The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 68,001-69,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
70749DATCLONEDHUMAN3H-Mazindoloxycodone>10000Olson KM, et al., 2019Jan 15, 2025Jan 15, 2025
70750DATCLONEDHUMAN3H-Mazindol3-((1R,2R)-2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenol>10000Olson KM, et al., 2019Jan 15, 2025Jan 15, 2025
70751DATCLONEDHUMAN3H-MazindolMorphine>10000Olson KM, et al., 2019Jan 15, 2025Jan 15, 2025
70752DATCLONEDHUMAN3H-Mazindolhydromorphone>10000Olson KM, et al., 2019Jan 15, 2025Jan 15, 2025
70753DATCLONEDHUMAN3H-MazindolHydrocodone>10000Olson KM, et al., 2019Jan 15, 2025Jan 15, 2025
70754DATCLONEDHUMAN3H-MazindolBUPRENORPHINE2000Olson KM, et al., 2019Jan 15, 2025Jan 15, 2025
707555-HT1A?CLONED? HUMAN3H-8-OH-DPAT1-Butanoyl-d-lysergic acid diethylamide345Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707565-HT2A?CLONED? HUMAN3H- Ketanserin1-Butanoyl-d-lysergic acid diethylamide87.7Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707575-HT2C?CLONED? HUMAN3H-MESULERGINE1-Butanoyl-d-lysergic acid diethylamide20.8Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707585-HT1A?CLONED? HUMAN3H-8-OH-DPAT1-propionyl-lysergic acid diethylamide637Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707595-HT2A?CLONED? HUMAN3H- Ketanserin1-propionyl-lysergic acid diethylamide196Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707605-HT2C?CLONED? HUMAN3H-MESULERGINE1-propionyl-lysergic acid diethylamide13Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707615-HT1A?CLONED? HUMAN3H-8-OH-DPAT1-Acetyl-D-lysergic acid diethylamide1054Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707625-HT2A?CLONED? HUMAN3H- Ketanserin1-Acetyl-D-lysergic acid diethylamide174Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707635-HT2C?CLONED? HUMAN3H-MESULERGINE1-Acetyl-D-lysergic acid diethylamide10.2Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707645-HT1A?CLONED? HUMAN3H-8-OH-DPATD-lysergic acid diethylamide (LSD)9.5Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707655-HT2A?CLONED? HUMAN3H- KetanserinD-lysergic acid diethylamide (LSD)14.7Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707665-HT2C?CLONED? HUMAN3H-MESULERGINED-lysergic acid diethylamide (LSD)45.3Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707675-HT1B?CLONED? HUMAN3H-GR-1257431-butanoyl-D-lysergic acid diethylamide (1B-LSD)1463Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707685-HT1D?CLONED? HUMAN3H-GR1257431-butanoyl-D-lysergic acid diethylamide (1B-LSD)295Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707695-HT2B?CLONED? HUMAN3H- LSD1-butanoyl-D-lysergic acid diethylamide (1B-LSD)3.5Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707705-HT5A?CLONED? HUMAN3H- LSD1-butanoyl-D-lysergic acid diethylamide (1B-LSD)158Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707715-HT6?CLONED? HUMAN3H- LSD1-butanoyl-D-lysergic acid diethylamide (1B-LSD)607Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
707725-HT7?CLONED? HUMAN3H- LSD1-butanoyl-D-lysergic acid diethylamide (1B-LSD)554Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
70773Alpha1A?CLONED? HUMAN3H-PRAZOSIN1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70774Alpha1B?CLONED? HUMAN3H-PRAZOSIN1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70775Alpha1D?CLONED? HUMAN3H-PRAZOSIN1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70776Alpha2A?CLONED? HUMAN3H-RAUWOLSCINE1-butanoyl-D-lysergic acid diethylamide (1B-LSD)537Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70777Alpha2B?CLONED? HUMAN3H-RAUWOLSCINE1-butanoyl-D-lysergic acid diethylamide (1B-LSD)2656Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70778Alpha2C?CLONED? HUMAN3H-RAUWOLSCINE1-butanoyl-D-lysergic acid diethylamide (1B-LSD)812Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70779Beta 1?CLONED? HUMAN125I-Pindolol1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
70780Beta 2?CLONED? HUMAN3H-CGP-121771-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 15, 2025
70781Beta3?CLONED? HUMAN3H-CGP121771-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70782D1?CLONED? HUMAN3H-SCH233901-butanoyl-D-lysergic acid diethylamide (1B-LSD)1167Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70783D2?CLONED? HUMAN3H-Methylspiperone1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70784D3?CLONED? HUMAN3H-N-Methylspiperone1-butanoyl-D-lysergic acid diethylamide (1B-LSD)352Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70785D4?CLONED? HUMAN3H-N-Methylspiperone1-butanoyl-D-lysergic acid diethylamide (1B-LSD)2271Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70786D5?CLONED? HUMAN3H-SCH233901-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70787H1?CLONED? HUMAN3H-PYRILAMINE1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
707885-HT1D?CLONED? HUMAN3H-TIOTIDINE1-butanoyl-D-lysergic acid diethylamide (1B-LSD)842Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70789H3?CLONEDGUINEA PIG3H-Alpha-methylhistamine1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70790H4?CLONED? HUMAN3H-Histamine1-butanoyl-D-lysergic acid diethylamide (1B-LSD)>10000Halberstadt AL, et al., 2019Jan 15, 2025Jan 28, 2025
70791DATSTRIATUMRAT3H-dopamineD-57816.2Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70792NETCEREBRAL CORTEXRAT3H-dopamineD-5783.23Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70793SERTCEREBRAL CORTEXRAT3H-5-HTD-57816.2Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70794DATSTRIATUMRAT3H-dopamineFLUOXETINE1092Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70795SERTCEREBRAL CORTEXRAT3H-5-HTFLUOXETINE12.2Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70796NETCEREBRAL CORTEXRAT3H-dopamineFLUOXETINE770Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70797DATSTRIATUMRAT3H-dopamineReboxetine2908Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70798SERTCEREBRAL CORTEXRAT3H-5HTReboxetine503Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70799NETCEREBRAL CORTEXRAT3H-dopamineReboxetine0.79Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70800DATSTRIATUMRAT3H-dopamineDESIPRAMINE1567Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70801SERTCEREBRAL CORTEXRAT3H-5HTDESIPRAMINE106Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70802NETCEREBRAL CORTEXRAT3H-dopamineDESIPRAMINE1.3Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70803DATSTRIATUMRAT3H-dopamineIMIPRAMINE1696Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70804SERTCEREBRAL CORTEXRAT3H-5HTIMIPRAMINE20Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70805NETCEREBRAL CORTEXRAT3H-dopamineIMIPRAMINE170Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70806DATHEK293 cellsHUMAN3H-dopamineD-57829.6Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70807SERTHEK293 cellsHUMAN3H-SerotoninD-57820.6Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70808NETHEK293 cellsHUMAN3H-dopamineD-5786.1Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70809SERTHEK293 cellsHUMAN3H-5HTFLUOXETINE14.4Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70810NETHEK293 cellsHUMAN3H-dopamineDESIPRAMINE0.86Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70811SERTHEK293 cellsHUMAN3H-5HTCITALOPRAM3.66Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70812D2CLONEDHUMAN3H-N-MethylspiporoneD-578773Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70813D3CLONEDHUMAN3H-N-MethylspiporoneD-5782615Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
708145-HT1DCLONEDHUMAN3H-GR-125743D-578702Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
708155-HT2ACLONEDHUMAN3H-KETANSERIND-5781639Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
708165-HT2BCLONEDHUMAN3H-LSDD-578425Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
708175-HT2CCLONEDHUMAN3H-MESULERGINED-57873Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70818Alpha2CCLONEDHUMAN3H-CLONIDINED-5782014Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70819Beta2CLONEDHUMAN125I-IodopindololD-578>10000Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70820Beta3CLONEDHUMAN125I-IodopindololD-5782703Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70821KORCLONEDHUMAN3H-BremazocineD-5781387Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
708225-HT1DCLONEDHUMAN3H-TiotodineD-57842Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70823M1CLONEDHUMAN3H-QNBD-578>10000Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70824M4CLONEDHUMAN3H-QNBD-578>10000Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70825M5CLONEDHUMAN3H-QNBD-578>10000Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70826mGluR5CLONEDHUMAN3H-MPEPD-578600Dutta A, et al. 2019Jan 15, 2025Jan 28, 2025
70827OTCLONEDHUMAN3H-OxytocinD-578>10000Dutta A, et al. 2019Jan 15, 2025Jan 15, 2025
70828TMEM97Sf9Insect3H-DTGDTG19.6Alon A et al 2017Jan 15, 2025Jan 15, 2025
70829TMEM97Sf9Insect3H-DTGHALOPERIDOL54.1Alon A et al 2017Jan 15, 2025Jan 15, 2025
70830TMEM97Sf9Insect3H-DTGPB-282Alon A et al 2017Jan 15, 2025Jan 15, 2025
70831TMEM97Sf9Insect3H-DTGPENTAZOCINE (+)2467Alon A et al 2017Jan 15, 2025Jan 15, 2025
70832TMEM97Sf9Insect3H-DTGSKF 10,047 (+)>10000Alon A et al 2017Jan 15, 2025Jan 15, 2025
70833TMEM97Sf9Insect3H-DTGSAS-112125.2Alon A et al 2017Jan 15, 2025Jan 15, 2025
70834TMEM97Sf9Insect3H-DTGElacridar6.5Alon A et al 2017Jan 15, 2025Jan 15, 2025
70835TMEM97Sf9Insect3H-DTGRo 48-8071971Alon A et al 2017Jan 15, 2025Jan 15, 2025
70836Sigma 2CLONEDHUMAN3H-DTGDTG21.2Alon A et al 2017Jan 15, 2025Jan 28, 2025
70837Sigma 2CLONEDHUMAN3H-DTGHALOPERIDOL48.7Alon A et al 2017Jan 15, 2025Jan 28, 2025
70838Sigma 2CLONEDHUMAN3H-DTGPB-281.8Alon A et al 2017Jan 15, 2025Jan 28, 2025
70839Sigma 2CLONEDHUMAN3H-DTGSAS-112123.8Alon A et al 2017Jan 15, 2025Jan 28, 2025
70840Sigma 2CLONEDHUMAN3H-DTGElacridar4.7Alon A et al 2017Jan 15, 2025Jan 28, 2025
70841Sigma 2CLONEDHUMAN3H-DTGRo 48-8071817Alon A et al 2017Jan 15, 2025Jan 28, 2025
708425-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-bromo-2,5-dimethoxyphenyl)ethanamine0.21Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708435-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-bromo-2,5-dimethoxyphenyl)ethanamine2.5Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708445-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-bromo-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride3.3Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708455-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-bromo-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride39Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708465-HT2A?CLONED? HUMAN3H- KetanserinN-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride (3)1.5Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708475-HT2C?CLONED? HUMAN3H-MESULERGINEN-(4-fluoro-2-methoxybenzyl)-2-(4-iodo-2,5-dimethoxyphenyl)ethan-1-amine hydrochloride18Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708485-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-chloro-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride7.7Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708495-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-chloro-2,5-dimethoxyphenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride67Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708505-HT2A?CLONED? HUMAN3H- Ketanserin2-(2,5-dimethoxy-4-nitrophenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride30Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708515-HT2C?CLONED? HUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-nitrophenyl)-N-(4-fluoro-2-methoxybenzyl)ethan-1-amine hydrochloride250Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708525-HT2A?CLONED? HUMAN3H- Ketanserin4-(2-((4-fluoro-2-methoxybenzyl)amino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride120Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
708535-HT2C?CLONED? HUMAN3H-MESULERGINE4-(2-((4-fluoro-2-methoxybenzyl)amino)ethyl)-2,5-dimethoxybenzonitrile hydrochloride>10000Petersen IN et al 2016Jan 15, 2025Jan 15, 2025
70854Sigma 2?CLONED? HUMAN3H-DTG(6S,7R)-7-(1H-Indol-3-yl)-4-methylene-1-azaspiro[5.5] undecane463Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70855Sigma 1?CLONED? HUMAN3H-Pentazocine(+)(6S,7R)-7-(1H-Indol-3-yl)-4-methylene-1-azaspiro[5.5] undecane1446Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70856Sigma 2?CLONED? HUMAN3H-DTG(6R,7S)-1-benzyl-4-methylene-7-phenyl-1,9-diazaspiro[5.5] undecane502Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70857Sigma 1?CLONED? HUMAN3H-Pentazocine(+)(6R,7S)-1-benzyl-4-methylene-7-phenyl-1,9-diazaspiro[5.5] undecane542Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70858Sigma 2?CLONED? HUMAN3H-DTG((4R,6S,7R)-7-phenyl-1-azaspiro[5.5]undecan-4-yl)methanol452Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70859Sigma 1?CLONED? HUMAN3H-Pentazocine(+)((4R,6S,7R)-7-phenyl-1-azaspiro[5.5]undecan-4-yl)methanol2257Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70860Sigma 2?CLONED? HUMAN3H-DTG(4aS,14bR)-13-methoxy-6-methylene-1,2,3,4,5,6,7,8,10,14bdecahydropyrido[2,1-e]phenanthridine152Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70861Sigma 1?CLONED? HUMAN3H-Pentazocine(+)(4aS,14bR)-13-methoxy-6-methylene-1,2,3,4,5,6,7,8,10,14bdecahydropyrido[2,1-e]phenanthridine8Lepovitz L, et al., 2019Jan 15, 2025Jan 15, 2025
70862Sigma 2?CLONED? HUMAN3H-DTG(3aS,13bR)-12-methoxy-5-methylene-2,3,4,5,6,7,9,13boctahydro-1H-cyclopenta[c]pyrido[1,2-b]isoquinoline308Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
70863Sigma 1?CLONED? HUMAN3H-Pentazocine(+)(3aS,13bR)-12-methoxy-5-methylene-2,3,4,5,6,7,9,13boctahydro-1H-cyclopenta[c]pyrido[1,2-b]isoquinoline45Lepovitz L, et al., 2019Jan 15, 2025Jan 28, 2025
708645-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine1138Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708655-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine434Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708665-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine2313Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708675-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine450Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708685-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708695-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708705-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708715-HT2ACLONEDHUMAN3H-Ketaserin(R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine414Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708725-HT2BCLONEDHUMAN3H-LSD(R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine552Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708735-HT2BCLONEDHUMAN3H-LSD(R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine422Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708745-HT2BCLONEDHUMAN3H-LSD(R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine2681Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708755-HT2BCLONEDHUMAN3H-LSD(R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine102Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708765-HT2BCLONEDHUMAN3H-LSD(R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine3044Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708775-HT2BCLONEDHUMAN3H-LSD(R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708785-HT2BCLONEDHUMAN3H-LSD(R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708795-HT2BCLONEDHUMAN3H-LSD(R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine106Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708805-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-2-Methoxy-11-(2-fluoroethoxy)aporphine343Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708815-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-2-Methoxy-11-(3-fluoropropoxy)aporphine338Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708825-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-2-Methoxy-11-((4-fluorobenzyl)oxy)aporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708835-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-2-Methoxy-11-((4-fluorobenzoyl)oxy)aporphine32Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708845-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-N-Propyl-2-methoxy-11-(2-fluoroethoxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708855-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-N-Propyl-2-methoxy-11-(3-fluoropropoxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708865-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzyl)oxy)noraporphine>10000Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
708875-HT2CCLONEDHUMAN3H-MESULERGINE(R)-(-)-N-Propyl-2-methoxy-11-((4-fluorobenzoyl)oxy)noraporphine24Xu Y et al., 2019Jan 15, 2025Jan 15, 2025
70888MOROvaryHAMSTER125i-IBNtxAMorphine5Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70889MOROvaryHAMSTER125i-IBNtxAButyrylfentanyl18Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70890MOROvaryHAMSTER125i-IBNtxAU-4770057Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70891MOROvaryHAMSTER125i-IBNtxAMT-4544Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70892DOROvaryHAMSTER125i-IBNtxAButyrylfentanyl286Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70893DOROvaryHAMSTER125i-IBNtxAU-477001105Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70894DOROvaryHAMSTER125i-IBNtxAMT-45606Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70895KOROvaryHAMSTER125i-IBNtxAButyrylfentanyl3174Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70896KOROvaryHAMSTER125i-IBNtxAU-47700653Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70897KOROvaryHAMSTER125i-IBNtxAMT-45204Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70898MORCLONEDHUMAN3H-DAMGOMorphine3.5Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70899MORCLONEDHUMAN3H-DAMGOButyrylfentanyl18Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70900MORCLONEDHUMAN3H-DAMGOU-4770039Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70901MORCLONEDHUMAN3H-DAMGOMT-4544Baumann MH et al 2018Jan 15, 2025Jan 28, 2025
70902D1?CLONED? HUMAN3H-SCH233906-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione5.7Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70903D5?CLONED? HUMAN3H-SCH233906-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione6.7Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70904D1?CLONED? HUMAN3H-SCH233901-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione10Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70905D5?CLONED? HUMAN3H-SCH233901-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione15Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70906M2?CLONED? HUMAN3H-QNB1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)5-methylpyrimidine-2,4(1H,3H)-dione7700Martini ML et al 2019Jan 15, 2025Jan 15, 2025
70907D1?CLONED? HUMAN3H-SCH233906-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione70Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70908D5?CLONED? HUMAN3H-SCH233906-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione171Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70909Alpha2A?CLONED? HUMAN3H-RAUWOLSCINE6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione6900Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70910M2?CLONED? HUMAN3H-QNB6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methylphenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione6900Martini ML et al 2019Jan 15, 2025Jan 15, 2025
70911D1?CLONED? HUMAN3H-SCH233901,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione93Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70912D5?CLONED? HUMAN3H-SCH233901,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione185Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70913D1?CLONED? HUMAN3H-SCH233901,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione14Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70914D5?CLONED? HUMAN3H-SCH233901,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione90Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70915M3?CLONED? HUMAN3H-QNB1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione4200Martini ML et al 2019Jan 15, 2025Jan 15, 2025
70916D1?CLONED? HUMAN3H-SCH233901,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione5.1Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70917D5?CLONED? HUMAN3H-SCH233901,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione53Martini ML et al 2019Jan 15, 2025Jan 28, 2025
70918M3?CLONED? HUMAN3H-QNB1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)phenyl)pyrimidine-2,4(1H,3H)-dione4600Martini ML et al 2019Jan 15, 2025Jan 15, 2025
709195-HT2BCLONEDHUMAN3H-LSD4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione742Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709205-HT2BCLONEDHUMAN3H-LSD(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione840Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709215-HT2BCLONEDHUMAN3H-LSD(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione2051Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709225-HT2BCLONEDHUMAN3H-LSD(4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione231Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709235-HT7CLONEDHUMAN3H-LSD(4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione2765Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709245-HT7CLONEDHUMAN3H-LSD(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709255-HT7CLONEDHUMAN3H-LSD(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709265-HT7CLONEDHUMAN3H-LSD4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70927Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70928Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70929Alpha2ACLONEDHUMAN3H-RAUWOLSCINE(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70930Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione3364Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70931D4CLONEDHUMAN3H-Methylspiperone4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione1283Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70932D4CLONEDHUMAN3H-Methylspiperone(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70933D4CLONEDHUMAN3H-Methylspiperone(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70934D4CLONEDHUMAN3H-Methylspiperone(4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70935DATCLONEDHUMAN3H-WIN35428(4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70936DATCLONEDHUMAN3H-WIN35428(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70937DATCLONEDHUMAN3H-WIN35428((S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70938DATCLONEDHUMAN3H-WIN354284-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione2562Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
709395-HT1DCLONEDHUMAN125I-aminopotentidine4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione823Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
709405-HT1DCLONEDHUMAN125I-aminopotentidine(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
709415-HT1DCLONEDHUMAN125I-aminopotentidine(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione546Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
709425-HT1DCLONEDHUMAN125I-aminopotentidine4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70943KORCLONEDHUMAN3H-U695934-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70944KORCLONEDHUMAN3H-U69593(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70945KORCLONEDHUMAN3H-U69593(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70946KORCLONEDHUMAN3H-U695934-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione1707Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70947MORCLONEDHUMAN3H-DAMGO4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70948MORCLONEDHUMAN3H-DAMGO(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione1634Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70949MORCLONEDHUMAN3H-DAMGO(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione993Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70950MORCLONEDHUMAN3H-DAMGO4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 28, 2025
70951Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70952Sigma 1CLONEDHUMAN3H-Pentazocine(+)(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70953Sigma 1CLONEDHUMAN3H-Pentazocine(+)(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione58Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70954Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione8.6Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70955Sigma 2CLONEDHUMAN3H-DTG4-(2,6-Dimethylphenyl)-2,9-dimethyl-1,4,9-triazaspiro[5.5]undec-1-ene-3,5-dione696Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70956Sigma 2CLONEDHUMAN3H-DTG(S)-4-(2,6-dimethylphenyl)-2-(hydroxymethyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70957Sigma 2CLONEDHUMAN3H-DTG(S)-2-((1H-Indol-3-yl)methyl)-4-(2,6-dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70958Sigma 2CLONEDHUMAN3H-DTG4-(2,6-Dimethylphenyl)-9-methyl-1,4,9-triazaspiro[5.5]undecane-3,5-dione>10000Uprety R. et al., 2019Jan 15, 2025Jan 15, 2025
70959D3CLONEDHUMAN125I-IABNN-(4-(4-phenylpiperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide8Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70960D3CLONEDHUMAN125I-IABNN-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt0.55Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70961D3CLONEDHUMAN125I-IABNN-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide8.3Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70962D3CLONEDHUMAN125I-IABNN-(4-(4-(4-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide32.7Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70963D3CLONEDHUMAN125I-IABNN-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide0.89Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70964D3CLONEDHUMAN125I-IABNN-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide3.8Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70965D3CLONEDHUMAN125I-IABNN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide0.44Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70966D3CLONEDHUMAN125I-IABNN-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide18Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70967D3CLONEDHUMAN125I-IABNN-(4-(4-(3-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide0.47Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70968D3CLONEDHUMAN125I-IABNN-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide13.6Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70969D3CLONEDHUMAN125I-IABNN-(4-(4-(2-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal0.68Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70970D3CLONEDHUMAN125I-IABNN-(4-(4-(3-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide21.9Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70971D3CLONEDHUMAN125I-IABNN-(4-(4-(4-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide36.1Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70972D3CLONEDHUMAN125I-IABNN-(4-(4-(2-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt0.25Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70973D3CLONEDHUMAN125I-IABNN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt0.5Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70974D3CLONEDHUMAN125I-IABNN-(4-(4-(4-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt2378Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70975D3CLONEDHUMAN125I-IABNN-(4-(4-(2-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt1.5Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70976D3CLONEDHUMAN125I-IABNN-(4-(4-(3-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt0.41Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70977D3CLONEDHUMAN125I-IABNN-(4-(4-(4-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt:78.3Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70978D2CLONEDHUMAN125I-IABNN-(4-(4-phenylpiperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide8434Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70979D2CLONEDHUMAN125I-IABNN-(4-(4-(2-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt169Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70980D2CLONEDHUMAN125I-IABNN-(4-(4-(3-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70981D2CLONEDHUMAN125I-IABNN-(4-(4-(4-chlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70982D2CLONEDHUMAN125I-IABNN-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide63.1Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70983D2CLONEDHUMAN125I-IABNN-(4-(4-(2,4-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide757Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70984D2CLONEDHUMAN125I-IABNN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide2049Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70985D2CLONEDHUMAN125I-IABNN-(4-(4-(3-methoxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide)benzamide1832Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70986D2CLONEDHUMAN125I-IABNN-(4-(4-(3-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide140Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70987D2CLONEDHUMAN125I-IABNN-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide4753Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70988D2CLONEDHUMAN125I-IABNN-(4-(4-(2-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt190Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70989D2CLONEDHUMAN125I-IABNN-(4-(4-(3-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70990D2CLONEDHUMAN125I-IABNN-(4-(4-(4-methylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70991D2CLONEDHUMAN125I-IABNN-(4-(4-(2-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt92.9Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70992D2CLONEDHUMAN125I-IABNN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt743Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70993D2CLONEDHUMAN125I-IABNN-(4-(4-(4-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70994D2CLONEDHUMAN125I-IABNN-(4-(4-(2-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt261Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70995D2CLONEDHUMAN125I-IABNN-(4-(4-(3-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt:99.7Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70996D2CLONEDHUMAN125I-IABNN-(4-(4-(4-trifluoromethylphenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70997D1CLONEDHUMAN125I-IABNN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70998D4CLONEDHUMAN125I-IABNN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
70999D5CLONEDHUMAN125I-IABNN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71000D5CLONEDHUMAN125I-IABNN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71001D1CLONEDHUMAN125I-IABNN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71002D4CLONEDHUMAN125I-IABNN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate sal806Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
710035-HT1ACLONEDHUMAN3H-WAY100635N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide245Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710045-HT1BCLONEDHUMAN3H-GR-125743N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710055-HT1DCLONEDHUMAN3H-GR-125743N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710065-HT1ECLONEDHUMAN3H-5-HTN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710075-HT2ACLONEDHUMAN3H-KetaserinN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710085-HT2BCLONEDHUMAN3H-LSDN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710095-HT2CCLONEDHUMAN3H-MESULERGINEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710105-HT3CLONEDHUMAN3H-MESULERGINEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710115-HT3CLONEDHUMAN3H-GR65630N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710125-HT5ACLONEDHUMAN3H-LSDN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710135-HT6CLONEDHUMAN3H-LSDN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710145-HT7CLONEDHUMAN3H-LSDN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71015Alpha1ACLONEDHUMAN3H-PRAZOSINN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71016Alpha1BCLONEDHUMAN3H-PRAZOSINN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71017Alpha1DCLONEDHUMAN3H-PRAZOSINN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71018Alpha2ACLONEDHUMAN3H-RAUWOLSCINEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71019Alpha2BCLONEDHUMAN3H-RAUWOLSCINEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71020Alpha2CCLONEDHUMAN3H-RAUWOLSCINEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71021BZPCEREBRAL CORTEXRATFNZN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71022Beta 1CLONEDHUMAN125I-PindololN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71023Beta3CLONEDHUMAN125I-PindololN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71024Beta 2CLONEDHUMAN3H-CGP12177N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71025KORCEREBRAL CORTEXRAT3H-MUSCIMOLN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 27, 2025
71026H1CLONEDHUMAN3H-PYRILAMINEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
710275-HT1DCLONEDHUMAN125I-aminopotentidineN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71028H3CLONEDHUMAN3H-Alpha-methylhistamineN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71029H4CLONEDHUMAN3H-HistamineN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71030M1CLONEDHUMAN3H-QNBN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71031M2CLONEDHUMAN3H-QNBN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71032M3CLONEDHUMAN3H-QNBN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71033M4CLONEDHUMAN3H-QNBN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71034M5CLONEDHUMAN3H-QNBN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71035DORCLONEDHUMAN3H-DADLEN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71036KORCLONEDHUMAN3H-U69593N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71037MORCLONEDHUMAN3H-DAMGON-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71038Sigma 1CLONEDHUMAN3H-Pentazocine(+)N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71039Sigma 2CLONEDHUMAN3H-DTGN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71040SLC6A3CLONEDHUMAN3H-WIN 35,428N-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71041NETCLONEDHUMAN3H-NisoxetineN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71042SERTCLONEDHUMAN3H-CITALOPRAMN-(4-(4-(3,5-dichlorophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
710435-HT1ACLONEDHUMAN3H-WAY100635N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710445-HT1BCLONEDHUMAN3H-GR-125743N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710455-HT1DCLONEDHUMAN3H-GR-125743N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710465-HT2ACLONEDHUMAN3H-KETANSERINN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710475-HT2BCLONEDHUMAN3H-LSDN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710485-HT2CCLONEDHUMAN3H-LSDN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt20Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710495-HT3CLONEDHUMAN3H-GR-65630N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710505-HT5ACLONEDHUMAN3H-LSDN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710515-HT6CLONEDHUMAN3H-LSDN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
710525-HT7CLONEDHUMAN3H-LSDN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt187Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71053Alpha1ACLONEDHUMAN3H-PRAZOSINN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71054Alpha1BCLONEDHUMAN3H-PRAZOSINN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71055Alpha1DCLONEDHUMAN3H-PRAZOSINN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71056Alpha2ACLONEDHUMAN3H-RAUWOLSCINEN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71057Alpha2BCLONEDHUMAN3H-RAUWOLSCINEN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71058Alpha2CCLONEDHUMAN3H-RAUWOLSCINEN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71059BZPCEREBRAL CORTEXRATFNZN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 29, 2025
71060Beta 1CLONEDHUMAN125I-PindololN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71061Beta3CLONEDHUMAN125I-PindololN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71062Beta 2CLONEDHUMAN3H-CGP12177N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71063KORCORTICAL MEMBRANESRAT3H-MUSCIMOLN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 27, 2025
71064H1CLONEDHUMAN3H-PYRILAMINEN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt3112Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
710655-HT1DCLONEDHUMAN125I-aminopotentidineN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71066H3CLONEDHUMAN3H-Alpha-methylhistamineN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71067H4CLONEDHUMAN3H-HistamineN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71068M1CLONEDHUMAN3H-QNBN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71069M2CLONEDHUMAN3H-QNBN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71070M3CLONEDHUMAN3H-QNBN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71071M4CLONEDHUMAN3H-QNBN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71072M5CLONEDHUMAN3H-QNBN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71073DORCLONEDHUMAN3H-DADLEN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71074KORCLONEDHUMAN3H-U69593N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71075MORCLONEDHUMAN3H-DAMGON-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71076Sigma 1CLONEDHUMAN3H-Pentazocine(+)N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71077Sigma 2CLONEDHUMAN3H-DTGN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71078DATCLONEDHUMAN3H-WIN 35,428N-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71079NETCLONEDHUMAN3H-NisoxetineN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt>10000Chen PJ et al., 2019Jan 15, 2025Jan 15, 2025
71080SERTCLONEDHUMAN3H-CITALOPRAMN-(4-(4-(3-cyanophenyl)piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamide formate salt118Chen PJ et al., 2019Jan 15, 2025Jan 28, 2025
71081Sigma 2CLONEDHUMAN3H-DTG4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one5.6Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71082Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one24Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71083Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(4-chloropyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one30Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71084Sigma 2CLONEDHUMAN3H-DTG4-(4-(4-chloropyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one8Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71085Sigma 2CLONEDHUMAN3H-DTG4-(4-(pyridinel)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one32Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71086Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(pyridine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one453Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71087Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(pyrimidine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one63Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71088Sigma 2CLONEDHUMAN3H-DTG4-(4-(pyrimidine)-1,4-diazepan-1-yl)-1-(4-fluorophenyl)butan-1-one44Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71089Sigma 2CLONEDHUMAN3H-DTG(4-(4-(5-chloropyridin-2-yl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl) butan-1-one oxime2.7Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71090Sigma 1CLONEDHUMAN3H-Pentazocine(+)(4-(4-(5-chloropyridin-2-yl)-1,4-diazepan-1-yl)-1-(4-fluorophenyl) butan-1-one oxime113Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71091Sigma 1CLONEDHUMAN3H-Pentazocine(+)1-(4-fluorophenyl)-4-(4-(pyridin-2-yl)-1,4-diazepan-1-yl)butan-1- one oxime70Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71092Sigma 2CLONEDHUMAN3H-DTG1-(4-fluorophenyl)-4-(4-(pyridin-2-yl)-1,4-diazepan-1-yl)butan-1- one oxime13Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71093Sigma 2CLONEDHUMAN3H-DTG1-(4-fluorophenyl)-4-(4-(pyrimidin-2-yl)-1,4-diazepan-1-yl)butan1-one oxime26Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71094Sigma 1CLONEDHUMAN3H-Pentazocine(+)1-(4-fluorophenyl)-4-(4-(pyrimidin-2-yl)-1,4-diazepan-1-yl)butan1-one oxime148Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71095Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(5-chloropyridin-2-yl)piperazin-1-yl)-1-(4-fluorophenyl)butan1-one25Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71096Sigma 2CLONEDHUMAN3H-DTG4-(4-(5-chloropyridin-2-yl)piperazin-1-yl)-1-(4-fluorophenyl)butan1-one8Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71097Sigma 1CLONEDHUMAN3H-DTG1-(5-chloropyridin-2-yl)-4-(4-(4-fluorophenyl)butyl)piperazine95Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71098Sigma 2CLONEDHUMAN3H-Pentazocine(+)1-(5-chloropyridin-2-yl)-4-(4-(4-fluorophenyl)butyl)piperazine43Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71099Sigma 2CLONEDHUMAN3H-DTG1-(5-chloropyridin-2-yl)-4-(3-((4-fluorophenyl)thio) propyl)-1,4-diazepane hydrochloride2Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71100Sigma 1CLONEDHUMAN3H-Pentazocine(+)1-(5-chloropyridin-2-yl)-4-(3-((4-fluorophenyl)thio) propyl)-1,4-diazepane hydrochloride8Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71101Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one36Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71102Sigma 2CLONEDHUMAN3H-DTG4-[5-(4-Chloro-phenyl)-2,5-diaza-bicyclo[2.2.1]hept-2-yl]-1-(4-fluoro-phenyl)-butan-1-one52Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71103Sigma 2CLONEDHUMAN3H-DTG4-[4-(2-Pyrimidine)piperazin-1-yl]-1-(4-fluorophenyl)butan-1-one600Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71104Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-[4-(2-Pyrimidine)piperazin-1-yl]-1-(4-fluorophenyl)butan-1-one1148Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71105Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one51Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71106Sigma 2CLONEDHUMAN3H-DTG4-[4-(4-Chlorophenyl)-1,4-diazepan-1-yl]-1-(4-fluorophenyl)butan-1-one33Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71107Sigma 2CLONEDHUMAN3H-DTG4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one5Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71108Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-[3-(4-Chlorophenyl)-3,9-diazabicyclo[4.2.1]non-9-yl]-1-(4-fluorophenyl)butan-1-one42Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71109Sigma 1CLONEDHUMAN3H-Pentazocine(+)cis-2,5-Dicarboethoxy-1-[4-chlorophenyl]pyrrolidine22Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71110Sigma 2CLONEDHUMAN3H-DTGcis-2,5-Dicarboethoxy-1-[4-chlorophenyl]pyrrolidine27Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71111Sigma 2CLONEDHUMAN3H-DTG2-Benzylcarbamyl-5-carboethoxy-1-[4-chlorophenyl]pyrrolidine18Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71112Sigma 2CLONEDHUMAN3H-DTG2-Benzylcarbamyl-5-carboethoxy-1-[4-chlorophenyl]pyrrolidine166Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71113Sigma 2CLONEDHUMAN3H-DTG3-Benzyl-8-[4-chlorophenyl]-3,8-diazabicyclo[3.2.1]octane-2,4-dione29Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71114Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-Benzyl-8-[4-chlorophenyl]-3,8-diazabicyclo[3.2.1]octane-2,4-dione81Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71115Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-Benzyl-8-phenyl-3, 8-diazabicyclo[3.2.1]octane71Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71116Sigma 2CLONEDHUMAN3H-DTG3-Benzyl-8-phenyl-3, 8-diazabicyclo[3.2.1]octane8Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71117Sigma 2CLONEDHUMAN3H-DTG3-Carboethoxy-8-phenyl-3, 8-diazabicyclo[3.2.1]octane2.2Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71118Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-Carboethoxy-8-phenyl-3, 8-diazabicyclo[3.2.1]octane57Al-Ghanim L et al., 2019Jan 15, 2025Jan 28, 2025
71119MT1HEK293 cellsHUMAN3H-MelatoninN-{2-[(4-methoxypyrimidin-2-yl)(methyl)amino]ethyl}acetamide489.7Patel N et al 2020Jan 15, 2025Jan 29, 2025
71120MT1HEK293 cellsHUMAN3H-Melatoninrac-N-{[(1R,2R)-2-(3-methoxyphenyl)cyclopropyl]methyl}ethanediamide3801.8Patel N et al 2020Jan 15, 2025Jan 29, 2025
71121MT1HEK293 cellsHUMAN3H-Melatonin[2-(5-methoxy-1H-indol-3-yl)ethyl]urea16.5959Patel N et al 2020Jan 15, 2025Jan 29, 2025
71122MT1HEK293 cellsHUMAN3H-MelatoninN-{[1-(2-methylpyrimidin-4-yl)piperidin-2-yl]methyl}acetamide6025.6Patel N et al 2020Jan 15, 2025Jan 29, 2025
71123MT1HEK293 cellsHUMAN3H-Melatonin3-cyclopropyl-N-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-amine8511.38Patel N et al 2020Jan 15, 2025Jan 29, 2025
71124MT1HEK293 cellsHUMAN3H-Melatonin6-amino-1-[(3-methoxyphenyl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione>10000Patel N et al 2020Jan 15, 2025Jan 29, 2025
71125MT1HEK293 cellsHUMAN3H-Melatonin1-{6-amino-4-thia-2-azatricyclo[7.3.0.0³,⁷]dodeca-1(9),2,5,7-tetraen-5-yl}ethan-1-one>10000Patel N et al 2020Jan 15, 2025Jan 29, 2025
71126MT1HEK293 cellsHUMAN3H-Melatonin4-(2-chlorobenzoyl)-1H-pyrrole-2-carboxamide>10000Patel N et al 2020Jan 15, 2025Jan 29, 2025
71127MT1HEK293 cellsHUMAN3H-Melatoninmethyl 3-amino-6-methoxy-1H-indole-2-carboxylate9332.54Patel N et al 2020Jan 15, 2025Jan 29, 2025
71128MT1HEK293 cellsHUMAN3H-MelatoninN-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide>10000Patel N et al 2020Jan 15, 2025Jan 29, 2025
71129MT1HEK293 cellsHUMAN3H-Melatonin6-amino-1-(2-phenylethyl)-2-thioxo-2,3-dihydro-4(1H)-pyrimidinone>10000Patel N et al 2020Jan 15, 2025Jan 29, 2025
71130MT2HEK293 cellsHUMAN3H-MelatoninN-{2-[(4-methoxypyrimidin-2-yl)(methyl)amino]ethyl}acetamide123.027Patel N et al 2020Jan 15, 2025Jan 29, 2025
71131MT2HEK293 cellsHUMAN3H-Melatoninrac-N-{[(1R,2R)-2-(3-methoxyphenyl)cyclopropyl]methyl}ethanediamide2754.23Patel N et al 2020Jan 15, 2025Jan 29, 2025
71132MT2HEK293 cellsHUMAN3H-Melatonin[2-(5-methoxy-1H-indol-3-yl)ethyl]urea23.4423Patel N et al 2020Jan 15, 2025Jan 29, 2025
71133MT2HEK293 cellsHUMAN3H-MelatoninN-{[1-(2-methylpyrimidin-4-yl)piperidin-2-yl]methyl}acetamide2454.71Patel N et al 2020Jan 15, 2025Jan 29, 2025
71134MT2HEK293 cellsHUMAN3H-Melatonin3-cyclopropyl-N-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-amine3548.13Patel N et al 2020Jan 15, 2025Jan 29, 2025
71135MT2HEK293 cellsHUMAN3H-Melatonin6-amino-1-[(3-methoxyphenyl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione>10000Patel N et al 2020Jan 15, 2025Jan 29, 2025
71136MT2HEK293 cellsHUMAN3H-Melatonin1-{6-amino-4-thia-2-azatricyclo[7.3.0.0³,⁷]dodeca-1(9),2,5,7-tetraen-5-yl}ethan-1-one5495.41Patel N et al 2020Jan 15, 2025Jan 29, 2025
71137MT2HEK293 cellsHUMAN3H-Melatonin4-(2-chlorobenzoyl)-1H-pyrrole-2-carboxamide1230.27Patel N et al 2020Jan 15, 2025Jan 29, 2025
71138MT2HEK293 cellsHUMAN3H-Melatoninmethyl 3-amino-6-methoxy-1H-indole-2-carboxylate2754.23Patel N et al 2020Jan 15, 2025Jan 29, 2025
71139MT2HEK293 cellsHUMAN3H-MelatoninN-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carboxamide4265.79Patel N et al 2020Jan 15, 2025Jan 29, 2025
71140MT2HEK293 cellsHUMAN3H-Melatonin6-amino-1-(2-phenylethyl)-2-thioxo-2,3-dihydro-4(1H)-pyrimidinone3235.94Patel N et al 2020Jan 15, 2025Jan 29, 2025
711415-HT1ACLONEDHUMANWAY100635ARIPIPRAZOLE50.6Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711425-HT1ACLONEDHUMANWAY100635HALOPERIDOL3600Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711435-HT1ACLONEDHUMANWAY100635CLOZAPINE140Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711445-HT1ACLONEDHUMANWAY100635SYA013117Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711455-HT1ACLONEDHUMANWAY100635SYA1626310.1Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711465-HT2ACLONEDHUMAN125I-DOIARIPIPRAZOLE80.7Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711475-HT2ACLONEDHUMAN125I-DOIHALOPERIDOL120Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711485-HT2ACLONEDHUMAN125I-DOICLOZAPINE80.9Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711495-HT2ACLONEDHUMAN125I-DOISYA01323.6Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711505-HT2ACLONEDHUMAN125I-DOISYA1626350Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711515-HT7CLONEDHUMAN3H-LSDARIPIPRAZOLE10.3Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711525-HT7CLONEDHUMAN3H-LSDHALOPERIDOL1100Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711535-HT7CLONEDHUMAN3H-LSDCLOZAPINE66Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711545-HT7CLONEDHUMAN3H-LSDSYA01378Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711555-HT7CLONEDHUMAN3H-LSDSYA1626390Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
71156D1CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE1960Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71157D1CLONEDHUMAN3H-SCH23390HALOPERIDOL120Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71158D1CLONEDHUMAN3H-SCH23390CLOZAPINE290Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71159D1CLONEDHUMAN3H-SCH23390SYA013163Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71160D1CLONEDHUMAN3H-SCH23390SYA16263238Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71161D2CLONEDHUMAN3H-N-MethylspiperoneARIPIPRAZOLE30.3Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71162D2CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL10.4Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71163D2CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE130Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71164D2CLONEDHUMAN3H-N-MethylspiperoneSYA01343.3Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71165D2CLONEDHUMAN3H-N-MethylspiperoneSYA16263124Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71166D3CLONEDHUMAN3H-N-MethylspiperoneARIPIPRAZOLE90.7Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71167D3CLONEDHUMAN3H-N-MethylspiperoneHALOPERIDOL20.5Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71168D3CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE240Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71169D3CLONEDHUMAN3H-N-MethylspiperoneSYA013159Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71170D3CLONEDHUMAN3H-N-MethylspiperoneSYA1626386Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71171D4CLONEDHUMAN3H-N-MethylspiperoneARIPIPRAZOLE510Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71172D4CLONEDHUMAN3H-MethylspiperoneHALOPERIDOL30.3Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71173D4CLONEDHUMAN3H-N-MethylspiperoneCLOZAPINE54Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71174D4CLONEDHUMAN3H-N-MethylspiperoneSYA01360.6Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71175D4CLONEDHUMAN3H-N-MethylspiperoneSYA1626330.5Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71176D5CLONEDHUMAN3H-SCH23390ARIPIPRAZOLE2590Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71177D5CLONEDHUMAN3H-SCH23390HALOPERIDOL147Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71178D5CLONEDHUMAN3H-SCH23390CLOZAPINE454Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71179D5CLONEDHUMAN3H-SCH23390SYA162631451Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
711805-HT2CCLONEDHUMANUNKNOWNARIPIPRAZOLE76Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711815-HT2CCLONEDHUMANUNKNOWNHALOPERIDOL4700Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711825-HT2CCLONEDHUMANUNKNOWNCLOZAPINE17Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711835-HT2CCLONEDHUMANUNKNOWNSYA0131425Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711845-HT2CCLONEDHUMANUNKNOWNSYA16263>10000Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
71185H1CLONEDHUMAN3H-PYRILAMINEARIPIPRAZOLE25.1Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71186H1CLONEDHUMAN3H-PYRILAMINEHALOPERIDOL440Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71187H1CLONEDHUMAN3H-PYRILAMINECLOZAPINE10.8Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71188H1CLONEDHUMAN3H-PYRILAMINESYA013189Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71189H1CLONEDHUMAN3H-PYRILAMINESYA16263167Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71190M1CLONEDHUMAN3H-QNBARIPIPRAZOLE6780Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
71191M1CLONEDHUMAN3H-QNBHALOPERIDOL1600Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
71192M1CLONEDHUMAN3H-QNBCLOZAPINE1.8Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
71193M1CLONEDHUMAN3H-QNBSYA013872Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
71194D2CLONEDHUMAN3H-N-MethylspiperoneARIPIPRAZOLE3.3Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
71195D2CLONEDHUMAN3H-N-MethylspiperoneARIPIPRAZOLE3.9Bricker B.A., et al. 2019Jan 15, 2025Jan 28, 2025
711965-HT1ACLONEDHUMANWAY100635METHYSERGIDE25Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711975-HT1ACLONEDHUMANWAY100635SYA162631.1Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711985-HT1ACLONEDHUMANWAY100635SYA013117.4Bricker B.A., et al. 2019Jan 15, 2025Jan 15, 2025
711995-HT1ACLONEDHUMANWAY100635FEMPT0.2Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712005-HT1BCLONEDHUMAN3H-5-CTFEMPT122.5Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712015-HT2ACLONEDHUMAN125I-DOIFEMPT406Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712025-HT2BCLONEDHUMAN3H-LSDFEMPT12Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712035-HT2CCLONEDHUMANUNKNOWNFEMPT343Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712045-HT3CLONEDHUMANUNKNOWNFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712055-HT5ACLONEDHUMAN3H-LSDFEMPT2340Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712065-HT6CLONEDHUMAN3H-LSDFEMPT71Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712075-HT7CLONEDHUMAN3H-LSDFEMPT11Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71208CLONEDHUMAN3H-NECAFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71209CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71210CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71211BZPBRAINRATUNKNOWNFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 29, 2025
71212CLONEDHUMAN3H-NitrendipineFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71213AMPACLONEDHUMAN3H-QuisqualateFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 29, 2025
71214NETCLONEDHUMAN3H-NisoxetineFEMPT6980Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71215CLONEDHUMAN3H-SUBSTANCE PFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71216Sigma 1CLONEDHUMAN3H-PentazocineFEMPT1014Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71217CLONEDHUMAN3H-VASOPRESSINFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71218V2CLONEDHUMAN3H-VASOPRESSINFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 29, 2025
71219CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71220CB1CLONEDHUMAN3H-CP55940FEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71221CB2CLONEDHUMAN3H-CP55940FEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71222CLONEDHUMAN3H-PRAZOSINFEMPT180Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71223Alpha2ACLONEDHUMAN3H-RAUWOLSCINEFEMPT346Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71224Alpha2BCLONEDHUMAN3H-RAUWOLSCINEFEMPT403Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71225Alpha2CCLONEDHUMAN3H-RAUWOLSCINEFEMPT400Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71226Beta 1CLONEDHUMAN125I-iodo-pindololFEMPT1300Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71227Beta 2CLONEDHUMAN3H-CPG-12177 (-)FEMPT202Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71228Beta3CLONEDHUMAN125I-iodo-pindololFEMPT564Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71229Alpha1BCLONEDHUMAN125I-HEATFEMPT196Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71230Alpha1DCLONEDHUMAN125I-HEATFEMPT142Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71231H1CLONEDHUMAN3H-PYRILAMINEFEMPT11Collier TL et al 2017Jan 15, 2025Jan 28, 2025
712325-HT1DCLONEDHUMAN125I-iodoaminopotentidineFEMPT1364Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71233H3CLONEDHUMAN3H-Alpha-methylhistamineFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71234H4CLONEDHUMAN3H-HistamineFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71235hERGCLONEDHUMAN3H-DofetilideFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71236KORCLONEDHUMAN3H-U69,593FEMPT1423Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71237M1CLONEDHUMAN3H-QNBFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71238MDR1CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71239MORCLONEDHUMAN3H-DAMGOFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71240mGluR5BRAINRAT3H-MPEPFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71241NMDACLONEDHUMAN3H-MK-801FEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71242D1CLONEDHUMAN3H-SCH23390FEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71243D2CLONEDHUMAN3H-N-MethylspiperoneFEMPT80Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71244D3CLONEDHUMAN3H-N-MethylspiperoneFEMPT35Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71245D4CLONEDHUMAN3H-N-MethylspiperoneFEMPT24Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71246D5CLONEDHUMAN3H-SCH23390FEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71247DATCLONEDHUMAN3H-WIN 35,428FEMPT407.4Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71248Sigma 2CLONEDHUMAN3H-DTGFEMPT10Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71249DORCLONEDHUMAN3H-DADLEFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71250EP1CLONEDHUMAN3H-PGE2FEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 29, 2025
71251CLONEDHUMAN3H-MUSCIMOLFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71252SmoothenedCLONEDHUMAN3H-CyclopamineFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71253Y2CLONEDHUMANUNKNOWNFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71254SERTCLONEDHUMAN3H-CITALOPRAMFEMPT6144Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71255Sigma 2CLONEDHUMAN3H-DTGFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 28, 2025
71256VMAT1CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71257VMAT2CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71258CLONEDHUMANUNKNOWNFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
71259I1CLONEDHUMANUNDEFINEDFEMPT>10000Collier TL et al 2017Jan 15, 2025Jan 15, 2025
712605-HT1ACLONEDHUMANWAY100635N,N-diallyltryptamine100Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712615-HT1BCLONEDHUMAN3H-5CTN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712625-HT1DCLONEDHUMAN3H-5CTN,N-diallyltryptamine689Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712635-HT1ECLONEDHUMAN3H-5HTN,N-diallyltryptamine378Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712645-HT2ACLONEDHUMAN125I-DOIN,N-diallyltryptamine701Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712655-HT2BCLONEDHUMAN3H-LSDN,N-diallyltryptamine61Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712665-HT2CCLONEDHUMANUNKNOWNN,N-diallyltryptamine385Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712675-HT5ACLONEDHUMAN3H-LSDN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712685-HT6CLONEDHUMAN3H-LSDN,N-diallyltryptamine1718Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712695-HT7CLONEDHUMAN3H-LSDN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71270SERTCLONEDHUMAN3H-CITALOPRAMN,N-diallyltryptamine150Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71271Alpha1ACLONEDHUMAN125I-HEATN,N-diallyltryptamine1663Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71272Alpha1BCLONEDHUMAN125I-HEATN,N-diallyltryptamine1369Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71273Alpha1DCLONEDHUMAN125I-HEATN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71274Alpha2ACLONEDHUMAN3H-CLONIDINEN,N-diallyltryptamine124Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71275Alpha2BCLONEDHUMAN3H-CLONIDINEN,N-diallyltryptamine305Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71276Alpha2CCLONEDHUMAN3H-CLONIDINEN,N-diallyltryptamine901Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71277NETCLONEDHUMAN3H-NisoxetineN,N-diallyltryptamine1121Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71278D1CLONEDHUMAN3H-SCH23390N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71279D2CLONEDHUMAN3H-N-MethylspiperoneN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71280D3CLONEDHUMAN3H-N-MethylspiperoneN,N-diallyltryptamine672Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71281D4CLONEDHUMAN3H-N-MethylspiperoneN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71282D5CLONEDHUMAN3H-SCH23390N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71283DATCLONEDHUMAN3H-WIN 35,428N,N-diallyltryptamine1406Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71284MORCLONEDHUMAN3H-DAMGON,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71285DORCLONEDHUMAN3H-DADLEN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71286KORCLONEDHUMAN3H-U69,593N,N-diallyltryptamine2477Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71287PBRKIDNEYRAT3H-PK11195N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71288H1CLONEDHUMAN3H-PYRILAMINEN,N-diallyltryptamine127Klein LM et al 2018Jan 15, 2025Jan 28, 2025
712895-HT1DCLONEDHUMAN125I-iodoaminopotentidineN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71290H3CLONEDGUINEA PIG3H-Alpha-methylhistamineN,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71291Sigma 1BRAINRAT3H-PentazocineN,N-diallyltryptamine101Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71292Sigma 2PC12RAT3H-DTGN,N-diallyltryptamine356Klein LM et al 2018Jan 15, 2025Jan 28, 2025
712935-HT1ACLONEDHUMANWAY1006355-methoxy-N,N-diallyltryptamine19Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712945-HT1BCLONEDHUMAN3H-5CT5-methoxy-N,N-diallyltryptamine735Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712955-HT1DCLONEDHUMAN3H-5CT5-methoxy-N,N-diallyltryptamine107Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712965-HT1ECLONEDHUMAN3H-5HT5-methoxy-N,N-diallyltryptamine500Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712975-HT2ACLONEDHUMAN125I-DOI5-methoxy-N,N-diallyltryptamine218Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712985-HT2BCLONEDHUMAN3H-LSD5-methoxy-N,N-diallyltryptamine59Klein LM et al 2018Jan 15, 2025Jan 15, 2025
712995-HT2CCLONEDHUMANUNKNOWN5-methoxy-N,N-diallyltryptamine456Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713005-HT5ACLONEDHUMAN3H-LSD5-methoxy-N,N-diallyltryptamine3312Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713015-HT6CLONEDHUMAN3H-LSD5-methoxy-N,N-diallyltryptamine153Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713025-HT7CLONEDHUMAN3H-LSD5-methoxy-N,N-diallyltryptamine90Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71303SERTCLONEDHUMAN3H-CITALOPRAM5-methoxy-N,N-diallyltryptamine499Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71304Alpha1ACLONEDHUMAN125I-HEAT5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71305Alpha1BCLONEDHUMAN125I-HEAT5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71306Alpha1DCLONEDHUMAN125I-HEAT5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71307Alpha2ACLONEDHUMAN3H-CLONIDINE5-methoxy-N,N-diallyltryptamine215Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71308Alpha2BCLONEDHUMAN3H-CLONIDINE5-methoxy-N,N-diallyltryptamine726Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71309Alpha2CCLONEDHUMAN3H-CLONIDINE5-methoxy-N,N-diallyltryptamine1467Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71310NETCLONEDHUMAN3H-Nisoxetine5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71311D1CLONEDHUMAN3H-SCH233905-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71312D2CLONEDHUMAN3H-N-Methylspiperone5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71313D3CLONEDHUMAN3H-N-Methylspiperone5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71314D4CLONEDHUMAN3H-N-Methylspiperone5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71315D5CLONEDHUMAN3H-SCH233905-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71316DATCLONEDHUMANWIN354285-methoxy-N,N-diallyltryptamine3378Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71317MORCLONEDHUMAN3H-DAMGO5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71318DORCLONEDHUMAN3H-DADLE5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71319KORCLONEDHUMAN3H-U69,5935-methoxy-N,N-diallyltryptamine1132Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71320PBRKIDNEYRAT3H-PK111955-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71321H1CLONEDHUMAN3H-PYRILAMINE5-methoxy-N,N-diallyltryptamine505Klein LM et al 2018Jan 15, 2025Jan 28, 2025
713225-HT1DCLONEDHUMAN125I-iodoaminopotentidine5-methoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71323H3CLONEDGUINEA PIG3H-Alpha-methylhistamine5-methoxy-N,N-diallyltryptamine1712Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71324Sigma 1BRAINRAT3H-Pentazocine5-methoxy-N,N-diallyltryptamine301Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71325Sigma 2PC12RAT3H-DTG5-methoxy-N,N-diallyltryptamine253Klein LM et al 2018Jan 15, 2025Jan 28, 2025
713265-HT1ACLONEDHUMANWAY1006355-fluoro-N,N-diallyltryptamine80Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713275-HT1BCLONEDHUMAN3H-5CT5-fluoro-N,N-diallyltryptamine1787Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713285-HT1DCLONEDHUMAN3H-5CT5-fluoro-N,N-diallyltryptamine816Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713295-HT1ECLONEDHUMAN3H-5HT5-fluoro-N,N-diallyltryptamine474Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713305-HT2ACLONEDHUMAN125I-DOI5-fluoro-N,N-diallyltryptamine247Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713315-HT2BCLONEDHUMAN3H-LSD5-fluoro-N,N-diallyltryptamine16Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713325-HT2CCLONEDHUMANUNKNOWN5-fluoro-N,N-diallyltryptamine102Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713335-HT5ACLONEDHUMAN3H-LSD5-fluoro-N,N-diallyltryptamine4299Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713345-HT6CLONEDHUMAN3H-LSD5-fluoro-N,N-diallyltryptamine74Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713355-HT7CLONEDHUMAN3H-LSD5-fluoro-N,N-diallyltryptamine402Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71336SERTCLONEDHUMAN3H-CITALOPRAM5-fluoro-N,N-diallyltryptamine36Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71337Alpha1ACLONEDHUMAN125I-HEAT5-fluoro-N,N-diallyltryptamine1251Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71338Alpha1BCLONEDHUMAN125I-HEAT5-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71339Alpha1DCLONEDHUMAN125I-HEAT5-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71340Alpha2ACLONEDHUMAN3H-CLONIDINE5-fluoro-N,N-diallyltryptamine119Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71341Alpha2BCLONEDHUMAN3H-CLONIDINE5-fluoro-N,N-diallyltryptamine218Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71342Alpha2CCLONEDHUMAN3H-CLONIDINE5-fluoro-N,N-diallyltryptamine848Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71343NETCLONEDHUMAN3H-Nisoxetine5-fluoro-N,N-diallyltryptamine1818Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71344D1CLONEDHUMAN3H-SCH233905-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71345D2CLONEDHUMAN3H-N-Methylspiperone5-fluoro-N,N-diallyltryptamine2463Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71346D3CLONEDHUMAN3H-N-Methylspiperone5-fluoro-N,N-diallyltryptamine120Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71347D4CLONEDHUMAN3H-N-Methylspiperone5-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71348D5CLONEDHUMAN3H-SCH233905-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71349DATCLONEDHUMAN3H-WIN 35,4285-fluoro-N,N-diallyltryptamine2150Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71350MORCLONEDHUMAN3H-DAMGO5-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71351DORCLONEDHUMAN3H-DADLE5-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71352KORCLONEDHUMAN3H-U69,5935-fluoro-N,N-diallyltryptamine2184Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71353PBRKIDNEYRAT3H-PK111955-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71354H1CLONEDHUMAN3H-PYRILAMINE5-fluoro-N,N-diallyltryptamine83Klein LM et al 2018Jan 15, 2025Jan 28, 2025
713555-HT1DCLONEDHUMAN125I-iodoaminopotentidine5-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71356H3CLONEDGUINEA PIG3H-Alpha-methylhistamine5-fluoro-N,N-diallyltryptamine2093Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71357Sigma 1BRAINRAT3H-Pentazocine5-fluoro-N,N-diallyltryptamine86Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71358Sigma 2PC12RAT3H-DTG5-fluoro-N,N-diallyltryptamine303Klein LM et al 2018Jan 15, 2025Jan 28, 2025
713595-HT1ACLONEDHUMANWAY1006355-bromo-N,N-diallyltryptamine11Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713605-HT1BCLONEDHUMAN3H-5CT5-bromo-N,N-diallyltryptamine950Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713615-HT1DCLONEDHUMAN3H-5CT5-bromo-N,N-diallyltryptamine130Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713625-HT1ECLONEDHUMAN3H-5HT5-bromo-N,N-diallyltryptamine512Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713635-HT2ACLONEDHUMAN125I-DOI5-bromo-N,N-diallyltryptamine477Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713645-HT2BCLONEDHUMAN3H-LSD5-bromo-N,N-diallyltryptamine53Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713655-HT2CCLONEDHUMANUNKNOWN5-bromo-N,N-diallyltryptamine358Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713665-HT5ACLONEDHUMAN3H-LSD5-bromo-N,N-diallyltryptamine2389Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713675-HT6CLONEDHUMAN3H-LSD5-bromo-N,N-diallyltryptamine133Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713685-HT7CLONEDHUMAN3H-LSD5-bromo-N,N-diallyltryptamine49Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71369SERTCLONEDHUMAN3H-CITALOPRAM5-bromo-N,N-diallyltryptamine127Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71370Alpha1ACLONEDHUMAN125I-HEAT5-bromo-N,N-diallyltryptamine637Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71371Alpha1BCLONEDHUMAN125I-HEAT5-bromo-N,N-diallyltryptamine2050Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71372Alpha1DCLONEDHUMAN125I-HEAT5-bromo-N,N-diallyltryptamine1124Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71373Alpha2ACLONEDHUMAN3H-CLONIDINE5-bromo-N,N-diallyltryptamine83Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71374Alpha2BCLONEDHUMAN3H-CLONIDINE5-bromo-N,N-diallyltryptamine227Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71375Alpha2CCLONEDHUMAN3H-CLONIDINE5-bromo-N,N-diallyltryptamine356Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71376NETCLONEDHUMAN3H-Nisoxetine5-bromo-N,N-diallyltryptamine964Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71377D1CLONEDHUMAN3H-SCH233905-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71378D2CLONEDHUMAN3H-N-Methylspiperone5-bromo-N,N-diallyltryptamine4349Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71379D3CLONEDHUMAN3H-N-Methylspiperone5-bromo-N,N-diallyltryptamine240Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71380D4CLONEDHUMAN3H-N-Methylspiperone5-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71381D5CLONEDHUMAN3H-SCH233905-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71382DATCLONEDHUMAN3H-WIN 35,4285-bromo-N,N-diallyltryptamine2455Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71383MORCLONEDHUMAN3H-DAMGO5-bromo-N,N-diallyltryptamine1726Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71384DORCLONEDHUMAN3H-DADLE5-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71385KORCLONEDHUMAN3H-U69,5935-bromo-N,N-diallyltryptamine898Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71386PBRKIDNEYRAT3H-PK111955-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71387H1CLONEDHUMAN3H-PYRILAMINE5-bromo-N,N-diallyltryptamine106Klein LM et al 2018Jan 15, 2025Jan 28, 2025
713885-HT1DCLONEDHUMAN125I-iodoaminopotentidine5-bromo-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71389H3CLONEDGUINEA PIG3H-Alpha-methylhistamine5-bromo-N,N-diallyltryptamine1495Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71390Sigma 1BRAINRAT3H-Pentazocine5-bromo-N,N-diallyltryptamine101Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71391Sigma 2PC12RAT3H-DTG5-bromo-N,N-diallyltryptamine224Klein LM et al 2018Jan 15, 2025Jan 28, 2025
713925-HT1ACLONEDHUMANWAY1006354-hydroxy-N,N-diallyltryptamine319Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713935-HT1BCLONEDHUMAN3H-5CT4-hydroxy-N,N-diallyltryptamine2494Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713945-HT1DCLONEDHUMAN3H-5CT4-hydroxy-N,N-diallyltryptamine693Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713955-HT1ECLONEDHUMAN3H-5HT4-hydroxy-N,N-diallyltryptamine238Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713965-HT2ACLONEDHUMAN125I-DOI4-hydroxy-N,N-diallyltryptamine652Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713975-HT2BCLONEDHUMAN3H-LSD4-hydroxy-N,N-diallyltryptamine2593Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713985-HT2CCLONEDHUMANUNKNOWN4-hydroxy-N,N-diallyltryptamine2113Klein LM et al 2018Jan 15, 2025Jan 15, 2025
713995-HT5ACLONEDHUMAN3H-LSD4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714005-HT6CLONEDHUMAN3H-LSD4-hydroxy-N,N-diallyltryptamine213Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714015-HT7CLONEDHUMAN3H-LSD4-hydroxy-N,N-diallyltryptamine600Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71402SERTCLONEDHUMAN3H-CITALOPRAM4-hydroxy-N,N-diallyltryptamine5210Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71403Alpha1ACLONEDHUMAN125I-HEAT4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71404Alpha1BCLONEDHUMAN125I-HEAT4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71405Alpha1DCLONEDHUMAN125I-HEAT4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71406Alpha2ACLONEDHUMAN3H-CLONIDINE4-hydroxy-N,N-diallyltryptamine1206Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71407Alpha2BCLONEDHUMAN3H-CLONIDINE4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71408Alpha2CCLONEDHUMAN3H-CLONIDINE4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71409NETCLONEDHUMAN3H-Nisoxetine4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71410D1CLONEDHUMAN3H-SCH233904-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71411D2CLONEDHUMAN3H-N-Methylspiperone4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71412D3CLONEDHUMAN3H-N-Methylspiperone4-hydroxy-N,N-diallyltryptamine1570Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71413D4CLONEDHUMAN3H-N-Methylspiperone4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71414D5CLONEDHUMAN3H-SCH233904-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71415DATCLONEDHUMAN3H-WIN 35,4284-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71416MORCLONEDHUMAN3H-DAMGO4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71417DORCLONEDHUMAN3H-DADLE4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71418KORCLONEDHUMAN3H-U69,5934-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71419PBRKIDNEYRAT3H-PK111954-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71420H1CLONEDHUMAN3H-PYRILAMINE4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
714215-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71422H3CLONEDGUINEA PIG3H-Alpha-methylhistamine4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71423Sigma 1BRAINRAT3H-Pentazocine(+)4-hydroxy-N,N-diallyltryptamine2765Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71424Sigma 2PC12RAT3H-DTG4-hydroxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
714255-HT1ACLONEDHUMANWAY1006354-acetoxy-N,N-diallyltryptamine383Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714265-HT1BCLONEDHUMAN3H-5CT4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714275-HT1DCLONEDHUMAN3H-5CT4-acetoxy-N,N-diallyltryptamine801Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714285-HT1ECLONEDHUMAN3H-5HT4-acetoxy-N,N-diallyltryptamine467Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714295-HT2ACLONEDHUMAN125I-DOI4-acetoxy-N,N-diallyltryptamine565Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714305-HT2BCLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine63Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714315-HT2CCLONEDHUMANUNKNOWN4-acetoxy-N,N-diallyltryptamine1515Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714325-HT5ACLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine5844Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714335-HT6CLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine1791Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714345-HT7CLONEDHUMAN3H-LSD4-acetoxy-N,N-diallyltryptamine724Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71435SERTCLONEDHUMAN3H-CITALOPRAM4-acetoxy-N,N-diallyltryptamine1089Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71436Alpha1ACLONEDHUMAN125I-HEAT4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71437Alpha1BCLONEDHUMAN125I-HEAT4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71438Alpha1DCLONEDHUMAN125I-HEAT4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71439Alpha2ACLONEDHUMAN3H-CLONIDINE4-acetoxy-N,N-diallyltryptamine342Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71440Alpha2BCLONEDHUMAN3H-CLONIDINE4-acetoxy-N,N-diallyltryptamine170Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71441Alpha2CCLONEDHUMAN3H-CLONIDINE4-acetoxy-N,N-diallyltryptamine748Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71442NETCLONEDHUMAN3H-Nisoxetine4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71443D1CLONEDHUMAN3H-SCH233904-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71444D2CLONEDHUMAN3H-N-Methylspiperone4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71445D3CLONEDHUMAN3H-N-Methylspiperone4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71446D4CLONEDHUMAN3H-N-Methylspiperone4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71447D5CLONEDHUMAN3H-SCH233904-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71448DATCLONEDHUMAN3H-WIN 35,4284-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71449MORCLONEDHUMAN3H-DADLE4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71450KORCLONEDHUMAN3H-U69,5934-acetoxy-N,N-diallyltryptamine5235Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71451PBRKIDNEYRAT3H-PK111954-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71452H1CLONEDHUMAN3H-PYRILAMINE4-acetoxy-N,N-diallyltryptamine353Klein LM et al 2018Jan 15, 2025Jan 28, 2025
714535-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71454H3CLONEDGUINEA PIG3H-Alpha-methylhistamine4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71455Sigma 1BRAINRAT3H-Pentazocine(+)4-acetoxy-N,N-diallyltryptamine299Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71456Sigma 2PC12RAT3H-DTG4-acetoxy-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
714575-HT1ACLONEDHUMANWAY1006352-phenyl-N,N-diallyltryptamine402Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714585-HT1BCLONEDHUMAN3H-5CT2-phenyl-N,N-diallyltryptamine273Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714595-HT1DCLONEDHUMAN3H-5CT2-phenyl-N,N-diallyltryptamine204Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714605-HT1ECLONEDHUMAN3H-5HT2-phenyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714615-HT2ACLONEDHUMAN125I-DOI2-phenyl-N,N-diallyltryptamine13Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714625-HT2BCLONEDHUMAN3H-LSD2-phenyl-N,N-diallyltryptamine192Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714635-HT2CCLONEDHUMANUNKNOWN2-phenyl-N,N-diallyltryptamine278Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714645-HT5ACLONEDHUMAN3H-LSD2-phenyl-N,N-diallyltryptamine1670Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714655-HT6CLONEDHUMAN3H-LSD2-phenyl-N,N-diallyltryptamine68Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714665-HT7CLONEDHUMAN3H-LSD2-phenyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71467SERTCLONEDHUMAN3H-CITALOPRAM2-phenyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71468Alpha1ACLONEDHUMAN125I-HEAT2-phenyl-N,N-diallyltryptamine75Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71469Alpha1BCLONEDHUMAN125I-HEAT2-phenyl-N,N-diallyltryptamine904Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71470Alpha1DCLONEDHUMAN125I-HEAT2-phenyl-N,N-diallyltryptamine243Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71471Alpha2ACLONEDHUMAN3H-CLONIDINE2-phenyl-N,N-diallyltryptamine85Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71472Alpha2BCLONEDHUMAN3H-CLONIDINE2-phenyl-N,N-diallyltryptamine78Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71473Alpha2CCLONEDHUMAN3H-CLONIDINE2-phenyl-N,N-diallyltryptamine159Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71474NETCLONEDHUMAN3H-Nisoxetine2-phenyl-N,N-diallyltryptamine420Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71475D1CLONEDHUMAN3H-SCH233902-phenyl-N,N-diallyltryptamine2793Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71476D2CLONEDHUMAN3H-N-Methylspiperone2-phenyl-N,N-diallyltryptamine388Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71477D3CLONEDHUMAN3H-N-Methylspiperone2-phenyl-N,N-diallyltryptamine342Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71478D4CLONEDHUMAN3H-N-Methylspiperone2-phenyl-N,N-diallyltryptamine1000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71479D5CLONEDHUMAN3H-SCH233902-phenyl-N,N-diallyltryptamine2003Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71480DATCLONEDHUMAN3H-WIN 35,4282-phenyl-N,N-diallyltryptamine746Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71481MORCLONEDHUMAN3H-DAMGO2-phenyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71482DORCLONEDHUMAN3H-DADLE2-phenyl-N,N-diallyltryptamine6789Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71483KORCLONEDHUMAN3H-U69,5932-phenyl-N,N-diallyltryptamine589Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71484PBRKIDNEYRAT3H-PK111952-phenyl-N,N-diallyltryptamine1929Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71485H1CLONEDHUMAN3H-PYRILAMINE2-phenyl-N,N-diallyltryptamine79Klein LM et al 2018Jan 15, 2025Jan 28, 2025
714865-HT1DCLONEDHUMAN125I-iodoaminopotentidine2-phenyl-N,N-diallyltryptamine367Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71487H3CLONEDGUINEA PIG3H-Alpha-methylhistamine2-phenyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71488Sigma 1BRAINRAT3H-Pentazocine(+)2-phenyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71489Sigma 2PC12RAT3H-DTG2-phenyl-N,N-diallyltryptamine717Klein LM et al 2018Jan 15, 2025Jan 28, 2025
714905-HT1ACLONEDHUMANWAY1006355-methoxy-2-methyl-N,N-diallyltryptamine267Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714915-HT1BCLONEDHUMAN3H-5CT5-methoxy-2-methyl-N,N-diallyltryptamine2267Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714925-HT1DCLONEDHUMAN3H-5CT5-methoxy-2-methyl-N,N-diallyltryptamine900Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714935-HT1ECLONEDHUMAN3H-5HT5-methoxy-2-methyl-N,N-diallyltryptamine1594Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714945-HT2ACLONEDHUMAN125I-DOI5-methoxy-2-methyl-N,N-diallyltryptamine1153Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714955-HT2BCLONEDHUMAN3H-LSD5-methoxy-2-methyl-N,N-diallyltryptamine241Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714965-HT2CCLONEDHUMANUNKNOWN5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714975-HT5ACLONEDHUMAN3H-LSD5-methoxy-2-methyl-N,N-diallyltryptamine1822Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714985-HT6CLONEDHUMAN3H-LSD5-methoxy-2-methyl-N,N-diallyltryptamine206Klein LM et al 2018Jan 15, 2025Jan 15, 2025
714995-HT7CLONEDHUMAN3H-LSD5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71500SERTCLONEDHUMAN3H-CITALOPRAM5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71501Alpha1ACLONEDHUMAN125I-HEAT5-methoxy-2-methyl-N,N-diallyltryptamine1198Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71502Alpha1BCLONEDHUMAN125I-HEAT5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71503Alpha1DCLONEDHUMAN3H-CLONIDINE5-methoxy-2-methyl-N,N-diallyltryptamine2405Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71504Alpha2ACLONEDHUMAN3H-CLONIDINE5-methoxy-2-methyl-N,N-diallyltryptamine189Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71505Alpha2BCLONEDHUMAN3H-CLONIDINE5-methoxy-2-methyl-N,N-diallyltryptamine335Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71506Alpha2CCLONEDHUMAN3H-CLONIDINE5-methoxy-2-methyl-N,N-diallyltryptamine888Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71507NETCLONEDHUMAN3H-Nisoxetine5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71508D1CLONEDHUMAN3H-SCH233905-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71509D2CLONEDHUMAN3H-N-Methylspiperone5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71510D3CLONEDHUMAN3H-N-Methylspiperone5-methoxy-2-methyl-N,N-diallyltryptamine2399Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71511D4CLONEDHUMAN3H-N-Methylspiperone5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71512D5CLONEDHUMAN3H-SCH233905-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71513DATCLONEDHUMAN3H-WIN 35,4285-methoxy-2-methyl-N,N-diallyltryptamine2413Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71514MORCLONEDHUMAN3H-DAMGO5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71515DORCLONEDHUMAN3H-DADLE5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71516KORCLONEDHUMAN3H-U69,5935-methoxy-2-methyl-N,N-diallyltryptamine391Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71517PBRKIDNEYRAT3H-PK111955-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71518H1CLONEDHUMAN3H-PYRILAMINE5-methoxy-2-methyl-N,N-diallyltryptamine847Klein LM et al 2018Jan 15, 2025Jan 28, 2025
715195-HT1DCLONEDHUMAN125I-iodoaminopotentidine5-methoxy-2-methyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71520H3CLONEDGUINEA PIG3H-Alpha-methylhistamine5-methoxy-2-methyl-N,N-diallyltryptamine1134Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71521Sigma 1BRAINRAT3H-Pentazocine(+)5-methoxy-2-methyl-N,N-diallyltryptamine427Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71522Sigma 2PC12RAT3H-DTG5-methoxy-2-methyl-N,N-diallyltryptamine1235Klein LM et al 2018Jan 15, 2025Jan 28, 2025
715235-HT1ACLONEDHUMANWAY1006355-methoxy-2-fluoro-N,N-diallyltryptamine318Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715245-HT1BCLONEDHUMAN3H-5CT5-methoxy-2-fluoro-N,N-diallyltryptamine2011Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715255-HT1DCLONEDHUMAN3H-5CT5-methoxy-2-fluoro-N,N-diallyltryptamine1592Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715265-HT1ECLONEDHUMAN3H-5HT5-methoxy-2-fluoro-N,N-diallyltryptamine1273Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715275-HT2ACLONEDHUMAN125I-DOI5-methoxy-2-fluoro-N,N-diallyltryptamine655Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715285-HT2BCLONEDHUMAN3H-LSD5-methoxy-2-fluoro-N,N-diallyltryptamine17Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715295-HT2CCLONEDHUMANUNKNOWN5-methoxy-2-fluoro-N,N-diallyltryptamine541Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715305-HT5ACLONEDHUMAN3H-LSD5-methoxy-2-fluoro-N,N-diallyltryptamine1916Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715315-HT6CLONEDHUMAN3H-LSD5-methoxy-2-fluoro-N,N-diallyltryptamine168Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715325-HT7CLONEDHUMAN3H-LSD5-methoxy-2-fluoro-N,N-diallyltryptamine493Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71533SERTCLONEDHUMAN3H-CITALOPRAM5-methoxy-2-fluoro-N,N-diallyltryptamine983Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71534Alpha1ACLONEDHUMAN125I-HEAT5-methoxy-2-fluoro-N,N-diallyltryptamine1570Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71535Alpha1BCLONEDHUMAN125I-HEAT5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71536Alpha1DCLONEDHUMAN125I-HEAT5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71537Alpha2ACLONEDHUMAN3H-CLONIDINE5-methoxy-2-fluoro-N,N-diallyltryptamine53Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71538Alpha2BCLONEDHUMAN3H-CLONIDINE5-methoxy-2-fluoro-N,N-diallyltryptamine108Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71539Alpha2CCLONEDHUMAN3H-CLONIDINE5-methoxy-2-fluoro-N,N-diallyltryptamine184Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71540NETCLONEDHUMAN3H-Nisoxetine5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71541D1CLONEDHUMAN3H-SCH233905-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71542D2CLONEDHUMAN3H-N-Methylspiperone5-methoxy-2-fluoro-N,N-diallyltryptamine4416Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71543D3CLONEDHUMAN3H-N-Methylspiperone5-methoxy-2-fluoro-N,N-diallyltryptamine414Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71544D4CLONEDHUMAN3H-N-Methylspiperone5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71545D5CLONEDHUMAN3H-SCH233905-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71546DATCLONEDHUMAN3H-WIN 35,4285-methoxy-2-fluoro-N,N-diallyltryptamine2208Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71547MORCLONEDHUMAN3H-DAMGO5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71548DORCLONEDHUMAN3H-DADLE5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71549KORCLONEDHUMAN3H-U69,5935-methoxy-2-fluoro-N,N-diallyltryptamine580Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71550PBRKIDNEYRAT3H-PK111955-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71551H1CLONEDHUMAN3H-PYRILAMINE5-methoxy-2-fluoro-N,N-diallyltryptamine435Klein LM et al 2018Jan 15, 2025Jan 28, 2025
715525-HT1DCLONEDHUMAN125I-iodoaminopotentidine5-methoxy-2-fluoro-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71553H3CLONEDGUINEA PIG3H-Alpha-methylhistamine5-methoxy-2-fluoro-N,N-diallyltryptamine1397Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71554Sigma 1BRAINRAT3H-Pentazocine(+)5-methoxy-2-fluoro-N,N-diallyltryptamine531Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71555Sigma 2PC12RAT3H-DTG5-methoxy-2-fluoro-N,N-diallyltryptamine396Klein LM et al 2018Jan 15, 2025Jan 28, 2025
715565-HT1ACLONEDHUMANWAY1006357-ethyl-N,N-diallyltryptamine1013Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715575-HT1BCLONEDHUMAN3H-5CT7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715585-HT1DCLONEDHUMAN3H-5CT7-ethyl-N,N-diallyltryptamine2691Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715595-HT1ECLONEDHUMAN3H-5HT7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715605-HT2ACLONEDHUMAN125I-DOI7-ethyl-N,N-diallyltryptamine1515Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715615-HT2BCLONEDHUMAN3H-LSD7-ethyl-N,N-diallyltryptamine65Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715625-HT2CCLONEDHUMANUNKNOWN7-ethyl-N,N-diallyltryptamine443Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715635-HT5ACLONEDHUMAN3H-LSD7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715645-HT6CLONEDHUMAN3H-LSD7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
715655-HT7CLONEDHUMAN3H-LSD7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71566SERTCLONEDHUMAN3H-CITALOPRAM7-ethyl-N,N-diallyltryptamine795Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71567Alpha1ACLONEDHUMAN125I-HEAT7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71568Alpha1BCLONEDHUMAN125I-HEAT7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71569Alpha1DCLONEDHUMAN125I-HEAT7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71570Alpha2ACLONEDHUMAN3H-CLONIDINE7-ethyl-N,N-diallyltryptamine141Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71571Alpha2BCLONEDHUMAN3H-CLONIDINE7-ethyl-N,N-diallyltryptamine489Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71572Alpha2CCLONEDHUMAN3H-CLONIDINE7-ethyl-N,N-diallyltryptamine682Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71573NETCLONEDHUMAN3H-Nisoxetine7-ethyl-N,N-diallyltryptamine1879Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71574D1CLONEDHUMAN3H-SCH233907-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71575D2CLONEDHUMAN3H-N-Methylspiperone7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71576D3CLONEDHUMAN3H-N-Methylspiperone7-ethyl-N,N-diallyltryptamine1082Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71577D4CLONEDHUMAN3H-N-Methylspiperone7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71578D5CLONEDHUMAN3H-SCH233907-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71579DATCLONEDHUMAN3H-WIN 35,4287-ethyl-N,N-diallyltryptamine1725Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71580MORCLONEDHUMAN3H-DAMGO7-ethyl-N,N-diallyltryptamine2674Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71581DORCLONEDHUMAN3H-DADLE7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71582KORCLONEDHUMAN3H-U69,5937-ethyl-N,N-diallyltryptamine580Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71583PBRKIDNEYRAT3H-PK111957-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 15, 2025
71584H1CLONEDHUMAN3H-PYRILAMINE7-ethyl-N,N-diallyltryptamine913Klein LM et al 2018Jan 15, 2025Jan 28, 2025
715855-HT1DCLONEDHUMAN125I-iodoaminopotentidine7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71586H3CLONEDGUINEA PIG3H-Alpha-methylhistamine7-ethyl-N,N-diallyltryptamine>10000Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71587Sigma 1BRAINRAT3H-Pentazocine(+)7-ethyl-N,N-diallyltryptamine22Klein LM et al 2018Jan 15, 2025Jan 28, 2025
71588Sigma 2PC12RAT3H-DTG7-ethyl-N,N-diallyltryptamine136Klein LM et al 2018Jan 15, 2025Jan 28, 2025
715895-HT7HEK293 cellsHUMAN3H-LSD3-Phenyl-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine322Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715905-HT7HEK293 cellsHUMAN3H-LSD3-(2-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine714Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715915-HT7HEK293 cellsHUMAN3H-LSD3-(3-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine1243Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715925-HT7HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine104Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715935-HT7HEK293 cellsHUMAN3H-LSD3-(2-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine386Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715945-HT7HEK293 cellsHUMAN3H-LSD3-(3-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine883Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715955-HT7HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine30Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715965-HT7HEK293 cellsHUMAN3H-LSD3-(o-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine881Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715975-HT7HEK293 cellsHUMAN3H-LSD3-(m-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepin1436Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715985-HT7HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine47Kim Y et al 2018Jan 15, 2025Jan 15, 2025
715995-HT7HEK293 cellsHUMAN3H-LSD3-Phenyl-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine319Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716005-HT7HEK293 cellsHUMAN3H-LSD3-(2-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine366Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716015-HT7HEK293 cellsHUMAN3H-LSD3-(3-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine1407Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716025-HT7HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine53Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716035-HT7HEK293 cellsHUMAN3H-LSD3-(2-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine425Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716045-HT7HEK293 cellsHUMAN3H-LSD3-(3-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine369Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716055-HT7HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine70Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716065-HT7HEK293 cellsHUMAN3H-LSD3-(m-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine506Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716075-HT7HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine16Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716085-HT1AHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine1866Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716095-HT1BHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716105-HT1DHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine636Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716115-HT1EHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine793Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716125-HT2AHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine175Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716135-HT2BHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine97Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716145-HT2CHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine200Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716155-HT3HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716165-HT4HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716175-HT5AHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716185-HT6HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine416Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716195-HT1AHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716205-HT1BHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716215-HT1DHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine2112Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716225-HT1EHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine1366Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716235-HT2AHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine187Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716245-HT2BHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine100Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716255-HT2CHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine799Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716265-HT3HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716275-HT4HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716285-HT5AHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716295-HT6HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine248Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716305-HT1AHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716315-HT1EHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716325-HT1DHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine165Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716335-HT1EHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine890Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716345-HT2AHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine159Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716355-HT2BHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine106Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716365-HT2CHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine296Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716375-HT3HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716385-HT4HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716395-HT5AHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716405-HT6HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepine109Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716415-HT1AHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716425-HT1BHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716435-HT1DHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716445-HT1EHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716455-HT2AHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine471Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716465-HT2BHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine505Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716475-HT2CHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine785Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716485-HT3HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine703Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716495-HT4HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716505-HT5AHEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine1231Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716515-HT6HEK293 cellsHUMAN3H-LSD3-(4-Fluorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716525-HT1AHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716535-HT1BHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716545-HT1DHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716555-HT1EHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716565-HT2AHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine399Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716575-HT2BHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine247Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716585-HT2CHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine1099Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716595-HT3HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine303Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716605-HT4HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716615-HT5AHEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716625-HT6HEK293 cellsHUMAN3H-LSD3-(4-Chlorophenyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]-azepine360Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716635-HT1AHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716645-HT1BHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716655-HT1DHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine147Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716665-HT1EHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine1787Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716675-HT2AHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine138Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716685-HT2BHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine150Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716695-HT2CHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine20Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716705-HT3HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine420Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716715-HT4HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine>10000Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716725-HT5AHEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine1135Kim Y et al 2018Jan 15, 2025Jan 15, 2025
716735-HT6HEK293 cellsHUMAN3H-LSD3-(p-Tolyl)-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepine492Kim Y et al 2018Jan 15, 2025Jan 15, 2025
71674Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate63Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71675Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl(5S)-8-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2- carboxylate841Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71676Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate8.7Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71677Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate230Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71678Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate3.6Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71679Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate473Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71680Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate10.1Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71681Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate208.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71682Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate4.6Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71683Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate129.8Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71684Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate5.6Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71685Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate23Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71686Sigma 1BRAINGUINEA PIG3H-Pentazocine(±)-Benzyl-7-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate10.5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71687Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate29.8Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71688Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate14.2Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71689Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate118.7Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71690Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate12.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71691Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate931Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71692Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate18.5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71693Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate413Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71694Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate69.7Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71695Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-8-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate2145.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71696Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-Benzyl-7-(4-(3-ethoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate107.7Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71697Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-(5S)-8-(4-Methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine6659.6Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71698Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-2-((3,5-Dichlorophenyl)sulfonyl)-7-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine3.4Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71699Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-7-yl)morpholine38a16.5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71700Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-2-((3,5-Dichlorophenyl)sulfonyl)-8-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine582Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71701Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)4-((5S)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-8-yl)morpholine2840Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71702Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-2-Benzyl-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine11.1Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71703Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)(±)-2-Benzyl-8-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine2491.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71704Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate269Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71705Sigma 2PC12RAT3H-DTG(±)-Benzyl(5S)-8-(4-methylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2- carboxylate89.7Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71706Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate29.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71707Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-propylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate5.1Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71708Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate8.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71709Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-isopropylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate14.5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71710Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate42.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71711Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-cyclobutylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71712Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate11.1Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71713Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-cyclopentylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate3.6Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71714Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate26Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71715Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-(cyclopentylmethyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine-2-carboxylate6.2Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71716Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate4.9Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71717Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-cyclohexylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate12.5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71718Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate90Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71719Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-benzylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo[c]azepine2-carboxylate80.8Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71720Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate172Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71721Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-allylpiperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5-methanobenzo-[c]azepine-2- carboxylate76.4Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71722Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate46.7Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71723Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-(2-methylallyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate17.5Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71724Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate297Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71725Sigma 2PC12RAT3H-DTG(±)-Benzyl-8-(4-(3-methoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate8.8Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71726Sigma 2PC12RAT3H-DTG(±)-Benzyl-7-(4-(3-ethoxy-3-oxopropyl)piperazin-1-yl)-1,3,4,5-tetrahydro-2H-1,5- methanobenzo[c]azepine-2-carboxylate111.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71727Sigma 2PC12RAT3H-DTG(±)-(5S)-8-(4-Methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine23.8Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71728Sigma 2PC12RAT3H-DTG(±)-2-((3,5-Dichlorophenyl)sulfonyl)-7-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine48Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71729Sigma 2PC12RAT3H-DTG(±)-2-((3,5-Dichlorophenyl)sulfonyl)-8-(4-methylpiperazin-1-yl)-2,3,4,5-tetrahydro-1H-1,5- methanobenzo[c]azepine67Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71730Sigma 2PC12RAT3H-DTG(±)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-7-yl)morpholine38a562.3Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71731Sigma 2PC12RAT3H-DTG4-((5S)-2-Benzyl-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepin-8-yl)morpholine1183Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71732Sigma 2PC12RAT3H-DTG(±)-2-Benzyl-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine121Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71733Sigma 2PC12RAT3H-DTG(±)-2-Benzyl-8-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1H-1,5-methanobenzo[c]azepine1548Sahn JJ et al 2017Jan 15, 2025Jan 28, 2025
71734Sigma 2PC12RAT3H-DTGSAS-013290Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71735Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)SAS-0132841Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71736Sigma 2PC12RAT3H-DTGUKH-111446Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71737Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)UKH-11141279Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71738Sigma 2PC12RAT3H-DTGJVW-103423Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71739Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)JVW-1034248Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71740Sigma 2PC12RAT3H-DTGDKR-16775.1Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
71741Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)DKR-1677230Vázquez-Rosa E et al 2019Jan 15, 2025Jan 28, 2025
717425-HT1ACLONEDHUMAN3H-WAY100635DKR-16771187Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025
717435-HT1BCLONEDHUMAN3H-5CTDKR-1677>10000Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025
717445-HT1DCLONEDHUMAN3H-5CTDKR-16771913Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025
717455-HT1ECLONEDHUMAN3H-5HTDKR-16777741Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025
717465-HT2ACLONEDHUMAN125I-DOIDKR-16771274Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025
717475-HT2BCLONEDHUMAN3H-LSDDKR-1677868Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025
717485-HT2CCLONEDHUMANUNKNOWNDKR-16772138Vázquez-Rosa E et al 2019Jan 15, 2025Jan 15, 2025