67749 5-HT1A CEREBRAL CORTEX RAT 3H-8-OH-DPAT ICS 205930 >10000 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67750 5-HT2C Choroid Plexus PIG 3H-5-HT D,L-Trimipramine 537.032 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67751 5-HT2C Choroid Plexus PIG 3H-5-HT CLOZAPINE 3.98107 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67752 5-HT2C Choroid Plexus PIG 3H-5-HT 5-Hydroxy Tryptamine 8.51138 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67753 5-HT2C Choroid Plexus PIG 3H-5-HT MESULERGINE 1.38038 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67754 5-HT2C Choroid Plexus PIG 3H-5-HT KETANSERIN 199.526 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67755 5-HT1D STRIATUM PIG 3H-5-HT D,L-Trimipramine >10000 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67756 5-HT1D STRIATUM PIG 3H-5-HT CLOZAPINE 2089.3 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67757 5-HT1D STRIATUM PIG 3H-5-HT 5-Hydroxy Tryptamine 1.8197 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67758 5-HT1D STRIATUM PIG 3H-5-HT KETANSERIN >10000 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67759 5-HT1D STRIATUM PIG 3H-5-HT METERGOLINE 107.152 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67760 5-HT1D STRIATUM PIG 3H-5-HT ICS 205930 >10000 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67761 CEREBRAL CORTEX RAT 3H-KETANSERIN D,L-Trimipramine 19.4984 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67762 CEREBRAL CORTEX RAT 3H-KETANSERIN L-Trimipramine 16.2181 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67763 CEREBRAL CORTEX RAT 3H-KETANSERIN D-Trimipramine 104.713 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67764 CEREBRAL CORTEX RAT 3H-KETANSERIN CLOZAPINE 14.4544 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67765 CEREBRAL CORTEX RAT 3H-KETANSERIN KETANSERIN 1.02329 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67766 5-HT3 Entorhinal Cortex RAT 3H-GR65630 D,L-Trimipramine 9120.11 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67767 5-HT3 Entorhinal Cortex RAT 3H-GR65630 CLOZAPINE 100 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67768 5-HT3 Entorhinal Cortex RAT 3H-GR65630 5-Hydroxy Tryptamine 131.826 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67769 5-HT3 Entorhinal Cortex RAT 3H-GR65630 ICS 205930 8.31764 Weltrowska et al., 2010 Jan 15, 2025 Jan 15, 2025
67770 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 56 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67771 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 24 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67772 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 348 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67773 5-HT7 CLONED HUMAN 3H-5-CT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 51 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67774 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 10 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67775 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 28 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67776 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 29 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67777 5-HT6 CLONED HUMAN 3H-LSD (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 949 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67778 5-HT7 CLONED HUMAN 3H-5-CT (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 52 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67779 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67780 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 24 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67781 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 35 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67782 5-HT6 CLONED HUMAN 3H-LSD (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 1259 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67783 5-HT7 CLONED HUMAN 3H-5-CT (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 69 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67784 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67785 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 48 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67786 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 30 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67787 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 457 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67788 5-HT7 CLONED HUMAN 3H-5-CT (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 17 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67789 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67790 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 50 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67791 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 26 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67792 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 623 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67793 5-HT7 CLONED HUMAN 3H-5CT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67794 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67795 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline 9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67796 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67797 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline 130 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67798 5-HT7 CLONED HUMAN 3H-5-CT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline 45 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67799 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline 24 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67800 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline 16 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67801 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline 16 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67802 5-HT6 CLONED HUMAN 3H-LSD (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline 104 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67803 5-HT7 CLONED HUMAN 3H-5CT (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline 31 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67804 D2 CLONED HUMAN 3H-5CT (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline 29 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67805 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline 15 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67806 5-HT2B CLONED HUMAN 3H-KETANSERIN (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline 35 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67807 5-HT6 CLONED HUMAN 3H-LSD (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline 337 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67808 5-HT7 CLONED HUMAN 3H-5-CT (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline 22 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67809 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline 21 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67810 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl) 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67811 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl) 64 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67812 5-HT6 CLONED HUMAN 3H-LSD (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl) 221 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67813 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl) 32 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67814 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl) 23 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67815 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl) 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67816 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl) 51 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67817 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl) 176 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67818 5-HT7 CLONED HUMAN 3H-5-CT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl) 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67819 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl) 10 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67820 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline 8 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67821 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline 29 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67822 5-HT6 CLONED HUMAN 3H-LSD (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline 190 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67823 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline 24 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67824 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67825 5-HT1A CLONED HUMAN 3H-WAY100635 HALOPERIDOL 1703 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67826 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 23 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67827 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 2453 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67828 5-HT6 CLONED HUMAN 3H-LSD (S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 3912 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67829 5-HT7 CLONED HUMAN 3H-5-CT (S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 1119 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67830 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67831 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 27 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67832 5-HT2A CLONED HUMAN 3H-KETANSERIN S)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 2040 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67833 5-HT6 CLONED HUMAN 3H-LSD S)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 2990 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67834 5-HT7 CLONED HUMAN 3H-5-CT S)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 672 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67835 D2 CLONED HUMAN 3H-RACLOPRIDE S)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67836 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 36 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67837 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 1970 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67838 5-HT6 CLONED HUMAN 3H-LSD (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 1810 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67839 5-HT7 CLONED HUMAN 3H-5-CT (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 1340 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67840 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d] 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67841 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67842 5-HT2A CLONED HUMAN 3H-Ketaserin (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 110 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67843 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 2533 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67844 5-HT7 CLONED HUMAN 3H-5CT (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 349 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67845 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67846 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67847 5-HT7 CLONED HUMAN 3H-5-CT S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 142 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67848 5-HT2A CLONED HUMAN 3H-KETANSERIN S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 91 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67849 5-HT6 CLONED HUMAN 3H-LSD S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 1483 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67850 D2 CLONED HUMAN 3H-RACLOPRIDE S)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67851 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67852 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 296 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67853 5-HT6 CLONED HUMAN 3H-LSD (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 996 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67854 5-HT7 CLONED HUMAN 3H-5CT (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 66 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67855 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67856 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67857 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 390 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67858 5-HT6 CLONED HUMAN 3H-LSD (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 1263 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67859 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 52 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67860 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 22 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67861 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 146 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67862 5-HT2A CLONED HUMAN 3H-Ketaserin (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 1400 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67863 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 77 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67864 5-HT7 CLONED HUMAN 3H-5-CT (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 65 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67865 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl) 11 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67866 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 66 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67867 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 238 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67868 5-HT6 CLONED HUMAN 3H-LSD (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline ) 60 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67869 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline ) 97 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67870 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67871 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 91 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67872 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 1150 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67873 5-HT6 CLONED HUMAN 3H-LSD (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 18 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67874 5-HT7 CLONED HUMAN 3H-5-CT (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67875 D2 CLONED HUMAN 3H-5-CT (R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 15 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67876 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 147 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67877 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 1904 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67878 5-HT6 CLONED HUMAN 3H-LSD (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 23 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67879 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 8 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67880 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67881 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 147 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67882 5-HT2A CLONED HUMAN 3H-Ketaserin (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67883 5-HT6 CLONED HUMAN 3H-LSD 1-(Aminomethyl)dibenzo[b,e]bicyclo[2.2.2]octadiene Hydrochloride 169 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67884 5-HT7 CLONED HUMAN 3H-5CT (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67885 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 1.7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67886 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 111 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67887 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67888 5-HT6 CLONED HUMAN 3H-LSD (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 137 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67889 5-HT7 CLONED HUMAN 3H-5-CT (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 0.4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67890 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 0.1 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67891 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 120 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67892 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67893 5-HT6 CLONED HUMAN 3H-LSD (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 45 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67894 5-HT7 CLONED HUMAN 3H-5-CT (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67895 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole 2 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67896 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 25 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67897 5-HT2A CLONED HUMAN 3H-KETANSERIN S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 16 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67898 5-HT6 CLONED HUMAN 3H-LSD S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 311 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67899 5-HT7 CLONED HUMAN 3H-5-CT S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67900 D2 CLONED HUMAN 3H-RACLOPRIDE S)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 1 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67901 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 37 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67902 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67903 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 313 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67904 5-HT7 CLONED HUMAN 3H-5-CT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67905 D2 CLONED HUMAN 3H-R-ZACOPRIDE (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 0.14 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67906 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 37 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67907 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 18 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67908 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 360 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67909 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 0.5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67910 5-HT7 CLONED HUMAN 3H-5-CT (S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 12 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67911 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 24 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67912 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 21 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67913 5-HT6 CLONED HUMAN 3H-LSD (R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 38 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67914 5-HT7 CLONED HUMAN 3H-5-CT (R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 1 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67915 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 0.7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67916 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 14 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67917 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 10 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67918 5-HT6 CLONED HUMAN 3H-LSD (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 40 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67919 5-HT7 CLONED HUMAN 3H-5-CT (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67920 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 0.9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67921 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 16 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67922 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 15 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67923 5-HT6 CLONED HUMAN 3H-LSD (R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 40 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67924 5-HT7 CLONED HUMAN 3H-5CT (R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 1 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67925 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 0.3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67926 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 179 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67927 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 49 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67928 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 291 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67929 5-HT7 CLONED HUMAN 3H-5CT (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67930 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67931 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 96 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67932 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 33 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67933 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 497 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67934 5-HT7 CLONED HUMAN 3H-5-CT (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67935 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67936 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 86 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67937 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 41 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67938 5-HT6 CLONED HUMAN 3H-LSD (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 92 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67939 5-HT7 CLONED HUMAN 3H-5-CT (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 10 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67940 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole 3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67941 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67942 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 36 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67943 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 82 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67944 5-HT7 CLONED HUMAN 3H-5-CT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67945 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 16 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67946 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 18 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67947 5-HT2A CLONED HUMAN 3H-KETANSERIN S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67948 5-HT6 CLONED HUMAN 3H-LSD S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 116 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67949 5-HT7 CLONED HUMAN 3H-5-CT S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67950 D2 CLONED HUMAN 3H-RACLOPRIDE S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 11 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67951 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 10 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67952 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67953 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 72 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67954 5-HT7 CLONED HUMAN 3H-5CT (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 23 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67955 D2 CLONED HUMAN 3H-R-ZACOPRIDE (S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67956 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 15 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67957 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 56 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67958 5-HT6 CLONED HUMAN 3H-LSD (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67959 5-HT7 CLONED HUMAN 3H-5-CT (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 1 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67960 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67961 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 24 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67962 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 26 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67963 5-HT6 CLONED HUMAN 3H-LSD (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 11 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67964 5-HT7 CLONED HUMAN 3H-5-CT (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67965 D2 CLONED HUMAN 3H-R-ZACOPRIDE (R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67966 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67967 5-HT2A CLONED HUMAN 3H-KETANSERIN (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 19 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67968 5-HT6 CLONED HUMAN 3H-LSD (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 9 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67969 5-HT7 CLONED HUMAN 3H-5CT (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67970 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67971 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 14 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67972 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 244 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67973 5-HT6 CLONED HUMAN 3H-LSD (S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 2310 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67974 5-HT7 CLONED HUMAN 3H-5-CT (S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 165 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67975 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 42 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67976 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 8 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67977 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 82 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67978 5-HT6 CLONED HUMAN 3H-LSD (S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 2057 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67979 5-HT7 CLONED HUMAN 3H-5-CT (S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 75 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67980 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline 37 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67981 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67982 5-HT2A CLONED HUMAN 3H-Ketaserin (R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 451 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67983 5-HT6 CLONED HUMAN 3H-LSD (R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 641 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67984 5-HT7 CLONED HUMAN 3H-5CT (R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 14 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67985 D2 CLONED HUMAN 3H-RACLOPRIDE (R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline 8 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67986 5-HT1A CLONED HUMAN 3H-8-OH-DPAT R)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67987 5-HT2A CLONED HUMAN 3H-KETANSERIN R)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 76 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67988 5-HT6 CLONED HUMAN 3H-LSD R)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 766 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67989 5-HT7 CLONED HUMAN 3H-5-CT R)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67990 D2 CLONED HUMAN 3H-RACLOPRIDE R)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl) 3 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67991 5-HT2A CLONED HUMAN 3H-KETANSERIN HALOPERIDOL 89 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67992 5-HT6 CLONED HUMAN 3H-LSD HALOPERIDOL 1083 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67993 5-HT7 CLONED HUMAN 3H-5-CT HALOPERIDOL 408 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67994 D2 CLONED HUMAN 3H-RACLOPRIDE HALOPERIDOL 2 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
67995 5-HT1A CLONED HUMAN 3H-8-OH-DPAT CLOZAPINE 143 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67996 5-HT2A CLONED HUMAN 3H-KETANSERIN CLOZAPINE 13 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67997 5-HT6 CLONED HUMAN 3H-LSD CLOZAPINE 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67998 5-HT7 CLONED HUMAN 3H-5CT CLOZAPINE >10000 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
67999 D2 CLONED HUMAN 3H-RACLOPRIDE CLOZAPINE 71 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68000 5-HT1A CLONED HUMAN 3H-8-OH-DPAT RISPERIDONE 1169 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68001 5-HT2A CLONED HUMAN 3H-KETANSERIN RISPERIDONE 0.5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68002 5-HT6 CLONED HUMAN 3H-LSD RISPERIDONE 1107 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68003 5-HT7 CLONED HUMAN 3H-5-CT RISPERIDONE 0.4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68004 D2 CLONED HUMAN 3H-RACLOPRIDE RISPERIDONE 0.6 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68005 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Ziprasidone 2 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68006 5-HT2A CLONED HUMAN 3H-KETANSERIN Ziprasidone 1.7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68007 5-HT6 CLONED HUMAN 3H-LSD Ziprasidone 20 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68008 5-HT7 CLONED HUMAN 3H-5-CT Ziprasidone 5 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68009 D2 CLONED HUMAN 3H-RACLOPRIDE Ziprasidone 0.8 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68010 5-HT1A CLONED HUMAN 3H-8-OH-DPAT OLANZAPINE 3442 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68011 5-HT2A CLONED HUMAN 3H-KETANSERIN OLANZAPINE 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68012 5-HT6 CLONED HUMAN 3H-LSD OLANZAPINE 7 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68013 5-HT7 CLONED HUMAN 3H-5-CT OLANZAPINE 206 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68014 D2 CLONED HUMAN 3H-RACLOPRIDE OLANZAPINE 4 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68015 5-HT1A CLONED HUMAN 3H-8-OH-DPAT ARIPIPRAZOLE 30 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68016 5-HT2A CLONED HUMAN 3H-KETANSERIN ARIPIPRAZOLE 63 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68017 5-HT6 CLONED HUMAN 3H-LSD ARIPIPRAZOLE 89 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68018 5-HT7 CLONED HUMAN 3H-5-CT ARIPIPRAZOLE 44 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68019 D2 CLONED HUMAN 3H-RACLOPRIDE ARIPIPRAZOLE 0.8 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68020 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 54 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68021 5-HT2A CLONED HUMAN 3H-KETANSERIN (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 30 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68022 5-HT6 CLONED HUMAN 3H-LSD (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 344 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68023 5-HT7 CLONED HUMAN 3H-5-CT (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 57 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 15, 2025
68024 D2 CLONED HUMAN 3H-RACLOPRIDE (S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole 11 Zajdel, Pawel et. al, 2018 Jan 15, 2025 Jan 28, 2025
68025 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 10.9648 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68026 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 5248.07 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68027 CCK2 CLONED HUMAN 125I-BH-CCK-8 GW5823 1000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68028 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(Benzo[d]isoxazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 89.1251 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68029 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(Benzo[d]isoxazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide >10000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68030 CCK1 CLONED HUMAN 125I-BH-CCK-8 GW5823 22.9087 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68031 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 8.31764 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68032 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide >10000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68033 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 13.8038 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68034 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide >10000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68035 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(N-Methylindol-3-yl)methyl]-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 17.7828 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68036 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-terahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 13.1826 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68037 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-terahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide >10000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68038 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamideisopropyl 14.4544 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68039 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamideisopropyl 3630.78 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68040 CCK1 CLONED HUMAN 125I-BH-CCK-8 N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]acetamide 42.658 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68041 CCK2 CLONED HUMAN 125I-BH-CCK-8 N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]acetamide 2398.83 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68042 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(1-Benzyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 309.03 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68043 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(1-Benzyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide >10000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68044 CCK1 CLONED HUMAN 125I-BH-CCK-8 N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]acetamide 38.9045 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68045 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[2,4-Dioxo-5-phenyl-3-[(1H-pyrazolo[3,4-b]pyridin-4-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 112.202 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68046 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[2,4-Dioxo-5-phenyl-3-[(1H-pyrazolo[3,4-b]pyridin-4-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide >10000 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68047 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[2,4-Dioxo-5-phenyl-3-[(4,5,6,7-tetrahydro-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-N-(4-methoxyphenyl)acetamide 128.825 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68048 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[2,4-Dioxo-5-phenyl-3-[(4,5,6,7-tetrahydro-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-N-(4-methoxyphenyl)acetamide 2951.21 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68049 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(4-Fluoro-1H-indazol-3-yl)methyl]methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 17.378 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68050 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(4-Fluoro-1H-indazol-3-yl)methyl]methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 1698.24 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68051 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(5-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 42.658 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68052 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(5-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 2511.89 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68053 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(6-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide 29.5121 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68054 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(6-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide 588.844 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68055 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(7-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 20.893 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68056 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-[(7-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide 1047.13 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68057 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide 87.0964 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68058 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide 177.828 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68059 CCK1 CLONED HUMAN 125I-BH-CCK-8 N-(4-Fluorophenyl)-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropylacetamide 138.038 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68060 CCK2 CLONED HUMAN 125I-BH-CCK-8 N-(4-Fluorophenyl)-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropylacetamide 478.63 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68061 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[4-(trifluoromethyl)phenyl]acetamide 660.693 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68062 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[4-(trifluoromethyl)phenyl]acetamide 1659.59 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68063 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(3-methoxyphenyl)acetamide 478.63 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68064 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(3-methoxyphenyl)acetamide 190.546 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68065 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(2-methoxyphenyl)acetamide 1584.89 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68066 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(2-methoxyphenyl)acetamide 128.825 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68067 CCK1 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[3,4-(methylenedioxy)phenyl]acetamide 354.813 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68068 CCK2 CLONED HUMAN 125I-BH-CCK-8 2-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[3,4-(methylenedioxy)phenyl]acetamide 724.436 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68069 CCK1 CLONED HUMAN 125I-BH-CCK-8 N-Cyclopentyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-(4-methoxyphenyl)acetamide 16.9824 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68070 CCK2 CLONED HUMAN 125I-BH-CCK-8 N-Cyclopentyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-(4-methoxyphenyl)acetamide 776.247 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68071 CCK1 CLONED HUMAN 125I-BH-CCK-8 N-Cyclopropyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacetamide 524.807 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68072 CCK2 CLONED HUMAN 125I-BH-CCK-8 N-Cyclopropyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacetamide 25.1189 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68073 CCK1 CLONED HUMAN 125I-BH-CCK-8 N-tert-Butyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacetamide 891.251 Henke BR et al., 1997 Jan 15, 2025 Jan 15, 2025
68074 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY, human 0.08 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68075 Y1 CLONED Rhesus Monkey [125I] - Peptide YY PYY, human 0.22 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68076 Y1 CLONED Rhesus Monkey [125I] - Peptide YY PP, human 50 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68077 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY 3-36, human 55 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68078 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY 13-36, human 30 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68079 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY Leu31, Pro34, human 0.08 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68080 Y1 CLONED Rhesus Monkey [125I] - Peptide YY NPY D-Trp32, human 1000 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68081 Y1 CLONED Rhesus Monkey [125I] - Peptide YY BIBP3226 6.9 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68082 Y1 CLONED HUMAN [125I] - Peptide YY NPY, human 0.18 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68083 Y1 CLONED HUMAN [125I] - Peptide YY PYY, human 0.14 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68084 Y1 CLONED HUMAN [125I] - Peptide YY PP, human 19 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68085 Y1 CLONED HUMAN [125I] - Peptide YY NPY 3-36, human 50 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68086 Y1 CLONED HUMAN [125I] - Peptide YY NPY Leu31, Pro34, human 0.11 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68087 Y1 CLONED HUMAN [125I] - Peptide YY NPY D-Trp32, human 1000 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68088 Y1 CLONED HUMAN [125I] - Peptide YY BIBP3226 9.7 Gehlert DR, et al., 2001 Jan 15, 2025 Jan 15, 2025
68089 AMPA BRAIN RAT 3H-AMPA AMPA 40 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68090 AMPA BRAIN RAT 3H-AMPA thio-AMPA 1800 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68091 AMPA BRAIN RAT 3H-AMPA ATPA 2100 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68092 AMPA BRAIN RAT 3H-AMPA Thio-ATPA 630 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68093 AMPA BRAIN RAT 3H-AMPA (RS)-HIBO 1500 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68094 AMPA BRAIN RAT 3H-AMPA Br-HIBO 650 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68095 AMPA BRAIN RAT 3H-AMPA 2-Amino-3-(4-bromo-3-hydroxyisothiazol-5-yl)-propionic Acid Hyrochloride >10000 Matzen L, et.al., 1997 Jan 15, 2025 Jan 15, 2025
68096 M2 UNDEFINED UNDEFINED 3H-AF-DX384 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68097 M3 UNDEFINED UNDEFINED 3H-4-DAMP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68098 M4 UNDEFINED UNDEFINED 3H-4-DAMP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68099 M5 UNDEFINED UNDEFINED 3H-4-DAMP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68100 Alpha1A UNDEFINED UNDEFINED 3H-PRAZOSIN ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68101 Alpha1B UNDEFINED UNDEFINED 3H-PRAZOSIN ABT-594 890 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68102 Alpha1D UNDEFINED UNDEFINED 3H-PRAZOSIN ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68103 Alpha2B UNDEFINED UNDEFINED 3H-RAUWOLSCINE ABT-594 597 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68104 Alpha2A UNDEFINED UNDEFINED 3H-RAUWOLSCINE ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68105 Alpha2C UNDEFINED UNDEFINED 3H-RAUWOLSCINE ABT-594 342 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68106 5-HT1A UNDEFINED UNDEFINED 3H-8-OH-DPAT ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68107 5-HT1B UNDEFINED UNDEFINED 125I-CYP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68108 5-HT2A UNDEFINED UNDEFINED 125I-DOI ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68109 5-HT2C UNDEFINED UNDEFINED 3H-MESULERGINE ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68110 5-HT3 UNDEFINED UNDEFINED 3H-BRL 43694 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68111 5-HT6 UNDEFINED UNDEFINED 3H-LSD ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68112 5-HT7 UNDEFINED UNDEFINED 3H-LSD ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68113 A1 UNDEFINED UNDEFINED 3H-CCPA ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68114 UNDEFINED UNDEFINED 3H-CGS-21680 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68115 A3 UNDEFINED UNDEFINED 3H-AB-MECA ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68116 Beta1 UNDEFINED UNDEFINED 3H-CPG-12177 (-) ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68117 Beta2 UNDEFINED UNDEFINED 3H-CPG-12177 (-) ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 28, 2025
68118 Beta3 UNDEFINED UNDEFINED 125I-CYP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68119 D1 UNDEFINED UNDEFINED 3H-SCH23390 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68120 D2 UNDEFINED UNDEFINED 3H-SPIPERONE ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68121 D3 UNDEFINED UNDEFINED 3H-SPIPERONE ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68122 D4 UNDEFINED UNDEFINED 3H-SPIPERONE ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 27, 2025
68123 D5 UNDEFINED UNDEFINED 3H-SCH23390 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68124 KOR UNDEFINED UNDEFINED 3H-MUSCIMOL ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 27, 2025
68125 GABAB UNDEFINED UNDEFINED 3H-GABA(+50 mM isoguvacine to block GABAA) ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68126 H3 UNDEFINED UNDEFINED 3H-Alpha-Me-histamine-(R) ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68127 UNDEFINED UNDEFINED 3H-DTG ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68128 AT1 UNDEFINED UNDEFINED 3H-A II ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 28, 2025
68129 UNDEFINED UNDEFINED 125I-ANP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68130 UNDEFINED UNDEFINED 3H-V1-antagonist ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68131 B2 UNDEFINED UNDEFINED 3H-NPC 17731 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68132 CCK1 UNDEFINED UNDEFINED 3H-Devazepide ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68133 ETA UNDEFINED UNDEFINED 125I-Endothelin 1 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68134 GCCR UNDEFINED UNDEFINED 125I-Glucagon ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68135 UNDEFINED UNDEFINED 125I-Tyr11-somatostatin ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68136 Y1 UNDEFINED UNDEFINED 125I-Peptide YY ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68137 Y2 UNDEFINED UNDEFINED 125I-Peptide YY ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68138 NK1 UNDEFINED UNDEFINED 3H-SP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68139 NK2 UNDEFINED UNDEFINED 125I-NKA ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68140 NK3 UNDEFINED UNDEFINED 3H-SENKTIDE ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68141 UNDEFINED UNDEFINED 125I-Neurotensin ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68142 Calcium channel UNDEFINED UNDEFINED 3H-D-888 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 29, 2025
68143 Chloride channel UNDEFINED UNDEFINED 3H-TBPS ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68144 UNDEFINED UNDEFINED 125I-Charybdotoxin ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68145 UNDEFINED UNDEFINED 3H-TCP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68146 UNDEFINED UNDEFINED 3H-Saxitoxin ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68147 UNDEFINED UNDEFINED 3H-Batrachotoxinin ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68148 PBR UNDEFINED UNDEFINED 3H-PK11195 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68149 BZP UNDEFINED UNDEFINED FNZ ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68150 GlyR UNDEFINED UNDEFINED 3H-Strychnine ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 27, 2025
68151 AMPA UNDEFINED UNDEFINED 3H-AMPA ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68152 KA UNDEFINED UNDEFINED 3H-Kainic acid ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68153 NMDA UNDEFINED UNDEFINED 3H-MK-801 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68154 NMDA UNDEFINED UNDEFINED 3H-CGP39653 ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 28, 2025
68155 NET UNDEFINED UNDEFINED 3H-Nisoxetine ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68156 UNDEFINED UNDEFINED 3H-GABA ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68157 UNDEFINED UNDEFINED 3H-Choline Chloride ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68158 SLC6A3 UNDEFINED UNDEFINED 3H-BTCP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68159 UNDEFINED UNDEFINED 3H-NBTI ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68160 PDE1, PDE2, PDE3, PDE4 UNDEFINED UNDEFINED 3H-cAMP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68161 PDE5 UNDEFINED UNDEFINED 3H-cGMP ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68162 MOA UNDEFINED UNDEFINED Kynuramine ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 29, 2025
68163 MOA UNDEFINED UNDEFINED Benzylamine ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 29, 2025
68164 COS-1 UNDEFINED UNDEFINED Indomethacin ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68165 COX-2 UNDEFINED UNDEFINED Nimesulfide ABT-594 1000 Donnelly-Roberts DL, et al., 1998 Jan 15, 2025 Jan 15, 2025
68166 A1 BRAIN RAT 3H-cyclohexyladenosine CPA 0.59 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
68167 Striatal Membranes RAT 3H-NECA CPA 462 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
68168 A1 BRAIN RAT 3H-cyclohexyladenosine N6-(2-endo-norbornyl)-adenosine 0.42 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
68169 Striatal Membranes RAT 3H-NECA N6-(2-endo-norbornyl)-adenosine 750 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
68170 Striatal Membranes RAT 3H-NECA 2-exo-norbornyl isomer 970 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
68171 A1 BRAIN RAT 3H-cyclohexyladenosine 2-exo-norbornyl isomer 0.91 Trivedi BK et al., 1989 Jan 15, 2025 Jan 15, 2025
68172 CLONED RAT 3H-GLUTAMATE (S)-BrHlbo >10000 Thomsen C, et.al., 1994a Jan 15, 2025 Jan 15, 2025
68173 CLONED RAT [3H]AP4 (S)-BrHlbo 1000 Thomsen C, et.al., 1994a Jan 15, 2025 Jan 15, 2025
68174 CLONED RAT [3H]AP4 (R)-BrHlbo 1100 Thomsen C, et.al., 1994a Jan 15, 2025 Jan 15, 2025
68175 A1 BRAIN RAT 3H-PIA NB-Benzyladenosine-5-N-methyluronamide 898 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68176 A1 Striatal Membranes RAT 3H-CGS-21680 NB-Benzyladenosine-5-N-methyluronamide 597 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68177 Striatal Membranes RAT 3H-CGS-21680 NB-Benzyladenosine-5-N-methyluronamide 597 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68178 A3 CLONED RAT 125I-APNEA NB-Benzyladenosine-5-N-methyluronamide 16 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68179 A1 BRAIN RAT 3H-PIA M- (3-Iodoben zy1)adenosine- N-methyluronamide 54 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68180 Striatal Membranes RAT 3H-CGS-21680 M- (3-Iodoben zy1)adenosine- N-methyluronamide 56 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68181 A3 CLONED RAT 125I-APNEA M- (3-Iodoben zy1)adenosine- N-methyluronamide 1.1 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68182 A1 BRAIN RAT 3H-PIA N6-( 3-Aminobenzyl)adenosine-N-methyluronamide 1000 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68183 Striatal Membranes RAT 3H-CGS-21680 N6-( 3-Aminobenzyl)adenosine-5-N-methyluronamide 794 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68184 A3 CLONED RAT 125I-APNEA N6-( 3-Aminobenzyl)adenosine-5-N-methyluronamide 28 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68185 A1 BRAIN RAT 3H-PIA N6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide 2970 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68186 Striatal Membranes RAT 3H-CGS-21680 N6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide 988 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68187 A3 CLONED RAT 125I-APNEA N6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide 41.4 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68188 A1 BRAIN RAT 3H-PIA N6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide 496 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68189 Striatal Membranes RAT 3H-CGS-21680 N6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide 574 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68190 A3 CLONED RAT 125I-APNEA N6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide 31 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68191 A1 BRAIN RAT 3H-PIA N6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide 18 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68192 Striatal Membranes RAT 3H-CGS-21680 N6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide 197 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68193 A3 CLONED RAT 125I-APNEA N6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide 1.27 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68194 A1 BRAIN RAT 3H-PIA N6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt >10000 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68195 Striatal Membranes RAT 3H-CGS-21680 N6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt 9070 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68196 A3 CLONED RAT 125I-APNEA N6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt 1310 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68197 A3 CLONED RAT 125I-APNEA N6-( 4-Sulfobenzyl)adenosine-5-N-methyluronamide 4500 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68198 A1 BRAIN RAT 3H-PIA (R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide 3.2 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68199 Striatal Membranes RAT 3H-CGS-21680 (R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide 259 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68200 A3 CLONED RAT 125I-APNEA (R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide 18 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68201 A1 BRAIN RAT 3H-PIA (S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide 65 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68202 Striatal Membranes RAT 3H-CGS-21680 (S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide 1650 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68203 A3 CLONED RAT 125I-APNEA (S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide 494 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68204 A1 BRAIN RAT 3H-PIA N6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide 51 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68205 Striatal Membranes RAT 3H-CGS-21680 N6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide 32 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68206 A3 CLONED RAT 125I-APNEA N6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide 10.7 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68207 A1 BRAIN RAT 3H-PIA N6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide 22 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68208 Striatal Membranes RAT 3H-CGS-21680 N6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide 19 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68209 A3 CLONED RAT 125I-APNEA N6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide 1.1 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68210 A1 BRAIN RAT 3H-PIA N6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide 31 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68211 Striatal Membranes RAT 3H-CGS-21680 N6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide 24 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68212 A3 CLONED RAT 125I-APNEA N6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide 2.8 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68213 A1 BRAIN RAT 3H-PIA N6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide 78 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68214 Striatal Membranes RAT 3H-CGS-21680 N6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide 35 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68215 A3 Striatal Membranes RAT 125I-APNEA N6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide 8.7 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68216 A1 BRAIN RAT 3H-PIA N6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide 49 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68217 Striatal Membranes RAT 3H-CGS-21680 N6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide 574 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68218 A3 Striatal Membranes RAT 125I-APNEA N6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide 9 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68219 A3 BRAIN RAT 3H-PIA N6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide 209 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68220 A1 BRAIN RAT 3H-PIA N6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide 209 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68221 Striatal Membranes RAT 3H-CGS-21680 N6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide 609 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68222 A3 CLONED RAT 125I-APNEA N6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide 11 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68223 A3 CLONED RAT 125I-APNEA N6-Benzyladenosine-5-N-cyclopropyluronamide 103 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68224 Striatal Membranes RAT 3H-CGS-21680 N6-Benzyladenosine-5-N-cyclopropyluronamide 55 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68225 A1 BRAIN RAT 3H-PIA N6-Benzyladenosine-5-N-cyclopropyluronamide 112 Gallo-Rodriguez C et al., 1994 Jan 15, 2025 Jan 15, 2025
68226 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-2- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate 377 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68227 CCK2 PANCREAS RAT 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-2- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate 48 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68228 CCK2 PANCREAS RAT 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-1- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate 210 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68229 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-1- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate 785 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68230 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-2-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate 775 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68231 CCK2 PANCREAS RAT 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-2-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate 6.4 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68232 CCK2 PANCREAS RAT 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-1-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate 21.6 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68233 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Tricyclo[3.3.1.1-3,7]dec-1-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate 1040 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68234 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]- cyclohexyl ester 625 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68235 CCK2 PANCREAS RAT 125I-BH-CCK-8 carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]- cyclohexyl ester 517 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68236 CCK2 PANCREAS RAT 125I-BH-CCK-8 carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]-2-chlorocyclohexyl ester trans (+/-) 49 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68237 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]-2-chlorocyclohexyl ester trans (+/-) 196 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68238 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester 66 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68239 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester 15 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68240 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester (isomer I) 140 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68241 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester (isomer I) 118 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68242 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester 288 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68243 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester 36 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68244 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S) 149 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68245 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S) 251 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68246 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S)[(-)-isomer] 266 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68247 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S)[(-)-isomer] 23 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68248 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester 16 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68249 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester 66 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68250 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1S-[1 alpha [S*(R*)], 2 beta]] 75 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68251 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1S-[1 alpha [S*(R*)], 2 beta]] 73 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68252 CCK2 PANCREAS RAT 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1R-[1 alpha [R*(S*)], 2 beta]] 9.3 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68253 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1R-[1 alpha [R*(S*)], 2 beta]] 288 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68254 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 2-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1S-[1 alpha[S*R*(E)]],-2beta]] 47 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68255 CCK2 PANCREAS RAT 125I-BH-CCK-8 2-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1S-[1 alpha[S*R*(E)]],-2beta]] 6.5 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68256 CCK2 PANCREAS RAT 125I-BH-CCK-8 2-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*(E)]],-2beta]] 1.2 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68257 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 2-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*(E)]],-2beta]] 154 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68258 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]] 391 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68259 CCK2 PANCREAS RAT 125I-BH-CCK-8 Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]] 13 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68260 CCK2 PANCREAS RAT 125I-BH-CCK-8 Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]] 3.9 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68261 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]] 1810 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68262 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta(E)]] 511 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68263 CCK2 PANCREAS RAT 125I-BH-CCK-8 Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta(E)]] 4 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68264 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring centers are trans (+/-)) 0.6 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68265 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring centers are trans (+/-)) 8.9 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68266 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1S-trans) 3.9 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68267 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1S-trans) 4.2 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68268 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1-R-trans) 0.34 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68269 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1-R-trans) 18 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68270 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans) 12 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68271 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans) 815 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68272 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans) 1260 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68273 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-( 1-S- trans) 1260 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68274 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-( 1-S- trans) 20 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68275 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl) 7.9 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68276 CCK2 PANCREAS RAT 125I-BH-CCK-8 Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl) 1160 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68277 CCK1 CEREBRAL CORTEX RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester 0.15 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68278 CCK1 CEREBRAL CORTEX RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester 25.5 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68279 CCK2 PANCREAS RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester 0.15 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68280 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester 25.5 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68281 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl) 186 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68282 CCK2 PANCREAS RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl) 9.3 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68283 CCK2 PANCREAS RAT 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-L-3(phenylmethyl) 13.2 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68284 CCK1 CEREBRAL CORTEX MOUSE 125I-BH-CCK-8 beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-L-3(phenylmethyl) 539 Boden PR et al., 1993 Jan 15, 2025 Jan 15, 2025
68285 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)glycine 14 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68286 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)glycine 1518 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68287 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-D-tryptophanyl]-N-(2-phenylethyl)glycine 224 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68288 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-D-tryptophanyl]-N-(2-phenylethyl)glycine 2842 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68289 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-2-phenylethylamine 87 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68290 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-2-phenylethylamine 1889 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68291 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)-3-aminopropionic Acid 36 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68292 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)-3-aminopropionic Acid 1323 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68293 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]glycine 986 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68294 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]glycine 4000 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68295 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]aniline 407 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68296 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]aniline 6082 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68297 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]benzylamine 231 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68298 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]benzylamine 4097 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68299 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](3-phenylpropyl)amine 182 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68300 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](3-phenylpropyl)amine 4249 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68301 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](2-naphthyl)amine 402 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68302 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](2-naphthyl)amine 2356 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68303 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(1-naphthyl)ethyl]amine 89 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68304 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(1-naphthyl)ethyl]amine 2367 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68305 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(1-naphthyl)alaninyl]-N-(2-phenylethyl)glycine 134 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68306 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(1-naphthyl)alaninyl]-N-(2-phenylethyl)glycine 2013 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68307 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methylphenyl-alaninyl]-N-(2-phenylethyl)glycine 87 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68308 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methylphenyl-alaninyl]-N-(2-phenylethyl)glycine 3798 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68309 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(2-naphthyl)alaninyl]-N-(2-phenylethyl)glycine 70 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68310 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(2-naphthyl)alaninyl]-N-(2-phenylethyl)glycine 3006 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68311 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(4-bromophenyl)alaninyl]-N-(2-phenylethyl)glycine 50 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68312 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(4-bromophenyl)alaninyl]-N-(2-phenylethyl)glycine 3414 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68313 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(4-Chlorophenyl)-DL-a-methyltryptophanyl][(2phenylethyl)amino]urea >10000 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68314 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(4-Chlorophenyl)-DL-a-methyltryptophanyl][(2phenylethyl)amino]urea 6329 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68315 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-methoxyphenyl)ethyl]amine 115 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68316 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-methoxyphenyl)ethyl]amine 3121 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68317 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-chlorophenyl)ethyl]amine 39 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68318 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-chlorophenyl)ethyl]amine 1614 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68319 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(3,4-dichlorophenyl)ethyl]amine 184 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68320 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(3,4-dichlorophenyl)ethyl]amine 1540 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68321 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-bromophenyl)ethyl]amine 51 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68322 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-bromophenyl)ethyl]amine 2141 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68323 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(2,4-dichlorophenyl)ethyl]amine 27 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68324 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(2,4-dichlorophenyl)ethyl]amine 3161 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68325 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-nitrophenyl)ethyl]amine 79 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68326 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-nitrophenyl)ethyl]amine 2352 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68327 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine 6.5 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68328 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine 1129 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68329 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-D-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine 6.1 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68330 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-D-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine 1060 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68331 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-L-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine 36 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68332 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-L-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine 1039 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68333 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(2,4-dichlorophenyl)ethyl]glycine 12.3 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68334 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(2,4-dichlorophenyl)ethyl]glycine 3045 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68335 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Naphthyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea 3478 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68336 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Naphthyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea 769 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68337 CCK2 BRAIN GUINEA PIG 3H-pCCK8 N-[(2-Triphenylmethyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea >10000 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68338 CCK1 PANCREAS GUINEA PIG 3H-pCCK8 N-[(2-Triphenylmethyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea 1777 Blommaert AG et al., 1993 Jan 15, 2025 Jan 15, 2025
68339 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 5.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68340 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 4.9 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68341 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 4.3 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68342 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine Free Janty EC Liquid 167.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68343 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine Free NicVape EC Liquid 886.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68344 nAChR BRAIN RAT 3H-Epibatidine Nicotine 9.3 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68345 nAChR BRAIN RAT 3H-Epibatidine Janty EC Liquid 9 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68346 nAChR BRAIN RAT 3H-Epibatidine NicVape EC Liquid 7.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68347 nAChR BRAIN RAT 3H-Epibatidine Nicotine Free Janty EC Liquid 267.1 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68348 nAChR BRAIN RAT 3H-Epibatidine Nicotine Free NicVape EC Liquid 1890 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68349 nAChR7 KIDNEY HUMAN 3H-Epibatidine Nicotine 208.7 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68350 nAChR7 KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 277.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68351 nAChR7 KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 352.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68352 nAChR7 BRAIN RAT 3H-Epibatidine Nicotine 9.2 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68353 nAChR7 BRAIN RAT 3H-Epibatidine Janty EC Liquid 6.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68354 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 303.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68355 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 288.4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68356 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 307.1 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68357 nAChR7 BRAIN RAT 3H-Epibatidine NicVape EC Liquid 6.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68358 nAChR7 BRAIN RAT 3H-Epibatidine Nicotine Free Janty EC Liquid 178 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68359 nAChR7 BRAIN RAT 3H-Epibatidine Nicotine Free NicVape EC Liquid 1008 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68360 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 4 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68361 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 3.8 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68362 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 4.8 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68363 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine Free Janty EC Liquid 111.9 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68364 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine Free NicVape EC Liquid 681.9 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68365 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 73.3 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68366 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 52.8 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68367 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 88.7 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68368 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 7.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68369 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 6.9 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68370 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 6.1 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68371 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine Free Janty EC Liquid 258.5 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68372 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine Free NicVape EC Liquid 1603 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68373 nAChR KIDNEY HUMAN 3H-Epibatidine Nicotine 22.6 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68374 nAChR KIDNEY HUMAN 3H-Epibatidine Janty EC Liquid 23.2 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68375 nAChR KIDNEY HUMAN 3H-Epibatidine NicVape EC Liquid 23.8 Harris, AC. et, al. 2018 Jan 15, 2025 Jan 29, 2025
68376 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68377 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68378 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68379 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.25893 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68380 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 6.60693 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68381 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68382 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 67.6083 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68383 5-HT1A CLONED HUMAN 3H-8-OH-DPAT 1-hydroxyindane 1.62181 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68384 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 23.4423 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68385 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 1.25893 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68386 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 6.60693 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68387 5-HT1A CLONED HUMAN 3H-8-OH-DPAT (-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-01 1.02329 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68388 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piperazine 1.28825 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68389 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 22.9087 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68390 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-01 0.831764 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68391 5-HT1A CLONED HUMAN 3H-8-OH-DPAT cis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 4-hydroxy piperid-1-yl] 5-fluoroindan-1-01 1000 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68392 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperid-1-yl] indan-1-01 0.707946 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68393 5-HT1A CLONED HUMAN 3H-8-OH-DPAT Piperidine 0.288403 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68394 5-HT1A CLONED HUMAN 3H-8-OH-DPAT trans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) piperid-1-yl] 6-nitroindan-1-01 0.74131 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68395 5-HT1A CLONED HUMAN 3H-8-OH-DPAT S 15535 0.794328 Peglion JL, et.al., 2002 Jan 15, 2025 Jan 15, 2025
68396 Alpha1A CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 182 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68397 Alpha2A CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 0.13 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68398 Alpha2B CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 1.03 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68399 Alpha2C CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 0.15 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68400 D2 CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 81 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68401 D3 CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 228 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68402 D4 CLONED HUMAN [11C[R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 158 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68403 5-HT1A CLONED HUMAN [11C[R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 1478 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68404 5-HT1B CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 1286 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68405 5-HT1D CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 48 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68406 5-HT1E CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 3330 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68407 5-HT1F CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 1678 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68408 5-HT2A CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 434 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68409 5-HT2C CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 97 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68410 5-HT4 CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 1003 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 27, 2025
68411 5-HT5A CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 352 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68412 5-HT6 CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 3056 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68413 5-HT7 CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 5 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68414 CLONED RAT [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 5118 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68415 CLONED HUMAN [11C]R107474 2-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one 1412 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68416 Alpha1A CLONED HUMAN [C11]R107474 mirtazapine 1815 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68417 Alpha2A CLONED HUMAN [C11]R107474 mirtazapine 20 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68418 Alpha2B CLONED HUMAN [11C]R107474 mirtazapine 88 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68419 Alpha2C CLONED HUMAN [11C]R107474 mirtazapine 18 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68420 Beta1 CLONED HUMAN [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68421 Beta2 CLONED HUMAN [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68422 Beta3 CLONED HUMAN [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68423 D1 CLONED RAT [11C]R107474 mirtazapine 4167 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68424 D2 CLONED HUMAN [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68425 D3 CLONED HUMAN [11C]R107474 mirtazapine 5723 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68426 D4 CLONED HUMAN [11C]R107474 mirtazapine 2518 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68427 5-HT1A CLONED HUMAN [11C]R107474 mirtazapine 3334 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68428 5-HT1B CLONED HUMAN [11C]R107474 mirtazapine 3534 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68429 5-HT1D CLONED HUMAN [11C]R107474 mirtazapine 955 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68430 5-HT1E CLONED HUMAN [11C]R107474 mirtazapine 728 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68431 5-HT1F CLONED HUMAN [11C]R107474 mirtazapine 583 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68432 5-HT2A CLONED HUMAN [11C]R107474 mirtazapine 70 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68433 5-HT2C CLONED HUMAN [11C]R107474 mirtazapine 40 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68434 5-HT3 CLONED MOUSE [11C]R107474 mirtazapine 170 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68435 5-HT4 CLONED HUMAN [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 27, 2025
68436 5-HT5A CLONED HUMAN [11C]R107474 mirtazapine 670 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68437 5-HT7 CLONED HUMAN [11C]R107474 mirtazapine 265 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68438 H1 CLONED HUMAN [11C]R107474 mirtazapine 1.6 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68439 CLONED RAT [11C]R107474 mirtazapine 1100 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68440 CLONED RAT [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68441 CLONED RAT [11C]R107474 mirtazapine 6905 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68442 SLC6A3 CLONED RAT [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68443 SERT CLONED RAT [11C]R107474 mirtazapine >10000 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 28, 2025
68444 NET CLONED RAT [11C]R107474 mirtazapine 1640 Van der Mey. et, al. 2006 Jan 15, 2025 Jan 15, 2025
68445 5-HT1A CLONED HUMAN 3H-WAY100635 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68446 5-HT1B CLONED HUMAN 3H-5CT N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68447 5-HT1D CLONED HUMAN 3H-5CT N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68448 5-HT1E CLONED HUMAN 3H-5HT N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68449 5-HT2A CLONED HUMAN 3H-KETANSERIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68450 5-HT2C CLONED HUMAN 3H-MESULERGINE N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68451 5-HT2B CLONED HUMAN 3H-LSD N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 415 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68452 5-HT3 CLONED HUMAN 3H-GR-65630 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68453 5-HT5A CLONED HUMAN 3H-LSD N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68454 5-HT6 CLONED HUMAN 3H-LSD N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68455 5-HT7 CLONED HUMAN 3H-LSD N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68456 Alpha1A CLONED HUMAN 3H-PRAZOSIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68457 Alpha1B CLONED HUMAN 3H-PRAZOSIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68458 Alpha1D CLONED HUMAN 3H-PRAZOSIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68459 Alpha2A CLONED HUMAN 3H-RAUWOLSCINE N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 1416 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68460 Alpha2C CLONED HUMAN 3H-RAUWOLSCINE N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 575 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68461 Alpha2B CLONED HUMAN 3H-RAUWOLSCINE N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68462 Beta1 CLONED HUMAN 125I-Iodopindolol N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68463 Beta3 CLONED HUMAN 125I-Iodopindolol N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68464 Beta2 CLONED HUMAN 3H-CPG-12177 (-) N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68465 BZP CLONED HUMAN FNZ N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68466 D1 CLONED HUMAN 3H-SCH23390 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68467 D5 CLONED HUMAN 3H-SCH23390 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68468 D2 CLONED HUMAN 3H-N-Methylspiperone N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68469 D3 CLONED HUMAN 3H-N-Methylspiperone N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68470 D4 CLONED HUMAN 3H-N-Methylspiperone N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68471 DAT CLONED HUMAN 3H-WIN35428 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68472 DOR CLONED HUMAN 3H-DADLE N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68473 KOR CLONED HUMAN 3H-MUSCIMOL N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 27, 2025
68474 H1 CLONED HUMAN 3H-PYRILAMINE N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68475 5-HT1D CLONED HUMAN 125I-aminopotentidine N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 443 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68476 H3 CLONED HUMAN 3H-Alpha-methylhistamine N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68477 H4 CLONED HUMAN 3H-Histamine N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68478 KOR CLONED HUMAN 3H-U69,593 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 1208 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68479 M1 CLONED HUMAN 3H-QNB N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68480 M2 CLONED HUMAN 3H-QNB N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68481 M3 CLONED HUMAN 3H-QNB N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68482 M4 CLONED HUMAN 3H-QNB N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68483 M5 CLONED HUMAN 3H-QNB N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 1749 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68484 mGluR5 CLONED HUMAN 3H-MPEP N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68485 MOR CLONED HUMAN 3H-DAMGO N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68486 NET CLONED HUMAN 3H-Nisoxetine N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 1289 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68487 OT CLONED HUMAN 3H-Oxytocin N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68488 PBR CLONED HUMAN 3H-PK11195 N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68489 SERT CLONED HUMAN 3H-CITALOPRAM N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 2495 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68490 Sigma 1 CLONED HUMAN 3H-Pentazocine(+) N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 1806 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68491 Sigma 2 CLONED HUMAN 3H-DTG N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide 984 He, S. et, al. 2017 Jan 15, 2025 Jan 28, 2025
68492 V1A CLONED HUMAN 3H-VASOPRESSIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68493 V1B CLONED HUMAN 3H-VASOPRESSIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68494 V2 CLONED HUMAN 3H-VASOPRESSIN N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide >10000 He, S. et, al. 2017 Jan 15, 2025 Jan 15, 2025
68495 5-HT3 CLONED HUMAN 3H-GR-65630 Ondansetron HCl 3.6 PDSP Certified Data Jan 15, 2025 Jan 15, 2025
68496 BRAIN RAT 3H-RAUWOLSCINE (+-)Org3770 112.202 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68497 BRAIN RAT 3H-RAUWOLSCINE (+)Org3770 63.0957 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68498 BRAIN RAT 3H-RAUWOLSCINE (-)Org3770 2344.23 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68499 BRAIN RAT 3H-RAUWOLSCINE (+-)Mianserin 109.648 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68500 BRAIN RAT 3H-RAUWOLSCINE (+)Mianserin 57.544 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68501 BRAIN RAT 3H-RAUWOLSCINE (-)Mianserin 363.078 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68502 BRAIN RAT 3H-MIANSERIN (+-)Org3770 8.91251 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68503 BRAIN RAT 3H-MIANSERIN (+)Org3770 4.7863 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68504 BRAIN RAT 3H-MIANSERIN (-)Org3770 60.256 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68505 BRAIN RAT 3H-MIANSERIN (+-)Mianserin 0.363078 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68506 BRAIN RAT 3H-MIANSERIN (+)Mianserin 0.416869 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68507 BRAIN RAT 3H-MIANSERIN (-)Mianserin 18.6209 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68508 D2 BRAIN RAT 3H-SPIPERONE (+-)Org3770 3981.07 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68509 D2 BRAIN RAT 3H-SPIPERONE (+)Org3770 5011.87 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68510 D2 BRAIN RAT 3H-SPIPERONE (-)Org3770 3981.07 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68511 D2 BRAIN RAT 3H-SPIPERONE (+-)Mianserin >10000 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68512 H1 BRAIN RAT 3H-MEPYRAMINE (+-)Org3770 0.501187 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68513 H1 BRAIN RAT 3H-MEPYRAMINE (+)Org3770 0.316228 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68514 H1 BRAIN RAT 3H-MEPYRAMINE (-)Org3770 0.630957 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68515 H1 BRAIN RAT 3H-MEPYRAMINE (+-)Mianserin 1.77828 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68516 H1 BRAIN RAT 3H-MEPYRAMINE (+)Mianserin 1 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68517 BRAIN RAT 3H-QNB (+)Mianserin 3981.07 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68518 BRAIN RAT 3H-QNB (-)Mianserin 151.356 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68519 BRAIN RAT 3H-QNB (+-)Mianserin 501.187 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68520 BRAIN RAT 3H-QNB (+-)Org3770 794.328 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68521 BRAIN RAT 3H-QNB (+)Org3770 7079.46 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68522 BRAIN RAT 3H-QNB (-)Org3770 251.189 De Boer TH, et al., 1988 Jan 15, 2025 Jan 15, 2025
68523 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-fluorobenzamide 10.1 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68524 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-fluorobenzamide 1.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68525 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-fluorobenzamide 8.8 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68526 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-fluorobenzamide 1.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68527 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-fluorobenzamide 6.1 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68528 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-fluorobenzamide 1 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68529 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-chlorobenzamide 10.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68530 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-chlorobenzamide 1.3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68531 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-chlorobenzamide 15 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68532 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-chlorobenzamide 2.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68533 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-chlorobenzamide 17.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68534 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-chlorobenzamide 2.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68535 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-iodobenzamide 10.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68536 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-iodobenzamide 3.8 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68537 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-iodobenzamide 28.1 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68538 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-iodobenzamide 3.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68539 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-iodobenzamide 35.4 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68540 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-iodobenzamide 3.4 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68541 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-methoxy-benzamide 3.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68542 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-methoxy-benzamide 0.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68543 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-methoxy-benzamide 39.1 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68544 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-methoxy-benzamide 3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68545 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-methoxy-benzamide 30.4 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68546 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-methoxy-benzamide 1.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68547 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-hydroxy-benzamide 6.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68548 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-hydroxy-benzamide 0.8 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68549 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-hydroxy-benzamide 13.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68550 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-hydroxy-benzamide 0.4 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68551 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-nitrobenzamide 7.4 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68552 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-nitrobenzamide 3.4 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68553 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-nitrobenzamide 21.9 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68554 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-nitrobenzamide 2.3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68555 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-nitrobenzamide 19.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68556 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-nitrobenzamide 0.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68557 D2 CLONED HUMAN 125I-IABN 2-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 18.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68558 D3 CLONED HUMAN 125I-IABN 2-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 2.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68559 D2 CLONED HUMAN 125I-IABN 3-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 29 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68560 D3 CLONED HUMAN 125I-IABN 3-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide 2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68561 D2 CLONED HUMAN 125I-IABN Pyridine-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 16.9 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68562 D3 CLONED HUMAN 125I-IABN Pyridine-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 2.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68563 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-nicotinamide 19.6 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68564 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-nicotinamide 2.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68565 D2 CLONED HUMAN 125I-IABN Pyridine-4-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 31.2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68566 D3 CLONED HUMAN 125I-IABN Pyridine-4-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 2 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68567 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide 93.3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68568 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide 0.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68569 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide 54.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68570 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide 0.9 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68571 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-4-yl-benzamide 43.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68572 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-4-yl-benzamide 0.9 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68573 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyrimidin-2-yl-benzamide 45.7 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68574 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyrimidin-2-yl-benzamide 1.3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68575 D2 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-(1H-imidazol-2-yl)-benzamide 8 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68576 D3 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-(1H-imidazol-2-yl)-benzamide 0.3 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68577 D2 CLONED HUMAN 125I-IABN Quinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 65.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68578 D3 CLONED HUMAN 125I-IABN Quinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 3.8 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68579 D2 CLONED HUMAN 125I-IABN Benzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 149 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68580 D3 CLONED HUMAN 125I-IABN Benzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 1.1 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68581 D2 CLONED HUMAN 125I-IABN 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 76.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68582 D3 CLONED HUMAN 125I-IABN 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 1.5 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68583 D4 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide 375 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68584 D4 CLONED HUMAN 125I-IABN N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide 520 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68585 D4 CLONED HUMAN 125I-IABN Quinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 1110 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68586 D4 CLONED HUMAN 125I-IABN Benzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 1770 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68587 D4 CLONED HUMAN 125I-IABN 2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide 1070 Grundt P, et al., 2005 Jan 15, 2025 Jan 15, 2025
68588 nAChR Striatal Membranes RAT 3H-NICOTINE N-methylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68589 nAChR Striatal Membranes RAT 3H-NICOTINE N-ethylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68590 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-propylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68591 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-butylpyridinium iodide 9650 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68592 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-pentylpyridinium iodide 8720 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68593 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-hexylpyridinium iodide 9070 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68594 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-heptylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68595 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-octylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68596 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-nonylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68597 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-decylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68598 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-undecylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68599 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-dodecylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68600 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-pentadecylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68601 nAChR Striatal Membranes RAT 3H-NICOTINE N-n-eicosylpyridinium iodide >10000 Grinevich VP, et al., 2003 Jan 15, 2025 Jan 15, 2025
68602 recombinant HUMAN 3H-AdoMet SKF 29661 550 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68603 recombinant HUMAN 3H-AdoMet p-chlorophenyl moiety 2600 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68604 recombinant HUMAN 3H-AdoMet 7-((N-Methylamino)sulfonyl)-1,2,3,4-tetrahydroisoquinoline 4600 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68605 recombinant HUMAN 3H-AdoMet 7-(N-(Methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline 4800 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68606 recombinant HUMAN 3H-AdoMet 7-(N,N-Bis(methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68607 recombinant HUMAN 3H-AdoMet 7-((N-(Methylsulfonyl)amino)methyl)-1,2,3,4-tetrahydroisoquinoline >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68608 recombinant HUMAN 3H-AdoMet 8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 980 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68609 recombinant HUMAN 3H-AdoMet 1-(Aminomethyl)-6-methoxynaphthalene 1500 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68610 recombinant HUMAN 3H-AdoMet 1-(Aminomethyl)-6-hydroxynaphthalene 8400 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68611 recombinant HUMAN 3H-AdoMet 8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 1400 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68612 CORTEX RAT 3H-CLONIDINE SKF 29661 >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68613 CORTEX RAT 3H-CLONIDINE p-chlorophenyl moiety 6300 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68614 CORTEX RAT 3H-CLONIDINE 7-((N-Methylamino)sulfonyl)-1,2,3,4-tetrahydroisoquinoline >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68615 CORTEX RAT 3H-CLONIDINE 7-(N-(Methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68616 CORTEX RAT 3H-CLONIDINE 7-(N,N-Bis(methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68617 CORTEX RAT 3H-CLONIDINE 7-((N-(Methylsulfonyl)amino)methyl)-1,2,3,4-tetrahydroisoquinoline >10000 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68618 CORTEX RAT 3H-CLONIDINE 8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 78 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68619 CORTEX RAT 3H-CLONIDINE 1-(Aminomethyl)-6-methoxynaphthalene 4600 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68620 CORTEX RAT 3H-CLONIDINE 1-(Aminomethyl)-6-hydroxynaphthalene 2100 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68621 CORTEX RAT 3H-CLONIDINE 8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline 840 Grunewald GL, et al., 1997 Jan 15, 2025 Jan 15, 2025
68622 UT CLONED HUMAN I125-urotensin II U-II (H-Glu-Thr-Pro-Asp-cyclo[Cys-Phe-Trp-Lys-Tyr-Cys]-Val-OH) 0.794328 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68623 UT CLONED HUMAN I125-urotensin II H-U-II(4-11)-Asp-C[Cys-Phe-Trp-Lys-Tyr-Cys]Val-OH 0.251189 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68624 UT CLONED HUMAN I125-urotensin II H-P5U-Asp-C[Pen-Phe-Trp-Lys-Tyr-Cys]Val-OH 0.199526 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68625 UT CLONED HUMAN I125-urotensin II H-Asp-C[Pen-Phe-DTrp-Lys-Tyr-Cys]Val-OH 1.25893 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68626 UT CLONED HUMAN I125-urotensin II H-Asp-C[Cys-Phe-DTrp-Lys-Tyr-Cys]Val-OH 1.25893 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68627 UT CLONED HUMAN I125-urotensin II H-Asp-C[Pen-Phe-Trp-Orn-Tyr-Cys]Val-OH 15.8489 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68628 UT CLONED HUMAN I125-urotensin II H-Asp-C[Cys-Phe-Trp-Orn-Tyr-Cys]Val-OH 10 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68629 UT CLONED HUMAN I125-urotensin II H-Asp-C[Pen-Phe-DTrp-Orn-Tyr-Cys]Val-OH 5.01187 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68630 UT CLONED HUMAN I125-urotensin II H-Asp-C[Cys-Phe-DTrp-Orn-Tyr-Cys]Val-OH 12.5893 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68631 UT CLONED HUMAN I125-urotensin II H-Asp-C[DPen-Phe-DTrp-Orn-Tyr-Cys]Val-OH 1995.26 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68632 UT CLONED HUMAN I125-urotensin II H-Asp-C[Pen-Phe-DTrp-DOrn-Tyr-Cys]Val-OH 398.107 Grieco P, et al., 2005 Jan 15, 2025 Jan 29, 2025
68633 recombinant HUMAN UNKNOWN Brassinin >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68634 recombinant HUMAN UNKNOWN N-[2-(Indol-3-yl)ethyl]-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68635 recombinant HUMAN UNKNOWN N-[2-(Benzo[b]thiophen-3-yl)ethyl]-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68636 recombinant HUMAN UNKNOWN N-[3-(Indol-3-yl)propyl]-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68637 recombinant HUMAN UNKNOWN N-(Indan-2-yl)-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68638 recombinant HUMAN UNKNOWN N-(Adamant-2-yl)-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68639 recombinant HUMAN UNKNOWN N-[(Naphth-2-yl)methyl]-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68640 recombinant HUMAN UNKNOWN N-Benzyl-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68641 recombinant HUMAN UNKNOWN N-Phenethyl-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68642 recombinant HUMAN UNKNOWN N-4-Fluorophenethyl-S-methyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68643 recombinant HUMAN UNKNOWN N,S-Dimethyl-N-phenethyldithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68644 recombinant HUMAN UNKNOWN S-Allyl-brassinin >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68645 recombinant HUMAN UNKNOWN S-Benzyl-brassinin >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68646 recombinant HUMAN UNKNOWN S-Hexyl-brassinin >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68647 recombinant HUMAN UNKNOWN N-[2-(Indol-3-yl)ethyl]-S-benzyl-dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68648 recombinant HUMAN UNKNOWN N-[2-(Indol-3-yl)ethyl]-S-[(naphth-2-yl)methyl]dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68649 recombinant HUMAN UNKNOWN N-[2-(Indol-3-yl)ethyl]-S-[(pyrid-3-yl)methyl]dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68650 recombinant HUMAN UNKNOWN N-[2-(Indol-3-yl)ethyl]-S-[(pyrid-4-yl)methyl]dithiocarbamate >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68651 recombinant HUMAN UNKNOWN N-[1-(Indol-3-yl)ethyl]-N'-methyl-thiourea >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68652 recombinant HUMAN UNKNOWN N-[(Indol-3-yl)methyl]propanethioamide >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68653 recombinant HUMAN UNKNOWN 4-[(Indol-3-yl)methyl]thiazole >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68654 recombinant HUMAN UNKNOWN 4-[(Indol-3-yl)methyl]-2-methyl-thiazole >10000 Gaspari P, et al., 2006 Jan 15, 2025 Jan 15, 2025
68655 DOR BRAIN RAT 3H-DPDPE DPI-5201 150.3 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68656 DOR BRAIN RAT 3H-DPDPE DPI-673 384.7 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68657 DOR BRAIN RAT 3H-DPDPE DPI-5402 12.7 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68658 DOR BRAIN RAT 3H-DPDPE DPI-5336 41.8 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68659 DOR BRAIN RAT 3H-DPDPE DPI-5337 429.9 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68660 DOR BRAIN RAT 3H-DPDPE DPI-5701 119.3 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68661 DOR BRAIN RAT 3H-DPDPE DPI-5702 3.8 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68662 MOR BRAIN RAT 3H-DAMGO DPI-3290 0.46 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68663 MOR BRAIN RAT 3H-DAMGO DPI-5201 1000 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68664 MOR BRAIN RAT 3H-DAMGO DPI-673 64.4 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68665 MOR BRAIN RAT 3H-DAMGO DPI-5402 7.3 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68666 MOR BRAIN RAT 3H-DAMGO DPI-5336 6.4 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68667 MOR BRAIN RAT 3H-DAMGO DPI-5337 320.2 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68668 MOR BRAIN RAT 3H-DAMGO DPI-5701 405.5 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68669 MOR BRAIN RAT 3H-DAMGO DPI-5702 11.6 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68670 KOR BRAIN RAT 3H-U69,593 DPI-3290 0.62 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68671 KOR BRAIN RAT 3H-U69,593 DPI-673 306.8 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68672 KOR BRAIN RAT 3H-U69,593 DPI-5402 13.8 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68673 KOR BRAIN RAT 3H-U69,593 DPI-5336 414.2 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68674 KOR BRAIN RAT 3H-U69,593 DPI-5337 1000 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68675 KOR BRAIN RAT 3H-U69,593 DPI-5701 231.4 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68676 KOR BRAIN RAT 3H-U69,593 DPI-5702 19.1 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68677 DOR BRAIN RAT 3H-DPDPE DPI-3290 0.18 Gengo PJ, et.al.,2003 Jan 15, 2025 Jan 15, 2025
68678 5-HT5A CLONED HUMAN 3H-5CT 5-Hydroxy Tryptamine 126 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68679 5-HT5A CLONED MOUSE I125-2-iodo LSD 2-Br LSD 2 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68680 5-HT5A CLONED MOUSE I125-2-iodo LSD METHYSERGIDE 63 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68681 5-HT5A CLONED HUMAN 3H-5CT METERGOLINE 630 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68682 5-HT5A CLONED HUMAN 3H-5CT 5-CT 20 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68683 5-HT5A CLONED HUMAN 3H-5CT SUMATRIPTAN 5000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68684 5-HT5A CLONED HUMAN 3H-5CT 8-OH-DPAT 2500 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68685 5-HT5A CLONED MOUSE 3H-LSD 2-Methyl 5-HT >10000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68686 5-HT5A CLONED HUMAN 3H-5CT METHIOTHEPIN 1 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68687 5-HT5A CLONED HUMAN 3H-5CT KETANSERIN >10000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68688 5-HT5A CLONED MOUSE 3H-LSD QUIPAZINE >10000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68689 5-HT5A CLONED MOUSE 3H-LSD 1-NP 40 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68690 5-HT5A CLONED HUMAN 3H-5CT SPIPERONE >10000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68691 5-HT5A CLONED HUMAN 3H-5CT CLOZAPINE 1000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68692 5-HT6 CLONED HUMAN 3H-LSD 5-Hydroxy Tryptamine 65 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68693 5-HT6 CLONED HUMAN 125I-2-iodo LSD 2-Br LSD 17 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68694 5-HT6 CLONED HUMAN 3H-LSD METHYSERGIDE 180 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68695 5-HT6 CLONED HUMAN 3H-LSD METERGOLINE 400 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68696 5-HT6 CLONED HUMAN 3H-LSD 5-CT 720 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68697 5-HT6 CLONED HUMAN 3H-LSD SUMATRIPTAN 2600 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68698 5-HT6 CLONED HUMAN 3H-LSD 8-OH-DPAT >10000 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68699 5-HT6 CLONED HUMAN 125I-2-iodo LSD 2-Methyl 5-HT 400 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68700 5-HT6 CLONED HUMAN 3H-LSD METHIOTHEPIN 0.4 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68701 5-HT6 CLONED HUMAN 3H-LSD KETANSERIN 2800 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68702 5-HT6 CLONED HUMAN 3H-LSD QUIPAZINE 3600 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68703 5-HT6 CLONED HUMAN 125I-2-iodo LSD 1-NP 104 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68704 5-HT6 CLONED HUMAN 3H-LSD SPIPERONE 1595 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68705 5-HT6 CLONED HUMAN 3H-LSD CLOZAPINE 9.5 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68706 5-HT6 CLONED HUMAN 3H-LSD MIANSERIN 55 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68707 5-HT7 CLONED HUMAN 3H-5HT 5-Hydroxy Tryptamine 8.1 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68708 5-HT7 CLONED HUMAN 3H-5HT 2-Br LSD 30 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68709 5-HT7 CLONED HUMAN 3H-5HT METHYSERGIDE 83 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68710 5-HT7 CLONED HUMAN 3H-5HT METERGOLINE 6.4 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68711 5-HT7 CLONED HUMAN 3H-5HT 5-CT 0.9 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68712 5-HT7 CLONED HUMAN 3H-5HT SUMATRIPTAN 950 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68713 5-HT7 CLONED HUMAN 3H-5HT 8-OH-DPAT 466 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68714 5-HT7 CLONED HUMAN 3H-LSD 2-Methyl 5-HT 1258 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68715 5-HT7 CLONED HUMAN 3H-5HT METHIOTHEPIN 3.7 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68716 5-HT7 CLONED HUMAN 3H-5HT KETANSERIN 1334 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68717 5-HT7 CLONED HUMAN 3H-LSD QUIPAZINE 3033 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68718 5-HT7 CLONED HUMAN 3H-5HT 1-NP 83 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68719 5-HT7 CLONED HUMAN 3H-5HT SPIPERONE 110 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68720 5-HT7 CLONED HUMAN 3H-LSD CLOZAPINE 40 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68721 5-HT7 CLONED HUMAN 3H-5HT MIANSERIN 8010 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68722 5-HT7 CLONED RAT 3H-5HT SPIPERONE 10 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68723 5-HT7 CLONED MOUSE 3H-5HT SPIPERONE 63 Glennon RA, 2003 Jan 15, 2025 Jan 15, 2025
68724 D1 KIDNEY Monkey 3H-SCH23390 SCH 23390 0.6 Grandy DK, et al., 1991 Jan 15, 2025 Jan 15, 2025
68725 D1 KIDNEY Monkey 3H-SCH23390 BUTACLAMOL,(+) 9.1 Grandy DK, et al., 1991 Jan 15, 2025 Jan 15, 2025
68726 D1 KIDNEY Monkey 3H-SCH23390 cis-flupenthixol 23.6 Grandy DK, et al., 1991 Jan 15, 2025 Jan 15, 2025
68727 D1 KIDNEY Monkey 3H-SCH23390 HALOPERIDOL 156 Grandy DK, et al., 1991 Jan 15, 2025 Jan 15, 2025
68728 D1 KIDNEY Monkey 3H-SCH23390 CLOZAPINE 406 Grandy DK, et al., 1991 Jan 15, 2025 Jan 15, 2025
68729 D1 KIDNEY Monkey 3H-SCH23390 BUTACLAMOL, (-) >10000 Grandy DK, et al., 1991 Jan 15, 2025 Jan 15, 2025
68730 M5 CLONED HUMAN 3H-NMS xanomeline >10000 Grant MK, et al., 2005 Jan 15, 2025 Jan 15, 2025
68731 CRF1 CLONED HUMAN 125I-Sauvagine Antalarmin 3.1 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68732 CRF1 CLONED HUMAN 125I-Sauvagine 1-(2,4-Dichloro-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 5.1 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68733 CRF1 CLONED HUMAN 125I-Sauvagine 1-(2-Bromo-4-isopropyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 1.1 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68734 CRF1 CLONED HUMAN 125I-Sauvagine 1-(4-Chloro-phenyl)-7-methyl-5-(1-propylbutyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 12 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68735 CRF1 CLONED HUMAN 125I-Sauvagine 1-(4-Methanesulfonyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 460 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68736 CRF1 CLONED HUMAN 125I-Sauvagine 1-(4-Methoxycarbonyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 920 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68737 CRF1 CLONED HUMAN 125I-Sauvagine 1-(4-Methoxy-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 2 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68738 CRF1 CLONED HUMAN 125I-Sauvagine 1-(5-Chloro-pyridin-2-yl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 23 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68739 CRF1 CLONED HUMAN 125I-Sauvagine 1-(6-Methoxy-pyridin-3-yl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 60 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68740 CRF1 CLONED HUMAN 125I-Sauvagine 5-Isopropyl-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one >10000 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68741 CRF1 CLONED HUMAN 125I-Sauvagine 5-Butyl-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 8800 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68742 CRF1 CLONED HUMAN 125I-Sauvagine 5-(1-Ethyl-propyl)-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 8 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68743 CRF1 CLONED HUMAN 125I-Sauvagine 5-(1-Methoxymethyl-propyl)-1-(4-methoxyphenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 150 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68744 CRF1 CLONED HUMAN 125I-Sauvagine 5-(1-Ethyl-propyl)-7-methyl-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 170 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68745 CRF1 CLONED HUMAN 125I-Sauvagine 5-(1-Ethyl-propyl)-1-(4-methoxy-2-methyl-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one 20 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68746 CRF1 CLONED HUMAN 125I-Sauvagine 1-(4-Chloro-phenyl)-5-(1-methoxymethyl-propyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one trifluoroacetate 200 Guo Z, et al., 2005 Jan 15, 2025 Jan 15, 2025
68747 5-HT4 CAUDATE PIG 3H-GR-113808 GR 125487 0.19 Schiavi, GB et al., 1994 Jan 15, 2025 Jan 15, 2025
68748 5-HT4 CAUDATE PIG 3H-GR-113808 GR 113808 0.32 Schiavi, GB et al., 1994 Jan 15, 2025 Jan 15, 2025