The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 52,001-53,000 of 98,685 items.

Kᵢ Database

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Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
54749SLC6A4UNDEFINEDHUMANUNDEFINED2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)acetamide5977Strappaghetti G et al., 2008Jan 15, 2025Jan 15, 2025
54750SLC6A4UNDEFINEDHUMANUNDEFINED2-(3-(1H-imidazol-1-yl)-6-oxopyridazin-1(6H)-yl)-N-(2-(4-(2-isopropoxyphenyl)piperazin-1-yl)ethyl)acetamide1000Strappaghetti G et al., 2008Jan 15, 2025Jan 15, 2025
54751SLC6A4UNDEFINEDHUMANUNDEFINEDPAROXETINE0.08Strappaghetti G et al., 2008Jan 15, 2025Jan 15, 2025
547525-HT2AUNDEFINEDUNDEFINEDUNDEFINED6-(1H-indol-1-yl)-2-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one83Strappaghetti G et al., 2008Jan 15, 2025Jan 15, 2025
547535-HT2AUNDEFINEDUNDEFINEDUNDEFINED6-(1H-imidazol-1-yl)-2-(4-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)butyl)pyridazin-3(2H)-one166Strappaghetti G et al., 2008Jan 15, 2025Jan 15, 2025
54754MT2UNDEFINEDHUMANUNDEFINEDMELATONIN0.41Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54755MT2UNDEFINEDHUMANUNDEFINEDS 200980.27Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54756MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-phenyl-7-methoxynaphth-1-yl)ethyl] acetamide0.37Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54757MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(2-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide1.86Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54758MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl] acetamide0.36Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54759MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(4-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide23Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54760MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]propionamide0.52Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54761MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]butyramide0.28Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54762MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Hydroxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]cyclobutyl carboxamide48.3Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54763MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Methoxymethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.95Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54764MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Formylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.42Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54765MT2UNDEFINEDHUMANUNDEFINED3-[4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl]benzoic acid methyl ester0.64Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54766MT2UNDEFINEDHUMANUNDEFINED3-(4-(2-Acetylaminoethyl)-6-methoxynaphth-2-yl)benzoic acid43.3Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54767MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Bromomethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.56Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54768MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Iodomethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.71Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54769MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Aminomethylphenyl)-7-methoxynaphth-1-yl)ethyl]acetamide3.4Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54770MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Aminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.27Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54771MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Methylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.51Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54772MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Dimethylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide0.94Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54773MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Ethoxycarbonylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide8.3Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54774MT2UNDEFINEDHUMANUNDEFINEDN-[2-(3-(3-Acetylaminophenyl)-7-methoxynaphth-1-yl)ethyl]acetamide7.54Poissonnier-Durieux S et al., 2008Jan 15, 2025Jan 15, 2025
54775D2UNDEFINEDHUMANUNDEFINED1-(2,4-Dimethyl-phenyl)-4-(2-phenyl-cyclopropylmethyl)-piperazine; hydrobromide540Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54776D2UNDEFINEDHUMANUNDEFINEDHALOPERIDOL5.09Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54777D2UNDEFINEDHUMANUNDEFINED(1S,2S)-1-[(S)-2-[4-(2,4-Dimethylphenyl)piperazyl]-ethyl]-2-methyl-2-phenylcyclopropane>10000Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54778D2UNDEFINEDHUMANUNDEFINED(1S,2S)-1-[(R)-2-[4-(2,4-Dimethylphenyl)piperazyl]-ethyl]-2-methyl-2-phenylcyclopropane>10000Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54779D2UNDEFINEDHUMANUNDEFINED(1S,2S)-1-[4-(2,4-Dimethylphenyl)piperazyl]methyl-2-methyl-2-phenylcyclopropane>10000Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54780D2UNDEFINEDHUMANUNDEFINED1-(2,4-dimethylphenyl)-4-(((1R,2S)-2-phenylcyclopropyl)methyl)piperazine515Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54781D2UNDEFINEDHUMANUNDEFINED1-(2,4-dimethylphenyl)-4-(((1S,2R)-2-phenylcyclopropyl)methyl)piperazine935Yamaguchi K et al., 2008Jan 15, 2025Jan 15, 2025
54782D2UNDEFINEDHUMANUNDEFINEDDOPAMINE450Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54783D2UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide220Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54784D2UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide5500Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54785D2UNDEFINEDHUMANUNDEFINEDN-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide40Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54786D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine690Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54787D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine210Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54788D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine610Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54789D2UNDEFINEDHUMANUNDEFINEDN-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine4100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54790D2UNDEFINEDHUMANUNDEFINEDN-(4-Propylaminobutyl)-4-biphenylcarboxamide>10000Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54791D2UNDEFINEDHUMANUNDEFINEDN-(4-Dipropylaminobutyl)-4-biphenylcarboxamide9700Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54792D2UNDEFINEDHUMANUNDEFINEDN-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide4700Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54793D2UNDEFINEDHUMANUNDEFINEDDOPAMINE360Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54794D2UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide360Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54795D2UNDEFINEDHUMANUNDEFINEDN-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide43Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54796D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine670Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54797D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine180Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54798D2UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine170Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54799D2UNDEFINEDHUMANUNDEFINEDN-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine2100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54800D2UNDEFINEDHUMANUNDEFINEDN-(4-Propylaminobutyl)-4-biphenylcarboxamide>10000Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54801D2UNDEFINEDHUMANUNDEFINEDN-(4-Dipropylaminobutyl)-4-biphenylcarboxamide8800Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54802D2UNDEFINEDHUMANUNDEFINEDN-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide6300Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54803D2UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide4700Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54804D3UNDEFINEDHUMANUNDEFINEDDOPAMINE240Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54805D3UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide4.4Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54806D3UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide300Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54807D3UNDEFINEDHUMANUNDEFINEDN-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide0.21Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54808D3UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine13Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54809D3UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine150Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54810D3UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine1.3Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54811D3UNDEFINEDHUMANUNDEFINEDN-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine280Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54812D3UNDEFINEDHUMANUNDEFINEDN-(4-Propylaminobutyl)-4-biphenylcarboxamide>10000Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54813D3UNDEFINEDHUMANUNDEFINEDN-(4-Dipropylaminobutyl)-4-biphenylcarboxamide950Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54814D3UNDEFINEDHUMANUNDEFINEDN-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide140Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54815D3UNDEFINEDHUMANUNDEFINEDBiphenyl-4-carboxylic acid {4-[(5-hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amino]-butyl}-amide0.2Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54816D4UNDEFINEDHUMANUNDEFINEDDOPAMINE6.2Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54817D4UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide69Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54818D4UNDEFINEDHUMANUNDEFINEDN-[N'-Propyl-N'-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]-4-aminobutyl]-4-biphenylcarboxamide3100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54819D4UNDEFINEDHUMANUNDEFINEDN-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide4.3Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54820D4UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-trimethylsilylethynyl)cyclohex-3-en-1-yl]amine1800Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54821D4UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-[4-(2-phenylethynyl)cyclohex-3-en-1-yl]amine1100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54822D4UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine190Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54823D4UNDEFINEDHUMANUNDEFINEDN-[4-(4-Methyltriazol-1-yl)butyl]-N-propyl-N-(4-propyn-1-ylcyclohex-3-en-1-yl)amine100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54824D4UNDEFINEDHUMANUNDEFINEDN-(4-Propylaminobutyl)-4-biphenylcarboxamide6100Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54825D4UNDEFINEDHUMANUNDEFINEDN-(4-Dipropylaminobutyl)-4-biphenylcarboxamide1400Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54826D4UNDEFINEDHUMANUNDEFINEDN-[(N'-(4-Cyclohexyl)-N'-propyl)aminobutyl]-4-biphenylcarboxamide670Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54827D3UNDEFINEDHUMANUNDEFINEDDOPAMINE72Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54828D3UNDEFINEDHUMANUNDEFINEDN-[N'-(4-Ethynylcyclohex-3-en-1-yl)-N'-propyl-4-aminobutyl]-4-biphenylcarboxamide0.78Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54829D3UNDEFINEDHUMANUNDEFINEDN-[4-[4-(4-Biphenyl)triazol-1-yl]butyl]-N-propyl-N-(4-ethynylcyclohex-3-en-1-yl)amine2.5Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54830D3UNDEFINEDHUMANUNDEFINED(4-Ethynyl-cyclohex-3-enyl)-dipropyl-amine190Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54831D3UNDEFINEDHUMANUNDEFINED7-OH-DPAT3.6Dörfler M et al., 2008Jan 15, 2025Jan 15, 2025
54832SLC6A4UNDEFINEDRATUNDEFINEDrac-[3-(5-fluoro-1H-indol-3-yl)-propyl]-(5-methoxy-chroman-3-yl)-propyl-amine9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54833SLC6A4UNDEFINEDRATUNDEFINED8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine12.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54834SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine17.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54835SLC6A4UNDEFINEDRATUNDEFINED(3S)-(+)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine13.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54836SLC6A4UNDEFINEDRATUNDEFINEDrac-8-fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide7.1Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54837SLC6A4UNDEFINEDRATUNDEFINED(R)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide8Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54838SLC6A4UNDEFINEDRATUNDEFINED(S)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide4.7Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54839SLC6A4UNDEFINEDRATUNDEFINED8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}-N-methylchromane-5-carboxamide2.4Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54840SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)-amino}-N-methylchromane-5-carboxamide11.3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54841SLC6A4UNDEFINEDRATUNDEFINED3-{[3-(5-Fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide23.4Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54842SLC6A4UNDEFINEDRATUNDEFINEDFLUOXETINE3.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54843SLC6A4UNDEFINEDRATUNDEFINEDrac-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine13Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54844SLC6A4UNDEFINEDRATUNDEFINED(3R)-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-3,4-dihydro-2H-chromen-41.4Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54845SLC6A4UNDEFINEDRATUNDEFINEDrac-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54846SLC6A4UNDEFINEDRATUNDEFINED(3R)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide1.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54847SLC6A4UNDEFINEDRATUNDEFINED8-Chloro-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-chromane-5-carboxamide3.74Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54848SLC6A4UNDEFINEDRATUNDEFINED8-Chloro-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-chromane-5-carboxamide1.98Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54849SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide9.55Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54850SLC6A4UNDEFINEDRATUNDEFINED(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54851SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide7.2Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54852SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide8.3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54853SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide10.2Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54854SLC6A4UNDEFINEDRATUNDEFINEDMethyl-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxylate161Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54855SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxylic Acid498.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54856SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-ethyl-8-fluorochromane-5-carboxamide9.47Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54857SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-propylchromane-5-carboxamide7.96Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54858SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-isopropylchromane-5-carboxamide11.28Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54859SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopropyl-8-fluorochromane-5-carboxamide8.05Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54860SLC6A4UNDEFINEDRATUNDEFINEDN-Cyclobutyl-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]-amino}-8-fluorochromane-5-carboxamide7.26Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54861SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopentyl-8-fluorochromane-5-carboxamide19.8Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54862SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-(cyclopropylmethyl)-8-fluorochromane-5-carboxamide6.91Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54863SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N,N-dimethylchromane-5-carboxamide28.8Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54864SLC6A4UNDEFINEDRATUNDEFINED(3S)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide5.3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54865SLC6A4UNDEFINEDRATUNDEFINED(-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide2.44Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54866SLC6A4UNDEFINEDRATUNDEFINED(-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide9.05Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54867SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(5-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide1000Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54868SLC6A4UNDEFINEDRATUNDEFINED3-[[3-(5-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide75.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54869SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(6-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide237.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54870SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[3-(7-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide1000Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54871SLC6A4UNDEFINEDRATUNDEFINED3-[[3-(7-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide66Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54872SLC6A4UNDEFINEDRATUNDEFINED(-)-3-{Cyclobutyl[3-(5,7-difluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide3.34Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54873SLC6A4UNDEFINEDRATUNDEFINED(-)-3-{Cyclobutyl[3-(5,7-difluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide12.15Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54874SLC6A4UNDEFINEDRATUNDEFINED8-Fluoro-3-[[4-(4-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide210.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54875SLC6A4UNDEFINEDRATUNDEFINED8-Fluoro-3-[[4-(5-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide114Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54876SLC6A4UNDEFINEDRATUNDEFINED8-Fluoro-3-[[4-(6-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide70Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54877SLC6A4UNDEFINEDRATUNDEFINED8-Fluoro-3-[[4-(7-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide32.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54878SLC6A4UNDEFINEDRATUNDEFINED3-{(Cyclopropylmethyl)[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide160Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54879SLC6A4UNDEFINEDRATUNDEFINED3-{(Cyclopropylmethyl)[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide77Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54880SLC6A4UNDEFINEDRATUNDEFINED3-{(Cyclopropylmethyl)[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide9.96Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54881SLC6A4UNDEFINEDRATUNDEFINED3-{(Cyclopropylmethyl)[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide38.7Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54882SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide288.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54883SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide241.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54884SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide123.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54885SLC6A4UNDEFINEDRATUNDEFINED3-{Cyclobutyl[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide39.3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54886SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-8-Fluoro-3-{[(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl]amino}chromane-5-carboxamide20.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54887SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-8-Fluoro-3-{[(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl]amino}chromane-5-carboxamide47.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54888SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-8-Fluoro-3-[{[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}(propyl)amino]chromane-5-carboxamide1000Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54889SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-8-Fluoro-3-[{[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}(propyl)amino]chromane-5-carboxamide180.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54890SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-3-((Cyclopropylmethyl){[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}amino)-8-fluorochromane-5-carboxamide347Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54891SLC6A4UNDEFINEDRATUNDEFINED(3R)-(-)-3-((Cyclopropylmethyl){[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}amino)-8-fluorochromane-5-carboxamide116Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54892SLC6A4UNDEFINEDRATUNDEFINED(-)-3-{(Cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)-1-methylpropyl]amino}-8-fluorochromane-5-carboxamide10.2Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54893SLC6A4UNDEFINEDRATUNDEFINED(-)-3-{(Cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)-1-methylpropyl]amino}-8-fluorochromane-5-carboxamide46.7Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
548945-HT1AUNDEFINEDHUMANUNDEFINEDrac-[3-(5-fluoro-1H-indol-3-yl)-propyl]-(5-methoxy-chroman-3-yl)-propyl-amine15.8Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
548955-HT1AUNDEFINEDHUMANUNDEFINED8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine19.4Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
548965-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine10.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
548975-HT1AUNDEFINEDHUMANUNDEFINED(3S)-(+)-8-Fluoro-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-N-propylchroman-3-amine12.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
548985-HT1AUNDEFINEDHUMANUNDEFINEDrac-8-fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide3.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
548995-HT1AUNDEFINEDHUMANUNDEFINED(R)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide1.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549005-HT1AUNDEFINEDHUMANUNDEFINED(S)-8-fluoro-3-((3-(5-fluoro-1H-indol-3-yl)propyl)(propyl)amino)-3,4-dihydro-2H-chromene-5-carboxamide3.2Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549015-HT1AUNDEFINEDHUMANUNDEFINED8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)amino}-N-methylchromane-5-carboxamide0.81Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549025-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-3-{[3-(5-fluoro-1H-indol-3-yl)propyl](propyl)-amino}-N-methylchromane-5-carboxamide2.64Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549035-HT1AUNDEFINEDHUMANUNDEFINED3-{[3-(5-Fluoro-1H-indol-3-yl)propyl](propyl)amino}chromane-5-carboxamide0.93Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549045-HT1AUNDEFINEDHUMANUNDEFINEDN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-N-(pyridin-2-yl)cyclohexanecarboxamide trihydrochloride0.96Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549055-HT1AUNDEFINEDHUMANUNDEFINED8-OH-DPAT3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549065-HT1AUNDEFINEDHUMANUNDEFINEDrac-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxychroman-3-amine15.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549075-HT1AUNDEFINEDHUMANUNDEFINED(3R)-N-cyclobutyl-N-[3-(5-fluoro-1H-indol-3-yl)propyl]-5-methoxy-3,4-dihydro-2H-chromen-2.14Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549085-HT1AUNDEFINEDHUMANUNDEFINEDrac-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide9.3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549095-HT1AUNDEFINEDHUMANUNDEFINED(3R)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide1.2Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549105-HT1AUNDEFINEDHUMANUNDEFINED8-Chloro-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-chromane-5-carboxamide6.21Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549115-HT1AUNDEFINEDHUMANUNDEFINED8-Chloro-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-chromane-5-carboxamide10.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549125-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide1.75Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549135-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-0.66Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549145-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}chromane-5-carboxamide29.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549155-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide5.35Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549165-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-methylchromane-5-carboxamide1.32Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549175-HT1AUNDEFINEDHUMANUNDEFINEDMethyl-3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxylate73.8Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549185-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-ethyl-8-fluorochromane-5-carboxamide17.8Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549195-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-propylchromane-5-carboxamide196Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549205-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N-isopropylchromane-5-carboxamide46.1Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549215-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-cyclopropyl-8-fluorochromane-5-carboxamide19.2Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549225-HT1AUNDEFINEDHUMANUNDEFINEDN-Cyclobutyl-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]-amino}-8-fluorochromane-5-carboxamide213.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549235-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-N-(cyclopropylmethyl)-8-fluorochromane-5-carboxamide160.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549245-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluoro-N,N-dimethylchromane-5-carboxamide372Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549255-HT1AUNDEFINEDHUMANUNDEFINED(3S)-3-{cyclobutyl[3-(5-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide253Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549265-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide1.98Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549275-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-[[3-(5-Cyano-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide258Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549285-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(5-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide1.19Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549295-HT1AUNDEFINEDHUMANUNDEFINED3-[[3-(5-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide3.98Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549305-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(6-fluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide5.02Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549315-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[3-(7-methoxy-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide3.22Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549325-HT1AUNDEFINEDHUMANUNDEFINED3-[[3-(7-Chloro-1H-indol-3-yl)propyl](cyclobutyl)amino]-8-fluorochromane-5-carboxamide26.1Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549335-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-{Cyclobutyl[3-(5,7-difluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide1.73Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549345-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-{Cyclobutyl[3-(5,7-difluoro-1H-indol-3-yl)propyl]amino}-8-fluorochromane-5-carboxamide68.9Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549355-HT1AUNDEFINEDHUMANUNDEFINED8-Fluoro-3-[[4-(4-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide14Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549365-HT1AUNDEFINEDHUMANUNDEFINED8-Fluoro-3-[[4-(5-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide6.54Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549375-HT1AUNDEFINEDHUMANUNDEFINED8-Fluoro-3-[[4-(6-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide10.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549385-HT1AUNDEFINEDHUMANUNDEFINED8-Fluoro-3-[[4-(7-fluoro-1H-indol-1-yl)butyl](propyl)amino]chromane-5-carboxamide16.6Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549395-HT1AUNDEFINEDHUMANUNDEFINED3-{(Cyclopropylmethyl)[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide9.64Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549405-HT1AUNDEFINEDHUMANUNDEFINED3-{(Cyclopropylmethyl)[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide5.44Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549415-HT1AUNDEFINEDHUMANUNDEFINED3-{(Cyclopropylmethyl)[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide3.25Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549425-HT1AUNDEFINEDHUMANUNDEFINED3-{(Cyclopropylmethyl)[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide19.25Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549435-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[4-(4-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide17.35Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549445-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[4-(5-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide10.78Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549455-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[4-(6-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide12.83Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549465-HT1AUNDEFINEDHUMANUNDEFINED3-{Cyclobutyl[4-(7-fluoro-1H-indol-1-yl)butyl]amino}-8-fluorochromane-5-carboxamide39.95Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549475-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-3-{[(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl]amino}chromane-5-carboxamide38.05Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549485-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-3-{[(6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl)methyl]amino}chromane-5-carboxamide31.4Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549495-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-3-[{[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}(propyl)amino]chromane-5-carboxamide60.3Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549505-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-8-Fluoro-3-[{[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}(propyl)amino]chromane-5-carboxamide7.34Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549515-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-3-((Cyclopropylmethyl){[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}amino)-8-fluorochromane-5-carboxamide117.5Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549525-HT1AUNDEFINEDHUMANUNDEFINED(3R)-(-)-3-((Cyclopropylmethyl){[6-fluoro-2,3,4,9-tetrahydro-1H-carbazol-3-yl]methyl}amino)-8-fluorochromane-5-carboxamide9.48Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549535-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-{(Cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)-1-methylpropyl]amino}-8-fluorochromane-5-carboxamide1.88Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
549545-HT1AUNDEFINEDHUMANUNDEFINED(-)-3-{(Cyclopropylmethyl)[3-(5-fluoro-1H-indol-3-yl)-1-methylpropyl]amino}-8-fluorochromane-5-carboxamide31.65Hatzenbuhler NT et al., 2008Jan 15, 2025Jan 15, 2025
54955Beta2UNDEFINEDHUMANUNDEFINEDCARAZOLOL0.114Sabio M et al., 2008Jan 15, 2025Jan 28, 2025
54956Beta2UNDEFINEDHUMANUNDEFINED4-[3-(4-Benzhydryl-piperazin-1-yl)-2-hydroxy-propoxy]-1H-indole-2-carbonitrile57.3Sabio M et al., 2008Jan 15, 2025Jan 28, 2025
54957Beta2UNDEFINEDHUMANUNDEFINED2-(4-(3-(tert-butylamino)-2-hydroxypropoxy)-1H-indol-3-yl)acetamide23.5Sabio M et al., 2008Jan 15, 2025Jan 28, 2025
54958Beta2UNDEFINEDHUMANUNDEFINED1-(4-benzhydrylpiperazin-1-yl)-3-(3-methyl-1H-indol-4-yloxy)propan-2-ol0.311Sabio M et al., 2008Jan 15, 2025Jan 28, 2025
54959Beta2UNDEFINEDHUMANUNDEFINEDGNF-Pf-16940.145Sabio M et al., 2008Jan 15, 2025Jan 28, 2025
549605-HT2AUNDEFINEDUNDEFINEDUNDEFINEDC-(9,10-Dihydro-anthracen-9-yl)-methylamine20Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549615-HT2AUNDEFINEDUNDEFINEDUNDEFINEDKETANSERIN0.4Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549625-HT2AUNDEFINEDUNDEFINEDUNDEFINEDDOI0.92Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549635-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(4-hexylphenyl)-2-phenylethanamine200Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549645-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(4-bromophenyl)-2-phenylethanamine260Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549655-HT2AUNDEFINEDUNDEFINEDUNDEFINED2,2-Diphenyl-ethylamine4610Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549665-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(4-hexylphenyl)ethanamine78Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549675-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-[4-(3-Phenyl-propyl)-phenyl]-ethylamine60Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549685-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(4-bromophenyl)ethylamine1770Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549695-HT2AUNDEFINEDUNDEFINEDUNDEFINEDPhenylethylamine>10000Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549705-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-(2-Amino-propyl)-2,5-dimethoxy-phenol>10000Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549715-HT2AUNDEFINEDUNDEFINEDUNDEFINED1-Methyl-2-(2,4,5-trimethoxy-phenyl)-ethylamine1200Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549725-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(4-Hexyl-2,5-dimethoxy-phenyl)-1-methyl-ethylamine : (Hydrochloride)2.5Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549735-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-[2,5-Dimethoxy-4-(3-phenyl-propyl)-phenyl]-1-methyl-ethylamine10Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549745-HT2AUNDEFINEDUNDEFINEDUNDEFINEDDOB41Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549755-HT2AUNDEFINEDUNDEFINEDUNDEFINED2-(2,5-Dimethoxy-phenyl)-1-methyl-ethylamine5200Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549765-HT2AUNDEFINEDUNDEFINEDUNDEFINED3-n-Hexyl-6-methoxy-9-aminomethyl-9,10-dihydroanthracene43Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549775-HT2AUNDEFINEDUNDEFINEDUNDEFINED3-Hydroxy-9-aminomethyl-9,10-dihydroanthracene107Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549785-HT2AUNDEFINEDUNDEFINEDUNDEFINED3-n-Pentyloxy-9-aminomethyl-9,10-dihydroanthracene fumarate23Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549795-HT2AUNDEFINEDUNDEFINEDUNDEFINED3-methoxy-9-aminomethyl-9,10-dihydroanthracene7.5Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549805-HT2AUNDEFINEDUNDEFINEDUNDEFINEDC-(3-Hexyl-9,10-dihydro-anthracen-9-yl)-methylamine7Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549815-HT2AUNDEFINEDUNDEFINEDUNDEFINEDC-[3-(3-Phenyl-propyl)-9,10-dihydro-anthracen-9-yl]-methylamine3.2Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549825-HT2AUNDEFINEDUNDEFINEDUNDEFINEDC-(3-Bromo-9,10-dihydro-anthracen-9-yl)-methylamine1.3Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549835-HT2AUNDEFINEDUNDEFINEDUNDEFINEDDOB0.29Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549845-HT2AUNDEFINEDUNDEFINEDUNDEFINEDDOB1.9Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549855-HT2CUNDEFINEDUNDEFINEDUNDEFINEDC-(9,10-Dihydro-anthracen-9-yl)-methylamine43Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549865-HT2CUNDEFINEDUNDEFINEDUNDEFINEDC-(3-Bromo-9,10-dihydro-anthracen-9-yl)-methylamine3.3Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
549875-HT2CUNDEFINEDUNDEFINEDUNDEFINEDC-(3-Hexyl-9,10-dihydro-anthracen-9-yl)-methylamine62Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54988D2UNDEFINEDUNDEFINEDUNDEFINEDC-(9,10-Dihydro-anthracen-9-yl)-methylamine>10000Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54989D2UNDEFINEDUNDEFINEDUNDEFINEDC-(3-Bromo-9,10-dihydro-anthracen-9-yl)-methylamine>10000Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54990D2UNDEFINEDUNDEFINEDUNDEFINEDC-(3-Hexyl-9,10-dihydro-anthracen-9-yl)-methylamine6280Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54991SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDC-(9,10-Dihydro-anthracen-9-yl)-methylamine>10000Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54992SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDC-(3-Bromo-9,10-dihydro-anthracen-9-yl)-methylamine1200Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54993SLC6A4UNDEFINEDUNDEFINEDUNDEFINEDC-(3-Hexyl-9,10-dihydro-anthracen-9-yl)-methylamine490Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54994SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDC-(9,10-Dihydro-anthracen-9-yl)-methylamine>10000Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54995SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDC-(3-Bromo-9,10-dihydro-anthracen-9-yl)-methylamine4490Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54996SLC6A2UNDEFINEDUNDEFINEDUNDEFINEDC-(3-Hexyl-9,10-dihydro-anthracen-9-yl)-methylamine845Runyon SP et al., 2008Jan 15, 2025Jan 15, 2025
54997D1UNDEFINEDRATUNDEFINEDPramipexole>10000Chen J et al., 2008Jan 15, 2025Jan 15, 2025
54998D1UNDEFINEDRATUNDEFINEDN-(4-{2-[((S)-2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-propyl-amino]-ethyl}-cyclohexyl)-3-phenyl-acrylamide>10000Chen J et al., 2008Jan 15, 2025Jan 15, 2025
54999D1UNDEFINEDRATUNDEFINEDBenzofuran-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-propyl-amino]-ethyl}-cyclohexyl)-amide4900Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55000D1UNDEFINEDRATUNDEFINEDNaphthalene-2-carboxylic acid {4-[2-((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-ylamino)-ethyl]-cyclohexyl}-amide>10000Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55001D1UNDEFINEDRATUNDEFINEDNaphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-(2-cyclohexyl-ethyl)-amino]-ethyl}-cyclohexyl)-amide4400Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55002D1UNDEFINEDRATUNDEFINEDNaphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-(3-methyl-butyl)-amino]-ethyl}-cyclohexyl)-amide>10000Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55003D1UNDEFINEDRATUNDEFINEDNaphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-butyl-amino]-ethyl}-cyclohexyl)-amide5400Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55004D1UNDEFINEDRATUNDEFINEDNaphthalene-2-carboxylic acid (4-{2-[((S)-2-amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-propyl-amino]-ethyl}-cyclohexyl)-amide3400Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55005D1UNDEFINEDRATUNDEFINED(S)-N-(4-((2-amino-4,5,6,7-tetrahydrobenzo[d]thiazol-6-yl)(propyl)amino)butyl)-2-naphthamide>10000Chen J et al., 2008Jan 15, 2025Jan 15, 2025
55006D1UNDEFINEDRATUNDEFINEDNaphthalene-2-carboxylic acid {4-[2-((R)-8-methoxy-1,2,4,4a,5,6-hexahydro-pyrazino[1,2-a]quinolin-3-yl)-ethyl]-cyclohexyl}-amide>10000Chen J et al., 2008Jan 15, 2025Jan 15, 2025
550075-HT7UNDEFINEDRATUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide71Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550085-HT7UNDEFINEDRATUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide76Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550095-HT7UNDEFINEDRATUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide5.7Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550105-HT7UNDEFINEDRATUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide148Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550115-HT7UNDEFINEDRATUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide296Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550125-HT7UNDEFINEDRATUNDEFINEDN-(4-Cyanophenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide8.6Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550135-HT7UNDEFINEDRATUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide0.58Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550145-HT7UNDEFINEDRATUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide9Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550155-HT7UNDEFINEDRATUNDEFINED4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide389Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550165-HT7UNDEFINEDRATUNDEFINED4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide5.1Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550175-HT7UNDEFINEDRATUNDEFINED4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide0.98Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550185-HT7UNDEFINEDRATUNDEFINED4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide34.8Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550195-HT7UNDEFINEDRATUNDEFINEDN-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide224Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550205-HT7UNDEFINEDRATUNDEFINEDN-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide215Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550215-HT7UNDEFINEDRATUNDEFINEDN-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide0.8Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550225-HT7UNDEFINEDRATUNDEFINEDN-Benzyl-4-(2-methylthiophenyl)-1-piperazinehexanamide22Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550235-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline31Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550245-HT7UNDEFINEDRATUNDEFINED5-CT0.5Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550255-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline6Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550265-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline3.81Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550275-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline32.9Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550285-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline179Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550295-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]isoindoline54Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550305-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline8.3Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550315-HT7UNDEFINEDRATUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]isoindoline42Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550325-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide29Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550335-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide57Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550345-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide106Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550355-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide10.3Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550365-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide43Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550375-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide53Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550385-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide188Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550395-HT1AUNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide94Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550405-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide19Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550415-HT1AUNDEFINEDHUMANUNDEFINED4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide325Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550425-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide70Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550435-HT1AUNDEFINEDHUMANUNDEFINED4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide8.2Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550445-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide13Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550455-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide139Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550465-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide161Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550475-HT1AUNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-methylthiophenyl)-1-piperazinehexanamide12Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550485-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline40Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550495-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline3.7Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550505-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline95Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550515-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline2.04Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550525-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline3.2Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550535-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]isoindoline22Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550545-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline124Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550555-HT1AUNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]isoindoline1.07Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
550565-HT1AUNDEFINEDHUMANUNDEFINED8-OH-DPAT2.1Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55057D2UNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide91Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55058D2UNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide7.8Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55059D2UNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide723Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55060D2UNDEFINEDHUMANUNDEFINEDN-(4-Methanesulfonyloxyphenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide30Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55061D2UNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-methoxyphenyl)-1-piperazinehexanamide311Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55062D2UNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide20Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55063D2UNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-diphenyl)-1-piperazinehexanamide142Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55064D2UNDEFINEDHUMANUNDEFINEDN-(4-Cyanophenylmethyl)-4-(2-methylthiophenyl)-1-piperazinehexanamide5.3Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55065D2UNDEFINEDHUMANUNDEFINED4-(2-Methoxyphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide501Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55066D2UNDEFINEDHUMANUNDEFINED4-[2-(1-Methylethyl)phenyl]-N-(4-pyridinylmethyl)-1-piperazinehexanamide21Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55067D2UNDEFINEDHUMANUNDEFINED4-(2-Diphenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide185Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55068D2UNDEFINEDHUMANUNDEFINED4-(2-Methylthiophenyl)-N-(4-pyridinylmethyl)-1-piperazinehexanamide64Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55069D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-methoxyphenyl)-1-piperazinehexanamide226Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55070D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-[2-(1-methylethyl)phenyl]-1-piperazinehexanamide9.2Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55071D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-diphenyl)-1-piperazinehexanamide503Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55072D2UNDEFINEDHUMANUNDEFINEDN-Benzyl-4-(2-methylthiophenyl)-1-piperazinehexanamide33Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55073D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline22Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55074D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline1.3Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55075D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline362Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55076D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]-1,2,3,4-tetrahydroisoquinoline40Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55077D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methoxyphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline730Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55078D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-(1-Methylethyl)phenyl)-1-piperazinyl]-1-oxohexyl]isoindoline65Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55079D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Diphenyl)-1-piperazinyl]-1-oxohexyl]isoindoline93Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55080D2UNDEFINEDHUMANUNDEFINED2-[6-[4-(2-Methylthiophenyl)-1-piperazinyl]-1-oxohexyl]isoindoline96Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55081D2UNDEFINEDHUMANUNDEFINEDHALOPERIDOL4.2Leopoldo M et al., 2008Jan 15, 2025Jan 15, 2025
55082H3UNDEFINEDHUMANUNDEFINEDAMITRIPTYLINE1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55083H3UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide4.9von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55084H3UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide3.5von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55085H3UNDEFINEDHUMANUNDEFINED[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine0.25von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55086H3UNDEFINEDHUMANUNDEFINEDMAPROTILINE1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55087H3UNDEFINEDHUMANUNDEFINEDmethyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen-1-yl}propyl)amine0.358von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55088H3UNDEFINEDHUMANUNDEFINEDCHLORPROMAZINE1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55089H3UNDEFINEDHUMANUNDEFINED[3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine1.21von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55090H3UNDEFINEDHUMANUNDEFINEDCHLORPROTHIXENE1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55091H3UNDEFINEDHUMANUNDEFINED{3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine1.54von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55092H3UNDEFINEDHUMANUNDEFINEDCLOZAPINE1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55093H3UNDEFINEDHUMANUNDEFINED8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine3.27von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55094H3UNDEFINEDHUMANUNDEFINEDFLUPHENAZINE1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55095H3UNDEFINEDHUMANUNDEFINED4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester0.042von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55096H1UNDEFINEDHUMANUNDEFINEDAMITRIPTYLINE1.12von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55097H1UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide559von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55098H1UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide686von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55099H1UNDEFINEDHUMANUNDEFINED[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine79von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55100H1UNDEFINEDHUMANUNDEFINEDMAPROTILINE1.67von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55101H1UNDEFINEDHUMANUNDEFINEDmethyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen-1-yl}propyl)amine40von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55102H1UNDEFINEDHUMANUNDEFINEDCHLORPROMAZINE4.25von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55103H1UNDEFINEDHUMANUNDEFINED[3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine205von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55104H1UNDEFINEDHUMANUNDEFINEDCHLORPROTHIXENE3.75von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55105H1UNDEFINEDHUMANUNDEFINED{3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine295von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55106H1UNDEFINEDHUMANUNDEFINEDCLOZAPINE2.38von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55107H1UNDEFINEDHUMANUNDEFINED8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine190von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55108H1UNDEFINEDHUMANUNDEFINEDFLUPHENAZINE40von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55109H1UNDEFINEDHUMANUNDEFINED4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester390von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55110D1UNDEFINEDHUMANUNDEFINEDAMITRIPTYLINE89von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55111D1UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide879von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55112D1UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55113D1UNDEFINEDHUMANUNDEFINED[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine305von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55114D1UNDEFINEDHUMANUNDEFINEDMAPROTILINE402von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55115D1UNDEFINEDHUMANUNDEFINEDmethyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen-1-yl}propyl)amine203von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55116D1UNDEFINEDHUMANUNDEFINEDCHLORPROMAZINE96von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55117D1UNDEFINEDHUMANUNDEFINED[3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine232von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55118D1UNDEFINEDHUMANUNDEFINED{3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine248von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55119D1UNDEFINEDHUMANUNDEFINEDCLOZAPINE89von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55120D1UNDEFINEDHUMANUNDEFINED8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine866von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55121D1UNDEFINEDHUMANUNDEFINEDFLUPHENAZINE179von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55122D1UNDEFINEDHUMANUNDEFINED4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester203von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55123D1UNDEFINEDHUMANUNDEFINEDCHLORPROTHIXENE18von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55124D5UNDEFINEDHUMANUNDEFINEDAMITRIPTYLINE170von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55125D5UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55126D5UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55127D5UNDEFINEDHUMANUNDEFINED[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine273von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55128D5UNDEFINEDHUMANUNDEFINEDMAPROTILINE429von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55129D5UNDEFINEDHUMANUNDEFINEDmethyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen-1-yl}propyl)amine265von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55130D5UNDEFINEDHUMANUNDEFINEDCHLORPROMAZINE172von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55131D5UNDEFINEDHUMANUNDEFINED[3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine153von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55132D5UNDEFINEDHUMANUNDEFINEDCHLORPROTHIXENE9von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55133D5UNDEFINEDHUMANUNDEFINED{3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine297von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55134D5UNDEFINEDHUMANUNDEFINEDCLOZAPINE198von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55135D5UNDEFINEDHUMANUNDEFINED8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine921von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55136D5UNDEFINEDHUMANUNDEFINEDFLUPHENAZINE21von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55137D5UNDEFINEDHUMANUNDEFINED4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester265von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55138D2UNDEFINEDHUMANUNDEFINEDAMITRIPTYLINE196von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55139D2UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide904von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55140D2UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide1000von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55141D2UNDEFINEDHUMANUNDEFINED[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine101von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55142D2UNDEFINEDHUMANUNDEFINEDMAPROTILINE665von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55143D2UNDEFINEDHUMANUNDEFINEDmethyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen-1-yl}propyl)amine146von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55144D2UNDEFINEDHUMANUNDEFINEDCHLORPROMAZINE4.06von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55145D2UNDEFINEDHUMANUNDEFINED[3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine41von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55146D2UNDEFINEDHUMANUNDEFINEDCHLORPROTHIXENE2.96von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55147D2UNDEFINEDHUMANUNDEFINED{3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine52von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55148D2UNDEFINEDHUMANUNDEFINEDCLOZAPINE83von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55149D2UNDEFINEDHUMANUNDEFINED8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine285von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55150D2UNDEFINEDHUMANUNDEFINEDFLUPHENAZINE1.44von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55151D2UNDEFINEDHUMANUNDEFINED4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester47von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55152D3UNDEFINEDHUMANUNDEFINEDAMITRIPTYLINE206von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55153D3UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-acetamide326von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55154D3UNDEFINEDHUMANUNDEFINEDN-[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-N-methyl-4-(3-piperidin-1-yl-propoxy)-benzamide243von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55155D3UNDEFINEDHUMANUNDEFINED[3-(10,11-Dihydro-dibenzo[a,d]cyclohepten-5-ylidene)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine67von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55156D3UNDEFINEDHUMANUNDEFINEDMAPROTILINE504von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55157D3UNDEFINEDHUMANUNDEFINEDmethyl({4-[3-(piperidin-1-yl)propoxy]phenyl}methyl)(3-{tetracyclo[6.6.2.0^{2,7}.0^{9,14}]hexadeca-2(7),3,5,9(14),10,12-hexaen-1-yl}propyl)amine149von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55158D3UNDEFINEDHUMANUNDEFINEDCHLORPROMAZINE6.9von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55159D3UNDEFINEDHUMANUNDEFINED[3-(2-Chloro-phenothiazin-10-yl)-propyl]-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine50von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55160D3UNDEFINEDHUMANUNDEFINEDCHLORPROTHIXENE4.56von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55161D3UNDEFINEDHUMANUNDEFINED{3-[2-Chloro-thioxanthenylidene]-propyl}-methyl-[4-(3-piperidin-1-yl-propoxy)-benzyl]-amine50von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55162D3UNDEFINEDHUMANUNDEFINEDCLOZAPINE295von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55163D3UNDEFINEDHUMANUNDEFINED8-Chloro-11-{4-[4-(3-piperidin-1-yl-propoxy)-benzyl]-piperazin-1-yl}-5H-dibenzo[b,e][1,4]diazepine223von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55164D3UNDEFINEDHUMANUNDEFINEDFLUPHENAZINE3.21von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
55165D3UNDEFINEDHUMANUNDEFINED4-(3-Piperidin-1-yl-propoxy)-benzoic acid 2-{4-[3-(2-trifluoromethyl-phenothiazin-10-yl)-propyl]-piperazin-1-yl}-ethyl ester15von Coburg Y et al., 2009Jan 15, 2025Jan 15, 2025
551665-HT1AUNDEFINEDHUMANUNDEFINEDBUSPIRONE15Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551675-HT1AUNDEFINEDHUMANUNDEFINED(+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine75.3Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551685-HT1AUNDEFINEDHUMANUNDEFINED(+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(cyclopropylmethyl)pyrimidin-2-amine21.3Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551695-HT1AUNDEFINEDHUMANUNDEFINED(+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(1-cyclopropylethyl)pyrimidin-2-amine7.4Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551705-HT1AUNDEFINEDHUMANUNDEFINED(+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(1-methylcyclopropyl)pyrimidin-2-amine32Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551715-HT1AUNDEFINEDHUMANUNDEFINED(+/-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-tert-butylpyrimidin-2-amine5.2Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551725-HT1AUNDEFINEDHUMANUNDEFINED(-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-propylpyrimidin-2-amine11.2Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551735-HT1AUNDEFINEDHUMANUNDEFINED(-)-4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-propylpyrimidin-2-amine16.3Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551745-HT1AUNDEFINEDHUMANUNDEFINEDN-cyclopropyl-4-(1-(2-(5-fluoro-1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine23.6Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551755-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(2-(5-chloro-1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine10.4Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551765-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine26.6Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551775-HT1AUNDEFINEDHUMANUNDEFINEDN-cyclopropyl-4-(1-(2-(7-fluoro-1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine35.1Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551785-HT1AUNDEFINEDHUMANUNDEFINEDN-cyclopropyl-4-(1-(2-(6-fluoro-1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine64.5Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551795-HT1AUNDEFINEDHUMANUNDEFINEDN-cyclopropyl-4-(1-(2-((S)-2,3-dihydrobenzo[b][1,4]dioxin-2-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine37.8Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551805-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(2-(benzo[b]thiophen-3-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine38.5Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551815-HT1AUNDEFINEDHUMANUNDEFINEDN-cyclopropyl-4-(1-(2-(2,3-dihydro-1H-inden-2-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine42.5Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551825-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(1-(1H-indol-3-yl)propan-2-yl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine40.2Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551835-HT1AUNDEFINEDHUMANUNDEFINED2-(3-(2-(cyclopropylamino)pyrimidin-4-yl)piperidin-1-yl)-1-(1H-indol-3-yl)ethanone3420Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551845-HT1AUNDEFINEDHUMANUNDEFINEDN-cyclopropyl-4-(1-(2-(thiazol-4-yl)ethyl)piperidin-3-yl)pyrimidin-2-amine780Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551855-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(2-(1H-pyrazol-4-yl)ethyl)piperidin-3-yl)-N-cyclopropylpyrimidin-2-amine4450Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551865-HT1AUNDEFINEDHUMANUNDEFINED3-(4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)pyrimidin-2-ylamino)propan-1-ol175Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551875-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(3-methoxypropyl)pyrimidin-2-amine78.3Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
551885-HT1AUNDEFINEDHUMANUNDEFINED4-(1-(2-(1H-indol-3-yl)ethyl)piperidin-3-yl)-N-(2-methoxyethyl)pyrimidin-2-amine66.3Dounay AB et al., 2009Jan 15, 2025Jan 15, 2025
55189OPRL1UNDEFINEDHUMANUNDEFINEDFLUSPIRILENE500Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55190OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one23Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55191OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one31Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55192OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one84Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55193OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one34Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55194OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one57Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55195OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-isopropyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one66Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55196OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclopropylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one83Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55197OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclobutylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one53Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55198OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclohexylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one89Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55199OPRL1UNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-(prop-2-ynyl)-1,3,8-triazaspiro[4.5]decan-4-one234Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55200OPRL1UNDEFINEDHUMANUNDEFINED3-allyl-8-benzhydryl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one203Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55201OPRL1UNDEFINEDHUMANUNDEFINED8-[bis-(2-chloro-phenyl)-methyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one6.8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55202OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one48.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55203OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-isopentyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one56Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55204OPRL1UNDEFINEDHUMANUNDEFINEDmethyl 2-(8-(bis(2-chlorophenyl)methyl)-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl)acetate19.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55205OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one18.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55206OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-methoxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one26Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55207OPRL1UNDEFINEDHUMANUNDEFINED3-(2-aminoethyl)-8-(bis(2-chlorophenyl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one47.8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55208OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one4.05Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55209OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2.1Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55210OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2.55Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55211OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one8.65Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55212OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55213OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(dimethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one3.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55214OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one3.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55215OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(diisopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one12.1Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55216OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(butylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2.15Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55217OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2.75Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55218OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylmethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one3.8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55219OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one2.25Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55220OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(3-(pyrrolidin-1-yl)propyl)-1,3,8-triazaspiro[4.5]decan-4-one3.2Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55221OPRL1UNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(piperidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55222OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichloro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one2.3Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55223OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55224OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55225OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55226OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55227OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55228OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one0.6Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55229OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55230OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.4Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55231OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55232OPRL1UNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one2.3Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55233OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one1.3Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55234OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one5.4Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55235OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one4.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55236OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55237OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2.1Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55238OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1.6Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55239OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1.4Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55240OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclopentylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.9Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55241OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.9Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55242OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one1Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55243OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(allylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.9Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55244OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55245OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55246OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55247OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(diisopropylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one6.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55248OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one1.4Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55249OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.5Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55250OPRL1UNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.4Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55251OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.7Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55252OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(benzylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one3.6Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55253OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one15.9Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55254OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(5-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1.8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55255OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6-chloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one0.6Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55256OPRL1UNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6,7-dichloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one12.2Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55257DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55258DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55259DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55260DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55261DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55262DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-isopropyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one9111Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55263DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclopropylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one5412Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55264DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclobutylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one8210Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55265DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclohexylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55266DORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-(prop-2-ynyl)-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55267DORUNDEFINEDHUMANUNDEFINED3-allyl-8-benzhydryl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55268DORUNDEFINEDHUMANUNDEFINED8-[bis-(2-chloro-phenyl)-methyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55269DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55270DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-isopentyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55271DORUNDEFINEDHUMANUNDEFINEDmethyl 2-(8-(bis(2-chlorophenyl)methyl)-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl)acetate>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55272DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one5612Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55273DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-methoxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55274DORUNDEFINEDHUMANUNDEFINED3-(2-aminoethyl)-8-(bis(2-chlorophenyl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one32Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55275DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one578Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55276DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one868Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55277DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one955Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55278DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1525Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55279DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one759Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55280DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(dimethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one933Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55281DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1136Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55282DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(diisopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one4758Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55283DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(butylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1033Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55284DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one878Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55285DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylmethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1535Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55286DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one906Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55287DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(3-(pyrrolidin-1-yl)propyl)-1,3,8-triazaspiro[4.5]decan-4-one2381Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55288DORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(piperidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one3176Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55289DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichloro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one1633Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55290DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2270Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55291DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1676Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55292DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1080Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55293DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one445Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55294DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one370Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55295DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one516Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55296DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one376Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55297DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one867Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55298DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one379Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55299DORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one538Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55300DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one1790Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55301DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one3103Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55302DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one795Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55303DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2639Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55304DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1298Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55305DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2064Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55306DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one5016Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55307DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopentylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1615Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55308DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1951Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55309DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one2340Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55310DORUNDEFINEDHUMANUNDEFINED3-(2-(allylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2515Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55311DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2096Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55312DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2879Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55313DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1802Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55314DORUNDEFINEDHUMANUNDEFINED3-(2-(diisopropylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2980Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55315DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one1224Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55316DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one3948Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55317DORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2600Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55318DORUNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1693Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55319DORUNDEFINEDHUMANUNDEFINED3-(2-(benzylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1279Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55320DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1062Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55321DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(5-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1316Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55322DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6-chloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one883Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55323DORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6,7-dichloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one5022Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55324KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one137Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55325KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one150Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55326KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one506Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55327KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one1342Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55328KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one773Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55329KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-isopropyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one543Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55330KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclopropylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one633Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55331KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclobutylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1846Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55332KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclohexylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2316Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55333KORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-(prop-2-ynyl)-1,3,8-triazaspiro[4.5]decan-4-one1268Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55334KORUNDEFINEDHUMANUNDEFINED3-allyl-8-benzhydryl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one694Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55335KORUNDEFINEDHUMANUNDEFINED8-[bis-(2-chloro-phenyl)-methyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one5887Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55336KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55337KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-isopentyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55338KORUNDEFINEDHUMANUNDEFINEDmethyl 2-(8-(bis(2-chlorophenyl)methyl)-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl)acetate2274Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55339KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1747Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55340KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-methoxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1830Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55341KORUNDEFINEDHUMANUNDEFINED3-(2-aminoethyl)-8-(bis(2-chlorophenyl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one852Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55342KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one871Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55343KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one497Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55344KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one469Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55345KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one247Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55346KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one224Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55347KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(dimethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one320Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55348KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1014Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55349KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(diisopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one674Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55350KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(butylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one165Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55351KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one238Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55352KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylmethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one271Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55353KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one254Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55354KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(3-(pyrrolidin-1-yl)propyl)-1,3,8-triazaspiro[4.5]decan-4-one64Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55355KORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(piperidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one279Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55356KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichloro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one52Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55357KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one68Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55358KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one54Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55359KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one40Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55360KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one25Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55361KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one29Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55362KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one13Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55363KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one8Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55364KORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one10Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55365KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one56Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55366KORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one15Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55367KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one540Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55368KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one1392Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55369KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one56Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55370KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one655Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55371KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one48Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55372KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one39Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55373KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one68Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55374KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopentylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one49Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55375KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one33Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55376KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one45Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55377KORUNDEFINEDHUMANUNDEFINED3-(2-(allylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one208Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55378KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one45Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55379KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one174Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55380KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one65Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55381KORUNDEFINEDHUMANUNDEFINED3-(2-(diisopropylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one86Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55382KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one169Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55383KORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one138Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55384KORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one82Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55385KORUNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one26Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55386KORUNDEFINEDHUMANUNDEFINED3-(2-(benzylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one151Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55387KORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one11Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55388KORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(5-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one14Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55389KORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6-chloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one25Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55390KORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6,7-dichloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one158Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55391MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one489Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55392MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one692Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55393MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2283Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55394MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55395MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one8438Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55396MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-isopropyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one4042Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55397MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-3-(cyclopropylmethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one5279Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55398MORUNDEFINEDHUMANUNDEFINED8-benzhydryl-1-phenyl-3-(prop-2-ynyl)-1,3,8-triazaspiro[4.5]decan-4-one4314Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55399MORUNDEFINEDHUMANUNDEFINED3-allyl-8-benzhydryl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55400MORUNDEFINEDHUMANUNDEFINED8-[bis-(2-chloro-phenyl)-methyl]-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one5945Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55401MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-butyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55402MORUNDEFINEDHUMANUNDEFINEDmethyl 2-(8-(bis(2-chlorophenyl)methyl)-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl)acetate683Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55403MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one483Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55404MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-methoxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one726Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55405MORUNDEFINEDHUMANUNDEFINED3-(2-aminoethyl)-8-(bis(2-chlorophenyl)methyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one886Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55406MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1069Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55407MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one776Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55408MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one745Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55409MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one625Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55410MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one400Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55411MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(dimethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one421Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55412MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one978Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55413MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(diisopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1921Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55414MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(butylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one2546Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55415MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1376Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55416MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-(2-(cyclohexylmethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one1800Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55417MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one436Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55418MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(3-(pyrrolidin-1-yl)propyl)-1,3,8-triazaspiro[4.5]decan-4-one436Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55419MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-1-phenyl-3-(2-(piperidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one683Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55420MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichloro-benzyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one29Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55421MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one146Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55422MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one167Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55423MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one136Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55424MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one89Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55425MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one112Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55426MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one28Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55427MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one26Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55428MORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(2,6-dichlorobenzyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one36Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55429MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-3-(2-(diethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one122Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55430MORUNDEFINEDHUMANUNDEFINED8-(2,6-dichlorobenzyl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one37Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55431MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one48Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55432MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-propyl-1,3,8-triazaspiro[4.5]decan-4-one142Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55433MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-oxopropyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one14Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55434MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-hydroxyethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one59Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55435MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(methylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one35Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55436MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(ethylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one37Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55437MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopropylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one69Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55438MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopentylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one96Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55439MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one120Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55440MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(propylamino)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one43Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55441MORUNDEFINEDHUMANUNDEFINED3-(2-(allylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one198Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55442MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclobutylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one64Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55443MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclopropylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one239Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55444MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isobutylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one61Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55445MORUNDEFINEDHUMANUNDEFINED3-(2-(diisopropylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one82Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55446MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-3-(2-(pyrrolidin-1-yl)ethyl)-1,3,8-triazaspiro[4.5]decan-4-one69Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55447MORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one66Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55448MORUNDEFINEDHUMANUNDEFINED8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(2-(isopentylamino)ethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one204Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55449MORUNDEFINEDHUMANUNDEFINED3-(2-(cyclohexylmethylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one102Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55450MORUNDEFINEDHUMANUNDEFINED3-(2-(benzylamino)ethyl)-8-(4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one139Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55451MORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(7-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one297Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55452MORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(5-chloro-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one141Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55453MORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6-chloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one50Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55454MORUNDEFINEDHUMANUNDEFINED3-(2-(butylamino)ethyl)-8-(6,7-dichloro-4,4-dimethyl-1,2,3,4-tetrahydronaphthalen-1-yl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one306Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55455MORUNDEFINEDHUMANUNDEFINED8-(bis(2-chlorophenyl)methyl)-3-isopentyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Caldwell JP et al., 2009Jan 15, 2025Jan 15, 2025
55456D3UNDEFINEDHUMANUNDEFINED4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one5.1Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55457D3UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-8-(4-fluorobenzyl)-8-azabicyclo[3.2.1]octan-3-ol172Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55458D3UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-8-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-8-azabicyclo[3.2.1]octan-3-ol128Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55459D3UNDEFINEDHUMANUNDEFINEDendo-8-(1H-Indol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo-[3.2.1]octan-3-ol25Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55460D3UNDEFINEDHUMANUNDEFINED8-(2-(1H-indol-3-yl)ethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol18Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55461D3UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-1-(1H-indol-3-ylmethyl)pyrrolidin-3-ol2874Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55462D3UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-1-[2-(1H-indol-3-yl)ethyl]pyrrolidin-3-ol3074Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55463D3UNDEFINEDHUMANUNDEFINED3-{[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]methyl}-1Hpyrrolo[2,3-b]pyridine370Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55464D3UNDEFINEDHUMANUNDEFINED9-[(1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]-3-(4-chlorophenyl)-3,9-diazabicyclo[4.2.1]nonane335.5Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55465D3UNDEFINEDHUMANUNDEFINED4-(6-(4-chlorophenyl)-2,6-diazabicyclo[2.2.1]heptan-2-yl)-1-(4-fluorophenyl)butan-1-one220Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55466D3UNDEFINEDHUMANUNDEFINED2-{(1H-Pyrrolo[2,3-b]pyridin-3-yl)methyl}-5-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane11Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55467D3UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one200Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55468D3UNDEFINEDHUMANUNDEFINED3-{(4-(Pyrimidin-2-yl)piperazin-1-yl)methyl}-1H-pyrrolo[2,3-b]pyridine1500Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55469D3UNDEFINEDHUMANUNDEFINEDHALOPERIDOL5.5Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55470D3UNDEFINEDHUMANUNDEFINED2-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)ethanone>10000Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55471D2UNDEFINEDHUMANUNDEFINED4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one1.6Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55472D2UNDEFINEDHUMANUNDEFINED2-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)ethanone1231Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55473D2UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-8-(4-fluorobenzyl)-8-azabicyclo[3.2.1]octan-3-ol1050Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55474D2UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-8-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-8-azabicyclo[3.2.1]octan-3-ol588Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55475D2UNDEFINEDHUMANUNDEFINEDendo-8-(1H-Indol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo-[3.2.1]octan-3-ol160.3Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55476D2UNDEFINEDHUMANUNDEFINED8-(2-(1H-indol-3-yl)ethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol53Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55477D2UNDEFINEDHUMANUNDEFINED3-{[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]methyl}-1Hpyrrolo[2,3-b]pyridine970Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55478D2UNDEFINEDHUMANUNDEFINED9-[(1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]-3-(4-chlorophenyl)-3,9-diazabicyclo[4.2.1]nonane>10000Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55479D2UNDEFINEDHUMANUNDEFINED4-(6-(4-chlorophenyl)-2,6-diazabicyclo[2.2.1]heptan-2-yl)-1-(4-fluorophenyl)butan-1-one170Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55480D2UNDEFINEDHUMANUNDEFINED2-{(1H-Pyrrolo[2,3-b]pyridin-3-yl)methyl}-5-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane62Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55481D2UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one33Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55482D2UNDEFINEDHUMANUNDEFINED3-{(4-(Pyrimidin-2-yl)piperazin-1-yl)methyl}-1H-pyrrolo[2,3-b]pyridine1170Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55483D2UNDEFINEDHUMANUNDEFINEDHALOPERIDOL1.1Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55484D2UNDEFINEDHUMANUNDEFINED4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one254Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55485D2UNDEFINEDHUMANUNDEFINED4-(4-Chloro-phenyl)-1-(1H-indol-3-ylmethyl)-piperidin-4-ol11.2Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55486D2UNDEFINEDHUMANUNDEFINEDL-745870960Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
554875-HT1AUNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one2332Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
554885-HT2AUNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one194.8Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
554895-HT2CUNDEFINEDHUMANUNDEFINED4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one3513Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55490D4UNDEFINEDHUMANUNDEFINED4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one5.3Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55491D4UNDEFINEDHUMANUNDEFINED2-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)ethanone789Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55492D4UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-8-(4-fluorobenzyl)-8-azabicyclo[3.2.1]octan-3-ol1015Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55493D4UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-8-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-8-azabicyclo[3.2.1]octan-3-ol7873Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55494D4UNDEFINEDHUMANUNDEFINEDendo-8-(1H-Indol-3-ylmethyl)-3-(4-chlorophenyl)-8-azabicyclo-[3.2.1]octan-3-ol3007Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55495D4UNDEFINEDHUMANUNDEFINED8-(2-(1H-indol-3-yl)ethyl)-3-(4-chlorophenyl)-8-azabicyclo[3.2.1]octan-3-ol277.5Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55496D4UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-1-(1H-indol-3-ylmethyl)pyrrolidin-3-ol816.5Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55497D4UNDEFINEDHUMANUNDEFINED3-{[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]methyl}-1Hpyrrolo[2,3-b]pyridine18.6Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55498D4UNDEFINEDHUMANUNDEFINED9-[(1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]-3-(4-chlorophenyl)-3,9-diazabicyclo[4.2.1]nonane583.7Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55499D4UNDEFINEDHUMANUNDEFINED4-(6-(4-chlorophenyl)-2,6-diazabicyclo[2.2.1]heptan-2-yl)-1-(4-fluorophenyl)butan-1-one513Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55500D4UNDEFINEDHUMANUNDEFINED2-{(1H-Pyrrolo[2,3-b]pyridin-3-yl)methyl}-5-(4-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptane69Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55501D4UNDEFINEDHUMANUNDEFINED4-[3-(4-Chloro-phenyl)-3-hydroxy-pyrrolidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one11Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55502D4UNDEFINEDHUMANUNDEFINED3-(4-Chlorophenyl)-1-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrrolidin-3-ol1213Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55503D4UNDEFINEDHUMANUNDEFINED3-{(4-(Pyrimidin-2-yl)piperazin-1-yl)methyl}-1H-pyrrolo[2,3-b]pyridine56Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55504D4UNDEFINEDHUMANUNDEFINEDHALOPERIDOL12.7Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55505D4UNDEFINEDHUMANUNDEFINED4-(4-(4-chlorophenyl)piperazin-1-yl)-1-(4-fluorophenyl)butan-1-one17Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55506D4UNDEFINEDHUMANUNDEFINED4-(4-Chloro-phenyl)-1-(1H-indol-3-ylmethyl)-piperidin-4-ol1520.7Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
55507D4UNDEFINEDHUMANUNDEFINEDL-7458700.43Sikazwe DM et al., 2009Jan 15, 2025Jan 15, 2025
555085-HT2AUNDEFINEDUNDEFINEDUNDEFINED1-Methoxy-4-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.2.0*2,6*]undec-8-ene-3,5-dione1390Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555095-HT2AUNDEFINEDUNDEFINEDUNDEFINEDAcetic acid 4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-8,8-dimethyl-3,5,11-trioxo-4-aza-tricyclo[5.2.2.0*2,6*]undec-1-yl ester770Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555105-HT2AUNDEFINEDUNDEFINEDUNDEFINED1-Ethoxy-4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-4-aza-tricyclo[5.2.2.0*2,6*]undecane-3,5,8-trione2790Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555115-HT2AUNDEFINEDUNDEFINEDUNDEFINEDBUSPIRONE851Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555125-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate737Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555135-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate6019Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555145-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate965Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555155-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[4-(4-Phenylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate286Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555165-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate170Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555175-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[4-(4-Benzylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate9720Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555185-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione522Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555195-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione3380Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555205-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione577Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555215-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[4-(4-Phenylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione181Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555225-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)] undecane-3,5,8-trione102Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555235-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[4-(4-Benzylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione2092Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555245-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate1024Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555255-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate575Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555265-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione429Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555275-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione292Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555285-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate681Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555295-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Pyridyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate1836Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555305-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propoxy]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate375Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555315-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate1073Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555325-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate376Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555335-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione637Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555345-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propoxy]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione300Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555355-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione910Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555365-HT2AUNDEFINEDUNDEFINEDUNDEFINED4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione110Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555375-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione1516Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555385-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione25Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555395-HT1AUNDEFINEDRATUNDEFINED4-[4-(4-Benzylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate1416Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555405-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate286Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555415-HT1AUNDEFINEDRATUNDEFINED4-[4-(4-Phenylpiperazin-1-yl)butyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate34Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555425-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate97Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555435-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(2-Pyrimidyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate800Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555445-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-ylacetate10Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555455-HT1AUNDEFINEDRATUNDEFINED1-Methoxy-4-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]-propoxy}-4-aza-tricyclo[5.2.2.0*2,6*]undec-8-ene-3,5-dione31Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555465-HT1AUNDEFINEDRATUNDEFINEDAcetic acid 4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-8,8-dimethyl-3,5,11-trioxo-4-aza-tricyclo[5.2.2.0*2,6*]undec-1-yl ester22Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555475-HT1AUNDEFINEDRATUNDEFINED1-Ethoxy-4-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-4-aza-tricyclo[5.2.2.0*2,6*]undecane-3,5,8-trione26Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555485-HT1AUNDEFINEDRATUNDEFINEDBUSPIRONE3.8Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555495-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(2-Pyridyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione202Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555505-HT1AUNDEFINEDRATUNDEFINED4-[4-(4-Phenylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione50Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555515-HT1AUNDEFINEDRATUNDEFINED4-{4-[4-(4-Fluorophenyl)piperazin-1-yl]butyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)] undecane-3,5,8-trione521Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555525-HT1AUNDEFINEDRATUNDEFINED4-[4-(4-Benzylpiperazin-1-yl)butyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione2730Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555535-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate35Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555545-HT1AUNDEFINEDRATUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propyl]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate294Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555555-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propyl}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione44Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555565-HT1AUNDEFINEDRATUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propyl]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione344Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555575-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate27Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555585-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Pyridyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate200Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555595-HT1AUNDEFINEDRATUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propoxy]-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate115Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555605-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate80Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555615-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-8,11-dimethyl-3,5-dioxo-4-azatricyclo[5.2.2.0(2,6)]undec-8-en-1-yl acetate37Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555625-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Methoxyphenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione124Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555635-HT1AUNDEFINEDRATUNDEFINED4-[3-(4-Phenylpiperazin-1-yl)propoxy]-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione616Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555645-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(2-Fluorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione331Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
555655-HT1AUNDEFINEDRATUNDEFINED4-{3-[4-(3-Chlorophenyl)piperazin-1-yl]propoxy}-1,11-dimethyl-4-azatricyclo[5.2.2.0(2,6)]undecane-3,5,8-trione92Bojarski AJ et al., 2009Jan 15, 2025Jan 15, 2025
55566Beta2UNDEFINEDHUMANUNDEFINED(6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one320Kern C et al., 2009Jan 15, 2025Jan 28, 2025
55567Beta2UNDEFINEDHUMANUNDEFINED(6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one580Kern C et al., 2009Jan 15, 2025Jan 28, 2025
55568Beta2UNDEFINEDHUMANUNDEFINEDClenbuterol570Kern C et al., 2009Jan 15, 2025Jan 28, 2025
55569Beta2UNDEFINEDHUMANUNDEFINED4-(1-hydroxy-2-(4-(4-hydroxyphenyl)butan-2-ylamino)ethyl)phenol180Kern C et al., 2009Jan 15, 2025Jan 28, 2025
55570Beta2UNDEFINEDHUMANUNDEFINEDAlbuterol510Kern C et al., 2009Jan 15, 2025Jan 28, 2025
55571Beta2UNDEFINEDHUMANUNDEFINEDICI 118,5511Kern C et al., 2009Jan 15, 2025Jan 28, 2025
55572MORUNDEFINEDHUMANUNDEFINED(6S,7S)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride7000Kern C et al., 2009Jan 15, 2025Jan 15, 2025
55573MORUNDEFINEDHUMANUNDEFINED(6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride>10000Kern C et al., 2009Jan 15, 2025Jan 15, 2025
55574MORUNDEFINEDHUMANUNDEFINED(6R,7R)-4,5,6,7-Tetrahydro-7-hydroxy-6-[(1-methylethyl)amino]imidazo[4,5,1-jk][1]benzazepin-2(1H)-one Hydrochloride>10000Kern C et al., 2009Jan 15, 2025Jan 15, 2025
55575MORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone2.5Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55576MORUNDEFINEDHUMANUNDEFINED14-O-phenylpropylnaltrexone0.34Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55577MORUNDEFINEDHUMANUNDEFINEDclocinnamox3Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55578MORUNDEFINEDHUMANUNDEFINEDMC-CAM4.8Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55579MORUNDEFINEDHUMANUNDEFINEDNaltrexone0.2Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55580MORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-methylcinnamoyloxy-7,8-dihydrocodeinone4.2Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55581MORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-chlorocinnamoyloxy-7,8-dihydrocodeinone3.5Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55582DORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone180Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55583DORUNDEFINEDHUMANUNDEFINED14-O-phenylpropylnaltrexone0.48Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55584DORUNDEFINEDHUMANUNDEFINEDclocinnamox2.7Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55585DORUNDEFINEDHUMANUNDEFINEDMC-CAM4.8Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55586DORUNDEFINEDHUMANUNDEFINEDNaltrexone11Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55587DORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-methylcinnamoyloxy-7,8-dihydrocodeinone270Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55588DORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-chlorocinnamoyloxy-7,8-dihydrocodeinone110Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55589KORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-cinnamoyloxy-7,8-dihydrocodeinone4.3Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55590KORUNDEFINEDHUMANUNDEFINED14-O-phenylpropylnaltrexone0.41Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55591KORUNDEFINEDHUMANUNDEFINEDclocinnamox1.4Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55592KORUNDEFINEDHUMANUNDEFINEDMC-CAM16Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55593KORUNDEFINEDHUMANUNDEFINEDNaltrexone0.4Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55594KORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-methylcinnamoyloxy-7,8-dihydrocodeinone36Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55595KORUNDEFINEDHUMANUNDEFINEDN-Cyclopropylmethyl-14beta-4'-chlorocinnamoyloxy-7,8-dihydrocodeinone52Moynihan H et al., 2009Jan 15, 2025Jan 15, 2025
55596SLC6A3UNDEFINEDHUMANUNDEFINED2-(Aminoethyl)-5-(2'-methoxy-5'-fluorophenethyl)tetrahydrofuran6500Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55597SLC6A3UNDEFINEDHUMANUNDEFINED2-Aminoethyl-5-(3'-(2''-methoxy-5''-fluorophenyl)-1'-propyl)tetrahydrofuran7307Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55598SLC6A3UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55599SLC6A3UNDEFINEDHUMANUNDEFINEDcis-(+/-)-2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55600SLC6A3UNDEFINEDHUMANUNDEFINEDcis-(+/-)-2-{5-[3-(5-fluoro-2-methoxyphenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl]-4,5,8,8a-tetrahydro-2H-phthalazin-1-one2478Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55601SLC6A3UNDEFINEDHUMANUNDEFINEDCis-(+/-)-2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-propyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one5340Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55602SLC6A3UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester371Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55603SLC6A3UNDEFINEDHUMANUNDEFINEDFLUOXETINE6670Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55604SLC6A3UNDEFINEDHUMANUNDEFINED2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-methyl-amine>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55605SLC6A4UNDEFINEDHUMANUNDEFINED2-(Aminoethyl)-5-(2'-methoxy-5'-fluorophenethyl)tetrahydrofuran2.1Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55606SLC6A4UNDEFINEDHUMANUNDEFINED2-Aminoethyl-5-(3'-(2''-methoxy-5''-fluorophenyl)-1'-propyl)tetrahydrofuran1.1Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55607SLC6A4UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55608SLC6A4UNDEFINEDHUMANUNDEFINEDcis-(+/-)-2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55609SLC6A4UNDEFINEDHUMANUNDEFINEDcis-(+/-)-2-{5-[3-(5-fluoro-2-methoxyphenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl]-4,5,8,8a-tetrahydro-2H-phthalazin-1-one156Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55610SLC6A4UNDEFINEDHUMANUNDEFINEDCis-(+/-)-2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-propyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one194Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55611SLC6A4UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester276Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55612SLC6A4UNDEFINEDHUMANUNDEFINEDFLUOXETINE1.1Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55613SLC6A4UNDEFINEDHUMANUNDEFINED2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-methyl-amine21.2Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55614SLC6A2UNDEFINEDHUMANUNDEFINED2-(Aminoethyl)-5-(2'-methoxy-5'-fluorophenethyl)tetrahydrofuran2440Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55615SLC6A2UNDEFINEDHUMANUNDEFINED2-Aminoethyl-5-(3'-(2''-methoxy-5''-fluorophenyl)-1'-propyl)tetrahydrofuran>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55616SLC6A2UNDEFINEDHUMANUNDEFINED4-(3,4-dimethoxy-phenyl)-4a,5,8,8a-tetrahydro-2Hphthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55617SLC6A2UNDEFINEDHUMANUNDEFINEDcis-(+/-)-2-(5-Bromo-pentyl)-4-(3,4-dimethoxy-phenyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55618SLC6A2UNDEFINEDHUMANUNDEFINEDcis-(+/-)-2-{5-[3-(5-fluoro-2-methoxyphenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl]-4,5,8,8a-tetrahydro-2H-phthalazin-1-one1748Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55619SLC6A2UNDEFINEDHUMANUNDEFINEDCis-(+/-)-2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-propyl]-tetrahydro-furan-2-yl}-ethylamine)-pentyl-4a,5,8,8a-tetrahydro-2H-phthalazin-1-one7441Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55620SLC6A2UNDEFINEDHUMANUNDEFINED3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2-carboxylic acid methyl ester1115Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55621SLC6A2UNDEFINEDHUMANUNDEFINEDFLUOXETINE1560Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55622SLC6A2UNDEFINEDHUMANUNDEFINED2-{5-[3-(5-Fluoro-2-methoxy-phenyl)-ethyl]-tetrahydro-furan-2-yl}-ethylamine)-methyl-amine>10000Cashman JR et al., 2009Jan 15, 2025Jan 15, 2025
55623CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Ethoxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride0.035Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55624CHRNA4UNDEFINEDRATUNDEFINEDcis-3-(5-Propyloxy-3-pyridinyl)-3,7-diazabicyclo[3.3.0]octane Semifumarate0.041Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55625CHRNA4UNDEFINEDRATUNDEFINEDEpibatidine0.047Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55626CHRNA4UNDEFINEDRATUNDEFINEDcis-3-(5-Isopropyloxy-3-pyridinyl)-3,7-diazabicyclo[3.3.0]octane Semi(fumarate)0.051Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55627CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-(Benzyloxy)pyridin-3-yl)octahydropyrrolo[3,4-c]pyrrole0.058Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55628CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Bromopyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate0.06Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55629CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Methoxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride0.081Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55630CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(3-Pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride0.12Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55631CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Phenylpyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bistrifluoroacetate0.16Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55632CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(6-Chloro-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Hydrochloride0.2Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55633CHRNA4UNDEFINEDRATUNDEFINEDcis-5-(6-Bromo-pyridin-3-yl)-hexahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate0.28Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55634CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Hydroxy-3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride0.75Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55635CHRNA4UNDEFINEDRATUNDEFINEDNicotine0.94Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55636CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(3-pyridinyl)octahydropyrrolo[3,4-c]pyrrole Dihydrochloride26Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55637CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(6-Chloro-3-pyridinyl)-5-methyloctahydropyrrolo[3,4-c]-pyrrole38Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55638CHRNA4UNDEFINEDRATUNDEFINEDcis-4-(5-(Hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)pyridin-3-yl)morpholine Sesqui-fumarate47Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55639CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Phenylpyridin-3-yl)-5-methyl-octahydro-pyrrolo[3,4-c]-pyrrole Sesqui-fumarate51Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55640CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(6-Phenyl-pyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate96Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55641CHRNA4UNDEFINEDRATUNDEFINEDcis-5-(6-Chloropyridin-3-yl)-2,2-dimethyloctahydropyrrolo[3,4-c]-pyrrol-2-ium Iodide210Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55642CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(Pyridin-2-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate260Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55643CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(6-m-tolyl-pyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-L-tartrate750Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55644CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-[6-(3-nitrophenyl)-pyridin-3-yl]-octahydro-pyrrolo[3,4-c]pyrrole p-toluenesulfonate2600Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55645CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(6-Phenyl-pyridazin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate5320Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55646CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(6-Biphenyl-3-yl-pyridin-3-yl)-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole p-Toluenesulfonate9800Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55647CHRNA4UNDEFINEDRATUNDEFINEDcis-3-[6-(5-Methyl-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl)-pyridazin-3-yl]-phenol dihydrochloride>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55648CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(6-phenyl-pyridin-3-yl)-octahydro-pyrrolo[3,4-c]pyrrole L-Tartrate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55649CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(Pyridin-4-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55650CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Biphenyl-4-yl-octahydro-pyrrolo[3,4-c]pyrrole Trifluoroacetate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55651CHRNA4UNDEFINEDRATUNDEFINEDcis-5-(6-Phenylpyridazin-3-yl)-2,2-dimethyloctahydropyrrolo[3,4-c]pyrrol-2-ium Iodide>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55652CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(6-(2-methylphenyl)pyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole Bis-L-tartrate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55653CHRNA4UNDEFINEDRATUNDEFINEDcis-4-[6-(5-Methyl-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl)-pyridazin-3-yl]-phenol Bis-p-toluenesulfonate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55654CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(5-Phenyl-pyridin-2-yl)-octahydro-pyrrolo[3,4-c]pyrrole Bis-trifluoroacetate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55655CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(5-phenyl-pyridin-2-yl)-octahydro-pyrrolo[3,4-c]pyrrole 4-Toluenesulfonate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55656CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Biphenyl-4-yl-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole Dihydrochloride>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55657CHRNA4UNDEFINEDRATUNDEFINEDcis-2-(6-Phenyl-pyridazin-3-yl)-5-methyloctahydro-pyrrolo[3,4-c]-pyrrole>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55658CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Ethyl-5-(6-phenyl-pyridazin-3-yl)-octahydro-pyrrolo[3,4-c]-pyrrole Bis-p-toluenesulfonate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55659CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(6-(4-methylphenyl)pyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole Dihydrochloride>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55660CHRNA4UNDEFINEDRATUNDEFINEDcis-2-Methyl-5-(6-(3-methylphenyl)pyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole Dihydrochloride>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55661CHRNA4UNDEFINEDRATUNDEFINEDcis-2-[6-(3,5-(Dimethylphenyl)pyridazin-3-yl]-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole Dihydrochloride>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55662CHRNA4UNDEFINEDRATUNDEFINEDcis-2-[6-(4-Methoxy-phenyl)-pyridazin-3-yl]-5-methyl-octahydro-pyrrolo[3,4-c]pyrrole p-Toluenesulfonate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55663CHRNA4UNDEFINEDRATUNDEFINEDcis-2-[6-(3-Methoxy-phenyl)-pyridin-3-yl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole Bis-L-tartrate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55664CHRNA4UNDEFINEDRATUNDEFINEDcis-5-[6-(5-Methyl-hexahydro-pyrrolo[3,4-c]pyrrol-2-yl)-pyridazin-3-yl]-1H-indole Bis-p-toluenesulfonate>10000Bunnelle WH et al., 2009Jan 15, 2025Jan 15, 2025
55665AChEUNDEFINEDHUMANUNDEFINED1,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene1.63Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55666AChEUNDEFINEDHUMANUNDEFINED1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}-5-methylbenzene7.45Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55667AChEUNDEFINEDHUMANUNDEFINED3,4-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}furan13.27Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55668AChEUNDEFINEDHUMANUNDEFINEDTacrine36Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55669AChEUNDEFINEDHUMANUNDEFINED2,6-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}pyridine0.768Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55670AChEUNDEFINEDHUMANUNDEFINED1,3-bis{[(1,2,3,4-Tetrahydroacridin-9-yl)amino]ethyl}benzene1.718Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55671AChEUNDEFINEDHUMANUNDEFINED1,4-bis[3-(1,2,3,4-Tetrahydroacridin-9-yl)aminopropyl]piperazine0.1359Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55672AChEUNDEFINEDHUMANUNDEFINEDN-(2-Hydroxyethyl)-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine0.1191Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55673AChEUNDEFINEDHUMANUNDEFINEDN-Ethyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine0.162Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55674AChEUNDEFINEDHUMANUNDEFINEDN-Methyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine0.0118Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55675AChEUNDEFINEDHUMANUNDEFINEDN-{4-[(1,2,3,4-Tetrahydroacridin-9-yl)amino]butyl}-N{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}acetamide0.223Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55676AChEUNDEFINEDHUMANUNDEFINEDN-(1,2,3,4-Tetrahydroacridin-9-yl)-N-(3-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)propyl)-1,4-butanediamine2.672Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55677AChEUNDEFINEDHUMANUNDEFINEDN-{4-[(1,2,3, 4-Tetrahydroacridin-9-yl)amino]butyl}-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)sulfanyl]propyl}acetamide20.877Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55678AChEUNDEFINEDHUMANUNDEFINED6-(1,2,3,4-Tetrahydro-acridin-9-ylamino)-hexanoic acid [3-(acridin-9-ylsulfanyl)-propyl]-amide5.15Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55679AChEUNDEFINEDHUMANUNDEFINEDN-[3-(Acridin-9-ylsulfanyl)-propyl]-N''-(1,2,3,4-tetrahydro-acridin-9-yl)-pentane-1,5-diamine3.99Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55680AChEUNDEFINEDHUMANUNDEFINED5-(1,2,3,4-Tetrahydro-acridin-9-ylamino)-pentanoic acid [3-(acridin-9-ylsulfanyl)-propyl]-amide13.37Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55681AChEUNDEFINEDHUMANUNDEFINEDN-Methyl-N'-(1,2,3,4-tetrahydro-acridin-9-yl)-N-[3-(1,2,3,4-tetrahydro-acridin-9-ylamino)-propyl]-propane-1,3-diamine0.54Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55682AChEUNDEFINEDHUMANUNDEFINED(1,2,3,4-Tetrahydro-acridin-9-yl)-[8-(1,2,3,4-tetrahydro-acridin-9-ylsulfanyl)-octyl]-amine27.95Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55683AChEUNDEFINEDHUMANUNDEFINEDN-Allyl-N-(1,2,3,4-tetrahydroacridin-9-yl)-N-{3-[(1,2,3,4-tetrahydroacridin-9-yl)amino]propyl}-1,4-butanediamine0.0847Butini S et al., 2008Jan 15, 2025Jan 28, 2025
55684AChEUNDEFINEDHUMANUNDEFINEDhuprine X0.67Butini S et al., 2008Jan 15, 2025Jan 28, 2025
556855-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[3-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-indol-5-yl)benzamide>10000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556865-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[6-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)hexyl]piperidin-4-yl}-1H-indol-5-yl)benzamide100Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556875-HT1BUNDEFINEDHUMANUNDEFINED5-Hydroxy Tryptamine1.1Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556885-HT1BUNDEFINEDHUMANUNDEFINEDSUMATRIPTAN9.1Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556895-HT1BUNDEFINEDHUMANUNDEFINED4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-benzamide83Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556905-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-{3-[1-({3-[(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)methyl]phenyl}methyl)piperidin-4-yl]-1H-indol-5-yl}benzamide453Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556915-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[(2E)-4-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)but-2-en-1-yl]piperidin-4-yl}-1H-indol-5-yl)benzamide103Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556925-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[2-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethoxy)ethyl]piperidin-4-yl}-1H-indol-5-yl)benzamide32Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556935-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-{3-[1-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethyl)piperidin-4-yl]-1H-indol-5-yl}benzamide18Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556945-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[12-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)dodecyl]piperidin-4-yl}-1H-indol-5-yl)benzamide>10000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556955-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[11-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)undecyl]piperidin-4-yl}-1H-indol-5-yl)benzamide126Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556965-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[10-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)decyl]piperidin-4-yl}-1H-indol-5-yl)benzamide38Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556975-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[9-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)nonyl]piperidin-4-yl}-1H-indol-5-yl)benzamide126Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556985-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[7-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)heptyl]piperidin-4-yl}-1H-indol-5-yl)benzamide79Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
556995-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[3,3,3-trifluoro-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557005-HT1BUNDEFINEDHUMANUNDEFINED10-(4-(5-(4-fluorobenzamido)-1H-indol-3-yl)piperidin-1-yl)decanoic acid1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557015-HT1BUNDEFINEDHUMANUNDEFINEDN-(3-(1-(3-(dimethylamino)propyl)piperidin-4-yl)-1H-indol-5-yl)-4-fluorobenzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557025-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-(1-(2-(piperidin-1-yl)ethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557035-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-(1-(2-hydroxyethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557045-HT1BUNDEFINEDHUMANUNDEFINEDN-(3-(1-benzylpiperidin-4-yl)-1H-indol-5-yl)-4-fluorobenzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557055-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-(1-octylpiperidin-4-yl)-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557065-HT1BUNDEFINEDHUMANUNDEFINEDN-(3-{1-[2-carbamoyl-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)-4-fluorobenzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557075-HT1BUNDEFINEDHUMANUNDEFINEDN1,N3-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)malonamide16Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557085-HT1BUNDEFINEDHUMANUNDEFINED5-amino-3-(N-methylpiperidin-4-yl)-1H-indole353Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557095-HT1BUNDEFINEDHUMANUNDEFINEDN1,N16-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)hexadecanediamide0.81Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557105-HT1BUNDEFINEDHUMANUNDEFINEDN1,N15-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)pentadecanediamide0.58Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557115-HT1BUNDEFINEDHUMANUNDEFINEDN1,N14-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tetradecanediamide0.5Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557125-HT1BUNDEFINEDHUMANUNDEFINEDN1,N13-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)tridecanediamide0.1Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557135-HT1BUNDEFINEDHUMANUNDEFINEDN1,N11-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)undecanediamide1.3Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557145-HT1BUNDEFINEDHUMANUNDEFINEDN1,N10-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)decanediamide0.79Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557155-HT1BUNDEFINEDHUMANUNDEFINEDN1,N8-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)octanediamide1.3Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557165-HT1BUNDEFINEDHUMANUNDEFINEDN1,N5-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)glutaramide0.76Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557175-HT1BUNDEFINEDHUMANUNDEFINED2-(5-{4-[3-(2-Amino-ethyl)-1H-indol-5-yloxymethyl]-benzyloxy}-1H-indol-3-yl)-ethylamine0.1Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557185-HT1BUNDEFINEDHUMANUNDEFINED2-(5-{2-[8-(4-Methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethoxy}-1H-indol-3-yl)-ethylamine0.76Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557195-HT1BUNDEFINEDHUMANUNDEFINEDC-[3-(2-Dimethylamino-ethyl)-1H-indol-5-yl]-N-[4-({[3-(2-dimethylamino-ethyl)-1H-indol-5-ylmethanesulfonyl]-methyl-amino}-methyl)-benzyl]-N-methyl-methanesulfonamide0.64Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557205-HT1BUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)benzamide>10000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557215-HT1DUNDEFINEDHUMANUNDEFINED(S)-1-{2-[4-(4-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-isochroman-6-carboxylic acid methylamide0.9Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557225-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)benzamide219Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557235-HT1DUNDEFINEDHUMANUNDEFINED5-Hydroxy Tryptamine0.5Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557245-HT1DUNDEFINEDHUMANUNDEFINEDSUMATRIPTAN1.2Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557255-HT1DUNDEFINEDHUMANUNDEFINED4-Fluoro-N-[3-(1-methyl-piperidin-4-yl)-1H-indol-5-yl]-benzamide137Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557265-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[3,3,3-trifluoro-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557275-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-{3-[1-({3-[(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)methyl]phenyl}methyl)piperidin-4-yl]-1H-indol-5-yl}benzamide151Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557285-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[(2E)-4-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)but-2-en-1-yl]piperidin-4-yl}-1H-indol-5-yl)benzamide24Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557295-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[2-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethoxy)ethyl]piperidin-4-yl}-1H-indol-5-yl)benzamide3.9Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557305-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-{3-[1-(2-{2-[2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethoxy]ethoxy}ethyl)piperidin-4-yl]-1H-indol-5-yl}benzamide1.5Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557315-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[12-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)dodecyl]piperidin-4-yl}-1H-indol-5-yl)benzamide13Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557325-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[11-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)undecyl]piperidin-4-yl}-1H-indol-5-yl)benzamide13Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557335-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[10-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)decyl]piperidin-4-yl}-1H-indol-5-yl)benzamide13Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557345-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[9-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)nonyl]piperidin-4-yl}-1H-indol-5-yl)benzamide1Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557355-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[7-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)heptyl]piperidin-4-yl}-1H-indol-5-yl)benzamide0.3Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557365-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[6-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)hexyl]piperidin-4-yl}-1H-indol-5-yl)benzamide0.6Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557375-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-{1-[3-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)propyl]piperidin-4-yl}-1H-indol-5-yl)benzamide79Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557385-HT1DUNDEFINEDHUMANUNDEFINED10-(4-(5-(4-fluorobenzamido)-1H-indol-3-yl)piperidin-1-yl)decanoic acid1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557395-HT1DUNDEFINEDHUMANUNDEFINEDN-(3-(1-(3-(dimethylamino)propyl)piperidin-4-yl)-1H-indol-5-yl)-4-fluorobenzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557405-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-(1-(2-(piperidin-1-yl)ethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557415-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-(1-(2-hydroxyethyl)piperidin-4-yl)-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557425-HT1DUNDEFINEDHUMANUNDEFINEDN-(3-(1-benzylpiperidin-4-yl)-1H-indol-5-yl)-4-fluorobenzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557435-HT1DUNDEFINEDHUMANUNDEFINED4-fluoro-N-(3-(1-octylpiperidin-4-yl)-1H-indol-5-yl)benzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557445-HT1DUNDEFINEDHUMANUNDEFINEDN-(3-{1-[2-carbamoyl-2-(4-{5-[(4-fluorobenzene)amido]-1H-indol-3-yl}piperidin-1-yl)ethyl]piperidin-4-yl}-1H-indol-5-yl)-4-fluorobenzamide1000Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557455-HT1DUNDEFINEDHUMANUNDEFINEDN1,N3-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)malonamide3.4Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557465-HT1DUNDEFINEDHUMANUNDEFINED5-amino-3-(N-methylpiperidin-4-yl)-1H-indole39.6Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557475-HT1DUNDEFINEDHUMANUNDEFINEDN1,N16-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)hexadecanediamide11.3Choi SK et al., 2008Jan 15, 2025Jan 15, 2025
557485-HT1DUNDEFINEDHUMANUNDEFINEDN1,N15-bis(3-(1-methylpiperidin-4-yl)-1H-indol-5-yl)pentadecanediamide2.3Choi SK et al., 2008Jan 15, 2025Jan 15, 2025