The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

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Showing 93,001-94,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
957495-HT5ACLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957505-HT6CLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957515-HT7CLONEDHUMAN3H-LSDTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957525-HT5ACLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957535-HT6CLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957545-HT7CLONEDHUMAN3H-LSD6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957555-HT5ACLONEDHUMAN3H-LSDN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957565-HT6CLONEDHUMAN3H-LSDN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957575-HT7CLONEDHUMAN3H-LSDN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957585-HT5ACLONEDHUMAN3H-LSDtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957595-HT6CLONEDHUMAN3H-LSDtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957605-HT7CLONEDHUMAN3H-LSDtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957615-HT5ACLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957625-HT6CLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957635-HT7CLONEDHUMAN3H-LSD4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957645-HT5ACLONEDHUMAN3H-LSD2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957655-HT6CLONEDHUMAN3H-LSD2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
957665-HT7CLONEDHUMAN3H-LSD2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95767Alpha1ACLONEDHUMAN3H-PRAZOSIN6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95768Alpha1BCLONEDHUMAN3H-PRAZOSIN6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95769Alpha1DCLONEDHUMAN3H-PRAZOSIN6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95770Alpha1ACLONEDHUMAN3H-PRAZOSINTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95771Alpha1BCLONEDHUMAN3H-PRAZOSINTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95772Alpha1DCLONEDHUMAN3H-PRAZOSINTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95773Alpha1ACLONEDHUMAN3H-PRAZOSINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95774Alpha1BCLONEDHUMAN3H-PRAZOSINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95775Alpha1DCLONEDHUMAN3H-PRAZOSINTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95776Alpha1ACLONEDHUMAN3H-PRAZOSIN6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95777Alpha1BCLONEDHUMAN3H-PRAZOSIN6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95778Alpha1DCLONEDHUMAN3H-PRAZOSIN6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95779Alpha1ACLONEDHUMAN3H-PRAZOSINN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95780Alpha1BCLONEDHUMAN3H-PRAZOSINN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95781Alpha1DCLONEDHUMAN3H-PRAZOSINN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95782Alpha1ACLONEDHUMAN3H-PRAZOSINtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95783Alpha1BCLONEDHUMAN3H-PRAZOSINtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95784Alpha1DCLONEDHUMAN3H-PRAZOSINtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95785Alpha1ACLONEDHUMAN3H-PRAZOSIN4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95786Alpha1BCLONEDHUMAN3H-PRAZOSIN4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95787Alpha1DCLONEDHUMAN3H-PRAZOSIN4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95788Alpha1ACLONEDHUMAN3H-PRAZOSIN2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95789Alpha1BCLONEDHUMAN3H-PRAZOSIN2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95790Alpha1DCLONEDHUMAN3H-PRAZOSIN2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95791Alpha2ACLONEDHUMAN3H-RAUWOLSCINE6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene4800Jung et al 2021Jan 15, 2025Jan 28, 2025
95792Alpha2ACLONEDHUMAN3H-RAUWOLSCINETrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane4700Jung et al 2021Jan 15, 2025Jan 28, 2025
95793Alpha2ACLONEDHUMAN3H-RAUWOLSCINE6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95794Alpha2ACLONEDHUMAN3H-RAUWOLSCINEN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide2200Jung et al 2021Jan 15, 2025Jan 28, 2025
95795Alpha2ACLONEDHUMAN3H-RAUWOLSCINEtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate940Jung et al 2021Jan 15, 2025Jan 28, 2025
95796Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid1800Jung et al 2021Jan 15, 2025Jan 28, 2025
95797Alpha2ACLONEDHUMAN3H-RAUWOLSCINE2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione650Jung et al 2021Jan 15, 2025Jan 28, 2025
95798Alpha2BCLONEDHUMAN3H-RAUWOLSCINE6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95799Alpha2BCLONEDHUMAN3H-RAUWOLSCINETrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95800Alpha2BCLONEDHUMAN3H-RAUWOLSCINETriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95801Alpha2BCLONEDHUMAN3H-RAUWOLSCINE6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95802Alpha2BCLONEDHUMAN3H-RAUWOLSCINEN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide6700Jung et al 2021Jan 15, 2025Jan 28, 2025
95803Alpha2BCLONEDHUMAN3H-RAUWOLSCINEtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95804Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid1000Jung et al 2021Jan 15, 2025Jan 28, 2025
95805Alpha2BCLONEDHUMAN3H-RAUWOLSCINE2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione4700Jung et al 2021Jan 15, 2025Jan 28, 2025
95806Alpha2CCLONEDHUMAN3H-RAUWOLSCINE6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95807Alpha2CCLONEDHUMAN3H-RAUWOLSCINETrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95808Alpha2CCLONEDHUMAN3H-RAUWOLSCINETriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95809Alpha2CCLONEDHUMAN3H-RAUWOLSCINE6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95810Alpha2CCLONEDHUMAN3H-RAUWOLSCINEN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95811Alpha2CCLONEDHUMAN3H-RAUWOLSCINEtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95812Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid2600Jung et al 2021Jan 15, 2025Jan 28, 2025
95813Alpha2CCLONEDHUMAN3H-RAUWOLSCINE2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95814Beta 1CLONEDHUMAN125I-iodo-pindolol6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95815Beta3CLONEDHUMAN125I-iodo-pindolol6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95816Beta 1CLONEDHUMAN125I-iodo-pindololTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95817Beta3CLONEDHUMAN125I-iodo-pindololTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95818Beta 1CLONEDHUMAN125I-iodo-pindololTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95819Beta3CLONEDHUMAN125I-iodo-pindololTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95820Beta 1CLONEDHUMAN125I-iodo-pindolol6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95821Beta3CLONEDHUMAN125I-iodo-pindolol6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95822Beta 1CLONEDHUMAN125I-iodo-pindololN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95823Beta3CLONEDHUMAN125I-iodo-pindololN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95824Beta 1CLONEDHUMAN125I-iodo-pindololtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95825Beta3CLONEDHUMAN125I-iodo-pindololtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95826Beta 1CLONEDHUMAN125I-iodo-pindolol4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95827Beta3CLONEDHUMAN125I-iodo-pindolol4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95828Beta 1CLONEDHUMAN125I-iodo-pindolol2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95829Beta3CLONEDHUMAN125I-iodo-pindolol2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95830Beta 2CLONEDHUMAN3H-CGP-121776-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95831Beta 2CLONEDHUMAN3H-CGP-12177Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95832Beta 2CLONEDHUMAN3H-CGP-12177Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95833Beta 2CLONEDHUMAN3H-CGP-121776-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95834Beta 2CLONEDHUMAN3H-CGP-12177N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95835Beta 2CLONEDHUMAN3H-CGP-12177tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95836Beta 2CLONEDHUMAN3H-CGP-121774-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95837Beta 2CLONEDHUMAN3H-CGP-121772-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95838BZPCORTICAL MEMBRANESRATFNZ6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95839BZPCORTICAL MEMBRANESRATFNZTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95840BZPCORTICAL MEMBRANESRATFNZTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95841BZPCORTICAL MEMBRANESRATFNZ6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95842BZPCORTICAL MEMBRANESRATFNZN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95843BZPCORTICAL MEMBRANESRATFNZtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95844BZPCORTICAL MEMBRANESRATFNZ4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95845BZPCORTICAL MEMBRANESRATFNZ2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95846D1CLONEDHUMAN3H-SCH233906-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95847D5CLONEDHUMAN3H-SCH233906-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene1600Jung et al 2021Jan 15, 2025Jan 28, 2025
95848D5CLONEDHUMAN3H-SCH23390Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane4200Jung et al 2021Jan 15, 2025Jan 28, 2025
95849D1CLONEDHUMAN3H-SCH23390Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95850D1CLONEDHUMAN3H-SCH23390Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95851D5CLONEDHUMAN3H-SCH23390Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95852D5CLONEDHUMAN3H-SCH233906-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene2100Jung et al 2021Jan 15, 2025Jan 28, 2025
95853D1CLONEDHUMAN3H-SCH233906-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95854D1CLONEDHUMAN3H-SCH23390N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95855D5CLONEDHUMAN3H-SCH23390N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide1100Jung et al 2021Jan 15, 2025Jan 28, 2025
95856D5CLONEDHUMAN3H-SCH23390tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate1250Jung et al 2021Jan 15, 2025Jan 28, 2025
95857D1CLONEDHUMAN3H-SCH23390tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95858D1CLONEDHUMAN3H-SCH233904-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid1100Jung et al 2021Jan 15, 2025Jan 28, 2025
95859D5CLONEDHUMAN3H-SCH233904-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid2100Jung et al 2021Jan 15, 2025Jan 28, 2025
95860D5CLONEDHUMAN3H-SCH233902-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione1400Jung et al 2021Jan 15, 2025Jan 28, 2025
95861D1CLONEDHUMAN3H-SCH233902-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95862D2CLONEDHUMAN3H-Methylspiperone6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95863D3CLONEDHUMAN3H-Methylspiperone6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95864D4CLONEDHUMAN3H-Methylspiperone6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95865D2CLONEDHUMAN3H-MethylspiperoneTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95866D3CLONEDHUMAN3H-MethylspiperoneTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95867D4CLONEDHUMAN3H-MethylspiperoneTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95868D2CLONEDHUMAN3H-Methylspiperone6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95869D3CLONEDHUMAN3H-Methylspiperone6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95870D4CLONEDHUMAN3H-Methylspiperone6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95871D2CLONEDHUMAN3H-MethylspiperoneN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95872D3CLONEDHUMAN3H-MethylspiperoneN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95873D4CLONEDHUMAN3H-MethylspiperoneN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95874D2CLONEDHUMAN3H-Methylspiperonetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95875D3CLONEDHUMAN3H-Methylspiperonetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate1700Jung et al 2021Jan 15, 2025Jan 28, 2025
95876D4CLONEDHUMAN3H-Methylspiperonetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95877D2CLONEDHUMAN3H-Methylspiperone4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95878D3CLONEDHUMAN3H-Methylspiperone4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95879D4CLONEDHUMAN3H-Methylspiperone4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95880D2CLONEDHUMAN3H-Methylspiperone2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95881D3CLONEDHUMAN3H-Methylspiperone2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95882D4CLONEDHUMAN3H-Methylspiperone2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95883KORCEREBRAL CORTEXRAT3H-MUSCIMOL6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95884KORCEREBRAL CORTEXRAT3H-MUSCIMOLTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95885KORCEREBRAL CORTEXRAT3H-MUSCIMOLTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95886KORCEREBRAL CORTEXRAT3H-MUSCIMOL6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95887KORCEREBRAL CORTEXRAT3H-MUSCIMOLN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95888KORCEREBRAL CORTEXRAT3H-MUSCIMOLtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95889KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95890KORCEREBRAL CORTEXRAT3H-MUSCIMOL2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 27, 2025
95891H1CLONEDHUMAN3H-PYRILAMINE6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95892H1CLONEDHUMAN3H-PYRILAMINETrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95893H1CLONEDHUMAN3H-PYRILAMINETriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95894H1CLONEDHUMAN3H-PYRILAMINE6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95895H1CLONEDHUMAN3H-PYRILAMINEN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95896H1CLONEDHUMAN3H-PYRILAMINEtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95897H1CLONEDHUMAN3H-PYRILAMINE4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95898H1CLONEDHUMAN3H-PYRILAMINE2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
958995-HT1DCLONEDHUMAN125I-iodoaminopotentidine6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959005-HT1DCLONEDHUMAN125I-iodoaminopotentidineTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959015-HT1DCLONEDHUMAN125I-iodoaminopotentidineTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959025-HT1DCLONEDHUMAN125I-iodoaminopotentidine6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959035-HT1DCLONEDHUMAN125I-iodoaminopotentidineN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959045-HT1DCLONEDHUMAN125I-iodoaminopotentidinetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959055-HT1DCLONEDHUMAN125I-iodoaminopotentidine4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
959065-HT1DCLONEDHUMAN125I-iodoaminopotentidine2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95907H3CLONEDHUMAN3H-Alpha-methylhistamine6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95908H3CLONEDHUMAN3H-Alpha-methylhistamineTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95909H3CLONEDHUMAN3H-Alpha-methylhistamineTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95910H3CLONEDHUMAN3H-Alpha-methylhistamine6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95911H3CLONEDHUMAN3H-Alpha-methylhistaminetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95912H3CLONEDHUMAN3H-Alpha-methylhistamine4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95913H3CLONEDHUMAN3H-Alpha-methylhistamine2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95914H4CLONEDHUMAN3H-Histamine6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95915H4CLONEDHUMAN3H-HistamineTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95916H4CLONEDHUMAN3H-HistamineTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95917H4CLONEDHUMAN3H-Histamine6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95918H4CLONEDHUMAN3H-HistamineN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95919H4CLONEDHUMAN3H-Histaminetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95920H4CLONEDHUMAN3H-Histamine4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95921H4CLONEDHUMAN3H-Histamine2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95922M1CLONEDHUMAN3H-QNB6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95923M2CLONEDHUMAN3H-QNB6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95924M3CLONEDHUMAN3H-QNB6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95925M4CLONEDHUMAN3H-QNB6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95926M5CLONEDHUMAN3H-QNB6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95927M1CLONEDHUMAN3H-QNBTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95928M2CLONEDHUMAN3H-QNBTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95929M3CLONEDHUMAN3H-QNBTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95930M4CLONEDHUMAN3H-QNBTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95931M5CLONEDHUMAN3H-QNBTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95932M1CLONEDHUMAN3H-QNBTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95933M2CLONEDHUMAN3H-QNBTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95934M3CLONEDHUMAN3H-QNBTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95935M4CLONEDHUMAN3H-QNBTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95936M5CLONEDHUMAN3H-QNBTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95937M1CLONEDHUMAN3H-QNB6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95938M2CLONEDHUMAN3H-QNB6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95939M3CLONEDHUMAN3H-QNB6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95940M4CLONEDHUMAN3H-QNB6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95941M5CLONEDHUMAN3H-QNB6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95942M1CLONEDHUMAN3H-QNBN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95943M2CLONEDHUMAN3H-QNBN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95944M3CLONEDHUMAN3H-QNBN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95945M4CLONEDHUMAN3H-QNBN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95946M5CLONEDHUMAN3H-QNBN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95947M1CLONEDHUMAN3H-QNBtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95948M2CLONEDHUMAN3H-QNBtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95949M3CLONEDHUMAN3H-QNBtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95950M4CLONEDHUMAN3H-QNBtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95951M5CLONEDHUMAN3H-QNBtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95952M1CLONEDHUMAN3H-QNB4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95953M2CLONEDHUMAN3H-QNB4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95954M3CLONEDHUMAN3H-QNB4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95955M4CLONEDHUMAN3H-QNB4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95956M5CLONEDHUMAN3H-QNB4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95957M1CLONEDHUMAN3H-QNB2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95958M2CLONEDHUMAN3H-QNB2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95959M3CLONEDHUMAN3H-QNB2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95960M4CLONEDHUMAN3H-QNB2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95961M5CLONEDHUMAN3H-QNB2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
95962DORCLONEDHUMAN3H-DADLE6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95963DORCLONEDHUMAN3H-DADLETrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95964DORCLONEDHUMAN3H-DADLETriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95965DORCLONEDHUMAN3H-DADLEN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95966DORCLONEDHUMAN3H-DADLEtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95967DORCLONEDHUMAN3H-DADLE4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95968DORCLONEDHUMAN3H-DADLE2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95969KORCLONEDHUMAN3H-U695936-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95970KORCLONEDHUMAN3H-U69593Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95971KORCLONEDHUMAN3H-U69593Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95972KORCLONEDHUMAN3H-U695936-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95973KORCLONEDHUMAN3H-U69593N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95974KORCLONEDHUMAN3H-U69593tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95975KORCLONEDHUMAN3H-U695934-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95976KORCLONEDHUMAN3H-U695932-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95977MORCLONEDHUMAN3H-DAMGO6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95978MORCLONEDHUMAN3H-DAMGOTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95979MORCLONEDHUMAN3H-DAMGOTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95980MORCLONEDHUMAN3H-DAMGO6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95981MORCLONEDHUMAN3H-DAMGON-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95982MORCLONEDHUMAN3H-DAMGOtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95983MORCLONEDHUMAN3H-DAMGO4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid4200Jung et al 2021Jan 15, 2025Jan 28, 2025
95984MORCLONEDHUMAN3H-DAMGO2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95985Sigma 1CLONEDHUMAN3H-Pentazocine(+)6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene2100Jung et al 2021Jan 15, 2025Jan 28, 2025
95986Sigma 1CLONEDHUMAN3H-Pentazocine(+)Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane1400Jung et al 2021Jan 15, 2025Jan 28, 2025
95987Sigma 1CLONEDHUMAN3H-Pentazocine(+)Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95988Sigma 1CLONEDHUMAN3H-Pentazocine(+)6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95989Sigma 1CLONEDHUMAN3H-Pentazocine(+)N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide4400Jung et al 2021Jan 15, 2025Jan 28, 2025
95990Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95991Sigma 1CLONEDHUMAN3H-Pentazocine(+)2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95992Sigma 2CLONEDHUMAN3H-DTG6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95993Sigma 2CLONEDHUMAN3H-DTGTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95994Sigma 2CLONEDHUMAN3H-DTGTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95995Sigma 2CLONEDHUMAN3H-DTG6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95996Sigma 2CLONEDHUMAN3H-DTGN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95997Sigma 2CLONEDHUMAN3H-DTGtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95998Sigma 2CLONEDHUMAN3H-DTG4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
95999Sigma 2CLONEDHUMAN3H-DTG2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96000DATCLONEDHUMAN3H-WIN 35,4286-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96001DATCLONEDHUMAN3H-WIN 35,428Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96002DATCLONEDHUMAN3H-WIN 35,428Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96003DATCLONEDHUMAN3H-WIN 35,4286-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96004DATCLONEDHUMAN3H-WIN 35,428N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96005DATCLONEDHUMAN3H-WIN 35,428tert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96006DATCLONEDHUMAN3H-WIN 35,4284-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96007DATCLONEDHUMAN3H-WIN 35,4282-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96008NETCLONEDHUMAN3H-Nisoxetine6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96009NETCLONEDHUMAN3H-NisoxetineTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96010NETCLONEDHUMAN3H-NisoxetineTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96011NETCLONEDHUMAN3H-Nisoxetine6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96012NETCLONEDHUMAN3H-NisoxetineN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96013NETCLONEDHUMAN3H-Nisoxetinetert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96014NETCLONEDHUMAN3H-Nisoxetine4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96015NETCLONEDHUMAN3H-Nisoxetine2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96016SERTCLONEDHUMAN3H-CITALOPRAM6-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96017SERTCLONEDHUMAN3H-CITALOPRAMTrimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96018SERTCLONEDHUMAN3H-CITALOPRAMTriethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96019SERTCLONEDHUMAN3H-CITALOPRAM6-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96020SERTCLONEDHUMAN3H-CITALOPRAMN-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96021SERTCLONEDHUMAN3H-CITALOPRAMtert-Butyl (3-(3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)carbamate>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96022SERTCLONEDHUMAN3H-CITALOPRAM4-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96023SERTCLONEDHUMAN3H-CITALOPRAM2-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 28, 2025
96024PBRKidney membranesRAT3H-PK111956-Iodo-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96025PBRKidney membranesRAT3H-PK11195Trimethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96026PBRKidney membranesRAT3H-PK11195Triethyl((3-nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)silane>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96027PBRKidney membranesRAT3H-PK111956-(3,3-Dimethylbut-1-yn-1-yl)-3-nitro-2-(trifluoromethyl)-2H-chromene>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96028PBRKidney membranesRAT3H-PK11195N-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)acetamide>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96029PBRKidney membranesRAT3H-PK111954-((3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)ethynyl)benzoic acid>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96030PBRKidney membranesRAT3H-PK111952-(3-(3-Nitro-2-(trifluoromethyl)-2H-chromen-6-yl)prop-2-yn-1-yl)isoindoline-1,3-dione>10000Jung et al 2021Jan 15, 2025Jan 15, 2025
96031MORCLONEDHUMAN3H-DAMGO4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96032MORCLONEDHUMAN3H-DAMGO4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96033MORCLONEDHUMAN3H-DAMGO4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96034MORCLONEDHUMAN3H-DAMGO4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96035MORCLONEDHUMAN3H-DAMGO4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96036MORCLONEDHUMAN3H-DAMGO4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96037MORCLONEDHUMAN3H-DAMGO4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96038MORCLONEDHUMAN3H-DAMGO4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96039MORCLONEDHUMAN3H-DAMGO4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96040MORCLONEDHUMAN3H-DAMGO3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96041Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96042Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96043Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96044Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid660Jung et al 2020Jan 15, 2025Jan 28, 2025
96045Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96046Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96047Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96048Sigma 1CLONEDHUMAN3H-Pentazocine(+)4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96049Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid500Jung et al 2020Jan 15, 2025Jan 28, 2025
96050Sigma 1CLONEDHUMAN3H-Pentazocine(+)4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96051Sigma 1CLONEDHUMAN3H-Pentazocine(+)3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid1110Jung et al 2020Jan 15, 2025Jan 28, 2025
96052Sigma 2CLONEDHUMAN3H-DTG4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid6200Jung et al 2020Jan 15, 2025Jan 28, 2025
96053Sigma 2CLONEDHUMAN3H-DTG4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96054Sigma 2CLONEDHUMAN3H-DTG4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96055Sigma 2CLONEDHUMAN3H-DTG4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid560Jung et al 2020Jan 15, 2025Jan 28, 2025
96056Sigma 2CLONEDHUMAN3H-DTG4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid2290Jung et al 2020Jan 15, 2025Jan 28, 2025
96057Sigma 2CLONEDHUMAN3H-DTG4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid1350Jung et al 2020Jan 15, 2025Jan 28, 2025
96058Sigma 2CLONEDHUMAN3H-DTG4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid300Jung et al 2020Jan 15, 2025Jan 28, 2025
96059Sigma 2CLONEDHUMAN3H-DTG4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate400Jung et al 2020Jan 15, 2025Jan 28, 2025
96060Sigma 2CLONEDHUMAN3H-DTG4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid2960Jung et al 2020Jan 15, 2025Jan 28, 2025
96061Sigma 2CLONEDHUMAN3H-DTG4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96062Sigma 2CLONEDHUMAN3H-DTG3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96063DATCLONEDHUMAN3H-WIN 35,4284′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96064DATCLONEDHUMAN3H-WIN 35,4284-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96065DATCLONEDHUMAN3H-WIN 35,4284-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96066DATCLONEDHUMAN3H-WIN 35,4284-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96067DATCLONEDHUMAN3H-WIN 35,4284-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96068DATCLONEDHUMAN3H-WIN 35,4284′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96069DATCLONEDHUMAN3H-WIN 35,4284′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96070DATCLONEDHUMAN3H-WIN 35,4284-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96071DATCLONEDHUMAN3H-WIN 35,4284′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96072DATCLONEDHUMAN3H-WIN 35,4284′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96073DATCLONEDHUMAN3H-WIN 35,4283-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96074NETCLONEDHUMAN3H-Nisoxetine4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96075NETCLONEDHUMAN3H-Nisoxetine4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96076NETCLONEDHUMAN3H-Nisoxetine4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96077NETCLONEDHUMAN3H-Nisoxetine4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96078NETCLONEDHUMAN3H-Nisoxetine4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96079NETCLONEDHUMAN3H-Nisoxetine4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96080NETCLONEDHUMAN3H-Nisoxetine4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96081NETCLONEDHUMAN3H-Nisoxetine4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96082NETCLONEDHUMAN3H-Nisoxetine4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96083NETCLONEDHUMAN3H-Nisoxetine4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96084NETCLONEDHUMAN3H-Nisoxetine3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96085SERTCLONEDHUMAN3H-CITALOPRAM4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96086SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96087SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96088SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96089SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96090SERTCLONEDHUMAN3H-CITALOPRAM4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96091SERTCLONEDHUMAN3H-CITALOPRAM4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96092SERTCLONEDHUMAN3H-CITALOPRAM4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96093SERTCLONEDHUMAN3H-CITALOPRAM4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96094SERTCLONEDHUMAN3H-CITALOPRAM4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96095SERTCLONEDHUMAN3H-CITALOPRAM3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96096PBRKidney membranesRAT3H-PK111954′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96097PBRKidney membranesRAT3H-PK111954-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96098PBRKidney membranesRAT3H-PK111954-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96099PBRKidney membranesRAT3H-PK111954-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96100PBRKidney membranesRAT3H-PK111954-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96101PBRKidney membranesRAT3H-PK111954′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96102PBRKidney membranesRAT3H-PK111954′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96103PBRKidney membranesRAT3H-PK111954-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96104PBRKidney membranesRAT3H-PK111954′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96105PBRKidney membranesRAT3H-PK111954′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96106PBRKidney membranesRAT3H-PK111953-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961075-HT1ACLONEDHUMAN3H-WAY1006354′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961085-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961095-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961105-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961115-HT1ACLONEDHUMAN3H-WAY1006354-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961125-HT1ACLONEDHUMAN3H-WAY1006354′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961135-HT1ACLONEDHUMAN3H-WAY1006354′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961145-HT1ACLONEDHUMAN3H-WAY1006354-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961155-HT1ACLONEDHUMAN3H-WAY1006354′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961165-HT1ACLONEDHUMAN3H-WAY1006354′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961175-HT1ACLONEDHUMAN3H-WAY1006353-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961185-HT1BCLONEDHUMAN3H-GR-1257434′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961195-HT1BCLONEDHUMAN3H-GR-1257434-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961205-HT1BCLONEDHUMAN3H-GR-1257434-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961215-HT1BCLONEDHUMAN3H-GR-1257434-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961225-HT1BCLONEDHUMAN3H-GR-1257434-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961235-HT1BCLONEDHUMAN3H-GR-1257434′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961245-HT1BCLONEDHUMAN3H-GR-1257434′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961255-HT1BCLONEDHUMAN3H-GR-1257434-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961265-HT1BCLONEDHUMAN3H-GR-1257434′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961275-HT1BCLONEDHUMAN3H-GR-1257434′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961285-HT1BCLONEDHUMAN3H-GR-1257433-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961295-HT1DCLONEDHUMAN3H-GR-1257434′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961305-HT1DCLONEDHUMAN3H-GR-1257434-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961315-HT1DCLONEDHUMAN3H-GR-1257434-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961325-HT1DCLONEDHUMAN3H-GR-1257434-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961335-HT1DCLONEDHUMAN3H-GR-1257434-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961345-HT1DCLONEDHUMAN3H-GR-1257434′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961355-HT1DCLONEDHUMAN3H-GR-1257434′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961365-HT1DCLONEDHUMAN3H-GR-1257434-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961375-HT1DCLONEDHUMAN3H-GR-1257434′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961385-HT1DCLONEDHUMAN3H-GR-1257434′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961395-HT1DCLONEDHUMAN3H-GR-1257433-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961405-HT1ECLONEDHUMAN3H-5-HT4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961415-HT1ECLONEDHUMAN3H-5-HT4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961425-HT1ECLONEDHUMAN3H-5-HT4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961435-HT1ECLONEDHUMAN3H-5-HT4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961445-HT1ECLONEDHUMAN3H-5-HT4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961455-HT1ECLONEDHUMAN3H-5-HT4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961465-HT1ECLONEDHUMAN3H-5-HT4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961475-HT1ECLONEDHUMAN3H-5-HT4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961485-HT1ECLONEDHUMAN3H-5-HT4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961495-HT1ECLONEDHUMAN3H-5-HT4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961505-HT1ECLONEDHUMAN3H-5-HT3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961515-HT2ACLONEDHUMAN3H-KETANSERIN4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961525-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961535-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961545-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid1370Jung et al 2020Jan 15, 2025Jan 15, 2025
961555-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961565-HT2ACLONEDHUMAN3H-KETANSERIN4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961575-HT2ACLONEDHUMAN3H-KETANSERIN4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961585-HT2ACLONEDHUMAN3H-KETANSERIN4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961595-HT2ACLONEDHUMAN3H-KETANSERIN4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961605-HT2ACLONEDHUMAN3H-KETANSERIN4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961615-HT2ACLONEDHUMAN3H-KETANSERIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961625-HT2BCLONEDHUMAN3H-LSD4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961635-HT2BCLONEDHUMAN3H-LSD4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961645-HT2BCLONEDHUMAN3H-LSD4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961655-HT2BCLONEDHUMAN3H-LSD4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961665-HT2BCLONEDHUMAN3H-LSD4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961675-HT2BCLONEDHUMAN3H-LSD4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961685-HT2BCLONEDHUMAN3H-LSD4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961695-HT2BCLONEDHUMAN3H-LSD4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961705-HT2BCLONEDHUMAN3H-LSD4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961715-HT2BCLONEDHUMAN3H-LSD4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961725-HT2BCLONEDHUMAN3H-LSD3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961735-HT2CCLONEDHUMAN3H-MESULERGINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961745-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961755-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961765-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961775-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961785-HT2CCLONEDHUMAN3H-MESULERGINE4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961795-HT2CCLONEDHUMAN3H-MESULERGINE4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961805-HT2CCLONEDHUMAN3H-MESULERGINE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961815-HT2CCLONEDHUMAN3H-MESULERGINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961825-HT2CCLONEDHUMAN3H-MESULERGINE4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961835-HT2CCLONEDHUMAN3H-MESULERGINE3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961845-HT3CLONEDHUMAN3H-GR-656304′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961855-HT3CLONEDHUMAN3H-GR-656304-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961865-HT3CLONEDHUMAN3H-GR-656304-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961875-HT3CLONEDHUMAN3H-GR-656304-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961885-HT3CLONEDHUMAN3H-GR-656304-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961895-HT3CLONEDHUMAN3H-GR-656304′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961905-HT3CLONEDHUMAN3H-GR-656304′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961915-HT3CLONEDHUMAN3H-GR-656304-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961925-HT3CLONEDHUMAN3H-GR-656304′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961935-HT3CLONEDHUMAN3H-GR-656304′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961945-HT3CLONEDHUMAN3H-GR-656303-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961955-HT5ACLONEDHUMAN3H-LSD4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961965-HT6CLONEDHUMAN3H-LSD4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961975-HT7CLONEDHUMAN3H-LSD4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961985-HT5ACLONEDHUMAN3H-LSD4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
961995-HT6CLONEDHUMAN3H-LSD4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962005-HT7CLONEDHUMAN3H-LSD4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962015-HT5ACLONEDHUMAN3H-LSD4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962025-HT6CLONEDHUMAN3H-LSD4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962035-HT7CLONEDHUMAN3H-LSD4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962045-HT5ACLONEDHUMAN3H-LSD4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962055-HT6CLONEDHUMAN3H-LSD4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962065-HT7CLONEDHUMAN3H-LSD4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962075-HT5ACLONEDHUMAN3H-LSD4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962085-HT6CLONEDHUMAN3H-LSD4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962095-HT7CLONEDHUMAN3H-LSD4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962105-HT5ACLONEDHUMAN3H-LSD4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962115-HT6CLONEDHUMAN3H-LSD4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962125-HT7CLONEDHUMAN3H-LSD4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962135-HT5ACLONEDHUMAN3H-LSD4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962145-HT6CLONEDHUMAN3H-LSD4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962155-HT7CLONEDHUMAN3H-LSD4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962165-HT5ACLONEDHUMAN3H-LSD4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962175-HT6CLONEDHUMAN3H-LSD4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962185-HT7CLONEDHUMAN3H-LSD4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962195-HT5ACLONEDHUMAN3H-LSD4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962205-HT6CLONEDHUMAN3H-LSD4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962215-HT7CLONEDHUMAN3H-LSD4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962225-HT5ACLONEDHUMAN3H-LSD4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962235-HT6CLONEDHUMAN3H-LSD4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962245-HT7CLONEDHUMAN3H-LSD4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962255-HT5ACLONEDHUMAN3H-LSD3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962265-HT6CLONEDHUMAN3H-LSD3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
962275-HT7CLONEDHUMAN3H-LSD3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96228Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96229Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96230Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96231Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96232Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96233Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96234Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96235Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96236Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96237Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96238Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96239Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96240Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96241Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96242Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96243Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96244Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96245Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96246Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96247Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96248Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96249Alpha1ACLONEDHUMAN3H-PRAZOSIN4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96250Alpha1BCLONEDHUMAN3H-PRAZOSIN4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96251Alpha1DCLONEDHUMAN3H-PRAZOSIN4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96252Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96253Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96254Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96255Alpha1ACLONEDHUMAN3H-PRAZOSIN4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96256Alpha1BCLONEDHUMAN3H-PRAZOSIN4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96257Alpha1DCLONEDHUMAN3H-PRAZOSIN4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96258Alpha1ACLONEDHUMAN3H-PRAZOSIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96259Alpha1BCLONEDHUMAN3H-PRAZOSIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96260Alpha1DCLONEDHUMAN3H-PRAZOSIN3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96261Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96262Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96263Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96264Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96265Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96266Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96267Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96268Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96269Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96270Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96271Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96272Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96273Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96274Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96275Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96276Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96277Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96278Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96279Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96280Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96281Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96282Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96283Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96284Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96285Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96286Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96287Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96288Alpha2ACLONEDHUMAN3H-RAUWOLSCINE4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid960Jung et al 2020Jan 15, 2025Jan 28, 2025
96289Alpha2BCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid5800Jung et al 2020Jan 15, 2025Jan 28, 2025
96290Alpha2CCLONEDHUMAN3H-RAUWOLSCINE4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid2710Jung et al 2020Jan 15, 2025Jan 28, 2025
96291Alpha2ACLONEDHUMAN3H-RAUWOLSCINE3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96292Alpha2BCLONEDHUMAN3H-RAUWOLSCINE3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96293Alpha2CCLONEDHUMAN3H-RAUWOLSCINE3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96294Beta 1CLONEDHUMAN125I-iodo-pindolol4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96295Beta3CLONEDHUMAN125I-iodo-pindolol4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96296Beta 1CLONEDHUMAN125I-iodo-pindolol4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96297Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96298Beta 1CLONEDHUMAN125I-iodo-pindolol4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96299Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96300Beta 1CLONEDHUMAN125I-iodo-pindolol4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96301Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96302Beta 1CLONEDHUMAN125I-iodo-pindolol4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96303Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96304Beta 1CLONEDHUMAN125I-iodo-pindolol4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96305Beta3CLONEDHUMAN125I-iodo-pindolol4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96306Beta 1CLONEDHUMAN125I-iodo-pindolol4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96307Beta3CLONEDHUMAN125I-iodo-pindolol4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96308Beta 1CLONEDHUMAN125I-iodo-pindolol4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96309Beta3CLONEDHUMAN125I-iodo-pindolol4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96310Beta 1CLONEDHUMAN125I-iodo-pindolol4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96311Beta3CLONEDHUMAN125I-iodo-pindolol4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96312Beta 1CLONEDHUMAN125I-iodo-pindolol4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96313Beta3CLONEDHUMAN125I-iodo-pindolol4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96314Beta 1CLONEDHUMAN125I-iodo-pindolol3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96315Beta3CLONEDHUMAN125I-iodo-pindolol3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96316Beta 2CLONEDHUMAN3H-CGP121774′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96317Beta 2CLONEDHUMAN3H-CGP121774-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96318Beta 2CLONEDHUMAN3H-CGP121774-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96319Beta 2CLONEDHUMAN3H-CGP121774-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96320Beta 2CLONEDHUMAN3H-CGP121774-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96321Beta 2CLONEDHUMAN3H-CGP121774′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96322Beta 2CLONEDHUMAN3H-CGP121774′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96323Beta 2CLONEDHUMAN3H-CGP121774-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96324Beta 2CLONEDHUMAN3H-CGP121774′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96325Beta 2CLONEDHUMAN3H-CGP121774′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96326Beta 2CLONEDHUMAN3H-CGP121773-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96327BZPCEREBRAL CORTEXRATFNZ4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96328BZPCEREBRAL CORTEXRATFNZ4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96329BZPCEREBRAL CORTEXRATFNZ4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96330BZPCEREBRAL CORTEXRATFNZ4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96331BZPCEREBRAL CORTEXRATFNZ4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96332BZPCEREBRAL CORTEXRATFNZ4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96333BZPCEREBRAL CORTEXRATFNZ4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96334BZPCEREBRAL CORTEXRATFNZ4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96335BZPCEREBRAL CORTEXRATFNZ4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96336BZPCEREBRAL CORTEXRATFNZ4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96337BZPCEREBRAL CORTEXRATFNZ3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96338D1CLONEDHUMAN3H-SCH233904′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96339D5CLONEDHUMAN3H-SCH233904′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96340D1CLONEDHUMAN3H-SCH233904-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96341D5CLONEDHUMAN3H-SCH233904-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96342D1CLONEDHUMAN3H-SCH233904-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96343D5CLONEDHUMAN3H-SCH233904-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96344D1CLONEDHUMAN3H-SCH233904-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96345D5CLONEDHUMAN3H-SCH233904-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96346D1CLONEDHUMAN3H-SCH233904-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96347D5CLONEDHUMAN3H-SCH233904-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96348D1CLONEDHUMAN3H-SCH233904′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96349D5CLONEDHUMAN3H-SCH233904′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96350D1CLONEDHUMAN3H-SCH233904′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96351D5CLONEDHUMAN3H-SCH233904′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96352D1CLONEDHUMAN3H-SCH233904-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96353D5CLONEDHUMAN3H-SCH233904-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96354D1CLONEDHUMAN3H-SCH233904′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96355D5CLONEDHUMAN3H-SCH233904′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96356D1CLONEDHUMAN3H-SCH233904′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96357D5CLONEDHUMAN3H-SCH233904′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96358D1CLONEDHUMAN3H-SCH233903-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96359D5CLONEDHUMAN3H-SCH233903-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96360D2CLONEDHUMAN3H-N-Methylspiperone4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96361D3CLONEDHUMAN3H-N-Methylspiperone4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96362D4CLONEDHUMAN3H-N-Methylspiperone4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96363D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96364D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96365D4CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96366D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96367D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96368D4CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96369D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96370D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96371D4CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96372D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96373D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96374D4CLONEDHUMAN3H-N-Methylspiperone4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96375D2CLONEDHUMAN3H-N-Methylspiperone4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96376D3CLONEDHUMAN3H-N-Methylspiperone4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96377D4CLONEDHUMAN3H-N-Methylspiperone4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96378D2CLONEDHUMAN3H-N-Methylspiperone4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96379D3CLONEDHUMAN3H-N-Methylspiperone4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96380D4CLONEDHUMAN3H-N-Methylspiperone4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96381D2CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96382D3CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96383D4CLONEDHUMAN3H-N-Methylspiperone4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96384D2CLONEDHUMAN3H-N-Methylspiperone4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96385D3CLONEDHUMAN3H-N-Methylspiperone4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96386D4CLONEDHUMAN3H-N-Methylspiperone4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96387D2CLONEDHUMAN3H-N-Methylspiperone4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96388D3CLONEDHUMAN3H-N-Methylspiperone4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96389D4CLONEDHUMAN3H-N-Methylspiperone4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96390D2CLONEDHUMAN3H-N-Methylspiperone3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96391D3CLONEDHUMAN3H-N-Methylspiperone3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96392D4CLONEDHUMAN3H-N-Methylspiperone3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96393DORCLONEDHUMAN3H-DADLE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96394DORCLONEDHUMAN3H-DADLE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96395DORCLONEDHUMAN3H-DADLE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96396DORCLONEDHUMAN3H-DADLE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96397DORCLONEDHUMAN3H-DADLE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96398DORCLONEDHUMAN3H-DADLE4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96399DORCLONEDHUMAN3H-DADLE4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid2630Jung et al 2020Jan 15, 2025Jan 28, 2025
96400DORCLONEDHUMAN3H-DADLE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96401DORCLONEDHUMAN3H-DADLE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid2480Jung et al 2020Jan 15, 2025Jan 28, 2025
96402DORCLONEDHUMAN3H-DADLE4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid3790Jung et al 2020Jan 15, 2025Jan 28, 2025
96403DORCLONEDHUMAN3H-DADLE3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid2960Jung et al 2020Jan 15, 2025Jan 28, 2025
96404KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96405KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96406KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96407KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96408KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96409KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96410KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96411KORCEREBRAL CORTEXRAT3H-MUSCIMOL4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96412KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96413KORCEREBRAL CORTEXRAT3H-MUSCIMOL4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96414KORCEREBRAL CORTEXRAT3H-MUSCIMOL3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 27, 2025
96415H1CLONEDHUMAN3H-PYRILAMINE4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96416H1CLONEDHUMAN3H-PYRILAMINE4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96417H1CLONEDHUMAN3H-PYRILAMINE4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96418H1CLONEDHUMAN3H-PYRILAMINE4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96419H1CLONEDHUMAN3H-PYRILAMINE4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96420H1CLONEDHUMAN3H-PYRILAMINE4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96421H1CLONEDHUMAN3H-PYRILAMINE4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96422H1CLONEDHUMAN3H-PYRILAMINE4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96423H1CLONEDHUMAN3H-PYRILAMINE4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96424H1CLONEDHUMAN3H-PYRILAMINE4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96425H1CLONEDHUMAN3H-PYRILAMINE3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964265-HT1DCLONEDHUMAN125I-aminopotentidine4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964275-HT1DCLONEDHUMAN125I-aminopotentidine4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964285-HT1DCLONEDHUMAN125I-aminopotentidine4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964295-HT1DCLONEDHUMAN125I-aminopotentidine4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964305-HT1DCLONEDHUMAN125I-aminopotentidine4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964315-HT1DCLONEDHUMAN125I-aminopotentidine4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964325-HT1DCLONEDHUMAN125I-aminopotentidine4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964335-HT1DCLONEDHUMAN125I-aminopotentidine4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964345-HT1DCLONEDHUMAN125I-aminopotentidine4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964355-HT1DCLONEDHUMAN125I-aminopotentidine4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
964365-HT1DCLONEDHUMAN125I-aminopotentidine3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96437H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96438H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96439H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96440H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96441H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96442H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96443H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96444H3CLONEDHUMAN3H-Alpha-methylhistamine4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96445H3CLONEDHUMAN3H-Alpha-methylhistamine4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96446H3CLONEDHUMAN3H-Alpha-methylhistamine4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96447H3CLONEDHUMAN3H-Alpha-methylhistamine3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96448H4CLONEDHUMAN3H-Histamine4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96449H4CLONEDHUMAN3H-Histamine4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96450H4CLONEDHUMAN3H-Histamine4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96451H4CLONEDHUMAN3H-Histamine4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96452H4CLONEDHUMAN3H-Histamine4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96453H4CLONEDHUMAN3H-Histamine4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96454H4CLONEDHUMAN3H-Histamine4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96455H4CLONEDHUMAN3H-Histamine4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96456H4CLONEDHUMAN3H-Histamine4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96457H4CLONEDHUMAN3H-Histamine4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96458H4CLONEDHUMAN3H-Histamine3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96459KORCLONEDHUMAN3H-U695934′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96460KORCLONEDHUMAN3H-U695934-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96461KORCLONEDHUMAN3H-U695934-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96462KORCLONEDHUMAN3H-U695934-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid1790Jung et al 2020Jan 15, 2025Jan 28, 2025
96463KORCLONEDHUMAN3H-U695934-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96464KORCLONEDHUMAN3H-U695934′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96465KORCLONEDHUMAN3H-U695934′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96466KORCLONEDHUMAN3H-U695934-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96467KORCLONEDHUMAN3H-U695934′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96468KORCLONEDHUMAN3H-U695934′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96469KORCLONEDHUMAN3H-U695933-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96470M1CLONEDHUMAN3H-QNB4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96471M2CLONEDHUMAN3H-QNB4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96472M5CLONEDHUMAN3H-QNB4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96473M1CLONEDHUMAN3H-QNB4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96474M2CLONEDHUMAN3H-QNB4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96475M5CLONEDHUMAN3H-QNB4-(4-(1-Propylpiperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)- phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96476M1CLONEDHUMAN3H-QNB4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96477M2CLONEDHUMAN3H-QNB4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96478M5CLONEDHUMAN3H-QNB4-(4-(1-(Hex-5-yn-1-yl)pipe ridin-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96479M1CLONEDHUMAN3H-QNB4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96480M2CLONEDHUMAN3H-QNB4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96481M5CLONEDHUMAN3H-QNB4-(4-(1-(1-Amino-3,6,9,12,15,18-hexaoxahenicosan-21-oyl)- piperidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2-naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96482M1CLONEDHUMAN3H-QNB4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96483M2CLONEDHUMAN3H-QNB4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96484M5CLONEDHUMAN3H-QNB4-(4-(Quinuclidin-4-yl)phenyl)-7-(4-(trifluoromethyl)phenyl)-2- naphthoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96485M1CLONEDHUMAN3H-QNB4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96486M2CLONEDHUMAN3H-QNB4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96487M5CLONEDHUMAN3H-QNB4′-(Quinuclidin-4-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3- triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96488M1CLONEDHUMAN3H-QNB4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96489M2CLONEDHUMAN3H-QNB4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96490M5CLONEDHUMAN3H-QNB4′-(3-Azabicyclo[4.1.0]heptan-6-yl)-5-(4-(4-(trifluoromethyl)- phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96491M1CLONEDHUMAN3H-QNB4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96492M2CLONEDHUMAN3H-QNB4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96493M5CLONEDHUMAN3H-QNB4-(4-(1-Methylquinuclidin-1-ium-4-yl)phenyl)-7-(4- (trifluoromethyl)phenyl)-2-naphthoate>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96494M1CLONEDHUMAN3H-QNB4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96495M2CLONEDHUMAN3H-QNB4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96496M5CLONEDHUMAN3H-QNB4′-Carbamoyl-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96497M1CLONEDHUMAN3H-QNB4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96498M2CLONEDHUMAN3H-QNB4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96499M5CLONEDHUMAN3H-QNB4′-(Piperidin-4-yl)-5-(1-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96500M1CLONEDHUMAN3H-QNB3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96501M2CLONEDHUMAN3H-QNB3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96502M5CLONEDHUMAN3H-QNB3-(5-((3-Aminopropyl)carbamoyl)thiophen-2-yl)-5-(1-(4- (trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)benzoic Acid>10000Jung et al 2020Jan 15, 2025Jan 15, 2025
96503MORCLONEDHUMAN3H-DAMGO4′-(Piperazin-1-yl)-5-(4-(4-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-1-yl)-[1,1′-biphenyl]-3-carboxylic Acid>10000Jung et al 2020Jan 15, 2025Jan 28, 2025
96504D1CLONEDHUMAN[3H]-SCH233906-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione5.7Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96505D2CLONEDHUMAN[3H]-N-methylspiperone6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96506D3CLONEDHUMAN[3H]-N-methylspiperone6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96507D4CLONEDHUMAN[3H]-N-methylspiperone6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96508D5CLONEDHUMAN[3H]-SCH233906-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione6.7Martini ML et al 2019aJan 15, 2025Jan 28, 2025
965095-HT1ACLONEDHUMAN[3H]-Way1006356-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965105-HT1BCLONEDHUMAN[3H]5-CT6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965115-HT1DCLONEDHUMAN[3H]5-CT6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965125-HT1ECLONEDHUMAN[3H]5-HT6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965135-HT2ACLONEDHUMAN[3H]-ketanserin6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965145-HT2BCLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965155-HT3CLONEDHUMAN[3H]GR656306-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965165-HT4CLONEDHUMAN[3H]GR1138086-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965175-HT5ACLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965185-HT6CLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965195-HT7CLONEDHUMAN[3H]-LSD6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96520Alpha1ACLONEDHUMAN[3H]-prazosin6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96521Alpha1BCLONEDHUMAN[3H]-prazosin6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96522Alpha2ACLONEDHUMAN[3H]-rauwolscine6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96523Beta1CLONEDHUMAN[125I]-Pindolol6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96524Beta2CLONEDHUMAN[3H]-CGP121776-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96525MORCLONEDHUMAN[3H]-DAMGO6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96526KORCLONEDHUMAN[3H]-U695936-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96527M1CLONEDHUMAN[3H]-NMS6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96528M2CLONEDHUMAN[3H]-NMS6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96529M3CLONEDHUMAN[3H]-NMS6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96530Sigma 1CLONEDHUMAN[3H]-Pentazocine6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96531H1CLONEDHUMAN[3H]-Pyrilamine6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
965325-HT1DCLONEDHUMAN[125I]-Iodoaminopotentidine6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96533DATCLONEDHUMAN[3H]-Win354286-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96534SERTCLONEDHUMAN[3H]-citalopram6-(4-(Furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-1,5-dimethyl-pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96535D1CLONEDHUMAN[3H]-SCH233901-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione10Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96536D2CLONEDHUMAN[3H]-N-methylspiperone1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96537D3CLONEDHUMAN[3H]-N-methylspiperone1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96538D4CLONEDHUMAN[3H]-N-methylspiperone1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96539D5CLONEDHUMAN[3H]-SCH233901-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione15Martini ML et al 2019aJan 15, 2025Jan 28, 2025
965405-HT1ACLONEDHUMAN[3H]-Way1006351-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965415-HT1BCLONEDHUMAN[3H]5-CT1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965425-HT1DCLONEDHUMAN[3H]5-CT1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965435-HT1ECLONEDHUMAN[3H]5-HT1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965445-HT2ACLONEDHUMAN[3H]-ketanserin1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965455-HT2BCLONEDHUMAN[3H]-LSD1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965465-HT3CLONEDHUMAN[3H]GR656301-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965475-HT4CLONEDHUMAN[3H]GR1138081-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965485-HT5ACLONEDHUMAN[3H]-LSD1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965495-HT6CLONEDHUMAN[3H]-LSD1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965505-HT7CLONEDHUMAN[3H]-LSD1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96551Alpha1ACLONEDHUMAN[3H]-prazosin1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96552Alpha1BCLONEDHUMAN[3H]-prazosin1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96553Alpha2ACLONEDHUMAN[3H]-rauwolscine1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96554Beta1CLONEDHUMAN[125I]-Pindolol1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96555Beta2CLONEDHUMAN[3H]-CGP121771-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96556MORCLONEDHUMAN[3H]-DAMGO1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96557KORCLONEDHUMAN[3H]-U695931-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96558M1CLONEDHUMAN[3H]-NMS1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96559M2CLONEDHUMAN[3H]-NMS1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione7700Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96560M3CLONEDHUMAN[3H]-NMS1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96561Sigma 1CLONEDHUMAN[3H]-Pentazocine1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96562H1CLONEDHUMAN[3H]-Pyrilamine1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
965635-HT1DCLONEDHUMAN[125I]-Iodoaminopotentidine1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96564DATCLONEDHUMAN[3H]-Win354281-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96565SERTCLONEDHUMAN[3H]-citalopram1-Cyclopropyl-6-(4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl)-5-methylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96566D1CLONEDHUMAN[3H]-SCH233906-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione70Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96567D2CLONEDHUMAN[3H]-N-methylspiperone6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96568D3CLONEDHUMAN[3H]-N-methylspiperone6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96569D4CLONEDHUMAN[3H]-N-methylspiperone6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96570D5CLONEDHUMAN[3H]-SCH233906-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione171Martini ML et al 2019aJan 15, 2025Jan 28, 2025
965715-HT1ACLONEDHUMAN[3H]-Way1006356-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965725-HT1BCLONEDHUMAN[3H]5-CT6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965735-HT1DCLONEDHUMAN[3H]5-CT6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965745-HT1ECLONEDHUMAN[3H]5-HT6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965755-HT2ACLONEDHUMAN[3H]-ketanserin6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965765-HT2BCLONEDHUMAN[3H]-LSD6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965775-HT3CLONEDHUMAN[3H]GR656306-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965785-HT4CLONEDHUMAN[3H]GR1138086-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965795-HT5ACLONEDHUMAN[3H]-LSD6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965805-HT6CLONEDHUMAN[3H]-LSD6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
965815-HT7CLONEDHUMAN[3H]-LSD6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96582Alpha1ACLONEDHUMAN[3H]-prazosin6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96583Alpha1BCLONEDHUMAN[3H]-prazosin6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96584Alpha2ACLONEDHUMAN[3H]-rauwolscine6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione6900Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96585Beta1CLONEDHUMAN[125I]-Pindolol6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96586Beta2CLONEDHUMAN[3H]-CGP121776-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96587MORCLONEDHUMAN[3H]-DAMGO6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96588KORCLONEDHUMAN[3H]-U695936-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96589M1CLONEDHUMAN[3H]-NMS6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96590M2CLONEDHUMAN[3H]-NMS6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione6900Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96591M3CLONEDHUMAN[3H]-NMS6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96592Sigma 1CLONEDHUMAN[3H]-Pentazocine6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96593H1CLONEDHUMAN[3H]-Pyrilamine6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
965945-HT1DCLONEDHUMAN[125I]-Iodoaminopotentidine6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96595DATCLONEDHUMAN[3H]-Win354286-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96596SERTCLONEDHUMAN[3H]-citalopram6-(4-((4-Methoxy-3-(trifluoromethyl)pyridin-2-yl)oxy)-2-methyl-phenyl)-1,5-dimethylpyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96597D1CLONEDHUMAN[3H]-SCH233901,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione93Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96598D2CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96599D3CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96600D4CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96601D5CLONEDHUMAN[3H]-SCH233901,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione185Martini ML et al 2019aJan 15, 2025Jan 28, 2025
966025-HT1ACLONEDHUMAN[3H]-Way1006351,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966035-HT1BCLONEDHUMAN[3H]5-CT1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966045-HT1DCLONEDHUMAN[3H]5-CT1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966055-HT1ECLONEDHUMAN[3H]5-HT1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966065-HT2ACLONEDHUMAN[3H]-ketanserin1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966075-HT2BCLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966085-HT3CLONEDHUMAN[3H]GR656301,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966095-HT4CLONEDHUMAN[3H]GR1138081,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966105-HT5ACLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966115-HT6CLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966125-HT7CLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96613Alpha1ACLONEDHUMAN[3H]-prazosin1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96614Alpha1BCLONEDHUMAN[3H]-prazosin1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96615Alpha2ACLONEDHUMAN[3H]-rauwolscine1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96616Beta1CLONEDHUMAN[125I]-Pindolol1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96617Beta2CLONEDHUMAN[3H]-CGP121771,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96618MORCLONEDHUMAN[3H]-DAMGO1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96619KORCLONEDHUMAN[3H]-U695931,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96620M1CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96621M2CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96622M3CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96623Sigma 1CLONEDHUMAN[3H]-Pentazocine1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96624H1CLONEDHUMAN[3H]-Pyrilamine1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
966255-HT1DCLONEDHUMAN[125I]-Iodoaminopotentidine1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96626DATCLONEDHUMAN[3H]-Win354281,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96627SERTCLONEDHUMAN[3H]-citalopram1,5-Dimethyl-6-(2-methyl-4-((2-methylfuro[3,2-c]pyridin-4-yl)-oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96628D1CLONEDHUMAN[3H]-SCH233901,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione14Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96629D2CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96630D3CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96631D4CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96632D5CLONEDHUMAN[3H]-SCH233901,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione90Martini ML et al 2019aJan 15, 2025Jan 28, 2025
966335-HT1ACLONEDHUMAN[3H]-Way1006351,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966345-HT1BCLONEDHUMAN[3H]5-CT1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966355-HT1DCLONEDHUMAN[3H]5-CT1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966365-HT1ECLONEDHUMAN[3H]5-HT1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966375-HT2ACLONEDHUMAN[3H]-ketanserin1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966385-HT2BCLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966395-HT3CLONEDHUMAN[3H]GR656301,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966405-HT4CLONEDHUMAN[3H]GR1138081,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966415-HT5ACLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966425-HT6CLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966435-HT7CLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96644Alpha1ACLONEDHUMAN[3H]-prazosin1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96645Alpha1BCLONEDHUMAN[3H]-prazosin1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96646Alpha2ACLONEDHUMAN[3H]-rauwolscine1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96647Beta1CLONEDHUMAN[125I]-Pindolol1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96648Beta2CLONEDHUMAN[3H]-CGP121771,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96649MORCLONEDHUMAN[3H]-DAMGO1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96650KORCLONEDHUMAN[3H]-U695931,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96651M1CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96652M2CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96653M3CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione4200Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96654Sigma 1CLONEDHUMAN[3H]-Pentazocine1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96655H1CLONEDHUMAN[3H]-Pyrilamine1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96656DATCLONEDHUMAN[3H]-Win354281,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96657SERTCLONEDHUMAN[3H]-citalopram1,5-Dimethyl-6-(2-methyl-4-((1-methyl-1H-pyrrolo[3,2-c]pyridin-4-yl)oxy)phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96658D1CLONEDHUMAN[3H]-SCH233901,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione5.1Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96659D2CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96660D3CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96661D4CLONEDHUMAN[3H]-N-methylspiperone1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96662D5CLONEDHUMAN[3H]-SCH233901,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione53Martini ML et al 2019aJan 15, 2025Jan 28, 2025
966635-HT1ACLONEDHUMAN[3H]-Way1006351,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966645-HT1BCLONEDHUMAN[3H]5-CT1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966655-HT1DCLONEDHUMAN[3H]5-CT1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966665-HT1ECLONEDHUMAN[3H]5-HT1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966675-HT2ACLONEDHUMAN[3H]-ketanserin1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966685-HT2BCLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966695-HT3CLONEDHUMAN[3H]GR656301,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966705-HT4CLONEDHUMAN[3H]GR1138081,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966715-HT5ACLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966725-HT6CLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
966735-HT7CLONEDHUMAN[3H]-LSD1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96674Alpha1ACLONEDHUMAN[3H]-prazosin1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96675Alpha1BCLONEDHUMAN[3H]-prazosin1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96676Alpha2ACLONEDHUMAN[3H]-rauwolscine1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96677Beta1CLONEDHUMAN[125I]-Pindolol1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96678Beta2CLONEDHUMAN[3H]-CGP121771,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 29, 2025
96679MORCLONEDHUMAN[3H]-DAMGO1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96680KORCLONEDHUMAN[3H]-U695931,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96681M1CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96682M2CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96683M3CLONEDHUMAN[3H]-NMS1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione4600Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96684Sigma 1CLONEDHUMAN[3H]-Pentazocine1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96685H1CLONEDHUMAN[3H]-Pyrilamine1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
966865-HT1DCLONEDHUMAN[125I]-Iodoaminopotentidine1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96687DATCLONEDHUMAN[3H]-Win354281,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 15, 2025
96688SERTCLONEDHUMAN[3H]-citalopram1,5-Dimethyl-6-(2-methyl-4-(thieno[2,3-c]pyridin-7-yloxy)-phenyl)pyrimidine-2,4(1H,3H)-dione>10000Martini ML et al 2019aJan 15, 2025Jan 28, 2025
96689D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propoxy)phenyl)acetamide167.2Huang L et al 2020Jan 15, 2025Jan 28, 2025
96690D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)phenyl) Acetamide>10000Huang L et al 2020Jan 15, 2025Jan 28, 2025
96691D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(pyridin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 28, 2025
96692D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)acetamide467.3Huang L et al 2020Jan 15, 2025Jan 28, 2025
96693D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide498.2Huang L et al 2020Jan 15, 2025Jan 28, 2025
96694D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide2.1Huang L et al 2020Jan 15, 2025Jan 28, 2025
96695D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)propoxy)phenyl) acetamide79.1Huang L et al 2020Jan 15, 2025Jan 28, 2025
96696D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(benzo[b]thiophen-4-yl)piperazin-1-yl)propoxy)phenyl)acetamide16.3Huang L et al 2020Jan 15, 2025Jan 28, 2025
96697D2STRIATUMRAT[3H]spiperoneRISPERIDONE3.8Huang L et al 2020Jan 15, 2025Jan 28, 2025
96698D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) propionamide>10000Huang L et al 2020Jan 15, 2025Jan 28, 2025
96699D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) benzamide>10000Huang L et al 2020Jan 15, 2025Jan 28, 2025
96700D2STRIATUMRAT[3H]spiperoneN-(2-fluoro-4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide148.3Huang L et al 2020Jan 15, 2025Jan 28, 2025
96701D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)-2-methylphenyl)acetamide150.3Huang L et al 2020Jan 15, 2025Jan 28, 2025
96702D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)benzyl)acetamide1589Huang L et al 2020Jan 15, 2025Jan 28, 2025
96703D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)-N-methylacetamide20.6Huang L et al 2020Jan 15, 2025Jan 28, 2025
96704D2STRIATUMRAT[3H]spiperoneN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide1143Huang L et al 2020Jan 15, 2025Jan 28, 2025
96705D2STRIATUMRAT[3H]spiperoneN-(4-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 28, 2025
96706D2STRIATUMRAT[3H]spiperoneN-(3-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 28, 2025
96707D2STRIATUMRAT[3H]spiperoneN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-2-hydroxypropoxy)phenyl)acetamide119.2Huang L et al 2020Jan 15, 2025Jan 28, 2025
967085-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967095-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)phenyl) Acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967105-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(pyridin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide1988Huang L et al 2020Jan 15, 2025Jan 15, 2025
967115-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967125-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967135-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide3.5Huang L et al 2020Jan 15, 2025Jan 15, 2025
967145-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)propoxy)phenyl) acetamide69.7Huang L et al 2020Jan 15, 2025Jan 15, 2025
967155-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(benzo[b]thiophen-4-yl)piperazin-1-yl)propoxy)phenyl)acetamide258Huang L et al 2020Jan 15, 2025Jan 15, 2025
967165-HT1ACORTEXRAT[3H]8-OH-DPATRISPERIDONE271Huang L et al 2020Jan 15, 2025Jan 15, 2025
967175-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) propionamide76.3Huang L et al 2020Jan 15, 2025Jan 15, 2025
967185-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) benzamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967195-HT1ACORTEXRAT[3H]8-OH-DPATN-(2-fluoro-4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide122.1Huang L et al 2020Jan 15, 2025Jan 15, 2025
967205-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)-2-methylphenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967215-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)benzyl)acetamide2142Huang L et al 2020Jan 15, 2025Jan 15, 2025
967225-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)-N-methylacetamide21.3Huang L et al 2020Jan 15, 2025Jan 15, 2025
967235-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide1232Huang L et al 2020Jan 15, 2025Jan 15, 2025
967245-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967255-HT1ACORTEXRAT[3H]8-OH-DPATN-(3-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967265-HT1ACORTEXRAT[3H]8-OH-DPATN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-2-hydroxypropoxy)phenyl)acetamide155.6Huang L et al 2020Jan 15, 2025Jan 15, 2025
967275-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propoxy)phenyl)acetamide288.9Huang L et al 2020Jan 15, 2025Jan 15, 2025
967285-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propoxy)phenyl) Acetamide447.9Huang L et al 2020Jan 15, 2025Jan 15, 2025
967295-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(pyridin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide2341Huang L et al 2020Jan 15, 2025Jan 15, 2025
967305-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967315-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967325-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide7.8Huang L et al 2020Jan 15, 2025Jan 15, 2025
967335-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)propoxy)phenyl) acetamide116.9Huang L et al 2020Jan 15, 2025Jan 15, 2025
967345-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(benzo[b]thiophen-4-yl)piperazin-1-yl)propoxy)phenyl)acetamide109Huang L et al 2020Jan 15, 2025Jan 15, 2025
967355-HT2ACORTEXRAT[3H]ketanserinRISPERIDONE0.39Huang L et al 2020Jan 15, 2025Jan 15, 2025
967365-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) propionamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967375-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) benzamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967385-HT2ACORTEXRAT[3H]ketanserinN-(2-fluoro-4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide41.8Huang L et al 2020Jan 15, 2025Jan 15, 2025
967395-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)-2-methylphenyl)acetamide135.2Huang L et al 2020Jan 15, 2025Jan 15, 2025
967405-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)benzyl)acetamide141.1Huang L et al 2020Jan 15, 2025Jan 15, 2025
967415-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)-N-methylacetamide12.7Huang L et al 2020Jan 15, 2025Jan 15, 2025
967425-HT2ACORTEXRAT[3H]ketanserinN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide223.7Huang L et al 2020Jan 15, 2025Jan 15, 2025
967435-HT2ACORTEXRAT[3H]ketanserinN-(4-(2-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)ethoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967445-HT2ACORTEXRAT[3H]ketanserinN-(3-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl)acetamide>10000Huang L et al 2020Jan 15, 2025Jan 15, 2025
967455-HT2ACORTEXRAT[3H]ketanserinN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)-2-hydroxypropoxy)phenyl)acetamide72.2Huang L et al 2020Jan 15, 2025Jan 15, 2025
967465-HT6CLONEDHUMAN[3H]lysergic acid diethylamideN-(4-(3-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)propoxy)phenyl) acetamide12.9Huang L et al 2020Jan 15, 2025Jan 15, 2025
967475-HT6CLONEDHUMAN[3H]lysergic acid diethylamideRISPERIDONE1190Huang L et al 2020Jan 15, 2025Jan 15, 2025
967485-HT6CLONEDHUMAN[3H]lysergic acid diethylamideN-(4-(4-(4-(6-fluorobenzo[d]isoxazol-3-yl)piperidin-1-yl)butoxy)phenyl)acetamide765Huang L et al 2020Jan 15, 2025Jan 15, 2025