The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

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Showing 97,001-98,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
99749DORCLONEDHUMAN3H-DPDPE(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide0.8Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99750DORCLONEDHUMAN3H-DPDPE(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99751DORCLONEDHUMAN3H-DPDPE(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide1.4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99752DORCLONEDHUMAN3H-DPDPE(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl] propyl}-Nmethylpropanamide1.6Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99753DORCLONEDHUMAN3H-DPDPE(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide57Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99754KORCLONEDHUMAN3H-U69593(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide86Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99755KORCLONEDHUMAN3H-U69593(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl] propyl}-Nmethylpropanamide43Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99756KORCLONEDHUMAN3H-U69593(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide68Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99757KORCLONEDHUMAN3H-U69593(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide37Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99758KORCLONEDHUMAN3H-U69593(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide3Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99759KORCLONEDHUMAN3H-U69593(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4- chloroph enyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4- tetrahydroisoquinoline-391Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99760KORCLONEDHUMAN3H-U69593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4- chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1- yl]propyl}(methyl) amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3- carboxamide13Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99761KORCLONEDHUMAN3H-U69593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car9Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99762KORCLONEDHUMAN3H-U69593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide230Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99763Alpha1ACLONEDHUMAN125I-HEAT(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide6800Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99764Alpha1ACLONEDHUMAN125I-HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide6600Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99765Alpha1ACLONEDHUMAN125I-HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide4600Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99766Alpha1ACLONEDHUMAN125I-HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99767Alpha1ACLONEDHUMAN125I-HEAT(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99768Alpha1ACLONEDHUMAN125I-HEAT(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99769Alpha2ACLONEDHUMAN125I-Clonidine(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99770Alpha2ACLONEDHUMAN125I-Clonidine(S)-2-[(S)-2-Amino-3-(tetrahydroisoquinoline-3-carboxamide)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4->10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99771Alpha2ACLONEDHUMAN125I-Clonidine(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99772Alpha2ACLONEDHUMAN125I-Clonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide4700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99773Alpha2ACLONEDHUMAN125I-Clonidine(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99774Alpha2ACLONEDHUMAN125I-Clonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99775Alpha2CCLONEDHUMAN125I-Clonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99776Alpha2CCLONEDHUMAN125I-Clonidine(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99777Alpha2CCLONEDHUMAN125I-Clonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide240Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99778Alpha2CCLONEDHUMAN125I-Clonidine(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide280Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99779Alpha2CCLONEDHUMAN125I-Clonidine(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-ca>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99780Alpha2CCLONEDHUMAN125I-Clonidine(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99781D2CLONEDHUMAN3H-N-Methylspiperone(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99782D2CLONEDHUMAN3H-N-Methylspiperone(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99783D2CLONEDHUMAN3H-N-Methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99784D2CLONEDHUMAN3H-N-Methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide2200Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99785D2CLONEDHUMAN3H-N-Methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99786D2CLONEDHUMAN3H-N-Methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99787D3CLONEDHUMAN3H-N-Methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99788D3CLONEDHUMAN3H-N-Methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide4300Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99789D3CLONEDHUMAN3H-N-Methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide890Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99790D3CLONEDHUMAN3H-N-Methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99791D3CLONEDHUMAN3H-N-Methylspiperone(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car6700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99792D3CLONEDHUMAN3H-N-Methylspiperone(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99793NETCLONEDHUMAN3H-Nisoxetine(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99794NETCLONEDHUMAN3H-Nisoxetine(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4tetrahydroisoquinoline-3-car>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99795NETCLONEDHUMAN3H-Nisoxetine(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99796NETCLONEDHUMAN3H-Nisoxetine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99797NETCLONEDHUMAN3H-Nisoxetine(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2400Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99798NETCLONEDHUMAN3H-Nisoxetine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide750Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99799SERTCLONEDHUMAN3H-CITALOPRAM(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide280Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99800SERTCLONEDHUMAN3H-CITALOPRAM(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99801SERTCLONEDHUMAN3H-CITALOPRAM(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99802SERTCLONEDHUMAN3H-CITALOPRAM(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99803SERTCLONEDHUMAN3H-CITALOPRAM(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-ca5700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99804SERTCLONEDHUMAN3H-CITALOPRAM(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide1400Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99805Sigma 1CLONEDHUMAN3H-Pentazocine(+)(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5- cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99806Sigma 1CLONEDHUMAN3H-Pentazocine(+)(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-ca>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99807Sigma 1CLONEDHUMAN3H-Pentazocine(+)(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl} (methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide1900Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99808Sigma 1CLONEDHUMAN3H-Pentazocine(+)(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6- dimethylphenyl)propanamido]propanami do}acetamido)-3-(4-chlorophenyl)-N-{3- [(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenz ofuran-1-yl]propyl}-Nmethylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99809Sigma 1CLONEDHUMAN3H-Pentazocine(+)(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1- (4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4- fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide47Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99810Sigma 1CLONEDHUMAN3H-Pentazocine(+)(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4- hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4- fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide410Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99811MORCLONEDRAT[3H]DAMGO(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide88Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99812MORCLONEDRAT[3H]DAMGO(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide7Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99813MORCLONEDRAT[3H]DAMGO(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide16Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99814MORCLONEDRAT[3H]DAMGO(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide12Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99815MORCLONEDRAT[3H]DAMGO(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide1Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99816MORCLONEDRAT[3H]DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb35Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99817MORCLONEDRAT[3H]DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide10Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99818MORCLONEDRAT[3H]DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb7Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99819MORCLONEDRAT[3H]DAMGO(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide0.4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99820MORCLONEDRAT[3H]DAMGOYaGF-NH22.8Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99821MORCLONEDRAT[3H]DAMGODALEA7.7Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99822DORCLONEDHUMAN[3H]DPDPE(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide57Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99823DORCLONEDHUMAN[3H]DPDPE(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide1.6Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99824DORCLONEDHUMAN[3H]DPDPE(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide1.4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99825DORCLONEDHUMAN[3H]DPDPE(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99826DORCLONEDHUMAN[3H]DPDPE(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide0.8Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99827DORCLONEDHUMAN[3H]DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb20Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99828DORCLONEDHUMAN[3H]DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide0.88Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99829DORCLONEDHUMAN[3H]DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb0.91Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99830DORCLONEDHUMAN[3H]DPDPE(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide13Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99831DORCLONEDHUMAN[3H]DPDPEYaGF-NH2300Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99832DORCLONEDHUMAN[3H]DPDPEDALEA2.4Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99833KORCLONEDHUMAN[3H]U69,593(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide86Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99834KORCLONEDHUMAN[3H]U69,593(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-3-(4-chlorophenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide43Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99835KORCLONEDHUMAN[3H]U69,593(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide68Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99836KORCLONEDHUMAN[3H]U69,593(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide37Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99837KORCLONEDHUMAN[3H]U69,593(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide3Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99838KORCLONEDHUMAN[3H]U69,593(S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]-N-(2-{[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb91Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99839KORCLONEDHUMAN[3H]U69,593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-3-(4-chlorophenyl)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide13Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99840KORCLONEDHUMAN[3H]U69,593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb9Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99841KORCLONEDHUMAN[3H]U69,593(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide230Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99842Alpha1ACLONEDHUMAN[125I] HEAT(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide6800Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99843Alpha1ACLONEDHUMAN[125I] HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide6600Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99844Alpha1ACLONEDHUMAN[125I] HEAT(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide4600Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99845Alpha1ACLONEDHUMAN[125I] HEAT(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99846Alpha2ACLONEDHUMAN[125I] iodoclonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide4700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99847Alpha2CCLONEDHUMAN[125I] iodoclonidine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide240Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99848Alpha2CCLONEDHUMAN[125I] iodoclonidine(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide280Mehr-un-Nisa et al 2015Jan 15, 2025Jan 29, 2025
99849D2CLONEDHUMAN[3H]N-methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide2200Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99850D2CLONEDHUMAN[3H]N-methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99851D3CLONEDHUMAN[3H]N-methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99852D3CLONEDHUMAN[3H]N-methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide4300Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99853D3CLONEDHUMAN[3H]N-methylspiperone(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide890Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99854D3CLONEDHUMAN[3H]N-methylspiperone(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99855D3CLONEDHUMAN[3H]N-methylspiperone(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb6700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99856NETCLONEDHUMAN[3H] Nisoxetine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide750Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99857NETCLONEDHUMAN[3H] Nisoxetine(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide2400Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99858SERTCLONEDHUMAN[3H] Citalopram(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide280Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99859SERTCLONEDHUMAN[3H] Citalopram(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-(2-{[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)-1,2,3,4-tetrahydroisoquinoline-3-carb5700Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99860SERTCLONEDHUMAN[3H] Citalopram(S)-2-[(S)-2-Amino-3-(4-hydroxy-3,5-dimethylphenyl)propanoyl]-N-[(R)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide1400Mehr-un-Nisa et al 2015Jan 15, 2025Jan 28, 2025
99861Sigma 1CLONEDHUMAN[3H] pentazocine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]propanamido}acetamido)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methyl-3-phenylpropanamide410Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99862Sigma 1CLONEDHUMAN[3H] pentazocine(R)-2-[(S)-2-Amino-3-(4-hydroxyphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-fluorophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide47Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99863Sigma 1CLONEDHUMAN[3H] pentazocine(S)-2-(2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimeth-ylphenyl)propanamido]propanamido}acetamido)-3-(4-chloro-phenyl)-N-{3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}-N-methylpropanamide>10000Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
99864Sigma 1CLONEDHUMAN[3H] pentazocine(R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethylphenyl)propanamido]-N-(2-{[(S)-1-({3-[(S)-5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofuran-1-yl]propyl}(methyl)amino)-3-(4-flu-orophenyl)-1-oxopropan-2-yl]amino}-2-oxoethyl)hexanamide1900Mehr-un-Nisa et al 2015Jan 15, 2025Jan 15, 2025
998655-HT1AHIPPOCAMPUSMOUSE3H-8-OH-DPAT1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride138Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998665-HT2AHIPPOCAMPUSMOUSE3H-KETANSERIN1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride77Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998675-HT7HYPOTHALAMUSMOUSE3H-5-CT1,3-di-methyl-8-morpholin-4-yl-7-[4-(4-phenyl-pi-perazin-1-yl)-butyl]-3,7-dihydro-purine-2,6-dio-ne hydrochloride1277Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998685-HT2AHIPPOCAMPUSMOUSE3H- Ketanserin7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride205Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998695-HT1AHIPPOCAMPUSMOUSE3H-8-OH-DPAT7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride7Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998705-HT1AHIPPOCAMPUSMOUSE3H-8-OH-DPAT7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride22Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998715-HT7HYPOTHALAMUSMOUSE3H-5-CT7-{4-[4-(3-chloro-phe-nyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-mor-pholin-4-yl-3,7-dihydro-purine-2,6-dione hydro-chloride112Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998725-HT7HYPOTHALAMUSMOUSE3H-5-CT7-{4-[4-(2-metho-xy-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride335Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
998735-HT2AHIPPOCAMPUSMOUSE3H- Ketanserin(7-{4-[4-(3-chloro-phenyl)-piperazin-1-yl]-butyl}-1,3-dimethyl-8-morpholin-4-yl-3,7-dihydro-purine-2,6-dione hydrochloride)21Jastrzębska-Więsek, Magdalena, et al., 2011Jan 15, 2025Jan 15, 2025
99874B1CORTICAL MEMBRANESRat brain3H-BRADYKININABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99875ETACORTICAL MEMBRANESRat brain125I-ENDOTHELINABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99876ETBCORTICAL MEMBRANESRat brain125I-ENDOTHELINABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99877NK1CORTICAL MEMBRANESRat brain3H-Leu,4,5 Substance PABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99878CORTICAL MEMBRANESRat brain125I-NPYABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99879CORTICAL MEMBRANESRat brain3H-NeurotensinABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99880CORTICAL MEMBRANESRat brain125I-VIPABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99881CORTICAL MEMBRANESRat brain125I-Omega-ConotoxinABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99882CORTICAL MEMBRANESRat brain3H-NitrendipineABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99883CORTICAL MEMBRANESRat brain3H-TBOBABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99884CORTICAL MEMBRANESRat brain125I-ApaminABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99885CORTICAL MEMBRANESRat brain3H-GlibenclamideABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99886CORTICAL MEMBRANESRat brain3H-CharybdotoxinABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99887NETCORTICAL MEMBRANESRat brain3H-NisoxetineABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99888SLC6A4CORTICAL MEMBRANESRat brain3H-CITALOPRAMABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99889CORTICAL MEMBRANESRat brain3H-GABAABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99890CORTICAL MEMBRANESRat brain3H-Choline ChlorideABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99891SLC6A3CORTICAL MEMBRANESRat brain3H-WIN 35,428ABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99892AChECORTICAL MEMBRANESRat brainUNDEFINEDABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 28, 2025
99893MOACORTICAL MEMBRANESRat brain14C-5-HTABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 29, 2025
99894MOACORTICAL MEMBRANESRat brain14C-PhenylethylamineABT-089 >10000Sullivan, JP et al., 1997Jan 15, 2025Jan 29, 2025
99895nAChR7CLONEDHUMAN125I-Alpha-bgtNicotine2000Sullivan, JP et al., 1997Jan 15, 2025Jan 15, 2025
99896IPHEK293 cellsHUMAN3H-ILOPROSTTreprostinil32.1Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99897EP1HEK293 cellsHUMAN3H-PGE2Treprostinil212Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99898EP2HEK293 cellsHUMAN3H-PGE2Treprostinil3.6Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99899EP3HEK293 cellsHUMAN3H-PGE2Treprostinil2505Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99900EP4CHO cellsHUMAN3H-PGE2Treprostinil826Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99901DP11321N1HUMAN3H-PGD2Treprostinil4.4Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99902FPHEK293 cellsHUMAN3H-PGF2Treprostinil4680Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99903IPHEK293 cellsHUMAN3H-ILOPROSTILOPROST3.9Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99904EP1HEK293 cellsHUMAN3H-PGE2ILOPROST1.1Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99905EP2HEK293 cellsHUMAN3H-PGE2ILOPROST1172Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99906EP3HEK293 cellsHUMAN3H-PGE2ILOPROST208Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99907EP4CHO cellsHUMAN3H-PGE2ILOPROST212Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99908DP11321N1HUMAN3H-PGD2ILOPROST1016Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99909FPHEK293 cellsHUMAN3H-PGF2ILOPROST131Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99910TPHEK293 cellsHUMAN3H-SQ-29548ILOPROST3778Whittle BJ et al 2012Jan 15, 2025Jan 29, 2025
99911MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride542Erli F et al 2017Jan 15, 2025Jan 28, 2025
99912KORCLONEDHUMAN3H-U695933-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride0.49Erli F et al 2017Jan 15, 2025Jan 28, 2025
99913DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride2268Erli F et al 2017Jan 15, 2025Jan 28, 2025
99914DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride2139Erli F et al 2017Jan 15, 2025Jan 28, 2025
99915MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride537Erli F et al 2017Jan 15, 2025Jan 28, 2025
99916KORCLONEDHUMAN3H-U695933-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride0.061Erli F et al 2017Jan 15, 2025Jan 28, 2025
99917KORCLONEDHUMAN3H-U695933-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride0.71Erli F et al 2017Jan 15, 2025Jan 28, 2025
99918MORCLONEDHUMAN3H-DAMGO3-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride463Erli F et al 2017Jan 15, 2025Jan 28, 2025
99919DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Benzyl)(phenethyl)amino]ethyl]phenol Hydrochloride1862Erli F et al 2017Jan 15, 2025Jan 28, 2025
99920DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride3539Erli F et al 2017Jan 15, 2025Jan 28, 2025
99921MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride670Erli F et al 2017Jan 15, 2025Jan 28, 2025
99922KORCLONEDHUMAN3H-U695933-[2-[(Cyclobutyl)(phenethyl)amino]ethyl]phenol Hydrochloride10.3Erli F et al 2017Jan 15, 2025Jan 28, 2025
99923KORCLONEDHUMAN3H-U695933-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride2.69Erli F et al 2017Jan 15, 2025Jan 28, 2025
99924MORCLONEDHUMAN3H-DAMGO3-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride259Erli F et al 2017Jan 15, 2025Jan 28, 2025
99925DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Isoamyl)(phenethyl)amino]ethyl]phenol Hydrochloride2743Erli F et al 2017Jan 15, 2025Jan 28, 2025
99926DORCLONEDHUMAN3H-Diprenorphine3,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride3340Erli F et al 2017Jan 15, 2025Jan 28, 2025
99927MORCLONEDHUMAN3H-DAMGO3,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride230Erli F et al 2017Jan 15, 2025Jan 28, 2025
99928KORCLONEDHUMAN3H-U695933,3′-[2,2′-(Cyclobutylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride0.38Erli F et al 2017Jan 15, 2025Jan 28, 2025
99929KORCLONEDHUMAN3H-U695933,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride4.62Erli F et al 2017Jan 15, 2025Jan 28, 2025
99930MORCLONEDHUMAN3H-DAMGO3,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride631Erli F et al 2017Jan 15, 2025Jan 28, 2025
99931DORCLONEDHUMAN3H-Diprenorphine3,3′-[2,2′-(Cyclopropylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride2850Erli F et al 2017Jan 15, 2025Jan 28, 2025
99932DORCLONEDHUMAN3H-Diprenorphine3,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride738Erli F et al 2017Jan 15, 2025Jan 28, 2025
99933MORCLONEDHUMAN3H-DAMGO3,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride358Erli F et al 2017Jan 15, 2025Jan 28, 2025
99934KORCLONEDHUMAN3H-U695933,3′-[2,2′-(Allylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride19.1Erli F et al 2017Jan 15, 2025Jan 28, 2025
99935KORCLONEDHUMAN3H-U695933,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride0.14Erli F et al 2017Jan 15, 2025Jan 28, 2025
99936MORCLONEDHUMAN3H-DAMGO3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride167Erli F et al 2017Jan 15, 2025Jan 28, 2025
99937DORCLONEDHUMAN3H-Diprenorphine3,3′-[2,2′-(Cyclohexylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride1432Erli F et al 2017Jan 15, 2025Jan 28, 2025
99938DORCLONEDHUMAN3H-Diprenorphine3,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 2775Erli F et al 2017Jan 15, 2025Jan 28, 2025
99939MORCLONEDHUMAN3H-DAMGO3,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 584Erli F et al 2017Jan 15, 2025Jan 28, 2025
99940KORCLONEDHUMAN3H-U695933,3′-[2,2′-(Cyclopentylmethylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride 0.31Erli F et al 2017Jan 15, 2025Jan 28, 2025
99941KORCLONEDHUMAN3H-U695933,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride2.1Erli F et al 2017Jan 15, 2025Jan 28, 2025
99942MORCLONEDHUMAN3H-DAMGO3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride211Erli F et al 2017Jan 15, 2025Jan 28, 2025
99943DORCLONEDHUMAN3H-Diprenorphine3,3′-[2,2′-(Isoamylazanediyl)bis(ethane-2,1-diyl)]diphenol Hydrochloride1469Erli F et al 2017Jan 15, 2025Jan 28, 2025
99944DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride428Erli F et al 2017Jan 15, 2025Jan 28, 2025
99945MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride16.1Erli F et al 2017Jan 15, 2025Jan 28, 2025
99946KORCLONEDHUMAN3H-U695933-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride3.43Erli F et al 2017Jan 15, 2025Jan 28, 2025
99947KORCLONEDHUMAN3H-U695933-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride1.85Erli F et al 2017Jan 15, 2025Jan 28, 2025
99948MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride234Erli F et al 2017Jan 15, 2025Jan 28, 2025
99949DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclohexylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride1637Erli F et al 2017Jan 15, 2025Jan 28, 2025
99950DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride1099Erli F et al 2017Jan 15, 2025Jan 28, 2025
99951MORCLONEDHUMAN3H-DAMGO3-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride192Erli F et al 2017Jan 15, 2025Jan 28, 2025
99952KORCLONEDHUMAN3H-U695933-[2-[(Allyl)(2-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride43.5Erli F et al 2017Jan 15, 2025Jan 28, 2025
99953KORCLONEDHUMAN3H-U695933-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride3.56Erli F et al 2017Jan 15, 2025Jan 28, 2025
99954MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride460Erli F et al 2017Jan 15, 2025Jan 28, 2025
99955DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclopropylmethyl)(4-hydroxyphenethyl)amino]ethyl]phenol Hydrochloride>10000Erli F et al 2017Jan 15, 2025Jan 28, 2025
99956DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride>10000Erli F et al 2017Jan 15, 2025Jan 28, 2025
99957MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride398Erli F et al 2017Jan 15, 2025Jan 28, 2025
99958KORCLONEDHUMAN3H-U695933-[2-[(Cyclobutylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride0.072Erli F et al 2017Jan 15, 2025Jan 28, 2025
99959KORCLONEDHUMAN3H-U695933-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride0.04Erli F et al 2017Jan 15, 2025Jan 28, 2025
99960MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride851Erli F et al 2017Jan 15, 2025Jan 28, 2025
99961DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclohexylmethyl)(phenethyl)amino]ethyl]-2-fluorophenol Hydrochloride>10000Erli F et al 2017Jan 15, 2025Jan 28, 2025
99962DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride >10000Erli F et al 2017Jan 15, 2025Jan 28, 2025
99963MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 557Erli F et al 2017Jan 15, 2025Jan 28, 2025
99964KORCLONEDHUMAN3H-U695933-[2-[(Cyclobutylmethyl)(3-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride 0.12Erli F et al 2017Jan 15, 2025Jan 28, 2025
99965KORCLONEDHUMAN3H-U695933-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride3.37Erli F et al 2017Jan 15, 2025Jan 28, 2025
99966MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride523Erli F et al 2017Jan 15, 2025Jan 28, 2025
99967DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclobutylmethyl)(4-hydroxyphenethyl)amino]ethyl]-2-fluorophenol Hydrochloride1312Erli F et al 2017Jan 15, 2025Jan 28, 2025
99968DORCLONEDHUMAN3H-DiprenorphineN-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine2178Erli F et al 2017Jan 15, 2025Jan 28, 2025
99969MORCLONEDHUMAN3H-DAMGON-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine1065Erli F et al 2017Jan 15, 2025Jan 28, 2025
99970KORCLONEDHUMAN3H-U69593N-(Cyclobutylmethyl)-N-phenethyl-2-phenylethanamine79.1Erli F et al 2017Jan 15, 2025Jan 28, 2025
99971KORCLONEDHUMAN3H-U695933-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride5.9Erli F et al 2017Jan 15, 2025Jan 28, 2025
99972MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride826Erli F et al 2017Jan 15, 2025Jan 28, 2025
99973DORCLONEDHUMAN3H-Diprenorphine3-[2-[(Cyclopropylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride>10000Erli F et al 2017Jan 15, 2025Jan 28, 2025
99974KORCLONEDHUMAN3H-U695933-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride0.017Erli F et al 2017Jan 15, 2025Jan 28, 2025
99975MORCLONEDHUMAN3H-DAMGO3-[2-[(Cyclopentylmethyl)(phenethyl)amino]ethyl]phenol Hydrochloride826Erli F et al 2017Jan 15, 2025Jan 28, 2025
999765-HT1ACLONEDHUMAN3H-WAY1006355,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999775-HT1ACLONEDHUMAN3H-WAY1006355,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999785-HT1BCLONEDHUMAN3H-5CT5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999795-HT1BCLONEDHUMAN3H-5CT5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999805-HT1DCLONEDHUMAN3H-5CT5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999815-HT1DCLONEDHUMAN3H-5CT5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999825-HT1ECLONEDHUMAN3H-5HT5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999835-HT1ECLONEDHUMAN3H-5HT5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999845-HT2ACLONEDHUMAN125I-DOI5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999855-HT2ACLONEDHUMAN125I-DOI5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999865-HT2BCLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999875-HT2BCLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999885-HT2CCLONEDHUMAN3H-MESULERGINE5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999895-HT2CCLONEDHUMAN3H-MESULERGINE5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999905-HT3CLONEDHUMAN3H-LY 2785845,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999915-HT3CLONEDHUMAN3H-LY 2785845,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999925-HT5ACLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999935-HT5ACLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999945-HT6CLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999955-HT6CLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999965-HT7CLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
999975-HT7CLONEDHUMAN3H-LSD5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
99998Alpha1ACLONEDHUMAN125I-HEAT5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
99999Alpha1ACLONEDHUMAN125I-HEAT5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100000Alpha1BCLONEDHUMAN125I-HEAT5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100001Alpha1BCLONEDHUMAN125I-HEAT5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100002Alpha1DCLONEDHUMAN125I-HEAT5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100003Alpha1DCLONEDHUMAN125I-HEAT5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100004Alpha2ACLONEDHUMAN3H-CLONIDINE5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100005Alpha2ACLONEDHUMAN3H-CLONIDINE5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100006Alpha2BCLONEDHUMAN3H-CLONIDINE5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100007Alpha2BCLONEDHUMAN3H-CLONIDINE5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100008Alpha2CCLONEDHUMAN3H-CLONIDINE5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100009Alpha2CCLONEDHUMAN3H-CLONIDINE5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100010Beta 1CLONEDHUMAN125I-Pindolol5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100011Beta 1CLONEDHUMAN125I-Pindolol5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100012Beta 2CLONEDHUMAN3H-CGP-121775,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100013Beta 2CLONEDHUMAN3H-CGP-121775,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100014Beta3CLONEDHUMAN125I-Pindolol5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100015Beta3CLONEDHUMAN125I-Pindolol5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100016CB1CLONEDHUMAN3H-CP559405,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100017CB1CLONEDHUMAN3H-CP559405,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100018CB2CLONEDHUMAN3H-CP559405,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100019CB2CLONEDHUMAN3H-CP559405,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100020D1CLONEDHUMAN3H-SCH233905,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100021D1CLONEDHUMAN3H-SCH233905,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100022D2CLONEDHUMAN3H-NMS5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100023D2CLONEDHUMAN3H-NMS5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100024D3CLONEDHUMAN3H-NMS5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100025D3CLONEDHUMAN3H-NMS5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100026D4CLONEDHUMAN3H-NMS5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100027D4CLONEDHUMAN3H-NMS5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100028D5CLONEDHUMAN3H-SCH233905,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100029D5CLONEDHUMAN3H-SCH233905,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100030H1CLONEDHUMAN3H-PYRILAMINE5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100031H1CLONEDHUMAN3H-PYRILAMINE5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
1000325-HT1DCLONEDHUMAN125I-iodoaminopotentidine5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
1000335-HT1DCLONEDHUMAN125I-iodoaminopotentidine5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100034KORCLONEDHUMAN3H-U69,5935,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100035KORCLONEDHUMAN3H-U69,5935,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100036MORCLONEDHUMAN3H-DAMGO5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100037MORCLONEDHUMAN3H-DAMGO5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100038DORCLONEDHUMAN3H-DADLE5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100039DORCLONEDHUMAN3H-DADLE5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100040M1CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100041M1CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100042M2CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100043M2CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100044M3CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100045M3CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100046M4CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100047M4CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100048M5CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100049M5CLONEDHUMAN3H-QNB5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100050NMDACLONEDHUMAN3H-MK-8015,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100051NMDACLONEDHUMAN3H-MK-8015,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100052Sigma 1CLONEDHUMAN3H-Pentazocine(+)5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100053Sigma 1CLONEDHUMAN3H-Pentazocine(+)5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100054Sigma 2CLONEDHUMAN3H-DTG5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100055Sigma 2CLONEDHUMAN3H-DTG5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100056mGluR5BRAINRAT3H-MPEP5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100057mGluR5BRAINRAT3H-MPEP5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100058BZPBRAINRATFNZ5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 29, 2025
100059BZPBRAINRATFNZ5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 29, 2025
100060DATCLONEDHUMAN3H-WIN 35,4285,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100061DATCLONEDHUMAN3H-WIN 35,4285,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100062GABAACLONEDHUMAN3H-MUSCIMOL5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 29, 2025
100063GABAACLONEDHUMAN3H-MUSCIMOL5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 29, 2025
100064NETCLONEDHUMAN3H-Nisoxetine5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100065NETCLONEDHUMAN3H-Nisoxetine5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide245Sundaresan A et al 2015Jan 15, 2025Jan 15, 2025
100066SERTCLONEDHUMAN3H-CITALOPRAM5,6-Dimethoxy-3-methylbenzofuran-2-yl)(piperidin-1-yl) Methanone>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
100067SERTCLONEDHUMAN3H-CITALOPRAM5,6-Dimethoxy-3-methyl-N-phenylbenzofuran-2-carboxamide>10000Sundaresan A et al 2015Jan 15, 2025Jan 28, 2025
1000725-HT1ACLONEDHUMAN[3H]WAY100635Perospirone0.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1000735-HT1ACLONEDHUMAN3H-WAY100635Cariprazine1.4PDSP Certified DataJan 15, 2025Jan 15, 2025
1000745-HT1BCLONEDHUMAN3H-5-CTCariprazine926PDSP Certified DataJan 15, 2025Jan 15, 2025
1000755-HT1DCLONEDHUMAN3H-5-CTCariprazine296PDSP Certified DataJan 15, 2025Jan 15, 2025
1000765-HT2ACLONEDHUMAN3H-KETANSERINCariprazine37PDSP Certified DataJan 15, 2025Jan 15, 2025
1000775-HT2BCLONEDHUMAN3H-LSDCariprazine0.71PDSP Certified DataJan 15, 2025Jan 15, 2025
1000785-HT2CCLONEDHUMAN3H-MESULERGINECariprazine414PDSP Certified DataJan 15, 2025Jan 15, 2025
1000795-HT5ACLONEDHUMAN3H-LSDCariprazine2316PDSP Certified DataJan 15, 2025Jan 15, 2025
1000805-HT6CLONEDHUMAN3H-LSDCariprazine854PDSP Certified DataJan 15, 2025Jan 15, 2025
1000815-HT7CLONEDHUMAN3H-LSDCariprazine20PDSP Certified DataJan 15, 2025Jan 15, 2025
100082Alpha1ACLONEDHUMAN3H-PRAZOSINCariprazine379PDSP Certified DataJan 15, 2025Jan 28, 2025
100083Alpha1BCLONEDHUMAN3H-PRAZOSINCariprazine969PDSP Certified DataJan 15, 2025Jan 28, 2025
100084Alpha1DCLONEDHUMAN3H-PRAZOSINCariprazine1411PDSP Certified DataJan 15, 2025Jan 28, 2025
100085Alpha2ACLONEDHUMAN3H-RAUWOLSCINECariprazine88PDSP Certified DataJan 15, 2025Jan 28, 2025
100086Alpha2BCLONEDHUMAN3H-RAUWOLSCINECariprazine640PDSP Certified DataJan 15, 2025Jan 28, 2025
100087Alpha2CCLONEDHUMAN3H-RAUWOLSCINECariprazine1229PDSP Certified DataJan 15, 2025Jan 28, 2025
100088Beta1CLONEDHUMAN125I-PindololCariprazine325PDSP Certified DataJan 15, 2025Jan 28, 2025
100089Beta3CLONEDHUMAN125I-PindololCariprazine1882PDSP Certified DataJan 15, 2025Jan 28, 2025
100090D3CLONEDHUMAN3H-N-MethylspiperoneCariprazine2.1PDSP Certified DataJan 15, 2025Jan 28, 2025
100091D4CLONEDHUMAN3H-N-MethylspiperoneCariprazine1047PDSP Certified DataJan 15, 2025Jan 28, 2025
100092H1CLONEDHUMAN3H-PYRILAMINECariprazine10PDSP Certified DataJan 15, 2025Jan 28, 2025
1000935-HT1DCLONEDHUMAN125I-Iodo-aminopotentidineCariprazine710PDSP Certified DataJan 15, 2025Jan 28, 2025
100094M4CLONEDHUMAN3H-QNBCariprazine1356PDSP Certified DataJan 15, 2025Jan 15, 2025
100095M5CLONEDHUMAN3H-QNBCariprazine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100096SERTCLONEDHUMAN3H-CITALOPRAMCariprazine3597PDSP Certified DataJan 15, 2025Jan 28, 2025
100097Sigma 1CLONEDHUMAN3H-Pentazocine(+)Cariprazine29PDSP Certified DataJan 15, 2025Jan 28, 2025
100098Sigma 2CLONEDHUMAN3H-DTGCariprazine1531PDSP Certified DataJan 15, 2025Jan 28, 2025
100099D1CLONEDHUMAN3H-SCH23390Cariprazine3749PDSP Certified DataJan 15, 2025Jan 28, 2025
100100D2CLONEDHUMAN3H-N-MethylspiperoneCariprazine18PDSP Certified DataJan 15, 2025Jan 28, 2025
1001015-HT1ACLONEDHUMAN3H-WAY100635Quetiapine267PDSP Certified DataJan 15, 2025Jan 15, 2025
1001025-HT2ACLONEDHUMAN3H-KETANSERINQuetiapine352PDSP Certified DataJan 15, 2025Jan 15, 2025
1001035-HT2BCLONEDHUMAN3H-LSDQuetiapine86PDSP Certified DataJan 15, 2025Jan 15, 2025
1001045-HT2CCLONEDHUMAN3H-MESULERGINEQuetiapine3624PDSP Certified DataJan 15, 2025Jan 15, 2025
1001055-HT3CLONEDHUMAN3H-GR65630Quetiapine4330PDSP Certified DataJan 15, 2025Jan 15, 2025
1001065-HT5ACLONEDHUMAN3H-LSDQuetiapine2300PDSP Certified DataJan 15, 2025Jan 15, 2025
1001075-HT6CLONEDHUMAN3H-LSDQuetiapine1777PDSP Certified DataJan 15, 2025Jan 15, 2025
1001085-HT7CLONEDHUMAN3H-LSDQuetiapine168PDSP Certified DataJan 15, 2025Jan 15, 2025
100109Alpha1ACLONEDHUMAN3H-PRAZOSINQuetiapine261PDSP Certified DataJan 15, 2025Jan 28, 2025
100110Alpha1BCLONEDHUMAN3H-PRAZOSINQuetiapine141PDSP Certified DataJan 15, 2025Jan 28, 2025
100111Alpha1DCLONEDHUMAN3H-PRAZOSINQuetiapine752PDSP Certified DataJan 15, 2025Jan 28, 2025
100112Alpha2ACLONEDHUMAN3H-RAUWOLSCINEQuetiapine1207PDSP Certified DataJan 15, 2025Jan 28, 2025
100113Alpha2BCLONEDHUMAN3H-RAUWOLSCINEQuetiapine96PDSP Certified DataJan 15, 2025Jan 28, 2025
100114Alpha2CCLONEDHUMAN3H-RAUWOLSCINEQuetiapine166PDSP Certified DataJan 15, 2025Jan 28, 2025
100115D2CLONEDHUMAN3H-N-MethylspiperoneQuetiapine5037PDSP Certified DataJan 15, 2025Jan 28, 2025
100116D3CLONEDHUMAN3H-N-MethylspiperoneQuetiapine2193PDSP Certified DataJan 15, 2025Jan 28, 2025
100117D4CLONEDHUMAN3H-N-MethylspiperoneQuetiapine1651PDSP Certified DataJan 15, 2025Jan 28, 2025
100118D5CLONEDHUMAN3H-SCH23390Quetiapine2133PDSP Certified DataJan 15, 2025Jan 28, 2025
100119H1CLONEDHUMAN3H-PYRILAMINEQuetiapine9.1PDSP Certified DataJan 15, 2025Jan 28, 2025
1001205-HT1DCLONEDHUMAN125I-Iodo-aminopotentidineQuetiapine473PDSP Certified DataJan 15, 2025Jan 28, 2025
100121KORCLONEDHUMAN3H-U69593Quetiapine3489PDSP Certified DataJan 15, 2025Jan 28, 2025
100122M3CLONEDHUMAN3H-QNBQuetiapine1294PDSP Certified DataJan 15, 2025Jan 15, 2025
100123M4CLONEDHUMAN3H-QNBQuetiapine722PDSP Certified DataJan 15, 2025Jan 15, 2025
100124Sigma 1CLONEDHUMAN3H-Pentazocine(+)Quetiapine413PDSP Certified DataJan 15, 2025Jan 28, 2025
100125Sigma 2CLONEDHUMAN3H-DTGQuetiapine1566PDSP Certified DataJan 15, 2025Jan 28, 2025
100126D1CLONEDHUMAN3H-SCH23390Quetiapine381PDSP Certified DataJan 15, 2025Jan 28, 2025
1001275-HT1ACLONEDHUMAN3H-WAY100635Brexpiprazole1.1PDSP Certified DataJan 15, 2025Jan 15, 2025
1001285-HT1BCLONEDHUMAN3H-5CTBrexpiprazole365PDSP Certified DataJan 15, 2025Jan 15, 2025
1001295-HT1DCLONEDHUMAN3H-5CTBrexpiprazole23PDSP Certified DataJan 15, 2025Jan 15, 2025
1001305-HT1ECLONEDHUMAN3H-5HTBrexpiprazole>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1001315-HT2ACLONEDHUMAN3H-KETANSERINBrexpiprazole3.9PDSP Certified DataJan 15, 2025Jan 15, 2025
1001325-HT2BCLONEDHUMAN3H-LSDBrexpiprazole1.3PDSP Certified DataJan 15, 2025Jan 15, 2025
1001335-HT2CCLONEDHUMAN3H-MESULERGINEBrexpiprazole29PDSP Certified DataJan 15, 2025Jan 15, 2025
1001345-HT3CLONEDHUMAN3H-GR65630Brexpiprazole754PDSP Certified DataJan 15, 2025Jan 15, 2025
1001355-HT5ACLONEDHUMAN3H-LSDBrexpiprazole614PDSP Certified DataJan 15, 2025Jan 15, 2025
1001365-HT6CLONEDHUMAN3H-LSDBrexpiprazole117PDSP Certified DataJan 15, 2025Jan 15, 2025
1001375-HT7CLONEDHUMAN3H-LSDBrexpiprazole6.6PDSP Certified DataJan 15, 2025Jan 15, 2025
100138Alpha1ACLONEDHUMAN3H-PRAZOSINBrexpiprazole24PDSP Certified DataJan 15, 2025Jan 28, 2025
100139Alpha1BCLONEDHUMAN3H-PRAZOSINBrexpiprazole134PDSP Certified DataJan 15, 2025Jan 28, 2025
100140Alpha1DCLONEDHUMAN3H-PRAZOSINBrexpiprazole58PDSP Certified DataJan 15, 2025Jan 28, 2025
100141Alpha2ACLONEDHUMAN3H-RAUWOLSCINEBrexpiprazole39PDSP Certified DataJan 15, 2025Jan 28, 2025
100142Alpha2BCLONEDHUMAN3H-RAUWOLSCINEBrexpiprazole135PDSP Certified DataJan 15, 2025Jan 28, 2025
100143Alpha2CCLONEDHUMAN3H-RAUWOLSCINEBrexpiprazole24PDSP Certified DataJan 15, 2025Jan 28, 2025
100144Beta1CLONEDHUMAN125I-PindololBrexpiprazole699PDSP Certified DataJan 15, 2025Jan 28, 2025
100145Beta2CLONEDHUMAN3H-CGP12177Brexpiprazole>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
100146Beta3CLONEDHUMAN125I-PindololBrexpiprazole1653PDSP Certified DataJan 15, 2025Jan 28, 2025
100147D2CLONEDHUMAN3H-N-MethylspiperoneBrexpiprazole40PDSP Certified DataJan 15, 2025Jan 28, 2025
100148D3CLONEDHUMAN3H-N-MethylspiperoneBrexpiprazole30PDSP Certified DataJan 15, 2025Jan 28, 2025
100149D4CLONEDHUMAN3H-N-MethylspiperoneBrexpiprazole19PDSP Certified DataJan 15, 2025Jan 28, 2025
100150D5CLONEDHUMAN3H-SCH23390Brexpiprazole465PDSP Certified DataJan 15, 2025Jan 28, 2025
100151DATCLONEDHUMAN3H-WIN35428Brexpiprazole1799PDSP Certified DataJan 15, 2025Jan 15, 2025
100152H1CLONEDHUMAN3H-PYRILAMINEBrexpiprazole6.8PDSP Certified DataJan 15, 2025Jan 28, 2025
1001535-HT1DCLONEDHUMAN125I-Iodo-aminopotentidineBrexpiprazole365PDSP Certified DataJan 15, 2025Jan 28, 2025
100154NETCLONEDHUMAN3H-NisoxetineBrexpiprazole>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100155SERTCLONEDHUMAN3H-CITALOPRAMBrexpiprazole247PDSP Certified DataJan 15, 2025Jan 28, 2025
100156Sigma 1CLONEDHUMAN3H-Pentazocine(+)Brexpiprazole287PDSP Certified DataJan 15, 2025Jan 28, 2025
100157Sigma 2CLONEDHUMAN3H-DTGBrexpiprazole40PDSP Certified DataJan 15, 2025Jan 28, 2025
100158D1CLONEDHUMAN3H-SCH23390Brexpiprazole>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
1001595-HT1ACLONEDHUMAN3H-WAY100635Amisulpride3546PDSP Certified DataJan 15, 2025Jan 15, 2025
1001605-HT2ACLONEDHUMAN3H-KETANSERINAmisulpride746PDSP Certified DataJan 15, 2025Jan 15, 2025
1001615-HT2BCLONEDHUMAN3H-LSDAmisulpride74PDSP Certified DataJan 15, 2025Jan 15, 2025
1001625-HT6CLONEDHUMAN3H-LSDAmisulpride1356PDSP Certified DataJan 15, 2025Jan 15, 2025
1001635-HT7CLONEDHUMAN3H-LSDAmisulpride35PDSP Certified DataJan 15, 2025Jan 15, 2025
100164Alpha2ACLONEDHUMAN3H-RAUWOLSCINEAmisulpride101PDSP Certified DataJan 15, 2025Jan 28, 2025
100165Alpha2BCLONEDHUMAN3H-RAUWOLSCINEAmisulpride465PDSP Certified DataJan 15, 2025Jan 28, 2025
100166Alpha2CCLONEDHUMAN3H-RAUWOLSCINEAmisulpride992PDSP Certified DataJan 15, 2025Jan 28, 2025
100167D2CLONEDHUMAN3H-N-MethylspiperoneAmisulpride2407PDSP Certified DataJan 15, 2025Jan 28, 2025
100168D4CLONEDHUMAN3H-N-MethylspiperoneAmisulpride1591PDSP Certified DataJan 15, 2025Jan 28, 2025
100169D3CLONEDHUMAN3H-N-MethylspiperoneAmisulpride17PDSP Certified DataJan 15, 2025Jan 28, 2025
100170Sigma 1CLONEDHUMAN3H-Pentazocine(+)Amisulpride3709PDSP Certified DataJan 15, 2025Jan 28, 2025
1001715-HT1ACLONEDHUMAN3H-WAY100635Perospirone0.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1001725-HT1ACLONEDHUMAN3H-WAY100635Ziprasidone1.5PDSP Certified DataJan 15, 2025Jan 15, 2025
1001735-HT1ACLONEDHUMAN3H-WAY100635Asenapine4.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1001745-HT1ACLONEDHUMAN3H-WAY100635NEMONAPRIDE5.8PDSP Certified DataJan 15, 2025Jan 15, 2025
1001755-HT1ACLONEDHUMAN3H-WAY100635ARIPIPRAZOLE13PDSP Certified DataJan 15, 2025Jan 15, 2025
1001765-HT1ACLONEDHUMAN3H-WAY100635ILOPERIDONE27PDSP Certified DataJan 15, 2025Jan 15, 2025
1001775-HT1ACLONEDHUMAN3H-WAY100635Lurasidone HCl53PDSP Certified DataJan 15, 2025Jan 15, 2025
1001785-HT1ACLONEDHUMAN3H-WAY100635CLOZAPINE104PDSP Certified DataJan 15, 2025Jan 15, 2025
1001795-HT1ACLONEDHUMAN3H-WAY100635ZOTEPINE131PDSP Certified DataJan 15, 2025Jan 15, 2025
1001805-HT1ACLONEDHUMAN3H-WAY100635RISPERIDONE158PDSP Certified DataJan 15, 2025Jan 15, 2025
1001815-HT1ACLONEDHUMAN3H-WAY100635SERTINDOLE236PDSP Certified DataJan 15, 2025Jan 15, 2025
1001825-HT1ACLONEDHUMAN3H-WAY100635Paliperidone404PDSP Certified DataJan 15, 2025Jan 15, 2025
1001835-HT1ACLONEDHUMAN3H-WAY100635OLANZAPINE1114PDSP Certified DataJan 15, 2025Jan 15, 2025
1001845-HT1ACLONEDHUMAN3H-WAY100635Blonanserin1215PDSP Certified DataJan 15, 2025Jan 15, 2025
1001855-HT1ACLONEDHUMAN3H-WAY100635Melperone HCl1328PDSP Certified DataJan 15, 2025Jan 15, 2025
1001865-HT1ACLONEDHUMAN3H-WAY100635Remoxapride2989PDSP Certified DataJan 15, 2025Jan 15, 2025
1001875-HT1ACLONEDHUMAN3H-WAY100635RS-(+/-)-Sulpriride7610PDSP Certified DataJan 15, 2025Jan 15, 2025
1001885-HT1BCLONEDHUMAN3H-5CTAsenapine55PDSP Certified DataJan 15, 2025Jan 15, 2025
1001895-HT1BCLONEDHUMAN3H-5CTZiprasidone58PDSP Certified DataJan 15, 2025Jan 15, 2025
1001905-HT1BCLONEDHUMAN3H-5CTILOPERIDONE99PDSP Certified DataJan 15, 2025Jan 15, 2025
1001915-HT1BCLONEDHUMAN3H-5CTZOTEPINE431PDSP Certified DataJan 15, 2025Jan 15, 2025
1001925-HT1BCLONEDHUMAN3H-5CTSERTINDOLE501PDSP Certified DataJan 15, 2025Jan 15, 2025
1001935-HT1BCLONEDHUMAN3H-5CTRISPERIDONE718PDSP Certified DataJan 15, 2025Jan 15, 2025
1001945-HT1BCLONEDHUMAN3H-5CTPaliperidone876PDSP Certified DataJan 15, 2025Jan 15, 2025
1001955-HT1BCLONEDHUMAN3H-5CTPerospirone1070PDSP Certified DataJan 15, 2025Jan 15, 2025
1001965-HT1BCLONEDHUMAN3H-5CTLurasidone HCl1675PDSP Certified DataJan 15, 2025Jan 15, 2025
1001975-HT1BCLONEDHUMAN3H-5CTCLOZAPINE2111PDSP Certified DataJan 15, 2025Jan 15, 2025
1001985-HT1BCLONEDHUMAN3H-5CTNEMONAPRIDE2812PDSP Certified DataJan 15, 2025Jan 15, 2025
1001995-HT1BCLONEDHUMAN3H-5CTOLANZAPINE3157PDSP Certified DataJan 15, 2025Jan 15, 2025
1002005-HT1BCLONEDHUMAN3H-5CTARIPIPRAZOLE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002015-HT1BCLONEDHUMAN3H-5CTBlonanserin>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002025-HT1DCLONEDHUMAN3H-5CTZiprasidone1.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1002035-HT1DCLONEDHUMAN3H-5CTAsenapine6.3PDSP Certified DataJan 15, 2025Jan 15, 2025
1002045-HT1DCLONEDHUMAN3H-5CTRISPERIDONE6.9PDSP Certified DataJan 15, 2025Jan 15, 2025
1002055-HT1DCLONEDHUMAN3H-5CTILOPERIDONE10PDSP Certified DataJan 15, 2025Jan 15, 2025
1002065-HT1DCLONEDHUMAN3H-5CTSERTINDOLE16PDSP Certified DataJan 15, 2025Jan 15, 2025
1002075-HT1DCLONEDHUMAN3H-5CTPaliperidone19PDSP Certified DataJan 15, 2025Jan 15, 2025
1002085-HT1DCLONEDHUMAN3H-5CTPerospirone20PDSP Certified DataJan 15, 2025Jan 15, 2025
1002095-HT1DCLONEDHUMAN3H-5CTZOTEPINE48PDSP Certified DataJan 15, 2025Jan 15, 2025
1002105-HT1DCLONEDHUMAN3H-5CTLurasidone HCl50PDSP Certified DataJan 15, 2025Jan 15, 2025
1002115-HT1DCLONEDHUMAN3H-5CTARIPIPRAZOLE176PDSP Certified DataJan 15, 2025Jan 15, 2025
1002125-HT1DCLONEDHUMAN3H-5CTNEMONAPRIDE295PDSP Certified DataJan 15, 2025Jan 15, 2025
1002135-HT1DCLONEDHUMAN3H-5CTCLOZAPINE474PDSP Certified DataJan 15, 2025Jan 15, 2025
1002145-HT1DCLONEDHUMAN3H-5CTBlonanserin1061PDSP Certified DataJan 15, 2025Jan 15, 2025
1002155-HT1DCLONEDHUMAN3H-5CTOLANZAPINE1062PDSP Certified DataJan 15, 2025Jan 15, 2025
1002165-HT1DCLONEDHUMAN3H-5CTMelperone HCl>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100217Alpha2ACLONEDHUMAN3H-RAUWOLSCINEBlonanserin1.6PDSP Certified DataJan 15, 2025Jan 28, 2025
100218Alpha2ACLONEDHUMAN3H-RAUWOLSCINEILOPERIDONE8.3PDSP Certified DataJan 15, 2025Jan 28, 2025
100219Alpha2ACLONEDHUMAN3H-RAUWOLSCINERISPERIDONE12PDSP Certified DataJan 15, 2025Jan 28, 2025
100220Alpha2ACLONEDHUMAN3H-RAUWOLSCINELurasidone HCl62PDSP Certified DataJan 15, 2025Jan 28, 2025
100221Alpha2ACLONEDHUMAN3H-RAUWOLSCINEMelperone HCl103PDSP Certified DataJan 15, 2025Jan 28, 2025
100222Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPerospirone108PDSP Certified DataJan 15, 2025Jan 28, 2025
100223Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPerospirone119PDSP Certified DataJan 15, 2025Jan 28, 2025
100224Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPerospirone123PDSP Certified DataJan 15, 2025Jan 28, 2025
100225Alpha2ACLONEDHUMAN3H-RAUWOLSCINEZOTEPINE156PDSP Certified DataJan 15, 2025Jan 28, 2025
100226Alpha2ACLONEDHUMAN3H-RAUWOLSCINEZiprasidone162PDSP Certified DataJan 15, 2025Jan 28, 2025
100227Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPerospirone183PDSP Certified DataJan 15, 2025Jan 28, 2025
100228Alpha2ACLONEDHUMAN3H-RAUWOLSCINEARIPIPRAZOLE190PDSP Certified DataJan 15, 2025Jan 28, 2025
100229Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPaliperidone222PDSP Certified DataJan 15, 2025Jan 28, 2025
100230Alpha2ACLONEDHUMAN3H-RAUWOLSCINECLOZAPINE306PDSP Certified DataJan 15, 2025Jan 28, 2025
100231Alpha2ACLONEDHUMAN3H-RAUWOLSCINERS-(+/-)-Sulpriride352PDSP Certified DataJan 15, 2025Jan 28, 2025
100232Alpha2ACLONEDHUMAN3H-RAUWOLSCINESERTINDOLE353PDSP Certified DataJan 15, 2025Jan 28, 2025
100233Alpha2ACLONEDHUMAN3H-RAUWOLSCINEOLANZAPINE472PDSP Certified DataJan 15, 2025Jan 28, 2025
100234Alpha2ACLONEDHUMAN3H-RAUWOLSCINENEMONAPRIDE1027PDSP Certified DataJan 15, 2025Jan 28, 2025
100235Alpha2ACLONEDHUMAN3H-RAUWOLSCINEAsenapine1624PDSP Certified DataJan 15, 2025Jan 28, 2025
100236Alpha2ACLONEDHUMAN3H-RAUWOLSCINEGMC 1-1162652PDSP Certified DataJan 15, 2025Jan 28, 2025
100237Alpha2ACLONEDHUMAN3H-RAUWOLSCINEGMC 1-1163899PDSP Certified DataJan 15, 2025Jan 28, 2025
1002385-HT1ECLONEDHUMAN3H-5HTAsenapine71PDSP Certified DataJan 15, 2025Jan 15, 2025
1002395-HT1ECLONEDHUMAN3H-5HTGMC 1-116324.94PDSP Certified DataJan 15, 2025Jan 15, 2025
1002405-HT1ECLONEDHUMAN3H-5HTSERTINDOLE7451PDSP Certified DataJan 15, 2025Jan 15, 2025
1002415-HT1ECLONEDHUMAN3H-5HTSERTINDOLE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002425-HT1ECLONEDHUMAN3H-5HTARIPIPRAZOLE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002435-HT1ECLONEDHUMAN3H-5HTCLOZAPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002445-HT1ECLONEDHUMAN3H-5HTSERTINDOLE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002455-HT1ECLONEDHUMAN3H-5HTZOTEPINE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
1002465-HT2ACLONEDHUMAN3H-KETANSERINAsenapine0.16PDSP Certified DataJan 15, 2025Jan 15, 2025
1002475-HT2ACLONEDHUMAN3H-KETANSERINZiprasidone0.31PDSP Certified DataJan 15, 2025Jan 15, 2025
1002485-HT2ACLONEDHUMAN3H-KETANSERINPerospirone0.44PDSP Certified DataJan 15, 2025Jan 15, 2025
1002495-HT2ACLONEDHUMAN3H-KETANSERINSERTINDOLE0.48PDSP Certified DataJan 15, 2025Jan 15, 2025
1002505-HT2ACLONEDHUMAN3H-KETANSERINRISPERIDONE0.64PDSP Certified DataJan 15, 2025Jan 15, 2025
1002515-HT2ACLONEDHUMAN3H-KETANSERINZOTEPINE0.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1002525-HT2ACLONEDHUMAN3H-KETANSERINILOPERIDONE0.8PDSP Certified DataJan 15, 2025Jan 15, 2025
1002535-HT2ACLONEDHUMAN3H-KETANSERINPaliperidone0.91PDSP Certified DataJan 15, 2025Jan 15, 2025
1002545-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE9.2PDSP Certified DataJan 15, 2025Jan 15, 2025
1002555-HT2ACLONEDHUMAN3H-KETANSERINCLOZAPINE13PDSP Certified DataJan 15, 2025Jan 15, 2025
1002565-HT2ACLONEDHUMAN3H-KETANSERINARIPIPRAZOLE15PDSP Certified DataJan 15, 2025Jan 15, 2025
1002575-HT2ACLONEDHUMAN3H-KETANSERINLurasidone HCl36PDSP Certified DataJan 15, 2025Jan 15, 2025
1002585-HT2ACLONEDHUMAN3H-KETANSERINBlonanserin41PDSP Certified DataJan 15, 2025Jan 15, 2025
1002595-HT2ACLONEDHUMAN3H-KETANSERINNEMONAPRIDE56PDSP Certified DataJan 15, 2025Jan 15, 2025
1002605-HT2ACLONEDHUMAN3H-KETANSERINMelperone HCl360PDSP Certified DataJan 15, 2025Jan 15, 2025
1002615-HT2ACLONEDHUMAN3H-KETANSERINRemoxapride6390PDSP Certified DataJan 15, 2025Jan 15, 2025
1002625-HT2BCLONEDHUMAN3H-LSDAsenapine0.21PDSP Certified DataJan 15, 2025Jan 15, 2025
1002635-HT2BCLONEDHUMAN3H-LSDZOTEPINE1.2PDSP Certified DataJan 15, 2025Jan 15, 2025
1002645-HT2BCLONEDHUMAN3H-LSDSERTINDOLE1.4PDSP Certified DataJan 15, 2025Jan 15, 2025
1002655-HT2BCLONEDHUMAN3H-LSDPerospirone2.9PDSP Certified DataJan 15, 2025Jan 15, 2025
1002665-HT2BCLONEDHUMAN3H-LSDARIPIPRAZOLE3.5PDSP Certified DataJan 15, 2025Jan 15, 2025
1002675-HT2BCLONEDHUMAN3H-LSDCLOZAPINE4PDSP Certified DataJan 15, 2025Jan 15, 2025
1002685-HT2BCLONEDHUMAN3H-LSDZiprasidone4.4PDSP Certified DataJan 15, 2025Jan 15, 2025
1002695-HT2BCLONEDHUMAN3H-LSDNEMONAPRIDE6.1PDSP Certified DataJan 15, 2025Jan 15, 2025
1002705-HT2BCLONEDHUMAN3H-LSDOLANZAPINE7.2PDSP Certified DataJan 15, 2025Jan 15, 2025
1002715-HT2BCLONEDHUMAN3H-LSDRISPERIDONE16PDSP Certified DataJan 15, 2025Jan 15, 2025
1002725-HT2BCLONEDHUMAN3H-LSDPaliperidone18PDSP Certified DataJan 15, 2025Jan 15, 2025
1002735-HT2BCLONEDHUMAN3H-LSDBlonanserin20PDSP Certified DataJan 15, 2025Jan 15, 2025
1002745-HT2BCLONEDHUMAN3H-LSDLurasidone HCl24PDSP Certified DataJan 15, 2025Jan 15, 2025
1002755-HT2BCLONEDHUMAN3H-LSDILOPERIDONE27PDSP Certified DataJan 15, 2025Jan 15, 2025
1002765-HT2BCLONEDHUMAN3H-LSDGMC 1-116148PDSP Certified DataJan 15, 2025Jan 15, 2025
1002775-HT2BCLONEDHUMAN3H-LSDRemoxapride194PDSP Certified DataJan 15, 2025Jan 15, 2025
1002785-HT2BCLONEDHUMAN3H-LSDS-(-)-Sulpride1976PDSP Certified DataJan 15, 2025Jan 15, 2025
1002795-HT2BCLONEDHUMAN3H-LSDMelperone HCl2264PDSP Certified DataJan 15, 2025Jan 15, 2025
1002805-HT2CCLONEDHUMAN3H-MESULERGINEAsenapine0.24PDSP Certified DataJan 15, 2025Jan 15, 2025
1002815-HT2CCLONEDHUMAN3H-MESULERGINESERTINDOLE1.6PDSP Certified DataJan 15, 2025Jan 15, 2025
1002825-HT2CCLONEDHUMAN3H-MESULERGINEZOTEPINE3.3PDSP Certified DataJan 15, 2025Jan 15, 2025
1002835-HT2CCLONEDHUMAN3H-MESULERGINEZiprasidone4PDSP Certified DataJan 15, 2025Jan 15, 2025
1002845-HT2CCLONEDHUMAN3H-MESULERGINEPerospirone5.2PDSP Certified DataJan 15, 2025Jan 15, 2025
1002855-HT2CCLONEDHUMAN3H-MESULERGINEOLANZAPINE16PDSP Certified DataJan 15, 2025Jan 15, 2025
1002865-HT2CCLONEDHUMAN3H-MESULERGINECLOZAPINE19PDSP Certified DataJan 15, 2025Jan 15, 2025
1002875-HT2CCLONEDHUMAN3H-MESULERGINERISPERIDONE24PDSP Certified DataJan 15, 2025Jan 15, 2025
1002885-HT2CCLONEDHUMAN3H-MESULERGINEPaliperidone38PDSP Certified DataJan 15, 2025Jan 15, 2025
1002895-HT2CCLONEDHUMAN3H-MESULERGINEILOPERIDONE46PDSP Certified DataJan 15, 2025Jan 15, 2025
1002905-HT2CCLONEDHUMAN3H-MESULERGINEARIPIPRAZOLE62PDSP Certified DataJan 15, 2025Jan 15, 2025
1002915-HT2CCLONEDHUMAN3H-MESULERGINEARIPIPRAZOLE86PDSP Certified DataJan 15, 2025Jan 15, 2025
1002925-HT2CCLONEDHUMAN3H-MESULERGINEBlonanserin251PDSP Certified DataJan 15, 2025Jan 15, 2025
1002935-HT2CCLONEDHUMAN3H-MESULERGINELurasidone HCl481PDSP Certified DataJan 15, 2025Jan 15, 2025
1002945-HT2CCLONEDHUMAN3H-MESULERGINENEMONAPRIDE481PDSP Certified DataJan 15, 2025Jan 15, 2025
1002955-HT2CCLONEDHUMAN3H-MESULERGINEGMC 1-116615PDSP Certified DataJan 15, 2025Jan 15, 2025
1002965-HT2CCLONEDHUMAN3H-MESULERGINERemoxapride3574PDSP Certified DataJan 15, 2025Jan 15, 2025
1002975-HT3CLONEDHUMAN3H-GR65630CLOZAPINE47PDSP Certified DataJan 15, 2025Jan 15, 2025
1002985-HT3CLONEDHUMAN3H-GR65630ARIPIPRAZOLE106PDSP Certified DataJan 15, 2025Jan 15, 2025
1002995-HT3CLONEDHUMAN3H-GR65630OLANZAPINE125PDSP Certified DataJan 15, 2025Jan 15, 2025
1003005-HT3CLONEDHUMAN3H-GR65630ZOTEPINE140PDSP Certified DataJan 15, 2025Jan 15, 2025
1003015-HT3CLONEDHUMAN3H-GR65630Asenapine336PDSP Certified DataJan 15, 2025Jan 15, 2025
1003025-HT3CLONEDHUMAN3H-GR65630NEMONAPRIDE410PDSP Certified DataJan 15, 2025Jan 15, 2025
1003035-HT3CLONEDHUMAN3H-GR65630SERTINDOLE2237PDSP Certified DataJan 15, 2025Jan 15, 2025
1003045-HT3CLONEDHUMAN3H-GR65630Ziprasidone3385PDSP Certified DataJan 15, 2025Jan 15, 2025
1003055-HT3CLONEDHUMAN3H-GR65630ILOPERIDONE3524PDSP Certified DataJan 15, 2025Jan 15, 2025
1003065-HT3CLONEDHUMAN3H-GR65630Lurasidone HCl5264PDSP Certified DataJan 15, 2025Jan 15, 2025
1003075-HT5ACLONEDHUMAN3H-LSDZOTEPINE134PDSP Certified DataJan 15, 2025Jan 15, 2025
1003085-HT5ACLONEDHUMAN3H-LSDRISPERIDONE195PDSP Certified DataJan 15, 2025Jan 15, 2025
1003095-HT5ACLONEDHUMAN3H-LSDARIPIPRAZOLE228PDSP Certified DataJan 15, 2025Jan 15, 2025
1003105-HT5ACLONEDHUMAN3H-LSDZiprasidone301PDSP Certified DataJan 15, 2025Jan 15, 2025
1003115-HT5ACLONEDHUMAN3H-LSDPerospirone321PDSP Certified DataJan 15, 2025Jan 15, 2025
1003125-HT5ACLONEDHUMAN3H-LSDILOPERIDONE394PDSP Certified DataJan 15, 2025Jan 15, 2025
1003135-HT5ACLONEDHUMAN3H-LSDAsenapine403PDSP Certified DataJan 15, 2025Jan 15, 2025
1003145-HT5ACLONEDHUMAN3H-LSDPaliperidone428PDSP Certified DataJan 15, 2025Jan 15, 2025
1003155-HT5ACLONEDHUMAN3H-LSDSERTINDOLE510PDSP Certified DataJan 15, 2025Jan 15, 2025
1003165-HT5ACLONEDHUMAN3H-LSDAsenapine540PDSP Certified DataJan 15, 2025Jan 15, 2025
1003175-HT5ACLONEDHUMAN3H-LSDILOPERIDONE550PDSP Certified DataJan 15, 2025Jan 15, 2025
1003185-HT5ACLONEDHUMAN3H-LSDBlonanserin1037PDSP Certified DataJan 15, 2025Jan 15, 2025
1003195-HT5ACLONEDHUMAN3H-LSDLurasidone HCl1198PDSP Certified DataJan 15, 2025Jan 15, 2025
1003205-HT5ACLONEDHUMAN3H-LSDGMC 1-1161357PDSP Certified DataJan 15, 2025Jan 15, 2025
1003215-HT5ACLONEDHUMAN3H-LSDOLANZAPINE1365PDSP Certified DataJan 15, 2025Jan 15, 2025
1003225-HT5ACLONEDHUMAN3H-LSDNEMONAPRIDE1538PDSP Certified DataJan 15, 2025Jan 15, 2025
1003235-HT5ACLONEDHUMAN3H-LSDGMC 1-1161856PDSP Certified DataJan 15, 2025Jan 15, 2025
1003245-HT6CLONEDHUMAN3H-LSDAsenapine0.62PDSP Certified DataJan 15, 2025Jan 15, 2025
1003255-HT6CLONEDHUMAN3H-LSDSERTINDOLE2.3PDSP Certified DataJan 15, 2025Jan 15, 2025
1003265-HT6CLONEDHUMAN3H-LSDZOTEPINE7.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1003275-HT6CLONEDHUMAN3H-LSDOLANZAPINE13PDSP Certified DataJan 15, 2025Jan 15, 2025
1003285-HT6CLONEDHUMAN3H-LSDCLOZAPINE14PDSP Certified DataJan 15, 2025Jan 15, 2025
1003295-HT6CLONEDHUMAN3H-LSDNEMONAPRIDE46PDSP Certified DataJan 15, 2025Jan 15, 2025
1003305-HT6CLONEDHUMAN3H-LSDZiprasidone51PDSP Certified DataJan 15, 2025Jan 15, 2025
1003315-HT6CLONEDHUMAN3H-LSDILOPERIDONE140.02PDSP Certified DataJan 15, 2025Jan 15, 2025
1003325-HT6CLONEDHUMAN3H-LSDARIPIPRAZOLE162PDSP Certified DataJan 15, 2025Jan 15, 2025
1003335-HT6CLONEDHUMAN3H-LSDILOPERIDONE183.19PDSP Certified DataJan 15, 2025Jan 15, 2025
1003345-HT6CLONEDHUMAN3H-LSDBlonanserin206PDSP Certified DataJan 15, 2025Jan 15, 2025
1003355-HT6CLONEDHUMAN3H-LSDPerospirone477PDSP Certified DataJan 15, 2025Jan 15, 2025
1003365-HT6CLONEDHUMAN3H-LSDGMC 1-116630.52PDSP Certified DataJan 15, 2025Jan 15, 2025
1003375-HT6CLONEDHUMAN3H-LSDPaliperidone681PDSP Certified DataJan 15, 2025Jan 15, 2025
1003385-HT6CLONEDHUMAN3H-LSDGMC 1-116781.27PDSP Certified DataJan 15, 2025Jan 15, 2025
1003395-HT6CLONEDHUMAN3H-LSDLurasidone HCl943PDSP Certified DataJan 15, 2025Jan 15, 2025
1003405-HT6CLONEDHUMAN3H-LSDRISPERIDONE962PDSP Certified DataJan 15, 2025Jan 15, 2025
1003415-HT6CLONEDHUMAN3H-LSDMelperone HCl1635PDSP Certified DataJan 15, 2025Jan 15, 2025
1003425-HT7CLONEDHUMAN3H-LSDAsenapine0.33PDSP Certified DataJan 15, 2025Jan 15, 2025
1003435-HT7CLONEDHUMAN3H-LSDPaliperidone2.8PDSP Certified DataJan 15, 2025Jan 15, 2025
1003445-HT7CLONEDHUMAN3H-LSDRISPERIDONE3.5PDSP Certified DataJan 15, 2025Jan 15, 2025
1003455-HT7CLONEDHUMAN3H-LSDPerospirone3.8PDSP Certified DataJan 15, 2025Jan 15, 2025
1003465-HT7CLONEDHUMAN3H-LSDZiprasidone4.7PDSP Certified DataJan 15, 2025Jan 15, 2025
1003475-HT7CLONEDHUMAN3H-LSDILOPERIDONE7.8PDSP Certified DataJan 15, 2025Jan 15, 2025
1003485-HT7CLONEDHUMAN3H-LSDZOTEPINE9.5PDSP Certified DataJan 15, 2025Jan 15, 2025
1003495-HT7CLONEDHUMAN3H-LSDCLOZAPINE21PDSP Certified DataJan 15, 2025Jan 15, 2025
1003505-HT7CLONEDHUMAN3H-LSDSERTINDOLE30PDSP Certified DataJan 15, 2025Jan 15, 2025
1003515-HT7CLONEDHUMAN3H-LSDLurasidone HCl32PDSP Certified DataJan 15, 2025Jan 15, 2025
1003525-HT7CLONEDHUMAN3H-LSDARIPIPRAZOLE38PDSP Certified DataJan 15, 2025Jan 15, 2025
1003535-HT7CLONEDHUMAN3H-LSDNEMONAPRIDE81PDSP Certified DataJan 15, 2025Jan 15, 2025
1003545-HT7CLONEDHUMAN3H-LSDOLANZAPINE157PDSP Certified DataJan 15, 2025Jan 15, 2025
1003555-HT7CLONEDHUMAN3H-LSDGMC 1-116200PDSP Certified DataJan 15, 2025Jan 15, 2025
1003565-HT7CLONEDHUMAN3H-LSDMelperone HCl346PDSP Certified DataJan 15, 2025Jan 15, 2025
1003575-HT7CLONEDHUMAN3H-LSDBlonanserin1010PDSP Certified DataJan 15, 2025Jan 15, 2025
1003585-HT7CLONEDHUMAN3H-LSDRS-(+/-)-Sulpriride1085PDSP Certified DataJan 15, 2025Jan 15, 2025
100359DATCLONEDHUMAN3H-WIN 35,428Cariprazine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100360NETCLONEDHUMAN3H-NisoxeneCariprazine>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100361Alpha2CCLONEDHUMAN3H-RAUWOLSCINEILOPERIDONE5.6PDSP Certified DataJan 15, 2025Jan 28, 2025
100362DATCLONEDHUMAN3H-WIN35428ILOPERIDONE>10000PDSP Certified DataJan 15, 2025Jan 15, 2025
100363NETCLONEDHUMAN3H-NisoxetineILOPERIDONE535PDSP Certified DataJan 15, 2025Jan 15, 2025
100364SERTCLONEDHUMAN3H-CITALOPRAMILOPERIDONE443PDSP Certified DataJan 15, 2025Jan 28, 2025
100365Alpha1ACLONEDHUMAN3H-PRAZOSINILOPERIDONE1.4PDSP Certified DataJan 15, 2025Jan 28, 2025
100366Alpha1BCLONEDHUMAN3H-PRAZOSINILOPERIDONE224PDSP Certified DataJan 15, 2025Jan 28, 2025
100367Alpha1DCLONEDHUMAN3H-PRAZOSINILOPERIDONE1.2PDSP Certified DataJan 15, 2025Jan 28, 2025
100368Alpha2BCLONEDHUMAN3H-RAUWOLSCINEILOPERIDONE11PDSP Certified DataJan 15, 2025Jan 28, 2025
100369Beta1CLONEDHUMAN125I-PindololILOPERIDONE>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
100370D2CLONEDHUMAN3H-N-MethylspiperoneILOPERIDONE369PDSP Certified DataJan 15, 2025Jan 28, 2025
100371D3CLONEDHUMAN3H-N-MethylspiperoneILOPERIDONE84PDSP Certified DataJan 15, 2025Jan 28, 2025
100372D4CLONEDHUMAN3H-N-MethylspiperoneILOPERIDONE33PDSP Certified DataJan 15, 2025Jan 28, 2025
100373D5CLONEDHUMAN3H-SCH23390ILOPERIDONE173PDSP Certified DataJan 15, 2025Jan 28, 2025
100374H1CLONEDHUMAN3H-PYRILAMINEILOPERIDONE1854PDSP Certified DataJan 15, 2025Jan 28, 2025
100375NETCLONEDHUMAN3H-NisoxetineBUPROPION>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100376SLC6A3CLONEDHUMAN3H-WIN 35,428CITALOPRAM>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100377SLC6A3CLONEDHUMAN3H-WIN 35,428Desmethylcitalopram>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100378SLC6A3CLONEDHUMAN3H-WIN 35,428DOXEPIN>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100379NETCLONEDHUMAN3H-NisoxetineEtoperidone>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100380SLC6A3CLONEDHUMAN3H-WIN 35,428Etoperidone>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100381SLC6A4CLONEDHUMAN3H-IMIPRAMINEIproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100382NETCLONEDHUMAN3H-NisoxetineIproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100383SLC6A3CLONEDHUMAN3H-WIN 35,428Iproniazid>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100384SLC6A3CLONEDHUMAN3H-WIN 35,428Lofepramine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100385SLC6A4CLONEDHUMAN3H-IMIPRAMINEmirtazepine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100386SLC6A3CLONEDHUMAN3H-WIN 35,428mirtazepine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100387SLC6A3CLONEDHUMAN3H-WIN 35,428mirtazepine(+)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100388SLC6A4CLONEDHUMAN3H-IMIPRAMINEmirtazepine(+)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100389SLC6A4CLONEDHUMAN3H-IMIPRAMINEmirtazepine(-)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100390NETCLONEDHUMAN3H-Nisoxetinemirtazepine(-)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100391SLC6A3CLONEDHUMAN3H-WIN 35,428mirtazepine(-)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100392SLC6A4CLONEDHUMAN3H-IMIPRAMINENORTRYPTYLINE18Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100393NETCLONEDHUMAN3H-NisoxetineNORTRYPTYLINE4.37Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100394SLC6A3CLONEDHUMAN3H-WIN 35,428NORTRYPTYLINE1140Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100395SLC6A4CLONEDHUMAN3H-IMIPRAMINEPhenelzine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100396NETCLONEDHUMAN3H-NisoxetinePhenelzine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100397SLC6A4CLONEDHUMAN3H-IMIPRAMINETRANYLCYPROMINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100398SLC6A4CLONEDHUMAN3H-IMIPRAMINEViloxazine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100399SLC6A3CLONEDHUMAN3H-WIN 35,428Viloxazine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100400SLC6A3CLONEDHUMAN3H-WIN 35,428ZIMELIDINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100401SLC6A4CLONEDHUMAN3H-IMIPRAMINEAlprazolam>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100402SLC6A4CLONEDHUMAN3H-IMIPRAMINEClonazepam>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100403SLC6A4CLONEDHUMAN3H-IMIPRAMINEacetazolamide>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100404SLC6A4CLONEDHUMAN3H-IMIPRAMINECARBAMAZEPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100405SLC6A4CLONEDHUMAN3H-IMIPRAMINENIFEDIPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100406SLC6A4CLONEDHUMAN3H-IMIPRAMINEVERAPAMIL245Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100407SLC6A4CLONEDHUMAN3H-IMIPRAMINERESERPINE1460Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100408SLC6A4CLONEDHUMAN3H-IMIPRAMINECOCAINE340Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100409SLC6A4CLONEDHUMAN3H-IMIPRAMINEMAZINDOL39Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100410SLC6A4CLONEDHUMAN3H-IMIPRAMINEMETHAMPHETAMINE (+)>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100411SLC6A4CLONEDHUMAN3H-IMIPRAMINEMETHYLPHENIDATE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100412SLC6A4CLONEDHUMAN3H-IMIPRAMINEGBR-12935940Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100413SLC6A4CLONEDHUMAN3H-IMIPRAMINECHLORPHENIRAMINE15.2Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100414SLC6A4CLONEDHUMAN3H-IMIPRAMINEDiphenhydramine3800Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100415SLC6A4CLONEDHUMAN3H-IMIPRAMINEDOPAMINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100416SLC6A4CLONEDHUMAN3H-IMIPRAMINENOREPINEPHRINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100417SLC6A4CLONEDHUMAN3H-IMIPRAMINE5-Hydroxy Tryptamine2100Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100418NETCLONEDHUMAN3H-NisoxetineAlprazolam>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100419NETCLONEDHUMAN3H-NisoxetineClonazepam>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100420NETCLONEDHUMAN3H-Nisoxetineacetazolamide>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100421NETCLONEDHUMAN3H-NisoxetineCARBAMAZEPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100422NETCLONEDHUMAN3H-NisoxetineNIFEDIPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100423NETCLONEDHUMAN3H-NisoxetineAmphetamine,(+)530Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100424NETCLONEDHUMAN3H-NisoxetineCOCAINE1420Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100425NETCLONEDHUMAN3H-NisoxetineMAZINDOL0.45Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100426NETCLONEDHUMAN3H-NisoxetineMETHAMPHETAMINE (+)660Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100427NETCLONEDHUMAN3H-NisoxetineMETHYLPHENIDATE234Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100428NETCLONEDHUMAN3H-NisoxetineGBR-12935310Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100429NETCLONEDHUMAN3H-NisoxetineCHLORPHENIRAMINE1440Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100430NETCLONEDHUMAN3H-NisoxetineDiphenhydramine960Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100431NETCLONEDHUMAN3H-NisoxetineDOPAMINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100432NETCLONEDHUMAN3H-NisoxetineNOREPINEPHRINE2200Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100433NETCLONEDHUMAN3H-Nisoxetine5-Hydroxy Tryptamine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100434SLC6A3CLONEDHUMAN3H-WIN 35,428Alprazolam>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100435SLC6A3CLONEDHUMAN3H-WIN 35,428Clonazepam>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100436SLC6A3CLONEDHUMAN3H-WIN 35,428acetazolamide>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100437SLC6A3CLONEDHUMAN3H-WIN 35,428CARBAMAZEPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100438SLC6A3CLONEDHUMAN3H-WIN 35,428NIFEDIPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100439SLC6A3CLONEDHUMAN3H-WIN 35,428VERAPAMIL>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100440SLC6A3CLONEDHUMAN3H-WIN 35,428RESERPINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100441SLC6A3CLONEDHUMAN3H-WIN 35,428Amphetamine,(+)2900Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100442SLC6A3CLONEDHUMAN3H-WIN 35,428COCAINE220Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100443SLC6A3CLONEDHUMAN3H-WIN 35,428MAZINDOL8.1Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100444SLC6A3CLONEDHUMAN3H-WIN 35,428METHAMPHETAMINE (+)2800Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100445SLC6A3CLONEDHUMAN3H-WIN 35,428METHYLPHENIDATE24Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100446SLC6A3CLONEDHUMAN3H-WIN 35,428GBR-1293527.2Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100447SLC6A3CLONEDHUMAN3H-WIN 35,428CHLORPHENIRAMINE1060Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100448SLC6A3CLONEDHUMAN3H-WIN 35,428Diphenhydramine2200Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100449SLC6A3CLONEDHUMAN3H-WIN 35,428DOPAMINE2400Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100450SLC6A3CLONEDHUMAN3H-WIN 35,428NOREPINEPHRINE>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100451SLC6A3CLONEDHUMAN3H-WIN 35,4285-Hydroxy Tryptamine>10000Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100452SLC6A3CLONEDHUMAN3H-WIN 35,428AMFONELIC ACID207Tatsumi M, et al., 1997Jan 15, 2025Jan 15, 2025
100453Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine110Niso M et al 2013Jan 15, 2025Jan 28, 2025
100454Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine8.67Niso M et al 2013Jan 15, 2025Jan 28, 2025
100455Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine373Niso M et al 2013Jan 15, 2025Jan 28, 2025
100456Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine35.9Niso M et al 2013Jan 15, 2025Jan 28, 2025
100457Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 7.43Niso M et al 2013Jan 15, 2025Jan 28, 2025
100458Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)cis-2,6-Dimethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine18.5Niso M et al 2013Jan 15, 2025Jan 28, 2025
100459Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine236Niso M et al 2013Jan 15, 2025Jan 28, 2025
100460Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-Pentazocine(+)2,2,6,6-Tetramethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 88.6Niso M et al 2013Jan 15, 2025Jan 28, 2025
100461Sigma 2LIVERRAT3H-DTGcis-2,6-Dimethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine90.9Niso M et al 2013Jan 15, 2025Jan 28, 2025
100462Sigma 2LIVERRAT3H-DTGcis-2,6-Dimethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine11.1Niso M et al 2013Jan 15, 2025Jan 28, 2025
100463Sigma 2LIVERRAT3H-DTG2,2,6,6-Tetramethyl-1-[3-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperidine641Niso M et al 2013Jan 15, 2025Jan 28, 2025
100464Sigma 2LIVERRAT3H-DTG2,2,6,6-Tetramethyl-1-[4-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)butyl]piperidine69.8Niso M et al 2013Jan 15, 2025Jan 28, 2025
100465Sigma 2LIVERRAT3H-DTGcis-2,6-Dimethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine 45.4Niso M et al 2013Jan 15, 2025Jan 28, 2025
100466Sigma 2LIVERRAT3H-DTGcis-2,6-Dimethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine13.8Niso M et al 2013Jan 15, 2025Jan 28, 2025
100467Sigma 2LIVERRAT3H-DTG2,2,6,6-Tetramethyl-1-[3-(6-methoxynaphthalen-1-yl)propyl]piperidine495Niso M et al 2013Jan 15, 2025Jan 28, 2025
100468Sigma 2LIVERRAT3H-DTG2,2,6,6-Tetramethyl-1-[4-(6-methoxynaphthalen-1-yl)butyl]piperidine 90.7Niso M et al 2013Jan 15, 2025Jan 28, 2025
100469Sigma 1CORTICAL MEMBRANESGUINEA PIG3H-PentazocinePENTAZOCINE (+)4.1Niso M et al 2013Jan 15, 2025Jan 28, 2025
100470Sigma 2LIVERRAT3H-DTGDTG30.2Niso M et al 2013Jan 15, 2025Jan 28, 2025
100471D1CLONEDHUMAN[3H]SCH23390F17464>10000Cosi C et al 2021Jan 15, 2025Jan 28, 2025
1004725-HT1ACLONEDHUMAN[3H]8-OH-DPATF174640.162181Cosi C et al 2021Jan 15, 2025Jan 15, 2025
100473D2CLONEDHUMAN[3H]spiperoneF174648.70964Cosi C et al 2021Jan 15, 2025Jan 29, 2025
100474D2CLONEDHUMAN[3H]spiperoneF1746412.0226Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100475D3CLONEDHUMAN[3H]spiperoneF174640.158489Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100476D4CLONEDHUMAN[3H]spiperoneF17464>10000Cosi C et al 2021Jan 15, 2025Jan 29, 2025
100477D2dorsal striatum RAT[3H]nemonaprideF174645.01187Cosi C et al 2021Jan 15, 2025Jan 28, 2025
1004785-HT1AHIPPOCAMPUSRAT[3H]8-OH-DPATF174641.25893Cosi C et al 2021Jan 15, 2025Jan 15, 2025
1004795-HT1DCLONEDHUMAN3H-GR125743F1746426.3027Cosi C et al 2021Jan 15, 2025Jan 15, 2025
1004805-HT2ACLONEDHUMAN3H-KETANSERINF17464436.516Cosi C et al 2021Jan 15, 2025Jan 15, 2025
1004815-HT2BCLONEDHUMAN[3H]mesulergineF174641548.82Cosi C et al 2021Jan 15, 2025Jan 15, 2025
1004825-HT2CCLONEDHUMAN[3H]mesulergineF174641995.26Cosi C et al 2021Jan 15, 2025Jan 15, 2025
100483Alpha1BCEREBRAL CORTEXPIG3H-PRAZOSINF17464794.328Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100484Alpha2ACLONEDHUMANUNDEFINEDF17464281.838Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100485Alpha2BCLONEDHUMANUNDEFINEDF17464208.93Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100486Alpha2CCLONEDHUMANUNDEFINEDF17464275.423Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100487Beta 2CLONEDHUMANUNDEFINEDF17464>10000Cosi C et al 2021Jan 15, 2025Jan 15, 2025
100488CLONEDRATUNDEFINEDF17464125.893Cosi C et al 2021Jan 15, 2025Jan 15, 2025
1004895-HT7CLONEDHUMANUNDEFINEDF17464>10000Cosi C et al 2021Jan 15, 2025Jan 29, 2025
1004905-HT1BCORTEXRATUNDEFINEDF174643981.07Cosi C et al 2021Jan 15, 2025Jan 15, 2025
100491H1CLONEDHUMANUNDEFINEDF1746421.3796Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100492MORCLONEDHUMANUNDEFINEDF17464141.254Cosi C et al 2021Jan 15, 2025Jan 28, 2025
100493M1CLONEDHUMANUNDEFINEDF17464>10000Cosi C et al 2021Jan 15, 2025Jan 15, 2025
100494M3CLONEDHUMANUNDEFINEDF17464>10000Cosi C et al 2021Jan 15, 2025Jan 15, 2025
100495Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100496Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide24Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100497Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100498Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide25.1Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100499Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100500Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)phenyl)-1H-1,2,3-triazole-4-carboxamide21.9Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100501Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100502Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide1.5Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100503Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100504Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide3Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100505Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100506Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide5.5Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100507Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100508Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1H-1,2,3-triazole-4-carboxamide1023Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100509Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100510Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(2-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide9.7Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100511Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100512Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide10.7Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100513Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide3345Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100514Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-methoxybenzyl)-1H-1,2,3-triazole-4-carboxamide5Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100515Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)1-Benzyl-N-(4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl)-1H-1,2,3-triazole-4-carboxamide4476Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100516Sigma 2LIVERRAT3H-DTG1-Benzyl-N-(4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl)-1H-1,2,3-triazole-4-carboxamide12.4Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100517Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide8082Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100518Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide22.5Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100519Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100520Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-hydroxybenzyl)-1H-1,2,3-triazole-4-carboxamide11.6Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100521Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100522Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(3-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide62.1Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100523Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100524Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl)-1-(4-(2-fluoroethoxy)benzyl)-1H-1,2,3-triazole-4-carboxamide48.2Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100525Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100526Sigma 2LIVERRAT3H-DTGN-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide150Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100527Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100528Sigma 2LIVERRAT3H-DTGN-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide180Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100529Sigma 2LIVERRAT3H-DTGN-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide410Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100530Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100531Sigma 2LIVERRAT3H-DTGN-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(2-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide156Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100532Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100533Sigma 2LIVERRAT3H-DTGN-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(3-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide214Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100534Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100535Sigma 2LIVERRAT3H-DTGN-(2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl)-1-(4-methoxybenthyl)-1H-1,2,3-triazole-4-carboxamide93.2Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100536Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100537Sigma 1LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)benzamide139Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100538Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-fluoroethoxy)ethyl)-1H-1,2,3-triazol-4-yl)benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100539Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-fluoroethoxy)ethyl)-1H-1,2,3-triazol-4-yl)benzamide137Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100540Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-(2-fluoroethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)-benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100541Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-(2-(2-fluoroethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)-benzamide212Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100542Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide8580Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100543Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(2-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide55Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100544Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100545Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide66.2Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100546Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(4-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100547Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-4-(1-(4-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide31.4Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100548Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide1752Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100549Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-(1-(3-methoxybenzyl)-1H-1,2,3-triazol-4-yl)benzamide66Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100550Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-(prop-2-ynyloxy)benzamide3678Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100551Sigma 2LIVERRAT3H-DTG5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-(prop-2-ynyloxy)benzamide12.2Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100552Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methoxy)-benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100553Sigma 2LIVERRAT3H-DTG5-Cyano-N-(4-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-butyl)-2-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methoxy)-benzamide31.9Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100554Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100555Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide56.8Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100556Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-2-methoxy-5-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-benzamide6359Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100557Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-2-methoxy-5-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-benzamide20.7Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100558Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((2-(2-fluoroethoxy)ethoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100559Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((2-(2-fluoroethoxy)ethoxy)methyl)-1H-1,2,3-triazol-1-yl)-2-methoxybenzamide66Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100560Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)N-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-(2-fluoroethoxy)benzamide>10000Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100561Sigma 2LIVERRAT3H-DTGN-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-5-(4-((dimethylamino)methyl)-1H-1,2,3-triazol-1-yl)-2-(2-fluoroethoxy)benzamide94Bai S, et al., 2014Jan 15, 2025Jan 15, 2025
100562GlyRCLONEDHUMAN3H-GlycineCHPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100563GlyRCLONEDHUMAN3H-GlycineCHPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100564GlyRCLONEDHUMAN3H-GlycineMCPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100565GlyRCLONEDHUMAN3H-GlycineCPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100566GlyRCLONEDHUMAN3H-GlycineL-glutamic acid>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100567GlyRCLONEDHUMAN3H-GlycineNMDA>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100568GlyRCLONEDHUMAN3H-GlycineCPP>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100569NMDACLONEDHUMAN[3H]CPPCHPG(RS)2089.3Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100570NMDACLONEDHUMAN[3H]CPPCHPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100571NMDACLONEDHUMAN[3H]CPPMCPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100572NMDACLONEDHUMAN[3H]CPPCPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100573NMDACLONEDHUMAN[3H]CPPL-glutamic acid218.776Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100574NMDACLONEDHUMAN[3H]CPPNMDA9120.11Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100575NMDACLONEDHUMAN[3H]CPPCPP69.1831Cavanni P, et.al., 1994Jan 15, 2025Jan 28, 2025
100576AMPACLONEDHUMANFunctionalCHPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100577AMPACLONEDHUMANFunctionalCHPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100578AMPACLONEDHUMANFunctionalMCPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100579AMPACLONEDHUMANFunctionalCPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100580AMPACLONEDHUMANFunctionalL-glutamic acid371.535Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100581AMPACLONEDHUMANFunctionalNMDA>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100582AMPACLONEDHUMANFunctionalCPP>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100583KACLONEDHUMAN3H-Kainic acidCHPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100584KACLONEDHUMAN3H-Kainic acidCHPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100585KACLONEDHUMAN3H-Kainic acidMCPG(RS)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100586KACLONEDHUMAN3H-Kainic acidCPG(S)>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100587KACLONEDHUMAN3H-Kainic acidL-glutamic acid107.152Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100588KACLONEDHUMAN3H-Kainic acidNMDA>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100589KACLONEDHUMAN3H-Kainic acidCPP>10000Cavanni P, et.al., 1994Jan 15, 2025Jan 15, 2025
100590CGRPCLONEDHUMAN1251-CGRPN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100591CGRPCLONEDHUMAN1251-CGRPN2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100592CGRPCLONEDHUMAN1251-CGRPN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100593CGRPCLONEDHUMAN1251-CGRPN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100594CGRPCLONEDHUMAN1251-CGRPN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-L-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100595CGRPCLONEDHUMAN1251-CGRPN2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysine-phenylamide Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100596CGRPCLONEDHUMAN1251-CGRP1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-phenyl-piperazine Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100597CGRPCLONEDHUMAN1251-CGRP1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-piperazine Dihydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100598CGRPCLONEDHUMAN1251-CGRP1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-(4-pyridinyl)piperazine>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100599CGRPCLONEDHUMAN1251-CGRPN2-[4-Amino-3,5-dibromo-N-(3-phenyl-1-oxopropyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrochloride>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100600CGRPCLONEDHUMAN1251-CGRPN2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100601CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine1000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100602CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine200Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100603CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperazinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 226Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100604CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate)250Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100605CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-[2(3H)-oxobenzoxazol-3-yl]-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate)44Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100606CGRPCLONEDHUMAN1251-CGRP1-[N2-[N-[[4-[N-(Aminocarbonyl)phenylamino]-1-piperidinyl]carbonyl]-3,5-dibromo-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate)4.7Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100607CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.2Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100608CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.03Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100609CGRPCLONEDHUMAN1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-4-phenyl-2(2H)-oxoimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.05Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100610CGRPSPLEENRAT1251-CGRP1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100611CGRPSPLEENRAT1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine56.7Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100612CGRPSPLEENmarmoset1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine2.7Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100613CGRPSPLEENRAT1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine6.4Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100614CGRPSPLEENmarmoset1251-CGRP1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.06Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100615CGRPCLONEDHUMANFunctionalN2-(3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-L-lysine-2-phenethylamide hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100616CGRPCLONEDHUMANFunctionalN2-[4-Amino-3,5-dibromo-N-(4-phenyl-1-oxobutyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100617CGRPCLONEDHUMANFunctionalN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-L-tyrosyl]-D-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100618CGRPCLONEDHUMANFunctionalN2-[3,5-Dibromo-N-(4-phenyl-1-oxobutyl)-D-tyrosyl]-D-lysine-2-phenethylamine>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100619CGRPCLONEDHUMANFunctionalN2-[3,5-Dibromo-N-(4-phenyl-1-oxybutyl)-L-tyrosyl]-L-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100620CGRPCLONEDHUMANFunctionalN2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysine-phenylamide Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100621CGRPCLONEDHUMANFunctional1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-4-phenyl-piperazine Hydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100622CGRPCLONEDHUMANFunctional1-[N2-[4-Amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl]-piperazine Dihydrobromide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100623CGRPCLONEDHUMANFunctional1-[N2-[4-amino-3,5-dibromo-N-(1-oxo-4-phenylbutyl)-D-phenylalanyl]-L-lysyl-4-(4-pyridinyl)piperazine>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100624CGRPCLONEDHUMANFunctionalN2-[4-Amino-3,5-dibromo-N-(3-phenyl-1-oxopropyl)-D-phenylalanyl]-L-lysine-2-phenethylamide Hydrochloride>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100625CGRPserumHUMANFunctionalN2-[3,5-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysine-2-phenethylamide>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100626CGRPserumHUMANFunctional1-[N2-[3,4-Dibromo-N-[[[2-(2-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]4-(4-pyridinyl)piperazine1000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100627CGRPserumHUMANFunctional1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine200Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100628CGRPserumHUMANFunctional1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperazinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine 226Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100629CGRPserumHUMANFunctional1-[N2-[3,5-Dibromo-N-[[4-(2-methoxyphenyl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate)250Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100630CGRPserumHUMANFunctional1-[N2-[3,5-Dibromo-N-[[4-[2(3H)-oxobenzoxazol-3-yl]-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate)44Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100631CGRPserumHUMANFunctional1-[N2-[N[[4-[N-(Aminocarbonyl)phenylamino]-1-piperidinyl]carbonyl]-3,5-dibromo-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine Bis(trifluoroacetate)4.7Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100632CGRPserumHUMANFunctional1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.2Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100633CGRPserumHUMANFunctional1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.03Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100634CGRPratclonedFunctional1-[N2-[3,5-Dibromo-N-[[[2-(3-methoxyphenyl)ethyl]amino]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine>10000Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100635CGRPratclonedFunctional1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidazol-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine56.7Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100636CGRPCLONEDRATFunctional1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine6.4Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100637CGRPSPLEENmarmosetFunctional1-[N2-[3,5-Dibromo-N-[[4-(1,3-dihydro-2(2H)-oxobenzimidal-1-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine2.7Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
100638CGRPSPLEENmarmosetFunctional1-[N2-[3,5-Dibromo-N-[[4-(3,4-dihydro-2(1H)-oxoquinazolin-3-yl)-1-piperidinyl]carbonyl]-D-tyrosyl]-L-lysyl]-4-(4-pyridinyl)piperazine0.06Rudolf K, et al., 2005Jan 15, 2025Jan 15, 2025
1006395-HT1ACLONEDHUMAN3H-WAY100635CYPROHEPTADINE50Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006405-HT1BCLONEDHUMAN3H-5CTCYPROHEPTADINE1600Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006415-HT1DCLONEDHUMAN3H-5CTCYPROHEPTADINE670Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006425-HT2ACLONEDHUMAN3H-KETANSERINCYPROHEPTADINE1.9Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006435-HT2BCLONEDHUMAN3H-LSDCYPROHEPTADINE2.6Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006445-HT2CCLONEDHUMAN3H-MESULERGINECYPROHEPTADINE18Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006455-HT3CLONEDHUMAN3H-GR-65630CYPROHEPTADINE235Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006465-HT5ACLONEDHUMAN3H-LSDCYPROHEPTADINE57Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006475-HT6CLONEDHUMAN3H-LSDCYPROHEPTADINE96Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006485-HT7CLONEDHUMAN3H-LSDCYPROHEPTADINE30Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100649D1CLONEDHUMAN3H-SCH23390CYPROHEPTADINE10Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100650D2CLONEDHUMAN3H-MethylspiperoneCYPROHEPTADINE74Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100651D4CLONEDHUMAN3H-MethylspiperoneCYPROHEPTADINE120Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100652D5CLONEDHUMAN3H-SCH23390CYPROHEPTADINE60Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100653SERTCLONEDHUMAN3H-CITALOPRAMCYPROHEPTADINE>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100654NETCLONEDHUMAN3H-NisoxetineCYPROHEPTADINE2550Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100655DATCLONEDHUMAN[3H]WIN35428CYPROHEPTADINE4100Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100656H1CLONEDHUMAN3H-PYRILAMINECYPROHEPTADINE2.3Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100657Alpha1ACLONEDHUMAN3H-PRAZOSINCYPROHEPTADINE45Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100658Alpha1BCLONEDHUMAN3H-PRAZOSINCYPROHEPTADINE>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100659Alpha2ACLONEDHUMAN3H-RAUWOLSCINECYPROHEPTADINE330Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100660Alpha2BCLONEDHUMAN3H-RAUWOLSCINECYPROHEPTADINE220Young, R., et. al., 2005Jan 15, 2025Jan 29, 2025
100661Alpha2CCLONEDHUMAN3H-RAUWOLSCINECYPROHEPTADINE160Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
1006625-HT1DCLONEDHUMAN[3H]TiotidineCYPROHEPTADINE4.8Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100663M1CLONEDHUMAN3H-QNBCYPROHEPTADINE19Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100664M2CLONEDHUMAN3H-QNBCYPROHEPTADINE18Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100665M3CLONEDHUMAN3H-QNBCYPROHEPTADINE12Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100666M4CLONEDHUMAN3H-QNBCYPROHEPTADINE19Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100667M5CLONEDHUMAN3H-QNBCYPROHEPTADINE4.5Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100668CLONEDHUMAN125I-ClonidineCYPROHEPTADINE204Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100669Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)CYPROHEPTADINE>10000Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100670Sigma 2PC12RAT3H-DTGCYPROHEPTADINE750Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006715-HT1ACLONEDHUMAN3H-WAY100635Pizotyline270Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006725-HT1BCLONEDHUMAN3H-5CTPizotyline1415Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006735-HT1DCLONEDHUMAN3H-5CTPizotyline770Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006745-HT1ECLONEDHUMAN3H-5HTPizotyline820Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006755-HT2ACLONEDHUMAN3H-KETANSERINPizotyline2Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006765-HT2BCLONEDHUMAN3H-LSDPizotyline2.3Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006775-HT2CCLONEDHUMAN3H-MESULERGINEPizotyline8.4Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006785-HT3CLONEDHUMAN3H-GR-65630Pizotyline95Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006795-HT5ACLONEDHUMAN3H-LSDPizotyline110Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006805-HT6CLONEDHUMAN3H-LSDPizotyline74Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
1006815-HT7CLONEDHUMAN3H-LSDPizotyline17Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100682D1CLONEDHUMAN3H-SCH23390Pizotyline3.5Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100683D2CLONEDHUMAN3H-N-MethylspiporonePizotyline87Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100684D4CLONEDHUMAN3H-N-MethylspiporonePizotyline64Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100685D5CLONEDHUMAN3H-SCH23390Pizotyline50Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100686SERTCLONEDHUMAN3H-CITALOPRAMPizotyline>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100687DATCLONEDHUMAN3H-WIN 35,428Pizotyline>10000Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100688NETCLONEDHUMAN3H-NisoxetinePizotyline710Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100689H1CLONEDHUMAN3H-PYRILAMINEPizotyline1.9Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
1006905-HT1DCLONEDHUMAN125I-aminopotentidinePizotyline1.4Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100691Alpha1ACLONEDHUMAN3H-PRAZOSINPizotyline65Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100692Alpha1BCLONEDHUMAN3H-PRAZOSINPizotyline>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100693Alpha2ACLONEDHUMAN3H-RAUWOLSCINEPizotyline660Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100694Alpha2BCLONEDHUMAN3H-RAUWOLSCINEPizotyline225Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100695Alpha2CCLONEDHUMAN3H-RAUWOLSCINEPizotyline390Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100696Beta1CLONEDHUMAN125I-PindololPizotyline>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100697Beta2CLONEDHUMAN3H-CGP-12177Pizotyline>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100698Beta1CLONEDHUMAN125I-PindololCYPROHEPTADINE>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100699Beta2CLONEDHUMAN3H-CGP-12177CYPROHEPTADINE>10000Young, R., et. al., 2005Jan 15, 2025Jan 28, 2025
100700M1CLONEDHUMAN3H-QNBPizotyline67Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100701M2CLONEDHUMAN3H-QNBPizotyline34Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100702M3CLONEDHUMAN3H-QNBPizotyline29Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100703M4CLONEDHUMAN3H-QNBPizotyline130Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100704M5CLONEDHUMAN3H-QNBPizotyline6.8Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100705I1CLONEDHUMAN125I-ClonidinePizotyline121Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100706Sigma 1BRAINGUINEA PIG3H-Pentazocine(+)Pizotyline>10000Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100707Sigma 2PC12RAT3H-DTGPizotyline6450Young, R., et. al., 2005Jan 15, 2025Jan 15, 2025
100708MT1C.H.O.HUMAN2-I125 iodomelatoninN-Propargyl-2-(5-methoxy-1H-indol-3-yl)acetamide14Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100709MT2C.H.O.HUMAN2-I125 iodomelatoninN-Propargyl-2-(5-methoxy-1H-indol-3-yl)acetamide3.8Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
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100712MT1C.H.O.HUMAN2-I125 iodomelatoninN-Allyl-2-(5-methoxy-1H-indol-3-yl)acetamide17Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
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100715MT2C.H.O.HUMAN2-I125 iodomelatoninN-Allyl-3-(5-methoxy-1H-indol-3-yl)propanamide0.45Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100716MT1C.H.O.HUMAN2-I125 iodomelatonin2-((5-Methoxy-1H-indol-3-yl)methyl)-5-methyloxazole280Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100717MT2C.H.O.HUMAN2-I125 iodomelatonin2-((5-Methoxy-1H-indol-3-yl)methyl)-5-methyloxazole1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100718MT1C.H.O.HUMAN2-I125 iodomelatonin2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyloxazole1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100719MT2C.H.O.HUMAN2-I125 iodomelatonin2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyloxazole498Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100720MT1C.H.O.HUMAN2-I125 iodomelatonin5-((5-Methoxy-1H-indol-3-yl)methyl)-3-methyl-1,2,4-oxadiazole170Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100721MT2C.H.O.HUMAN2-I125 iodomelatonin5-((5-Methoxy-1H-indol-3-yl)methyl)-3-methyl-1,2,4-oxadiazole44Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100722MT1C.H.O.HUMAN2-I125 iodomelatonin5-(2-(5-Methoxy-1H-indol-3-yl)-3-methyl-1,2,4-oxadiazole1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100723MT2C.H.O.HUMAN2-I125 iodomelatonin5-(2-(5-Methoxy-1H-indol-3-yl)-3-methyl-1,2,4-oxadiazole1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100724MT1C.H.O.HUMAN2-I125 iodomelatonin2-((5-Methoxy-1H-indol-3-yl)methyl)5-1,3,4-oxadiazole210Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100725MT2C.H.O.HUMAN2-I125 iodomelatonin2-((5-Methoxy-1H-indol-3-yl)methyl)5-1,3,4-oxadiazole16Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100726MT1C.H.O.HUMAN125I-Iodomelatonin2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyl-1,3,4-oxadiazole709Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100727MT2C.H.O.HUMAN125I-Iodomelatonin2-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-5-methyl-1,3,4-oxadiazole190Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100728MT1C.H.O.HUMAN125I-Iodomelatonin2-(2-(5-Methoxy-1H-indol-3-yl)ehtyl)-1,3,4-oxadiazole570Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100729MT2C.H.O.HUMAN125I-Iodomelatonin2-(2-(5-Methoxy-1H-indol-3-yl)ehtyl)-1,3,4-oxadiazole68Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100730MT1C.H.O.HUMAN125I-Iodomelatonin5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazol-2(3H)-one1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100731MT2C.H.O.HUMAN125I-Iodomelatonin5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazol-2(3H)-one160Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100732MT1C.H.O.HUMAN125I-Iodomelatonin5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazol-2(3H)-one35Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100733MT2C.H.O.HUMAN125I-Iodomelatonin5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazol-2(3H)-one4Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100734MT1C.H.O.HUMAN125I-Iodomelatonin5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazole-2(3H)-thione1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100735MT2C.H.O.HUMAN125I-Iodomelatonin5-((5-Methoxy-1H-indol-3-yl)methyl)-1,3,4,-oxadiazole-2(3H)-thione535Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100736MT1C.H.O.HUMAN125I-Iodomelatonin5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazole-2(3H)-thione1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100737MT2C.H.O.HUMAN125I-Iodomelatonin5-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-1,3,4-oxadiazole-2(3H)-thione530Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100738MT1C.H.O.HUMAN125I-Iodomelatonin3-((5-Methoxy-1H-indol-3-yl)methyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100739MT2C.H.O.HUMAN125I-Iodomelatonin3-((5-Methoxy-1H-indol-3-yl)methyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one560Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100740MT1C.H.O.HUMAN125I-Iodomelatonin3-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100741MT2C.H.O.HUMAN125I-Iodomelatonin3-(2-(5-Methoxy-1H-indol-3-yl)ethyl)-4-methyl-1H-1,2,4,-triazol-5(4H)-one1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100742MT1C.H.O.HUMAN125I-Iodomelatonin4-Ethyl-3-((5-methoxy-1H-indol-3-yl)methyl)1H-1,2,4-triazol-5(4H)-thione1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100743MT2C.H.O.HUMAN125I-Iodomelatonin4-Ethyl-3-((5-methoxy-1H-indol-3-yl)methyl)1H-1,2,4-triazol-5(4H)-thione220Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100744MT1C.H.O.HUMAN125I-Iodomelatonin4-Ethyl-3-(2-(5-methoxy-1H-indol-3-yl)ethyl)-1H-1,2,4-triazol-5(4H)-thione1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100745MT2C.H.O.HUMAN125I-Iodomelatonin4-Ethyl-3-(2-(5-methoxy-1H-indol-3-yl)ethyl)-1H-1,2,4-triazol-5(4H)-thione1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100746MT1C.H.O.HUMAN125I-IodomelatoninN-Ethyl-5-((5-methoxy-1H-indol-3-yl)methyl)-1,3,4-thiadiazol-2-amine1000Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100747MT2C.H.O.HUMAN125I-IodomelatoninN-Ethyl-5-((5-methoxy-1H-indol-3-yl)methyl)-1,3,4-thiadiazol-2-amine17Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100748MT1C.H.O.HUMAN125I-IodomelatoninDMT,5-MeO210Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100749MT2C.H.O.HUMAN125I-IodomelatoninDMT,5-MeO16Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100750MT1C.H.O.HUMAN125I-IodomelatoninMELATONIN0.091Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100751MT2C.H.O.HUMAN125I-IodomelatoninMELATONIN0.15Revenga, de la Fuente Mario, et. al. 2015Jan 15, 2025Jan 29, 2025
100752PDE1CLONEDHUMANFunctionalRoflumilast>10000Liu S, et al., 2005Jan 15, 2025Jan 15, 2025