99749 DOR CLONED HUMAN 3H-DPDPE (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 0.8 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99750 DOR CLONED HUMAN 3H-DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide 4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99751 DOR CLONED HUMAN 3H-DPDPE (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99752 DOR CLONED HUMAN 3H-DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl] propyl}-Nmethylpropanamide 1.6 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99753 DOR CLONED HUMAN 3H-DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 57 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99754 KOR CLONED HUMAN 3H-U69593 (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 86 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99755 KOR CLONED HUMAN 3H-U69593 (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl] propyl}-Nmethylpropanamide 43 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99756 KOR CLONED HUMAN 3H-U69593 (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 68 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99757 KOR CLONED HUMAN 3H-U69593 (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide 37 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99758 KOR CLONED HUMAN 3H-U69593 (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 3 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99759 KOR CLONED HUMAN 3H-U69593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4- chloroph enyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4- tetrahydroisoquinoline-3 91 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99760 KOR CLONED HUMAN 3H-U69593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4- chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3- carboxamide 13 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99761 KOR CLONED HUMAN 3H-U69593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car 9 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99762 KOR CLONED HUMAN 3H-U69593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 230 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99763 Alpha1A CLONED HUMAN 125I-HEAT (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 6800 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99764 Alpha1A CLONED HUMAN 125I-HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 6600 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99765 Alpha1A CLONED HUMAN 125I-HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 4600 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99766 Alpha1A CLONED HUMAN 125I-HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99767 Alpha1A CLONED HUMAN 125I-HEAT (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99768 Alpha1A CLONED HUMAN 125I-HEAT (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99769 Alpha2A CLONED HUMAN 125I-Clonidine (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99770 Alpha2A CLONED HUMAN 125I-Clonidine (S)-2-[(S)-2-Amino-3-(tetrahydroisoquinoline-3-carboxamide)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4- >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99771 Alpha2A CLONED HUMAN 125I-Clonidine (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99772 Alpha2A CLONED HUMAN 125I-Clonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide 4700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99773 Alpha2A CLONED HUMAN 125I-Clonidine (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99774 Alpha2A CLONED HUMAN 125I-Clonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99775 Alpha2C CLONED HUMAN 125I-Clonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99776 Alpha2C CLONED HUMAN 125I-Clonidine (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99777 Alpha2C CLONED HUMAN 125I-Clonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide 240 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99778 Alpha2C CLONED HUMAN 125I-Clonidine (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 280 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99779 Alpha2C CLONED HUMAN 125I-Clonidine (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-ca >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99780 Alpha2C CLONED HUMAN 125I-Clonidine (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99781 D2 CLONED HUMAN 3H-N-Methylspiperone (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99782 D2 CLONED HUMAN 3H-N-Methylspiperone (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99783 D2 CLONED HUMAN 3H-N-Methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99784 D2 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide 2200 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99785 D2 CLONED HUMAN 3H-N-Methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99786 D2 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99787 D3 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99788 D3 CLONED HUMAN 3H-N-Methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 4300 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99789 D3 CLONED HUMAN 3H-N-Methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide 890 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99790 D3 CLONED HUMAN 3H-N-Methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99791 D3 CLONED HUMAN 3H-N-Methylspiperone (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car 6700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99792 D3 CLONED HUMAN 3H-N-Methylspiperone (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99793 NET CLONED HUMAN 3H-Nisoxetine (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99794 NET CLONED HUMAN 3H-Nisoxetine (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99795 NET CLONED HUMAN 3H-Nisoxetine (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99796 NET CLONED HUMAN 3H-Nisoxetine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99797 NET CLONED HUMAN 3H-Nisoxetine (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2400 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99798 NET CLONED HUMAN 3H-Nisoxetine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 750 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99799 SERT CLONED HUMAN 3H-CITALOPRAM (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 280 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99800 SERT CLONED HUMAN 3H-CITALOPRAM (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99801 SERT CLONED HUMAN 3H-CITALOPRAM (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99802 SERT CLONED HUMAN 3H-CITALOPRAM (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99803 SERT CLONED HUMAN 3H-CITALOPRAM (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-ca 5700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99804 SERT CLONED HUMAN 3H-CITALOPRAM (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1400 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99805 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99806 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-ca >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99807 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1900 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99808 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99809 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 47 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99810 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 410 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99811 MOR CLONED RAT [3H]DAMGO (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 88 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99812 MOR CLONED RAT [3H]DAMGO (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 7 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99813 MOR CLONED RAT [3H]DAMGO (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 16 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99814 MOR CLONED RAT [3H]DAMGO (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 12 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99815 MOR CLONED RAT [3H]DAMGO (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99816 MOR CLONED RAT [3H]DAMGO (S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 35 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99817 MOR CLONED RAT [3H]DAMGO (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 10 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99818 MOR CLONED RAT [3H]DAMGO (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 7 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99819 MOR CLONED RAT [3H]DAMGO (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 0.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99820 MOR CLONED RAT [3H]DAMGO YaGF-NH2 2.8 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99821 MOR CLONED RAT [3H]DAMGO DALEA 7.7 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99822 DOR CLONED HUMAN [3H]DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 57 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99823 DOR CLONED HUMAN [3H]DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 1.6 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99824 DOR CLONED HUMAN [3H]DPDPE (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99825 DOR CLONED HUMAN [3H]DPDPE (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99826 DOR CLONED HUMAN [3H]DPDPE (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 0.8 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99827 DOR CLONED HUMAN [3H]DPDPE (S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 20 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99828 DOR CLONED HUMAN [3H]DPDPE (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 0.88 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99829 DOR CLONED HUMAN [3H]DPDPE (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 0.91 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99830 DOR CLONED HUMAN [3H]DPDPE (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 13 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99831 DOR CLONED HUMAN [3H]DPDPE YaGF-NH2 300 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99832 DOR CLONED HUMAN [3H]DPDPE DALEA 2.4 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99833 KOR CLONED HUMAN [3H]U69,593 (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 86 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99834 KOR CLONED HUMAN [3H]U69,593 (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 43 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99835 KOR CLONED HUMAN [3H]U69,593 (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 68 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99836 KOR CLONED HUMAN [3H]U69,593 (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 37 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99837 KOR CLONED HUMAN [3H]U69,593 (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 3 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99838 KOR CLONED HUMAN [3H]U69,593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 91 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99839 KOR CLONED HUMAN [3H]U69,593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 13 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99840 KOR CLONED HUMAN [3H]U69,593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 9 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99841 KOR CLONED HUMAN [3H]U69,593 (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 230 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99842 Alpha1A CLONED HUMAN [125I] HEAT (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 6800 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99843 Alpha1A CLONED HUMAN [125I] HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 6600 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99844 Alpha1A CLONED HUMAN [125I] HEAT (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 4600 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99845 Alpha1A CLONED HUMAN [125I] HEAT (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99846 Alpha2A CLONED HUMAN [125I] iodoclonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 4700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99847 Alpha2C CLONED HUMAN [125I] iodoclonidine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 240 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99848 Alpha2C CLONED HUMAN [125I] iodoclonidine (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 280 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 29, 2025
99849 D2 CLONED HUMAN [3H]N-methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 2200 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99850 D2 CLONED HUMAN [3H]N-methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99851 D3 CLONED HUMAN [3H]N-methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99852 D3 CLONED HUMAN [3H]N-methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 4300 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99853 D3 CLONED HUMAN [3H]N-methylspiperone (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide 890 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99854 D3 CLONED HUMAN [3H]N-methylspiperone (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99855 D3 CLONED HUMAN [3H]N-methylspiperone (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 6700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99856 NET CLONED HUMAN [3H] Nisoxetine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 750 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99857 NET CLONED HUMAN [3H] Nisoxetine (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 2400 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99858 SERT CLONED HUMAN [3H] Citalopram (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 280 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99859 SERT CLONED HUMAN [3H] Citalopram (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb 5700 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99860 SERT CLONED HUMAN [3H] Citalopram (S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1400 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 28, 2025
99861 Sigma 1 CLONED HUMAN [3H] pentazocine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide 410 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99862 Sigma 1 CLONED HUMAN [3H] pentazocine (R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 47 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99863 Sigma 1 CLONED HUMAN [3H] pentazocine (S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide >10000 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99864 Sigma 1 CLONED HUMAN [3H] pentazocine (R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide 1900 Mehr-un-Nisa et al 2015 Jan 15, 2025 Jan 15, 2025
99865 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride 138 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99866 5-HT2A HIPPOCAMPUS MOUSE 3H-KETANSERIN 1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride 77 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99867 5-HT7 HYPOTHALAMUS MOUSE 3H-5-CT 1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride 1277 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99868 5-HT2A HIPPOCAMPUS MOUSE 3H- Ketanserin 7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride 205 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99869 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride 7 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99870 5-HT1A HIPPOCAMPUS MOUSE 3H-8-OH-DPAT 7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride 22 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99871 5-HT7 HYPOTHALAMUS MOUSE 3H-5-CT 7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride 112 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99872 5-HT7 HYPOTHALAMUS MOUSE 3H-5-CT 7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride 335 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99873 5-HT2A HIPPOCAMPUS MOUSE 3H- Ketanserin (7-{4-[4-(3-chloro-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride) 21 Jastrzębska-Więsek, Magdalena, et al., 2011 Jan 15, 2025 Jan 15, 2025
99874 B1 CORTICAL MEMBRANES Rat brain 3H-BRADYKININ ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99875 ETA CORTICAL MEMBRANES Rat brain 125I-ENDOTHELIN ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99876 ETB CORTICAL MEMBRANES Rat brain 125I-ENDOTHELIN ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99877 NK1 CORTICAL MEMBRANES Rat brain 3H-Leu,4,5 Substance P ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99878 CORTICAL MEMBRANES Rat brain 125I-NPY ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99879 CORTICAL MEMBRANES Rat brain 3H-Neurotensin ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99880 CORTICAL MEMBRANES Rat brain 125I-VIP ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99881 CORTICAL MEMBRANES Rat brain 125I-Omega-Conotoxin ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99882 CORTICAL MEMBRANES Rat brain 3H-Nitrendipine ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99883 CORTICAL MEMBRANES Rat brain 3H-TBOB ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99884 CORTICAL MEMBRANES Rat brain 125I-Apamin ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99885 CORTICAL MEMBRANES Rat brain 3H-Glibenclamide ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99886 CORTICAL MEMBRANES Rat brain 3H-Charybdotoxin ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99887 NET CORTICAL MEMBRANES Rat brain 3H-Nisoxetine ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99888 SLC6A4 CORTICAL MEMBRANES Rat brain 3H-CITALOPRAM ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99889 CORTICAL MEMBRANES Rat brain 3H-GABA ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99890 CORTICAL MEMBRANES Rat brain 3H-Choline Chloride ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99891 SLC6A3 CORTICAL MEMBRANES Rat brain 3H-WIN 35,428 ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99892 AChE CORTICAL MEMBRANES Rat brain UNDEFINED ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 28, 2025
99893 MOA CORTICAL MEMBRANES Rat brain 14C-5-HT ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 29, 2025
99894 MOA CORTICAL MEMBRANES Rat brain 14C-Phenylethylamine ABT-089 >10000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 29, 2025
99895 nAChR7 CLONED HUMAN 125I-Alpha-bgt Nicotine 2000 Sullivan, JP et al., 1997 Jan 15, 2025 Jan 15, 2025
99896 IP HEK293 cells HUMAN 3H-ILOPROST Treprostinil 32.1 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99897 EP1 HEK293 cells HUMAN 3H-PGE2 Treprostinil 212 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99898 EP2 HEK293 cells HUMAN 3H-PGE2 Treprostinil 3.6 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99899 EP3 HEK293 cells HUMAN 3H-PGE2 Treprostinil 2505 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99900 EP4 CHO cells HUMAN 3H-PGE2 Treprostinil 826 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99901 DP1 1321N1 HUMAN 3H-PGD2 Treprostinil 4.4 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99902 FP HEK293 cells HUMAN 3H-PGF2 Treprostinil 4680 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99903 IP HEK293 cells HUMAN 3H-ILOPROST ILOPROST 3.9 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99904 EP1 HEK293 cells HUMAN 3H-PGE2 ILOPROST 1.1 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99905 EP2 HEK293 cells HUMAN 3H-PGE2 ILOPROST 1172 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99906 EP3 HEK293 cells HUMAN 3H-PGE2 ILOPROST 208 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99907 EP4 CHO cells HUMAN 3H-PGE2 ILOPROST 212 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99908 DP1 1321N1 HUMAN 3H-PGD2 ILOPROST 1016 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99909 FP HEK293 cells HUMAN 3H-PGF2 ILOPROST 131 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99910 TP HEK293 cells HUMAN 3H-SQ-29548 ILOPROST 3778 Whittle BJ et al 2012 Jan 15, 2025 Jan 29, 2025
99911 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 542 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99912 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 0.49 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99913 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 2268 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99914 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 2139 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99915 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 537 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99916 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 0.061 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99917 KOR CLONED HUMAN 3H-U69593 3-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride 0.71 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99918 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride 463 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99919 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride 1862 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99920 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride 3539 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99921 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride 670 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99922 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride 10.3 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99923 KOR CLONED HUMAN 3H-U69593 3-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride 2.69 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99924 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride 259 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99925 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride 2743 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99926 DOR CLONED HUMAN 3H-Diprenorphine 3,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 3340 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99927 MOR CLONED HUMAN 3H-DAMGO 3,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 230 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99928 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 0.38 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99929 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 4.62 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99930 MOR CLONED HUMAN 3H-DAMGO 3,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 631 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99931 DOR CLONED HUMAN 3H-Diprenorphine 3,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 2850 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99932 DOR CLONED HUMAN 3H-Diprenorphine 3,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 738 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99933 MOR CLONED HUMAN 3H-DAMGO 3,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 358 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99934 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 19.1 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99935 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 0.14 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99936 MOR CLONED HUMAN 3H-DAMGO 3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 167 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99937 DOR CLONED HUMAN 3H-Diprenorphine 3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 1432 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99938 DOR CLONED HUMAN 3H-Diprenorphine 3,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 2775 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99939 MOR CLONED HUMAN 3H-DAMGO 3,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 584 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99940 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 0.31 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99941 KOR CLONED HUMAN 3H-U69593 3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 2.1 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99942 MOR CLONED HUMAN 3H-DAMGO 3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 211 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99943 DOR CLONED HUMAN 3H-Diprenorphine 3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 1469 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99944 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 428 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99945 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 16.1 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99946 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 3.43 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99947 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 1.85 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99948 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 234 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99949 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 1637 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99950 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 1099 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99951 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 192 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99952 KOR CLONED HUMAN 3H-U69593 3-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 43.5 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99953 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 3.56 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99954 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride 460 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99955 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride >10000 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99956 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride >10000 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99957 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 398 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99958 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.072 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99959 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.04 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99960 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 851 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99961 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride >10000 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99962 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride >10000 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99963 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 557 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99964 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.12 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99965 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 3.37 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99966 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 523 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99967 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 1312 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99968 DOR CLONED HUMAN 3H-Diprenorphine N-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine 2178 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99969 MOR CLONED HUMAN 3H-DAMGO N-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine 1065 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99970 KOR CLONED HUMAN 3H-U69593 N-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine 79.1 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99971 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 5.9 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99972 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 826 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99973 DOR CLONED HUMAN 3H-Diprenorphine 3-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride >10000 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99974 KOR CLONED HUMAN 3H-U69593 3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 0.017 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99975 MOR CLONED HUMAN 3H-DAMGO 3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride 826 Erli F et al 2017 Jan 15, 2025 Jan 28, 2025
99976 5-HT1A CLONED HUMAN 3H-WAY100635 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99977 5-HT1A CLONED HUMAN 3H-WAY100635 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99978 5-HT1B CLONED HUMAN 3H-5CT 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99979 5-HT1B CLONED HUMAN 3H-5CT 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99980 5-HT1D CLONED HUMAN 3H-5CT 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99981 5-HT1D CLONED HUMAN 3H-5CT 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99982 5-HT1E CLONED HUMAN 3H-5HT 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99983 5-HT1E CLONED HUMAN 3H-5HT 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99984 5-HT2A CLONED HUMAN 125I-DOI 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99985 5-HT2A CLONED HUMAN 125I-DOI 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99986 5-HT2B CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99987 5-HT2B CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99988 5-HT2C CLONED HUMAN 3H-MESULERGINE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99989 5-HT2C CLONED HUMAN 3H-MESULERGINE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99990 5-HT3 CLONED HUMAN 3H-LY 278584 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99991 5-HT3 CLONED HUMAN 3H-LY 278584 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99992 5-HT5A CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99993 5-HT5A CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99994 5-HT6 CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99995 5-HT6 CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99996 5-HT7 CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99997 5-HT7 CLONED HUMAN 3H-LSD 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
99998 Alpha1A CLONED HUMAN 125I-HEAT 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
99999 Alpha1A CLONED HUMAN 125I-HEAT 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100000 Alpha1B CLONED HUMAN 125I-HEAT 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100001 Alpha1B CLONED HUMAN 125I-HEAT 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100002 Alpha1D CLONED HUMAN 125I-HEAT 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100003 Alpha1D CLONED HUMAN 125I-HEAT 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100004 Alpha2A CLONED HUMAN 3H-CLONIDINE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100005 Alpha2A CLONED HUMAN 3H-CLONIDINE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100006 Alpha2B CLONED HUMAN 3H-CLONIDINE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100007 Alpha2B CLONED HUMAN 3H-CLONIDINE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100008 Alpha2C CLONED HUMAN 3H-CLONIDINE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100009 Alpha2C CLONED HUMAN 3H-CLONIDINE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100010 Beta 1 CLONED HUMAN 125I-Pindolol 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100011 Beta 1 CLONED HUMAN 125I-Pindolol 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100012 Beta 2 CLONED HUMAN 3H-CGP-12177 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100013 Beta 2 CLONED HUMAN 3H-CGP-12177 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100014 Beta3 CLONED HUMAN 125I-Pindolol 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100015 Beta3 CLONED HUMAN 125I-Pindolol 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100016 CB1 CLONED HUMAN 3H-CP55940 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100017 CB1 CLONED HUMAN 3H-CP55940 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100018 CB2 CLONED HUMAN 3H-CP55940 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100019 CB2 CLONED HUMAN 3H-CP55940 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100020 D1 CLONED HUMAN 3H-SCH23390 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100021 D1 CLONED HUMAN 3H-SCH23390 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100022 D2 CLONED HUMAN 3H-NMS 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100023 D2 CLONED HUMAN 3H-NMS 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100024 D3 CLONED HUMAN 3H-NMS 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100025 D3 CLONED HUMAN 3H-NMS 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100026 D4 CLONED HUMAN 3H-NMS 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100027 D4 CLONED HUMAN 3H-NMS 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100028 D5 CLONED HUMAN 3H-SCH23390 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100029 D5 CLONED HUMAN 3H-SCH23390 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100030 H1 CLONED HUMAN 3H-PYRILAMINE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100031 H1 CLONED HUMAN 3H-PYRILAMINE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100032 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100033 5-HT1D CLONED HUMAN 125I-iodoaminopotentidine 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100034 KOR CLONED HUMAN 3H-U69,593 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100035 KOR CLONED HUMAN 3H-U69,593 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100036 MOR CLONED HUMAN 3H-DAMGO 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100037 MOR CLONED HUMAN 3H-DAMGO 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100038 DOR CLONED HUMAN 3H-DADLE 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100039 DOR CLONED HUMAN 3H-DADLE 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100040 M1 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100041 M1 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100042 M2 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100043 M2 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100044 M3 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100045 M3 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100046 M4 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100047 M4 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100048 M5 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100049 M5 CLONED HUMAN 3H-QNB 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100050 NMDA CLONED HUMAN 3H-MK-801 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100051 NMDA CLONED HUMAN 3H-MK-801 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100052 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100053 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100054 Sigma 2 CLONED HUMAN 3H-DTG 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100055 Sigma 2 CLONED HUMAN 3H-DTG 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100056 mGluR5 BRAIN RAT 3H-MPEP 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100057 mGluR5 BRAIN RAT 3H-MPEP 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100058 BZP BRAIN RAT FNZ 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 29, 2025
100059 BZP BRAIN RAT FNZ 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 29, 2025
100060 DAT CLONED HUMAN 3H-WIN 35,428 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100061 DAT CLONED HUMAN 3H-WIN 35,428 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100062 GABAA CLONED HUMAN 3H-MUSCIMOL 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 29, 2025
100063 GABAA CLONED HUMAN 3H-MUSCIMOL 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 29, 2025
100064 NET CLONED HUMAN 3H-Nisoxetine 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100065 NET CLONED HUMAN 3H-Nisoxetine 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide 245 Sundaresan A et al 2015 Jan 15, 2025 Jan 15, 2025
100066 SERT CLONED HUMAN 3H-CITALOPRAM 5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100067 SERT CLONED HUMAN 3H-CITALOPRAM 5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide >10000 Sundaresan A et al 2015 Jan 15, 2025 Jan 28, 2025
100072 5-HT1A CLONED HUMAN [3H]WAY100635 Perospirone 0.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100073 5-HT1A CLONED HUMAN 3H-WAY100635 Cariprazine 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100074 5-HT1B CLONED HUMAN 3H-5-CT Cariprazine 926 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100075 5-HT1D CLONED HUMAN 3H-5-CT Cariprazine 296 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100076 5-HT2A CLONED HUMAN 3H-KETANSERIN Cariprazine 37 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100077 5-HT2B CLONED HUMAN 3H-LSD Cariprazine 0.71 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100078 5-HT2C CLONED HUMAN 3H-MESULERGINE Cariprazine 414 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100079 5-HT5A CLONED HUMAN 3H-LSD Cariprazine 2316 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100080 5-HT6 CLONED HUMAN 3H-LSD Cariprazine 854 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100081 5-HT7 CLONED HUMAN 3H-LSD Cariprazine 20 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100082 Alpha1A CLONED HUMAN 3H-PRAZOSIN Cariprazine 379 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100083 Alpha1B CLONED HUMAN 3H-PRAZOSIN Cariprazine 969 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100084 Alpha1D CLONED HUMAN 3H-PRAZOSIN Cariprazine 1411 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100085 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Cariprazine 88 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100086 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Cariprazine 640 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100087 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Cariprazine 1229 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100088 Beta1 CLONED HUMAN 125I-Pindolol Cariprazine 325 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100089 Beta3 CLONED HUMAN 125I-Pindolol Cariprazine 1882 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100090 D3 CLONED HUMAN 3H-N-Methylspiperone Cariprazine 2.1 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100091 D4 CLONED HUMAN 3H-N-Methylspiperone Cariprazine 1047 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100092 H1 CLONED HUMAN 3H-PYRILAMINE Cariprazine 10 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100093 5-HT1D CLONED HUMAN 125I-Iodo-aminopotentidine Cariprazine 710 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100094 M4 CLONED HUMAN 3H-QNB Cariprazine 1356 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100095 M5 CLONED HUMAN 3H-QNB Cariprazine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100096 SERT CLONED HUMAN 3H-CITALOPRAM Cariprazine 3597 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100097 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) Cariprazine 29 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100098 Sigma 2 CLONED HUMAN 3H-DTG Cariprazine 1531 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100099 D1 CLONED HUMAN 3H-SCH23390 Cariprazine 3749 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100100 D2 CLONED HUMAN 3H-N-Methylspiperone Cariprazine 18 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100101 5-HT1A CLONED HUMAN 3H-WAY100635 Quetiapine 267 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100102 5-HT2A CLONED HUMAN 3H-KETANSERIN Quetiapine 352 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100103 5-HT2B CLONED HUMAN 3H-LSD Quetiapine 86 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100104 5-HT2C CLONED HUMAN 3H-MESULERGINE Quetiapine 3624 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100105 5-HT3 CLONED HUMAN 3H-GR65630 Quetiapine 4330 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100106 5-HT5A CLONED HUMAN 3H-LSD Quetiapine 2300 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100107 5-HT6 CLONED HUMAN 3H-LSD Quetiapine 1777 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100108 5-HT7 CLONED HUMAN 3H-LSD Quetiapine 168 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100109 Alpha1A CLONED HUMAN 3H-PRAZOSIN Quetiapine 261 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100110 Alpha1B CLONED HUMAN 3H-PRAZOSIN Quetiapine 141 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100111 Alpha1D CLONED HUMAN 3H-PRAZOSIN Quetiapine 752 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100112 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Quetiapine 1207 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100113 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Quetiapine 96 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100114 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Quetiapine 166 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100115 D2 CLONED HUMAN 3H-N-Methylspiperone Quetiapine 5037 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100116 D3 CLONED HUMAN 3H-N-Methylspiperone Quetiapine 2193 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100117 D4 CLONED HUMAN 3H-N-Methylspiperone Quetiapine 1651 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100118 D5 CLONED HUMAN 3H-SCH23390 Quetiapine 2133 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100119 H1 CLONED HUMAN 3H-PYRILAMINE Quetiapine 9.1 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100120 5-HT1D CLONED HUMAN 125I-Iodo-aminopotentidine Quetiapine 473 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100121 KOR CLONED HUMAN 3H-U69593 Quetiapine 3489 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100122 M3 CLONED HUMAN 3H-QNB Quetiapine 1294 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100123 M4 CLONED HUMAN 3H-QNB Quetiapine 722 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100124 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) Quetiapine 413 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100125 Sigma 2 CLONED HUMAN 3H-DTG Quetiapine 1566 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100126 D1 CLONED HUMAN 3H-SCH23390 Quetiapine 381 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100127 5-HT1A CLONED HUMAN 3H-WAY100635 Brexpiprazole 1.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100128 5-HT1B CLONED HUMAN 3H-5CT Brexpiprazole 365 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100129 5-HT1D CLONED HUMAN 3H-5CT Brexpiprazole 23 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100130 5-HT1E CLONED HUMAN 3H-5HT Brexpiprazole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100131 5-HT2A CLONED HUMAN 3H-KETANSERIN Brexpiprazole 3.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100132 5-HT2B CLONED HUMAN 3H-LSD Brexpiprazole 1.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100133 5-HT2C CLONED HUMAN 3H-MESULERGINE Brexpiprazole 29 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100134 5-HT3 CLONED HUMAN 3H-GR65630 Brexpiprazole 754 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100135 5-HT5A CLONED HUMAN 3H-LSD Brexpiprazole 614 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100136 5-HT6 CLONED HUMAN 3H-LSD Brexpiprazole 117 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100137 5-HT7 CLONED HUMAN 3H-LSD Brexpiprazole 6.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100138 Alpha1A CLONED HUMAN 3H-PRAZOSIN Brexpiprazole 24 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100139 Alpha1B CLONED HUMAN 3H-PRAZOSIN Brexpiprazole 134 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100140 Alpha1D CLONED HUMAN 3H-PRAZOSIN Brexpiprazole 58 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100141 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Brexpiprazole 39 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100142 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Brexpiprazole 135 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100143 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Brexpiprazole 24 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100144 Beta1 CLONED HUMAN 125I-Pindolol Brexpiprazole 699 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100145 Beta2 CLONED HUMAN 3H-CGP12177 Brexpiprazole >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100146 Beta3 CLONED HUMAN 125I-Pindolol Brexpiprazole 1653 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100147 D2 CLONED HUMAN 3H-N-Methylspiperone Brexpiprazole 40 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100148 D3 CLONED HUMAN 3H-N-Methylspiperone Brexpiprazole 30 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100149 D4 CLONED HUMAN 3H-N-Methylspiperone Brexpiprazole 19 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100150 D5 CLONED HUMAN 3H-SCH23390 Brexpiprazole 465 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100151 DAT CLONED HUMAN 3H-WIN35428 Brexpiprazole 1799 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100152 H1 CLONED HUMAN 3H-PYRILAMINE Brexpiprazole 6.8 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100153 5-HT1D CLONED HUMAN 125I-Iodo-aminopotentidine Brexpiprazole 365 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100154 NET CLONED HUMAN 3H-Nisoxetine Brexpiprazole >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100155 SERT CLONED HUMAN 3H-CITALOPRAM Brexpiprazole 247 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100156 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) Brexpiprazole 287 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100157 Sigma 2 CLONED HUMAN 3H-DTG Brexpiprazole 40 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100158 D1 CLONED HUMAN 3H-SCH23390 Brexpiprazole >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100159 5-HT1A CLONED HUMAN 3H-WAY100635 Amisulpride 3546 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100160 5-HT2A CLONED HUMAN 3H-KETANSERIN Amisulpride 746 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100161 5-HT2B CLONED HUMAN 3H-LSD Amisulpride 74 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100162 5-HT6 CLONED HUMAN 3H-LSD Amisulpride 1356 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100163 5-HT7 CLONED HUMAN 3H-LSD Amisulpride 35 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100164 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Amisulpride 101 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100165 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Amisulpride 465 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100166 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Amisulpride 992 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100167 D2 CLONED HUMAN 3H-N-Methylspiperone Amisulpride 2407 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100168 D4 CLONED HUMAN 3H-N-Methylspiperone Amisulpride 1591 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100169 D3 CLONED HUMAN 3H-N-Methylspiperone Amisulpride 17 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100170 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) Amisulpride 3709 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100171 5-HT1A CLONED HUMAN 3H-WAY100635 Perospirone 0.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100172 5-HT1A CLONED HUMAN 3H-WAY100635 Ziprasidone 1.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100173 5-HT1A CLONED HUMAN 3H-WAY100635 Asenapine 4.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100174 5-HT1A CLONED HUMAN 3H-WAY100635 NEMONAPRIDE 5.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100175 5-HT1A CLONED HUMAN 3H-WAY100635 ARIPIPRAZOLE 13 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100176 5-HT1A CLONED HUMAN 3H-WAY100635 ILOPERIDONE 27 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100177 5-HT1A CLONED HUMAN 3H-WAY100635 Lurasidone HCl 53 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100178 5-HT1A CLONED HUMAN 3H-WAY100635 CLOZAPINE 104 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100179 5-HT1A CLONED HUMAN 3H-WAY100635 ZOTEPINE 131 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100180 5-HT1A CLONED HUMAN 3H-WAY100635 RISPERIDONE 158 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100181 5-HT1A CLONED HUMAN 3H-WAY100635 SERTINDOLE 236 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100182 5-HT1A CLONED HUMAN 3H-WAY100635 Paliperidone 404 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100183 5-HT1A CLONED HUMAN 3H-WAY100635 OLANZAPINE 1114 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100184 5-HT1A CLONED HUMAN 3H-WAY100635 Blonanserin 1215 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100185 5-HT1A CLONED HUMAN 3H-WAY100635 Melperone HCl 1328 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100186 5-HT1A CLONED HUMAN 3H-WAY100635 Remoxapride 2989 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100187 5-HT1A CLONED HUMAN 3H-WAY100635 RS-(+/-)-Sulpriride 7610 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100188 5-HT1B CLONED HUMAN 3H-5CT Asenapine 55 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100189 5-HT1B CLONED HUMAN 3H-5CT Ziprasidone 58 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100190 5-HT1B CLONED HUMAN 3H-5CT ILOPERIDONE 99 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100191 5-HT1B CLONED HUMAN 3H-5CT ZOTEPINE 431 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100192 5-HT1B CLONED HUMAN 3H-5CT SERTINDOLE 501 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100193 5-HT1B CLONED HUMAN 3H-5CT RISPERIDONE 718 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100194 5-HT1B CLONED HUMAN 3H-5CT Paliperidone 876 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100195 5-HT1B CLONED HUMAN 3H-5CT Perospirone 1070 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100196 5-HT1B CLONED HUMAN 3H-5CT Lurasidone HCl 1675 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100197 5-HT1B CLONED HUMAN 3H-5CT CLOZAPINE 2111 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100198 5-HT1B CLONED HUMAN 3H-5CT NEMONAPRIDE 2812 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100199 5-HT1B CLONED HUMAN 3H-5CT OLANZAPINE 3157 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100200 5-HT1B CLONED HUMAN 3H-5CT ARIPIPRAZOLE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100201 5-HT1B CLONED HUMAN 3H-5CT Blonanserin >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100202 5-HT1D CLONED HUMAN 3H-5CT Ziprasidone 1.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100203 5-HT1D CLONED HUMAN 3H-5CT Asenapine 6.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100204 5-HT1D CLONED HUMAN 3H-5CT RISPERIDONE 6.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100205 5-HT1D CLONED HUMAN 3H-5CT ILOPERIDONE 10 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100206 5-HT1D CLONED HUMAN 3H-5CT SERTINDOLE 16 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100207 5-HT1D CLONED HUMAN 3H-5CT Paliperidone 19 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100208 5-HT1D CLONED HUMAN 3H-5CT Perospirone 20 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100209 5-HT1D CLONED HUMAN 3H-5CT ZOTEPINE 48 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100210 5-HT1D CLONED HUMAN 3H-5CT Lurasidone HCl 50 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100211 5-HT1D CLONED HUMAN 3H-5CT ARIPIPRAZOLE 176 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100212 5-HT1D CLONED HUMAN 3H-5CT NEMONAPRIDE 295 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100213 5-HT1D CLONED HUMAN 3H-5CT CLOZAPINE 474 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100214 5-HT1D CLONED HUMAN 3H-5CT Blonanserin 1061 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100215 5-HT1D CLONED HUMAN 3H-5CT OLANZAPINE 1062 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100216 5-HT1D CLONED HUMAN 3H-5CT Melperone HCl >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100217 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Blonanserin 1.6 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100218 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE ILOPERIDONE 8.3 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100219 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE RISPERIDONE 12 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100220 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Lurasidone HCl 62 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100221 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Melperone HCl 103 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100222 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Perospirone 108 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100223 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Perospirone 119 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100224 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Perospirone 123 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100225 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE ZOTEPINE 156 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100226 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Ziprasidone 162 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100227 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Perospirone 183 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100228 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE ARIPIPRAZOLE 190 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100229 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Paliperidone 222 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100230 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE CLOZAPINE 306 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100231 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE RS-(+/-)-Sulpriride 352 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100232 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE SERTINDOLE 353 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100233 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE OLANZAPINE 472 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100234 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE NEMONAPRIDE 1027 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100235 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Asenapine 1624 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100236 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE GMC 1-116 2652 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100237 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE GMC 1-116 3899 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100238 5-HT1E CLONED HUMAN 3H-5HT Asenapine 71 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100239 5-HT1E CLONED HUMAN 3H-5HT GMC 1-116 324.94 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100240 5-HT1E CLONED HUMAN 3H-5HT SERTINDOLE 7451 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100241 5-HT1E CLONED HUMAN 3H-5HT SERTINDOLE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100242 5-HT1E CLONED HUMAN 3H-5HT ARIPIPRAZOLE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100243 5-HT1E CLONED HUMAN 3H-5HT CLOZAPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100244 5-HT1E CLONED HUMAN 3H-5HT SERTINDOLE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100245 5-HT1E CLONED HUMAN 3H-5HT ZOTEPINE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100246 5-HT2A CLONED HUMAN 3H-KETANSERIN Asenapine 0.16 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100247 5-HT2A CLONED HUMAN 3H-KETANSERIN Ziprasidone 0.31 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100248 5-HT2A CLONED HUMAN 3H-KETANSERIN Perospirone 0.44 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100249 5-HT2A CLONED HUMAN 3H-KETANSERIN SERTINDOLE 0.48 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100250 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.64 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100251 5-HT2A CLONED HUMAN 3H-KETANSERIN ZOTEPINE 0.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100252 5-HT2A CLONED HUMAN 3H-KETANSERIN ILOPERIDONE 0.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100253 5-HT2A CLONED HUMAN 3H-KETANSERIN Paliperidone 0.91 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100254 5-HT2A CLONED HUMAN 3H-KETANSERIN OLANZAPINE 9.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100255 5-HT2A CLONED HUMAN 3H-KETANSERIN CLOZAPINE 13 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100256 5-HT2A CLONED HUMAN 3H-KETANSERIN ARIPIPRAZOLE 15 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100257 5-HT2A CLONED HUMAN 3H-KETANSERIN Lurasidone HCl 36 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100258 5-HT2A CLONED HUMAN 3H-KETANSERIN Blonanserin 41 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100259 5-HT2A CLONED HUMAN 3H-KETANSERIN NEMONAPRIDE 56 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100260 5-HT2A CLONED HUMAN 3H-KETANSERIN Melperone HCl 360 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100261 5-HT2A CLONED HUMAN 3H-KETANSERIN Remoxapride 6390 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100262 5-HT2B CLONED HUMAN 3H-LSD Asenapine 0.21 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100263 5-HT2B CLONED HUMAN 3H-LSD ZOTEPINE 1.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100264 5-HT2B CLONED HUMAN 3H-LSD SERTINDOLE 1.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100265 5-HT2B CLONED HUMAN 3H-LSD Perospirone 2.9 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100266 5-HT2B CLONED HUMAN 3H-LSD ARIPIPRAZOLE 3.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100267 5-HT2B CLONED HUMAN 3H-LSD CLOZAPINE 4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100268 5-HT2B CLONED HUMAN 3H-LSD Ziprasidone 4.4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100269 5-HT2B CLONED HUMAN 3H-LSD NEMONAPRIDE 6.1 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100270 5-HT2B CLONED HUMAN 3H-LSD OLANZAPINE 7.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100271 5-HT2B CLONED HUMAN 3H-LSD RISPERIDONE 16 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100272 5-HT2B CLONED HUMAN 3H-LSD Paliperidone 18 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100273 5-HT2B CLONED HUMAN 3H-LSD Blonanserin 20 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100274 5-HT2B CLONED HUMAN 3H-LSD Lurasidone HCl 24 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100275 5-HT2B CLONED HUMAN 3H-LSD ILOPERIDONE 27 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100276 5-HT2B CLONED HUMAN 3H-LSD GMC 1-116 148 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100277 5-HT2B CLONED HUMAN 3H-LSD Remoxapride 194 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100278 5-HT2B CLONED HUMAN 3H-LSD S-(-)-Sulpride 1976 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100279 5-HT2B CLONED HUMAN 3H-LSD Melperone HCl 2264 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100280 5-HT2C CLONED HUMAN 3H-MESULERGINE Asenapine 0.24 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100281 5-HT2C CLONED HUMAN 3H-MESULERGINE SERTINDOLE 1.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100282 5-HT2C CLONED HUMAN 3H-MESULERGINE ZOTEPINE 3.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100283 5-HT2C CLONED HUMAN 3H-MESULERGINE Ziprasidone 4 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100284 5-HT2C CLONED HUMAN 3H-MESULERGINE Perospirone 5.2 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100285 5-HT2C CLONED HUMAN 3H-MESULERGINE OLANZAPINE 16 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100286 5-HT2C CLONED HUMAN 3H-MESULERGINE CLOZAPINE 19 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100287 5-HT2C CLONED HUMAN 3H-MESULERGINE RISPERIDONE 24 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100288 5-HT2C CLONED HUMAN 3H-MESULERGINE Paliperidone 38 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100289 5-HT2C CLONED HUMAN 3H-MESULERGINE ILOPERIDONE 46 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100290 5-HT2C CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 62 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100291 5-HT2C CLONED HUMAN 3H-MESULERGINE ARIPIPRAZOLE 86 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100292 5-HT2C CLONED HUMAN 3H-MESULERGINE Blonanserin 251 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100293 5-HT2C CLONED HUMAN 3H-MESULERGINE Lurasidone HCl 481 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100294 5-HT2C CLONED HUMAN 3H-MESULERGINE NEMONAPRIDE 481 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100295 5-HT2C CLONED HUMAN 3H-MESULERGINE GMC 1-116 615 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100296 5-HT2C CLONED HUMAN 3H-MESULERGINE Remoxapride 3574 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100297 5-HT3 CLONED HUMAN 3H-GR65630 CLOZAPINE 47 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100298 5-HT3 CLONED HUMAN 3H-GR65630 ARIPIPRAZOLE 106 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100299 5-HT3 CLONED HUMAN 3H-GR65630 OLANZAPINE 125 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100300 5-HT3 CLONED HUMAN 3H-GR65630 ZOTEPINE 140 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100301 5-HT3 CLONED HUMAN 3H-GR65630 Asenapine 336 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100302 5-HT3 CLONED HUMAN 3H-GR65630 NEMONAPRIDE 410 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100303 5-HT3 CLONED HUMAN 3H-GR65630 SERTINDOLE 2237 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100304 5-HT3 CLONED HUMAN 3H-GR65630 Ziprasidone 3385 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100305 5-HT3 CLONED HUMAN 3H-GR65630 ILOPERIDONE 3524 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100306 5-HT3 CLONED HUMAN 3H-GR65630 Lurasidone HCl 5264 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100307 5-HT5A CLONED HUMAN 3H-LSD ZOTEPINE 134 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100308 5-HT5A CLONED HUMAN 3H-LSD RISPERIDONE 195 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100309 5-HT5A CLONED HUMAN 3H-LSD ARIPIPRAZOLE 228 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100310 5-HT5A CLONED HUMAN 3H-LSD Ziprasidone 301 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100311 5-HT5A CLONED HUMAN 3H-LSD Perospirone 321 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100312 5-HT5A CLONED HUMAN 3H-LSD ILOPERIDONE 394 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100313 5-HT5A CLONED HUMAN 3H-LSD Asenapine 403 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100314 5-HT5A CLONED HUMAN 3H-LSD Paliperidone 428 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100315 5-HT5A CLONED HUMAN 3H-LSD SERTINDOLE 510 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100316 5-HT5A CLONED HUMAN 3H-LSD Asenapine 540 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100317 5-HT5A CLONED HUMAN 3H-LSD ILOPERIDONE 550 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100318 5-HT5A CLONED HUMAN 3H-LSD Blonanserin 1037 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100319 5-HT5A CLONED HUMAN 3H-LSD Lurasidone HCl 1198 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100320 5-HT5A CLONED HUMAN 3H-LSD GMC 1-116 1357 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100321 5-HT5A CLONED HUMAN 3H-LSD OLANZAPINE 1365 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100322 5-HT5A CLONED HUMAN 3H-LSD NEMONAPRIDE 1538 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100323 5-HT5A CLONED HUMAN 3H-LSD GMC 1-116 1856 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100324 5-HT6 CLONED HUMAN 3H-LSD Asenapine 0.62 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100325 5-HT6 CLONED HUMAN 3H-LSD SERTINDOLE 2.3 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100326 5-HT6 CLONED HUMAN 3H-LSD ZOTEPINE 7.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100327 5-HT6 CLONED HUMAN 3H-LSD OLANZAPINE 13 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100328 5-HT6 CLONED HUMAN 3H-LSD CLOZAPINE 14 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100329 5-HT6 CLONED HUMAN 3H-LSD NEMONAPRIDE 46 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100330 5-HT6 CLONED HUMAN 3H-LSD Ziprasidone 51 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100331 5-HT6 CLONED HUMAN 3H-LSD ILOPERIDONE 140.02 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100332 5-HT6 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 162 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100333 5-HT6 CLONED HUMAN 3H-LSD ILOPERIDONE 183.19 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100334 5-HT6 CLONED HUMAN 3H-LSD Blonanserin 206 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100335 5-HT6 CLONED HUMAN 3H-LSD Perospirone 477 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100336 5-HT6 CLONED HUMAN 3H-LSD GMC 1-116 630.52 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100337 5-HT6 CLONED HUMAN 3H-LSD Paliperidone 681 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100338 5-HT6 CLONED HUMAN 3H-LSD GMC 1-116 781.27 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100339 5-HT6 CLONED HUMAN 3H-LSD Lurasidone HCl 943 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100340 5-HT6 CLONED HUMAN 3H-LSD RISPERIDONE 962 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100341 5-HT6 CLONED HUMAN 3H-LSD Melperone HCl 1635 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100342 5-HT7 CLONED HUMAN 3H-LSD Asenapine 0.33 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100343 5-HT7 CLONED HUMAN 3H-LSD Paliperidone 2.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100344 5-HT7 CLONED HUMAN 3H-LSD RISPERIDONE 3.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100345 5-HT7 CLONED HUMAN 3H-LSD Perospirone 3.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100346 5-HT7 CLONED HUMAN 3H-LSD Ziprasidone 4.7 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100347 5-HT7 CLONED HUMAN 3H-LSD ILOPERIDONE 7.8 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100348 5-HT7 CLONED HUMAN 3H-LSD ZOTEPINE 9.5 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100349 5-HT7 CLONED HUMAN 3H-LSD CLOZAPINE 21 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100350 5-HT7 CLONED HUMAN 3H-LSD SERTINDOLE 30 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100351 5-HT7 CLONED HUMAN 3H-LSD Lurasidone HCl 32 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100352 5-HT7 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 38 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100353 5-HT7 CLONED HUMAN 3H-LSD NEMONAPRIDE 81 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100354 5-HT7 CLONED HUMAN 3H-LSD OLANZAPINE 157 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100355 5-HT7 CLONED HUMAN 3H-LSD GMC 1-116 200 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100356 5-HT7 CLONED HUMAN 3H-LSD Melperone HCl 346 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100357 5-HT7 CLONED HUMAN 3H-LSD Blonanserin 1010 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100358 5-HT7 CLONED HUMAN 3H-LSD RS-(+/-)-Sulpriride 1085 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100359 DAT CLONED HUMAN 3H-WIN 35,428 Cariprazine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100360 NET CLONED HUMAN 3H-Nisoxene Cariprazine >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100361 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE ILOPERIDONE 5.6 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100362 DAT CLONED HUMAN 3H-WIN35428 ILOPERIDONE >10000 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100363 NET CLONED HUMAN 3H-Nisoxetine ILOPERIDONE 535 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
100364 SERT CLONED HUMAN 3H-CITALOPRAM ILOPERIDONE 443 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100365 Alpha1A CLONED HUMAN 3H-PRAZOSIN ILOPERIDONE 1.4 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100366 Alpha1B CLONED HUMAN 3H-PRAZOSIN ILOPERIDONE 224 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100367 Alpha1D CLONED HUMAN 3H-PRAZOSIN ILOPERIDONE 1.2 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100368 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE ILOPERIDONE 11 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100369 Beta1 CLONED HUMAN 125I-Pindolol ILOPERIDONE >10000 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100370 D2 CLONED HUMAN 3H-N-Methylspiperone ILOPERIDONE 369 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100371 D3 CLONED HUMAN 3H-N-Methylspiperone ILOPERIDONE 84 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100372 D4 CLONED HUMAN 3H-N-Methylspiperone ILOPERIDONE 33 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100373 D5 CLONED HUMAN 3H-SCH23390 ILOPERIDONE 173 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100374 H1 CLONED HUMAN 3H-PYRILAMINE ILOPERIDONE 1854 PDSP Certified Data Jan 15, 2025 Jan 28, 2025
100375 NET CLONED HUMAN 3H-Nisoxetine BUPROPION >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100376 SLC6A3 CLONED HUMAN 3H-WIN 35,428 CITALOPRAM >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100377 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Desmethylcitalopram >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100378 SLC6A3 CLONED HUMAN 3H-WIN 35,428 DOXEPIN >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100379 NET CLONED HUMAN 3H-Nisoxetine Etoperidone >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100380 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Etoperidone >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100381 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100382 NET CLONED HUMAN 3H-Nisoxetine Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100383 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Iproniazid >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100384 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Lofepramine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100385 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE mirtazepine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100386 SLC6A3 CLONED HUMAN 3H-WIN 35,428 mirtazepine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100387 SLC6A3 CLONED HUMAN 3H-WIN 35,428 mirtazepine(+) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100388 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE mirtazepine(+) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100389 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE mirtazepine(-) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100390 NET CLONED HUMAN 3H-Nisoxetine mirtazepine(-) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100391 SLC6A3 CLONED HUMAN 3H-WIN 35,428 mirtazepine(-) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100392 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NORTRYPTYLINE 18 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100393 NET CLONED HUMAN 3H-Nisoxetine NORTRYPTYLINE 4.37 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100394 SLC6A3 CLONED HUMAN 3H-WIN 35,428 NORTRYPTYLINE 1140 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100395 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Phenelzine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100396 NET CLONED HUMAN 3H-Nisoxetine Phenelzine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100397 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE TRANYLCYPROMINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100398 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Viloxazine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100399 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Viloxazine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100400 SLC6A3 CLONED HUMAN 3H-WIN 35,428 ZIMELIDINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100401 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Alprazolam >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100402 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Clonazepam >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100403 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE acetazolamide >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100404 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE CARBAMAZEPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100405 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NIFEDIPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100406 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE VERAPAMIL 245 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100407 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE RESERPINE 1460 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100408 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE COCAINE 340 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100409 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE MAZINDOL 39 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100410 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE METHAMPHETAMINE (+) >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100411 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE METHYLPHENIDATE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100412 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE GBR-12935 940 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100413 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE CHLORPHENIRAMINE 15.2 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100414 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE Diphenhydramine 3800 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100415 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE DOPAMINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100416 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE NOREPINEPHRINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100417 SLC6A4 CLONED HUMAN 3H-IMIPRAMINE 5-Hydroxy Tryptamine 2100 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100418 NET CLONED HUMAN 3H-Nisoxetine Alprazolam >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100419 NET CLONED HUMAN 3H-Nisoxetine Clonazepam >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100420 NET CLONED HUMAN 3H-Nisoxetine acetazolamide >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100421 NET CLONED HUMAN 3H-Nisoxetine CARBAMAZEPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100422 NET CLONED HUMAN 3H-Nisoxetine NIFEDIPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100423 NET CLONED HUMAN 3H-Nisoxetine Amphetamine,(+) 530 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100424 NET CLONED HUMAN 3H-Nisoxetine COCAINE 1420 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100425 NET CLONED HUMAN 3H-Nisoxetine MAZINDOL 0.45 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100426 NET CLONED HUMAN 3H-Nisoxetine METHAMPHETAMINE (+) 660 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100427 NET CLONED HUMAN 3H-Nisoxetine METHYLPHENIDATE 234 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100428 NET CLONED HUMAN 3H-Nisoxetine GBR-12935 310 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100429 NET CLONED HUMAN 3H-Nisoxetine CHLORPHENIRAMINE 1440 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100430 NET CLONED HUMAN 3H-Nisoxetine Diphenhydramine 960 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100431 NET CLONED HUMAN 3H-Nisoxetine DOPAMINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100432 NET CLONED HUMAN 3H-Nisoxetine NOREPINEPHRINE 2200 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100433 NET CLONED HUMAN 3H-Nisoxetine 5-Hydroxy Tryptamine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100434 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Alprazolam >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100435 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Clonazepam >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100436 SLC6A3 CLONED HUMAN 3H-WIN 35,428 acetazolamide >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100437 SLC6A3 CLONED HUMAN 3H-WIN 35,428 CARBAMAZEPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100438 SLC6A3 CLONED HUMAN 3H-WIN 35,428 NIFEDIPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100439 SLC6A3 CLONED HUMAN 3H-WIN 35,428 VERAPAMIL >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100440 SLC6A3 CLONED HUMAN 3H-WIN 35,428 RESERPINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100441 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Amphetamine,(+) 2900 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100442 SLC6A3 CLONED HUMAN 3H-WIN 35,428 COCAINE 220 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100443 SLC6A3 CLONED HUMAN 3H-WIN 35,428 MAZINDOL 8.1 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100444 SLC6A3 CLONED HUMAN 3H-WIN 35,428 METHAMPHETAMINE (+) 2800 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100445 SLC6A3 CLONED HUMAN 3H-WIN 35,428 METHYLPHENIDATE 24 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100446 SLC6A3 CLONED HUMAN 3H-WIN 35,428 GBR-12935 27.2 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100447 SLC6A3 CLONED HUMAN 3H-WIN 35,428 CHLORPHENIRAMINE 1060 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100448 SLC6A3 CLONED HUMAN 3H-WIN 35,428 Diphenhydramine 2200 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100449 SLC6A3 CLONED HUMAN 3H-WIN 35,428 DOPAMINE 2400 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100450 SLC6A3 CLONED HUMAN 3H-WIN 35,428 NOREPINEPHRINE >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100451 SLC6A3 CLONED HUMAN 3H-WIN 35,428 5-Hydroxy Tryptamine >10000 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100452 SLC6A3 CLONED HUMAN 3H-WIN 35,428 AMFONELIC ACID 207 Tatsumi M, et al., 1997 Jan 15, 2025 Jan 15, 2025
100453 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-2,6-Dimethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine 110 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100454 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-2,6-Dimethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine 8.67 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100455 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) 2,2,6,6-Tetramethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine 373 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100456 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) 2,2,6,6-Tetramethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine 35.9 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100457 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-2,6-Dimethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 7.43 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100458 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) cis-2,6-Dimethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 18.5 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100459 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) 2,2,6,6-Tetramethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 236 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100460 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine(+) 2,2,6,6-Tetramethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 88.6 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100461 Sigma 2 LIVER RAT 3H-DTG cis-2,6-Dimethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine 90.9 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100462 Sigma 2 LIVER RAT 3H-DTG cis-2,6-Dimethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine 11.1 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100463 Sigma 2 LIVER RAT 3H-DTG 2,2,6,6-Tetramethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine 641 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100464 Sigma 2 LIVER RAT 3H-DTG 2,2,6,6-Tetramethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine 69.8 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100465 Sigma 2 LIVER RAT 3H-DTG cis-2,6-Dimethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 45.4 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100466 Sigma 2 LIVER RAT 3H-DTG cis-2,6-Dimethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 13.8 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100467 Sigma 2 LIVER RAT 3H-DTG 2,2,6,6-Tetramethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 495 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100468 Sigma 2 LIVER RAT 3H-DTG 2,2,6,6-Tetramethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 90.7 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100469 Sigma 1 CORTICAL MEMBRANES GUINEA PIG 3H-Pentazocine PENTAZOCINE (+) 4.1 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100470 Sigma 2 LIVER RAT 3H-DTG DTG 30.2 Niso M et al 2013 Jan 15, 2025 Jan 28, 2025
100471 D1 CLONED HUMAN [3H]SCH23390 F17464 >10000 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100472 5-HT1A CLONED HUMAN [3H]8-OH-DPAT F17464 0.162181 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100473 D2 CLONED HUMAN [3H]spiperone F17464 8.70964 Cosi C et al 2021 Jan 15, 2025 Jan 29, 2025
100474 D2 CLONED HUMAN [3H]spiperone F17464 12.0226 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100475 D3 CLONED HUMAN [3H]spiperone F17464 0.158489 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100476 D4 CLONED HUMAN [3H]spiperone F17464 >10000 Cosi C et al 2021 Jan 15, 2025 Jan 29, 2025
100477 D2 dorsal striatum RAT [3H]nemonapride F17464 5.01187 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100478 5-HT1A HIPPOCAMPUS RAT [3H]8-OH-DPAT F17464 1.25893 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100479 5-HT1D CLONED HUMAN 3H-GR125743 F17464 26.3027 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100480 5-HT2A CLONED HUMAN 3H-KETANSERIN F17464 436.516 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100481 5-HT2B CLONED HUMAN [3H]mesulergine F17464 1548.82 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100482 5-HT2C CLONED HUMAN [3H]mesulergine F17464 1995.26 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100483 Alpha1B CEREBRAL CORTEX PIG 3H-PRAZOSIN F17464 794.328 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100484 Alpha2A CLONED HUMAN UNDEFINED F17464 281.838 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100485 Alpha2B CLONED HUMAN UNDEFINED F17464 208.93 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100486 Alpha2C CLONED HUMAN UNDEFINED F17464 275.423 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100487 Beta 2 CLONED HUMAN UNDEFINED F17464 >10000 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100488 CLONED RAT UNDEFINED F17464 125.893 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100489 5-HT7 CLONED HUMAN UNDEFINED F17464 >10000 Cosi C et al 2021 Jan 15, 2025 Jan 29, 2025
100490 5-HT1B CORTEX RAT UNDEFINED F17464 3981.07 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100491 H1 CLONED HUMAN UNDEFINED F17464 21.3796 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100492 MOR CLONED HUMAN UNDEFINED F17464 141.254 Cosi C et al 2021 Jan 15, 2025 Jan 28, 2025
100493 M1 CLONED HUMAN UNDEFINED F17464 >10000 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100494 M3 CLONED HUMAN UNDEFINED F17464 >10000 Cosi C et al 2021 Jan 15, 2025 Jan 15, 2025
100495 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100496 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide 24 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100497 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100498 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide 25.1 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100499 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100500 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide 21.9 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100501 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100502 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 1.5 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100503 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100504 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 3 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100505 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100506 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 5.5 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100507 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100508 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1H-1,2,3-triazole-4-carboxamide 1023 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100509 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100510 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide 9.7 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100511 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100512 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide 10.7 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100513 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide 3345 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100514 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide 5 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100515 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 1-Benzyl-N-(4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl)-1H-1,2,3-triazole-4-carboxamide 4476 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100516 Sigma 2 LIVER RAT 3H-DTG 1-Benzyl-N-(4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl)-1H-1,2,3-triazole-4-carboxamide 12.4 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100517 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide 8082 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100518 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide 22.5 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100519 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100520 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide 11.6 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100521 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100522 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide 62.1 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100523 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100524 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide 48.2 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100525 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100526 Sigma 2 LIVER RAT 3H-DTG N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 150 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100527 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100528 Sigma 2 LIVER RAT 3H-DTG N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 180 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100529 Sigma 2 LIVER RAT 3H-DTG N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide 410 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100530 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100531 Sigma 2 LIVER RAT 3H-DTG N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide 156 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100532 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100533 Sigma 2 LIVER RAT 3H-DTG N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide 214 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100534 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100535 Sigma 2 LIVER RAT 3H-DTG N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide 93.2 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100536 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100537 Sigma 1 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)benzamide 139 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100538 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-fluoroethoxy)ethyl)-1H-1,2,3-triazol-4-yl)benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100539 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-fluoroethoxy)ethyl)-1H-1,2,3-triazol-4-yl)benzamide 137 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100540 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-(2-fluoroethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)-benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100541 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-(2-fluoroethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)-benzamide 212 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100542 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide 8580 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100543 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide 55 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100544 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100545 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide 66.2 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100546 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(4-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100547 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(4-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide 31.4 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100548 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide 1752 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100549 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide 66 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100550 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-(prop-2-ynyloxy)benzamide 3678 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100551 Sigma 2 LIVER RAT 3H-DTG 5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-(prop-2-ynyloxy)benzamide 12.2 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100552 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) 5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methoxy)-benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100553 Sigma 2 LIVER RAT 3H-DTG 5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methoxy)-benzamide 31.9 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100554 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100555 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide 56.8 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100556 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-2-methoxy-5-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-benzamide 6359 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100557 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-2-methoxy-5-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-benzamide 20.7 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100558 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((2-(2-fluoroethoxy)ethoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100559 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((2-(2-fluoroethoxy)ethoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide 66 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100560 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-(2-fluoroethoxy)benzamide >10000 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100561 Sigma 2 LIVER RAT 3H-DTG N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-(2-fluoroethoxy)benzamide 94 Bai S, et al., 2014 Jan 15, 2025 Jan 15, 2025
100562 GlyR CLONED HUMAN 3H-Glycine CHPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100563 GlyR CLONED HUMAN 3H-Glycine CHPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100564 GlyR CLONED HUMAN 3H-Glycine MCPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100565 GlyR CLONED HUMAN 3H-Glycine CPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100566 GlyR CLONED HUMAN 3H-Glycine L-glutamic acid >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100567 GlyR CLONED HUMAN 3H-Glycine NMDA >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100568 GlyR CLONED HUMAN 3H-Glycine CPP >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100569 NMDA CLONED HUMAN [3H]CPP CHPG(RS) 2089.3 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100570 NMDA CLONED HUMAN [3H]CPP CHPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100571 NMDA CLONED HUMAN [3H]CPP MCPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100572 NMDA CLONED HUMAN [3H]CPP CPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100573 NMDA CLONED HUMAN [3H]CPP L-glutamic acid 218.776 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100574 NMDA CLONED HUMAN [3H]CPP NMDA 9120.11 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100575 NMDA CLONED HUMAN [3H]CPP CPP 69.1831 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 28, 2025
100576 AMPA CLONED HUMAN Functional CHPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100577 AMPA CLONED HUMAN Functional CHPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100578 AMPA CLONED HUMAN Functional MCPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100579 AMPA CLONED HUMAN Functional CPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100580 AMPA CLONED HUMAN Functional L-glutamic acid 371.535 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100581 AMPA CLONED HUMAN Functional NMDA >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100582 AMPA CLONED HUMAN Functional CPP >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100583 KA CLONED HUMAN 3H-Kainic acid CHPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100584 KA CLONED HUMAN 3H-Kainic acid CHPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100585 KA CLONED HUMAN 3H-Kainic acid MCPG(RS) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100586 KA CLONED HUMAN 3H-Kainic acid CPG(S) >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100587 KA CLONED HUMAN 3H-Kainic acid L-glutamic acid 107.152 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100588 KA CLONED HUMAN 3H-Kainic acid NMDA >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100589 KA CLONED HUMAN 3H-Kainic acid CPP >10000 Cavanni P, et.al., 1994 Jan 15, 2025 Jan 15, 2025
100590 CGRP CLONED HUMAN 1251-CGRP N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100591 CGRP CLONED HUMAN 1251-CGRP N2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100592 CGRP CLONED HUMAN 1251-CGRP N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100593 CGRP CLONED HUMAN 1251-CGRP N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100594 CGRP CLONED HUMAN 1251-CGRP N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-L-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100595 CGRP CLONED HUMAN 1251-CGRP N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysine-phenylamide Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100596 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-phenyl-piperazine Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100597 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-piperazine Dihydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100598 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-(4-pyridinyl)piperazine >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100599 CGRP CLONED HUMAN 1251-CGRP N2-[4-Amino-3,5-dibromo-N-(3-phenyl-1-oxopropyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrochloride >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100600 CGRP CLONED HUMAN 1251-CGRP N2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100601 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 1000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100602 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 200 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100603 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperazinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 226 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100604 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate) 250 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100605 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-[2(3H)-oxobenzoxazol-3-yl]-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate) 44 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100606 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[N-[[4-[N-(Aminocarbonyl)phenylamino]-1-piperidinyl]carbonyl]-3,5-dibromo-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate) 4.7 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100607 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.2 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100608 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.03 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100609 CGRP CLONED HUMAN 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-4-phenyl-2(2H)-oxoimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.05 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100610 CGRP SPLEEN RAT 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100611 CGRP SPLEEN RAT 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 56.7 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100612 CGRP SPLEEN marmoset 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 2.7 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100613 CGRP SPLEEN RAT 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 6.4 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100614 CGRP SPLEEN marmoset 1251-CGRP 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.06 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100615 CGRP CLONED HUMAN Functional N2-(3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100616 CGRP CLONED HUMAN Functional N2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100617 CGRP CLONED HUMAN Functional N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100618 CGRP CLONED HUMAN Functional N2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamine >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100619 CGRP CLONED HUMAN Functional N2-[3,5-Dibromo-N-(4-phenyl-1-oxybutyl)-L-tyrosyl]-L-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100620 CGRP CLONED HUMAN Functional N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysine-phenylamide Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100621 CGRP CLONED HUMAN Functional 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-phenyl-piperazine Hydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100622 CGRP CLONED HUMAN Functional 1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-piperazine Dihydrobromide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100623 CGRP CLONED HUMAN Functional 1-[N2-[4-amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl-4-(4-pyridinyl)piperazine >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100624 CGRP CLONED HUMAN Functional N2-[4-Amino-3,5-dibromo-N-(3-phenyl-1-oxopropyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrochloride >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100625 CGRP serum HUMAN Functional N2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysine-2-phenethylamide >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100626 CGRP serum HUMAN Functional 1-[N2-[3,4-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]4-(4-pyridinyl)piperazine 1000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100627 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 200 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100628 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperazinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 226 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100629 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate) 250 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100630 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-[2(3H)-oxobenzoxazol-3-yl]-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate) 44 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100631 CGRP serum HUMAN Functional 1-[N2-[N[[4-[N-(Aminocarbonyl)phenylamino]-1-piperidinyl]carbonyl]-3,5-dibromo-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate) 4.7 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100632 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.2 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100633 CGRP serum HUMAN Functional 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.03 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100634 CGRP rat cloned Functional 1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine >10000 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100635 CGRP rat cloned Functional 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 56.7 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100636 CGRP CLONED RAT Functional 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 6.4 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100637 CGRP SPLEEN marmoset Functional 1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidal-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 2.7 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100638 CGRP SPLEEN marmoset Functional 1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 0.06 Rudolf K, et al., 2005 Jan 15, 2025 Jan 15, 2025
100639 5-HT1A CLONED HUMAN 3H-WAY100635 CYPROHEPTADINE 50 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100640 5-HT1B CLONED HUMAN 3H-5CT CYPROHEPTADINE 1600 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100641 5-HT1D CLONED HUMAN 3H-5CT CYPROHEPTADINE 670 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100642 5-HT2A CLONED HUMAN 3H-KETANSERIN CYPROHEPTADINE 1.9 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100643 5-HT2B CLONED HUMAN 3H-LSD CYPROHEPTADINE 2.6 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100644 5-HT2C CLONED HUMAN 3H-MESULERGINE CYPROHEPTADINE 18 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100645 5-HT3 CLONED HUMAN 3H-GR-65630 CYPROHEPTADINE 235 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100646 5-HT5A CLONED HUMAN 3H-LSD CYPROHEPTADINE 57 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100647 5-HT6 CLONED HUMAN 3H-LSD CYPROHEPTADINE 96 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100648 5-HT7 CLONED HUMAN 3H-LSD CYPROHEPTADINE 30 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100649 D1 CLONED HUMAN 3H-SCH23390 CYPROHEPTADINE 10 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100650 D2 CLONED HUMAN 3H-Methylspiperone CYPROHEPTADINE 74 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100651 D4 CLONED HUMAN 3H-Methylspiperone CYPROHEPTADINE 120 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100652 D5 CLONED HUMAN 3H-SCH23390 CYPROHEPTADINE 60 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100653 SERT CLONED HUMAN 3H-CITALOPRAM CYPROHEPTADINE >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100654 NET CLONED HUMAN 3H-Nisoxetine CYPROHEPTADINE 2550 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100655 DAT CLONED HUMAN [3H]WIN35428 CYPROHEPTADINE 4100 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100656 H1 CLONED HUMAN 3H-PYRILAMINE CYPROHEPTADINE 2.3 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100657 Alpha1A CLONED HUMAN 3H-PRAZOSIN CYPROHEPTADINE 45 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100658 Alpha1B CLONED HUMAN 3H-PRAZOSIN CYPROHEPTADINE >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100659 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE CYPROHEPTADINE 330 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100660 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE CYPROHEPTADINE 220 Young, R., et. al., 2005 Jan 15, 2025 Jan 29, 2025
100661 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE CYPROHEPTADINE 160 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100662 5-HT1D CLONED HUMAN [3H]Tiotidine CYPROHEPTADINE 4.8 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100663 M1 CLONED HUMAN 3H-QNB CYPROHEPTADINE 19 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100664 M2 CLONED HUMAN 3H-QNB CYPROHEPTADINE 18 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100665 M3 CLONED HUMAN 3H-QNB CYPROHEPTADINE 12 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100666 M4 CLONED HUMAN 3H-QNB CYPROHEPTADINE 19 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100667 M5 CLONED HUMAN 3H-QNB CYPROHEPTADINE 4.5 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100668 CLONED HUMAN 125I-Clonidine CYPROHEPTADINE 204 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100669 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) CYPROHEPTADINE >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100670 Sigma 2 PC12 RAT 3H-DTG CYPROHEPTADINE 750 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100671 5-HT1A CLONED HUMAN 3H-WAY100635 Pizotyline 270 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100672 5-HT1B CLONED HUMAN 3H-5CT Pizotyline 1415 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100673 5-HT1D CLONED HUMAN 3H-5CT Pizotyline 770 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100674 5-HT1E CLONED HUMAN 3H-5HT Pizotyline 820 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100675 5-HT2A CLONED HUMAN 3H-KETANSERIN Pizotyline 2 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100676 5-HT2B CLONED HUMAN 3H-LSD Pizotyline 2.3 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100677 5-HT2C CLONED HUMAN 3H-MESULERGINE Pizotyline 8.4 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100678 5-HT3 CLONED HUMAN 3H-GR-65630 Pizotyline 95 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100679 5-HT5A CLONED HUMAN 3H-LSD Pizotyline 110 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100680 5-HT6 CLONED HUMAN 3H-LSD Pizotyline 74 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100681 5-HT7 CLONED HUMAN 3H-LSD Pizotyline 17 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100682 D1 CLONED HUMAN 3H-SCH23390 Pizotyline 3.5 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100683 D2 CLONED HUMAN 3H-N-Methylspiporone Pizotyline 87 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100684 D4 CLONED HUMAN 3H-N-Methylspiporone Pizotyline 64 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100685 D5 CLONED HUMAN 3H-SCH23390 Pizotyline 50 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100686 SERT CLONED HUMAN 3H-CITALOPRAM Pizotyline >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100687 DAT CLONED HUMAN 3H-WIN 35,428 Pizotyline >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100688 NET CLONED HUMAN 3H-Nisoxetine Pizotyline 710 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100689 H1 CLONED HUMAN 3H-PYRILAMINE Pizotyline 1.9 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100690 5-HT1D CLONED HUMAN 125I-aminopotentidine Pizotyline 1.4 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100691 Alpha1A CLONED HUMAN 3H-PRAZOSIN Pizotyline 65 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100692 Alpha1B CLONED HUMAN 3H-PRAZOSIN Pizotyline >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100693 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE Pizotyline 660 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100694 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE Pizotyline 225 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100695 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE Pizotyline 390 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100696 Beta1 CLONED HUMAN 125I-Pindolol Pizotyline >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100697 Beta2 CLONED HUMAN 3H-CGP-12177 Pizotyline >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100698 Beta1 CLONED HUMAN 125I-Pindolol CYPROHEPTADINE >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100699 Beta2 CLONED HUMAN 3H-CGP-12177 CYPROHEPTADINE >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 28, 2025
100700 M1 CLONED HUMAN 3H-QNB Pizotyline 67 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100701 M2 CLONED HUMAN 3H-QNB Pizotyline 34 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100702 M3 CLONED HUMAN 3H-QNB Pizotyline 29 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100703 M4 CLONED HUMAN 3H-QNB Pizotyline 130 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100704 M5 CLONED HUMAN 3H-QNB Pizotyline 6.8 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100705 I1 CLONED HUMAN 125I-Clonidine Pizotyline 121 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100706 Sigma 1 BRAIN GUINEA PIG 3H-Pentazocine(+) Pizotyline >10000 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100707 Sigma 2 PC12 RAT 3H-DTG Pizotyline 6450 Young, R., et. al., 2005 Jan 15, 2025 Jan 15, 2025
100708 MT1 C.H.O. HUMAN 2-I125 iodomelatonin N-Propargyl-2-(5-methoxy-1H-indol-3-yl)acetamide 14 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100709 MT2 C.H.O. HUMAN 2-I125 iodomelatonin N-Propargyl-2-(5-methoxy-1H-indol-3-yl)acetamide 3.8 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100710 MT1 C.H.O. HUMAN 2-I125 iodomelatonin N-Propargyl-3-(5-methoxy-1H-indol-3-yl)propanamide 5 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100711 MT2 C.H.O. HUMAN 2-I125 iodomelatonin N-Propargyl-3-(5-methoxy-1H-indol-3-yl)propanamide 1 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100712 MT1 C.H.O. HUMAN 2-I125 iodomelatonin N-Allyl-2-(5-methoxy-1H-indol-3-yl)acetamide 17 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100713 MT2 C.H.O. HUMAN 2-I125 iodomelatonin N-Allyl-2-(5-methoxy-1H-indol-3-yl)acetamide 4.9 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100714 MT1 C.H.O. HUMAN 2-I125 iodomelatonin N-Allyl-3-(5-methoxy-1H-indol-3-yl)propanamide 2.5 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100715 MT2 C.H.O. HUMAN 2-I125 iodomelatonin N-Allyl-3-(5-methoxy-1H-indol-3-yl)propanamide 0.45 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100716 MT1 C.H.O. HUMAN 2-I125 iodomelatonin 2-((5-Methoxy-1H-indol-3-yl)methyl)-5-methyloxazole 280 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100717 MT2 C.H.O. HUMAN 2-I125 iodomelatonin 2-((5-Methoxy-1H-indol-3-yl)methyl)-5-methyloxazole 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100718 MT1 C.H.O. HUMAN 2-I125 iodomelatonin 2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyloxazole 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100719 MT2 C.H.O. HUMAN 2-I125 iodomelatonin 2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyloxazole 498 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100720 MT1 C.H.O. HUMAN 2-I125 iodomelatonin 5-((5-Methoxy-1H-indol-3-yl)methyl)-3-methyl-1,2,4-oxadiazole 170 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100721 MT2 C.H.O. HUMAN 2-I125 iodomelatonin 5-((5-Methoxy-1H-indol-3-yl)methyl)-3-methyl-1,2,4-oxadiazole 44 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100722 MT1 C.H.O. HUMAN 2-I125 iodomelatonin 5-(2-(5-Methoxy-1H-indol-3-yl)-3-methyl-1,2,4-oxadiazole 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100723 MT2 C.H.O. HUMAN 2-I125 iodomelatonin 5-(2-(5-Methoxy-1H-indol-3-yl)-3-methyl-1,2,4-oxadiazole 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100724 MT1 C.H.O. HUMAN 2-I125 iodomelatonin 2-((5-Methoxy-1H-indol-3-yl)methyl)5-1,3,4-oxadiazole 210 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100725 MT2 C.H.O. HUMAN 2-I125 iodomelatonin 2-((5-Methoxy-1H-indol-3-yl)methyl)5-1,3,4-oxadiazole 16 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100726 MT1 C.H.O. HUMAN 125I-Iodomelatonin 2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyl-1,3,4-oxadiazole 709 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100727 MT2 C.H.O. HUMAN 125I-Iodomelatonin 2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyl-1,3,4-oxadiazole 190 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100728 MT1 C.H.O. HUMAN 125I-Iodomelatonin 2-(2-(5-Methoxy-1H-indol-3-yl)ehtyl)-1,3,4-oxadiazole 570 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100729 MT2 C.H.O. HUMAN 125I-Iodomelatonin 2-(2-(5-Methoxy-1H-indol-3-yl)ehtyl)-1,3,4-oxadiazole 68 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100730 MT1 C.H.O. HUMAN 125I-Iodomelatonin 5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazol-2(3H)-one 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100731 MT2 C.H.O. HUMAN 125I-Iodomelatonin 5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazol-2(3H)-one 160 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100732 MT1 C.H.O. HUMAN 125I-Iodomelatonin 5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazol-2(3H)-one 35 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100733 MT2 C.H.O. HUMAN 125I-Iodomelatonin 5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazol-2(3H)-one 4 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100734 MT1 C.H.O. HUMAN 125I-Iodomelatonin 5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazole-2(3H)-thione 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100735 MT2 C.H.O. HUMAN 125I-Iodomelatonin 5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazole-2(3H)-thione 535 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100736 MT1 C.H.O. HUMAN 125I-Iodomelatonin 5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazole-2(3H)-thione 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100737 MT2 C.H.O. HUMAN 125I-Iodomelatonin 5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazole-2(3H)-thione 530 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100738 MT1 C.H.O. HUMAN 125I-Iodomelatonin 3-((5-Methoxy-1H-indol-3-yl)methyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100739 MT2 C.H.O. HUMAN 125I-Iodomelatonin 3-((5-Methoxy-1H-indol-3-yl)methyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one 560 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100740 MT1 C.H.O. HUMAN 125I-Iodomelatonin 3-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100741 MT2 C.H.O. HUMAN 125I-Iodomelatonin 3-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100742 MT1 C.H.O. HUMAN 125I-Iodomelatonin 4-Ethyl-3-((5-methoxy-1H-indol-3-yl)methyl)1H-1,2,4-triazol-5(4H)-thione 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100743 MT2 C.H.O. HUMAN 125I-Iodomelatonin 4-Ethyl-3-((5-methoxy-1H-indol-3-yl)methyl)1H-1,2,4-triazol-5(4H)-thione 220 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100744 MT1 C.H.O. HUMAN 125I-Iodomelatonin 4-Ethyl-3-(2-(5-methoxy-1H-indol-3-yl)ethyl)-1H-1,2,4-triazol-5(4H)-thione 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100745 MT2 C.H.O. HUMAN 125I-Iodomelatonin 4-Ethyl-3-(2-(5-methoxy-1H-indol-3-yl)ethyl)-1H-1,2,4-triazol-5(4H)-thione 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100746 MT1 C.H.O. HUMAN 125I-Iodomelatonin N-Ethyl-5-((5-methoxy-1H-indol-3-yl)methyl)-1,3,4-thiadiazol-2-amine 1000 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100747 MT2 C.H.O. HUMAN 125I-Iodomelatonin N-Ethyl-5-((5-methoxy-1H-indol-3-yl)methyl)-1,3,4-thiadiazol-2-amine 17 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100748 MT1 C.H.O. HUMAN 125I-Iodomelatonin DMT,5-MeO 210 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100749 MT2 C.H.O. HUMAN 125I-Iodomelatonin DMT,5-MeO 16 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100750 MT1 C.H.O. HUMAN 125I-Iodomelatonin MELATONIN 0.091 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100751 MT2 C.H.O. HUMAN 125I-Iodomelatonin MELATONIN 0.15 Revenga, de la Fuente Mario, et. al. 2015 Jan 15, 2025 Jan 29, 2025
100752 PDE1 CLONED HUMAN Functional Roflumilast >10000 Liu S, et al., 2005 Jan 15, 2025 Jan 15, 2025