70749 DAT CLONED HUMAN 3H-Mazindol oxycodone >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 15, 2025
70750 DAT CLONED HUMAN 3H-Mazindol 3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 15, 2025
70751 DAT CLONED HUMAN 3H-Mazindol Morphine >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 15, 2025
70752 DAT CLONED HUMAN 3H-Mazindol hydromorphone >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 15, 2025
70753 DAT CLONED HUMAN 3H-Mazindol Hydrocodone >10000 Olson KM, et al., 2019 Jan 15, 2025 Jan 15, 2025
70754 DAT CLONED HUMAN 3H-Mazindol BUPRENORPHINE 2000 Olson KM, et al., 2019 Jan 15, 2025 Jan 15, 2025
70755 5-HT1A ?CLONED ? HUMAN 3H-8-OH-DPAT 1-Butanoyl-d-lysergic acid diethylamide 345 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70756 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-Butanoyl-d-lysergic acid diethylamide 87.7 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70757 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-Butanoyl-d-lysergic acid diethylamide 20.8 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70758 5-HT1A ?CLONED ? HUMAN 3H-8-OH-DPAT 1-propionyl-lysergic acid diethylamide 637 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70759 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-propionyl-lysergic acid diethylamide 196 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70760 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-propionyl-lysergic acid diethylamide 13 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70761 5-HT1A ?CLONED ? HUMAN 3H-8-OH-DPAT 1-Acetyl-D-lysergic acid diethylamide 1054 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70762 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 1-Acetyl-D-lysergic acid diethylamide 174 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70763 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 1-Acetyl-D-lysergic acid diethylamide 10.2 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70764 5-HT1A ?CLONED ? HUMAN 3H-8-OH-DPAT D-lysergic acid diethylamide (LSD) 9.5 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70765 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin D-lysergic acid diethylamide (LSD) 14.7 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70766 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE D-lysergic acid diethylamide (LSD) 45.3 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70767 5-HT1B ?CLONED ? HUMAN 3H-GR-125743 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 1463 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70768 5-HT1D ?CLONED ? HUMAN 3H-GR125743 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 295 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70769 5-HT2B ?CLONED ? HUMAN 3H- LSD 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 3.5 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70770 5-HT5A ?CLONED ? HUMAN 3H- LSD 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 158 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70771 5-HT6 ?CLONED ? HUMAN 3H- LSD 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 607 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70772 5-HT7 ?CLONED ? HUMAN 3H- LSD 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 554 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70773 Alpha1A ?CLONED ? HUMAN 3H-PRAZOSIN 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70774 Alpha1B ?CLONED ? HUMAN 3H-PRAZOSIN 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70775 Alpha1D ?CLONED ? HUMAN 3H-PRAZOSIN 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70776 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 537 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70777 Alpha2B ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 2656 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70778 Alpha2C ?CLONED ? HUMAN 3H-RAUWOLSCINE 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 812 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70779 Beta 1 ?CLONED ? HUMAN 125I-Pindolol 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70780 Beta 2 ?CLONED ? HUMAN 3H-CGP-12177 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 15, 2025
70781 Beta3 ?CLONED ? HUMAN 3H-CGP12177 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70782 D1 ?CLONED ? HUMAN 3H-SCH23390 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 1167 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70783 D2 ?CLONED ? HUMAN 3H-Methylspiperone 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70784 D3 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 352 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70785 D4 ?CLONED ? HUMAN 3H-N-Methylspiperone 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 2271 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70786 D5 ?CLONED ? HUMAN 3H-SCH23390 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70787 H1 ?CLONED ? HUMAN 3H-PYRILAMINE 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70788 5-HT1D ?CLONED ? HUMAN 3H-TIOTIDINE 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) 842 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70789 H3 ?CLONED GUINEA PIG 3H-Alpha-methylhistamine 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70790 H4 ?CLONED ? HUMAN 3H-Histamine 1-butanoyl-D-lysergic acid diethylamide (1B-LSD) >10000 Halberstadt AL, et al., 2019 Jan 15, 2025 Jan 28, 2025
70791 DAT STRIATUM RAT 3H-dopamine D-578 16.2 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70792 NET CEREBRAL CORTEX RAT 3H-dopamine D-578 3.23 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70793 SERT CEREBRAL CORTEX RAT 3H-5-HT D-578 16.2 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70794 DAT STRIATUM RAT 3H-dopamine FLUOXETINE 1092 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70795 SERT CEREBRAL CORTEX RAT 3H-5-HT FLUOXETINE 12.2 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70796 NET CEREBRAL CORTEX RAT 3H-dopamine FLUOXETINE 770 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70797 DAT STRIATUM RAT 3H-dopamine Reboxetine 2908 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70798 SERT CEREBRAL CORTEX RAT 3H-5HT Reboxetine 503 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70799 NET CEREBRAL CORTEX RAT 3H-dopamine Reboxetine 0.79 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70800 DAT STRIATUM RAT 3H-dopamine DESIPRAMINE 1567 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70801 SERT CEREBRAL CORTEX RAT 3H-5HT DESIPRAMINE 106 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70802 NET CEREBRAL CORTEX RAT 3H-dopamine DESIPRAMINE 1.3 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70803 DAT STRIATUM RAT 3H-dopamine IMIPRAMINE 1696 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70804 SERT CEREBRAL CORTEX RAT 3H-5HT IMIPRAMINE 20 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70805 NET CEREBRAL CORTEX RAT 3H-dopamine IMIPRAMINE 170 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70806 DAT HEK293 cells HUMAN 3H-dopamine D-578 29.6 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70807 SERT HEK293 cells HUMAN 3H-Serotonin D-578 20.6 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70808 NET HEK293 cells HUMAN 3H-dopamine D-578 6.1 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70809 SERT HEK293 cells HUMAN 3H-5HT FLUOXETINE 14.4 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70810 NET HEK293 cells HUMAN 3H-dopamine DESIPRAMINE 0.86 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70811 SERT HEK293 cells HUMAN 3H-5HT CITALOPRAM 3.66 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70812 D2 CLONED HUMAN 3H-N-Methylspiporone D-578 773 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70813 D3 CLONED HUMAN 3H-N-Methylspiporone D-578 2615 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70814 5-HT1D CLONED HUMAN 3H-GR-125743 D-578 702 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70815 5-HT2A CLONED HUMAN 3H-KETANSERIN D-578 1639 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70816 5-HT2B CLONED HUMAN 3H-LSD D-578 425 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70817 5-HT2C CLONED HUMAN 3H-MESULERGINE D-578 73 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70818 Alpha2C CLONED HUMAN 3H-CLONIDINE D-578 2014 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70819 Beta2 CLONED HUMAN 125I-Iodopindolol D-578 >10000 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70820 Beta3 CLONED HUMAN 125I-Iodopindolol D-578 2703 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70821 KOR CLONED HUMAN 3H-Bremazocine D-578 1387 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70822 5-HT1D CLONED HUMAN 3H-Tiotodine D-578 42 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70823 M1 CLONED HUMAN 3H-QNB D-578 >10000 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70824 M4 CLONED HUMAN 3H-QNB D-578 >10000 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70825 M5 CLONED HUMAN 3H-QNB D-578 >10000 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70826 mGluR5 CLONED HUMAN 3H-MPEP D-578 600 Dutta A, et al. 2019 Jan 15, 2025 Jan 28, 2025
70827 OT CLONED HUMAN 3H-Oxytocin D-578 >10000 Dutta A, et al. 2019 Jan 15, 2025 Jan 15, 2025
70828 TMEM97 Sf9 Insect 3H-DTG DTG 19.6 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70829 TMEM97 Sf9 Insect 3H-DTG HALOPERIDOL 54.1 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70830 TMEM97 Sf9 Insect 3H-DTG PB-28 2 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70831 TMEM97 Sf9 Insect 3H-DTG PENTAZOCINE (+) 2467 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70832 TMEM97 Sf9 Insect 3H-DTG SKF 10,047 (+) >10000 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70833 TMEM97 Sf9 Insect 3H-DTG SAS-1121 25.2 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70834 TMEM97 Sf9 Insect 3H-DTG Elacridar 6.5 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70835 TMEM97 Sf9 Insect 3H-DTG Ro 48-8071 971 Alon A et al 2017 Jan 15, 2025 Jan 15, 2025
70836 Sigma 2 CLONED HUMAN 3H-DTG DTG 21.2 Alon A et al 2017 Jan 15, 2025 Jan 28, 2025
70837 Sigma 2 CLONED HUMAN 3H-DTG HALOPERIDOL 48.7 Alon A et al 2017 Jan 15, 2025 Jan 28, 2025
70838 Sigma 2 CLONED HUMAN 3H-DTG PB-28 1.8 Alon A et al 2017 Jan 15, 2025 Jan 28, 2025
70839 Sigma 2 CLONED HUMAN 3H-DTG SAS-1121 23.8 Alon A et al 2017 Jan 15, 2025 Jan 28, 2025
70840 Sigma 2 CLONED HUMAN 3H-DTG Elacridar 4.7 Alon A et al 2017 Jan 15, 2025 Jan 28, 2025
70841 Sigma 2 CLONED HUMAN 3H-DTG Ro 48-8071 817 Alon A et al 2017 Jan 15, 2025 Jan 28, 2025
70842 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 2-(4-bromo-2,5-dimethoxyphenyl)ethanamine 0.21 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70843 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)ethanamine 2.5 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70844 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 2-(4-bromo-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 3.3 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70845 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 39 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70846 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin N-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride (3) 1.5 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70847 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE N-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride 18 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70848 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 2-(4-chloro-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 7.7 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70849 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 2-(4-chloro-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 67 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70850 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 2-(2,5-dimethoxy-4-nitrophenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 30 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70851 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-nitrophenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride 250 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70852 5-HT2A ?CLONED ? HUMAN 3H- Ketanserin 4-(2-((4-fluoro-2-methoxybenzyl)amino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride 120 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70853 5-HT2C ?CLONED ? HUMAN 3H-MESULERGINE 4-(2-((4-fluoro-2-methoxybenzyl)amino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride >10000 Petersen IN et al 2016 Jan 15, 2025 Jan 15, 2025
70854 Sigma 2 ?CLONED ? HUMAN 3H-DTG (6S,7R)-7-(1H-Indol-3-yl)-4-methylene-1-azaspiro[5.5] undecane 463 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70855 Sigma 1 ?CLONED ? HUMAN 3H-Pentazocine(+) (6S,7R)-7-(1H-Indol-3-yl)-4-methylene-1-azaspiro[5.5] undecane 1446 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70856 Sigma 2 ?CLONED ? HUMAN 3H-DTG (6R,7S)-1-benzyl-4-methylene-7-phenyl-1,9-diazaspiro[5.5] undecane 502 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70857 Sigma 1 ?CLONED ? HUMAN 3H-Pentazocine(+) (6R,7S)-1-benzyl-4-methylene-7-phenyl-1,9-diazaspiro[5.5] undecane 542 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70858 Sigma 2 ?CLONED ? HUMAN 3H-DTG ((4R,6S,7R)-7-phenyl-1-azaspiro[5.5]undecan-4-yl)methanol 452 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70859 Sigma 1 ?CLONED ? HUMAN 3H-Pentazocine(+) ((4R,6S,7R)-7-phenyl-1-azaspiro[5.5]undecan-4-yl)methanol 2257 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70860 Sigma 2 ?CLONED ? HUMAN 3H-DTG (4aS,14bR)-13-methoxy-6-methylene-1,2,3,4,5,6,7,8,10,14bdecahydropyrido[2,1-e]phenanthridine 152 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70861 Sigma 1 ?CLONED ? HUMAN 3H-Pentazocine(+) (4aS,14bR)-13-methoxy-6-methylene-1,2,3,4,5,6,7,8,10,14bdecahydropyrido[2,1-e]phenanthridine 8 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 15, 2025
70862 Sigma 2 ?CLONED ? HUMAN 3H-DTG (3aS,13bR)-12-methoxy-5-methylene-2,3,4,5,6,7,9,13boctahydro-1H-cyclopenta[c]pyrido[1,2-b]isoquinoline 308 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70863 Sigma 1 ?CLONED ? HUMAN 3H-Pentazocine(+) (3aS,13bR)-12-methoxy-5-methylene-2,3,4,5,6,7,9,13boctahydro-1H-cyclopenta[c]pyrido[1,2-b]isoquinoline 45 Lepovitz L, et al., 2019 Jan 15, 2025 Jan 28, 2025
70864 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine 1138 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70865 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine 434 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70866 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine 2313 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70867 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine 450 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70868 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70869 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70870 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70871 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine 414 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70872 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine 552 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70873 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine 422 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70874 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine 2681 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70875 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine 102 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70876 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine 3044 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70877 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70878 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70879 5-HT2B CLONED HUMAN 3H-LSD (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine 106 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70880 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine 343 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70881 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine 338 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70882 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70883 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine 32 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70884 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70885 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70886 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine >10000 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70887 5-HT2C CLONED HUMAN 3H-MESULERGINE (R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine 24 Xu Y et al., 2019 Jan 15, 2025 Jan 15, 2025
70888 MOR Ovary HAMSTER 125i-IBNtxA Morphine 5 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70889 MOR Ovary HAMSTER 125i-IBNtxA Butyrylfentanyl 18 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70890 MOR Ovary HAMSTER 125i-IBNtxA U-47700 57 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70891 MOR Ovary HAMSTER 125i-IBNtxA MT-45 44 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70892 DOR Ovary HAMSTER 125i-IBNtxA Butyrylfentanyl 286 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70893 DOR Ovary HAMSTER 125i-IBNtxA U-47700 1105 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70894 DOR Ovary HAMSTER 125i-IBNtxA MT-45 606 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70895 KOR Ovary HAMSTER 125i-IBNtxA Butyrylfentanyl 3174 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70896 KOR Ovary HAMSTER 125i-IBNtxA U-47700 653 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70897 KOR Ovary HAMSTER 125i-IBNtxA MT-45 204 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70898 MOR CLONED HUMAN 3H-DAMGO Morphine 3.5 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70899 MOR CLONED HUMAN 3H-DAMGO Butyrylfentanyl 18 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70900 MOR CLONED HUMAN 3H-DAMGO U-47700 39 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70901 MOR CLONED HUMAN 3H-DAMGO MT-45 44 Baumann MH et al 2018 Jan 15, 2025 Jan 28, 2025
70902 D1 ?CLONED ? HUMAN 3H-SCH23390 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 5.7 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70903 D5 ?CLONED ? HUMAN 3H-SCH23390 6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6.7 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70904 D1 ?CLONED ? HUMAN 3H-SCH23390 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione 10 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70905 D5 ?CLONED ? HUMAN 3H-SCH23390 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione 15 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70906 M2 ?CLONED ? HUMAN 3H-QNB 1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione 7700 Martini ML et al 2019 Jan 15, 2025 Jan 15, 2025
70907 D1 ?CLONED ? HUMAN 3H-SCH23390 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 70 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70908 D5 ?CLONED ? HUMAN 3H-SCH23390 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 171 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70909 Alpha2A ?CLONED ? HUMAN 3H-RAUWOLSCINE 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6900 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70910 M2 ?CLONED ? HUMAN 3H-QNB 6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione 6900 Martini ML et al 2019 Jan 15, 2025 Jan 15, 2025
70911 D1 ?CLONED ? HUMAN 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 93 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70912 D5 ?CLONED ? HUMAN 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 185 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70913 D1 ?CLONED ? HUMAN 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 14 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70914 D5 ?CLONED ? HUMAN 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 90 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70915 M3 ?CLONED ? HUMAN 3H-QNB 1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione 4200 Martini ML et al 2019 Jan 15, 2025 Jan 15, 2025
70916 D1 ?CLONED ? HUMAN 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione 5.1 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70917 D5 ?CLONED ? HUMAN 3H-SCH23390 1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione 53 Martini ML et al 2019 Jan 15, 2025 Jan 28, 2025
70918 M3 ?CLONED ? HUMAN 3H-QNB 1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione 4600 Martini ML et al 2019 Jan 15, 2025 Jan 15, 2025
70919 5-HT2B CLONED HUMAN 3H-LSD 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 742 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70920 5-HT2B CLONED HUMAN 3H-LSD (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 840 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70921 5-HT2B CLONED HUMAN 3H-LSD (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 2051 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70922 5-HT2B CLONED HUMAN 3H-LSD (4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 231 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70923 5-HT7 CLONED HUMAN 3H-LSD (4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 2765 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70924 5-HT7 CLONED HUMAN 3H-LSD (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70925 5-HT7 CLONED HUMAN 3H-LSD (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70926 5-HT7 CLONED HUMAN 3H-LSD 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70927 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70928 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70929 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70930 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 3364 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70931 D4 CLONED HUMAN 3H-Methylspiperone 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 1283 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70932 D4 CLONED HUMAN 3H-Methylspiperone (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70933 D4 CLONED HUMAN 3H-Methylspiperone (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70934 D4 CLONED HUMAN 3H-Methylspiperone (4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70935 DAT CLONED HUMAN 3H-WIN35428 (4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70936 DAT CLONED HUMAN 3H-WIN35428 (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70937 DAT CLONED HUMAN 3H-WIN35428 ((S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70938 DAT CLONED HUMAN 3H-WIN35428 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 2562 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70939 5-HT1D CLONED HUMAN 125I-aminopotentidine 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 823 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70940 5-HT1D CLONED HUMAN 125I-aminopotentidine (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70941 5-HT1D CLONED HUMAN 125I-aminopotentidine (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 546 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70942 5-HT1D CLONED HUMAN 125I-aminopotentidine 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70943 KOR CLONED HUMAN 3H-U69593 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70944 KOR CLONED HUMAN 3H-U69593 (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70945 KOR CLONED HUMAN 3H-U69593 (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70946 KOR CLONED HUMAN 3H-U69593 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 1707 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70947 MOR CLONED HUMAN 3H-DAMGO 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70948 MOR CLONED HUMAN 3H-DAMGO (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 1634 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70949 MOR CLONED HUMAN 3H-DAMGO (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 993 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70950 MOR CLONED HUMAN 3H-DAMGO 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 28, 2025
70951 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70952 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70953 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione 58 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70954 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 8.6 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70955 Sigma 2 CLONED HUMAN 3H-DTG 4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione 696 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70956 Sigma 2 CLONED HUMAN 3H-DTG (S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70957 Sigma 2 CLONED HUMAN 3H-DTG (S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70958 Sigma 2 CLONED HUMAN 3H-DTG 4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione >10000 Uprety R. et al., 2019 Jan 15, 2025 Jan 15, 2025
70959 D3 CLONED HUMAN 125I-IABN N-(4-(4-phenylpiperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 8 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70960 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 0.55 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70961 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 8.3 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70962 D3 CLONED HUMAN 125I-IABN N-(4-(4-(4-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 32.7 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70963 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 0.89 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70964 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 3.8 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70965 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 0.44 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70966 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 18 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70967 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 0.47 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70968 D3 CLONED HUMAN 125I-IABN N-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 13.6 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70969 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal 0.68 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70970 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 21.9 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70971 D3 CLONED HUMAN 125I-IABN N-(4-(4-(4-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 36.1 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70972 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 0.25 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70973 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 0.5 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70974 D3 CLONED HUMAN 125I-IABN N-(4-(4-(4-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 2378 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70975 D3 CLONED HUMAN 125I-IABN N-(4-(4-(2-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 1.5 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70976 D3 CLONED HUMAN 125I-IABN N-(4-(4-(3-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 0.41 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70977 D3 CLONED HUMAN 125I-IABN N-(4-(4-(4-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt: 78.3 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70978 D2 CLONED HUMAN 125I-IABN N-(4-(4-phenylpiperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 8434 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70979 D2 CLONED HUMAN 125I-IABN N-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 169 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70980 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70981 D2 CLONED HUMAN 125I-IABN N-(4-(4-(4-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70982 D2 CLONED HUMAN 125I-IABN N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 63.1 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70983 D2 CLONED HUMAN 125I-IABN N-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 757 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70984 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 2049 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70985 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide)benzamide 1832 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70986 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 140 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70987 D2 CLONED HUMAN 125I-IABN N-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 4753 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70988 D2 CLONED HUMAN 125I-IABN N-(4-(4-(2-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 190 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70989 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70990 D2 CLONED HUMAN 125I-IABN N-(4-(4-(4-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70991 D2 CLONED HUMAN 125I-IABN N-(4-(4-(2-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 92.9 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70992 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 743 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70993 D2 CLONED HUMAN 125I-IABN N-(4-(4-(4-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70994 D2 CLONED HUMAN 125I-IABN N-(4-(4-(2-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 261 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70995 D2 CLONED HUMAN 125I-IABN N-(4-(4-(3-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt: 99.7 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70996 D2 CLONED HUMAN 125I-IABN N-(4-(4-(4-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70997 D1 CLONED HUMAN 125I-IABN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70998 D4 CLONED HUMAN 125I-IABN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
70999 D5 CLONED HUMAN 125I-IABN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71000 D5 CLONED HUMAN 125I-IABN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71001 D1 CLONED HUMAN 125I-IABN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71002 D4 CLONED HUMAN 125I-IABN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal 806 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71003 5-HT1A CLONED HUMAN 3H-WAY100635 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide 245 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71004 5-HT1B CLONED HUMAN 3H-GR-125743 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71005 5-HT1D CLONED HUMAN 3H-GR-125743 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71006 5-HT1E CLONED HUMAN 3H-5-HT N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71007 5-HT2A CLONED HUMAN 3H-Ketaserin N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71008 5-HT2B CLONED HUMAN 3H-LSD N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71009 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71010 5-HT3 CLONED HUMAN 3H-MESULERGINE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71011 5-HT3 CLONED HUMAN 3H-GR65630 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71012 5-HT5A CLONED HUMAN 3H-LSD N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71013 5-HT6 CLONED HUMAN 3H-LSD N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71014 5-HT7 CLONED HUMAN 3H-LSD N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71015 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71016 Alpha1B CLONED HUMAN 3H-PRAZOSIN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71017 Alpha1D CLONED HUMAN 3H-PRAZOSIN N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71018 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71019 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71020 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71021 BZP CEREBRAL CORTEX RAT FNZ N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71022 Beta 1 CLONED HUMAN 125I-Pindolol N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71023 Beta3 CLONED HUMAN 125I-Pindolol N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71024 Beta 2 CLONED HUMAN 3H-CGP12177 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71025 KOR CEREBRAL CORTEX RAT 3H-MUSCIMOL N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 27, 2025
71026 H1 CLONED HUMAN 3H-PYRILAMINE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71027 5-HT1D CLONED HUMAN 125I-aminopotentidine N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71028 H3 CLONED HUMAN 3H-Alpha-methylhistamine N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71029 H4 CLONED HUMAN 3H-Histamine N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71030 M1 CLONED HUMAN 3H-QNB N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71031 M2 CLONED HUMAN 3H-QNB N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71032 M3 CLONED HUMAN 3H-QNB N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71033 M4 CLONED HUMAN 3H-QNB N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71034 M5 CLONED HUMAN 3H-QNB N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71035 DOR CLONED HUMAN 3H-DADLE N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71036 KOR CLONED HUMAN 3H-U69593 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71037 MOR CLONED HUMAN 3H-DAMGO N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71038 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71039 Sigma 2 CLONED HUMAN 3H-DTG N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71040 SLC6A3 CLONED HUMAN 3H-WIN 35,428 N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71041 NET CLONED HUMAN 3H-Nisoxetine N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71042 SERT CLONED HUMAN 3H-CITALOPRAM N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71043 5-HT1A CLONED HUMAN 3H-WAY100635 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71044 5-HT1B CLONED HUMAN 3H-GR-125743 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71045 5-HT1D CLONED HUMAN 3H-GR-125743 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71046 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71047 5-HT2B CLONED HUMAN 3H-LSD N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71048 5-HT2C CLONED HUMAN 3H-LSD N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 20 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71049 5-HT3 CLONED HUMAN 3H-GR-65630 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71050 5-HT5A CLONED HUMAN 3H-LSD N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71051 5-HT6 CLONED HUMAN 3H-LSD N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71052 5-HT7 CLONED HUMAN 3H-LSD N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 187 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71053 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71054 Alpha1B CLONED HUMAN 3H-PRAZOSIN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71055 Alpha1D CLONED HUMAN 3H-PRAZOSIN N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71056 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71057 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71058 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71059 BZP CEREBRAL CORTEX RAT FNZ N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 29, 2025
71060 Beta 1 CLONED HUMAN 125I-Pindolol N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71061 Beta3 CLONED HUMAN 125I-Pindolol N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71062 Beta 2 CLONED HUMAN 3H-CGP12177 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71063 KOR CORTICAL MEMBRANES RAT 3H-MUSCIMOL N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 27, 2025
71064 H1 CLONED HUMAN 3H-PYRILAMINE N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 3112 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71065 5-HT1D CLONED HUMAN 125I-aminopotentidine N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71066 H3 CLONED HUMAN 3H-Alpha-methylhistamine N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71067 H4 CLONED HUMAN 3H-Histamine N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71068 M1 CLONED HUMAN 3H-QNB N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71069 M2 CLONED HUMAN 3H-QNB N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71070 M3 CLONED HUMAN 3H-QNB N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71071 M4 CLONED HUMAN 3H-QNB N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71072 M5 CLONED HUMAN 3H-QNB N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71073 DOR CLONED HUMAN 3H-DADLE N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71074 KOR CLONED HUMAN 3H-U69593 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71075 MOR CLONED HUMAN 3H-DAMGO N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71076 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71077 Sigma 2 CLONED HUMAN 3H-DTG N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71078 DAT CLONED HUMAN 3H-WIN 35,428 N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71079 NET CLONED HUMAN 3H-Nisoxetine N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt >10000 Chen PJ et al., 2019 Jan 15, 2025 Jan 15, 2025
71080 SERT CLONED HUMAN 3H-CITALOPRAM N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt 118 Chen PJ et al., 2019 Jan 15, 2025 Jan 28, 2025
71081 Sigma 2 CLONED HUMAN 3H-DTG 4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 5.6 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71082 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 24 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71083 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(4-(4-chloropyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 30 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71084 Sigma 2 CLONED HUMAN 3H-DTG 4-(4-(4-chloropyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 8 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71085 Sigma 2 CLONED HUMAN 3H-DTG 4-(4-(pyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 32 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71086 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(4-(pyridine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 453 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71087 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(4-(pyrimidine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 63 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71088 Sigma 2 CLONED HUMAN 3H-DTG 4-(4-(pyrimidine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one 44 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71089 Sigma 2 CLONED HUMAN 3H-DTG (4-(4-(5-chloropyridin-2-yl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl) butan-1-one oxime 2.7 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71090 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (4-(4-(5-chloropyridin-2-yl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl) butan-1-one oxime 113 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71091 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 1-(4-fluorophenyl)-4-(4-(pyridin-2-yl)-1,4-diazepan-1-yl)butan-1- one oxime 70 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71092 Sigma 2 CLONED HUMAN 3H-DTG 1-(4-fluorophenyl)-4-(4-(pyridin-2-yl)-1,4-diazepan-1-yl)butan-1- one oxime 13 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71093 Sigma 2 CLONED HUMAN 3H-DTG 1-(4-fluorophenyl)-4-(4-(pyrimidin-2-yl)-1,4-diazepan-1-yl)butan1-one oxime 26 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71094 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 1-(4-fluorophenyl)-4-(4-(pyrimidin-2-yl)-1,4-diazepan-1-yl)butan1-one oxime 148 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71095 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-(4-(5-chloropyridin-2-yl)piperazin-1-yl)-1-(4-fluorophenyl)butan1-one 25 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71096 Sigma 2 CLONED HUMAN 3H-DTG 4-(4-(5-chloropyridin-2-yl)piperazin-1-yl)-1-(4-fluorophenyl)butan1-one 8 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71097 Sigma 1 CLONED HUMAN 3H-DTG 1-(5-chloropyridin-2-yl)-4-(4-(4-fluorophenyl)butyl)piperazine 95 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71098 Sigma 2 CLONED HUMAN 3H-Pentazocine(+) 1-(5-chloropyridin-2-yl)-4-(4-(4-fluorophenyl)butyl)piperazine 43 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71099 Sigma 2 CLONED HUMAN 3H-DTG 1-(5-chloropyridin-2-yl)-4-(3-((4-fluorophenyl)thio) propyl)-1,4-diazepane hydrochloride 2 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71100 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 1-(5-chloropyridin-2-yl)-4-(3-((4-fluorophenyl)thio) propyl)-1,4-diazepane hydrochloride 8 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71101 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one 36 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71102 Sigma 2 CLONED HUMAN 3H-DTG 4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one 52 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71103 Sigma 2 CLONED HUMAN 3H-DTG 4-[4-(2-Pyrimidine)piperazin-1-yl]-1-(4-fluorophenyl)butan-1-one 600 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71104 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-[4-(2-Pyrimidine)piperazin-1-yl]-1-(4-fluorophenyl)butan-1-one 1148 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71105 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one 51 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71106 Sigma 2 CLONED HUMAN 3H-DTG 4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one 33 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71107 Sigma 2 CLONED HUMAN 3H-DTG 4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one 5 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71108 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one 42 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71109 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) cis-2,5-Dicarboethoxy-1-[4-chlorophenyl]pyrrolidine 22 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71110 Sigma 2 CLONED HUMAN 3H-DTG cis-2,5-Dicarboethoxy-1-[4-chlorophenyl]pyrrolidine 27 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71111 Sigma 2 CLONED HUMAN 3H-DTG 2-Benzylcarbamyl-5-carboethoxy-1-[4-chlorophenyl]pyrrolidine 18 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71112 Sigma 2 CLONED HUMAN 3H-DTG 2-Benzylcarbamyl-5-carboethoxy-1-[4-chlorophenyl]pyrrolidine 166 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71113 Sigma 2 CLONED HUMAN 3H-DTG 3-Benzyl-8-[4-chlorophenyl]-3,8-diazabicyclo[3.2.1]octane-2,4-dione 29 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71114 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 3-Benzyl-8-[4-chlorophenyl]-3,8-diazabicyclo[3.2.1]octane-2,4-dione 81 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71115 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 3-Benzyl-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 71 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71116 Sigma 2 CLONED HUMAN 3H-DTG 3-Benzyl-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 8 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71117 Sigma 2 CLONED HUMAN 3H-DTG 3-Carboethoxy-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 2.2 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71118 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 3-Carboethoxy-8-phenyl-3, 8-diazabicyclo[3.2.1]octane 57 Al-Ghanim L et al., 2019 Jan 15, 2025 Jan 28, 2025
71119 MT1 HEK293 cells HUMAN 3H-Melatonin N-{2-[(4-methoxypyrimidin-2-yl)(methyl)amino]ethyl}acetamide 489.7 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71120 MT1 HEK293 cells HUMAN 3H-Melatonin rac-N-{[(1R,2R)-2-(3-methoxyphenyl)cyclopropyl]methyl}ethanediamide 3801.8 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71121 MT1 HEK293 cells HUMAN 3H-Melatonin [2-(5-methoxy-1H-indol-3-yl)ethyl]urea 16.5959 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71122 MT1 HEK293 cells HUMAN 3H-Melatonin N-{[1-(2-methylpyrimidin-4-yl)piperidin-2-yl]methyl}acetamide 6025.6 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71123 MT1 HEK293 cells HUMAN 3H-Melatonin 3-cyclopropyl-N-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-amine 8511.38 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71124 MT1 HEK293 cells HUMAN 3H-Melatonin 6-amino-1-[(3-methoxyphenyl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione >10000 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71125 MT1 HEK293 cells HUMAN 3H-Melatonin 1-{6-amino-4-thia-2-azatricyclo[7.3.0.0³,â·]dodeca-1(9),2,5,7-tetraen-5-yl}ethan-1-one >10000 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71126 MT1 HEK293 cells HUMAN 3H-Melatonin 4-(2-chlorobenzoyl)-1H-pyrrole-2-carboxamide >10000 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71127 MT1 HEK293 cells HUMAN 3H-Melatonin methyl 3-amino-6-methoxy-1H-indole-2-carboxylate 9332.54 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71128 MT1 HEK293 cells HUMAN 3H-Melatonin N-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide >10000 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71129 MT1 HEK293 cells HUMAN 3H-Melatonin 6-amino-1-(2-phenylethyl)-2-thioxo-2,3-dihydro-4(1H)-pyrimidinone >10000 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71130 MT2 HEK293 cells HUMAN 3H-Melatonin N-{2-[(4-methoxypyrimidin-2-yl)(methyl)amino]ethyl}acetamide 123.027 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71131 MT2 HEK293 cells HUMAN 3H-Melatonin rac-N-{[(1R,2R)-2-(3-methoxyphenyl)cyclopropyl]methyl}ethanediamide 2754.23 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71132 MT2 HEK293 cells HUMAN 3H-Melatonin [2-(5-methoxy-1H-indol-3-yl)ethyl]urea 23.4423 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71133 MT2 HEK293 cells HUMAN 3H-Melatonin N-{[1-(2-methylpyrimidin-4-yl)piperidin-2-yl]methyl}acetamide 2454.71 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71134 MT2 HEK293 cells HUMAN 3H-Melatonin 3-cyclopropyl-N-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-amine 3548.13 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71135 MT2 HEK293 cells HUMAN 3H-Melatonin 6-amino-1-[(3-methoxyphenyl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione >10000 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71136 MT2 HEK293 cells HUMAN 3H-Melatonin 1-{6-amino-4-thia-2-azatricyclo[7.3.0.0³,â·]dodeca-1(9),2,5,7-tetraen-5-yl}ethan-1-one 5495.41 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71137 MT2 HEK293 cells HUMAN 3H-Melatonin 4-(2-chlorobenzoyl)-1H-pyrrole-2-carboxamide 1230.27 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71138 MT2 HEK293 cells HUMAN 3H-Melatonin methyl 3-amino-6-methoxy-1H-indole-2-carboxylate 2754.23 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71139 MT2 HEK293 cells HUMAN 3H-Melatonin N-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide 4265.79 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71140 MT2 HEK293 cells HUMAN 3H-Melatonin 6-amino-1-(2-phenylethyl)-2-thioxo-2,3-dihydro-4(1H)-pyrimidinone 3235.94 Patel N et al 2020 Jan 15, 2025 Jan 29, 2025
71141 5-HT1A CLONED HUMAN WAY100635 ARIPIPRAZOLE 50.6 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71142 5-HT1A CLONED HUMAN WAY100635 HALOPERIDOL 3600 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71143 5-HT1A CLONED HUMAN WAY100635 CLOZAPINE 140 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71144 5-HT1A CLONED HUMAN WAY100635 SYA013 117 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71145 5-HT1A CLONED HUMAN WAY100635 SYA16263 10.1 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71146 5-HT2A CLONED HUMAN 125I-DOI ARIPIPRAZOLE 80.7 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71147 5-HT2A CLONED HUMAN 125I-DOI HALOPERIDOL 120 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71148 5-HT2A CLONED HUMAN 125I-DOI CLOZAPINE 80.9 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71149 5-HT2A CLONED HUMAN 125I-DOI SYA013 23.6 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71150 5-HT2A CLONED HUMAN 125I-DOI SYA16263 50 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71151 5-HT7 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 10.3 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71152 5-HT7 CLONED HUMAN 3H-LSD HALOPERIDOL 1100 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71153 5-HT7 CLONED HUMAN 3H-LSD CLOZAPINE 66 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71154 5-HT7 CLONED HUMAN 3H-LSD SYA013 78 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71155 5-HT7 CLONED HUMAN 3H-LSD SYA16263 90 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71156 D1 CLONED HUMAN 3H-SCH23390 ARIPIPRAZOLE 1960 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71157 D1 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 120 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71158 D1 CLONED HUMAN 3H-SCH23390 CLOZAPINE 290 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71159 D1 CLONED HUMAN 3H-SCH23390 SYA013 163 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71160 D1 CLONED HUMAN 3H-SCH23390 SYA16263 238 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71161 D2 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 30.3 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71162 D2 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 10.4 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71163 D2 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 130 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71164 D2 CLONED HUMAN 3H-N-Methylspiperone SYA013 43.3 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71165 D2 CLONED HUMAN 3H-N-Methylspiperone SYA16263 124 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71166 D3 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 90.7 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71167 D3 CLONED HUMAN 3H-N-Methylspiperone HALOPERIDOL 20.5 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71168 D3 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 240 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71169 D3 CLONED HUMAN 3H-N-Methylspiperone SYA013 159 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71170 D3 CLONED HUMAN 3H-N-Methylspiperone SYA16263 86 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71171 D4 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 510 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71172 D4 CLONED HUMAN 3H-Methylspiperone HALOPERIDOL 30.3 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71173 D4 CLONED HUMAN 3H-N-Methylspiperone CLOZAPINE 54 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71174 D4 CLONED HUMAN 3H-N-Methylspiperone SYA013 60.6 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71175 D4 CLONED HUMAN 3H-N-Methylspiperone SYA16263 30.5 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71176 D5 CLONED HUMAN 3H-SCH23390 ARIPIPRAZOLE 2590 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71177 D5 CLONED HUMAN 3H-SCH23390 HALOPERIDOL 147 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71178 D5 CLONED HUMAN 3H-SCH23390 CLOZAPINE 454 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71179 D5 CLONED HUMAN 3H-SCH23390 SYA16263 1451 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71180 5-HT2C CLONED HUMAN UNKNOWN ARIPIPRAZOLE 76 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71181 5-HT2C CLONED HUMAN UNKNOWN HALOPERIDOL 4700 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71182 5-HT2C CLONED HUMAN UNKNOWN CLOZAPINE 17 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71183 5-HT2C CLONED HUMAN UNKNOWN SYA013 1425 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71184 5-HT2C CLONED HUMAN UNKNOWN SYA16263 >10000 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71185 H1 CLONED HUMAN 3H-PYRILAMINE ARIPIPRAZOLE 25.1 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71186 H1 CLONED HUMAN 3H-PYRILAMINE HALOPERIDOL 440 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71187 H1 CLONED HUMAN 3H-PYRILAMINE CLOZAPINE 10.8 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71188 H1 CLONED HUMAN 3H-PYRILAMINE SYA013 189 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71189 H1 CLONED HUMAN 3H-PYRILAMINE SYA16263 167 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71190 M1 CLONED HUMAN 3H-QNB ARIPIPRAZOLE 6780 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71191 M1 CLONED HUMAN 3H-QNB HALOPERIDOL 1600 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71192 M1 CLONED HUMAN 3H-QNB CLOZAPINE 1.8 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71193 M1 CLONED HUMAN 3H-QNB SYA013 872 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71194 D2 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 3.3 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71195 D2 CLONED HUMAN 3H-N-Methylspiperone ARIPIPRAZOLE 3.9 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 28, 2025
71196 5-HT1A CLONED HUMAN WAY100635 METHYSERGIDE 25 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71197 5-HT1A CLONED HUMAN WAY100635 SYA16263 1.1 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71198 5-HT1A CLONED HUMAN WAY100635 SYA013 117.4 Bricker B.A., et al. 2019 Jan 15, 2025 Jan 15, 2025
71199 5-HT1A CLONED HUMAN WAY100635 FEMPT 0.2 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71200 5-HT1B CLONED HUMAN 3H-5-CT FEMPT 122.5 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71201 5-HT2A CLONED HUMAN 125I-DOI FEMPT 406 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71202 5-HT2B CLONED HUMAN 3H-LSD FEMPT 12 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71203 5-HT2C CLONED HUMAN UNKNOWN FEMPT 343 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71204 5-HT3 CLONED HUMAN UNKNOWN FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71205 5-HT5A CLONED HUMAN 3H-LSD FEMPT 2340 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71206 5-HT6 CLONED HUMAN 3H-LSD FEMPT 71 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71207 5-HT7 CLONED HUMAN 3H-LSD FEMPT 11 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71208 CLONED HUMAN 3H-NECA FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71209 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71210 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71211 BZP BRAIN RAT UNKNOWN FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 29, 2025
71212 CLONED HUMAN 3H-Nitrendipine FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71213 AMPA CLONED HUMAN 3H-Quisqualate FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 29, 2025
71214 NET CLONED HUMAN 3H-Nisoxetine FEMPT 6980 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71215 CLONED HUMAN 3H-SUBSTANCE P FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71216 Sigma 1 CLONED HUMAN 3H-Pentazocine FEMPT 1014 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71217 CLONED HUMAN 3H-VASOPRESSIN FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71218 V2 CLONED HUMAN 3H-VASOPRESSIN FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 29, 2025
71219 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71220 CB1 CLONED HUMAN 3H-CP55940 FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71221 CB2 CLONED HUMAN 3H-CP55940 FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71222 CLONED HUMAN 3H-PRAZOSIN FEMPT 180 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71223 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE FEMPT 346 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71224 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE FEMPT 403 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71225 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE FEMPT 400 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71226 Beta 1 CLONED HUMAN 125I-iodo-pindolol FEMPT 1300 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71227 Beta 2 CLONED HUMAN 3H-CPG-12177 (-) FEMPT 202 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71228 Beta3 CLONED HUMAN 125I-iodo-pindolol FEMPT 564 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71229 Alpha1B CLONED HUMAN 125I-HEAT FEMPT 196 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71230 Alpha1D CLONED HUMAN 125I-HEAT FEMPT 142 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71231 H1 CLONED HUMAN 3H-PYRILAMINE FEMPT 11 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71232 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine FEMPT 1364 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71233 H3 CLONED HUMAN 3H-Alpha-methylhistamine FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71234 H4 CLONED HUMAN 3H-Histamine FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71235 hERG CLONED HUMAN 3H-Dofetilide FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71236 KOR CLONED HUMAN 3H-U69,593 FEMPT 1423 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71237 M1 CLONED HUMAN 3H-QNB FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71238 MDR1 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71239 MOR CLONED HUMAN 3H-DAMGO FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71240 mGluR5 BRAIN RAT 3H-MPEP FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71241 NMDA CLONED HUMAN 3H-MK-801 FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71242 D1 CLONED HUMAN 3H-SCH23390 FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71243 D2 CLONED HUMAN 3H-N-Methylspiperone FEMPT 80 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71244 D3 CLONED HUMAN 3H-N-Methylspiperone FEMPT 35 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71245 D4 CLONED HUMAN 3H-N-Methylspiperone FEMPT 24 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71246 D5 CLONED HUMAN 3H-SCH23390 FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71247 DAT CLONED HUMAN 3H-WIN 35,428 FEMPT 407.4 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71248 Sigma 2 CLONED HUMAN 3H-DTG FEMPT 10 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71249 DOR CLONED HUMAN 3H-DADLE FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71250 EP1 CLONED HUMAN 3H-PGE2 FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 29, 2025
71251 CLONED HUMAN 3H-MUSCIMOL FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71252 Smoothened CLONED HUMAN 3H-Cyclopamine FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71253 Y2 CLONED HUMAN UNKNOWN FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71254 SERT CLONED HUMAN 3H-CITALOPRAM FEMPT 6144 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71255 Sigma 2 CLONED HUMAN 3H-DTG FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 28, 2025
71256 VMAT1 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71257 VMAT2 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71258 CLONED HUMAN UNKNOWN FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71259 I1 CLONED HUMAN UNDEFINED FEMPT >10000 Collier TL et al 2017 Jan 15, 2025 Jan 15, 2025
71260 5-HT1A CLONED HUMAN WAY100635 N,N-diallyltryptamine 100 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71261 5-HT1B CLONED HUMAN 3H-5CT N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71262 5-HT1D CLONED HUMAN 3H-5CT N,N-diallyltryptamine 689 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71263 5-HT1E CLONED HUMAN 3H-5HT N,N-diallyltryptamine 378 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71264 5-HT2A CLONED HUMAN 125I-DOI N,N-diallyltryptamine 701 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71265 5-HT2B CLONED HUMAN 3H-LSD N,N-diallyltryptamine 61 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71266 5-HT2C CLONED HUMAN UNKNOWN N,N-diallyltryptamine 385 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71267 5-HT5A CLONED HUMAN 3H-LSD N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71268 5-HT6 CLONED HUMAN 3H-LSD N,N-diallyltryptamine 1718 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71269 5-HT7 CLONED HUMAN 3H-LSD N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71270 SERT CLONED HUMAN 3H-CITALOPRAM N,N-diallyltryptamine 150 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71271 Alpha1A CLONED HUMAN 125I-HEAT N,N-diallyltryptamine 1663 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71272 Alpha1B CLONED HUMAN 125I-HEAT N,N-diallyltryptamine 1369 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71273 Alpha1D CLONED HUMAN 125I-HEAT N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71274 Alpha2A CLONED HUMAN 3H-CLONIDINE N,N-diallyltryptamine 124 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71275 Alpha2B CLONED HUMAN 3H-CLONIDINE N,N-diallyltryptamine 305 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71276 Alpha2C CLONED HUMAN 3H-CLONIDINE N,N-diallyltryptamine 901 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71277 NET CLONED HUMAN 3H-Nisoxetine N,N-diallyltryptamine 1121 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71278 D1 CLONED HUMAN 3H-SCH23390 N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71279 D2 CLONED HUMAN 3H-N-Methylspiperone N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71280 D3 CLONED HUMAN 3H-N-Methylspiperone N,N-diallyltryptamine 672 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71281 D4 CLONED HUMAN 3H-N-Methylspiperone N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71282 D5 CLONED HUMAN 3H-SCH23390 N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71283 DAT CLONED HUMAN 3H-WIN 35,428 N,N-diallyltryptamine 1406 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71284 MOR CLONED HUMAN 3H-DAMGO N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71285 DOR CLONED HUMAN 3H-DADLE N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71286 KOR CLONED HUMAN 3H-U69,593 N,N-diallyltryptamine 2477 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71287 PBR KIDNEY RAT 3H-PK11195 N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71288 H1 CLONED HUMAN 3H-PYRILAMINE N,N-diallyltryptamine 127 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71289 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71290 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71291 Sigma 1 BRAIN RAT 3H-Pentazocine N,N-diallyltryptamine 101 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71292 Sigma 2 PC12 RAT 3H-DTG N,N-diallyltryptamine 356 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71293 5-HT1A CLONED HUMAN WAY100635 5-methoxy-N,N-diallyltryptamine 19 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71294 5-HT1B CLONED HUMAN 3H-5CT 5-methoxy-N,N-diallyltryptamine 735 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71295 5-HT1D CLONED HUMAN 3H-5CT 5-methoxy-N,N-diallyltryptamine 107 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71296 5-HT1E CLONED HUMAN 3H-5HT 5-methoxy-N,N-diallyltryptamine 500 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71297 5-HT2A CLONED HUMAN 125I-DOI 5-methoxy-N,N-diallyltryptamine 218 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71298 5-HT2B CLONED HUMAN 3H-LSD 5-methoxy-N,N-diallyltryptamine 59 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71299 5-HT2C CLONED HUMAN UNKNOWN 5-methoxy-N,N-diallyltryptamine 456 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71300 5-HT5A CLONED HUMAN 3H-LSD 5-methoxy-N,N-diallyltryptamine 3312 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71301 5-HT6 CLONED HUMAN 3H-LSD 5-methoxy-N,N-diallyltryptamine 153 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71302 5-HT7 CLONED HUMAN 3H-LSD 5-methoxy-N,N-diallyltryptamine 90 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71303 SERT CLONED HUMAN 3H-CITALOPRAM 5-methoxy-N,N-diallyltryptamine 499 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71304 Alpha1A CLONED HUMAN 125I-HEAT 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71305 Alpha1B CLONED HUMAN 125I-HEAT 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71306 Alpha1D CLONED HUMAN 125I-HEAT 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71307 Alpha2A CLONED HUMAN 3H-CLONIDINE 5-methoxy-N,N-diallyltryptamine 215 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71308 Alpha2B CLONED HUMAN 3H-CLONIDINE 5-methoxy-N,N-diallyltryptamine 726 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71309 Alpha2C CLONED HUMAN 3H-CLONIDINE 5-methoxy-N,N-diallyltryptamine 1467 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71310 NET CLONED HUMAN 3H-Nisoxetine 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71311 D1 CLONED HUMAN 3H-SCH23390 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71312 D2 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71313 D3 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71314 D4 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71315 D5 CLONED HUMAN 3H-SCH23390 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71316 DAT CLONED HUMAN WIN35428 5-methoxy-N,N-diallyltryptamine 3378 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71317 MOR CLONED HUMAN 3H-DAMGO 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71318 DOR CLONED HUMAN 3H-DADLE 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71319 KOR CLONED HUMAN 3H-U69,593 5-methoxy-N,N-diallyltryptamine 1132 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71320 PBR KIDNEY RAT 3H-PK11195 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71321 H1 CLONED HUMAN 3H-PYRILAMINE 5-methoxy-N,N-diallyltryptamine 505 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71322 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5-methoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71323 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 5-methoxy-N,N-diallyltryptamine 1712 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71324 Sigma 1 BRAIN RAT 3H-Pentazocine 5-methoxy-N,N-diallyltryptamine 301 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71325 Sigma 2 PC12 RAT 3H-DTG 5-methoxy-N,N-diallyltryptamine 253 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71326 5-HT1A CLONED HUMAN WAY100635 5-fluoro-N,N-diallyltryptamine 80 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71327 5-HT1B CLONED HUMAN 3H-5CT 5-fluoro-N,N-diallyltryptamine 1787 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71328 5-HT1D CLONED HUMAN 3H-5CT 5-fluoro-N,N-diallyltryptamine 816 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71329 5-HT1E CLONED HUMAN 3H-5HT 5-fluoro-N,N-diallyltryptamine 474 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71330 5-HT2A CLONED HUMAN 125I-DOI 5-fluoro-N,N-diallyltryptamine 247 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71331 5-HT2B CLONED HUMAN 3H-LSD 5-fluoro-N,N-diallyltryptamine 16 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71332 5-HT2C CLONED HUMAN UNKNOWN 5-fluoro-N,N-diallyltryptamine 102 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71333 5-HT5A CLONED HUMAN 3H-LSD 5-fluoro-N,N-diallyltryptamine 4299 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71334 5-HT6 CLONED HUMAN 3H-LSD 5-fluoro-N,N-diallyltryptamine 74 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71335 5-HT7 CLONED HUMAN 3H-LSD 5-fluoro-N,N-diallyltryptamine 402 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71336 SERT CLONED HUMAN 3H-CITALOPRAM 5-fluoro-N,N-diallyltryptamine 36 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71337 Alpha1A CLONED HUMAN 125I-HEAT 5-fluoro-N,N-diallyltryptamine 1251 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71338 Alpha1B CLONED HUMAN 125I-HEAT 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71339 Alpha1D CLONED HUMAN 125I-HEAT 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71340 Alpha2A CLONED HUMAN 3H-CLONIDINE 5-fluoro-N,N-diallyltryptamine 119 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71341 Alpha2B CLONED HUMAN 3H-CLONIDINE 5-fluoro-N,N-diallyltryptamine 218 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71342 Alpha2C CLONED HUMAN 3H-CLONIDINE 5-fluoro-N,N-diallyltryptamine 848 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71343 NET CLONED HUMAN 3H-Nisoxetine 5-fluoro-N,N-diallyltryptamine 1818 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71344 D1 CLONED HUMAN 3H-SCH23390 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71345 D2 CLONED HUMAN 3H-N-Methylspiperone 5-fluoro-N,N-diallyltryptamine 2463 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71346 D3 CLONED HUMAN 3H-N-Methylspiperone 5-fluoro-N,N-diallyltryptamine 120 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71347 D4 CLONED HUMAN 3H-N-Methylspiperone 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71348 D5 CLONED HUMAN 3H-SCH23390 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71349 DAT CLONED HUMAN 3H-WIN 35,428 5-fluoro-N,N-diallyltryptamine 2150 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71350 MOR CLONED HUMAN 3H-DAMGO 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71351 DOR CLONED HUMAN 3H-DADLE 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71352 KOR CLONED HUMAN 3H-U69,593 5-fluoro-N,N-diallyltryptamine 2184 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71353 PBR KIDNEY RAT 3H-PK11195 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71354 H1 CLONED HUMAN 3H-PYRILAMINE 5-fluoro-N,N-diallyltryptamine 83 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71355 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71356 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 5-fluoro-N,N-diallyltryptamine 2093 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71357 Sigma 1 BRAIN RAT 3H-Pentazocine 5-fluoro-N,N-diallyltryptamine 86 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71358 Sigma 2 PC12 RAT 3H-DTG 5-fluoro-N,N-diallyltryptamine 303 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71359 5-HT1A CLONED HUMAN WAY100635 5-bromo-N,N-diallyltryptamine 11 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71360 5-HT1B CLONED HUMAN 3H-5CT 5-bromo-N,N-diallyltryptamine 950 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71361 5-HT1D CLONED HUMAN 3H-5CT 5-bromo-N,N-diallyltryptamine 130 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71362 5-HT1E CLONED HUMAN 3H-5HT 5-bromo-N,N-diallyltryptamine 512 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71363 5-HT2A CLONED HUMAN 125I-DOI 5-bromo-N,N-diallyltryptamine 477 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71364 5-HT2B CLONED HUMAN 3H-LSD 5-bromo-N,N-diallyltryptamine 53 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71365 5-HT2C CLONED HUMAN UNKNOWN 5-bromo-N,N-diallyltryptamine 358 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71366 5-HT5A CLONED HUMAN 3H-LSD 5-bromo-N,N-diallyltryptamine 2389 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71367 5-HT6 CLONED HUMAN 3H-LSD 5-bromo-N,N-diallyltryptamine 133 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71368 5-HT7 CLONED HUMAN 3H-LSD 5-bromo-N,N-diallyltryptamine 49 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71369 SERT CLONED HUMAN 3H-CITALOPRAM 5-bromo-N,N-diallyltryptamine 127 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71370 Alpha1A CLONED HUMAN 125I-HEAT 5-bromo-N,N-diallyltryptamine 637 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71371 Alpha1B CLONED HUMAN 125I-HEAT 5-bromo-N,N-diallyltryptamine 2050 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71372 Alpha1D CLONED HUMAN 125I-HEAT 5-bromo-N,N-diallyltryptamine 1124 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71373 Alpha2A CLONED HUMAN 3H-CLONIDINE 5-bromo-N,N-diallyltryptamine 83 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71374 Alpha2B CLONED HUMAN 3H-CLONIDINE 5-bromo-N,N-diallyltryptamine 227 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71375 Alpha2C CLONED HUMAN 3H-CLONIDINE 5-bromo-N,N-diallyltryptamine 356 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71376 NET CLONED HUMAN 3H-Nisoxetine 5-bromo-N,N-diallyltryptamine 964 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71377 D1 CLONED HUMAN 3H-SCH23390 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71378 D2 CLONED HUMAN 3H-N-Methylspiperone 5-bromo-N,N-diallyltryptamine 4349 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71379 D3 CLONED HUMAN 3H-N-Methylspiperone 5-bromo-N,N-diallyltryptamine 240 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71380 D4 CLONED HUMAN 3H-N-Methylspiperone 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71381 D5 CLONED HUMAN 3H-SCH23390 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71382 DAT CLONED HUMAN 3H-WIN 35,428 5-bromo-N,N-diallyltryptamine 2455 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71383 MOR CLONED HUMAN 3H-DAMGO 5-bromo-N,N-diallyltryptamine 1726 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71384 DOR CLONED HUMAN 3H-DADLE 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71385 KOR CLONED HUMAN 3H-U69,593 5-bromo-N,N-diallyltryptamine 898 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71386 PBR KIDNEY RAT 3H-PK11195 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71387 H1 CLONED HUMAN 3H-PYRILAMINE 5-bromo-N,N-diallyltryptamine 106 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71388 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5-bromo-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71389 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 5-bromo-N,N-diallyltryptamine 1495 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71390 Sigma 1 BRAIN RAT 3H-Pentazocine 5-bromo-N,N-diallyltryptamine 101 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71391 Sigma 2 PC12 RAT 3H-DTG 5-bromo-N,N-diallyltryptamine 224 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71392 5-HT1A CLONED HUMAN WAY100635 4-hydroxy-N,N-diallyltryptamine 319 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71393 5-HT1B CLONED HUMAN 3H-5CT 4-hydroxy-N,N-diallyltryptamine 2494 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71394 5-HT1D CLONED HUMAN 3H-5CT 4-hydroxy-N,N-diallyltryptamine 693 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71395 5-HT1E CLONED HUMAN 3H-5HT 4-hydroxy-N,N-diallyltryptamine 238 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71396 5-HT2A CLONED HUMAN 125I-DOI 4-hydroxy-N,N-diallyltryptamine 652 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71397 5-HT2B CLONED HUMAN 3H-LSD 4-hydroxy-N,N-diallyltryptamine 2593 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71398 5-HT2C CLONED HUMAN UNKNOWN 4-hydroxy-N,N-diallyltryptamine 2113 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71399 5-HT5A CLONED HUMAN 3H-LSD 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71400 5-HT6 CLONED HUMAN 3H-LSD 4-hydroxy-N,N-diallyltryptamine 213 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71401 5-HT7 CLONED HUMAN 3H-LSD 4-hydroxy-N,N-diallyltryptamine 600 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71402 SERT CLONED HUMAN 3H-CITALOPRAM 4-hydroxy-N,N-diallyltryptamine 5210 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71403 Alpha1A CLONED HUMAN 125I-HEAT 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71404 Alpha1B CLONED HUMAN 125I-HEAT 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71405 Alpha1D CLONED HUMAN 125I-HEAT 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71406 Alpha2A CLONED HUMAN 3H-CLONIDINE 4-hydroxy-N,N-diallyltryptamine 1206 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71407 Alpha2B CLONED HUMAN 3H-CLONIDINE 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71408 Alpha2C CLONED HUMAN 3H-CLONIDINE 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71409 NET CLONED HUMAN 3H-Nisoxetine 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71410 D1 CLONED HUMAN 3H-SCH23390 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71411 D2 CLONED HUMAN 3H-N-Methylspiperone 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71412 D3 CLONED HUMAN 3H-N-Methylspiperone 4-hydroxy-N,N-diallyltryptamine 1570 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71413 D4 CLONED HUMAN 3H-N-Methylspiperone 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71414 D5 CLONED HUMAN 3H-SCH23390 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71415 DAT CLONED HUMAN 3H-WIN 35,428 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71416 MOR CLONED HUMAN 3H-DAMGO 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71417 DOR CLONED HUMAN 3H-DADLE 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71418 KOR CLONED HUMAN 3H-U69,593 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71419 PBR KIDNEY RAT 3H-PK11195 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71420 H1 CLONED HUMAN 3H-PYRILAMINE 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71421 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71422 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71423 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4-hydroxy-N,N-diallyltryptamine 2765 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71424 Sigma 2 PC12 RAT 3H-DTG 4-hydroxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71425 5-HT1A CLONED HUMAN WAY100635 4-acetoxy-N,N-diallyltryptamine 383 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71426 5-HT1B CLONED HUMAN 3H-5CT 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71427 5-HT1D CLONED HUMAN 3H-5CT 4-acetoxy-N,N-diallyltryptamine 801 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71428 5-HT1E CLONED HUMAN 3H-5HT 4-acetoxy-N,N-diallyltryptamine 467 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71429 5-HT2A CLONED HUMAN 125I-DOI 4-acetoxy-N,N-diallyltryptamine 565 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71430 5-HT2B CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 63 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71431 5-HT2C CLONED HUMAN UNKNOWN 4-acetoxy-N,N-diallyltryptamine 1515 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71432 5-HT5A CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 5844 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71433 5-HT6 CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 1791 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71434 5-HT7 CLONED HUMAN 3H-LSD 4-acetoxy-N,N-diallyltryptamine 724 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71435 SERT CLONED HUMAN 3H-CITALOPRAM 4-acetoxy-N,N-diallyltryptamine 1089 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71436 Alpha1A CLONED HUMAN 125I-HEAT 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71437 Alpha1B CLONED HUMAN 125I-HEAT 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71438 Alpha1D CLONED HUMAN 125I-HEAT 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71439 Alpha2A CLONED HUMAN 3H-CLONIDINE 4-acetoxy-N,N-diallyltryptamine 342 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71440 Alpha2B CLONED HUMAN 3H-CLONIDINE 4-acetoxy-N,N-diallyltryptamine 170 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71441 Alpha2C CLONED HUMAN 3H-CLONIDINE 4-acetoxy-N,N-diallyltryptamine 748 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71442 NET CLONED HUMAN 3H-Nisoxetine 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71443 D1 CLONED HUMAN 3H-SCH23390 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71444 D2 CLONED HUMAN 3H-N-Methylspiperone 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71445 D3 CLONED HUMAN 3H-N-Methylspiperone 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71446 D4 CLONED HUMAN 3H-N-Methylspiperone 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71447 D5 CLONED HUMAN 3H-SCH23390 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71448 DAT CLONED HUMAN 3H-WIN 35,428 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71449 MOR CLONED HUMAN 3H-DADLE 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71450 KOR CLONED HUMAN 3H-U69,593 4-acetoxy-N,N-diallyltryptamine 5235 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71451 PBR KIDNEY RAT 3H-PK11195 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71452 H1 CLONED HUMAN 3H-PYRILAMINE 4-acetoxy-N,N-diallyltryptamine 353 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71453 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71454 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71455 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 4-acetoxy-N,N-diallyltryptamine 299 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71456 Sigma 2 PC12 RAT 3H-DTG 4-acetoxy-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71457 5-HT1A CLONED HUMAN WAY100635 2-phenyl-N,N-diallyltryptamine 402 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71458 5-HT1B CLONED HUMAN 3H-5CT 2-phenyl-N,N-diallyltryptamine 273 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71459 5-HT1D CLONED HUMAN 3H-5CT 2-phenyl-N,N-diallyltryptamine 204 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71460 5-HT1E CLONED HUMAN 3H-5HT 2-phenyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71461 5-HT2A CLONED HUMAN 125I-DOI 2-phenyl-N,N-diallyltryptamine 13 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71462 5-HT2B CLONED HUMAN 3H-LSD 2-phenyl-N,N-diallyltryptamine 192 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71463 5-HT2C CLONED HUMAN UNKNOWN 2-phenyl-N,N-diallyltryptamine 278 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71464 5-HT5A CLONED HUMAN 3H-LSD 2-phenyl-N,N-diallyltryptamine 1670 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71465 5-HT6 CLONED HUMAN 3H-LSD 2-phenyl-N,N-diallyltryptamine 68 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71466 5-HT7 CLONED HUMAN 3H-LSD 2-phenyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71467 SERT CLONED HUMAN 3H-CITALOPRAM 2-phenyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71468 Alpha1A CLONED HUMAN 125I-HEAT 2-phenyl-N,N-diallyltryptamine 75 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71469 Alpha1B CLONED HUMAN 125I-HEAT 2-phenyl-N,N-diallyltryptamine 904 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71470 Alpha1D CLONED HUMAN 125I-HEAT 2-phenyl-N,N-diallyltryptamine 243 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71471 Alpha2A CLONED HUMAN 3H-CLONIDINE 2-phenyl-N,N-diallyltryptamine 85 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71472 Alpha2B CLONED HUMAN 3H-CLONIDINE 2-phenyl-N,N-diallyltryptamine 78 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71473 Alpha2C CLONED HUMAN 3H-CLONIDINE 2-phenyl-N,N-diallyltryptamine 159 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71474 NET CLONED HUMAN 3H-Nisoxetine 2-phenyl-N,N-diallyltryptamine 420 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71475 D1 CLONED HUMAN 3H-SCH23390 2-phenyl-N,N-diallyltryptamine 2793 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71476 D2 CLONED HUMAN 3H-N-Methylspiperone 2-phenyl-N,N-diallyltryptamine 388 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71477 D3 CLONED HUMAN 3H-N-Methylspiperone 2-phenyl-N,N-diallyltryptamine 342 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71478 D4 CLONED HUMAN 3H-N-Methylspiperone 2-phenyl-N,N-diallyltryptamine 1000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71479 D5 CLONED HUMAN 3H-SCH23390 2-phenyl-N,N-diallyltryptamine 2003 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71480 DAT CLONED HUMAN 3H-WIN 35,428 2-phenyl-N,N-diallyltryptamine 746 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71481 MOR CLONED HUMAN 3H-DAMGO 2-phenyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71482 DOR CLONED HUMAN 3H-DADLE 2-phenyl-N,N-diallyltryptamine 6789 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71483 KOR CLONED HUMAN 3H-U69,593 2-phenyl-N,N-diallyltryptamine 589 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71484 PBR KIDNEY RAT 3H-PK11195 2-phenyl-N,N-diallyltryptamine 1929 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71485 H1 CLONED HUMAN 3H-PYRILAMINE 2-phenyl-N,N-diallyltryptamine 79 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71486 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 2-phenyl-N,N-diallyltryptamine 367 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71487 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 2-phenyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71488 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 2-phenyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71489 Sigma 2 PC12 RAT 3H-DTG 2-phenyl-N,N-diallyltryptamine 717 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71490 5-HT1A CLONED HUMAN WAY100635 5-methoxy-2-methyl-N,N-diallyltryptamine 267 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71491 5-HT1B CLONED HUMAN 3H-5CT 5-methoxy-2-methyl-N,N-diallyltryptamine 2267 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71492 5-HT1D CLONED HUMAN 3H-5CT 5-methoxy-2-methyl-N,N-diallyltryptamine 900 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71493 5-HT1E CLONED HUMAN 3H-5HT 5-methoxy-2-methyl-N,N-diallyltryptamine 1594 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71494 5-HT2A CLONED HUMAN 125I-DOI 5-methoxy-2-methyl-N,N-diallyltryptamine 1153 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71495 5-HT2B CLONED HUMAN 3H-LSD 5-methoxy-2-methyl-N,N-diallyltryptamine 241 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71496 5-HT2C CLONED HUMAN UNKNOWN 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71497 5-HT5A CLONED HUMAN 3H-LSD 5-methoxy-2-methyl-N,N-diallyltryptamine 1822 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71498 5-HT6 CLONED HUMAN 3H-LSD 5-methoxy-2-methyl-N,N-diallyltryptamine 206 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71499 5-HT7 CLONED HUMAN 3H-LSD 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71500 SERT CLONED HUMAN 3H-CITALOPRAM 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71501 Alpha1A CLONED HUMAN 125I-HEAT 5-methoxy-2-methyl-N,N-diallyltryptamine 1198 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71502 Alpha1B CLONED HUMAN 125I-HEAT 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71503 Alpha1D CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-methyl-N,N-diallyltryptamine 2405 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71504 Alpha2A CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-methyl-N,N-diallyltryptamine 189 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71505 Alpha2B CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-methyl-N,N-diallyltryptamine 335 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71506 Alpha2C CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-methyl-N,N-diallyltryptamine 888 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71507 NET CLONED HUMAN 3H-Nisoxetine 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71508 D1 CLONED HUMAN 3H-SCH23390 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71509 D2 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71510 D3 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-2-methyl-N,N-diallyltryptamine 2399 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71511 D4 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71512 D5 CLONED HUMAN 3H-SCH23390 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71513 DAT CLONED HUMAN 3H-WIN 35,428 5-methoxy-2-methyl-N,N-diallyltryptamine 2413 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71514 MOR CLONED HUMAN 3H-DAMGO 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71515 DOR CLONED HUMAN 3H-DADLE 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71516 KOR CLONED HUMAN 3H-U69,593 5-methoxy-2-methyl-N,N-diallyltryptamine 391 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71517 PBR KIDNEY RAT 3H-PK11195 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71518 H1 CLONED HUMAN 3H-PYRILAMINE 5-methoxy-2-methyl-N,N-diallyltryptamine 847 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71519 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5-methoxy-2-methyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71520 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 5-methoxy-2-methyl-N,N-diallyltryptamine 1134 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71521 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 5-methoxy-2-methyl-N,N-diallyltryptamine 427 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71522 Sigma 2 PC12 RAT 3H-DTG 5-methoxy-2-methyl-N,N-diallyltryptamine 1235 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71523 5-HT1A CLONED HUMAN WAY100635 5-methoxy-2-fluoro-N,N-diallyltryptamine 318 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71524 5-HT1B CLONED HUMAN 3H-5CT 5-methoxy-2-fluoro-N,N-diallyltryptamine 2011 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71525 5-HT1D CLONED HUMAN 3H-5CT 5-methoxy-2-fluoro-N,N-diallyltryptamine 1592 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71526 5-HT1E CLONED HUMAN 3H-5HT 5-methoxy-2-fluoro-N,N-diallyltryptamine 1273 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71527 5-HT2A CLONED HUMAN 125I-DOI 5-methoxy-2-fluoro-N,N-diallyltryptamine 655 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71528 5-HT2B CLONED HUMAN 3H-LSD 5-methoxy-2-fluoro-N,N-diallyltryptamine 17 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71529 5-HT2C CLONED HUMAN UNKNOWN 5-methoxy-2-fluoro-N,N-diallyltryptamine 541 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71530 5-HT5A CLONED HUMAN 3H-LSD 5-methoxy-2-fluoro-N,N-diallyltryptamine 1916 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71531 5-HT6 CLONED HUMAN 3H-LSD 5-methoxy-2-fluoro-N,N-diallyltryptamine 168 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71532 5-HT7 CLONED HUMAN 3H-LSD 5-methoxy-2-fluoro-N,N-diallyltryptamine 493 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71533 SERT CLONED HUMAN 3H-CITALOPRAM 5-methoxy-2-fluoro-N,N-diallyltryptamine 983 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71534 Alpha1A CLONED HUMAN 125I-HEAT 5-methoxy-2-fluoro-N,N-diallyltryptamine 1570 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71535 Alpha1B CLONED HUMAN 125I-HEAT 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71536 Alpha1D CLONED HUMAN 125I-HEAT 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71537 Alpha2A CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-fluoro-N,N-diallyltryptamine 53 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71538 Alpha2B CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-fluoro-N,N-diallyltryptamine 108 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71539 Alpha2C CLONED HUMAN 3H-CLONIDINE 5-methoxy-2-fluoro-N,N-diallyltryptamine 184 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71540 NET CLONED HUMAN 3H-Nisoxetine 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71541 D1 CLONED HUMAN 3H-SCH23390 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71542 D2 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-2-fluoro-N,N-diallyltryptamine 4416 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71543 D3 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-2-fluoro-N,N-diallyltryptamine 414 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71544 D4 CLONED HUMAN 3H-N-Methylspiperone 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71545 D5 CLONED HUMAN 3H-SCH23390 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71546 DAT CLONED HUMAN 3H-WIN 35,428 5-methoxy-2-fluoro-N,N-diallyltryptamine 2208 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71547 MOR CLONED HUMAN 3H-DAMGO 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71548 DOR CLONED HUMAN 3H-DADLE 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71549 KOR CLONED HUMAN 3H-U69,593 5-methoxy-2-fluoro-N,N-diallyltryptamine 580 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71550 PBR KIDNEY RAT 3H-PK11195 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71551 H1 CLONED HUMAN 3H-PYRILAMINE 5-methoxy-2-fluoro-N,N-diallyltryptamine 435 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71552 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5-methoxy-2-fluoro-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71553 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 5-methoxy-2-fluoro-N,N-diallyltryptamine 1397 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71554 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 5-methoxy-2-fluoro-N,N-diallyltryptamine 531 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71555 Sigma 2 PC12 RAT 3H-DTG 5-methoxy-2-fluoro-N,N-diallyltryptamine 396 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71556 5-HT1A CLONED HUMAN WAY100635 7-ethyl-N,N-diallyltryptamine 1013 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71557 5-HT1B CLONED HUMAN 3H-5CT 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71558 5-HT1D CLONED HUMAN 3H-5CT 7-ethyl-N,N-diallyltryptamine 2691 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71559 5-HT1E CLONED HUMAN 3H-5HT 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71560 5-HT2A CLONED HUMAN 125I-DOI 7-ethyl-N,N-diallyltryptamine 1515 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71561 5-HT2B CLONED HUMAN 3H-LSD 7-ethyl-N,N-diallyltryptamine 65 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71562 5-HT2C CLONED HUMAN UNKNOWN 7-ethyl-N,N-diallyltryptamine 443 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71563 5-HT5A CLONED HUMAN 3H-LSD 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71564 5-HT6 CLONED HUMAN 3H-LSD 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71565 5-HT7 CLONED HUMAN 3H-LSD 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71566 SERT CLONED HUMAN 3H-CITALOPRAM 7-ethyl-N,N-diallyltryptamine 795 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71567 Alpha1A CLONED HUMAN 125I-HEAT 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71568 Alpha1B CLONED HUMAN 125I-HEAT 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71569 Alpha1D CLONED HUMAN 125I-HEAT 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71570 Alpha2A CLONED HUMAN 3H-CLONIDINE 7-ethyl-N,N-diallyltryptamine 141 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71571 Alpha2B CLONED HUMAN 3H-CLONIDINE 7-ethyl-N,N-diallyltryptamine 489 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71572 Alpha2C CLONED HUMAN 3H-CLONIDINE 7-ethyl-N,N-diallyltryptamine 682 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71573 NET CLONED HUMAN 3H-Nisoxetine 7-ethyl-N,N-diallyltryptamine 1879 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71574 D1 CLONED HUMAN 3H-SCH23390 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71575 D2 CLONED HUMAN 3H-N-Methylspiperone 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71576 D3 CLONED HUMAN 3H-N-Methylspiperone 7-ethyl-N,N-diallyltryptamine 1082 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71577 D4 CLONED HUMAN 3H-N-Methylspiperone 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71578 D5 CLONED HUMAN 3H-SCH23390 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71579 DAT CLONED HUMAN 3H-WIN 35,428 7-ethyl-N,N-diallyltryptamine 1725 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71580 MOR CLONED HUMAN 3H-DAMGO 7-ethyl-N,N-diallyltryptamine 2674 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71581 DOR CLONED HUMAN 3H-DADLE 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71582 KOR CLONED HUMAN 3H-U69,593 7-ethyl-N,N-diallyltryptamine 580 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71583 PBR KIDNEY RAT 3H-PK11195 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 15, 2025
71584 H1 CLONED HUMAN 3H-PYRILAMINE 7-ethyl-N,N-diallyltryptamine 913 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71585 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71586 H3 CLONED GUINEA PIG 3H-Alpha-methylhistamine 7-ethyl-N,N-diallyltryptamine >10000 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71587 Sigma 1 BRAIN RAT 3H-Pentazocine(+) 7-ethyl-N,N-diallyltryptamine 22 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71588 Sigma 2 PC12 RAT 3H-DTG 7-ethyl-N,N-diallyltryptamine 136 Klein LM et al 2018 Jan 15, 2025 Jan 28, 2025
71589 5-HT7 HEK293 cells HUMAN 3H-LSD 3-Phenyl-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 322 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71590 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(2-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 714 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71591 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(3-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 1243 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71592 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 104 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71593 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(2-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 386 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71594 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(3-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 883 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71595 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 30 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71596 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(o-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 881 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71597 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(m-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepin 1436 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71598 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 47 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71599 5-HT7 HEK293 cells HUMAN 3H-LSD 3-Phenyl-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 319 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71600 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(2-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 366 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71601 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(3-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 1407 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71602 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 53 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71603 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(2-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 425 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71604 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(3-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 369 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71605 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 70 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71606 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(m-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 506 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71607 5-HT7 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 16 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71608 5-HT1A HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 1866 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71609 5-HT1B HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71610 5-HT1D HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 636 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71611 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 793 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71612 5-HT2A HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 175 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71613 5-HT2B HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 97 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71614 5-HT2C HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 200 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71615 5-HT3 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71616 5-HT4 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71617 5-HT5A HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71618 5-HT6 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 416 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71619 5-HT1A HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71620 5-HT1B HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71621 5-HT1D HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 2112 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71622 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 1366 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71623 5-HT2A HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 187 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71624 5-HT2B HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 100 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71625 5-HT2C HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 799 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71626 5-HT3 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71627 5-HT4 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71628 5-HT5A HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71629 5-HT6 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 248 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71630 5-HT1A HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71631 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71632 5-HT1D HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 165 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71633 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 890 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71634 5-HT2A HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 159 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71635 5-HT2B HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 106 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71636 5-HT2C HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 296 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71637 5-HT3 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71638 5-HT4 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71639 5-HT5A HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71640 5-HT6 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine 109 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71641 5-HT1A HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71642 5-HT1B HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71643 5-HT1D HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71644 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71645 5-HT2A HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 471 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71646 5-HT2B HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 505 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71647 5-HT2C HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 785 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71648 5-HT3 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 703 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71649 5-HT4 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71650 5-HT5A HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 1231 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71651 5-HT6 HEK293 cells HUMAN 3H-LSD 3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71652 5-HT1A HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71653 5-HT1B HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71654 5-HT1D HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71655 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71656 5-HT2A HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 399 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71657 5-HT2B HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 247 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71658 5-HT2C HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 1099 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71659 5-HT3 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 303 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71660 5-HT4 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71661 5-HT5A HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71662 5-HT6 HEK293 cells HUMAN 3H-LSD 3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine 360 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71663 5-HT1A HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71664 5-HT1B HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71665 5-HT1D HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 147 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71666 5-HT1E HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 1787 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71667 5-HT2A HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 138 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71668 5-HT2B HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 150 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71669 5-HT2C HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 20 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71670 5-HT3 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 420 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71671 5-HT4 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine >10000 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71672 5-HT5A HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 1135 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71673 5-HT6 HEK293 cells HUMAN 3H-LSD 3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine 492 Kim Y et al 2018 Jan 15, 2025 Jan 15, 2025
71674 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 63 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71675 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl(5S)-8-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2- carboxylate 841 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71676 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 8.7 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71677 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 230 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71678 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 3.6 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71679 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 473 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71680 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 10.1 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71681 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 208.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71682 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 4.6 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71683 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 129.8 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71684 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate 5.6 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71685 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate 23 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71686 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine (±)-Benzyl-7-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 10.5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71687 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 29.8 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71688 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 14.2 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71689 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 118.7 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71690 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate 12.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71691 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate 931 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71692 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 18.5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71693 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 413 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71694 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 69.7 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71695 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-8-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 2145.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71696 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-Benzyl-7-(4-(3-ethoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 107.7 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71697 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-(5S)-8-(4-Methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine 6659.6 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71698 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-2-((3,5-Dichlorophenyl)sulfonyl)-7-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine 3.4 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71699 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-7-yl)morpholine38a 16.5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71700 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-2-((3,5-Dichlorophenyl)sulfonyl)-8-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine 582 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71701 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 4-((5S)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-8-yl)morpholine 2840 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71702 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-2-Benzyl-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine 11.1 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71703 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) (±)-2-Benzyl-8-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine 2491.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71704 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 269 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71705 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl(5S)-8-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2- carboxylate 89.7 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71706 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 29.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71707 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 5.1 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71708 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 8.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71709 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 14.5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71710 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 42.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71711 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71712 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 11.1 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71713 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 3.6 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71714 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate 26 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71715 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate 6.2 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71716 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 4.9 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71717 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 12.5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71718 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 90 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71719 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate 80.8 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71720 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate 172 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71721 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate 76.4 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71722 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 46.7 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71723 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 17.5 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71724 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 297 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71725 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-8-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 8.8 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71726 Sigma 2 PC12 RAT 3H-DTG (±)-Benzyl-7-(4-(3-ethoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate 111.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71727 Sigma 2 PC12 RAT 3H-DTG (±)-(5S)-8-(4-Methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine 23.8 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71728 Sigma 2 PC12 RAT 3H-DTG (±)-2-((3,5-Dichlorophenyl)sulfonyl)-7-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine 48 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71729 Sigma 2 PC12 RAT 3H-DTG (±)-2-((3,5-Dichlorophenyl)sulfonyl)-8-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine 67 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71730 Sigma 2 PC12 RAT 3H-DTG (±)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-7-yl)morpholine38a 562.3 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71731 Sigma 2 PC12 RAT 3H-DTG 4-((5S)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-8-yl)morpholine 1183 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71732 Sigma 2 PC12 RAT 3H-DTG (±)-2-Benzyl-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine 121 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71733 Sigma 2 PC12 RAT 3H-DTG (±)-2-Benzyl-8-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine 1548 Sahn JJ et al 2017 Jan 15, 2025 Jan 28, 2025
71734 Sigma 2 PC12 RAT 3H-DTG SAS-0132 90 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71735 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) SAS-0132 841 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71736 Sigma 2 PC12 RAT 3H-DTG UKH-1114 46 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71737 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) UKH-1114 1279 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71738 Sigma 2 PC12 RAT 3H-DTG JVW-1034 23 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71739 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) JVW-1034 248 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71740 Sigma 2 PC12 RAT 3H-DTG DKR-1677 5.1 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71741 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) DKR-1677 230 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 28, 2025
71742 5-HT1A CLONED HUMAN 3H-WAY100635 DKR-1677 1187 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025
71743 5-HT1B CLONED HUMAN 3H-5CT DKR-1677 >10000 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025
71744 5-HT1D CLONED HUMAN 3H-5CT DKR-1677 1913 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025
71745 5-HT1E CLONED HUMAN 3H-5HT DKR-1677 7741 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025
71746 5-HT2A CLONED HUMAN 125I-DOI DKR-1677 1274 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025
71747 5-HT2B CLONED HUMAN 3H-LSD DKR-1677 868 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025
71748 5-HT2C CLONED HUMAN UNKNOWN DKR-1677 2138 Vázquez-Rosa E et al 2019 Jan 15, 2025 Jan 15, 2025