89749 nAChR CORTEX RAT 3H-Cytisine (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 29, 2025
89750 5-HT3 CLONED HUMAN 3H-GR-65630 (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89751 Calcium channel CLONED HUMAN 3H-Nitrendipine (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 28, 2025
89752 hERG CLONED HUMAN 3H-Dofetilide (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89753 Sodium Channel CLONED HUMAN 3H-Batrachotoxin (3-Chloro-4-fluorophenyl)(4-fluoro-4-(((2-(pyridin-2-yloxy)ethyl)- amino)methyl)piperidin-1-yl)methanone >10000 Sniecikowska J et al 2019 Jan 15, 2025 Jan 15, 2025
89754 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 38.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89755 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89756 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 957 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89757 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89758 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 194 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89759 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 5670 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89760 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 16.2 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89761 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 2500 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89762 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 171 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89763 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89764 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 13.1 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89765 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 60.2 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89766 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 1230 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89767 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 81 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89768 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89769 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 2840 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89770 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89771 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 28.2 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89772 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 293 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89773 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 5790 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89774 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 250 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89775 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89776 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 5700 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89777 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89778 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 141 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89779 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 838 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89780 nAChR CLONED HUMAN 3H-Epibatidine 3-[(1-Methyl-2(S)-azetidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89781 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride 445 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89782 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(piperidinyl)pyridine Hydrochloride 23.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89783 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89784 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride 4170 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89785 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89786 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride 297 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89787 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride 1570 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89788 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-(pyrrolidinyl)pyridine Hydrochloride 1680 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89789 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride 126 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89790 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89791 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride 8070 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89792 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89793 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride 54.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89794 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride 426 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89795 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(morpholinyl)pyridine Hydrochloride 8630 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89796 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride 61.8 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89797 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89798 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride 2130 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89799 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89800 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride 27.7 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89801 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride 213 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89802 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(thiomorpholinyl)pyridine Hydrochloride 4110 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89803 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 69.7 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89804 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 8870 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89805 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 166 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89806 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89807 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 39.2 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89808 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 104 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89809 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-pyrrolidinyl)methoxy]-5-(piperazinyl)pyridine Hydrochloride 7080 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89810 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 57.9 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89811 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 349 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89812 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 3220 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89813 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 6270 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89814 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 13.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89815 nAChR FOREBRAIN RAT 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 366 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89816 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-Indolinyl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 225 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89817 nAChR CLONED HUMAN 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 158 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89818 nAChR CLONED HUMAN 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89819 nAChR CLONED HUMAN 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 812 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89820 nAChR CLONED HUMAN 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89821 nAChR CLONED HUMAN 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 50.9 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89822 nAChR FOREBRAIN RAT 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 509 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89823 nAChR CLONED HUMAN 3H-Epibatidine 3-(1,3-Dihydro-2H-isoindol-2-yl)-5-[(2(S)-pyrrolidinyl)methoxy]pyridine Hydrochloride 3960 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89824 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 6.5 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89825 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 104 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89826 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 208 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89827 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 793 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89828 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 2.4 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89829 nAChR FOREBRAIN RAT 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 55.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89830 nAChR CLONED HUMAN 3H-Epibatidine 3-(1-indolyl)-5-(2(S)-pyrrolidinylmethoxy)pyridine Hydrochloride 70.6 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89831 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 20.5 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89832 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 4160 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89833 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 383 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89834 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89835 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 18.8 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89836 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 100 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89837 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-butylaminopyridine Hydrochloride 1790 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89838 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 1.7 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89839 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 559 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89840 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 40.6 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89841 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 5640 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89842 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 1.2 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89843 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 1.4 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89844 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-phenylaminopyridine Hydrochloride 16.9 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89845 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 12.5 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89846 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 937 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89847 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 150 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89848 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89849 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 13.2 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89850 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 63.4 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89851 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-benzylaminopyridine Hydrochloride 503 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89852 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 357 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89853 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 1970 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89854 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 1290 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89855 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89856 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 190 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89857 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 1150 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89858 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-diethylaminopyridine Hydrochloride 108 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89859 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 124 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89860 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 631 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89861 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 953 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89862 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 9520 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89863 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 59.3 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89864 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 374 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89865 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-ethyl-N-phenyl)amino]pyridine Hydrochloride 378 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89866 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 133 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89867 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 3400 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89868 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 628 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89869 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride >10000 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89870 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 48.8 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89871 nAChR FOREBRAIN RAT 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 380 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89872 nAChR CLONED HUMAN 3H-Epibatidine 3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(N-methyl-N-benzyl)amino]pyridine Hydrochloride 192 Liu J et al 2010 Jan 15, 2025 Jan 29, 2025
89873 nAChR CLONED HUMAN 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89874 nAChR CLONED HUMAN 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine 1820 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89875 nAChR CLONED HUMAN 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89876 nAChR CLONED HUMAN 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine 6100 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89877 nAChR CORTICAL MEMBRANES RAT 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89878 nAChR CLONED HUMAN 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine 5580 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89879 nAChR CLONED HUMAN 3H-Epibatidine 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine 2220 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89880 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine 103 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89881 Sigma 2 CLONED HUMAN 3H-DTG 3-[[3-(2(S)-Azetidinylmethoxy)isoxazol-5-yl]methoxy]-5-chloropyridine >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89882 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89883 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89884 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89885 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89886 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89887 nAChR CORTICAL MEMBRANES RAT 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89888 nAChR CLONED HUMAN 3H-Epibatidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 29, 2025
89889 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 4.1 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89890 Sigma 2 CLONED HUMAN 3H-DTG 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 1312 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89891 5-HT1A CLONED HUMAN 3H-WAY100635 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89892 5-HT1B CLONED HUMAN 3H-5-CT 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89893 5-HT1D CLONED HUMAN 3H-5-CT 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89894 5-HT1E CLONED HUMAN 3H-5-HT 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89895 5-HT2A CLONED HUMAN 3H-KETANSERIN 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 4406 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89896 5-HT2B CLONED HUMAN 3H-LSD 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 5097 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89897 5-HT2C CLONED HUMAN 3H-MESULERGINE 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89898 5-HT3 CLONED HUMAN 3H-GR-65630 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89899 5-HT5A CLONED HUMAN 3H-LSD 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89900 5-HT6 CLONED HUMAN 3H-LSD 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89901 5-HT7 CLONED HUMAN 3H-LSD 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89902 KOR CLONED HUMAN 3H-MUSCIMOL 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 27, 2025
89903 D1 CLONED HUMAN 3H-SCH23390 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89904 D5 CLONED HUMAN 3H-SCH23390 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89905 D2 CLONED HUMAN 3H-N-Methylspiperone 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89906 D3 CLONED HUMAN 3H-N-Methylspiperone 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89907 D4 CLONED HUMAN 3H-N-Methylspiperone 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89908 BZP CORTICAL MEMBRANES RAT FNZ 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89909 Alpha1A CLONED HUMAN 3H-PRAZOSIN 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89910 Alpha1B CLONED HUMAN 3H-PRAZOSIN 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89911 Alpha1D CLONED HUMAN 3H-PRAZOSIN 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89912 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89913 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89914 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89915 Beta 1 CLONED HUMAN 125I-Pindolol 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89916 Beta3 CLONED HUMAN 125I-Pindolol 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89917 Beta 2 CLONED HUMAN 3H-CGP-12177 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89918 H1 CLONED HUMAN 3H-PYRILAMINE 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89919 5-HT1D CLONED HUMAN 3H-Cimetidine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 5157 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89920 H3 CLONED HUMAN 3H-Alpha-methylhistamine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89921 H4 CLONED HUMAN 3H-Histamine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89922 M1 CLONED HUMAN 3H-QNB 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89923 M2 CLONED HUMAN 3H-QNB 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89924 M3 CLONED HUMAN 3H-QNB 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89925 M4 CLONED HUMAN 3H-QNB 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89926 M5 CLONED HUMAN 3H-QNB 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89927 DOR CLONED HUMAN 3H-DADLE 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89928 KOR CLONED HUMAN 3H-U69593 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89929 MOR CLONED HUMAN 3H-DAMGO 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89930 DAT CLONED HUMAN 3H-WIN35428 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 373 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89931 NET CLONED HUMAN 3H-Nisoxetine 5-(Phenoxymethyl)-3-(2(S)-pyrrolidinylmethoxy)isoxazole 203 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89932 5-HT1A CLONED HUMAN 3H-WAY100635 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89933 5-HT1B CLONED HUMAN 3H-5-CT 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89934 5-HT1D CLONED HUMAN 3H-5-CT 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89935 5-HT1E CLONED HUMAN 3H-5-HT 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89936 5-HT2A CLONED HUMAN 3H-KETANSERIN 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole 6405 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89937 5-HT2B CLONED HUMAN 3H-LSD 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89938 5-HT2C CLONED HUMAN 3H-MESULERGINE 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89939 5-HT3 CLONED HUMAN 3H-GR-65630 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89940 5-HT5A CLONED HUMAN 3H-LSD 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89941 5-HT6 CLONED HUMAN 3H-LSD 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89942 5-HT7 CLONED HUMAN 3H-LSD 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89943 KOR CLONED HUMAN 3H-MUSCIMOL 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 27, 2025
89944 D1 CLONED HUMAN 3H-SCH23390 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89945 D5 CLONED HUMAN 3H-SCH23390 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89946 D2 CLONED HUMAN 3H-N-Methylspiperone 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89947 D3 CLONED HUMAN 3H-N-Methylspiperone 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89948 D4 CLONED HUMAN 3H-N-Methylspiperone 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89949 BZP CORTICAL MEMBRANES RAT FNZ 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89950 Alpha1A CLONED HUMAN 3H-PRAZOSIN 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89951 Alpha1B CLONED HUMAN 3H-PRAZOSIN 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89952 Alpha1D CLONED HUMAN 3H-PRAZOSIN 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89953 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89954 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89955 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89956 Beta 1 CLONED HUMAN 125I-Pindolol 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89957 Beta3 CLONED HUMAN 125I-Pindolol 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89958 Beta 2 CLONED HUMAN 3H-CGP12177 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89959 H1 CLONED HUMAN 3H-PYRILAMINE 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89960 5-HT1D CLONED HUMAN 3H-Cimetidine 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89961 H3 CLONED HUMAN 3H-Alpha-methylhistamine 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89962 H4 CLONED HUMAN 3H-Histamine 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89963 M1 CLONED HUMAN 3H-QNB 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89964 M2 CLONED HUMAN 3H-QNB 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89965 M3 CLONED HUMAN 3H-QNB 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89966 M4 CLONED HUMAN 3H-QNB 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89967 M5 CLONED HUMAN 3H-QNB 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89968 DOR CLONED HUMAN 3H-DADLE 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89969 KOR CLONED HUMAN 3H-U69593 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89970 MOR CLONED HUMAN 3H-DAMGO 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89971 DAT CLONED HUMAN 3H-WIN 35,428 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole 24 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89972 NET CLONED HUMAN 3H-Nisoxetine 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole 191 Yu LF et al 2012 Jan 15, 2025 Jan 15, 2025
89973 SERT CLONED HUMAN 3H-CITALOPRAM 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole >10000 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89974 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 3-[(2(S)-Azetidinyl)methoxy]-5-(phenoxymethyl)isoxazole 33 Yu LF et al 2012 Jan 15, 2025 Jan 28, 2025
89975 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-Bromo-2,5-dimethoxyphenethylamine 240 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89976 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-chloro-2,5-dimethoxy)ethanamine 190 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89977 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5-dimethoxy-4-methyl) ethanamine 440 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89978 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 360 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89979 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxyphenethylamine 70 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89980 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 4-iodo-2,5-dimethoxyphenethylamine 180 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89981 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5- dimethoxy-4-nitro)ethanamine 2200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89982 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 110 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89983 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 370 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89984 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2,5-dimethoxy-4-isopropylthiophenethylamine 470 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89985 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 520 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89986 5-HT1A CLONED HUMAN 3H-8-OH-DPAT MESCALINE 4600 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89987 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3600 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89988 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 5000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89989 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89990 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3500 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89991 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89992 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1800 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89993 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89994 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1800 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89995 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89996 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2500 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89997 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1800 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89998 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
89999 5-HT1A CLONED HUMAN 3H-8-OH-DPAT LSD 3 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90000 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-Bromo-2,5-dimethoxyphenethylamine 8.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90001 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-chloro-2,5-dimethoxy)ethanamine 13 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90002 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxy-4-methyl) ethanamine 32.4 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90003 5-HT2A CLONED HUMAN 3H-KETANSERIN 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 10.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90004 5-HT2A CLONED HUMAN 3H-KETANSERIN 2,5-dimethoxyphenethylamin 1600 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90005 5-HT2A CLONED HUMAN 3H-KETANSERIN 4-iodo-2,5-dimethoxyphenethylamine 3.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90006 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5- dimethoxy-4-nitro)ethanamine 23.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90007 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxy-4-propylphenyl)ethanamine; 8.1 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90008 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 9 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90009 5-HT2A CLONED HUMAN 3H-KETANSERIN 2,5-dimethoxy-4-isopropylthiophenethylamine 27.9 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90010 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 6.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90011 5-HT2A CLONED HUMAN 3H-KETANSERIN MESCALINE 6300 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90012 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 0.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90013 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 0.7 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90014 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90015 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 0.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90016 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 16.4 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90017 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 0.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90018 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 0.8 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90019 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1.1 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90020 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 0.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90021 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90022 5-HT2A CLONED HUMAN 3H-KETANSERIN 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1.1 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90023 5-HT2A CLONED HUMAN 3H-KETANSERIN Mescaline-NBOMe 140 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90024 5-HT2A CLONED HUMAN 3H-KETANSERIN LSD 4.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90025 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-Bromo-2,5-dimethoxyphenethylamine 47 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90026 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-chloro-2,5-dimethoxy)ethanamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90027 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-methyl) ethanamine 150 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90028 5-HT2C CLONED HUMAN 3H-MESULERGINE 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90029 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,5-dimethoxyphenethylamine 4100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90030 5-HT2C CLONED HUMAN 3H-MESULERGINE 4-iodo-2,5-dimethoxyphenethylamine 40 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90031 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5- dimethoxy-4-nitro)ethanamine 370 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90032 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 40 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90033 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 69 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90034 5-HT2C CLONED HUMAN 3H-MESULERGINE 2,5-dimethoxy-4-isopropylthiophenethylamine 130 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90035 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 39 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90036 5-HT2C CLONED HUMAN 3H-MESULERGINE MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90037 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90038 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 5.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90039 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 13 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90040 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7.2 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90041 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 130 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90042 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4.6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90043 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 21 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90044 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90045 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6.5 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90046 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 16 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90047 5-HT2C CLONED HUMAN 3H-MESULERGINE 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 6.4 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90048 5-HT2C CLONED HUMAN 3H-MESULERGINE Mescaline-NBOMe 640 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90049 5-HT2C CLONED HUMAN 3H-MESULERGINE LSD 15 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90050 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2C-B, 4-bromo-2,5-dimethoxyphenethylamine 8200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90051 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90052 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90053 Alpha1A CLONED HUMAN 3H-PRAZOSIN 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 7400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90054 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2,5-dimethoxyphenethylamine 7900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90055 Alpha1A CLONED HUMAN 3H-PRAZOSIN 4-iodo-2,5-dimethoxyphenethylamine 5100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90056 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90057 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 3500 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90058 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90059 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90060 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90061 Alpha1A CLONED HUMAN 3H-PRAZOSIN MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90062 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 430 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90063 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 810 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90064 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90065 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 530 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90066 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 550 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90067 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 370 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90068 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 850 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90069 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 310 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90070 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 550 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90071 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 580 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90072 Alpha1A CLONED HUMAN 3H-PRAZOSIN 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 340 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90073 Alpha1A CLONED HUMAN 3H-PRAZOSIN Mescaline-NBOMe 3000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90074 Alpha1A CLONED HUMAN 3H-PRAZOSIN LSD 670 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90075 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-Bromo-2,5-dimethoxyphenethylamine 320 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90076 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-chloro-2,5-dimethoxy)ethanamine 530 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90077 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5-dimethoxy-4-methyl) ethanamine 290 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90078 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 110 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90079 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2,5-dimethoxyphenethylamine 1000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90080 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 4-iodo-2,5-dimethoxyphenethylamine 70 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90081 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5- dimethoxy-4-nitro)ethanamine 1300 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90082 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90083 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 230 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90084 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2,5-dimethoxy-4-isopropylthiophenethylamine 180 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90085 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE MESCALINE 1400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90086 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamin 430 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90087 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 560 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90088 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 370 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90089 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 260 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90090 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 530 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90091 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 320 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90092 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 590 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90093 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 410 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90094 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 450 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90095 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 260 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90096 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 360 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90097 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Mescaline-NBOMe 810 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90098 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE LSD 12 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90099 D1 CLONED HUMAN 3H-SCH23390 4-Bromo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90100 D1 CLONED HUMAN 3H-SCH23390 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90101 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90102 D1 CLONED HUMAN 3H-SCH23390 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90103 D1 CLONED HUMAN 3H-SCH23390 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90104 D1 CLONED HUMAN 3H-SCH23390 4-iodo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90105 D1 CLONED HUMAN 3H-SCH23390 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90106 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 8400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90107 D1 CLONED HUMAN 3H-SCH23390 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90108 D1 CLONED HUMAN 3H-SCH23390 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90109 D1 CLONED HUMAN 3H-SCH23390 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90110 D1 CLONED HUMAN 3H-SCH23390 MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90111 D1 CLONED HUMAN 3H-SCH23390 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 9300 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90112 D1 CLONED HUMAN 3H-SCH23390 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90113 D1 CLONED HUMAN 3H-SCH23390 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 8700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90114 D1 CLONED HUMAN 3H-SCH23390 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90115 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90116 D1 CLONED HUMAN 3H-SCH23390 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90117 D1 CLONED HUMAN 3H-SCH23390 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90118 D1 CLONED HUMAN 3H-SCH23390 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90119 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90120 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90121 D1 CLONED HUMAN 3H-SCH23390 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 4100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90122 D1 CLONED HUMAN 3H-SCH23390 Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90123 D1 CLONED HUMAN 3H-SCH23390 LSD 310 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90124 D2 CLONED HUMAN 3H-SPIPERONE 4-Bromo-2,5-dimethoxyphenethylamine 2200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90125 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-chloro-2,5-dimethoxy)ethanamine 2100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90126 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-methyl) ethanamine 7100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90127 D2 CLONED HUMAN 3H-SPIPERONE 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 3200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90128 D2 CLONED HUMAN 3H-SPIPERONE 2,5-dimethoxyphenethylamine 9000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90129 D2 CLONED HUMAN 3H-SPIPERONE 4-iodo-2,5-dimethoxyphenethylamine 2700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90130 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5- dimethoxy-4-nitro)ethanamine 6100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90131 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 2300 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90132 D2 CLONED HUMAN 3H-SPIPERONE 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 5100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90133 D2 CLONED HUMAN 3H-SPIPERONE 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90134 D2 CLONED HUMAN 3H-SPIPERONE 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 5000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90135 D2 CLONED HUMAN 3H-SPIPERONE MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90136 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 840 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90137 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1600 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90138 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2600 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90139 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1500 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90140 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90141 D2 CLONED HUMAN 3H-SPIPERONE , 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90142 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90143 D2 CLONED HUMAN 3H-SPIPERONE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 870 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90144 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1600 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90145 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90146 D2 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90147 D2 CLONED HUMAN 3H-SPIPERONE Mescaline-NBOMe 9600 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90148 D2 CLONED HUMAN 3H-SPIPERONE LSD 25 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90149 D3 CLONED HUMAN 3H-SPIPERONE 4-Bromo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90150 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90151 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90152 D3 CLONED HUMAN 3H-SPIPERONE 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90153 D3 CLONED HUMAN 3H-SPIPERONE 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90154 D3 CLONED HUMAN 3H-SPIPERONE 4-iodo-2,5-dimethoxyphenethylamine 5000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90155 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90156 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 5200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90157 D3 CLONED HUMAN 3H-SPIPERONE 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90158 D3 CLONED HUMAN 3H-SPIPERONE 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90159 D3 CLONED HUMAN 3H-SPIPERONE 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 7500 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90160 D3 CLONED HUMAN 3H-SPIPERONE MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90161 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90162 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 3500 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90163 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90164 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90165 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90166 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90167 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4500 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90168 D3 CLONED HUMAN 3H-SPIPERONE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2300 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90169 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90170 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90171 D3 CLONED HUMAN 3H-SPIPERONE 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90172 D3 CLONED HUMAN 3H-SPIPERONE Mescaline-NBOMe 1700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90173 D3 CLONED HUMAN 3H-SPIPERONE LSD 96 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90174 CLONED RAT 3H-RO5166017 4-Bromo-2,5-dimethoxyphenethylamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90175 CLONED RAT 3H-RO5166017 2-(4-chloro-2,5-dimethoxy)ethanamine 110 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90176 CLONED RAT 3H-RO5166017 2-(2,5-dimethoxy-4-methyl) ethanamine 150 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90177 CLONED RAT 3H-RO5166017 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 70 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90178 CLONED RAT 3H-RO5166017 2,5-dimethoxyphenethylamine 900 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90179 CLONED RAT 3H-RO5166017 4-iodo-2,5-dimethoxyphenethylamine 120 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90180 CLONED RAT 3H-RO5166017 2-(2,5- dimethoxy-4-nitro)ethanamine 340 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90181 CLONED RAT 3H-RO5166017 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 20 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90182 CLONED RAT 3H-RO5166017 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 40 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90183 CLONED RAT 3H-RO5166017 2,5-dimethoxy-4-isopropylthiophenethylamine 50 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90184 CLONED RAT 3H-RO5166017 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine; 30 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90185 CLONED RAT 3H-RO5166017 MESCALINE 3300 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90186 CLONED RAT 3H-RO5166017 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 280 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90187 CLONED RAT 3H-RO5166017 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 520 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90188 CLONED RAT 3H-RO5166017 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 810 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90189 CLONED RAT 3H-RO5166017 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 260 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90190 CLONED RAT 3H-RO5166017 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1400 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90191 CLONED RAT 3H-RO5166017 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 440 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90192 CLONED RAT 3H-RO5166017 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90193 CLONED RAT 3H-RO5166017 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 60 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90194 CLONED RAT 3H-RO5166017 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 350 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90195 CLONED RAT 3H-RO5166017 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 120 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90196 CLONED RAT 3H-RO5166017 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90197 CLONED RAT 3H-RO5166017 Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90198 CLONED RAT 3H-RO5166017 LSD 450 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90199 CLONED MOUSE 3H-RO5166017 4-Bromo-2,5-dimethoxyphenethylamine 3000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90200 CLONED MOUSE 3H-RO5166017 2-(4-chloro-2,5-dimethoxy)ethanamine 4100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90201 CLONED MOUSE 3H-RO5166017 2-(2,5-dimethoxy-4-methyl) ethanamine-(4-chloro-2,5-dimethoxy)ethanamine 3500 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90202 CLONED MOUSE 3H-RO5166017 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane 1200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90203 CLONED MOUSE 3H-RO5166017 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90204 CLONED MOUSE 3H-RO5166017 4-iodo-2,5-dimethoxyphenethylamine 3300 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90205 CLONED MOUSE 3H-RO5166017 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90206 CLONED MOUSE 3H-RO5166017 2-(2,5-dimethoxy-4-propylphenyl)ethanamine 280 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90207 CLONED MOUSE 3H-RO5166017 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine 2200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90208 CLONED MOUSE 3H-RO5166017 2,5-dimethoxy-4-isopropylthiophenethylamine 4500 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90209 CLONED MOUSE 3H-RO5166017 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine 560 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90210 CLONED MOUSE 3H-RO5166017 MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90211 CLONED MOUSE 3H-RO5166017 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4500 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90212 CLONED MOUSE 3H-RO5166017 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90213 CLONED MOUSE 3H-RO5166017 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90214 CLONED MOUSE 3H-RO5166017 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90215 CLONED MOUSE 3H-RO5166017 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90216 CLONED MOUSE 3H-RO5166017 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90217 CLONED MOUSE 3H-RO5166017 , 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90218 CLONED MOUSE 3H-RO5166017 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 240 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90219 CLONED MOUSE 3H-RO5166017 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90220 CLONED MOUSE 3H-RO5166017 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1600 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90221 CLONED MOUSE 3H-RO5166017 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90222 CLONED MOUSE 3H-RO5166017 Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90223 CLONED MOUSE 3H-RO5166017 LSD >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90224 NET CLONED HUMAN 3H-Nisoxetine 4-Bromo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90225 NET CLONED HUMAN 3H-Nisoxetine 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90226 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90227 NET CLONED HUMAN 3H-Nisoxetine 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90228 NET CLONED HUMAN 3H-Nisoxetine 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90229 NET CLONED HUMAN 3H-Nisoxetine 4-iodo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90230 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90231 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5-dimethoxy-4-propylphenyl)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90232 NET CLONED HUMAN 3H-Nisoxetine 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90233 NET CLONED HUMAN 3H-Nisoxetine 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90234 NET CLONED HUMAN 3H-Nisoxetine 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90235 NET CLONED HUMAN 3H-Nisoxetine MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90236 NET CLONED HUMAN 3H-Nisoxetine 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90237 NET CLONED HUMAN 3H-Nisoxetine 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1600 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90238 NET CLONED HUMAN 3H-Nisoxetine 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamin 2200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90239 NET CLONED HUMAN 3H-Nisoxetine 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 3000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90240 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5500 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90241 NET CLONED HUMAN 3H-Nisoxetine 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1300 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90242 NET CLONED HUMAN 3H-Nisoxetine 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90243 NET CLONED HUMAN 3H-Nisoxetine 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2800 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90244 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5900 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90245 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4300 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90246 NET CLONED HUMAN 3H-Nisoxetine 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 3700 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90247 NET CLONED HUMAN 3H-Nisoxetine Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90248 NET CLONED HUMAN 3H-Nisoxetine LSD >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90249 DAT CLONED HUMAN 3H-WIN 35,428 4-Bromo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90250 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90251 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90252 DAT CLONED HUMAN 3H-WIN 35,428 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90253 DAT CLONED HUMAN 3H-WIN 35,428 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90254 DAT CLONED HUMAN 3H-WIN 35,428 4-iodo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90255 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90256 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5-dimethoxy-4-propylphenyl)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90257 DAT CLONED HUMAN 3H-WIN 35,428 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamin >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90258 DAT CLONED HUMAN 3H-WIN 35,428 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90259 DAT CLONED HUMAN 3H-WIN 35,428 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90260 DAT CLONED HUMAN 3H-WIN 35,428 MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90261 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 7200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90262 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90263 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90264 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 8100 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90265 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90266 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5400 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90267 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90268 DAT CLONED HUMAN 3H-WIN 35,428 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4700 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90269 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 8600 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90270 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 6200 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90271 DAT CLONED HUMAN 3H-WIN 35,428 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 4800 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90272 DAT CLONED HUMAN 3H-WIN 35,428 Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90273 DAT CLONED HUMAN 3H-WIN 35,428 LSD >10000 Rickli A et al 2015 Jan 15, 2025 Jan 15, 2025
90274 SERT CLONED HUMAN 3H-CITALOPRAM 4-Bromo-2,5-dimethoxyphenethylamine 9700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90275 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90276 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90277 SERT CLONED HUMAN 3H-CITALOPRAM 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90278 SERT CLONED HUMAN 3H-CITALOPRAM 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90279 SERT CLONED HUMAN 3H-CITALOPRAM 4-iodo-2,5-dimethoxyphenethylamine 4900 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90280 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90281 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5-dimethoxy-4-propylphenyl)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90282 SERT CLONED HUMAN 3H-CITALOPRAM 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90283 SERT CLONED HUMAN 3H-CITALOPRAM 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90284 SERT CLONED HUMAN 3H-CITALOPRAM 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90285 SERT CLONED HUMAN 3H-CITALOPRAM MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90286 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 840 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90287 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1500 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90288 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90289 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90290 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 2300 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90291 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90292 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90293 SERT CLONED HUMAN 3H-CITALOPRAM 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90294 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90295 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 8100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90296 SERT CLONED HUMAN 3H-CITALOPRAM 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 3200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90297 SERT CLONED HUMAN 3H-CITALOPRAM Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90298 SERT CLONED HUMAN 3H-CITALOPRAM LSD >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90299 H1 CLONED HUMAN 3H-PYRILAMINE 4-Bromo-2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90300 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-chloro-2,5-dimethoxy)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90301 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5-dimethoxy-4-methyl) ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90302 H1 CLONED HUMAN 3H-PYRILAMINE 1-(2,5-dimethoxy-4-ethylphenyl)-2-aminoethane >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90303 H1 CLONED HUMAN 3H-PYRILAMINE 2,5-dimethoxyphenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90304 H1 CLONED HUMAN 3H-PYRILAMINE 4-iodo-2,5-dimethoxyphenethylamine 6100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90305 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5- dimethoxy-4-nitro)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90306 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5-dimethoxy-4-propylphenyl)ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90307 H1 CLONED HUMAN 3H-PYRILAMINE 2-[2,5-dimethoxy-4-(ethylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90308 H1 CLONED HUMAN 3H-PYRILAMINE 2,5-dimethoxy-4-isopropylthiophenethylamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90309 H1 CLONED HUMAN 3H-PYRILAMINE 2-[2,5-dimethoxy-4-(propylthio)phenyl]ethanamine >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90310 H1 CLONED HUMAN 3H-PYRILAMINE MESCALINE >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90311 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-bromo-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 80 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90312 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-chloro-2,5-dimethoxyphenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90313 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-methyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 630 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90314 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-ethyl-2,5- dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90315 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 4100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90316 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-iodo2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 90 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90317 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-nitro-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 210 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90318 H1 CLONED HUMAN 3H-PYRILAMINE 2-(4-propyl-2,5-dimethoxyphenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 1700 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90319 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5-dimethoxy-4-ethylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 490 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90320 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5-dimethoxy-4-isopropylthiophenyl)-N-[(2-methoxyphenyl)methyl] ethanamine 5400 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90321 H1 CLONED HUMAN 3H-PYRILAMINE 2-(2,5-dimethoxy-4-n-propylthiophenyl)-N-[(2- methoxyphenyl)methyl] ethanamine 1200 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90322 H1 CLONED HUMAN 3H-PYRILAMINE Mescaline-NBOMe >10000 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90323 H1 CLONED HUMAN 3H-PYRILAMINE LSD 1100 Rickli A et al 2015 Jan 15, 2025 Jan 28, 2025
90324 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide 113 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90325 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide 146 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90326 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide 509 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90327 A1 brain membranes RAT 3H-CCPA N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 120 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90328 A1 brain membranes RAT 3H-CCPA N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 136 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90329 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90330 A1 brain membranes RAT 3H-CCPA N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide 1370 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90331 A1 brain membranes RAT 3H-CCPA N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 145 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90332 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 563 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90333 A1 brain membranes RAT 3H-CCPA N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90334 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90335 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90336 A1 brain membranes RAT 3H-CCPA N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90337 A1 brain membranes RAT 3H-CCPA N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 605 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90338 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide 50.7 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90339 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide 24.8 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90340 A1 brain membranes RAT 3H-CCPA N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 320 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90341 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide 181 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90342 A1 brain membranes RAT 3H-CCPA N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 684 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90343 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1590 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90344 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1010 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90345 A1 brain membranes RAT 3H-CCPA N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 118 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90346 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 382 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90347 A1 brain membranes RAT 3H-CCPA N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 194 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90348 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide 36.6 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90349 A1 brain membranes RAT 3H-CCPA 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90350 A1 brain membranes RAT 3H-CCPA N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 593 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90351 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide 551 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90352 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide 320 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90353 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide 1120 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90354 A2A Striatal Membranes RAT 3H-MSX-2 N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 271 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90355 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 303 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90356 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90357 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide 807 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90358 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 335 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90359 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 1360 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90360 A2A Striatal Membranes RAT 3H-MSX-2 N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 3230 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90361 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1360 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90362 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide 1870 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90363 A2A Striatal Membranes RAT 3H-MSX-2 N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90364 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 637 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90365 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide 242 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90366 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide 318 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90367 A2A Striatal Membranes RAT 3H-MSX-2 N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1290 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90368 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide 671 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90369 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 6520 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90370 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1630 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90371 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide >10000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90372 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 1250 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90373 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 1070 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90374 A2A Striatal Membranes RAT 3H-MSX-2 N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 569 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90375 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide 455 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90376 A2A Striatal Membranes RAT 3H-MSX-2 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide 2270 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90377 A2A Striatal Membranes RAT 3H-MSX-2 N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 7310 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90378 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide 193 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90379 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide 452 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90380 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide 911 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90381 A2B CLONED HUMAN 3H-PSB-603 N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 179 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90382 A2B CLONED HUMAN 3H-PSB-603 N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 340 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90383 A2B CLONED HUMAN 3H-PSB-603 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 306 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90384 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90385 A2B CLONED HUMAN 3H-PSB-603 N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90386 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90387 A2B CLONED HUMAN 3H-PSB-603 N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90388 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90389 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90390 A2B CLONED HUMAN 3H-PSB-603 N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90391 A2B CLONED HUMAN 3H-PSB-603 N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 862 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90392 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide 113 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90393 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide 126 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90394 A2B CLONED HUMAN 3H-PSB-603 N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 578 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90395 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide 298 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90396 A2B CLONED HUMAN 3H-PSB-603 N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90397 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90398 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90399 A2B CLONED HUMAN 3H-PSB-603 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 215 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90400 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90401 A2B CLONED HUMAN 3H-PSB-603 N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 275 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90402 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide 66.3 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90403 A2B CLONED HUMAN 3H-PSB-603 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90404 A2B CLONED HUMAN 3H-PSB-603 N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90405 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)acet-amide 509 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90406 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-Dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-ylo)ethyl)phenoxy)-N-(3-(pyrrolidin-1-yl)- propyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90407 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- ylo)ethyl)phenoxy)-N-(2-morpholinoethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90408 A3 CLONED HUMAN 3H-PSB-11 N-(2-(diethylamino)ethyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 508 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90409 A3 CLONED HUMAN 3H-PSB-11 N-(3-(diethylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90410 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90411 A3 CLONED HUMAN 3H-PSB-11 N-(3-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide 572 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90412 A3 CLONED HUMAN 3H-PSB-11 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 458 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90413 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90414 A3 CLONED HUMAN 3H-PSB-11 N-benzyl-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90415 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90416 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90417 A3 CLONED HUMAN 3H-PSB-11 N-(4-chlorobenzyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin9(6H)-yl)ethyl)phenoxy)acetamide 1090 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90418 A3 CLONED HUMAN 3H-PSB-11 N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(2,4-dioxo-1,3-dipropyl-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90419 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(diethylamino)ethyl)acetamide 155 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90420 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(3-(diethylamino)propyl)- acetamide 248 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90421 A3 CLONED HUMAN 3H-PSB-11 N-benzyl-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 602 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90422 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-morpholinoethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90423 A3 CLONED HUMAN 3H-PSB-11 N-(3-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90424 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(3-methoxybenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90425 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-fluorobenzyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90426 A3 CLONED HUMAN 3H-PSB-11 N-(3-(cyclohexylamino)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 353 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90427 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(2-(pyridin-2-yl)ethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90428 A3 CLONED HUMAN 3H-PSB-11 N-(3-(1H-imidazol-1-yl)propyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1- f]purin-9(6H)-yl)ethyl)phenoxy)acetamide 868 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90429 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-Dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimidoij2,1-f ]purin-9IJ6H)-yl)ethyl)phenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)- acetamide 204 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90430 A3 CLONED HUMAN 3H-PSB-11 2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)-yl)ethyl)phenoxy)- N-(4-sulfamoylphenethyl)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90431 A3 CLONED HUMAN 3H-PSB-11 N-(4-chlorobenzyl)-2-(4-(2-(1,3-dibutyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyrimido[2,1-f]purin-9(6H)- yl)ethyl)phenoxy)acetamide 1000 Zaluski M et al 2018 Jan 15, 2025 Jan 15, 2025
90432 D2 CLONED HUMAN 125I-IABN 1-((1H-Indol-3-yl)methyl)-4-(1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate)piperidin-4-ol oxalate 3.8 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90433 D2 CLONED HUMAN 125I-IABN 4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 0.9 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90434 D2 CLONED HUMAN 125I-IABN 4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 0.9 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90435 D2 CLONED HUMAN 125I-IABN 1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate 1396 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90436 D2 CLONED HUMAN 125I-IABN 4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 27.7 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90437 D2 CLONED HUMAN 125I-IABN 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 13.8 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90438 D2 CLONED HUMAN 125I-IABN 1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 23.3 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90439 D2 CLONED HUMAN 125I-IABN 1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 12.5 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90440 D2 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 212 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90441 D2 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 61 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90442 D2 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate 254 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90443 D2 CLONED HUMAN 125I-IABN 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 17.3 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90444 D2 CLONED HUMAN 125I-IABN 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 14.3 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90445 D2 CLONED HUMAN 125I-IABN 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 46.8 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90446 D2 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 6.6 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90447 D2 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 2.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90448 D2 CLONED HUMAN 125I-IABN 1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 13.6 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90449 D2 CLONED HUMAN 125I-IABN 1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 37.8 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90450 D2 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 7.1 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90451 D2 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 8 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90452 D2 CLONED HUMAN 125I-IABN 8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 71.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90453 D2 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 2 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90454 D2 CLONED HUMAN 125I-IABN HALOPERIDOL 1.1 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90455 D3 CLONED HUMAN 125I-IABN HALOPERIDOL 12.7 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90456 D3 CLONED HUMAN 125I-IABN 1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 94.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90457 D4 CLONED HUMAN 125I-IABN 1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 53.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90458 D4 CLONED HUMAN 125I-IABN 4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 60.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90459 D3 CLONED HUMAN 125I-IABN 4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 122 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90460 D3 CLONED HUMAN 125I-IABN 4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 100 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90461 D4 CLONED HUMAN 125I-IABN 4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 129 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90462 D4 CLONED HUMAN 125I-IABN 1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90463 D3 CLONED HUMAN 125I-IABN 1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate 2927 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90464 D3 CLONED HUMAN 125I-IABN 4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 849 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90465 D4 CLONED HUMAN 125I-IABN 4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 668 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90466 D4 CLONED HUMAN 125I-IABN 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 344 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90467 D3 CLONED HUMAN 125I-IABN 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 188 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90468 D3 CLONED HUMAN 125I-IABN 1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 132 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90469 D4 CLONED HUMAN 125I-IABN 1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 1390 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90470 D4 CLONED HUMAN 125I-IABN 1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 2230 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90471 D3 CLONED HUMAN 125I-IABN 1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 68.2 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90472 D3 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 2983 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90473 D4 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 620 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90474 D4 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 634 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90475 D3 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1585 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90476 D3 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate 4938 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90477 D4 CLONED HUMAN 125I-IABN 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate 937 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90478 D4 CLONED HUMAN 125I-IABN 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 254 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90479 D3 CLONED HUMAN 125I-IABN 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 31.8 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90480 D3 CLONED HUMAN 125I-IABN 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 49 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90481 D4 CLONED HUMAN 125I-IABN 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 245 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90482 D4 CLONED HUMAN 125I-IABN 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 377 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90483 D3 CLONED HUMAN 125I-IABN 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 142 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90484 D3 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 10.9 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90485 D4 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 94.5 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90486 D4 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 40.4 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90487 D3 CLONED HUMAN 125I-IABN 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 11.2 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90488 D3 CLONED HUMAN 125I-IABN 1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 3 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90489 D4 CLONED HUMAN 125I-IABN 1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 163 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90490 D4 CLONED HUMAN 125I-IABN 1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 72.6 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90491 D3 CLONED HUMAN 125I-IABN 1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 46.7 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90492 D3 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 2.1 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90493 D4 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 492 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90494 D4 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 945 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90495 D3 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 9.3 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90496 D3 CLONED HUMAN 125I-IABN 8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 60.1 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90497 D4 CLONED HUMAN 125I-IABN 8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 352 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90498 D4 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 978 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90499 D3 CLONED HUMAN 125I-IABN 8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 0.9 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90500 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 2 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90501 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 881 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90502 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 197 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90503 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate 1527 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90504 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 3224 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90505 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 227 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90506 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 4129 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90507 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate 1768 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90508 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 15.1 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90509 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1.2 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90510 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate 8.07 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90511 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 2.45 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90512 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 1.41 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90513 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 2.13 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90514 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 0.59 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90515 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 0.51 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90516 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 1779 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90517 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate 1879 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90518 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 708 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90519 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 28 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90520 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 331 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90521 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) 8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate 802 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90522 Sigma 1 brain membranes GUINEA PIG 3H-Pentazocine(+) HALOPERIDOL 1.45 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90523 Sigma 2 liver membranes RAT 3H-DTG HALOPERIDOL 24.2 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90524 Sigma 2 liver membranes RAT 3H-DTG 1-((1H-Indol-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 2200 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90525 Sigma 2 liver membranes RAT 3H-DTG 4-(4-Iodophenyl)-1-((4-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 970 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90526 Sigma 2 liver membranes RAT 3H-DTG 4-(4-Iodophenyl)-1-((5-methoxy-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 3262 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90527 Sigma 2 liver membranes RAT 3H-DTG 1-((5-Methoxy-1H-indol-3-yl)methyl)-4-phenylpiperidin-4-ol oxalate 2761 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90528 Sigma 2 liver membranes RAT 3H-DTG 4-(4-Bromophenyl)-1-((4-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate 9510 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90529 Sigma 2 liver membranes RAT 3H-DTG 4-(4-Bromophenyl)-1-((5-(2-fluoroethoxy)-1H-indol-3-yl)methyl)piperidin-4-ol oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90530 Sigma 2 liver membranes RAT 3H-DTG 1-(1-((4-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90531 Sigma 2 liver membranes RAT 3H-DTG 1-(1-((5-Methoxy-1H-indol-3-yl)methyl)piperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90532 Sigma 2 liver membranes RAT 3H-DTG 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1.9 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90533 Sigma 2 liver membranes RAT 3H-DTG 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 5.53 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90534 Sigma 2 liver membranes RAT 3H-DTG 1-((1H-pyrrolo[2,3-b]pyridine-3-yl)methyl)-4-(4-(methylthio)phenyl)piperidin-4-ol oxalate 7.75 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90535 Sigma 2 liver membranes RAT 3H-DTG 1-(Benzofuran-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1398 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90536 Sigma 2 liver membranes RAT 3H-DTG 1-(Benzofuran-2-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 2368 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90537 Sigma 2 liver membranes RAT 3H-DTG 1-(Benzo[b]thiophen-2-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 1964 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90538 Sigma 2 liver membranes RAT 3H-DTG 1-(Benzofuran-3-ylmethyl)-4-(4-bromophenyl)piperidin-4-ol oxalate 377 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90539 Sigma 2 liver membranes RAT 3H-DTG 1-(Benzofuran-3-ylmethyl)-4-(4-iodophenyl)piperidin-4-ol oxalate 393 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90540 Sigma 2 liver membranes RAT 3H-DTG 1-(1-(Benzofuran-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90541 Sigma 2 liver membranes RAT 3H-DTG 1-(1-(Benzo[b]thiophen-3-ylmethyl)piperidin-4-yl)-1H-benzo[d]imidazol-2-(3H)-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90542 Sigma 2 liver membranes RAT 3H-DTG 8-(Benzofuran-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90543 Sigma 2 liver membranes RAT 3H-DTG 8-(Benzofuran-3-ylmethyl)-3-(2-fluoroethyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90544 Sigma 2 liver membranes RAT 3H-DTG 8-(Benzo[b]thiophen-3-ylmethyl)-3-methyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90545 Sigma 2 liver membranes RAT 3H-DTG 8-(Benzofuran-3-ylmethyl)-3-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-1- phenyl-1,3,8-triazaspiro[4.5]decan-4-one oxalate >10000 Vangveravong S et al 2010 Jan 15, 2025 Jan 28, 2025
90546 A1 CORTICAL MEMBRANES RAT 3H-CCPA Preladenant (SCH420814) 68.7 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90547 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 422 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90548 A1 CORTICAL MEMBRANES RAT 3H-CCPA 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 367 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90549 A1 CORTICAL MEMBRANES RAT 3H-CCPA 3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1500 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90550 A1 CORTICAL MEMBRANES RAT 3H-CCPA 3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90551 A1 CORTICAL MEMBRANES RAT 3H-CCPA 3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90552 A1 CORTICAL MEMBRANES RAT 3H-CCPA 2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90553 A1 CORTICAL MEMBRANES RAT 3H-CCPA (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 205 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90554 A1 CORTICAL MEMBRANES RAT 3H-CCPA (E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90555 A1 CORTICAL MEMBRANES RAT 3H-CCPA 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90556 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 229 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90557 A1 CORTICAL MEMBRANES RAT 3H-CCPA 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 22.5 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90558 A1 CORTICAL MEMBRANES RAT 3H-CCPA 4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 898 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90559 A1 CORTICAL MEMBRANES RAT 3H-CCPA 4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 1500 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90560 A1 CORTICAL MEMBRANES RAT 3H-CCPA (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 53 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90561 A1 CORTICAL MEMBRANES RAT 3H-CCPA (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 11.2 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90562 A1 CORTICAL MEMBRANES RAT 3H-CCPA (E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide 11.4 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90563 A1 CORTICAL MEMBRANES RAT 3H-CCPA (E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide 1500 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90564 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 98.3 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90565 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90566 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90567 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90568 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 64.4 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90569 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90570 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 35.2 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90571 A1 CORTICAL MEMBRANES RAT 3H-CCPA N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90572 A2A Striatal Membranes RAT 3H-MSX-2 Preladenant (SCH420814) 0.66 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90573 A2A Striatal Membranes RAT 3H-MSX-2 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 103 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90574 A2A Striatal Membranes RAT 3H-MSX-2 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 294 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90575 A2A Striatal Membranes RAT 3H-MSX-2 3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90576 A2A Striatal Membranes RAT 3H-MSX-2 3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 2190 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90577 A2A Striatal Membranes RAT 3H-MSX-2 3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90578 A2A Striatal Membranes RAT 3H-MSX-2 2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90579 A2A Striatal Membranes RAT 3H-MSX-2 (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 253 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90580 A2A Striatal Membranes RAT 3H-MSX-2 (E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90581 A2A Striatal Membranes RAT 3H-MSX-2 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide 1720 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90582 A2A Striatal Membranes RAT 3H-MSX-2 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 423 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90583 A2A Striatal Membranes RAT 3H-MSX-2 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 558 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90584 A2A Striatal Membranes RAT 3H-MSX-2 4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90585 A2A Striatal Membranes RAT 3H-MSX-2 4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90586 A2A Striatal Membranes RAT 3H-MSX-2 (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 814 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90587 A2A Striatal Membranes RAT 3H-MSX-2 (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 317 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90588 A2A Striatal Membranes RAT 3H-MSX-2 (E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90589 A2A Striatal Membranes RAT 3H-MSX-2 (E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90590 A2A Striatal Membranes RAT 3H-MSX-2 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90591 A2A Striatal Membranes RAT 3H-MSX-2 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 84.7 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90592 A2A Striatal Membranes RAT 3H-MSX-2 4-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 488 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90593 A2A Striatal Membranes RAT 3H-MSX-2 N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90594 A2A Striatal Membranes RAT 3H-MSX-2 N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 6060 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90595 A2A Striatal Membranes RAT 3H-MSX-2 N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90596 A2A Striatal Membranes RAT 3H-MSX-2 N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90597 A2A Striatal Membranes RAT 3H-MSX-2 N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90598 A2A Striatal Membranes RAT 3H-MSX-2 N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90599 A2A Striatal Membranes RAT 3H-MSX-2 N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 693 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90600 A2A Striatal Membranes RAT 3H-MSX-2 N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90601 A1 CLONED HUMAN 3H-CCPA Preladenant (SCH420814) 295 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90602 A1 CLONED HUMAN 3H-CCPA N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 1050 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90603 A1 CLONED HUMAN 3H-CCPA 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1370 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90604 A1 CLONED HUMAN 3H-CCPA (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90605 A1 CLONED HUMAN 3H-CCPA N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 2500 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90606 A1 CLONED HUMAN 3H-CCPA 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 214 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90607 A1 CLONED HUMAN 3H-CCPA 4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide >10000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90608 A1 CLONED HUMAN 3H-CCPA (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 822 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90609 A1 CLONED HUMAN 3H-CCPA (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 500 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90610 A1 CLONED HUMAN 3H-CCPA (E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide 562 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90611 A1 CLONED HUMAN 3H-CCPA 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90612 A1 CLONED HUMAN 3H-CCPA 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90613 A1 CLONED HUMAN 3H-CCPA 4-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 4370 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90614 A1 CLONED HUMAN 3H-CCPA N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 785 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90615 A1 CLONED HUMAN 3H-CCPA N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 364 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90616 A2A CLONED HUMAN 3H-MSX-2 Preladenant (SCH420814) 0.884 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90617 A2A CLONED HUMAN 3H-MSX-2 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 80.9 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90618 A2A CLONED HUMAN 3H-MSX-2 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 64.9 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90619 A2A CLONED HUMAN 3H-MSX-2 (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 62.4 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90620 A2A CLONED HUMAN 3H-MSX-2 (E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90621 A2A CLONED HUMAN 3H-MSX-2 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90622 A2A CLONED HUMAN 3H-MSX-2 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 39.5 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90623 A2A CLONED HUMAN 3H-MSX-2 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 115 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90624 A2A CLONED HUMAN 3H-MSX-2 (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 118 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90625 A2A CLONED HUMAN 3H-MSX-2 (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 91.8 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90626 A2A CLONED HUMAN 3H-MSX-2 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90627 A2A CLONED HUMAN 3H-MSX-2 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 58.3 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90628 A2A CLONED HUMAN 3H-MSX-2 N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 82.5 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90629 A2B CLONED HUMAN 3H-PSB-603 Preladenant (SCH420814) 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90630 A2B CLONED HUMAN 3H-PSB-603 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 365 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90631 A2B CLONED HUMAN 3H-PSB-603 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 225 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90632 A2B CLONED HUMAN 3H-PSB-603 3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90633 A2B CLONED HUMAN 3H-PSB-603 3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 801 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90634 A2B CLONED HUMAN 3H-PSB-603 3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90635 A2B CLONED HUMAN 3H-PSB-603 2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90636 A2B CLONED HUMAN 3H-PSB-603 (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 679 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90637 A2B CLONED HUMAN 3H-PSB-603 (E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90638 A2B CLONED HUMAN 3H-PSB-603 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90639 A2B CLONED HUMAN 3H-PSB-603 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90640 A2B CLONED HUMAN 3H-PSB-603 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 302 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90641 A2B CLONED HUMAN 3H-PSB-603 4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90642 A2B CLONED HUMAN 3H-PSB-603 4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90643 A2B CLONED HUMAN 3H-PSB-603 (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 119 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90644 A2B CLONED HUMAN 3H-PSB-603 (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90645 A2B CLONED HUMAN 3H-PSB-603 (E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90646 A2B CLONED HUMAN 3H-PSB-603 (E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90647 A2B CLONED HUMAN 3H-PSB-603 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90648 A2B CLONED HUMAN 3H-PSB-603 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90649 A2B CLONED HUMAN 3H-PSB-603 4-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90650 A2B CLONED HUMAN 3H-PSB-603 N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90651 A2B CLONED HUMAN 3H-PSB-603 N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 408 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90652 A2B CLONED HUMAN 3H-PSB-603 N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90653 A2B CLONED HUMAN 3H-PSB-603 N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90654 A2B CLONED HUMAN 3H-PSB-603 N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90655 A2B CLONED HUMAN 3H-PSB-603 N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide 547 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90656 A2B CLONED HUMAN 3H-PSB-603 N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 361 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90657 A2B CLONED HUMAN 3H-PSB-603 N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90658 A3 CLONED HUMAN 3H-PSB-11 Preladenant (SCH420814) 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90659 A3 CLONED HUMAN 3H-PSB-11 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-3-phenylpropanamide 390 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90660 A3 CLONED HUMAN 3H-PSB-11 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 173 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90661 A3 CLONED HUMAN 3H-PSB-11 3-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90662 A3 CLONED HUMAN 3H-PSB-11 3-(2-Fluorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90663 A3 CLONED HUMAN 3H-PSB-11 3-(2-Bromophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90664 A3 CLONED HUMAN 3H-PSB-11 2-(3-Chlorophenoxy)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acetamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90665 A3 CLONED HUMAN 3H-PSB-11 (E)-3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90666 A3 CLONED HUMAN 3H-PSB-11 (E)-3-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- acrylamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90667 A3 CLONED HUMAN 3H-PSB-11 3-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- propiolamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90668 A3 CLONED HUMAN 3H-PSB-11 N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90669 A3 CLONED HUMAN 3H-PSB-11 4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 382 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90670 A3 CLONED HUMAN 3H-PSB-11 4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90671 A3 CLONED HUMAN 3H-PSB-11 4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- butanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90672 A3 CLONED HUMAN 3H-PSB-11 (E)-N-(4-Oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbut-3-enamide 158 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90673 A3 CLONED HUMAN 3H-PSB-11 (E)-4-(3-Methoxyphenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but3-enamide 115 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90674 A3 CLONED HUMAN 3H-PSB-11 (E)-4-(3-Chlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)but-3- enamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90675 A3 CLONED HUMAN 3H-PSB-11 (E)-4-(3,4-Dichlorophenyl)-N-(4-oxo-4H-3,1-benzothiazin-2-yl)- but-3-enamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90676 A3 CLONED HUMAN 3H-PSB-11 4-(4-(2-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90677 A3 CLONED HUMAN 3H-PSB-11 4-(4-(3-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90678 A3 CLONED HUMAN 3H-PSB-11 4-(4-(4-Chlorobenzyl)piperazine-1-carbonyl)-N-(4-oxo-4H-3,1- benzothiazin-2-yl)benzamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90679 A3 CLONED HUMAN 3H-PSB-11 N-Methyl-N-(4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90680 A3 CLONED HUMAN 3H-PSB-11 N-(6-Methyl-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 147 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90681 A3 CLONED HUMAN 3H-PSB-11 N-(6-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90682 A3 CLONED HUMAN 3H-PSB-11 N-(6-Bromo-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90683 A3 CLONED HUMAN 3H-PSB-11 N-(7-Chloro-4-oxo-4H-3,1-benzothiazin-2-yl)-4-phenylbutanamide 91.6 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90684 A3 CLONED HUMAN 3H-PSB-11 N-(4-Oxo-4H-thieno[3,2-d][1,3]thiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90685 A3 CLONED HUMAN 3H-PSB-11 N-(4-Oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90686 A3 CLONED HUMAN 3H-PSB-11 N-(5,6-Dimethyl-4-oxo-4H-thieno[2,3-d][1,3]thiazin-2-yl)-4-phenylbutanamide 1000 Stossel A et al 2013 Jan 15, 2025 Jan 15, 2025
90687 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 12 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90688 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 5.7 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90689 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 4.9 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90690 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 2.3 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90691 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 183 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90692 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 36 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90693 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine 15 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90694 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine 8.1 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90695 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 19 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90696 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 5.8 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90697 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine 3.1 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90698 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine 1.9 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90699 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 19 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90700 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine 20 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90701 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 8 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90702 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 8.2 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90703 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine 15 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90704 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 18 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90705 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 8 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90706 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 3.1 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90707 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine 262 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90708 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine 50 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90709 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) trans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 256 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90710 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 97 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90711 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) PENTAZOCINE (+) 5.4 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90712 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) DTG 71 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90713 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 53 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90714 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 67 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90715 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 81 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90716 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 33 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90717 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 161 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90718 Sigma 2 liver membranes RAT 3H-DTG cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 308 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90719 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine 361 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90720 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine 42 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90721 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 128 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90722 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-3-methoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 101 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90723 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2- benzopyran-1,1’-cyclohexan]-4’-amine 154 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90724 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine 12 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90725 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 133 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90726 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine 52 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90727 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 164 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90728 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 70 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90729 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]- 4’-amine 99 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90730 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 84 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90731 Sigma 2 liver membranes RAT 3H-DTG trans-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 175 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90732 Sigma 2 liver membranes RAT 3H-DTG cis-N-(Cyclohexylmethyl)-N-methyl-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 30 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90733 Sigma 2 liver membranes RAT 3H-DTG trans-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine 1000 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90734 Sigma 2 liver membranes RAT 3H-DTG cis-N-Benzyl-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]-4’-amine 751 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90735 Sigma 2 liver membranes RAT 3H-DTG trans-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 1000 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90736 Sigma 2 liver membranes RAT 3H-DTG cis-N-Benzyl-3,4-dihydrospiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 503 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90737 Sigma 2 liver membranes RAT 3H-DTG DTG 54 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90738 Sigma 2 CLONED HUMAN 3H-DTG trans-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 7 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90739 Sigma 2 CLONED HUMAN 3H-DTG cis-N-(Cyclohexylmethyl)spiro[[2]benzopyran-1,1’-cyclohexan]-4’-amine 6.7 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90740 Sigma 2 CLONED HUMAN 3H-DTG trans-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 16 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90741 Sigma 2 CLONED HUMAN 3H-DTG cis-N-(Cyclohexylmethyl)-N-methylspiro[[2]benzopyran-1,1’-cyclohexan]-4’- amine 4.6 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90742 Sigma 2 CLONED HUMAN 3H-DTG trans-N-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 16 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90743 Sigma 2 CLONED HUMAN 3H-DTG cis-(Cyclohexylmethyl)-3-ethoxy-3,4-dihydrospiro[[2]benzopyran-1,1’- cyclohexan]-4’-amine 46 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90744 Sigma 2 CLONED HUMAN 3H-DTG trans-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine 93 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90745 Sigma 2 CLONED HUMAN 3H-DTG cis-N-(Cyclohexylmethyl)-3-ethoxy-N-methyl-3,4-dihydrospiro[[2]benzopyran1,1’-cyclohexan]-4’-amine 14 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90746 Sigma 2 CLONED HUMAN 3H-DTG cis-N-(Cyclohexylmethyl)-3-methoxy-N-methyl-3,4-dihydrospiro[2-benzopyran1,1’-cyclohexan]-4’-amine 13 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90747 Sigma 2 CLONED HUMAN 3H-DTG trans-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’- cyclohexan]-4’-amine 39 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025
90748 Sigma 2 CLONED HUMAN 3H-DTG cis-N-(Cyclohexylmethyl)-3-methoxy-3H-spiro[[2]benzofuran-1,1’-cyclohexan]- 4’-amine 11 Kronenberg E et al 2019 Jan 15, 2025 Jan 28, 2025