The KᵢDB allows you to filter and search for various scientific entities, including receptors, sources, species, hot ligands, test ligands, and citations.

You can customize your search by selecting multiple items or using specific Kᵢ values for more targeted results.

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Showing 65,001-66,000 of 98,685 items.

Kᵢ Database

Kᵢ IDReceptorsSourcesSpeciesHot LigandsTest LigandsKᵢ ValueCitationsSubmitted AtUpdated At 
677495-HT1ACEREBRAL CORTEXRAT3H-8-OH-DPATICS 205930>10000Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677505-HT2CChoroid PlexusPIG3H-5-HTD,L-Trimipramine537.032Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677515-HT2CChoroid PlexusPIG3H-5-HTCLOZAPINE3.98107Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677525-HT2CChoroid PlexusPIG3H-5-HT5-Hydroxy Tryptamine8.51138Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677535-HT2CChoroid PlexusPIG3H-5-HTMESULERGINE1.38038Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677545-HT2CChoroid PlexusPIG3H-5-HTKETANSERIN199.526Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677555-HT1DSTRIATUMPIG3H-5-HTD,L-Trimipramine>10000Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677565-HT1DSTRIATUMPIG3H-5-HTCLOZAPINE2089.3Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677575-HT1DSTRIATUMPIG3H-5-HT5-Hydroxy Tryptamine1.8197Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677585-HT1DSTRIATUMPIG3H-5-HTKETANSERIN>10000Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677595-HT1DSTRIATUMPIG3H-5-HTMETERGOLINE107.152Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677605-HT1DSTRIATUMPIG3H-5-HTICS 205930>10000Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
67761CEREBRAL CORTEXRAT3H-KETANSERIND,L-Trimipramine19.4984Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
67762CEREBRAL CORTEXRAT3H-KETANSERINL-Trimipramine16.2181Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
67763CEREBRAL CORTEXRAT3H-KETANSERIND-Trimipramine104.713Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
67764CEREBRAL CORTEXRAT3H-KETANSERINCLOZAPINE14.4544Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
67765CEREBRAL CORTEXRAT3H-KETANSERINKETANSERIN1.02329Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677665-HT3Entorhinal CortexRAT3H-GR65630D,L-Trimipramine9120.11Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677675-HT3Entorhinal CortexRAT3H-GR65630CLOZAPINE100Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677685-HT3Entorhinal CortexRAT3H-GR656305-Hydroxy Tryptamine131.826Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677695-HT3Entorhinal CortexRAT3H-GR65630ICS 2059308.31764Weltrowska et al., 2010Jan 15, 2025Jan 15, 2025
677705-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole56Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677715-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole24Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677725-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole348Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677735-HT7CLONEDHUMAN3H-5-CT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole51Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67774D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole10Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
677755-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole28Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677765-HT2ACLONEDHUMAN3H-KETANSERIN(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole29Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677775-HT6CLONEDHUMAN3H-LSD(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole949Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677785-HT7CLONEDHUMAN3H-5-CT(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole52Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67779D2CLONEDHUMAN3H-RACLOPRIDE(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
677805-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole24Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677815-HT2ACLONEDHUMAN3H-KETANSERIN(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole35Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677825-HT6CLONEDHUMAN3H-LSD(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole1259Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677835-HT7CLONEDHUMAN3H-5-CT(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole69Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67784D2CLONEDHUMAN3H-RACLOPRIDE(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)piperidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
677855-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole48Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677865-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole30Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677875-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole457Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677885-HT7CLONEDHUMAN3H-5-CT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole17Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67789D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
677905-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole50Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677915-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole26Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677925-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole623Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677935-HT7CLONEDHUMAN3H-5CT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67794D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)azepan-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
677955-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677965-HT2ACLONEDHUMAN3H-KETANSERIN(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677975-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline130Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
677985-HT7CLONEDHUMAN3H-5-CT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline45Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67799D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)quinoline24Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678005-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline16Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678015-HT2ACLONEDHUMAN3H-KETANSERIN(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline16Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678025-HT6CLONEDHUMAN3H-LSD(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline104Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678035-HT7CLONEDHUMAN3H-5CT(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline31Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67804D2CLONEDHUMAN3H-5CT(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azetidin-1-yl)sulfonyl)isoquinoline29Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678055-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline15Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678065-HT2BCLONEDHUMAN3H-KETANSERIN(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline35Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678075-HT6CLONEDHUMAN3H-LSD(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline337Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678085-HT7CLONEDHUMAN3H-5-CT(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline22Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67809D2CLONEDHUMAN3H-RACLOPRIDE(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)quinoline21Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678105-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678115-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)64Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678125-HT6CLONEDHUMAN3H-LSD(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)221Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678135-HT7CLONEDHUMAN3H-5-CT(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)32Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67814D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)piperidin-1-yl)sulfonyl)23Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678155-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678165-HT2ACLONEDHUMAN3H-KETANSERIN(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)51Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678175-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)176Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678185-HT7CLONEDHUMAN3H-5-CT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67819D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)10Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678205-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline8Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678215-HT2ACLONEDHUMAN3H-KETANSERIN(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline29Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678225-HT6CLONEDHUMAN3H-LSD(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline190Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678235-HT7CLONEDHUMAN3H-5-CT(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline24Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67824D2CLONEDHUMAN3H-RACLOPRIDE(S)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)azepan-1-yl)sulfonyl)isoquinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678255-HT1ACLONEDHUMAN3H-WAY100635HALOPERIDOL1703Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678265-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]23Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678275-HT2ACLONEDHUMAN3H-KETANSERIN(S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]2453Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678285-HT6CLONEDHUMAN3H-LSD(S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]3912Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678295-HT7CLONEDHUMAN3H-5-CT(S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]1119Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67830D2CLONEDHUMAN3H-RACLOPRIDE(S)-7-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678315-HT1ACLONEDHUMAN3H-8-OH-DPATS)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one27Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678325-HT2ACLONEDHUMAN3H-KETANSERINS)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one2040Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678335-HT6CLONEDHUMAN3H-LSDS)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one2990Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678345-HT7CLONEDHUMAN3H-5-CTS)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one672Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67835D2CLONEDHUMAN3H-RACLOPRIDES)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]oxazol-2(3H)-one5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678365-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]36Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678375-HT2ACLONEDHUMAN3H-KETANSERIN(R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]1970Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678385-HT6CLONEDHUMAN3H-LSD(R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]1810Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678395-HT7CLONEDHUMAN3H-5-CT(R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]1340Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67840D2CLONEDHUMAN3H-RACLOPRIDE(R)-7-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)benzo[d]12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678415-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678425-HT2ACLONEDHUMAN3H-Ketaserin(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline110Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678435-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline2533Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678445-HT7CLONEDHUMAN3H-5CT(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline349Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67845D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl-pyrrolidin-1-yl)sulfonyl)quinoline13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678465-HT1ACLONEDHUMAN3H-8-OH-DPATS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678475-HT7CLONEDHUMAN3H-5-CTS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline142Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678485-HT2ACLONEDHUMAN3H-KETANSERINS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline91Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678495-HT6CLONEDHUMAN3H-LSDS)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline1483Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67850D2CLONEDHUMAN3H-RACLOPRIDES)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678515-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678525-HT2ACLONEDHUMAN3H-KETANSERIN(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline296Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678535-HT6CLONEDHUMAN3H-LSD(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline996Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678545-HT7CLONEDHUMAN3H-5CT(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline66Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67855D2CLONEDHUMAN3H-RACLOPRIDE(R)-5-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678565-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678575-HT2ACLONEDHUMAN3H-Ketaserin(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline390Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678585-HT6CLONEDHUMAN3H-LSD(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline1263Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678595-HT7CLONEDHUMAN3H-5-CT(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline52Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67860D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-((2-(2-(4-(2,3-Dihydrobenzo[b][1,4]dioxin-5-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline22Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678615-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)146Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678625-HT2ACLONEDHUMAN3H-Ketaserin(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)1400Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678635-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)77Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678645-HT7CLONEDHUMAN3H-5-CT(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)65Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67865D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)11Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678665-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline66Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678675-HT2ACLONEDHUMAN3H-KETANSERIN(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline238Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678685-HT6CLONEDHUMAN3H-LSD(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline )60Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678695-HT7CLONEDHUMAN3H-5-CT(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethylpyrrolidin-1-yl)sulfonyl)isoquinoline )97Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67870D2CLONEDHUMAN3H-RACLOPRIDE(S)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678715-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline91Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678725-HT2ACLONEDHUMAN3H-KETANSERIN(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline1150Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678735-HT6CLONEDHUMAN3H-LSD(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline18Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678745-HT7CLONEDHUMAN3H-5-CT(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67875D2CLONEDHUMAN3H-5-CT(R)-5-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline15Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678765-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline147Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678775-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline1904Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678785-HT6CLONEDHUMAN3H-LSD(R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline23Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678795-HT7CLONEDHUMAN3H-5-CT(R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline8Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67880D2CLONEDHUMAN3H-RACLOPRIDE(R)-4-((2-(2-(4-(5-Chloro-1H-indol-3-yl)-5,6-dihydropyridin-1(2H)-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678815-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole147Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678825-HT2ACLONEDHUMAN3H-Ketaserin(S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678835-HT6CLONEDHUMAN3H-LSD 1-(Aminomethyl)dibenzo[b,e]bicyclo[2.2.2]octadiene Hydrochloride169Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678845-HT7CLONEDHUMAN3H-5CT(S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67885D2CLONEDHUMAN3H-RACLOPRIDE(S)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole1.7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678865-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole111Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678875-HT2ACLONEDHUMAN3H-KETANSERIN(S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678885-HT6CLONEDHUMAN3H-LSD(S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole137Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678895-HT7CLONEDHUMAN3H-5-CT(S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole0.4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67890D2CLONEDHUMAN3H-RACLOPRIDE(S)-6-Fluoro-3-(1-(2-(1-(isoquinolin-4-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole0.1Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678915-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole120Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678925-HT2ACLONEDHUMAN3H-KETANSERIN(R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678935-HT6CLONEDHUMAN3H-LSD(R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole45Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678945-HT7CLONEDHUMAN3H-5-CT(R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67895D2CLONEDHUMAN3H-RACLOPRIDE(R)-6-Fluoro-3-(1-(2-(1-(quinolin-5-ylsulfonyl-pyrrolidin-2-yl)ethyl)piperidin-4-yl)-1,2-benzoxazole2Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
678965-HT1ACLONEDHUMAN3H-8-OH-DPATS)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole25Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678975-HT2ACLONEDHUMAN3H-KETANSERINS)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole16Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678985-HT6CLONEDHUMAN3H-LSDS)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole311Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
678995-HT7CLONEDHUMAN3H-5-CTS)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67900D2CLONEDHUMAN3H-RACLOPRIDES)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole1Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679015-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole37Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679025-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679035-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole313Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679045-HT7CLONEDHUMAN3H-5-CT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67905D2CLONEDHUMAN3H-R-ZACOPRIDE(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole0.14Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679065-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole37Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679075-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole18Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679085-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole360Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67909D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole0.5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679105-HT7CLONEDHUMAN3H-5-CT(S)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole12Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679115-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole24Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679125-HT2ACLONEDHUMAN3H-KETANSERIN(R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole21Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679135-HT6CLONEDHUMAN3H-LSD(R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole38Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679145-HT7CLONEDHUMAN3H-5-CT(R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole1Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67915D2CLONEDHUMAN3H-RACLOPRIDE(R)-3-(4-(2-(1-Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole0.7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679165-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole14Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679175-HT2ACLONEDHUMAN3H-KETANSERIN(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole10Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679185-HT6CLONEDHUMAN3H-LSD(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole40Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679195-HT7CLONEDHUMAN3H-5-CT(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67920D2CLONEDHUMAN3H-RACLOPRIDE(R)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole0.9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679215-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole16Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679225-HT2ACLONEDHUMAN3H-KETANSERIN(R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole15Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679235-HT6CLONEDHUMAN3H-LSD(R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole40Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679245-HT7CLONEDHUMAN3H-5CT(R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole1Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67925D2CLONEDHUMAN3H-RACLOPRIDE(R)-3-(4-(2-(1-(Isoquinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole0.3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679265-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole179Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679275-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole49Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679285-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole291Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679295-HT7CLONEDHUMAN3H-5CT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67930D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679315-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole96Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679325-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole33Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679335-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole497Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679345-HT7CLONEDHUMAN3H-5-CT(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67935D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Isoquinolin-4-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679365-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole86Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679375-HT2ACLONEDHUMAN3H-Ketaserin(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole41Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679385-HT6CLONEDHUMAN3H-LSD(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole92Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679395-HT7CLONEDHUMAN3H-5-CT(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole10Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67940D2CLONEDHUMAN3H-RACLOPRIDE(R)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)pyrrolidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzoxazole3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679415-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679425-HT2ACLONEDHUMAN3H-KETANSERIN(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)36Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679435-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)82Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679445-HT7CLONEDHUMAN3H-5-CT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67945D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)16Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679465-HT1ACLONEDHUMAN3H-8-OH-DPATS)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline18Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679475-HT2ACLONEDHUMAN3H-KETANSERINS)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679485-HT6CLONEDHUMAN3H-LSDS)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline116Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679495-HT7CLONEDHUMAN3H-5-CTS)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67950D2CLONEDHUMAN3H-RACLOPRIDES)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline11Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679515-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)10Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679525-HT2ACLONEDHUMAN3H-KETANSERIN(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679535-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)72Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679545-HT7CLONEDHUMAN3H-5CT(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)23Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67955D2CLONEDHUMAN3H-R-ZACOPRIDE(S)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679565-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)15Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679575-HT2ACLONEDHUMAN3H-KETANSERIN(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)56Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679585-HT6CLONEDHUMAN3H-LSD(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679595-HT7CLONEDHUMAN3H-5-CT(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)1Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67960D2CLONEDHUMAN3H-RACLOPRIDE(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679615-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline24Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679625-HT2ACLONEDHUMAN3H-KETANSERIN(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline26Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679635-HT6CLONEDHUMAN3H-LSD(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline11Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679645-HT7CLONEDHUMAN3H-5-CT(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67965D2CLONEDHUMAN3H-R-ZACOPRIDE(R)-4-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679665-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679675-HT2ACLONEDHUMAN3H-KETANSERIN(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)19Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679685-HT6CLONEDHUMAN3H-LSD(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)9Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679695-HT7CLONEDHUMAN3H-5CT(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67970D2CLONEDHUMAN3H-RACLOPRIDE(R)-5-((2-(2-(4-(Benzo[b]thiophen-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679715-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline14Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679725-HT2ACLONEDHUMAN3H-KETANSERIN(S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline244Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679735-HT6CLONEDHUMAN3H-LSD(S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline2310Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679745-HT7CLONEDHUMAN3H-5-CT(S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline165Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67975D2CLONEDHUMAN3H-RACLOPRIDE(S)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline42Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679765-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline8Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679775-HT2ACLONEDHUMAN3H-KETANSERIN(S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline82Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679785-HT6CLONEDHUMAN3H-LSD(S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline2057Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679795-HT7CLONEDHUMAN3H-5-CT(S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline75Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67980D2CLONEDHUMAN3H-RACLOPRIDE(S)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)isoquinoline37Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679815-HT1ACLONEDHUMAN3H-8-OH-DPAT(R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679825-HT2ACLONEDHUMAN3H-Ketaserin(R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline451Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679835-HT6CLONEDHUMAN3H-LSD(R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline641Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679845-HT7CLONEDHUMAN3H-5CT(R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline14Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67985D2CLONEDHUMAN3H-RACLOPRIDE(R)-5-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)quinoline8Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679865-HT1ACLONEDHUMAN3H-8-OH-DPATR)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679875-HT2ACLONEDHUMAN3H-KETANSERINR)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)76Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679885-HT6CLONEDHUMAN3H-LSDR)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)766Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679895-HT7CLONEDHUMAN3H-5-CTR)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67990D2CLONEDHUMAN3H-RACLOPRIDER)-4-((2-(2-(4-(1H-Indol-4-yl)piperazin-1-yl)ethyl)pyrrolidin-1-yl)sulfonyl)3Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679915-HT2ACLONEDHUMAN3H-KETANSERINHALOPERIDOL89Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679925-HT6CLONEDHUMAN3H-LSDHALOPERIDOL1083Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679935-HT7CLONEDHUMAN3H-5-CTHALOPERIDOL408Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67994D2CLONEDHUMAN3H-RACLOPRIDEHALOPERIDOL2Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
679955-HT1ACLONEDHUMAN3H-8-OH-DPATCLOZAPINE143Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679965-HT2ACLONEDHUMAN3H-KETANSERINCLOZAPINE13Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679975-HT6CLONEDHUMAN3H-LSDCLOZAPINE4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
679985-HT7CLONEDHUMAN3H-5CTCLOZAPINE>10000Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
67999D2CLONEDHUMAN3H-RACLOPRIDECLOZAPINE71Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
680005-HT1ACLONEDHUMAN3H-8-OH-DPATRISPERIDONE1169Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680015-HT2ACLONEDHUMAN3H-KETANSERINRISPERIDONE0.5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680025-HT6CLONEDHUMAN3H-LSDRISPERIDONE1107Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680035-HT7CLONEDHUMAN3H-5-CTRISPERIDONE0.4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68004D2CLONEDHUMAN3H-RACLOPRIDERISPERIDONE0.6Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
680055-HT1ACLONEDHUMAN3H-8-OH-DPATZiprasidone2Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680065-HT2ACLONEDHUMAN3H-KETANSERINZiprasidone1.7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680075-HT6CLONEDHUMAN3H-LSDZiprasidone20Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680085-HT7CLONEDHUMAN3H-5-CTZiprasidone5Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68009D2CLONEDHUMAN3H-RACLOPRIDEZiprasidone0.8Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
680105-HT1ACLONEDHUMAN3H-8-OH-DPATOLANZAPINE3442Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680115-HT2ACLONEDHUMAN3H-KETANSERINOLANZAPINE4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680125-HT6CLONEDHUMAN3H-LSDOLANZAPINE7Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680135-HT7CLONEDHUMAN3H-5-CTOLANZAPINE206Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68014D2CLONEDHUMAN3H-RACLOPRIDEOLANZAPINE4Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
680155-HT1ACLONEDHUMAN3H-8-OH-DPATARIPIPRAZOLE30Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680165-HT2ACLONEDHUMAN3H-KETANSERINARIPIPRAZOLE63Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680175-HT6CLONEDHUMAN3H-LSDARIPIPRAZOLE89Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680185-HT7CLONEDHUMAN3H-5-CTARIPIPRAZOLE44Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68019D2CLONEDHUMAN3H-RACLOPRIDEARIPIPRAZOLE0.8Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
680205-HT1ACLONEDHUMAN3H-8-OH-DPAT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole54Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680215-HT2ACLONEDHUMAN3H-KETANSERIN(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole30Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680225-HT6CLONEDHUMAN3H-LSD(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole344Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
680235-HT7CLONEDHUMAN3H-5-CT(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole57Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 15, 2025
68024D2CLONEDHUMAN3H-RACLOPRIDE(S)-3-(4-(2-(1-(Quinolin-5-ylsulfonyl)azetidin-2-yl)ethyl)piperazin-1-yl)-1,2-benzothiazole11Zajdel, Pawel et. al, 2018Jan 15, 2025Jan 28, 2025
68025CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide10.9648Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68026CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide5248.07Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68027CCK2CLONEDHUMAN125I-BH-CCK-8GW58231000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68028CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(Benzo[d]isoxazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide89.1251Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68029CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(Benzo[d]isoxazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide>10000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68030CCK1CLONEDHUMAN125I-BH-CCK-8GW582322.9087Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68031CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide8.31764Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68032CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide>10000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68033CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide13.8038Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68034CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide>10000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68035CCK1CLONEDHUMAN125I-BH-CCK-82-[3-[(N-Methylindol-3-yl)methyl]-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide17.7828Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68036CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-terahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide13.1826Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68037CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-terahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide>10000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68038CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamideisopropyl14.4544Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68039CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-3-methoxy-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamideisopropyl3630.78Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68040CCK1CLONEDHUMAN125I-BH-CCK-8N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]acetamide42.658Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68041CCK2CLONEDHUMAN125I-BH-CCK-8N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]acetamide2398.83Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68042CCK1CLONEDHUMAN125I-BH-CCK-82-[3-[(1-Benzyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide309.03Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68043CCK2CLONEDHUMAN125I-BH-CCK-82-[3-[(1-Benzyl-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide>10000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68044CCK1CLONEDHUMAN125I-BH-CCK-8N-Isopropyl-N-(4-methoxyphenyl)-2-[3-[(1-methyl-1H-indazol-3-yl)methyl]-3-methyl-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-benzo[b][1,4]diazepin-1-yl]acetamide38.9045Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68045CCK1CLONEDHUMAN125I-BH-CCK-82-[2,4-Dioxo-5-phenyl-3-[(1H-pyrazolo[3,4-b]pyridin-4-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide112.202Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68046CCK2CLONEDHUMAN125I-BH-CCK-82-[2,4-Dioxo-5-phenyl-3-[(1H-pyrazolo[3,4-b]pyridin-4-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide>10000Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68047CCK1CLONEDHUMAN125I-BH-CCK-82-[2,4-Dioxo-5-phenyl-3-[(4,5,6,7-tetrahydro-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-N-(4-methoxyphenyl)acetamide128.825Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68048CCK2CLONEDHUMAN125I-BH-CCK-82-[2,4-Dioxo-5-phenyl-3-[(4,5,6,7-tetrahydro-1H-indazol-3-yl)methyl]-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-N-(4-methoxyphenyl)acetamide2951.21Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68049CCK1CLONEDHUMAN125I-BH-CCK-82-[3-[(4-Fluoro-1H-indazol-3-yl)methyl]methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide17.378Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68050CCK2CLONEDHUMAN125I-BH-CCK-82-[3-[(4-Fluoro-1H-indazol-3-yl)methyl]methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide1698.24Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68051CCK1CLONEDHUMAN125I-BH-CCK-82-[3-[(5-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide42.658Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68052CCK2CLONEDHUMAN125I-BH-CCK-82-[3-[(5-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide2511.89Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68053CCK1CLONEDHUMAN125I-BH-CCK-82-[3-[(6-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide29.5121Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68054CCK2CLONEDHUMAN125I-BH-CCK-82-[3-[(6-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzotetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide588.844Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68055CCK1CLONEDHUMAN125I-BH-CCK-82-[3-[(7-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide20.893Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68056CCK2CLONEDHUMAN125I-BH-CCK-82-[3-[(7-Fluoro-1H-indazol-3-yl)methyl]-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(4-methoxyphenyl)acetamide1047.13Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68057CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide87.0964Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68058CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-phenylacetamide177.828Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68059CCK1CLONEDHUMAN125I-BH-CCK-8N-(4-Fluorophenyl)-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropylacetamide138.038Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68060CCK2CLONEDHUMAN125I-BH-CCK-8N-(4-Fluorophenyl)-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropylacetamide478.63Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68061CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[4-(trifluoromethyl)phenyl]acetamide660.693Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68062CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[4-(trifluoromethyl)phenyl]acetamide1659.59Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68063CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(3-methoxyphenyl)acetamide478.63Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68064CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(3-methoxyphenyl)acetamide190.546Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68065CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(2-methoxyphenyl)acetamide1584.89Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68066CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-(2-methoxyphenyl)acetamide128.825Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68067CCK1CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[3,4-(methylenedioxy)phenyl]acetamide354.813Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68068CCK2CLONEDHUMAN125I-BH-CCK-82-[3-(1H-Indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydrobenzo[b][1,4]diazepin-1-yl]-N-isopropyl-N-[3,4-(methylenedioxy)phenyl]acetamide724.436Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68069CCK1CLONEDHUMAN125I-BH-CCK-8N-Cyclopentyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-(4-methoxyphenyl)acetamide16.9824Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68070CCK2CLONEDHUMAN125I-BH-CCK-8N-Cyclopentyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-(4-methoxyphenyl)acetamide776.247Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68071CCK1CLONEDHUMAN125I-BH-CCK-8N-Cyclopropyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacetamide524.807Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68072CCK2CLONEDHUMAN125I-BH-CCK-8N-Cyclopropyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacetamide25.1189Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68073CCK1CLONEDHUMAN125I-BH-CCK-8N-tert-Butyl-2-[3-(1H-indazol-3-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5,5a,9a-hexahydrobenzo[b][1,4]diazepin-1-yl]-N-phenylacetamide891.251Henke BR et al., 1997Jan 15, 2025Jan 15, 2025
68074Y1CLONEDRhesus Monkey[125I] - Peptide YYNPY, human0.08Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68075Y1CLONEDRhesus Monkey[125I] - Peptide YYPYY, human0.22Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68076Y1CLONEDRhesus Monkey[125I] - Peptide YYPP, human50Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68077Y1CLONEDRhesus Monkey[125I] - Peptide YYNPY 3-36, human55Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68078Y1CLONEDRhesus Monkey[125I] - Peptide YYNPY 13-36, human30Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68079Y1CLONEDRhesus Monkey[125I] - Peptide YYNPY Leu31, Pro34, human0.08Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68080Y1CLONEDRhesus Monkey[125I] - Peptide YYNPY D-Trp32, human1000Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68081Y1CLONEDRhesus Monkey[125I] - Peptide YYBIBP32266.9Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68082Y1CLONEDHUMAN[125I] - Peptide YYNPY, human0.18Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68083Y1CLONEDHUMAN[125I] - Peptide YYPYY, human0.14Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68084Y1CLONEDHUMAN[125I] - Peptide YYPP, human19Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68085Y1CLONEDHUMAN[125I] - Peptide YYNPY 3-36, human50Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68086Y1CLONEDHUMAN[125I] - Peptide YYNPY Leu31, Pro34, human0.11Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68087Y1CLONEDHUMAN[125I] - Peptide YYNPY D-Trp32, human1000Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68088Y1CLONEDHUMAN[125I] - Peptide YYBIBP32269.7Gehlert DR, et al., 2001Jan 15, 2025Jan 15, 2025
68089AMPABRAINRAT3H-AMPAAMPA40Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68090AMPABRAINRAT3H-AMPAthio-AMPA1800Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68091AMPABRAINRAT3H-AMPAATPA2100Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68092AMPABRAINRAT3H-AMPAThio-ATPA630Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68093AMPABRAINRAT3H-AMPA(RS)-HIBO1500Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68094AMPABRAINRAT3H-AMPABr-HIBO650Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68095AMPABRAINRAT3H-AMPA2-Amino-3-(4-bromo-3-hydroxyisothiazol-5-yl)-propionic Acid Hyrochloride>10000Matzen L, et.al., 1997Jan 15, 2025Jan 15, 2025
68096M2UNDEFINEDUNDEFINED3H-AF-DX384ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68097M3UNDEFINEDUNDEFINED3H-4-DAMPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68098M4UNDEFINEDUNDEFINED3H-4-DAMPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68099M5UNDEFINEDUNDEFINED3H-4-DAMPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68100Alpha1AUNDEFINEDUNDEFINED3H-PRAZOSINABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68101Alpha1BUNDEFINEDUNDEFINED3H-PRAZOSINABT-594890Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68102Alpha1DUNDEFINEDUNDEFINED3H-PRAZOSINABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68103Alpha2BUNDEFINEDUNDEFINED3H-RAUWOLSCINEABT-594597Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68104Alpha2AUNDEFINEDUNDEFINED3H-RAUWOLSCINEABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68105Alpha2CUNDEFINEDUNDEFINED3H-RAUWOLSCINEABT-594342Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681065-HT1AUNDEFINEDUNDEFINED3H-8-OH-DPATABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681075-HT1BUNDEFINEDUNDEFINED125I-CYPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681085-HT2AUNDEFINEDUNDEFINED125I-DOIABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681095-HT2CUNDEFINEDUNDEFINED3H-MESULERGINEABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681105-HT3UNDEFINEDUNDEFINED3H-BRL 43694ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681115-HT6UNDEFINEDUNDEFINED3H-LSDABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
681125-HT7UNDEFINEDUNDEFINED3H-LSDABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68113A1UNDEFINEDUNDEFINED3H-CCPAABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68114UNDEFINEDUNDEFINED3H-CGS-21680ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68115A3UNDEFINEDUNDEFINED3H-AB-MECAABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68116Beta1UNDEFINEDUNDEFINED3H-CPG-12177 (-)ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68117Beta2UNDEFINEDUNDEFINED3H-CPG-12177 (-)ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 28, 2025
68118Beta3UNDEFINEDUNDEFINED125I-CYPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68119D1UNDEFINEDUNDEFINED3H-SCH23390ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68120D2UNDEFINEDUNDEFINED3H-SPIPERONEABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68121D3UNDEFINEDUNDEFINED3H-SPIPERONEABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68122D4UNDEFINEDUNDEFINED3H-SPIPERONEABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 27, 2025
68123D5UNDEFINEDUNDEFINED3H-SCH23390ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68124KORUNDEFINEDUNDEFINED3H-MUSCIMOLABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 27, 2025
68125GABABUNDEFINEDUNDEFINED3H-GABA(+50 mM isoguvacine to block GABAA)ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68126H3UNDEFINEDUNDEFINED3H-Alpha-Me-histamine-(R)ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68127UNDEFINEDUNDEFINED3H-DTGABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68128AT1UNDEFINEDUNDEFINED3H-A IIABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 28, 2025
68129UNDEFINEDUNDEFINED125I-ANPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68130UNDEFINEDUNDEFINED3H-V1-antagonistABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68131B2UNDEFINEDUNDEFINED3H-NPC 17731ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68132CCK1UNDEFINEDUNDEFINED3H-DevazepideABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68133ETAUNDEFINEDUNDEFINED125I-Endothelin 1ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68134GCCRUNDEFINEDUNDEFINED125I-GlucagonABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68135UNDEFINEDUNDEFINED125I-Tyr11-somatostatinABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68136Y1UNDEFINEDUNDEFINED125I-Peptide YYABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68137Y2UNDEFINEDUNDEFINED125I-Peptide YYABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68138NK1UNDEFINEDUNDEFINED3H-SPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68139NK2UNDEFINEDUNDEFINED125I-NKAABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68140NK3UNDEFINEDUNDEFINED3H-SENKTIDEABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68141UNDEFINEDUNDEFINED125I-NeurotensinABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68142Calcium channelUNDEFINEDUNDEFINED3H-D-888ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 29, 2025
68143Chloride channelUNDEFINEDUNDEFINED3H-TBPSABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68144UNDEFINEDUNDEFINED125I-CharybdotoxinABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68145UNDEFINEDUNDEFINED3H-TCPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68146UNDEFINEDUNDEFINED3H-SaxitoxinABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68147UNDEFINEDUNDEFINED3H-BatrachotoxininABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68148PBRUNDEFINEDUNDEFINED3H-PK11195ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68149BZPUNDEFINEDUNDEFINEDFNZABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68150GlyRUNDEFINEDUNDEFINED3H-StrychnineABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 27, 2025
68151AMPAUNDEFINEDUNDEFINED3H-AMPAABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68152KAUNDEFINEDUNDEFINED3H-Kainic acidABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68153NMDAUNDEFINEDUNDEFINED3H-MK-801ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68154NMDAUNDEFINEDUNDEFINED3H-CGP39653ABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 28, 2025
68155NETUNDEFINEDUNDEFINED3H-NisoxetineABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68156UNDEFINEDUNDEFINED3H-GABAABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68157UNDEFINEDUNDEFINED3H-Choline ChlorideABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68158SLC6A3UNDEFINEDUNDEFINED3H-BTCPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68159UNDEFINEDUNDEFINED3H-NBTIABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68160PDE1, PDE2, PDE3, PDE4UNDEFINEDUNDEFINED3H-cAMPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68161PDE5UNDEFINEDUNDEFINED3H-cGMPABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68162MOAUNDEFINEDUNDEFINEDKynuramineABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 29, 2025
68163MOAUNDEFINEDUNDEFINEDBenzylamineABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 29, 2025
68164COS-1UNDEFINEDUNDEFINEDIndomethacinABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68165COX-2UNDEFINEDUNDEFINEDNimesulfideABT-5941000Donnelly-Roberts DL, et al., 1998Jan 15, 2025Jan 15, 2025
68166A1BRAINRAT3H-cyclohexyladenosineCPA0.59Trivedi BK et al., 1989Jan 15, 2025Jan 15, 2025
68167Striatal MembranesRAT3H-NECACPA462Trivedi BK et al., 1989Jan 15, 2025Jan 15, 2025
68168A1BRAINRAT3H-cyclohexyladenosineN6-(2-endo-norbornyl)-adenosine0.42Trivedi BK et al., 1989Jan 15, 2025Jan 15, 2025
68169Striatal MembranesRAT3H-NECAN6-(2-endo-norbornyl)-adenosine750Trivedi BK et al., 1989Jan 15, 2025Jan 15, 2025
68170Striatal MembranesRAT3H-NECA2-exo-norbornyl isomer970Trivedi BK et al., 1989Jan 15, 2025Jan 15, 2025
68171A1BRAINRAT3H-cyclohexyladenosine2-exo-norbornyl isomer0.91Trivedi BK et al., 1989Jan 15, 2025Jan 15, 2025
68172CLONEDRAT3H-GLUTAMATE(S)-BrHlbo>10000Thomsen C, et.al., 1994aJan 15, 2025Jan 15, 2025
68173CLONEDRAT[3H]AP4(S)-BrHlbo1000Thomsen C, et.al., 1994aJan 15, 2025Jan 15, 2025
68174CLONEDRAT[3H]AP4(R)-BrHlbo1100Thomsen C, et.al., 1994aJan 15, 2025Jan 15, 2025
68175A1BRAINRAT3H-PIANB-Benzyladenosine-5-N-methyluronamide898Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68176A1Striatal MembranesRAT3H-CGS-21680NB-Benzyladenosine-5-N-methyluronamide597Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68177Striatal MembranesRAT3H-CGS-21680NB-Benzyladenosine-5-N-methyluronamide597Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68178A3CLONEDRAT125I-APNEANB-Benzyladenosine-5-N-methyluronamide16Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68179A1BRAINRAT3H-PIAM- (3-Iodoben zy1)adenosine- N-methyluronamide54Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68180Striatal MembranesRAT3H-CGS-21680M- (3-Iodoben zy1)adenosine- N-methyluronamide56Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68181A3CLONEDRAT125I-APNEAM- (3-Iodoben zy1)adenosine- N-methyluronamide1.1Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68182A1BRAINRAT3H-PIAN6-( 3-Aminobenzyl)adenosine-N-methyluronamide1000Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68183Striatal MembranesRAT3H-CGS-21680N6-( 3-Aminobenzyl)adenosine-5-N-methyluronamide794Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68184A3CLONEDRAT125I-APNEAN6-( 3-Aminobenzyl)adenosine-5-N-methyluronamide28Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68185A1BRAINRAT3H-PIAN6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide2970Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68186Striatal MembranesRAT3H-CGS-21680N6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide988Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68187A3CLONEDRAT125I-APNEAN6- (3-Acetamidobenzyl)adenosine-5- N-methyluronamide41.4Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68188A1BRAINRAT3H-PIAN6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide496Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68189Striatal MembranesRAT3H-CGS-21680N6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide574Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68190A3CLONEDRAT125I-APNEAN6--(3-(Trifluoromethyl)benzyl)adenosine-5-N-methyluronamide31Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68191A1BRAINRAT3H-PIAN6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide18Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68192Striatal MembranesRAT3H-CGS-21680N6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide197Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68193A3CLONEDRAT125I-APNEAN6---( 4-Amino-3-iodobenzyl)adenosine-5-N-methyluronamide1.27Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68194A1BRAINRAT3H-PIAN6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt>10000Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68195Striatal MembranesRAT3H-CGS-21680N6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt9070Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68196A3CLONEDRAT125I-APNEAN6-( 3-Sulfobenzyl)adenosine-5-N-methyluronamide Triethylammonium Salt1310Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68197A3CLONEDRAT125I-APNEAN6-( 4-Sulfobenzyl)adenosine-5-N-methyluronamide4500Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68198A1BRAINRAT3H-PIA(R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide3.2Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68199Striatal MembranesRAT3H-CGS-21680(R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide259Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68200A3CLONEDRAT125I-APNEA(R)-N6-( l-Phenylethyl)adenosine-5-N-ethyluronamide18Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68201A1BRAINRAT3H-PIA(S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide65Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68202Striatal MembranesRAT3H-CGS-21680(S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide1650Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68203A3CLONEDRAT125I-APNEA(S)-N6-( 1-P henylethyl)adenosine-5-N-ethyluronamide494Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68204A1BRAINRAT3H-PIAN6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide51Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68205Striatal MembranesRAT3H-CGS-21680N6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide32Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68206A3CLONEDRAT125I-APNEAN6-(3-Fluorobenzyl)adenosine-5-N-ethyluronamide10.7Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68207A1BRAINRAT3H-PIAN6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide22Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68208Striatal MembranesRAT3H-CGS-21680N6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide19Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68209A3CLONEDRAT125I-APNEAN6-(3-Chlorobenzyl)adenosine-5- N-ethyluronamide1.1Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68210A1BRAINRAT3H-PIAN6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide31Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68211Striatal MembranesRAT3H-CGS-21680N6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide24Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68212A3CLONEDRAT125I-APNEAN6-(2-Nitrobenzyl)adenosine-5-N-ethyluronamide2.8Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68213A1BRAINRAT3H-PIAN6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide78Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68214Striatal MembranesRAT3H-CGS-21680N6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide35Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68215A3Striatal MembranesRAT125I-APNEAN6-(3-Nitrobenzyl)adenosine-5-N-ethyluronamide8.7Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68216A1BRAINRAT3H-PIAN6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide49Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68217Striatal MembranesRAT3H-CGS-21680N6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide574Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68218A3Striatal MembranesRAT125I-APNEAN6-(4-Nitrobenzyl)adenosine-5-N-ethyluronamide9Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68219A3BRAINRAT3H-PIAN6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide209Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68220A1BRAINRAT3H-PIAN6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide209Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68221Striatal MembranesRAT3H-CGS-21680N6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide609Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68222A3CLONEDRAT125I-APNEAN6-(4 Methoxybenzyl)adenosine-5-N-ethyluronamide11Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68223A3CLONEDRAT125I-APNEAN6-Benzyladenosine-5-N-cyclopropyluronamide103Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68224Striatal MembranesRAT3H-CGS-21680N6-Benzyladenosine-5-N-cyclopropyluronamide55Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68225A1BRAINRAT3H-PIAN6-Benzyladenosine-5-N-cyclopropyluronamide112Gallo-Rodriguez C et al., 1994Jan 15, 2025Jan 15, 2025
68226CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-2- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate377Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68227CCK2PANCREASRAT125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-2- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate48Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68228CCK2PANCREASRAT125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-1- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate210Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68229CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-1- (+/-)-[1-(1H-indol-3-ylmethyl)-1-methyl-2-oxo-2-[(2-phenylethyl)amino] ethyl] carbamate785Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68230CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-2-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate775Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68231CCK2PANCREASRAT125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-2-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate6.4Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68232CCK2PANCREASRAT125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-1-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate21.6Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68233CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Tricyclo[3.3.1.1-3,7]dec-1-yl [R-(R*S*0-[2[[1-(hydroxy-methyl)-2-phenylethyl]amino]-1-(1H-indol-3-ylmethyl)-1-methyl-2-oxoethyl]carbamate1040Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68234CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]- cyclohexyl ester625Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68235CCK2PANCREASRAT125I-BH-CCK-8carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]- cyclohexyl ester517Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68236CCK2PANCREASRAT125I-BH-CCK-8carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]-2-chlorocyclohexyl ester trans (+/-)49Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68237CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8carbamic acid,[1-(1H-indol-3-ylmethyl)-1-methyl-2oxo 2-[(2-phenylethyl)amino] ethyl]-2-chlorocyclohexyl ester trans (+/-)196Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68238CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester66Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68239CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester15Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68240CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester (isomer I)140Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68241CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-chlorocyclohexyl ester (isomer I)118Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68242CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester288Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68243CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester36Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68244CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S)149Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68245CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S)251Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68246CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S)[(-)-isomer]266Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68247CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2-fluorocyclohexyl ester(indole center is R, hydroxymethyl center is S)[(-)-isomer]23Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68248CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester16Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68249CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester66Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68250CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1S-[1 alpha [S*(R*)], 2 beta]]75Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68251CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1S-[1 alpha [S*(R*)], 2 beta]]73Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68252CCK2PANCREASRAT125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1R-[1 alpha [R*(S*)], 2 beta]]9.3Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68253CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Carbamic acid, [2-[[ l-(hydroxymethyl)-2-phenylethyl]-amino)-1-(1H-indol-3-ylmethyl)-1methyl-2-oxoethyl]-, 2- methylcyclohexyl ester, [1R-[1 alpha [R*(S*)], 2 beta]]288Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68254CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-82-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1S-[1 alpha[S*R*(E)]],-2beta]]47Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68255CCK2PANCREASRAT125I-BH-CCK-82-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1S-[1 alpha[S*R*(E)]],-2beta]]6.5Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68256CCK2PANCREASRAT125I-BH-CCK-82-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*(E)]],-2beta]]1.2Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68257CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-82-Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*(E)]],-2beta]]154Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68258CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]]391Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68259CCK2PANCREASRAT125I-BH-CCK-8Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-3-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]]13Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68260CCK2PANCREASRAT125I-BH-CCK-8Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]]3.9Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68261CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta]]1810Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68262CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta(E)]]511Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68263CCK2PANCREASRAT125I-BH-CCK-8Butenoic Acid, 4-[[2-[[3-(1H-Indol-3-yl)-2-methyl-2-[[[(2-methylcyclohexyl)oxy]carbonyl]amino]-1-oxopropyl]-amino]-1-phenylpropyl]amino]-4-oxo-,[1R-[1 alpha[R*S*]],-2beta(E)]]4Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68264CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring centers are trans (+/-))0.6Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68265CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring centers are trans (+/-))8.9Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68266CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1S-trans)3.9Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68267CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-csrbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1S-trans)4.2Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68268CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1-R-trans)0.34Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68269CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(1-R-trans)18Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68270CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans)12Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68271CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans)815Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68272CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-(ring mixtures are trans)1260Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68273CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-( 1-S- trans)1260Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68274CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)-( 1-S- trans)20Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68275CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)7.9Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68276CCK2PANCREASRAT125I-BH-CCK-8Beta-alaine, N-[alpha-Methyl-N[[(2-methylcyclohexyl)oxy]-carbonyl]-D-3-tryptophyl]-L-3-(phenylmethyl)1160Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68277CCK1CEREBRAL CORTEXRAT125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester0.15Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68278CCK1CEREBRAL CORTEXRAT125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester25.5Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68279CCK2PANCREASRAT125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester0.15Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68280CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)-phenylmethyl ester25.5Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68281CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)186Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68282CCK2PANCREASRAT125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-D-3(phenylmethyl)9.3Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68283CCK2PANCREASRAT125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-L-3(phenylmethyl)13.2Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68284CCK1CEREBRAL CORTEXMOUSE125I-BH-CCK-8beta-alaine, N-[alpha-methyl-N-[(tricyclo[3.3.1.13,7] dec-2-yloxy)carbonyl]-L-3(phenylmethyl)539Boden PR et al., 1993Jan 15, 2025Jan 15, 2025
68285CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)glycine14Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68286CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)glycine1518Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68287CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-D-tryptophanyl]-N-(2-phenylethyl)glycine224Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68288CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-D-tryptophanyl]-N-(2-phenylethyl)glycine2842Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68289CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-2-phenylethylamine87Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68290CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-2-phenylethylamine1889Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68291CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)-3-aminopropionic Acid36Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68292CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-(2-phenylethyl)-3-aminopropionic Acid1323Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68293CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]glycine986Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68294CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]glycine4000Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68295CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]aniline407Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68296CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]aniline6082Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68297CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]benzylamine231Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68298CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]benzylamine4097Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68299CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](3-phenylpropyl)amine182Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68300CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](3-phenylpropyl)amine4249Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68301CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](2-naphthyl)amine402Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68302CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl](2-naphthyl)amine2356Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68303CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(1-naphthyl)ethyl]amine89Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68304CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(1-naphthyl)ethyl]amine2367Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68305CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(1-naphthyl)alaninyl]-N-(2-phenylethyl)glycine134Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68306CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(1-naphthyl)alaninyl]-N-(2-phenylethyl)glycine2013Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68307CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methylphenyl-alaninyl]-N-(2-phenylethyl)glycine87Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68308CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methylphenyl-alaninyl]-N-(2-phenylethyl)glycine3798Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68309CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(2-naphthyl)alaninyl]-N-(2-phenylethyl)glycine70Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68310CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(2-naphthyl)alaninyl]-N-(2-phenylethyl)glycine3006Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68311CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(4-bromophenyl)alaninyl]-N-(2-phenylethyl)glycine50Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68312CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyl-3-(4-bromophenyl)alaninyl]-N-(2-phenylethyl)glycine3414Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68313CCK2BRAINGUINEA PIG3H-pCCK8N-[(4-Chlorophenyl)-DL-a-methyltryptophanyl][(2phenylethyl)amino]urea>10000Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68314CCK1PANCREASGUINEA PIG3H-pCCK8N-[(4-Chlorophenyl)-DL-a-methyltryptophanyl][(2phenylethyl)amino]urea6329Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68315CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-methoxyphenyl)ethyl]amine115Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68316CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-methoxyphenyl)ethyl]amine3121Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68317CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-chlorophenyl)ethyl]amine39Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68318CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-chlorophenyl)ethyl]amine1614Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68319CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(3,4-dichlorophenyl)ethyl]amine184Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68320CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(3,4-dichlorophenyl)ethyl]amine1540Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68321CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-bromophenyl)ethyl]amine51Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68322CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-bromophenyl)ethyl]amine2141Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68323CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(2,4-dichlorophenyl)ethyl]amine27Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68324CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(2,4-dichlorophenyl)ethyl]amine3161Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68325CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-nitrophenyl)ethyl]amine79Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68326CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl][2-(4-nitrophenyl)ethyl]amine2352Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68327CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine6.5Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68328CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine1129Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68329CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-D-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine6.1Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68330CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-D-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine1060Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68331CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-L-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine36Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68332CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-L-a-methyltryptophanyl]-N-[2-(4-chlorophenyl)ethyl]glycine1039Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68333CCK2BRAINGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(2,4-dichlorophenyl)ethyl]glycine12.3Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68334CCK1PANCREASGUINEA PIG3H-pCCK8N-[N-[(2-Adamantyloxy)carbonyl]-DL-a-methyltryptophanyl]-N-[2-(2,4-dichlorophenyl)ethyl]glycine3045Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68335CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Naphthyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea3478Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68336CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Naphthyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea769Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68337CCK2BRAINGUINEA PIG3H-pCCK8N-[(2-Triphenylmethyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea>10000Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68338CCK1PANCREASGUINEA PIG3H-pCCK8N-[(2-Triphenylmethyl)-DL-a-methyltryptophanyl][2-phenylethyl)amino]urea1777Blommaert AG et al., 1993Jan 15, 2025Jan 15, 2025
68339nAChRKIDNEYHUMAN3H-EpibatidineNicotine5.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68340nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid4.9Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68341nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid4.3Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68342nAChRKIDNEYHUMAN3H-EpibatidineNicotine Free Janty EC Liquid167.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68343nAChRKIDNEYHUMAN3H-EpibatidineNicotine Free NicVape EC Liquid886.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68344nAChRBRAINRAT3H-EpibatidineNicotine9.3Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68345nAChRBRAINRAT3H-EpibatidineJanty EC Liquid9Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68346nAChRBRAINRAT3H-EpibatidineNicVape EC Liquid7.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68347nAChRBRAINRAT3H-EpibatidineNicotine Free Janty EC Liquid267.1Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68348nAChRBRAINRAT3H-EpibatidineNicotine Free NicVape EC Liquid1890Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68349nAChR7KIDNEYHUMAN3H-EpibatidineNicotine208.7Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68350nAChR7KIDNEYHUMAN3H-EpibatidineJanty EC Liquid277.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68351nAChR7KIDNEYHUMAN3H-EpibatidineNicVape EC Liquid352.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68352nAChR7BRAINRAT3H-EpibatidineNicotine9.2Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68353nAChR7BRAINRAT3H-EpibatidineJanty EC Liquid6.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68354nAChRKIDNEYHUMAN3H-EpibatidineNicotine303.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68355nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid288.4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68356nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid307.1Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68357nAChR7BRAINRAT3H-EpibatidineNicVape EC Liquid6.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68358nAChR7BRAINRAT3H-EpibatidineNicotine Free Janty EC Liquid178Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68359nAChR7BRAINRAT3H-EpibatidineNicotine Free NicVape EC Liquid1008Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68360nAChRKIDNEYHUMAN3H-EpibatidineNicotine4Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68361nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid3.8Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68362nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid4.8Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68363nAChRKIDNEYHUMAN3H-EpibatidineNicotine Free Janty EC Liquid111.9Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68364nAChRKIDNEYHUMAN3H-EpibatidineNicotine Free NicVape EC Liquid681.9Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68365nAChRKIDNEYHUMAN3H-EpibatidineNicotine73.3Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68366nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid52.8Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68367nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid88.7Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68368nAChRKIDNEYHUMAN3H-EpibatidineNicotine7.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68369nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid6.9Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68370nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid6.1Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68371nAChRKIDNEYHUMAN3H-EpibatidineNicotine Free Janty EC Liquid258.5Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68372nAChRKIDNEYHUMAN3H-EpibatidineNicotine Free NicVape EC Liquid1603Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68373nAChRKIDNEYHUMAN3H-EpibatidineNicotine22.6Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68374nAChRKIDNEYHUMAN3H-EpibatidineJanty EC Liquid23.2Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
68375nAChRKIDNEYHUMAN3H-EpibatidineNicVape EC Liquid23.8Harris, AC. et, al. 2018Jan 15, 2025Jan 29, 2025
683765-HT1ACLONEDHUMAN3H-8-OH-DPATcis 1-hydroxyindane67.6083Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683775-HT1ACLONEDHUMAN3H-8-OH-DPATtrans 1-hydroxyindane1.62181Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683785-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol23.4423Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683795-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol1.25893Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683805-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol6.60693Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683815-HT1ACLONEDHUMAN3H-8-OH-DPAT(-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin1-yl] 5-methoxyindan-1-ol1.02329Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683825-HT1ACLONEDHUMAN3H-8-OH-DPAT1-hydroxyindane67.6083Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683835-HT1ACLONEDHUMAN3H-8-OH-DPAT1-hydroxyindane1.62181Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683845-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo [1,4]dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-0123.4423Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683855-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-011.25893Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683865-HT1ACLONEDHUMAN3H-8-OH-DPAT(+)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-016.60693Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683875-HT1ACLONEDHUMAN3H-8-OH-DPAT(-)-trans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperazin-1-yl] 5-methoxyindan-1-011.02329Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683885-HT1ACLONEDHUMAN3H-8-OH-DPATPiperazine1.28825Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683895-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-0122.9087Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683905-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 3,6-dihydro-2H-pyridin-1-yl] indan-1-010.831764Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683915-HT1ACLONEDHUMAN3H-8-OH-DPATcis-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) 4-hydroxy piperid-1-yl] 5-fluoroindan-1-011000Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683925-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo [1,4] dioxin-5-yl) piperid-1-yl] indan-1-010.707946Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683935-HT1ACLONEDHUMAN3H-8-OH-DPATPiperidine0.288403Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683945-HT1ACLONEDHUMAN3H-8-OH-DPATtrans-2-[4-(2,3-Dihydrobenzo[1,4] dioxin-5-yl) piperid-1-yl] 6-nitroindan-1-010.74131Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
683955-HT1ACLONEDHUMAN3H-8-OH-DPATS 155350.794328Peglion JL, et.al., 2002Jan 15, 2025Jan 15, 2025
68396Alpha1ACLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one182Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68397Alpha2ACLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one0.13Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68398Alpha2BCLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1.03Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68399Alpha2CCLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one0.15Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68400D2CLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one81Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68401D3CLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one228Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68402D4CLONEDHUMAN[11C[R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one158Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
684035-HT1ACLONEDHUMAN[11C[R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1478Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684045-HT1BCLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1286Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684055-HT1DCLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one48Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684065-HT1ECLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one3330Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684075-HT1FCLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1678Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684085-HT2ACLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one434Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684095-HT2CCLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one97Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684105-HT4CLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1003Van der Mey. et, al. 2006Jan 15, 2025Jan 27, 2025
684115-HT5ACLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one352Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684125-HT6CLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one3056Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684135-HT7CLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one5Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68414CLONEDRAT[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one5118Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68415CLONEDHUMAN[11C]R1074742-methyl-3-[2-(1,2,3,4-tetrahydrobenzo[4,5]furo[3,2-c]pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidin-4-one1412Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68416Alpha1ACLONEDHUMAN[C11]R107474mirtazapine1815Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68417Alpha2ACLONEDHUMAN[C11]R107474mirtazapine20Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68418Alpha2BCLONEDHUMAN[11C]R107474mirtazapine88Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68419Alpha2CCLONEDHUMAN[11C]R107474mirtazapine18Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68420Beta1CLONEDHUMAN[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68421Beta2CLONEDHUMAN[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68422Beta3CLONEDHUMAN[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68423D1CLONEDRAT[11C]R107474mirtazapine4167Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68424D2CLONEDHUMAN[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68425D3CLONEDHUMAN[11C]R107474mirtazapine5723Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68426D4CLONEDHUMAN[11C]R107474mirtazapine2518Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
684275-HT1ACLONEDHUMAN[11C]R107474mirtazapine3334Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684285-HT1BCLONEDHUMAN[11C]R107474mirtazapine3534Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684295-HT1DCLONEDHUMAN[11C]R107474mirtazapine955Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684305-HT1ECLONEDHUMAN[11C]R107474mirtazapine728Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684315-HT1FCLONEDHUMAN[11C]R107474mirtazapine583Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684325-HT2ACLONEDHUMAN[11C]R107474mirtazapine70Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684335-HT2CCLONEDHUMAN[11C]R107474mirtazapine40Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684345-HT3CLONEDMOUSE[11C]R107474mirtazapine170Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684355-HT4CLONEDHUMAN[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 27, 2025
684365-HT5ACLONEDHUMAN[11C]R107474mirtazapine670Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684375-HT7CLONEDHUMAN[11C]R107474mirtazapine265Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68438H1CLONEDHUMAN[11C]R107474mirtazapine1.6Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68439CLONEDRAT[11C]R107474mirtazapine1100Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68440CLONEDRAT[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68441CLONEDRAT[11C]R107474mirtazapine6905Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68442SLC6A3CLONEDRAT[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
68443SERTCLONEDRAT[11C]R107474mirtazapine>10000Van der Mey. et, al. 2006Jan 15, 2025Jan 28, 2025
68444NETCLONEDRAT[11C]R107474mirtazapine1640Van der Mey. et, al. 2006Jan 15, 2025Jan 15, 2025
684455-HT1ACLONEDHUMAN3H-WAY100635N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684465-HT1BCLONEDHUMAN3H-5CTN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684475-HT1DCLONEDHUMAN3H-5CTN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684485-HT1ECLONEDHUMAN3H-5HTN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684495-HT2ACLONEDHUMAN3H-KETANSERINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684505-HT2CCLONEDHUMAN3H-MESULERGINEN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684515-HT2BCLONEDHUMAN3H-LSDN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide415He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684525-HT3CLONEDHUMAN3H-GR-65630N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684535-HT5ACLONEDHUMAN3H-LSDN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684545-HT6CLONEDHUMAN3H-LSDN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684555-HT7CLONEDHUMAN3H-LSDN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68456Alpha1ACLONEDHUMAN3H-PRAZOSINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68457Alpha1BCLONEDHUMAN3H-PRAZOSINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68458Alpha1DCLONEDHUMAN3H-PRAZOSINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68459Alpha2ACLONEDHUMAN3H-RAUWOLSCINEN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide1416He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68460Alpha2CCLONEDHUMAN3H-RAUWOLSCINEN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide575He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68461Alpha2BCLONEDHUMAN3H-RAUWOLSCINEN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68462Beta1CLONEDHUMAN125I-IodopindololN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68463Beta3CLONEDHUMAN125I-IodopindololN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68464Beta2CLONEDHUMAN3H-CPG-12177 (-)N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68465BZPCLONEDHUMANFNZN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68466D1CLONEDHUMAN3H-SCH23390N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68467D5CLONEDHUMAN3H-SCH23390N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68468D2CLONEDHUMAN3H-N-MethylspiperoneN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68469D3CLONEDHUMAN3H-N-MethylspiperoneN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68470D4CLONEDHUMAN3H-N-MethylspiperoneN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68471DATCLONEDHUMAN3H-WIN35428N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68472DORCLONEDHUMAN3H-DADLEN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68473KORCLONEDHUMAN3H-MUSCIMOLN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 27, 2025
68474H1CLONEDHUMAN3H-PYRILAMINEN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
684755-HT1DCLONEDHUMAN125I-aminopotentidineN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide443He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68476H3CLONEDHUMAN3H-Alpha-methylhistamineN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68477H4CLONEDHUMAN3H-HistamineN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68478KORCLONEDHUMAN3H-U69,593N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide1208He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68479M1CLONEDHUMAN3H-QNBN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68480M2CLONEDHUMAN3H-QNBN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68481M3CLONEDHUMAN3H-QNBN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68482M4CLONEDHUMAN3H-QNBN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68483M5CLONEDHUMAN3H-QNBN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide1749He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68484mGluR5CLONEDHUMAN3H-MPEPN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68485MORCLONEDHUMAN3H-DAMGON-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68486NETCLONEDHUMAN3H-NisoxetineN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide1289He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68487OTCLONEDHUMAN3H-OxytocinN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68488PBRCLONEDHUMAN3H-PK11195N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68489SERTCLONEDHUMAN3H-CITALOPRAMN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide2495He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68490Sigma 1CLONEDHUMAN3H-Pentazocine(+)N-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide1806He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68491Sigma 2CLONEDHUMAN3H-DTGN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide984He, S. et, al. 2017Jan 15, 2025Jan 28, 2025
68492V1ACLONEDHUMAN3H-VASOPRESSINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68493V1BCLONEDHUMAN3H-VASOPRESSINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
68494V2CLONEDHUMAN3H-VASOPRESSINN-(3-(cis-3,5-Dimethylpiperidin-1-yl)propyl)-1-((2-(2-chloro-6-methylphenyl)-5-methyloxazol-4-yl)methyl)piperidine-4-carboxamide>10000He, S. et, al. 2017Jan 15, 2025Jan 15, 2025
684955-HT3CLONEDHUMAN3H-GR-65630Ondansetron HCl3.6PDSP Certified DataJan 15, 2025Jan 15, 2025
68496BRAINRAT3H-RAUWOLSCINE(+-)Org3770112.202De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68497BRAINRAT3H-RAUWOLSCINE(+)Org377063.0957De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68498BRAINRAT3H-RAUWOLSCINE(-)Org37702344.23De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68499BRAINRAT3H-RAUWOLSCINE(+-)Mianserin109.648De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68500BRAINRAT3H-RAUWOLSCINE(+)Mianserin57.544De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68501BRAINRAT3H-RAUWOLSCINE(-)Mianserin363.078De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68502BRAINRAT3H-MIANSERIN(+-)Org37708.91251De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68503BRAINRAT3H-MIANSERIN(+)Org37704.7863De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68504BRAINRAT3H-MIANSERIN(-)Org377060.256De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68505BRAINRAT3H-MIANSERIN(+-)Mianserin0.363078De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68506BRAINRAT3H-MIANSERIN(+)Mianserin0.416869De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68507BRAINRAT3H-MIANSERIN(-)Mianserin18.6209De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68508D2BRAINRAT3H-SPIPERONE(+-)Org37703981.07De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68509D2BRAINRAT3H-SPIPERONE(+)Org37705011.87De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68510D2BRAINRAT3H-SPIPERONE(-)Org37703981.07De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68511D2BRAINRAT3H-SPIPERONE(+-)Mianserin>10000De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68512H1BRAINRAT3H-MEPYRAMINE(+-)Org37700.501187De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68513H1BRAINRAT3H-MEPYRAMINE(+)Org37700.316228De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68514H1BRAINRAT3H-MEPYRAMINE(-)Org37700.630957De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68515H1BRAINRAT3H-MEPYRAMINE(+-)Mianserin1.77828De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68516H1BRAINRAT3H-MEPYRAMINE(+)Mianserin1De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68517BRAINRAT3H-QNB(+)Mianserin3981.07De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68518BRAINRAT3H-QNB(-)Mianserin151.356De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68519BRAINRAT3H-QNB(+-)Mianserin501.187De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68520BRAINRAT3H-QNB(+-)Org3770794.328De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68521BRAINRAT3H-QNB(+)Org37707079.46De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68522BRAINRAT3H-QNB(-)Org3770251.189De Boer TH, et al., 1988Jan 15, 2025Jan 15, 2025
68523D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-fluorobenzamide10.1Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68524D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-fluorobenzamide1.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68525D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-fluorobenzamide8.8Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68526D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-fluorobenzamide1.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68527D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-fluorobenzamide6.1Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68528D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-fluorobenzamide1Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68529D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-chlorobenzamide10.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68530D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-chlorobenzamide1.3Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68531D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-chlorobenzamide15Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68532D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-chlorobenzamide2.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68533D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-chlorobenzamide17.5Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68534D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-chlorobenzamide2.6Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68535D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-iodobenzamide10.6Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68536D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-iodobenzamide3.8Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68537D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-iodobenzamide28.1Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68538D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-iodobenzamide3.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68539D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-iodobenzamide35.4Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68540D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-iodobenzamide3.4Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68541D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-methoxy-benzamide3.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68542D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-methoxy-benzamide0.6Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68543D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-methoxy-benzamide39.1Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68544D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-methoxy-benzamide3Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68545D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-methoxy-benzamide30.4Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68546D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-methoxy-benzamide1.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68547D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-hydroxy-benzamide6.6Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68548D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-hydroxy-benzamide0.8Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68549D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-hydroxy-benzamide13.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68550D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-hydroxy-benzamide0.4Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68551D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-nitrobenzamide7.4Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68552D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-2-nitrobenzamide3.4Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68553D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-nitrobenzamide21.9Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68554D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-3-nitrobenzamide2.3Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68555D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-nitrobenzamide19.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68556D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-nitrobenzamide0.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68557D2CLONEDHUMAN125I-IABN2-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide18.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68558D3CLONEDHUMAN125I-IABN2-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide2.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68559D2CLONEDHUMAN125I-IABN3-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide29Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68560D3CLONEDHUMAN125I-IABN3-Amino-N-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-benzamide2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68561D2CLONEDHUMAN125I-IABNPyridine-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide16.9Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68562D3CLONEDHUMAN125I-IABNPyridine-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide2.6Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68563D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-nicotinamide19.6Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68564D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-nicotinamide2.5Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68565D2CLONEDHUMAN125I-IABNPyridine-4-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide31.2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68566D3CLONEDHUMAN125I-IABNPyridine-4-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide2Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68567D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide93.3Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68568D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide0.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68569D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide54.5Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68570D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide0.9Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68571D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-4-yl-benzamide43.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68572D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-4-yl-benzamide0.9Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68573D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyrimidin-2-yl-benzamide45.7Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68574D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyrimidin-2-yl-benzamide1.3Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68575D2CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-(1H-imidazol-2-yl)-benzamide8Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68576D3CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-(1H-imidazol-2-yl)-benzamide0.3Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68577D2CLONEDHUMAN125I-IABNQuinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide65.5Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68578D3CLONEDHUMAN125I-IABNQuinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide3.8Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68579D2CLONEDHUMAN125I-IABNBenzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide149Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68580D3CLONEDHUMAN125I-IABNBenzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide1.1Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68581D2CLONEDHUMAN125I-IABN2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide76.5Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68582D3CLONEDHUMAN125I-IABN2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide1.5Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68583D4CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-2-yl-benzamide375Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68584D4CLONEDHUMAN125I-IABNN-{4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-4-pyridine-3-yl-benzamide520Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68585D4CLONEDHUMAN125I-IABNQuinoxaline-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide1110Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68586D4CLONEDHUMAN125I-IABNBenzo[b]thiophene-2-carboxylic acid-{4-[4-(2,3-dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide1770Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68587D4CLONEDHUMAN125I-IABN2-Benzofuran-2-carboxylic acid {4-[4-(2,3-Dichlorophenyl)-piperazin-1-yl]-trans-but-2-enyl}-amide1070Grundt P, et al., 2005Jan 15, 2025Jan 15, 2025
68588nAChRStriatal MembranesRAT3H-NICOTINEN-methylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68589nAChRStriatal MembranesRAT3H-NICOTINEN-ethylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68590nAChRStriatal MembranesRAT3H-NICOTINEN-n-propylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68591nAChRStriatal MembranesRAT3H-NICOTINEN-n-butylpyridinium iodide9650Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68592nAChRStriatal MembranesRAT3H-NICOTINEN-n-pentylpyridinium iodide8720Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68593nAChRStriatal MembranesRAT3H-NICOTINEN-n-hexylpyridinium iodide9070Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68594nAChRStriatal MembranesRAT3H-NICOTINEN-n-heptylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68595nAChRStriatal MembranesRAT3H-NICOTINEN-n-octylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68596nAChRStriatal MembranesRAT3H-NICOTINEN-n-nonylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68597nAChRStriatal MembranesRAT3H-NICOTINEN-n-decylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68598nAChRStriatal MembranesRAT3H-NICOTINEN-n-undecylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68599nAChRStriatal MembranesRAT3H-NICOTINEN-n-dodecylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68600nAChRStriatal MembranesRAT3H-NICOTINEN-n-pentadecylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68601nAChRStriatal MembranesRAT3H-NICOTINEN-n-eicosylpyridinium iodide>10000Grinevich VP, et al., 2003Jan 15, 2025Jan 15, 2025
68602recombinantHUMAN3H-AdoMetSKF 29661550Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68603recombinantHUMAN3H-AdoMetp-chlorophenyl moiety2600Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68604recombinantHUMAN3H-AdoMet7-((N-Methylamino)sulfonyl)-1,2,3,4-tetrahydroisoquinoline4600Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68605recombinantHUMAN3H-AdoMet7-(N-(Methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline4800Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68606recombinantHUMAN3H-AdoMet7-(N,N-Bis(methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68607recombinantHUMAN3H-AdoMet7-((N-(Methylsulfonyl)amino)methyl)-1,2,3,4-tetrahydroisoquinoline>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68608recombinantHUMAN3H-AdoMet8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline980Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68609recombinantHUMAN3H-AdoMet1-(Aminomethyl)-6-methoxynaphthalene1500Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68610recombinantHUMAN3H-AdoMet1-(Aminomethyl)-6-hydroxynaphthalene8400Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68611recombinantHUMAN3H-AdoMet8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline1400Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68612CORTEXRAT3H-CLONIDINESKF 29661>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68613CORTEXRAT3H-CLONIDINEp-chlorophenyl moiety6300Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68614CORTEXRAT3H-CLONIDINE7-((N-Methylamino)sulfonyl)-1,2,3,4-tetrahydroisoquinoline>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68615CORTEXRAT3H-CLONIDINE7-(N-(Methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68616CORTEXRAT3H-CLONIDINE7-(N,N-Bis(methylsulfonyl)amino)-1,2,3,4-tetrahydroisoquinoline>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68617CORTEXRAT3H-CLONIDINE7-((N-(Methylsulfonyl)amino)methyl)-1,2,3,4-tetrahydroisoquinoline>10000Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68618CORTEXRAT3H-CLONIDINE8-Hydroxy-1,2,3,4-tetrahydrobenz[h]isoquinoline78Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68619CORTEXRAT3H-CLONIDINE1-(Aminomethyl)-6-methoxynaphthalene4600Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68620CORTEXRAT3H-CLONIDINE1-(Aminomethyl)-6-hydroxynaphthalene2100Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68621CORTEXRAT3H-CLONIDINE8-Methoxy-1,2,3,4-tetrahydrobenz[h]isoquinoline840Grunewald GL, et al., 1997Jan 15, 2025Jan 15, 2025
68622UTCLONEDHUMANI125-urotensin IIU-II (H-Glu-Thr-Pro-Asp-cyclo[Cys-Phe-Trp-Lys-Tyr-Cys]-Val-OH) 0.794328Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68623UTCLONEDHUMANI125-urotensin IIH-U-II(4-11)-Asp-C[Cys-Phe-Trp-Lys-Tyr-Cys]Val-OH0.251189Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68624UTCLONEDHUMANI125-urotensin IIH-P5U-Asp-C[Pen-Phe-Trp-Lys-Tyr-Cys]Val-OH0.199526Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68625UTCLONEDHUMANI125-urotensin IIH-Asp-C[Pen-Phe-DTrp-Lys-Tyr-Cys]Val-OH1.25893Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68626UTCLONEDHUMANI125-urotensin IIH-Asp-C[Cys-Phe-DTrp-Lys-Tyr-Cys]Val-OH1.25893Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68627UTCLONEDHUMANI125-urotensin IIH-Asp-C[Pen-Phe-Trp-Orn-Tyr-Cys]Val-OH15.8489Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68628UTCLONEDHUMANI125-urotensin IIH-Asp-C[Cys-Phe-Trp-Orn-Tyr-Cys]Val-OH10Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68629UTCLONEDHUMANI125-urotensin IIH-Asp-C[Pen-Phe-DTrp-Orn-Tyr-Cys]Val-OH5.01187Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68630UTCLONEDHUMANI125-urotensin IIH-Asp-C[Cys-Phe-DTrp-Orn-Tyr-Cys]Val-OH12.5893Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68631UTCLONEDHUMANI125-urotensin IIH-Asp-C[DPen-Phe-DTrp-Orn-Tyr-Cys]Val-OH1995.26Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68632UTCLONEDHUMANI125-urotensin IIH-Asp-C[Pen-Phe-DTrp-DOrn-Tyr-Cys]Val-OH398.107Grieco P, et al., 2005Jan 15, 2025Jan 29, 2025
68633recombinantHUMANUNKNOWNBrassinin>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68634recombinantHUMANUNKNOWNN-[2-(Indol-3-yl)ethyl]-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68635recombinantHUMANUNKNOWNN-[2-(Benzo[b]thiophen-3-yl)ethyl]-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68636recombinantHUMANUNKNOWNN-[3-(Indol-3-yl)propyl]-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68637recombinantHUMANUNKNOWNN-(Indan-2-yl)-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68638recombinantHUMANUNKNOWNN-(Adamant-2-yl)-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68639recombinantHUMANUNKNOWNN-[(Naphth-2-yl)methyl]-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68640recombinantHUMANUNKNOWNN-Benzyl-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68641recombinantHUMANUNKNOWNN-Phenethyl-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68642recombinantHUMANUNKNOWNN-4-Fluorophenethyl-S-methyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68643recombinantHUMANUNKNOWNN,S-Dimethyl-N-phenethyldithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68644recombinantHUMANUNKNOWNS-Allyl-brassinin>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68645recombinantHUMANUNKNOWNS-Benzyl-brassinin>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68646recombinantHUMANUNKNOWNS-Hexyl-brassinin>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68647recombinantHUMANUNKNOWNN-[2-(Indol-3-yl)ethyl]-S-benzyl-dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68648recombinantHUMANUNKNOWNN-[2-(Indol-3-yl)ethyl]-S-[(naphth-2-yl)methyl]dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68649recombinantHUMANUNKNOWNN-[2-(Indol-3-yl)ethyl]-S-[(pyrid-3-yl)methyl]dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68650recombinantHUMANUNKNOWNN-[2-(Indol-3-yl)ethyl]-S-[(pyrid-4-yl)methyl]dithiocarbamate>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68651recombinantHUMANUNKNOWNN-[1-(Indol-3-yl)ethyl]-N'-methyl-thiourea>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68652recombinantHUMANUNKNOWNN-[(Indol-3-yl)methyl]propanethioamide>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68653recombinantHUMANUNKNOWN4-[(Indol-3-yl)methyl]thiazole>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68654recombinantHUMANUNKNOWN4-[(Indol-3-yl)methyl]-2-methyl-thiazole>10000Gaspari P, et al., 2006Jan 15, 2025Jan 15, 2025
68655DORBRAINRAT3H-DPDPEDPI-5201150.3Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68656DORBRAINRAT3H-DPDPEDPI-673384.7Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68657DORBRAINRAT3H-DPDPEDPI-540212.7Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68658DORBRAINRAT3H-DPDPEDPI-533641.8Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68659DORBRAINRAT3H-DPDPEDPI-5337429.9Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68660DORBRAINRAT3H-DPDPEDPI-5701119.3Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68661DORBRAINRAT3H-DPDPEDPI-57023.8Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68662MORBRAINRAT3H-DAMGODPI-32900.46Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68663MORBRAINRAT3H-DAMGODPI-52011000Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68664MORBRAINRAT3H-DAMGODPI-67364.4Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68665MORBRAINRAT3H-DAMGODPI-54027.3Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68666MORBRAINRAT3H-DAMGODPI-53366.4Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68667MORBRAINRAT3H-DAMGODPI-5337320.2Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68668MORBRAINRAT3H-DAMGODPI-5701405.5Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68669MORBRAINRAT3H-DAMGODPI-570211.6Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68670KORBRAINRAT3H-U69,593DPI-32900.62Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68671KORBRAINRAT3H-U69,593DPI-673306.8Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68672KORBRAINRAT3H-U69,593DPI-540213.8Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68673KORBRAINRAT3H-U69,593DPI-5336414.2Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68674KORBRAINRAT3H-U69,593DPI-53371000Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68675KORBRAINRAT3H-U69,593DPI-5701231.4Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68676KORBRAINRAT3H-U69,593DPI-570219.1Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
68677DORBRAINRAT3H-DPDPEDPI-32900.18Gengo PJ, et.al.,2003Jan 15, 2025Jan 15, 2025
686785-HT5ACLONEDHUMAN3H-5CT5-Hydroxy Tryptamine126Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686795-HT5ACLONEDMOUSEI125-2-iodo LSD2-Br LSD2Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686805-HT5ACLONEDMOUSEI125-2-iodo LSDMETHYSERGIDE63Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686815-HT5ACLONEDHUMAN3H-5CTMETERGOLINE630Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686825-HT5ACLONEDHUMAN3H-5CT5-CT20Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686835-HT5ACLONEDHUMAN3H-5CTSUMATRIPTAN5000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686845-HT5ACLONEDHUMAN3H-5CT8-OH-DPAT2500Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686855-HT5ACLONEDMOUSE3H-LSD2-Methyl 5-HT>10000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686865-HT5ACLONEDHUMAN3H-5CTMETHIOTHEPIN1Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686875-HT5ACLONEDHUMAN3H-5CTKETANSERIN>10000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686885-HT5ACLONEDMOUSE3H-LSDQUIPAZINE>10000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686895-HT5ACLONEDMOUSE3H-LSD1-NP40Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686905-HT5ACLONEDHUMAN3H-5CTSPIPERONE>10000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686915-HT5ACLONEDHUMAN3H-5CTCLOZAPINE1000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686925-HT6CLONEDHUMAN3H-LSD5-Hydroxy Tryptamine65Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686935-HT6CLONEDHUMAN125I-2-iodo LSD2-Br LSD17Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686945-HT6CLONEDHUMAN3H-LSDMETHYSERGIDE180Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686955-HT6CLONEDHUMAN3H-LSDMETERGOLINE400Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686965-HT6CLONEDHUMAN3H-LSD5-CT720Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686975-HT6CLONEDHUMAN3H-LSDSUMATRIPTAN2600Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686985-HT6CLONEDHUMAN3H-LSD8-OH-DPAT>10000Glennon RA, 2003Jan 15, 2025Jan 15, 2025
686995-HT6CLONEDHUMAN125I-2-iodo LSD2-Methyl 5-HT400Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687005-HT6CLONEDHUMAN3H-LSDMETHIOTHEPIN0.4Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687015-HT6CLONEDHUMAN3H-LSDKETANSERIN2800Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687025-HT6CLONEDHUMAN3H-LSDQUIPAZINE3600Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687035-HT6CLONEDHUMAN125I-2-iodo LSD1-NP104Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687045-HT6CLONEDHUMAN3H-LSDSPIPERONE1595Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687055-HT6CLONEDHUMAN3H-LSDCLOZAPINE9.5Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687065-HT6CLONEDHUMAN3H-LSDMIANSERIN55Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687075-HT7CLONEDHUMAN3H-5HT5-Hydroxy Tryptamine8.1Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687085-HT7CLONEDHUMAN3H-5HT2-Br LSD30Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687095-HT7CLONEDHUMAN3H-5HTMETHYSERGIDE83Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687105-HT7CLONEDHUMAN3H-5HTMETERGOLINE6.4Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687115-HT7CLONEDHUMAN3H-5HT5-CT0.9Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687125-HT7CLONEDHUMAN3H-5HTSUMATRIPTAN950Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687135-HT7CLONEDHUMAN3H-5HT8-OH-DPAT466Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687145-HT7CLONEDHUMAN3H-LSD2-Methyl 5-HT1258Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687155-HT7CLONEDHUMAN3H-5HTMETHIOTHEPIN3.7Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687165-HT7CLONEDHUMAN3H-5HTKETANSERIN1334Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687175-HT7CLONEDHUMAN3H-LSDQUIPAZINE3033Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687185-HT7CLONEDHUMAN3H-5HT1-NP83Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687195-HT7CLONEDHUMAN3H-5HTSPIPERONE110Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687205-HT7CLONEDHUMAN3H-LSDCLOZAPINE40Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687215-HT7CLONEDHUMAN3H-5HTMIANSERIN8010Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687225-HT7CLONEDRAT3H-5HTSPIPERONE10Glennon RA, 2003Jan 15, 2025Jan 15, 2025
687235-HT7CLONEDMOUSE3H-5HTSPIPERONE63Glennon RA, 2003Jan 15, 2025Jan 15, 2025
68724D1KIDNEYMonkey3H-SCH23390SCH 233900.6Grandy DK, et al., 1991Jan 15, 2025Jan 15, 2025
68725D1KIDNEYMonkey3H-SCH23390BUTACLAMOL,(+)9.1Grandy DK, et al., 1991Jan 15, 2025Jan 15, 2025
68726D1KIDNEYMonkey3H-SCH23390cis-flupenthixol23.6Grandy DK, et al., 1991Jan 15, 2025Jan 15, 2025
68727D1KIDNEYMonkey3H-SCH23390HALOPERIDOL156Grandy DK, et al., 1991Jan 15, 2025Jan 15, 2025
68728D1KIDNEYMonkey3H-SCH23390CLOZAPINE406Grandy DK, et al., 1991Jan 15, 2025Jan 15, 2025
68729D1KIDNEYMonkey3H-SCH23390BUTACLAMOL, (-)>10000Grandy DK, et al., 1991Jan 15, 2025Jan 15, 2025
68730M5CLONEDHUMAN3H-NMSxanomeline>10000Grant MK, et al., 2005Jan 15, 2025Jan 15, 2025
68731CRF1CLONEDHUMAN125I-SauvagineAntalarmin3.1Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68732CRF1CLONEDHUMAN125I-Sauvagine1-(2,4-Dichloro-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one5.1Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68733CRF1CLONEDHUMAN125I-Sauvagine1-(2-Bromo-4-isopropyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one1.1Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68734CRF1CLONEDHUMAN125I-Sauvagine1-(4-Chloro-phenyl)-7-methyl-5-(1-propylbutyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one12Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68735CRF1CLONEDHUMAN125I-Sauvagine1-(4-Methanesulfonyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one460Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68736CRF1CLONEDHUMAN125I-Sauvagine1-(4-Methoxycarbonyl-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one920Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68737CRF1CLONEDHUMAN125I-Sauvagine1-(4-Methoxy-phenyl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one2Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68738CRF1CLONEDHUMAN125I-Sauvagine1-(5-Chloro-pyridin-2-yl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one23Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68739CRF1CLONEDHUMAN125I-Sauvagine1-(6-Methoxy-pyridin-3-yl)-7-methyl-5-(1-propyl-butyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one60Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68740CRF1CLONEDHUMAN125I-Sauvagine5-Isopropyl-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one>10000Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68741CRF1CLONEDHUMAN125I-Sauvagine5-Butyl-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one8800Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68742CRF1CLONEDHUMAN125I-Sauvagine5-(1-Ethyl-propyl)-1-(4-methoxy-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one8Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68743CRF1CLONEDHUMAN125I-Sauvagine5-(1-Methoxymethyl-propyl)-1-(4-methoxyphenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one150Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68744CRF1CLONEDHUMAN125I-Sauvagine5-(1-Ethyl-propyl)-7-methyl-1-(4-trifluoromethyl-phenyl)-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one170Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68745CRF1CLONEDHUMAN125I-Sauvagine5-(1-Ethyl-propyl)-1-(4-methoxy-2-methyl-phenyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one20Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
68746CRF1CLONEDHUMAN125I-Sauvagine1-(4-Chloro-phenyl)-5-(1-methoxymethyl-propyl)-7-methyl-4,5-dihydro-1H,3H-1,2a,5,8-tetraaza-acenaphthylen-2-one trifluoroacetate200Guo Z, et al., 2005Jan 15, 2025Jan 15, 2025
687475-HT4CAUDATEPIG3H-GR-113808GR 1254870.19Schiavi, GB et al., 1994Jan 15, 2025Jan 15, 2025
687485-HT4CAUDATEPIG3H-GR-113808GR 1138080.32Schiavi, GB et al., 1994Jan 15, 2025Jan 15, 2025