[leu13]pMOT(1-19)0.977237Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42523CLONEDHUMANFunctional[leu13]pMOT(1-22)1Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42524CLONEDHUMANFunctional[ala1,leu13]pMOT(1-14)588.844Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42525CLONEDHUMANFunctional[ala3,leu13]pMOT(1-14)1.31826Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42526CLONEDHUMANFunctional[ala4,leu13]pMOT(1-14)2570.4Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42527CLONEDHUMANFunctional[ala5,leu13]pMOT(1-14)28.8403Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42528CLONEDHUMANFunctional[ala6,leu13]pMOT(1-14)46.7735Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42529CLONEDHUMANFunctional[ala7,leu13]pMOT(1-14)1445.44Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42530CLONEDHUMANFunctional[ala8,leu13]pMOT(1-14)36.3078Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42531CLONEDHUMANFunctional[ala9,leu13]pMOT(1-14)75.8578Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42532CLONEDHUMANFunctional[ala10,leu13]pMOT(1-14)5.01187Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42533CLONEDHUMANFunctional[ala11,leu13]pMOT(1-14)4.57088Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42534CLONEDHUMANFunctional[ala12,leu13]pMOT(1-14)6.30957Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42535CLONEDHUMANFunctional[ala13,leu13]pMOT(1-14)7.24436Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42536CLONEDHUMANFunctional[ala14,leu13]pMOT(1-14)7.07946Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42537CLONEDHUMANFunctionalerythromycin-A77.6247Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42538CLONEDHUMANFunctionalN-ethyl, N-Methyl Erythromycin-A239.883Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42539CLONEDHUMANFunctionalErythromycin-A enol ether8.31764Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42540CLONEDHUMANFunctionalErythromycin-B144.544Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42541CLONEDHUMANFunctionalErythromycin-B enol ether7.58578Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42542CLONEDHUMANFunctionalN-ethyl, N-methyl Erythromycin-A enol ether6.0256Thielemans L, et al., 2002Jan 15, 2025Jan 15, 2025
42543UNDEFINEDUNDEFINEDFunctionalLY-36494759Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42544UNDEFINEDUNDEFINEDFunctional5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42545UNDEFINEDUNDEFINEDFunctional1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole4100Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42546UNDEFINEDUNDEFINEDFunctional1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42547UNDEFINEDUNDEFINEDFunctional6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole47Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42548UNDEFINEDUNDEFINEDFunctional6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole68Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42549UNDEFINEDUNDEFINEDFunctionalLY-364947400Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42550UNDEFINEDUNDEFINEDFunctional5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42551UNDEFINEDUNDEFINEDFunctional1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42552UNDEFINEDUNDEFINEDFunctional1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42553UNDEFINEDUNDEFINEDFunctional6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole1300Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42554UNDEFINEDUNDEFINEDFunctional6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole409Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42555UNDEFINEDUNDEFINEDFunctionalLY-3649471400Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42556UNDEFINEDUNDEFINEDFunctional5-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42557UNDEFINEDUNDEFINEDFunctional1-Methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42558UNDEFINEDUNDEFINEDFunctional1-Methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42559UNDEFINEDUNDEFINEDFunctional6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole>10000Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42560UNDEFINEDUNDEFINEDFunctional6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole9450Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42561UNDEFINEDUNDEFINEDFunctionalLY-36494740Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42562UNDEFINEDUNDEFINEDFunctional6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole15Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42563UNDEFINEDUNDEFINEDFunctional6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole57Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42564UNDEFINEDUNDEFINEDFunctionalLY-36494781Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42565UNDEFINEDUNDEFINEDFunctional6-[2-(6-Methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-benzoimidazole42Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42566UNDEFINEDUNDEFINEDFunctional6-(2-Pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole118Li HY, et al., 2006Jan 15, 2025Jan 15, 2025
42567Alpha1ACLONEDUNDEFINEDUNDEFINEDPRAZOSIN0.2Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42568Alpha1ACLONEDUNDEFINEDUNDEFINEDTerazosin6.3Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42569Alpha1ACLONEDUNDEFINEDUNDEFINEDDoxazosin3.16Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42570Alpha1ACLONEDUNDEFINEDUNDEFINEDAlfuzosin10Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42571Alpha1ACLONEDUNDEFINEDUNDEFINEDUrapidil-5-methyl0.63Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42572Alpha1ACLONEDUNDEFINEDUNDEFINEDRS-1009751Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42573Alpha1ACLONEDUNDEFINEDUNDEFINEDWB 41010.16Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42574Alpha1ACLONEDUNDEFINEDUNDEFINEDRS-170530.6Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42575Alpha1BCLONEDUNDEFINEDUNDEFINEDPRAZOSIN0.25Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42576Alpha1BCLONEDUNDEFINEDUNDEFINEDTerazosin2Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42577Alpha1BCLONEDUNDEFINEDUNDEFINEDDoxazosin1Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42578Alpha1BCLONEDUNDEFINEDUNDEFINEDAlfuzosin10Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42579Alpha1BCLONEDUNDEFINEDUNDEFINEDUrapidil-5-methyl40Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42580Alpha1BCLONEDUNDEFINEDUNDEFINEDRS-10097579Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42581Alpha1BCLONEDUNDEFINEDUNDEFINEDWB 41012.5Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42582Alpha1BCLONEDUNDEFINEDUNDEFINEDRS-1705316Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42583Alpha1CCLONEDUNDEFINEDUNDEFINEDPRAZOSIN0.32Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42584Alpha1CCLONEDUNDEFINEDUNDEFINEDTerazosin2.5Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42585Alpha1CCLONEDUNDEFINEDUNDEFINEDDoxazosin4Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42586Alpha1CCLONEDUNDEFINEDUNDEFINEDAlfuzosin3.16Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42587Alpha1CCLONEDUNDEFINEDUNDEFINEDUrapidil-5-methyl10Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42588Alpha1CCLONEDUNDEFINEDUNDEFINEDRS-100975100Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42589Alpha1CCLONEDUNDEFINEDUNDEFINEDWB 41010.25Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42590Alpha1CCLONEDUNDEFINEDUNDEFINEDRS-1705316Kinsella GK, et al., 2006Jan 15, 2025Jan 15, 2025
42591CLONEDHUMANFunctional2-amino-4-oxo-6-methyl-5-substituted pyrrolo[2,3-d]pyrimidine54Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42592CLONEDHUMANFunctional2-Amino-6-methyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine150Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42593CLONEDHUMANFunctionalN-[4-[(2-amino-6-ethyl-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidin-5-yl)thio]benzoyl]-L-glutamic acid90Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42594CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(3',4'-dichlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine230Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42595CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine240Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42596CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-fluorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine2700Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42597CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine3.1E-5Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42598CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine1000Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42599CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine>10000Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42600CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(3'-chlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine2600Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42601CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(3'-bromophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]p-yrimidine1100Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42602CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(3'-methoxyphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine3.2E-5Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42603CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(3',5'-trifluoromethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine2.2E-5Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42604CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(2',6'-dimethylphenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine>10000Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42605CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(1'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine5600Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42606CLONEDHUMANFunctional2-Amino-6-ethyl-5-[(2'-naphthyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine5600Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42607CLONEDHUMANFunctionalPDDF72Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42608CLONEDHUMANFunctionalraltitrexed380Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42609CLONEDHUMANFunctionalPemetrexed9500Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42610DHFRCLONEDHUMANFunctional2-amino-4-oxo-6-methyl-5-substituted pyrrolo[2,3-d]pyrimidine2100Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42611DHFRCLONEDHUMANFunctionalN-[4-[(2-amino-6-ethyl-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidin-5-yl)thio]benzoyl]-L-glutamic acid420Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42612DHFRCLONEDHUMANFunctional2-Amino-6-ethyl-5-[(3',4'-dichlorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine>10000Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42613DHFRCLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-nitrophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine>10000Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025
42614DHFRCLONEDHUMANFunctional2-Amino-6-ethyl-5-[(4'-fluorophenyl)sulfanyl]-3,4-dihydro-4-oxo-7H-pyrrolo[2,3-d]pyrimidine>10000Gangjee A, et al., 2006Jan 15, 2025Jan 15, 2025