The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

Selecting a hot ligand or test ligand from the table will redirect you to the specifications of the chosen entity.

Selecting a citation from the table will open its respective PubMed link.

Showing 82,001-83,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
84749MORCLONEDHUMAN3H-DAMGO(±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84750DORCLONEDHUMAN3H-DADLE(±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84751KORCLONEDHUMAN3H-U69593(±)-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carbonyl)-L-phenylalanine>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84752DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84753MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84754MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-methyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84755DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-methyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84756KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-methyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84757KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-benzyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84758DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-benzyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84759MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-benzyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84760MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84761DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84762KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84763KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84764DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84765MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84766MORCLONEDHUMAN3H-DAMGO±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84767DORCLONEDHUMAN3H-DADLE±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84768KORCLONEDHUMAN3H-U69593±)-(4aS,8R,8aS)-1-oxo-N-(pyridin-3-yl)-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84769KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84770DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84771MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84772MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-benzyl-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84773DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-benzyl-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84774DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84775MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84776MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84777DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84778DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84779MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84780MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84781DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84782KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-methyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84783KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N,N-dicyclohexyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84784DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N,N-dicyclohexyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84785MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N,N-dicyclohexyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84786MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84787DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chloro-4-methylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84788DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84789MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84790MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84791DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84792DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-bemzyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84793MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-bemzyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84794KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-bemzyl-N-methyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84795KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N,N-dicyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84796MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N,N-dicyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84797DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N,N-dicyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84798DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N,2-dibenzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84799MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N,2-dibenzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84800DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(3-chloro-4-methylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84801DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-nitro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84802DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84803MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(pyridin-3-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84804MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84805DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84806KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84807KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84808DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84809MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84810MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84811DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84812KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84813KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84814DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84815MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84816MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(2,4,6-trimethylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84817DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(2,4,6-trimethylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84818KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(2,4,6-trimethylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84819DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84820MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84821MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84822DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84823KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84824DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84825MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84826MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84827DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84828KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84829KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84830DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84831MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84832MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84833DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84834KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84835DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84836MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84837MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-nitrophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84838DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-nitrophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84839DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84840MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-iodophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84841MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84842DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-bromobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84843DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84844MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-methylbenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84845MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84846DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84847DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84848MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84849KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(adamantan-1-yl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84850KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84851DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84852MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-nitrophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84853DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-iodophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84854DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(3-bromobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84855DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84856MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-methylbenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84857MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84858DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(2,4,6-trimethylphenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84859DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84860MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84861MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84862DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84863DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84864MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84865MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84866DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84867DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84868MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84869MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84870DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84871DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N,2-bis(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84872MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N,2-bis(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84873MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84874DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84875DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84876MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84877MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84878DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84879DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-8-(pyrrolidine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84880MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-8-(pyrrolidine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84881MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N-(cyclopropylmethyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84882DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-N-(cyclopropylmethyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84883DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N,N-dimethyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84884MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N,N-dimethyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84885MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84886DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chlorophenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84887DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84888MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84889MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84890DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-8-(pyrrolidine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84891DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-2-benzyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84892MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-(4aS,8R,8aS)-2-benzyl-N-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84893MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84894DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N,N-dimethyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84895DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-chlorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84896DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84897MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3,4,5-trifluorophenyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84898MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-allyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84899DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-allyl-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84900DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84901MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84902MORCLONEDHUMAN3H-DAMGOethyl 4-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84903DORCLONEDHUMAN3H-DADLEethyl 4-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84904DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-methyl-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84905MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-methyl-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84906KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-methyl-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84907KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84908DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84909MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-N-phenyl-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84910MORCLONEDHUMAN3H-DAMGOethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1R)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84911DORCLONEDHUMAN3H-DADLEethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1R)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84912KORCLONEDHUMAN3H-U69593ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1R)-2-((±)-(4aS,8R,8aS)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamido)cyclohexane-1-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84913DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-allyl-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84914MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-allyl-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84915MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84916DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84917KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84918KORCLONEDHUMAN3H-U69593ethyl 4-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84919DORCLONEDHUMAN3H-DADLEethyl 4-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84920MORCLONEDHUMAN3H-DAMGOethyl 4-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84921MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84922DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84923DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84924MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84925KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84926DORCLONEDHUMAN3H-DADLEethyl (1S)-2-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84927MORCLONEDHUMAN3H-DAMGOethyl (1S)-2-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84928MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-allyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84929DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-allyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84930KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-allyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84931DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84932MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(2-carbamoylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84933MORCLONEDHUMAN3H-DAMGOethyl 4-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84934DORCLONEDHUMAN3H-DADLEethyl 4-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84935KORCLONEDHUMAN3H-U69593ethyl 4-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84936DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-methyl-1-oxo-N,2-diphenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84937MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-methyl-1-oxo-N,2-diphenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84938MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84939DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84940KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3,4-dimethoxybenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84941KORCLONEDHUMAN3H-U69593ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyla>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84942DORCLONEDHUMAN3H-DADLEethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyla>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84943MORCLONEDHUMAN3H-DAMGOethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyla>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84944MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-allyl-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84945DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-allyl-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84946DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(2-carbamoylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84947MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(2-carbamoylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84948MORCLONEDHUMAN3H-DAMGOethyl 4-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84949DORCLONEDHUMAN3H-DADLEethyl 4-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)benzoate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84950DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84951MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84952MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84953DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dimethoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84954DORCLONEDHUMAN3H-DADLEethyl (1S)-2-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyla>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84955MORCLONEDHUMAN3H-DAMGOethyl (1S)-2-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxylate and ethyl (1S)-2-((±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamido)cyclohexane-1-carboxyla>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84956MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydro-1H-isochromen-1-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84957DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydro-1H-isochromen-1-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84958KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydro-1H-isochromen-1-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84959KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84960DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84961MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84962MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamid>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84963DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamid>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84964KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamid>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84965DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclohexylmethyl)-N-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84966MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclohexylmethyl)-N-isopropyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84967MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84968DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84969KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84970DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84971MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84972MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84973DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84974KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84975DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84976MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84977MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-cyclohexyl-N-isopropyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84978DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-cyclohexyl-N-isopropyl-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84979DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84980MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84981KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-8-(4-methylpiperazine-1-carbonyl)-2-phenyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84982DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84983MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3,4-dichlorobenzyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84984MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84985DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84986KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-hexylphenyl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84987KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84988DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84989MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-1-oxo-2-phenyl-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84990MORCLONEDHUMAN3H-DAMGO±)-(4aS,8R,8aS)-2-benzyl-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84991DORCLONEDHUMAN3H-DADLE±)-(4aS,8R,8aS)-2-benzyl-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84992KORCLONEDHUMAN3H-U69593±)-(4aS,8R,8aS)-2-benzyl-8-(4-methylpiperazine-1-carbonyl)-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84993DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(3,4-dichlorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84994DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84995MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84996KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(4-hexylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84997KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-N-(pyrazin-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84998MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
84999DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-cyclohexyl-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85000DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85001MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85002MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85003DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85004DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85005MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-N-(3,4-difluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85006MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85007DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85008DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85009MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(cyclopropylmethyl)-1-oxo-N-(thiazol-2-yl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85010MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85011DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-cyclohexyl-N-methyl-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85012DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85013MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85014MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-((R)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85015DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS,8R,8aS)-N-(3-chlorophenyl)-1-oxo-2-((R)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85016DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-((R)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85017MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS,8R,8aS)-N-(3,4-difluorophenyl)-1-oxo-2-((R)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85018MORCLONEDHUMAN3H-DAMGO±)-(4aS,8R,8aS)-N-(thiazol-2-yl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS,8R,8aS)-N-(thiazol-2-yl)-1-oxo-2-((R)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85019DORCLONEDHUMAN3H-DADLE±)-(4aS,8R,8aS)-N-(thiazol-2-yl)-1-oxo-2-((S)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide and (±)-(4aS,8R,8aS)-N-(thiazol-2-yl)-1-oxo-2-((R)-1-phenylethyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85020DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85021DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3-bromobenzyl)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85022DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85023MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclopropylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85024MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85025DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85026DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85027MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85028KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85029DORCLONEDHUMAN3H-DADLE4-chloro-3-(trifluoromethyl)phenyl (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85030MORCLONEDHUMAN3H-DAMGO4-chloro-3-(trifluoromethyl)phenyl (±)-(4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85031MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluoro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85032DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-fluoro-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85033DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85034DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(2,3-difluoro-4-methylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85035MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(2,3-difluoro-4-methylphenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85036MORCLONEDHUMAN3H-DAMGO4-chloro-3-(trifluoromethyl)phenyl (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85037DORCLONEDHUMAN3H-DADLE4-chloro-3-(trifluoromethyl)phenyl (±)-(4aS,8R,8aS)-2-(cyclohexylmethyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxylate>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85038DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-fluorobenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85039DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(2-fluorobenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85040DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85041MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85042KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85043DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(2-methoxybenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85044DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85045MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85046KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85047KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85048DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85049MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85050MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(2-fluoro-6-methoxybenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85051DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(2-fluoro-6-methoxybenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85052KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(2-fluoro-6-methoxybenzyl)-N-(4-methyl-3-(trifluoromethyl)phenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85053KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(2,3-difluoro-4-methylphenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85054DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(2,3-difluoro-4-methylphenyl)-2-(2-fluoro-6-methoxybenzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85055DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(2,3,4,5,6-pentafluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85056MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(2,3,4,5,6-pentafluorophenyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85057MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-N-phenyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85058DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-N-phenyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85059KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-2-benzyl-N-phenyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85060KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-2-benzyl-N-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85061DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-N-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85062MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-N-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85063MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-N-(3-chlorophenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85064DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-N-(3-chlorophenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85065KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-2-benzyl-N-(3-chlorophenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85066KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85067DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85068MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85069MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85070DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85071KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85072KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85073DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85074MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85075MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-phenyl-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85076DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-benzyl-1-oxo-N-phenyl-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85077DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-N,2-dicyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85078MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-N,2-dicyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85079MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-N-(3-chlorlophenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85080DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-N-(3-chlorlophenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85081DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85082MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85083KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-N-(4-bromo-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85084KORCLONEDHUMAN3H-U69593(±)-(5aS,9R,9aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85085DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85086MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-1-oxo-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85087MORCLONEDHUMAN3H-DAMGO(±)-(5aS,9R,9aS)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85088DORCLONEDHUMAN3H-DADLE(±)-(5aS,9R,9aS)-2-cyclohexyl-1-oxo-N-(thiazol-2-yl)-2,3,4,5,5a,8,9,9a-octahydro-1H-benzo[c]azepine-9-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85089DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-benzyl-3-oxo-N-phenyl-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85090DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-N-cyclohexyl-2-benzyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85091MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-N-cyclohexyl-2-benzyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85092KORCLONEDHUMAN3H-U69593(±)-(3aS,4R,7aS)-N-cyclohexyl-2-benzyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85093KORCLONEDHUMAN3H-U69593(±)-(3aS,4R,7aS)-2-benzyl-N-(3-chlorophenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85094DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-benzyl-N-(3-chlorophenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85095MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-benzyl-N-(3-chlorophenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85096MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85097DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-benzyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85098DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85099MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-benzyl-N-(4-chloro-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85100MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-benzyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85101DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-benzyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85102KORCLONEDHUMAN3H-U69593(±)-(3aS,4R,7aS)-2-benzyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85103DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-cyclohexyl-3-oxo-N-phenyl-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85104MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-cyclohexyl-3-oxo-N-phenyl-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85105MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-N,2-dicyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85106DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-N,2-dicyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85107DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-N-(3-chlorophenyl)-2-cyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85108MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-N-(3-chlorophenyl)-2-cyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85109MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-cyclohexyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85110DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-cyclohexyl-N-(4-bromo-3-(trifluoromethyl)phenyl)-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85111DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85112MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-cyclohexyl-3-oxo-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85113MORCLONEDHUMAN3H-DAMGO(±)-(3aS,4R,7aS)-2-cyclohexyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85114DORCLONEDHUMAN3H-DADLE(±)-(3aS,4R,7aS)-2-cyclohexyl-3-oxo-N-(thiazol-2-yl)-2,3,3a,4,5,7a-hexahydro-1H-isoindole-4-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85115DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-methoxy-N-methyl-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85116MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-methoxy-N-methyl-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85117KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-methoxy-N-methyl-1-oxo-2-phenethyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85118DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-([1,1-biphenyl]-2-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85119MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-([1,1-biphenyl]-2-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85120MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-([1,1-biphenyl]-2-yl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85121DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-([1,1-biphenyl]-2-yl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85122DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85123DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-3-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85124MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-3-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85125KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-3-yl)-1-oxo-3,4,4a,7,8,8a-hexahydro-1H-isochromene-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85126KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85127DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85128MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-2-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85129MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85130DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85131KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-chloro-3-(trifluoromethyl)phenyl)-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85132KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-phenyl-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85133DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-phenyl-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85134MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-phenyl-1-oxo-2-((4-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85135MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-((3-fluoro-4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85136DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-((3-fluoro-4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85137KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-((3-fluoro-4-methoxy-[1,1-biphenyl]-3-yl)methyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85138KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85139DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85140MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-N-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85141MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-4-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85142DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-4-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85143KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-N-(4-methyl-[1,1-biphenyl]-4-yl)-1-oxo-2-phenyl-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85144KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85145DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85146MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-((4-methyl-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85147DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-((4-acetamido-[1,1-biphenyl]-3-yl)methyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85148DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-((3-chloro-4-fluoro-[1,1-biphenyl]-3-yl)methyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85149DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-((3-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85150MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-((3-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85151KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-((3-(trifluoromethoxy)-[1,1-biphenyl]-3-yl)methyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85152DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-(3-(5-acetylthiophen-2-yl)benzyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85153DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-N-((4-acetyl-[1,1-biphenyl]-3-yl)methyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85154MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-N-((4-acetyl-[1,1-biphenyl]-3-yl)methyl)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85155DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-1-oxo-N-(3-(thiophen-2-yl)benzyl)-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85156DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-2-benzyl-N-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85157MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-2-benzyl-N-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85158KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-2-benzyl-N-(3-((E)-4-fluorostyryl)benzyl)-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinoline-8-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85159DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85160MORCLONEDHUMAN3H-DAMGO(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85161MORCLONEDHUMAN3H-DAMGO(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85162DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85163DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3-chlorobenzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85164DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3,5-dichlorobenzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85165DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-bromobenzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85166DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-(trifluoromethyl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85167DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-3-methylbenzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85168DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-3-chloro-4-methylbenzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85169DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-chloro-2-methylbenzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85170DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85171MORCLONEDHUMAN3H-DAMGO(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)thiazole-2-carboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85172DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-benzyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)-4-bromo-3-(trifluoromethyl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85173DORCLONEDHUMAN3H-DADLE(±)-(4aS,8R,8aS)-8-amino-2-benzyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85174MORCLONEDHUMAN3H-DAMGO(±)-(4aS,8R,8aS)-8-amino-2-benzyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85175KORCLONEDHUMAN3H-U69593(±)-(4aS,8R,8aS)-8-amino-2-benzyl-3,4,4a,7,8,8a-hexahydroisoquinolin-1(2H)-one>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85176MORCLONEDHUMAN3H-DAMGO(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85177MORCLONEDHUMAN3H-DAMGO(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85178DORCLONEDHUMAN3H-DADLE(±)-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)cyclohexanecarboxamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85179DORCLONEDHUMAN3H-DADLE(±)-3-chloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85180DORCLONEDHUMAN3H-DADLE(±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85181MORCLONEDHUMAN3H-DAMGO(±)-3,5-dichloro-N-((4aS,8R,8aS)-2-cyclohexyl-1-oxo-1,2,3,4,4a,7,8,8a-octahydroisoquinolin-8-yl)benzamide>10000PDSP Certified DataJan 15, 2025Jan 28, 2025
85182MT1NIH-3T3HUMAN125I-IodomelatoninTasimelteon0.35Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85183MT2NIH-3T3HUMAN125I-IodomelatoninTasimelteon0.17Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85184MT1CHO-K1HUMAN125I-IodomelatoninTasimelteon0.304Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85185MT2CHO-K1HUMAN125I-IodomelatoninTasimelteon0.0692Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85186A1recombinantHUMAN3H-DPCPXTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85187A1BRAINRAT3H-DPCPXTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85188A2ArecombinantHUMAN3H-CGS-21680Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85189A2ASTRIATUMRAT3H-CGS-21680Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85190A3recombinantHUMAN125I-AB-MECATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85191BRAINRAT3H-PRAZOSINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85192Alpha1ASUBMAXILLARY GLANDRAT3H-PRAZOSINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85193Alpha1BLIVERRAT3H-PRAZOSINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85194Alpha1DrecombinantHUMAN3H-PRAZOSINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85195CORTEXRAT3H-RAUWOLSCINETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85196Alpha2ArecombinantHUMAN3H-MK912Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85197Alpha2CrecombinantHUMAN3H-MK912Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85198Beta 1recombinantHUMAN125I-cyanopindololTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85199Beta 2recombinantHUMAN3H-CGP-12177Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85200Beta3recombinantHUMAN125I-cyanopindololTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85201recombinantHUMAN125I-AdrenomedullinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85202recombinantHUMAN125I-AdrenomedullinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85203KIDNEYRAT3H-D-AldosteroneTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85204recombinantHUMAN125I-C5a AnaphylatoxinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85205ARrecombinantRAT3H-miboleroneTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85206AT1recombinantHUMAN125I-AngiotensinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85207AT1ADRENALRABBIT3H-LosartanTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85208AT2recombinantHUMAN125I-CGP42112ATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85209ApelinrecombinantHUMAN125I-Apelin-13Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85210ADRENALGUINEA PIG125I-ANFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85211BB1recombinantHUMAN125I-BOMBESINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85212BB2recombinantHUMAN125I-BOMBESINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85213BB3recombinantHUMAN125I-BNTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85214B1IMR-90 cellsHUMAN3H-KallidinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85215B2recombinantHUMAN3H-BRADYKININTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85216B2ILEUMGUINEA PIG3H-BRADYKININTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85217T-47D cellsHUMAN125I-CalcitoninTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85218SK-N-MC CellsHUMAN125I-CGRPTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85219Calcium channelBRAINRAT3H-DiltiazemTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85220Calcium channelCEREBRAL CORTEXRAT3H-NitrendipineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85221Calcium channelBRAINRAT3H-D-888Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85222Calcium channelBrain Frontal LobeRAT125I-Omega-ConotoxinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85223CB1recombinantHUMAN3H-CP-55940Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85224CB2recombinantHUMAN3H-WIN 55,212-2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85225CCR1recombinantHUMAN125I-MIP-1AlphaTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85226CCR2recombinantHUMAN125I-MCP-1Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85227CCR4recombinantHUMAN125I-TARCTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85228CCR5recombinantHUMAN125I-MIP-1BetaTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85229CX3CR1recombinantHUMAN125I-FractalkineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85230CXCR2recombinantHUMAN125I-IL-8Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85231CCK1recombinantHUMAN3H-DevazepideTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85232CCK1PANCREASRAT3H-L364718Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85233CCK2FGS-7 JurkatHUMAN125I-CCK-8Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85234CCK2BRAINGUINEA PIG3H-CCK8Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85235BRAINRAT3H-ColcichineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85236CRF1recombinantHUMAN125I-CRFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85237D1recombinantHUMAN3H-SCH23390Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85238D2recombinantHUMAN3H-SPIPERONETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85239D2recombinantHUMAN3H-SPIPERONETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85240D3recombinantHUMAN3H-SPIPERONETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85241D4recombinantHUMAN3H-SPIPERONETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85242D5recombinantHUMAN3H-SCH23390Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85243ETAA10 cellsRAT125I-Endothelin 1Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85244ETArecombinantHUMAN125I-Endothelin 1Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85245ETBrecombinantHUMAN125I-Endothelin 1Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85246A431 CellsHUMAN125I-EGFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85247recombinantHUMAN125I-ErthropoietinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85248UterusCALF3H-EstradiolTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85249recombinantHUMAN3H-EstradiolTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85250recombinantHUMAN3H-EstradiolTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85251recombinantHUMAN125I-QRFP-43Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85252GPR8recombinantHUMAN125I-NPW-23Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85253GABAABRAINRAT3H-MUSCIMOLTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85254CEREBRAL CORTEXRAT3H-TBOBTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85255GABAABRAINRATFNZTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85256GABAABRAINRAT3H-MUSCIMOLTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85257GABABCEREBELLUMRAT3H-GABATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85258GABAArecombinantHUMAN3H-CGP 54626ATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85259GABAArecombinantHUMAN3H-CGP 54626ATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85260BRAIN CORTEXRAT3H-GabapentinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85261BRAINRAT125I-GALANINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85262GAL1recombinantHUMAN125I-GALANINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85263GAL2recombinantHUMAN125I-GALANINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85264HeLa S3 CellsHUMAN3H-dexamethasoneTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85265Jurkat cellsHUMAN3H-dexamethasoneTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85266AMPACEREBRAL CORTEXRAT3H-AMPATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85267BRAINRAT3H-Kainic acidTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85268NMDACEREBRAL CORTEXRAT3H-CGP39653Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85269NMDACEREBRAL CORTEXRAT3H-CGS-19755Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85270NMDACEREBRAL CORTEXRat brain3H-MDL-105519Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85271NMDACEREBRAL CORTEXRAT3H-TCPTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85272NMDACEREBRAL CORTEXRAT3H-IfenprodilTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85273BRAINRAT3H-L-GlutamateTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85274GlyRSpinal cordRAT3H-StrychnineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 27, 2025
85275GhrelinrecombinantHUMAN125I-ghrelinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85276H1recombinantHUMAN3H-PYRILAMINETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85277H1BRAINGUINEA PIG3H-PYRILAMINETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
852785-HT1DrecombinantHUMAN125I-iodoaminopotentidineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85279H3recombinantHUMAN3H-NAMHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85280H3BRAINRAT3H-R(-)-alpha-MethylhistamineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85281H4recombinantHUMAN3H-HistamineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85282recombinantHUMAN125I-Orexin-ATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85283recombinantHUMAN125I-Orexin-ATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85284CEREBRAL CORTEXRAT3H-IDAZOXANTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85285CEREBELLUMRAT3H-11,4,5-IP3Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85286LIVERRAT125I-InsulinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85287IL-13T3 CellsMOUSE125I-IL-1alphaTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85288IL-2CTLL-2 CellsMOUSE125I-IL-2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85289IL-2TIB-214MOUSE125I-IL-2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85290IL-6U266 CellsHUMAN125I-IL-6Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85291recombinantMOUSE125I-LeptinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85292U937 cellsHUMAN3H-LTB4Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85293NeutrophilRABBIT3H-LTB4Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85294CysLT1recombinantHUMAN3H-LTD4Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85295CysLT1recombinantHUMAN3H-LTC4Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85296MC1recombinantHUMAN125I-NDP-alpha-MSHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85297MC3recombinantHUMAN125I-NDP-alpha-MSHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85298MC4recombinantHUMAN125I-NDP-alpha-MSHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85299MC5recombinantHUMAN125I-NDP-alpha-MSHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85300MT1recombinantHUMAN125I-2-iodo-metatoninTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85301MT2recombinantHUMAN125I-2-iodo-metatoninTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85302recombinantHUMAN125I-MotilinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85303M1recombinantHUMAN3H-NMSTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85304M2recombinantHUMAN3H-NMSTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85305M3recombinantHUMAN3H-NMSTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85306M4recombinantHUMAN3H-NMSTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85307M5recombinantHUMAN3H-NMSTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85308FPR1recombinantHUMAN3H-fMLFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85309FPR2recombinantHUMAN125I-WKYMVmTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85310NK1SUBMAXILLARY GLANDGUINEA PIG3H-SUBSTANCE PTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85311NMU1recombinantHUMAN125I-Neuromedin U-25Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85312NMU2recombinantHUMAN125I-Neuromedin U-25Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85313Y1SK-N-MC CellsHUMAN125I-Peptide YYTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85314Y2KAN-TS CellsHUMAN125I-Peptide YYTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85315Y2Kidney MedullaRABBIT3H-Neuropeptide YTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85316NTSR1recombinantHUMAN125I-NeurotensinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85317IMR-32 CellsHUMAN125I-EpibatidineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85318CEREBRAL CORTEXRAT3H-CytisineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85319nAChRRD CellsHUMAN125I-Alpha-bgtTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85320nAChRBRAINRAT125I-Alpha-bgtTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85321DORrecombinantHUMAN3H-NaltrindoleTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85322DORBRAINGUINEA PIG3H-D-Penicillamine-enkephalinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85323KORrecombinantHUMAN3H-DiprenorphineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85324KORBRAINGUINEA PIG3H-U69,593Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85325MORrecombinantHUMAN3H-DiprenorphineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85326MORBRAINGUINEA PIG3H-EnkephalinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85327NOPrecombinantHUMAN3H-NociceptinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85328BRAINMOUSE3H-PDBUTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85329PAFPlateletsHUMAN3H-PAFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85330PAFPlateletsRABBIT3H-PAFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85331PDGF3T3 CellsMOUSE125I-PDGFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85332Potassium channelCEREBRAL CORTEXRAT125I-DendrotoxinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85333Potassium channelPancreatic HIT-T15 Beta CellsHAMSTER3H-GlyburideTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85334Potassium channelHIT-T15HAMSTER3H-GlyburideTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85335Potassium channelBRAINRAT125I-ApaminTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85336Potassium channelrecombinantHUMAN3H-AstemizoleTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85337UterusCALF3H-R-5020Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85338recombinantHUMAN3H-progesteroneTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85339Potassium channelrecombinantHUMAN3H-PGD2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85340recombinantHUMAN3H-PGD2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85341EP2recombinantHUMAN3H-PGE2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85342EP4recombinantHUMAN3H-PGE2Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85343recombinantHUMAN3H-SQ 29548Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85344P2XUrinary bladderRABBIT3H-alpha, beta-mATPTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85345P2YBRAINRAT35S-ATP-alphaSTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85346recombinantHUMAN3H-9-cis-Retinoic acidTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85347BRAINRAT3H-RolipramTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85348BRAINRAT3H-RyanodineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85349CEREBRAL CORTEXRAT3H-5HTTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853505-HT1ArecombinantHUMAN3H-8-OH-DPATTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853515-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853525-HT1BCEREBRAL CORTEXRAT125I-cyanopindololTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85353BRAINRAT3H-KETANSERINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853545-HT2ArecombinantHUMAN3H-KETANSERINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853555-HT2BrecombinantHUMAN3H-LSDTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853565-HT2CrecombinantHUMAN3H-MESULERGINETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853575-HT3recombinantHUMAN3H-GR-65630Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853585-HT3Ileum MuscularisRABBIT3H-GR-65630Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853595-HT4STRIATUMGUINEA PIG3H-GR-113808Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853605-HT5ArecombinantHUMAN3H-LSDTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853615-HT6recombinantHUMAN3H-LSDTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85362Sigma 1Jurkat cellsHUMAN3H-HaloperidolTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85363Sigma 1BRAINRAT3H-Pentazocine(+)Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85364Sigma 2BRAINRAT3H-IfenprodilTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85365BRAINGUINEA PIG3H-DTGTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85366Sodium ChannelBRAINRAT3H-BatrachotoxinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85367SST1recombinantHUMAN125I-SOMATOSTATIN 14Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85368SST2recombinantHUMAN125I-SOMATOSTATIN 14Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85369SST3recombinantHUMAN125I-SOMATOSTATIN 14Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85370SST4recombinantHUMAN125I-SOMATOSTATIN 14Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85371SST5recombinantHUMAN125I-SOMATOSTATIN 14Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85372NK1recombinantHUMAN3H-SR-140333Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85373NK2recombinantHUMAN3H-SR 48968Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85374NK3recombinantHUMAN125I-MePhe7-Neurokinin BTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85375Ventral ProstateRAT3H-miboleroneTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85376TPPlateletsRABBIT3H-SQ 29548Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85377LIVERRAT125I-TriiodothyronineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85378BRAINRAT3H-Me-TRHTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853793T3 Cells CCL-92MOUSE125I-TGF-beta1Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85380CEREBRAL CORTEXGUINEA PIG3H-NitrobenzylthioinosineTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85381STRIATUMRAT3H-Hemicholinium-3Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85382DATrecombinantHUMAN125I-RTI-55Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85383GABAACEREBRAL CORTEXRAT3H-GABATasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85384PlateletsRABBIT3H-KETANSERINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85385NETrecombinantHUMAN3H-RTI-55Tasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85386SERTrecombinantHUMAN3H-PAROXETINETasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 28, 2025
85387TNFU937 cellsHUMAN125I-TNF-alphaTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85388UTrecombinantHUMAN125I-Urotensin IITasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 29, 2025
85389Spinal cordRAT3H-ResiniferatoxinTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85390VEGFUmbilical Vein Endothelial CellsHUMAN125I-VEGFTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85391LUNGGUINEA PIG125I-VIPTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85392HT29 Colon Carcinoma CellsHUMAN125I-VIPTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85393V1ArecombinantHUMAN125I-PhenylacetylTyr(Me)PheGlnAsnArgProArgTyrTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85394V1BrecombinantHUMAN3H-VASOPRESSINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85395V2recombinantHUMAN3H-VASOPRESSINTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
85396recombinantHUMAN3H-1alpha, 25-Dihydroxyvitamin DTasimelteon>10000Lavedan C et al 2015Jan 15, 2025Jan 15, 2025
853975-HT1A?CLONED? HUMAN[3H] Way1006352-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole216Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
853985-HT2A?CLONED? HUMAN3H- Ketanserin2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole696Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85399SERT?CLONED? HUMAN3H-CITALOPRAM2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole34Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854005-HT2C?CLONED? HUMAN3H-MESULERGINE2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854015-HT7?CLONED? HUMAN3H- LSD2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole2060Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85402D2?CLONED? HUMAN3H-N-Methylspiperone2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85403D4?CLONED? HUMAN3H-N-Methylspiperone2-(3-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)propyl)benzo [d]thiazole431Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854045-HT1A?CLONED? HUMAN[3H] Way1006352-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole263Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854055-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole159Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854065-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole1420Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854075-HT7?CLONED? HUMAN3H-LSD2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole413Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85408SERT?CLONED? HUMAN3H-CITALOPRAM2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole65Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85409D2?CLONED? HUMAN3H-N-Methylspiperone2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole259Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85410D4?CLONED? HUMAN3H-N-Methylspiperone2-(4-(4-(4-Chlorophenyl)-1,4-diazepan-1-yl)butyl) benzo [d]thiazole28.6Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854115-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85412SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one5.3Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854135-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one1038Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854145-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854155-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one356Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85416D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one126Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85417D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854185-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one495Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85419SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one65Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854205-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one1003Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854215-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one5920Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854225-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one2810Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85423D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one1983Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85424D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)-1,4-diazepan-1-yl)pentan-1-one1215Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85425SERT?CLONED? HUMAN3H-CITALOPRAMFLUOXETINE1.1Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854265-HT2C?CLONED? HUMAN3H-MESULERGINEFLUOXETINE72Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854275-HT1A?CLONED? HUMAN[3H] Way100635Vilazodone0.3Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85428SERT?CLONED? HUMAN3H-CITALOPRAMVilazodone0.5Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85429D2?CLONED? HUMAN3H-N-MethylspiperoneVilazodone666Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854305-HT1A?CLONED? HUMAN[3H] Way1006352-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride312Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854315-HT2A?CLONED? HUMAN3H- Ketanserin2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride36Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854325-HT2C?CLONED? HUMAN3H-MESULERGINE2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride4647Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854335-HT7?CLONED? HUMAN3H-LSD2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride790Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85434D2?CLONED? HUMAN3H-Methylspiperone2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride2321Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85435D4?CLONED? HUMAN3H-Methylspiperone2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride31Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85436SERT?CLONED? HUMAN3H-CITALOPRAM2-(3-(4-(4-Chlorophenyl)piperazin-1-yl)propyl)benzo[d]thiazole hydrochloride1184Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854375-HT1A?CLONED? HUMAN[3H] Way1006352-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole90.5Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854385-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole132Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854395-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole6210Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854405-HT7?CLONED? HUMAN3H-LSD2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole329Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85441SERT?CLONED? HUMAN3H-CITALOPRAM2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole166Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85442D2?CLONED? HUMAN3H-N-Methylspiperone2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole219Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85443D4?CLONED? HUMAN3H-N-Methylspiperone2-(4-(4-(4-Chlorophenyl)piperazin-1-yl)butyl)benzo[d]thiazole4Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854445-HT1A?CLONED? HUMAN[3H] Way1006351-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol771Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854455-HT2A?CLONED? HUMAN3H- Ketanserin1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol4255Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854465-HT2C?CLONED? HUMAN3H-MESULERGINE1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854475-HT7?CLONED? HUMAN3H-LSD1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol983Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85448D2?CLONED? HUMAN3H-N-Methylspiperone1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol201Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85449D4?CLONED? HUMAN3H-N-Methylspiperone1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol140Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85450SERT?CLONED? HUMAN3H-CITALOPRAM1-(4-(Benzo[d]thiazol-2-yl)butyl)-4-(4-chlorophenyl)piperidin-4-ol922Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85451SERT?CLONED? HUMAN3H-CITALOPRAM2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854525-HT1A?CLONED? HUMAN[3H] Way1006352-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride6.6Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854535-HT2A?CLONED? HUMAN3H- Ketanserin2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride224Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854545-HT2C?CLONED? HUMAN3H-MESULERGINE2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854555-HT7?CLONED? HUMAN3H-LSD2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854565-HT7?CLONED? HUMAN3H-LSD2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride228.9Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85457D2?CLONED? HUMAN3H-N-Methylspiperone2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride26.5Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85458D4?CLONED? HUMAN3H-N-Methylspiperone2-[4-(4-Pyrimidin-2-yl-piperazin-1-yl)-butyl]-benzo[d]thiazole hydrochloride0.8Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854595-HT1A?CLONED? HUMAN[3H] Way1006352-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate5.1Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85460SERT?CLONED? HUMAN3H-CITALOPRAM2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate1325Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854615-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate3812Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854625-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate6265Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854635-HT7?CLONED? HUMAN3H-LSD2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate35.6Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85464D2?CLONED? HUMAN3H-N-Methylspiperone2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate30.8Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85465D4?CLONED? HUMAN3H-N-Methylspiperone2-(4-Benzo[d]thiazol-2-yl-butyl)-1,2,3,4-tetrahydro-isoquinoline p-toluenesulfonate65.5Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85466D4?CLONED? HUMAN3H-N-Methylspiperone2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride141Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85467D2?CLONED? HUMAN3H-N-Methylspiperone2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride990Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85468SERT?CLONED? HUMAN3H-CITALOPRAM2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride186Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854695-HT1A?CLONED? HUMAN[3H] Way1006352-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride111Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854705-HT7?CLONED? HUMAN3H- LSD2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride211Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854715-HT2A?CLONED? HUMAN3H- Ketanserin2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854725-HT2C?CLONED? HUMAN3H-MESULERGINE2-(4-(Isoindolin-2-yl)butyl)benzo[d]thiazole hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854735-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85474SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride491Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854755-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride1996Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854765-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854775-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85478D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride8355Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85479D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-(4-chlorophenyl)piperazin-1-yl)butan-1-one hydrochloride342Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85480D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85481D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854825-HT7?CLONED? HUMAN3H- LSD1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854835-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854845-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85485SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854865-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperazin-1-yl)-butan-1-one350Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854875-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride85Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85488SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride706Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854895-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride287Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854905-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854915-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride425.8Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85492D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride530Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85493D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-phenyl-piperidin-1-yl)-butan-1-one hydrochloride44.4Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85494D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride1522Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85495D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride51.5Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854965-HT1A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride63Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85497SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
854985-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride2206Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
854995-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855005-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-4-(4-pyrimidin-2-yl-piperazin-1-yl)-butan-1-one hydrochloride2467Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855015-HT1A?CLONED? HUMAN[3H] Way1006351-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one252Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85502SERT?CLONED? HUMAN3H-CITALOPRAM1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one565Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855035-HT2A?CLONED? HUMAN3H- Ketanserin1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one1564Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855045-HT7?CLONED? HUMAN3H- LSD1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one127Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855055-HT2C?CLONED? HUMAN3H-MESULERGINE1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85506D2?CLONED? HUMAN3H-N-Methylspiperone1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one217Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85507D4?CLONED? HUMAN3H-N-Methylspiperone1-(1-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)piperidin-4-yl)-5-chloro-1H-benzo[d]imidazol-2(3H)-one1710Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855085-HT1A?CLONED? HUMAN[3H] Way1006358-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one103Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85509SERT?CLONED? HUMAN3H-CITALOPRAM8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one284Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855105-HT2A?CLONED? HUMAN3H- Ketanserin8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one3720Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855115-HT7?CLONED? HUMAN3H- LSD8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one518Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85512D2?CLONED? HUMAN3H-N-Methylspiperone8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one25Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85513D4?CLONED? HUMAN3H-N-Methylspiperone8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one162Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855145-HT2C?CLONED? HUMAN3H-MESULERGINE8-(5-(Benzo[d]thiazol-2-yl)-5-oxopentyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855155-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride214Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85516SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride237Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855175-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855185-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855195-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride242Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85520D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride2931Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85521D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(isoindolin-2-yl)pentan-1-one hydrochloride512Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855225-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride28.3Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85523SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride81Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855245-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride523Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855255-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855265-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride2917Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85527D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride4793Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85528D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride100Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85529D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride346Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85530D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride505Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85531SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855325-HT2A?CLONED? HUMAN3H-KETANSERIN1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride6982Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855335-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855345-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-5-(4-pyrimidin-2-yl-piperazin-1-yl)-pentan-1-one hydrochloride337Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855355-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride3.6Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85536SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride298Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855375-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride204Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855385-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride2140Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855395-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride62.6Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85540D2?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride198Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85541D4?CLONED? HUMAN3H-N-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperazin-1-yl)-pentan-1-one hydrochloride105Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855425-HT1A?CLONED? HUMAN[3H] Way1006351-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride7.3Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85543SERT?CLONED? HUMAN3H-CITALOPRAM1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride64Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
855445-HT2A?CLONED? HUMAN3H- Ketanserin1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride3.4Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855455-HT2C?CLONED? HUMAN3H-MESULERGINE1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride3738Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
855465-HT7?CLONED? HUMAN3H-LSD1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride107Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85547D2?CLONED? HUMAN3H-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride642Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85548D4?CLONED? HUMAN3H-Methylspiperone1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride180Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85549NET?CLONED? HUMAN3H-Nisoxetine1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride49Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85550H1?CLONED? HUMAN3H-PYRILAMINE1-(Benzo[d]thiazol-2-yl)-5-(4-phenyl-piperidin-1-yl)-pentan-1-one hydrochloride52Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85551H1?CLONED? HUMAN3H-PYRILAMINE1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride46Zhu XY et al 2012Jan 15, 2025Jan 28, 2025
85552NET?CLONED? HUMAN3H-Nisoxetine1-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride>10000Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85553DAT?CLONED? HUMAN[3H] WIN354281-(Benzo[d]thiazol-2-yl)-5-(4-(4-chlorophenyl)piperazin-1-yl)pentan-1-one hydrochloride4742Zhu XY et al 2012Jan 15, 2025Jan 15, 2025
85554nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate0.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85555nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate233.4Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85556nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate2.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85557nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate6119Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85558nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate0.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85559nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate0.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85560nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(hydroxymethyl)cyclopropyl]pyridineTrifluoroacetate78.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85561nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate0.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85562nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate211.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85563nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate3.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85564nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate7514Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85565nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate0.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85566nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate0.4Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85567nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2S)-2-(3-hydroxypropyl)cyclopropyl]pyridine Trifluoroacetate88.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85568nAChRCLONEDHUMAN3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate0.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85569nAChRCLONEDHUMAN3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate318Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85570nAChRCLONEDHUMAN3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate10.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85571nAChRCLONEDHUMAN3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate4290Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85572nAChRCLONEDHUMAN3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate0.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85573nAChRFOREBRAINRAT3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate1.6Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85574nAChRCLONEDHUMAN3H-Epibatidine3-[(1S,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]propanoicAcid Trifluoroacetate75.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85575nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate1.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85576nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate20.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85577nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate17Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85578nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate612.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85579nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85580nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate3.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85581nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-trifluoromethoxyethyl)cyclopropyl]pyridine Trifluoroacetate4.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85582nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperidin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate15.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85583nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperidin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate224Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85584nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperidin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate11.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85585nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperidin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate9.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85586nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate14.9Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85587nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate>10000Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85588nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate403Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85589nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate4.6Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85590nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate10.4Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85591nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate2930Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85592nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate65.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85593nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate6.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85594nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate2.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85595nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate1.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85596nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1S,2R)-2-(2-(piperazin-1-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate6237Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85597nAChRCLONEDHUMAN3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate0.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85598nAChRCLONEDHUMAN3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate203Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85599nAChRCLONEDHUMAN3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate8.9Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85600nAChRCLONEDHUMAN3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate8830Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85601nAChRCLONEDHUMAN3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate0.4Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85602nAChRFOREBRAINRAT3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85603nAChRCLONEDHUMAN3H-EpibatidineEthyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate125Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85604nAChRCLONEDHUMAN3H-EpibatidineIsopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate0.6Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85605nAChRCLONEDHUMAN3H-EpibatidineIsopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate453Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85606nAChRCLONEDHUMAN3H-EpibatidineIsopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate11.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85607nAChRCLONEDHUMAN3H-EpibatidineIsopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate0.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85608nAChRFOREBRAINRAT3H-EpibatidineIsopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate1.4Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85609nAChRCLONEDHUMAN3H-EpibatidineIsopropyl [2-[(1R,2S)-2-[5-[((S)-Azetidin-2-yl)methoxy]pyridin-3-yl]cyclopropyl]ethyl]carbamate Trifluoroacetate158Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85610nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate89.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85611nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate7850Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85612nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate1190Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85613nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate56.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85614nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate91.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85615nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Azetidinyl)methoxy]-5-[(1R,2S)-2-(2-(morpholin-4-yl)ethyl)cyclopropyl]pyridine Trifluoroacetate2700Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85616nAChRCLONEDHUMAN3H-Epibatidine3-[2-(Isopropylamino)ethoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate2176Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85617nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85618nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate612Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85619nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate17.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85620nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.4Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85621nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate1.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85622nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate161Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85623nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate18.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85624nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate>10000Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85625nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate2534Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85626nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate38.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85627nAChRFOREBRAINRAT3H-Epibatidine3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate221Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85628nAChRCLONEDHUMAN3H-Epibatidine3-[(2(S)-Piperidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate>10000Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85629nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85630nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate129.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85631nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate21Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85632nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85633nAChRFOREBRAINRAT3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85634nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate584.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85635nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Ethyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate167.9Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85636nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Ethyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate49.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85637nAChRFOREBRAINRAT3H-Epibatidine3-[(1-Ethyl-2(S)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate173.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85638nAChRCLONEDHUMAN3H-Epibatidine3-[((1S,2S,5R)-3-Azabicyclo[3.1.0]hexan-2-yl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate43.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85639nAChRCLONEDHUMAN3H-Epibatidine3-[((1S,2S,5R)-3-Azabicyclo[3.1.0]hexan-2-yl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate2094Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85640nAChRCLONEDHUMAN3H-Epibatidine3-[((1S,2S,5R)-3-Azabicyclo[3.1.0]hexan-2-yl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate28.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85641nAChRFOREBRAINRAT3H-Epibatidine3-[((1S,2S,5R)-3-Azabicyclo[3.1.0]hexan-2-yl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate193.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85642nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate12.9Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85643nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate9959Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85644nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate472.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85645nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate21.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85646nAChRFOREBRAINRAT3H-Epibatidine3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate86.6Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85647nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(R)-pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate9475Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85648nAChRCLONEDHUMAN3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.04Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85649nAChRCLONEDHUMAN3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate50.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85650nAChRCLONEDHUMAN3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.8Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85651nAChRCLONEDHUMAN3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate2074Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85652nAChRCLONEDHUMAN3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.05Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85653nAChRFOREBRAINRAT3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate0.2Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85654nAChRCLONEDHUMAN3H-Epibatidine3-[(3(S)-Pyrrolidinyl)methoxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate30Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85655nAChRCLONEDHUMAN3H-Epibatidine3-[(3(R)-Pyrrolidinyl)oxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridineTrifluoroacetate6.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85656nAChRCLONEDHUMAN3H-Epibatidine3-[(3(R)-Pyrrolidinyl)oxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridineTrifluoroacetate191.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85657nAChRCLONEDHUMAN3H-Epibatidine3-[(3(R)-Pyrrolidinyl)oxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridineTrifluoroacetate90.9Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85658nAChRFOREBRAINRAT3H-Epibatidine3-[(3(R)-Pyrrolidinyl)oxy]-5-[(1S,2R)-2-(2-methoxyethyl)cyclopropyl]pyridineTrifluoroacetate40.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85659nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate3.5Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85660nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate546.6Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85661nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate137.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85662nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate3.3Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85663nAChRFOREBRAINRAT3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate15.7Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
85664nAChRCLONEDHUMAN3H-Epibatidine3-[(1-Methyl-2(S)-pyrrolidinyl)methoxy]-5-[(1R,2S)-2-(2-methoxyethyl)cyclopropyl]pyridine Trifluoroacetate234.1Zhang HK et al 2013Jan 15, 2025Jan 29, 2025
856655-HT1ACORTICAL MEMBRANESRAT3H-8-OH-DPATN-(2-(4-phenylpiperazin-1-yl)ethyl)picolinamide161Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856665-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-phenylpiperazin-1-yl)ethyl)picolinamide53.2Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856675-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-phenylpiperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856685-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856695-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide0.0224Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856705-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide599Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856715-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide138Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856725-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide9.33Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856735-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-methoxyphenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856745-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856755-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856765-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-ethoxyphenyl)piperazin-1-yl)ethyl)picolinamide55.4Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856775-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl)picolinamide74.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856785-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl)picolinamide616Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856795-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-cyanophenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856805-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl) picolinamide140Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856815-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl) picolinamide48.5Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856825-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl) picolinamide1320Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856835-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) picolinamide215Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856845-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856855-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2,3-dimethylphenyl)piperazin-1-yl)ethyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856865-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)picolinamide268Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856875-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856885-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-chlorophenyl)piperazin-1-yl)ethyl)picolinamide412Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856895-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)picolinamide267Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856905-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)picolinamide309Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856915-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(3-chlorophenyl)piperazin-1-yl)ethyl)picolinamide90.9Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856925-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide564Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856935-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide178Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856945-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-chlorophenyl)piperazin-1-yl)ethyl)isonicotinamide0.344Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856955-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide0.183Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856965-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide74.1Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856975-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(3,4-dichlorophenyl)piperazin-1-yl)ethyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856985-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
856995-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857005-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(2-fluorophenyl)piperazin-1-yl)ethyl)picolinamide158Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857015-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl)picolinamide82Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857025-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl)picolinamide241Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857035-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-fluorophenyl)piperazin-1-yl)ethyl)picolinamide79.4Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857045-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857055-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857065-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(pyridin-2-yl)piperazin-1-yl)ethyl)picolinamide32.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857075-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide0.046Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857085-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857095-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(pyrimidin-2-yl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857105-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(piperonyl)piperazin-1-yl)ethyl)picolinamide61.2Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857115-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(piperonyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857125-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(piperonyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857135-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(furoyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857145-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(furoyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857155-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(furoyl)piperazin-1-yl)ethyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857165-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) picolinamide49.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857175-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) picolinamide504Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857185-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(4-chlorobenzhydryl)piperazin-1-yl)ethyl) picolinamide540Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857195-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857205-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) picolinamide218Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857215-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)ethyl) picolinamide0.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857225-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl)picolinamide116Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857235-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl)picolinamide91.1Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857245-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(naphthalen-1-yl)piperazin-1-yl)ethyl)picolinamide20.8Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857255-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-phenylpiperazin-1-yl)propyl)picolinamide104Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857265-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-phenylpiperazin-1-yl)propyl)picolinamide277Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857275-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-phenylpiperazin-1-yl)propyl)picolinamide111Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857285-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) picolinamide128Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857295-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857305-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl) picolinamide40.1Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857315-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857325-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857335-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(4-methoxyphenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857345-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl)picolinamide80Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857355-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl)picolinamide119Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857365-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-ethoxyphenyl)piperazin-1-yl)propyl)picolinamide85.6Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857375-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl)picolinamide108Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857385-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl)picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857395-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-cyanophenyl)piperazin-1-yl)propyl)picolinamide128Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857405-HT2CFR. CORTEXRAT3H-MESULERGINEN-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857415-HT2AFR. CORTEXRAT3H-KETANSERINN-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857425-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)propyl) picolinamide17.9Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857435-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) picolinamide88.7Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857445-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) picolinamide1000Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857455-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl) picolinamide105Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857465-HT2CFR. CORTEXRAT3H-MESULERGINEN-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl)picolinamide1050Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857475-HT2AFR. CORTEXRAT3H-KETANSERINN-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl)picolinamide763Fiorino F et al 2017Jan 15, 2025Jan 15, 2025
857485-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATN-(3-(4-(2-chlorophenyl)piperazin-1-yl)propyl)picolinamide71.6Fiorino F et al 2017Jan 15, 2025Jan 15, 2025