The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 87,001-88,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
89749nAChRCORTEXRAT3H-Cytisine(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 29, 2025
897505-HT3CLONEDHUMAN3H-GR-65630(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89751Calcium channelCLONEDHUMAN3H-Nitrendipine(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 28, 2025
89752hERGCLONEDHUMAN3H-Dofetilide(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89753Sodium ChannelCLONEDHUMAN3H-Batrachotoxin(3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone>10000Sniecikowska J et al 2019Jan 15, 2025Jan 15, 2025
89754nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride38.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
89755nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89756nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride957Liu J et al 2010Jan 15, 2025Jan 29, 2025
89757nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89758nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride194Liu J et al 2010Jan 15, 2025Jan 29, 2025
89759nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride5670Liu J et al 2010Jan 15, 2025Jan 29, 2025
89760nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride16.2Liu J et al 2010Jan 15, 2025Jan 29, 2025
89761nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride2500Liu J et al 2010Jan 15, 2025Jan 29, 2025
89762nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride171Liu J et al 2010Jan 15, 2025Jan 29, 2025
89763nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89764nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride13.1Liu J et al 2010Jan 15, 2025Jan 29, 2025
89765nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride60.2Liu J et al 2010Jan 15, 2025Jan 29, 2025
89766nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride1230Liu J et al 2010Jan 15, 2025Jan 29, 2025
89767nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride81Liu J et al 2010Jan 15, 2025Jan 29, 2025
89768nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89769nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride2840Liu J et al 2010Jan 15, 2025Jan 29, 2025
89770nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89771nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride28.2Liu J et al 2010Jan 15, 2025Jan 29, 2025
89772nAChRFOREBRAINRAT3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride293Liu J et al 2010Jan 15, 2025Jan 29, 2025
89773nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride5790Liu J et al 2010Jan 15, 2025Jan 29, 2025
89774nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride250Liu J et al 2010Jan 15, 2025Jan 29, 2025
89775nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89776nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride5700Liu J et al 2010Jan 15, 2025Jan 29, 2025
89777nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89778nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride141Liu J et al 2010Jan 15, 2025Jan 29, 2025
89779nAChRFOREBRAINRAT3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride838Liu J et al 2010Jan 15, 2025Jan 29, 2025
89780nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89781nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride445Liu J et al 2010Jan 15, 2025Jan 29, 2025
89782nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride23.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
89783nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89784nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride4170Liu J et al 2010Jan 15, 2025Jan 29, 2025
89785nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89786nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride297Liu J et al 2010Jan 15, 2025Jan 29, 2025
89787nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride1570Liu J et al 2010Jan 15, 2025Jan 29, 2025
89788nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride1680Liu J et al 2010Jan 15, 2025Jan 29, 2025
89789nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride126Liu J et al 2010Jan 15, 2025Jan 29, 2025
89790nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89791nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride8070Liu J et al 2010Jan 15, 2025Jan 29, 2025
89792nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89793nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride54.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
89794nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride426Liu J et al 2010Jan 15, 2025Jan 29, 2025
89795nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride8630Liu J et al 2010Jan 15, 2025Jan 29, 2025
89796nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride61.8Liu J et al 2010Jan 15, 2025Jan 29, 2025
89797nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89798nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride2130Liu J et al 2010Jan 15, 2025Jan 29, 2025
89799nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89800nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride27.7Liu J et al 2010Jan 15, 2025Jan 29, 2025
89801nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride213Liu J et al 2010Jan 15, 2025Jan 29, 2025
89802nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride4110Liu J et al 2010Jan 15, 2025Jan 29, 2025
89803nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride69.7Liu J et al 2010Jan 15, 2025Jan 29, 2025
89804nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride8870Liu J et al 2010Jan 15, 2025Jan 29, 2025
89805nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride166Liu J et al 2010Jan 15, 2025Jan 29, 2025
89806nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89807nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride39.2Liu J et al 2010Jan 15, 2025Jan 29, 2025
89808nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride104Liu J et al 2010Jan 15, 2025Jan 29, 2025
89809nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride7080Liu J et al 2010Jan 15, 2025Jan 29, 2025
89810nAChRCLONEDHUMAN3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride57.9Liu J et al 2010Jan 15, 2025Jan 29, 2025
89811nAChRCLONEDHUMAN3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride349Liu J et al 2010Jan 15, 2025Jan 29, 2025
89812nAChRCLONEDHUMAN3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride3220Liu J et al 2010Jan 15, 2025Jan 29, 2025
89813nAChRCLONEDHUMAN3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride6270Liu J et al 2010Jan 15, 2025Jan 29, 2025
89814nAChRCLONEDHUMAN3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride13.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
89815nAChRFOREBRAINRAT3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride366Liu J et al 2010Jan 15, 2025Jan 29, 2025
89816nAChRCLONEDHUMAN3H-Epibatidine3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride225Liu J et al 2010Jan 15, 2025Jan 29, 2025
89817nAChRCLONEDHUMAN3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride158Liu J et al 2010Jan 15, 2025Jan 29, 2025
89818nAChRCLONEDHUMAN3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89819nAChRCLONEDHUMAN3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride812Liu J et al 2010Jan 15, 2025Jan 29, 2025
89820nAChRCLONEDHUMAN3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89821nAChRCLONEDHUMAN3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride50.9Liu J et al 2010Jan 15, 2025Jan 29, 2025
89822nAChRFOREBRAINRAT3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride509Liu J et al 2010Jan 15, 2025Jan 29, 2025
89823nAChRCLONEDHUMAN3H-Epibatidine3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride3960Liu J et al 2010Jan 15, 2025Jan 29, 2025
89824nAChRCLONEDHUMAN3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride6.5Liu J et al 2010Jan 15, 2025Jan 29, 2025
89825nAChRCLONEDHUMAN3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride104Liu J et al 2010Jan 15, 2025Jan 29, 2025
89826nAChRCLONEDHUMAN3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride208Liu J et al 2010Jan 15, 2025Jan 29, 2025
89827nAChRCLONEDHUMAN3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride793Liu J et al 2010Jan 15, 2025Jan 29, 2025
89828nAChRCLONEDHUMAN3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride2.4Liu J et al 2010Jan 15, 2025Jan 29, 2025
89829nAChRFOREBRAINRAT3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride55.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
89830nAChRCLONEDHUMAN3H-Epibatidine3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride70.6Liu J et al 2010Jan 15, 2025Jan 29, 2025
89831nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride20.5Liu J et al 2010Jan 15, 2025Jan 29, 2025
89832nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride4160Liu J et al 2010Jan 15, 2025Jan 29, 2025
89833nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride383Liu J et al 2010Jan 15, 2025Jan 29, 2025
89834nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89835nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride18.8Liu J et al 2010Jan 15, 2025Jan 29, 2025
89836nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride100Liu J et al 2010Jan 15, 2025Jan 29, 2025
89837nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride1790Liu J et al 2010Jan 15, 2025Jan 29, 2025
89838nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride1.7Liu J et al 2010Jan 15, 2025Jan 29, 2025
89839nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride559Liu J et al 2010Jan 15, 2025Jan 29, 2025
89840nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride40.6Liu J et al 2010Jan 15, 2025Jan 29, 2025
89841nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride5640Liu J et al 2010Jan 15, 2025Jan 29, 2025
89842nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride1.2Liu J et al 2010Jan 15, 2025Jan 29, 2025
89843nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride1.4Liu J et al 2010Jan 15, 2025Jan 29, 2025
89844nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride16.9Liu J et al 2010Jan 15, 2025Jan 29, 2025
89845nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride12.5Liu J et al 2010Jan 15, 2025Jan 29, 2025
89846nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride937Liu J et al 2010Jan 15, 2025Jan 29, 2025
89847nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride150Liu J et al 2010Jan 15, 2025Jan 29, 2025
89848nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89849nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride13.2Liu J et al 2010Jan 15, 2025Jan 29, 2025
89850nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride63.4Liu J et al 2010Jan 15, 2025Jan 29, 2025
89851nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride503Liu J et al 2010Jan 15, 2025Jan 29, 2025
89852nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride357Liu J et al 2010Jan 15, 2025Jan 29, 2025
89853nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride1970Liu J et al 2010Jan 15, 2025Jan 29, 2025
89854nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride1290Liu J et al 2010Jan 15, 2025Jan 29, 2025
89855nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89856nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride190Liu J et al 2010Jan 15, 2025Jan 29, 2025
89857nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride1150Liu J et al 2010Jan 15, 2025Jan 29, 2025
89858nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride108Liu J et al 2010Jan 15, 2025Jan 29, 2025
89859nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride124Liu J et al 2010Jan 15, 2025Jan 29, 2025
89860nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride631Liu J et al 2010Jan 15, 2025Jan 29, 2025
89861nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride953Liu J et al 2010Jan 15, 2025Jan 29, 2025
89862nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride9520Liu J et al 2010Jan 15, 2025Jan 29, 2025
89863nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride59.3Liu J et al 2010Jan 15, 2025Jan 29, 2025
89864nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride374Liu J et al 2010Jan 15, 2025Jan 29, 2025
89865nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride378Liu J et al 2010Jan 15, 2025Jan 29, 2025
89866nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride133Liu J et al 2010Jan 15, 2025Jan 29, 2025
89867nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride3400Liu J et al 2010Jan 15, 2025Jan 29, 2025
89868nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride628Liu J et al 2010Jan 15, 2025Jan 29, 2025
89869nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride>10000Liu J et al 2010Jan 15, 2025Jan 29, 2025
89870nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride48.8Liu J et al 2010Jan 15, 2025Jan 29, 2025
89871nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride380Liu J et al 2010Jan 15, 2025Jan 29, 2025
89872nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride192Liu J et al 2010Jan 15, 2025Jan 29, 2025
89873nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89874nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine1820Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89875nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89876nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine6100Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89877nAChRCORTICAL MEMBRANESRAT3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89878nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine5580Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89879nAChRCLONEDHUMAN3H-Epibatidine3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine2220Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89880Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine103Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89881Sigma 2CLONEDHUMAN3H-DTG3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89882nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89883nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89884nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89885nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89886nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89887nAChRCORTICAL MEMBRANESRAT3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89888nAChRCLONEDHUMAN3H-Epibatidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 29, 2025
89889Sigma 1CLONEDHUMAN3H-Pentazocine(+)5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole4.1Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89890Sigma 2CLONEDHUMAN3H-DTG5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole1312Yu LF et al 2012Jan 15, 2025Jan 28, 2025
898915-HT1ACLONEDHUMAN3H-WAY1006355-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898925-HT1BCLONEDHUMAN3H-5-CT5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898935-HT1DCLONEDHUMAN3H-5-CT5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898945-HT1ECLONEDHUMAN3H-5-HT5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898955-HT2ACLONEDHUMAN3H-KETANSERIN5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole4406Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898965-HT2BCLONEDHUMAN3H-LSD5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole5097Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898975-HT2CCLONEDHUMAN3H-MESULERGINE5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898985-HT3CLONEDHUMAN3H-GR-656305-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
898995-HT5ACLONEDHUMAN3H-LSD5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899005-HT6CLONEDHUMAN3H-LSD5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899015-HT7CLONEDHUMAN3H-LSD5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89902KORCLONEDHUMAN3H-MUSCIMOL5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 27, 2025
89903D1CLONEDHUMAN3H-SCH233905-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89904D5CLONEDHUMAN3H-SCH233905-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89905D2CLONEDHUMAN3H-N-Methylspiperone5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89906D3CLONEDHUMAN3H-N-Methylspiperone5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89907D4CLONEDHUMAN3H-N-Methylspiperone5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89908BZPCORTICAL MEMBRANESRATFNZ5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89909Alpha1ACLONEDHUMAN3H-PRAZOSIN5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89910Alpha1BCLONEDHUMAN3H-PRAZOSIN5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89911Alpha1DCLONEDHUMAN3H-PRAZOSIN5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89912Alpha2ACLONEDHUMAN3H-RAUWOLSCINE5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89913Alpha2BCLONEDHUMAN3H-RAUWOLSCINE5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89914Alpha2CCLONEDHUMAN3H-RAUWOLSCINE5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89915Beta 1CLONEDHUMAN125I-Pindolol5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89916Beta3CLONEDHUMAN125I-Pindolol5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89917Beta 2CLONEDHUMAN3H-CGP-121775-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89918H1CLONEDHUMAN3H-PYRILAMINE5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
899195-HT1DCLONEDHUMAN3H-Cimetidine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole5157Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89920H3CLONEDHUMAN3H-Alpha-methylhistamine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89921H4CLONEDHUMAN3H-Histamine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89922M1CLONEDHUMAN3H-QNB5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89923M2CLONEDHUMAN3H-QNB5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89924M3CLONEDHUMAN3H-QNB5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89925M4CLONEDHUMAN3H-QNB5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89926M5CLONEDHUMAN3H-QNB5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89927DORCLONEDHUMAN3H-DADLE5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89928KORCLONEDHUMAN3H-U695935-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89929MORCLONEDHUMAN3H-DAMGO5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89930DATCLONEDHUMAN3H-WIN354285-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole373Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89931NETCLONEDHUMAN3H-Nisoxetine5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole203Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899325-HT1ACLONEDHUMAN3H-WAY1006353-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899335-HT1BCLONEDHUMAN3H-5-CT3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899345-HT1DCLONEDHUMAN3H-5-CT3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899355-HT1ECLONEDHUMAN3H-5-HT3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899365-HT2ACLONEDHUMAN3H-KETANSERIN3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole6405Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899375-HT2BCLONEDHUMAN3H-LSD3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899385-HT2CCLONEDHUMAN3H-MESULERGINE3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899395-HT3CLONEDHUMAN3H-GR-656303-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899405-HT5ACLONEDHUMAN3H-LSD3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899415-HT6CLONEDHUMAN3H-LSD3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
899425-HT7CLONEDHUMAN3H-LSD3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89943KORCLONEDHUMAN3H-MUSCIMOL3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 27, 2025
89944D1CLONEDHUMAN3H-SCH233903-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89945D5CLONEDHUMAN3H-SCH233903-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89946D2CLONEDHUMAN3H-N-Methylspiperone3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89947D3CLONEDHUMAN3H-N-Methylspiperone3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89948D4CLONEDHUMAN3H-N-Methylspiperone3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89949BZPCORTICAL MEMBRANESRATFNZ3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89950Alpha1ACLONEDHUMAN3H-PRAZOSIN3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89951Alpha1BCLONEDHUMAN3H-PRAZOSIN3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89952Alpha1DCLONEDHUMAN3H-PRAZOSIN3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89953Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89954Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89955Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89956Beta 1CLONEDHUMAN125I-Pindolol3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89957Beta3CLONEDHUMAN125I-Pindolol3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89958Beta 2CLONEDHUMAN3H-CGP121773-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89959H1CLONEDHUMAN3H-PYRILAMINE3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
899605-HT1DCLONEDHUMAN3H-Cimetidine3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89961H3CLONEDHUMAN3H-Alpha-methylhistamine3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89962H4CLONEDHUMAN3H-Histamine3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89963M1CLONEDHUMAN3H-QNB3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89964M2CLONEDHUMAN3H-QNB3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89965M3CLONEDHUMAN3H-QNB3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89966M4CLONEDHUMAN3H-QNB3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89967M5CLONEDHUMAN3H-QNB3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89968DORCLONEDHUMAN3H-DADLE3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89969KORCLONEDHUMAN3H-U695933-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89970MORCLONEDHUMAN3H-DAMGO3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89971DATCLONEDHUMAN3H-WIN 35,4283-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole24Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89972NETCLONEDHUMAN3H-Nisoxetine3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole191Yu LF et al 2012Jan 15, 2025Jan 15, 2025
89973SERTCLONEDHUMAN3H-CITALOPRAM3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole>10000Yu LF et al 2012Jan 15, 2025Jan 28, 2025
89974Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole33Yu LF et al 2012Jan 15, 2025Jan 28, 2025
899755-HT1ACLONEDHUMAN3H-8-OH-DPAT4-Bromo-2,5-dimethoxyphenethylamine240Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899765-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-chloro-2,5-dimethoxy)ethanamine190Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899775-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-methyl) ethanamine440Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899785-HT1ACLONEDHUMAN3H-8-OH-DPAT1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane360Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899795-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxyphenethylamine70Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899805-HT1ACLONEDHUMAN3H-8-OH-DPAT4-iodo-2,5-dimethoxyphenethylamine180Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899815-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5- dimethoxy-4-nitro)ethanamine2200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899825-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-propylphenyl)ethanamine110Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899835-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine370Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899845-HT1ACLONEDHUMAN3H-8-OH-DPAT2,5-dimethoxy-4-isopropylthiophenethylamine470Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899855-HT1ACLONEDHUMAN3H-8-OH-DPAT2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine520Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899865-HT1ACLONEDHUMAN3H-8-OH-DPATMESCALINE4600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899875-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899885-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine5000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899895-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899905-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899915-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899925-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899935-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899945-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899955-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899965-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899975-HT1ACLONEDHUMAN3H-8-OH-DPAT2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899985-HT1ACLONEDHUMAN3H-8-OH-DPATMescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
899995-HT1ACLONEDHUMAN3H-8-OH-DPATLSD3Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900005-HT2ACLONEDHUMAN3H-KETANSERIN4-Bromo-2,5-dimethoxyphenethylamine8.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900015-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-chloro-2,5-dimethoxy)ethanamine13Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900025-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-methyl) ethanamine32.4Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900035-HT2ACLONEDHUMAN3H-KETANSERIN1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane10.5Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900045-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxyphenethylamin1600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900055-HT2ACLONEDHUMAN3H-KETANSERIN4-iodo-2,5-dimethoxyphenethylamine3.5Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900065-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5- dimethoxy-4-nitro)ethanamine23.5Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900075-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-propylphenyl)ethanamine;8.1Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900085-HT2ACLONEDHUMAN3H-KETANSERIN2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine9Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900095-HT2ACLONEDHUMAN3H-KETANSERIN2,5-dimethoxy-4-isopropylthiophenethylamine27.9Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900105-HT2ACLONEDHUMAN3H-KETANSERIN2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine6.5Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900115-HT2ACLONEDHUMAN3H-KETANSERINMESCALINE6300Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900125-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine0.5Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900135-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine0.7Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900145-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900155-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine0.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900165-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine16.4Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900175-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine0.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900185-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine0.8Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900195-HT2ACLONEDHUMAN3H-KETANSERIN2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1.1Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900205-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine0.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900215-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900225-HT2ACLONEDHUMAN3H-KETANSERIN2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1.1Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900235-HT2ACLONEDHUMAN3H-KETANSERINMescaline-NBOMe140Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900245-HT2ACLONEDHUMAN3H-KETANSERINLSD4.2Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900255-HT2CCLONEDHUMAN3H-MESULERGINE4-Bromo-2,5-dimethoxyphenethylamine47Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900265-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-chloro-2,5-dimethoxy)ethanamine90Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900275-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-methyl) ethanamine150Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900285-HT2CCLONEDHUMAN3H-MESULERGINE1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900295-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxyphenethylamine4100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900305-HT2CCLONEDHUMAN3H-MESULERGINE4-iodo-2,5-dimethoxyphenethylamine40Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900315-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5- dimethoxy-4-nitro)ethanamine370Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900325-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-propylphenyl)ethanamine40Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900335-HT2CCLONEDHUMAN3H-MESULERGINE2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine69Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900345-HT2CCLONEDHUMAN3H-MESULERGINE2,5-dimethoxy-4-isopropylthiophenethylamine130Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900355-HT2CCLONEDHUMAN3H-MESULERGINE2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine39Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900365-HT2CCLONEDHUMAN3H-MESULERGINEMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900375-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6.2Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900385-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine5.2Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900395-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine13Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900405-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7.2Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900415-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine130Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900425-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4.6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900435-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine21Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900445-HT2CCLONEDHUMAN3H-MESULERGINE2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900455-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6.5Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900465-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine16Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900475-HT2CCLONEDHUMAN3H-MESULERGINE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine6.4Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900485-HT2CCLONEDHUMAN3H-MESULERGINEMescaline-NBOMe640Rickli A et al 2015Jan 15, 2025Jan 15, 2025
900495-HT2CCLONEDHUMAN3H-MESULERGINELSD15Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90050Alpha1ACLONEDHUMAN3H-PRAZOSIN2C-B, 4-bromo-2,5-dimethoxyphenethylamine8200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90051Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90052Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90053Alpha1ACLONEDHUMAN3H-PRAZOSIN1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane7400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90054Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxyphenethylamine7900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90055Alpha1ACLONEDHUMAN3H-PRAZOSIN4-iodo-2,5-dimethoxyphenethylamine5100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90056Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90057Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-propylphenyl)ethanamine3500Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90058Alpha1ACLONEDHUMAN3H-PRAZOSIN2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90059Alpha1ACLONEDHUMAN3H-PRAZOSIN2,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90060Alpha1ACLONEDHUMAN3H-PRAZOSIN2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90061Alpha1ACLONEDHUMAN3H-PRAZOSINMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90062Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine430Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90063Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine810Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90064Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90065Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine530Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90066Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine550Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90067Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine370Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90068Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine850Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90069Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine310Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90070Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine550Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90071Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine580Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90072Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine340Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90073Alpha1ACLONEDHUMAN3H-PRAZOSINMescaline-NBOMe3000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90074Alpha1ACLONEDHUMAN3H-PRAZOSINLSD670Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90075Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-Bromo-2,5-dimethoxyphenethylamine320Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90076Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-chloro-2,5-dimethoxy)ethanamine530Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90077Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-methyl) ethanamine290Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90078Alpha2ACLONEDHUMAN3H-RAUWOLSCINE1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane110Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90079Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxyphenethylamine1000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90080Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-iodo-2,5-dimethoxyphenethylamine70Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90081Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5- dimethoxy-4-nitro)ethanamine1300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90082Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-propylphenyl)ethanamine90Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90083Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine230Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90084Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2,5-dimethoxy-4-isopropylthiophenethylamine180Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90085Alpha2ACLONEDHUMAN3H-RAUWOLSCINEMESCALINE1400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90086Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamin430Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90087Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine560Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90088Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine370Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90089Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine260Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90090Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine530Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90091Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine320Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90092Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine590Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90093Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine410Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90094Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine450Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90095Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine260Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90096Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine360Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90097Alpha2ACLONEDHUMAN3H-RAUWOLSCINEMescaline-NBOMe810Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90098Alpha2ACLONEDHUMAN3H-RAUWOLSCINELSD12Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90099D1CLONEDHUMAN3H-SCH233904-Bromo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90100D1CLONEDHUMAN3H-SCH233902-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90101D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90102D1CLONEDHUMAN3H-SCH233901-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90103D1CLONEDHUMAN3H-SCH233902,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90104D1CLONEDHUMAN3H-SCH233904-iodo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90105D1CLONEDHUMAN3H-SCH233902-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90106D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-propylphenyl)ethanamine8400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90107D1CLONEDHUMAN3H-SCH233902-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90108D1CLONEDHUMAN3H-SCH233902,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90109D1CLONEDHUMAN3H-SCH233902-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90110D1CLONEDHUMAN3H-SCH23390MESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90111D1CLONEDHUMAN3H-SCH233902-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine9300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90112D1CLONEDHUMAN3H-SCH233902-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90113D1CLONEDHUMAN3H-SCH233902-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine8700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90114D1CLONEDHUMAN3H-SCH233902-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90115D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90116D1CLONEDHUMAN3H-SCH233902-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90117D1CLONEDHUMAN3H-SCH233902-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90118D1CLONEDHUMAN3H-SCH233902-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90119D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90120D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90121D1CLONEDHUMAN3H-SCH233902-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine4100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90122D1CLONEDHUMAN3H-SCH23390Mescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90123D1CLONEDHUMAN3H-SCH23390LSD310Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90124D2CLONEDHUMAN3H-SPIPERONE4-Bromo-2,5-dimethoxyphenethylamine2200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90125D2CLONEDHUMAN3H-SPIPERONE2-(4-chloro-2,5-dimethoxy)ethanamine2100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90126D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-methyl) ethanamine7100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90127D2CLONEDHUMAN3H-SPIPERONE1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane3200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90128D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxyphenethylamine9000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90129D2CLONEDHUMAN3H-SPIPERONE4-iodo-2,5-dimethoxyphenethylamine2700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90130D2CLONEDHUMAN3H-SPIPERONE2-(2,5- dimethoxy-4-nitro)ethanamine6100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90131D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-propylphenyl)ethanamine2300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90132D2CLONEDHUMAN3H-SPIPERONE2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine5100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90133D2CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90134D2CLONEDHUMAN3H-SPIPERONE2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine5000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90135D2CLONEDHUMAN3H-SPIPERONEMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90136D2CLONEDHUMAN3H-SPIPERONE2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine840Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90137D2CLONEDHUMAN3H-SPIPERONE2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1600Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90138D2CLONEDHUMAN3H-SPIPERONE2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2600Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90139D2CLONEDHUMAN3H-SPIPERONE2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1500Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90140D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90141D2CLONEDHUMAN3H-SPIPERONE, 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90142D2CLONEDHUMAN3H-SPIPERONE2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90143D2CLONEDHUMAN3H-SPIPERONE2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine870Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90144D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1600Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90145D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90146D2CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90147D2CLONEDHUMAN3H-SPIPERONEMescaline-NBOMe9600Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90148D2CLONEDHUMAN3H-SPIPERONELSD25Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90149D3CLONEDHUMAN3H-SPIPERONE4-Bromo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90150D3CLONEDHUMAN3H-SPIPERONE2-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90151D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90152D3CLONEDHUMAN3H-SPIPERONE1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90153D3CLONEDHUMAN3H-SPIPERONE2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90154D3CLONEDHUMAN3H-SPIPERONE4-iodo-2,5-dimethoxyphenethylamine5000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90155D3CLONEDHUMAN3H-SPIPERONE2-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90156D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-propylphenyl)ethanamine5200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90157D3CLONEDHUMAN3H-SPIPERONE2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90158D3CLONEDHUMAN3H-SPIPERONE2,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90159D3CLONEDHUMAN3H-SPIPERONE2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine7500Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90160D3CLONEDHUMAN3H-SPIPERONEMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90161D3CLONEDHUMAN3H-SPIPERONE2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90162D3CLONEDHUMAN3H-SPIPERONE2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine3500Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90163D3CLONEDHUMAN3H-SPIPERONE2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90164D3CLONEDHUMAN3H-SPIPERONE2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90165D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90166D3CLONEDHUMAN3H-SPIPERONE2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90167D3CLONEDHUMAN3H-SPIPERONE2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4500Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90168D3CLONEDHUMAN3H-SPIPERONE2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90169D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90170D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90171D3CLONEDHUMAN3H-SPIPERONE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90172D3CLONEDHUMAN3H-SPIPERONEMescaline-NBOMe1700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90173D3CLONEDHUMAN3H-SPIPERONELSD96Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90174CLONEDRAT3H-RO51660174-Bromo-2,5-dimethoxyphenethylamine90Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90175CLONEDRAT3H-RO51660172-(4-chloro-2,5-dimethoxy)ethanamine110Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90176CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-methyl) ethanamine150Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90177CLONEDRAT3H-RO51660171-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane70Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90178CLONEDRAT3H-RO51660172,5-dimethoxyphenethylamine900Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90179CLONEDRAT3H-RO51660174-iodo-2,5-dimethoxyphenethylamine120Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90180CLONEDRAT3H-RO51660172-(2,5- dimethoxy-4-nitro)ethanamine340Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90181CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-propylphenyl)ethanamine20Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90182CLONEDRAT3H-RO51660172-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine40Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90183CLONEDRAT3H-RO51660172,5-dimethoxy-4-isopropylthiophenethylamine50Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90184CLONEDRAT3H-RO51660172-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine;30Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90185CLONEDRAT3H-RO5166017MESCALINE3300Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90186CLONEDRAT3H-RO51660172-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine280Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90187CLONEDRAT3H-RO51660172-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine520Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90188CLONEDRAT3H-RO51660172-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine810Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90189CLONEDRAT3H-RO51660172-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine260Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90190CLONEDRAT3H-RO51660172-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1400Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90191CLONEDRAT3H-RO51660172-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine440Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90192CLONEDRAT3H-RO51660172-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90193CLONEDRAT3H-RO51660172-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine60Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90194CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine350Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90195CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine120Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90196CLONEDRAT3H-RO51660172-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine90Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90197CLONEDRAT3H-RO5166017Mescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90198CLONEDRAT3H-RO5166017LSD450Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90199CLONEDMOUSE3H-RO51660174-Bromo-2,5-dimethoxyphenethylamine3000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90200CLONEDMOUSE3H-RO51660172-(4-chloro-2,5-dimethoxy)ethanamine4100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90201CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-methyl) ethanamine-(4-chloro-2,5-dimethoxy)ethanamine3500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90202CLONEDMOUSE3H-RO51660171-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane1200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90203CLONEDMOUSE3H-RO51660172,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90204CLONEDMOUSE3H-RO51660174-iodo-2,5-dimethoxyphenethylamine3300Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90205CLONEDMOUSE3H-RO51660172-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90206CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-propylphenyl)ethanamine280Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90207CLONEDMOUSE3H-RO51660172-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine2200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90208CLONEDMOUSE3H-RO51660172,5-dimethoxy-4-isopropylthiophenethylamine4500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90209CLONEDMOUSE3H-RO51660172-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine560Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90210CLONEDMOUSE3H-RO5166017MESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90211CLONEDMOUSE3H-RO51660172-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90212CLONEDMOUSE3H-RO51660172-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90213CLONEDMOUSE3H-RO51660172-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90214CLONEDMOUSE3H-RO51660172-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90215CLONEDMOUSE3H-RO51660172-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90216CLONEDMOUSE3H-RO51660172-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90217CLONEDMOUSE3H-RO5166017, 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90218CLONEDMOUSE3H-RO51660172-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine240Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90219CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90220CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90221CLONEDMOUSE3H-RO51660172-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90222CLONEDMOUSE3H-RO5166017Mescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90223CLONEDMOUSE3H-RO5166017LSD>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90224NETCLONEDHUMAN3H-Nisoxetine4-Bromo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90225NETCLONEDHUMAN3H-Nisoxetine2-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90226NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90227NETCLONEDHUMAN3H-Nisoxetine1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90228NETCLONEDHUMAN3H-Nisoxetine2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90229NETCLONEDHUMAN3H-Nisoxetine4-iodo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90230NETCLONEDHUMAN3H-Nisoxetine2-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90231NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-propylphenyl)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90232NETCLONEDHUMAN3H-Nisoxetine2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90233NETCLONEDHUMAN3H-Nisoxetine2,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90234NETCLONEDHUMAN3H-Nisoxetine2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90235NETCLONEDHUMAN3H-NisoxetineMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90236NETCLONEDHUMAN3H-Nisoxetine2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90237NETCLONEDHUMAN3H-Nisoxetine2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90238NETCLONEDHUMAN3H-Nisoxetine2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamin2200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90239NETCLONEDHUMAN3H-Nisoxetine 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine3000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90240NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5500Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90241NETCLONEDHUMAN3H-Nisoxetine2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1300Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90242NETCLONEDHUMAN3H-Nisoxetine2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90243NETCLONEDHUMAN3H-Nisoxetine2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90244NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5900Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90245NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4300Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90246NETCLONEDHUMAN3H-Nisoxetine2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine3700Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90247NETCLONEDHUMAN3H-NisoxetineMescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90248NETCLONEDHUMAN3H-NisoxetineLSD>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90249DATCLONEDHUMAN3H-WIN 35,4284-Bromo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90250DATCLONEDHUMAN3H-WIN 35,4282-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90251DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90252DATCLONEDHUMAN3H-WIN 35,4281-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90253DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90254DATCLONEDHUMAN3H-WIN 35,4284-iodo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90255DATCLONEDHUMAN3H-WIN 35,4282-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90256DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-propylphenyl)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90257DATCLONEDHUMAN3H-WIN 35,4282-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamin>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90258DATCLONEDHUMAN3H-WIN 35,4282,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90259DATCLONEDHUMAN3H-WIN 35,4282-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90260DATCLONEDHUMAN3H-WIN 35,428MESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90261DATCLONEDHUMAN3H-WIN 35,4282-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine7200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90262DATCLONEDHUMAN3H-WIN 35,4282-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90263DATCLONEDHUMAN3H-WIN 35,4282-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90264DATCLONEDHUMAN3H-WIN 35,4282-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine8100Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90265DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90266DATCLONEDHUMAN3H-WIN 35,4282-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5400Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90267DATCLONEDHUMAN3H-WIN 35,4282-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90268DATCLONEDHUMAN3H-WIN 35,4282-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4700Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90269DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine8600Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90270DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine6200Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90271DATCLONEDHUMAN3H-WIN 35,4282-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine4800Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90272DATCLONEDHUMAN3H-WIN 35,428Mescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90273DATCLONEDHUMAN3H-WIN 35,428LSD>10000Rickli A et al 2015Jan 15, 2025Jan 15, 2025
90274SERTCLONEDHUMAN3H-CITALOPRAM4-Bromo-2,5-dimethoxyphenethylamine9700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90275SERTCLONEDHUMAN3H-CITALOPRAM2-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90276SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90277SERTCLONEDHUMAN3H-CITALOPRAM1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90278SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90279SERTCLONEDHUMAN3H-CITALOPRAM4-iodo-2,5-dimethoxyphenethylamine4900Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90280SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90281SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-propylphenyl)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90282SERTCLONEDHUMAN3H-CITALOPRAM2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90283SERTCLONEDHUMAN3H-CITALOPRAM2,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90284SERTCLONEDHUMAN3H-CITALOPRAM2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90285SERTCLONEDHUMAN3H-CITALOPRAMMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90286SERTCLONEDHUMAN3H-CITALOPRAM2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine840Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90287SERTCLONEDHUMAN3H-CITALOPRAM2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1500Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90288SERTCLONEDHUMAN3H-CITALOPRAM2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90289SERTCLONEDHUMAN3H-CITALOPRAM2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90290SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine2300Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90291SERTCLONEDHUMAN3H-CITALOPRAM2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90292SERTCLONEDHUMAN3H-CITALOPRAM2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90293SERTCLONEDHUMAN3H-CITALOPRAM2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90294SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90295SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine8100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90296SERTCLONEDHUMAN3H-CITALOPRAM2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine3200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90297SERTCLONEDHUMAN3H-CITALOPRAMMescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90298SERTCLONEDHUMAN3H-CITALOPRAMLSD>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90299H1CLONEDHUMAN3H-PYRILAMINE4-Bromo-2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90300H1CLONEDHUMAN3H-PYRILAMINE2-(4-chloro-2,5-dimethoxy)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90301H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-methyl) ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90302H1CLONEDHUMAN3H-PYRILAMINE1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90303H1CLONEDHUMAN3H-PYRILAMINE2,5-dimethoxyphenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90304H1CLONEDHUMAN3H-PYRILAMINE4-iodo-2,5-dimethoxyphenethylamine6100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90305H1CLONEDHUMAN3H-PYRILAMINE2-(2,5- dimethoxy-4-nitro)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90306H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-propylphenyl)ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90307H1CLONEDHUMAN3H-PYRILAMINE2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90308H1CLONEDHUMAN3H-PYRILAMINE2,5-dimethoxy-4-isopropylthiophenethylamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90309H1CLONEDHUMAN3H-PYRILAMINE2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90310H1CLONEDHUMAN3H-PYRILAMINEMESCALINE>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90311H1CLONEDHUMAN3H-PYRILAMINE2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine80Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90312H1CLONEDHUMAN3H-PYRILAMINE2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine90Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90313H1CLONEDHUMAN3H-PYRILAMINE2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine630Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90314H1CLONEDHUMAN3H-PYRILAMINE2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90315H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine4100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90316H1CLONEDHUMAN3H-PYRILAMINE2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine90Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90317H1CLONEDHUMAN3H-PYRILAMINE2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine210Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90318H1CLONEDHUMAN3H-PYRILAMINE2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine1700Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90319H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine490Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90320H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine5400Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90321H1CLONEDHUMAN3H-PYRILAMINE2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine1200Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90322H1CLONEDHUMAN3H-PYRILAMINEMescaline-NBOMe>10000Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90323H1CLONEDHUMAN3H-PYRILAMINELSD1100Rickli A et al 2015Jan 15, 2025Jan 28, 2025
90324A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide113Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90325A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide146Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90326A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide509Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90327A1brain membranesRAT3H-CCPAN-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide120Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90328A1brain membranesRAT3H-CCPAN-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide136Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90329A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90330A1brain membranesRAT3H-CCPAN-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide1370Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90331A1brain membranesRAT3H-CCPAN-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide145Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90332A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide563Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90333A1brain membranesRAT3H-CCPAN-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90334A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90335A1brain membranesRAT3H-CCPA2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90336A1brain membranesRAT3H-CCPAN-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90337A1brain membranesRAT3H-CCPAN-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide605Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90338A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide50.7Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90339A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide24.8Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90340A1brain membranesRAT3H-CCPAN-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide320Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90341A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide181Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90342A1brain membranesRAT3H-CCPAN-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide684Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90343A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1590Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90344A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1010Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90345A1brain membranesRAT3H-CCPAN-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide118Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90346A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide382Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90347A1brain membranesRAT3H-CCPAN-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide194Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90348A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide36.6Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90349A1brain membranesRAT3H-CCPA2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90350A1brain membranesRAT3H-CCPAN-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide593Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90351A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide551Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90352A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide320Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90353A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide1120Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90354A2AStriatal MembranesRAT3H-MSX-2N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide271Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90355A2AStriatal MembranesRAT3H-MSX-2N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide303Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90356A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90357A2AStriatal MembranesRAT3H-MSX-2N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide807Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90358A2AStriatal MembranesRAT3H-MSX-2N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide335Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90359A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1360Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90360A2AStriatal MembranesRAT3H-MSX-2N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide3230Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90361A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1360Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90362A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide1870Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90363A2AStriatal MembranesRAT3H-MSX-2N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90364A2AStriatal MembranesRAT3H-MSX-2N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide637Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90365A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide242Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90366A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide318Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90367A2AStriatal MembranesRAT3H-MSX-2N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1290Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90368A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide671Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90369A2AStriatal MembranesRAT3H-MSX-2N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide6520Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90370A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1630Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90371A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide>10000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90372A2AStriatal MembranesRAT3H-MSX-2N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide1250Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90373A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1070Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90374A2AStriatal MembranesRAT3H-MSX-2N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide569Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90375A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide455Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90376A2AStriatal MembranesRAT3H-MSX-22-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide2270Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90377A2AStriatal MembranesRAT3H-MSX-2N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide7310Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90378A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide193Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90379A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide452Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90380A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide911Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90381A2BCLONEDHUMAN3H-PSB-603N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide179Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90382A2BCLONEDHUMAN3H-PSB-603N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide340Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90383A2BCLONEDHUMAN3H-PSB-603N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide306Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90384A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90385A2BCLONEDHUMAN3H-PSB-603N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90386A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90387A2BCLONEDHUMAN3H-PSB-603N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90388A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90389A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90390A2BCLONEDHUMAN3H-PSB-603N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90391A2BCLONEDHUMAN3H-PSB-603N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide862Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90392A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide113Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90393A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide126Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90394A2BCLONEDHUMAN3H-PSB-603N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide578Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90395A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide298Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90396A2BCLONEDHUMAN3H-PSB-603N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90397A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90398A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90399A2BCLONEDHUMAN3H-PSB-603N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide215Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90400A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90401A2BCLONEDHUMAN3H-PSB-603N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide275Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90402A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide66.3Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90403A2BCLONEDHUMAN3H-PSB-6032-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90404A2BCLONEDHUMAN3H-PSB-603N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90405A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide509Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90406A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90407A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90408A3CLONEDHUMAN3H-PSB-11N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide508Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90409A3CLONEDHUMAN3H-PSB-11N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90410A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90411A3CLONEDHUMAN3H-PSB-11N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide572Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90412A3CLONEDHUMAN3H-PSB-11N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide458Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90413A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90414A3CLONEDHUMAN3H-PSB-11N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90415A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90416A3CLONEDHUMAN3H-PSB-112-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90417A3CLONEDHUMAN3H-PSB-11N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide1090Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90418A3CLONEDHUMAN3H-PSB-11N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90419A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide155Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90420A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide248Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90421A3CLONEDHUMAN3H-PSB-11N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide602Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90422A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90423A3CLONEDHUMAN3H-PSB-11N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90424A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90425A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90426A3CLONEDHUMAN3H-PSB-11N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide353Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90427A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90428A3CLONEDHUMAN3H-PSB-11N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide868Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90429A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide204Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90430A3CLONEDHUMAN3H-PSB-112-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90431A3CLONEDHUMAN3H-PSB-11N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide1000Zaluski M et al 2018Jan 15, 2025Jan 15, 2025
90432D2CLONEDHUMAN125I-IABN1-((1H-Indol-3-yl)methyl)-4-(1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate)piperidin-4-ol oxalate3.8Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90433D2CLONEDHUMAN125I-IABN4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate0.9Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90434D2CLONEDHUMAN125I-IABN4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate0.9Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90435D2CLONEDHUMAN125I-IABN1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate1396Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90436D2CLONEDHUMAN125I-IABN4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate27.7Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90437D2CLONEDHUMAN125I-IABN4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate13.8Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90438D2CLONEDHUMAN125I-IABN1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate23.3Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90439D2CLONEDHUMAN125I-IABN1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate12.5Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90440D2CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate212Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90441D2CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate61Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90442D2CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate254Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90443D2CLONEDHUMAN125I-IABN1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate17.3Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90444D2CLONEDHUMAN125I-IABN1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate14.3Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90445D2CLONEDHUMAN125I-IABN1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate46.8Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90446D2CLONEDHUMAN125I-IABN1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate6.6Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90447D2CLONEDHUMAN125I-IABN1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate2.4Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90448D2CLONEDHUMAN125I-IABN1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate13.6Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90449D2CLONEDHUMAN125I-IABN1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate37.8Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90450D2CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate7.1Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90451D2CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate8Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90452D2CLONEDHUMAN125I-IABN8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate71.4Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90453D2CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate2Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90454D2CLONEDHUMAN125I-IABNHALOPERIDOL1.1Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90455D3CLONEDHUMAN125I-IABNHALOPERIDOL12.7Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90456D3CLONEDHUMAN125I-IABN1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate94.4Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90457D4CLONEDHUMAN125I-IABN1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate53.4Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90458D4CLONEDHUMAN125I-IABN4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate60.4Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90459D3CLONEDHUMAN125I-IABN4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate122Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90460D3CLONEDHUMAN125I-IABN4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate100Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90461D4CLONEDHUMAN125I-IABN4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate129Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90462D4CLONEDHUMAN125I-IABN1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90463D3CLONEDHUMAN125I-IABN1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate2927Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90464D3CLONEDHUMAN125I-IABN4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate849Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90465D4CLONEDHUMAN125I-IABN4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate668Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90466D4CLONEDHUMAN125I-IABN4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate344Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90467D3CLONEDHUMAN125I-IABN4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate188Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90468D3CLONEDHUMAN125I-IABN1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate132Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90469D4CLONEDHUMAN125I-IABN1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate1390Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90470D4CLONEDHUMAN125I-IABN1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate2230Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90471D3CLONEDHUMAN125I-IABN1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate68.2Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90472D3CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate2983Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90473D4CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate620Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90474D4CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate634Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90475D3CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate1585Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90476D3CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate4938Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90477D4CLONEDHUMAN125I-IABN1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate937Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90478D4CLONEDHUMAN125I-IABN1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate254Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90479D3CLONEDHUMAN125I-IABN1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate31.8Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90480D3CLONEDHUMAN125I-IABN1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate49Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90481D4CLONEDHUMAN125I-IABN1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate245Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90482D4CLONEDHUMAN125I-IABN1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate377Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90483D3CLONEDHUMAN125I-IABN1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate142Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90484D3CLONEDHUMAN125I-IABN1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate10.9Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90485D4CLONEDHUMAN125I-IABN1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate94.5Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90486D4CLONEDHUMAN125I-IABN1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate40.4Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90487D3CLONEDHUMAN125I-IABN1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate11.2Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90488D3CLONEDHUMAN125I-IABN1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate3Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90489D4CLONEDHUMAN125I-IABN1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate163Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90490D4CLONEDHUMAN125I-IABN1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate72.6Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90491D3CLONEDHUMAN125I-IABN1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate46.7Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90492D3CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate2.1Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90493D4CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate492Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90494D4CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate945Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90495D3CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate9.3Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90496D3CLONEDHUMAN125I-IABN8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate60.1Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90497D4CLONEDHUMAN125I-IABN8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate352Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90498D4CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate978Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90499D3CLONEDHUMAN125I-IABN8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate0.9Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90500Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate2Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90501Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate881Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90502Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate197Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90503Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate1527Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90504Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate3224Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90505Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate227Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90506Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate4129Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90507Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate1768Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90508Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate15.1Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90509Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate1.2Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90510Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate8.07Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90511Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate2.45Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90512Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate1.41Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90513Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate2.13Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90514Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate0.59Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90515Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate0.51Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90516Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate1779Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90517Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate1879Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90518Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate708Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90519Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate28Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90520Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate331Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90521Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate802Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90522Sigma 1brain membranesGUINEA PIG3H-Pentazocine(+)HALOPERIDOL1.45Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90523Sigma 2liver membranesRAT3H-DTGHALOPERIDOL24.2Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90524Sigma 2liver membranesRAT3H-DTG1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate2200Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90525Sigma 2liver membranesRAT3H-DTG4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate970Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90526Sigma 2liver membranesRAT3H-DTG4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate3262Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90527Sigma 2liver membranesRAT3H-DTG1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate2761Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90528Sigma 2liver membranesRAT3H-DTG4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate9510Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90529Sigma 2liver membranesRAT3H-DTG4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90530Sigma 2liver membranesRAT3H-DTG1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90531Sigma 2liver membranesRAT3H-DTG1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90532Sigma 2liver membranesRAT3H-DTG1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate1.9Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90533Sigma 2liver membranesRAT3H-DTG1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate5.53Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90534Sigma 2liver membranesRAT3H-DTG1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate7.75Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90535Sigma 2liver membranesRAT3H-DTG1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate1398Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90536Sigma 2liver membranesRAT3H-DTG1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate2368Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90537Sigma 2liver membranesRAT3H-DTG1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate1964Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90538Sigma 2liver membranesRAT3H-DTG1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate377Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90539Sigma 2liver membranesRAT3H-DTG1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate393Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90540Sigma 2liver membranesRAT3H-DTG1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90541Sigma 2liver membranesRAT3H-DTG1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90542Sigma 2liver membranesRAT3H-DTG8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90543Sigma 2liver membranesRAT3H-DTG8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90544Sigma 2liver membranesRAT3H-DTG8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90545Sigma 2liver membranesRAT3H-DTG8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate>10000Vangveravong S et al 2010Jan 15, 2025Jan 28, 2025
90546A1CORTICAL MEMBRANESRAT3H-CCPAPreladenant (SCH420814)68.7 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90547A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide422 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90548A1CORTICAL MEMBRANESRAT3H-CCPA3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide367 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90549A1CORTICAL MEMBRANESRAT3H-CCPA3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90550A1CORTICAL MEMBRANESRAT3H-CCPA3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90551A1CORTICAL MEMBRANESRAT3H-CCPA3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90552A1CORTICAL MEMBRANESRAT3H-CCPA2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90553A1CORTICAL MEMBRANESRAT3H-CCPA(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide205 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90554A1CORTICAL MEMBRANESRAT3H-CCPA(E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90555A1CORTICAL MEMBRANESRAT3H-CCPA3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90556A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide229 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90557A1CORTICAL MEMBRANESRAT3H-CCPA4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide22.5 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90558A1CORTICAL MEMBRANESRAT3H-CCPA4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide898 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90559A1CORTICAL MEMBRANESRAT3H-CCPA4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90560A1CORTICAL MEMBRANESRAT3H-CCPA(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide53 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90561A1CORTICAL MEMBRANESRAT3H-CCPA(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide11.2 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90562A1CORTICAL MEMBRANESRAT3H-CCPA(E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide11.4 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90563A1CORTICAL MEMBRANESRAT3H-CCPA(E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide1500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90564A1CORTICAL MEMBRANESRAT3H-CCPAN-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide98.3 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90565A1CORTICAL MEMBRANESRAT3H-CCPAN-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90566A1CORTICAL MEMBRANESRAT3H-CCPAN-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90567A1CORTICAL MEMBRANESRAT3H-CCPAN-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90568A1CORTICAL MEMBRANESRAT3H-CCPAN-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide64.4 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90569A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90570A1CORTICAL MEMBRANESRAT3H-CCPAN-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide35.2 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90571A1CORTICAL MEMBRANESRAT3H-CCPAN-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90572A2AStriatal MembranesRAT3H-MSX-2Preladenant (SCH420814)0.66 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90573A2AStriatal MembranesRAT3H-MSX-2N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide103 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90574A2AStriatal MembranesRAT3H-MSX-23-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide294 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90575A2AStriatal MembranesRAT3H-MSX-23-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90576A2AStriatal MembranesRAT3H-MSX-23-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide2190 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90577A2AStriatal MembranesRAT3H-MSX-23-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90578A2AStriatal MembranesRAT3H-MSX-22-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90579A2AStriatal MembranesRAT3H-MSX-2(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide253 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90580A2AStriatal MembranesRAT3H-MSX-2(E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90581A2AStriatal MembranesRAT3H-MSX-23-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide1720 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90582A2AStriatal MembranesRAT3H-MSX-2N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide423 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90583A2AStriatal MembranesRAT3H-MSX-24-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide558 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90584A2AStriatal MembranesRAT3H-MSX-24-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90585A2AStriatal MembranesRAT3H-MSX-24-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90586A2AStriatal MembranesRAT3H-MSX-2(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide814 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90587A2AStriatal MembranesRAT3H-MSX-2(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide317 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90588A2AStriatal MembranesRAT3H-MSX-2(E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90589A2AStriatal MembranesRAT3H-MSX-2(E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90590A2AStriatal MembranesRAT3H-MSX-24-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90591A2AStriatal MembranesRAT3H-MSX-24-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide84.7 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90592A2AStriatal MembranesRAT3H-MSX-24-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide488 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90593A2AStriatal MembranesRAT3H-MSX-2N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90594A2AStriatal MembranesRAT3H-MSX-2N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide6060 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90595A2AStriatal MembranesRAT3H-MSX-2N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90596A2AStriatal MembranesRAT3H-MSX-2N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90597A2AStriatal MembranesRAT3H-MSX-2N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90598A2AStriatal MembranesRAT3H-MSX-2N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90599A2AStriatal MembranesRAT3H-MSX-2N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide693 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90600A2AStriatal MembranesRAT3H-MSX-2N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90601A1CLONEDHUMAN3H-CCPAPreladenant (SCH420814)295 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90602A1CLONEDHUMAN3H-CCPAN-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide1050 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90603A1CLONEDHUMAN3H-CCPA3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1370 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90604A1CLONEDHUMAN3H-CCPA(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90605A1CLONEDHUMAN3H-CCPAN-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide2500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90606A1CLONEDHUMAN3H-CCPA4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide214 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90607A1CLONEDHUMAN3H-CCPA4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide>10000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90608A1CLONEDHUMAN3H-CCPA(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide822 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90609A1CLONEDHUMAN3H-CCPA(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide500 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90610A1CLONEDHUMAN3H-CCPA(E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide562 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90611A1CLONEDHUMAN3H-CCPA4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90612A1CLONEDHUMAN3H-CCPA4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90613A1CLONEDHUMAN3H-CCPA4-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide4370 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90614A1CLONEDHUMAN3H-CCPAN-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide785 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90615A1CLONEDHUMAN3H-CCPAN-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide364 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90616A2ACLONEDHUMAN3H-MSX-2Preladenant (SCH420814)0.884 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90617A2ACLONEDHUMAN3H-MSX-2N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide80.9 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90618A2ACLONEDHUMAN3H-MSX-23-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide64.9 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90619A2ACLONEDHUMAN3H-MSX-2(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide62.4 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90620A2ACLONEDHUMAN3H-MSX-2(E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90621A2ACLONEDHUMAN3H-MSX-23-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90622A2ACLONEDHUMAN3H-MSX-2N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide39.5 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90623A2ACLONEDHUMAN3H-MSX-24-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide115 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90624A2ACLONEDHUMAN3H-MSX-2(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide118 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90625A2ACLONEDHUMAN3H-MSX-2(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide91.8 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90626A2ACLONEDHUMAN3H-MSX-24-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90627A2ACLONEDHUMAN3H-MSX-24-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide58.3 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90628A2ACLONEDHUMAN3H-MSX-2N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide82.5 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90629A2BCLONEDHUMAN3H-PSB-603Preladenant (SCH420814)1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90630A2BCLONEDHUMAN3H-PSB-603N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide365 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90631A2BCLONEDHUMAN3H-PSB-6033-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide225 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90632A2BCLONEDHUMAN3H-PSB-6033-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90633A2BCLONEDHUMAN3H-PSB-6033-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide801 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90634A2BCLONEDHUMAN3H-PSB-6033-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90635A2BCLONEDHUMAN3H-PSB-6032-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90636A2BCLONEDHUMAN3H-PSB-603(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide679 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90637A2BCLONEDHUMAN3H-PSB-603(E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90638A2BCLONEDHUMAN3H-PSB-6033-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90639A2BCLONEDHUMAN3H-PSB-603N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90640A2BCLONEDHUMAN3H-PSB-6034-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide302 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90641A2BCLONEDHUMAN3H-PSB-6034-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90642A2BCLONEDHUMAN3H-PSB-6034-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90643A2BCLONEDHUMAN3H-PSB-603(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide119 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90644A2BCLONEDHUMAN3H-PSB-603(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90645A2BCLONEDHUMAN3H-PSB-603(E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90646A2BCLONEDHUMAN3H-PSB-603(E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90647A2BCLONEDHUMAN3H-PSB-6034-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90648A2BCLONEDHUMAN3H-PSB-6034-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90649A2BCLONEDHUMAN3H-PSB-6034-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90650A2BCLONEDHUMAN3H-PSB-603N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90651A2BCLONEDHUMAN3H-PSB-603N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide408 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90652A2BCLONEDHUMAN3H-PSB-603N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90653A2BCLONEDHUMAN3H-PSB-603N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90654A2BCLONEDHUMAN3H-PSB-603N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90655A2BCLONEDHUMAN3H-PSB-603N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide547 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90656A2BCLONEDHUMAN3H-PSB-603N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide361 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90657A2BCLONEDHUMAN3H-PSB-603N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90658A3CLONEDHUMAN3H-PSB-11Preladenant (SCH420814)1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90659A3CLONEDHUMAN3H-PSB-11N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide390 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90660A3CLONEDHUMAN3H-PSB-113-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide173 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90661A3CLONEDHUMAN3H-PSB-113-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90662A3CLONEDHUMAN3H-PSB-113-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90663A3CLONEDHUMAN3H-PSB-113-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90664A3CLONEDHUMAN3H-PSB-112-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90665A3CLONEDHUMAN3H-PSB-11(E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90666A3CLONEDHUMAN3H-PSB-11(E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90667A3CLONEDHUMAN3H-PSB-113-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90668A3CLONEDHUMAN3H-PSB-11N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90669A3CLONEDHUMAN3H-PSB-114-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide382 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90670A3CLONEDHUMAN3H-PSB-114-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90671A3CLONEDHUMAN3H-PSB-114-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90672A3CLONEDHUMAN3H-PSB-11(E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide158 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90673A3CLONEDHUMAN3H-PSB-11(E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide115 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90674A3CLONEDHUMAN3H-PSB-11(E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90675A3CLONEDHUMAN3H-PSB-11(E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90676A3CLONEDHUMAN3H-PSB-114-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90677A3CLONEDHUMAN3H-PSB-114-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90678A3CLONEDHUMAN3H-PSB-114-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90679A3CLONEDHUMAN3H-PSB-11N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90680A3CLONEDHUMAN3H-PSB-11N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide147 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90681A3CLONEDHUMAN3H-PSB-11N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90682A3CLONEDHUMAN3H-PSB-11N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90683A3CLONEDHUMAN3H-PSB-11N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide91.6 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90684A3CLONEDHUMAN3H-PSB-11N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90685A3CLONEDHUMAN3H-PSB-11N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90686A3CLONEDHUMAN3H-PSB-11N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide1000 Stossel A et al 2013Jan 15, 2025Jan 15, 2025
90687Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine12Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90688Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine5.7Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90689Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine4.9Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90690Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine2.3Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90691Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine183Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90692Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine36Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90693Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine15Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90694Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine8.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90695Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine19Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90696Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine5.8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90697Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine3.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90698Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine1.9Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90699Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine19Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90700Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine20Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90701Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90702Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine8.2Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90703Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine15Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90704Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine18Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90705Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine8Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90706Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine3.1Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90707Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine262Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90708Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine50Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90709Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)trans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine256Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90710Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine97Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90711Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)PENTAZOCINE (+)5.4Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90712Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)DTG71Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90713Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine53Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90714Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine67Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90715Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine81Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90716Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine33Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90717Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine161Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90718Sigma 2liver membranesRAT3H-DTGcis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine308Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90719Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine361Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90720Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine42Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90721Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine128Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90722Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine101Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90723Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine154Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90724Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine12Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90725Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine133Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90726Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine52Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90727Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine164Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90728Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine70Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90729Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine99Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90730Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine84Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90731Sigma 2liver membranesRAT3H-DTGtrans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine175Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90732Sigma 2liver membranesRAT3H-DTGcis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine30Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90733Sigma 2liver membranesRAT3H-DTGtrans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90734Sigma 2liver membranesRAT3H-DTGcis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine751Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90735Sigma 2liver membranesRAT3H-DTGtrans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine1000Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90736Sigma 2liver membranesRAT3H-DTGcis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine503Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90737Sigma 2liver membranesRAT3H-DTGDTG54Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90738Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine7Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90739Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine6.7Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90740Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine16Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90741Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine4.6Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90742Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine16Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90743Sigma 2CLONEDHUMAN3H-DTGcis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine46Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90744Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine93Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90745Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine14Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90746Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine13Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90747Sigma 2CLONEDHUMAN3H-DTGtrans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine39Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025
90748Sigma 2CLONEDHUMAN3H-DTGcis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine11Kronenberg E et al 2019Jan 15, 2025Jan 28, 2025